4wd5:A (GLY779) to (ARG973) CRYSTAL STRUCTURE OF EGFR 696-1022 T790M IN COMPLEX WITH QL-X138 | EGFR, T790M, GATEKEEPER MUTATION, INHIBITOR, TRANSFERASE-INHIBITOR COMPLEX
2auh:A (LEU1063) to (LEU1262) CRYSTAL STRUCTURE OF THE GRB14 BPS REGION IN COMPLEX WITH THE INSULIN RECEPTOR TYROSINE KINASE | TYROSINE KINASE, BPS REGION, TRANSFERASE/SIGNALING PROTEIN COMPLEX
4wkq:A (GLY779) to (ARG973) 1.85 ANGSTROM STRUCTURE OF EGFR KINASE DOMAIN WITH GEFITINIB | INHIBITOR, COMPLEX, KINASE, EPIDERMAL GROWTH FACTOR RECEPTOR, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2b4s:B (LEU1063) to (LEU1263) CRYSTAL STRUCTURE OF A COMPLEX BETWEEN PTP1B AND THE INSULIN RECEPTOR TYROSINE KINASE | HYDROLASE/TRANSFERASE, PHOSPHORYLATION, TYROSINE PROTEIN KINASE
4wrg:A (GLY779) to (ARG973) 1.9 ANGSTROM STRUCTURE OF EGFR KINASE DOMAIN | TRANSFERASE, KINASE DOMAIN
3emg:A (GLY437) to (TYR631) DISCOVERY AND SAR OF NOVEL 4-THIAZOLYL-2- PHENYLAMINOPYRIMIDINES AS POTENT INHIBITORS OF SPLEEN TYROSINE KINASE (SYK) | KINASE, SYK, ALTERNATIVE SPLICING, ATP-BINDING, HOST-VIRUS INTERACTION, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, UBL CONJUGATION
3eqp:B (GLY194) to (GLN389) CRYSTAL STRUCTURE OF ACK1 WITH COMPOUND T95 | ACK1, ALTERNATIVE SPLICING, ATP-BINDING, CELL MEMBRANE, KINASE, MAGNESIUM, MEMBRANE, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3eqr:A (GLY194) to (GLN389) CRYSTAL STRUCTURE OF ACK1 WITH COMPOUND T74 | ACK1, ALTERNATIVE SPLICING, ATP-BINDING, CELL MEMBRANE, KINASE, MAGNESIUM, MEMBRANE, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3eqr:B (GLY194) to (ALA388) CRYSTAL STRUCTURE OF ACK1 WITH COMPOUND T74 | ACK1, ALTERNATIVE SPLICING, ATP-BINDING, CELL MEMBRANE, KINASE, MAGNESIUM, MEMBRANE, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3f5p:J (VAL1062) to (ILE1266) COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR | IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
4hzr:A (GLY194) to (GLN389) CRYSTAL STRUCTURE OF ACK1 KINASE DOMAIN | ACTIVE STATE, PHOSPHOTRANSFER, TRANSFERASE
4hzr:B (GLY194) to (GLN389) CRYSTAL STRUCTURE OF ACK1 KINASE DOMAIN | ACTIVE STATE, PHOSPHOTRANSFER, TRANSFERASE
4xg2:A (GLY437) to (LEU636) CRYSTAL STRUCTURE OF LIGAND-FREE SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE
4xg3:A (GLY437) to (VAL634) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4xg3:B (GLY437) to (VAL633) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4xg4:A (GLY437) to (ASN635) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4i0r:A (GLY437) to (HIS639) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH 2-(3,4,5- TRIMETHOXY-PHENYL)-5H-PYRROLO[2,3-B]PYRAZINE-7-CARBOXYLIC ACID ISOPROPYLAMIDE | KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4xg6:A (GLY437) to (ASN635) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4i0s:A (GLY437) to (HIS639) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH 2-(6- CHLORO-1-METHYL-1H-INDAZOL-3-YL)-5H-PYRROLO[2,3-B]PYRAZINE-7- CARBOXYLIC ACID ISOPROPYLAMIDE | KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4xg7:A (GLY437) to (ASN635) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4i0t:A (GLY437) to (HIS639) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH 2-(5,6,7,8- TETRAHYDRO-IMIDAZO[1,5-A]PYRIDIN-1-YL)-5H-PYRROLO[2,3-B]PYRAZINE-7- CARBOXYLIC ACID TERT-BUTYLAMIDE | KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4xg8:A (GLY437) to (VAL634) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4xg8:C (GLY437) to (TYR629) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4xg9:A (GLY437) to (ASP632) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4xg9:B (GLY437) to (VAL634) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4i1z:A (HIS773) to (ARG973) CRYSTAL STRUCTURE OF THE MONOMERIC (V948R) FORM OF THE GEFITINIB/ERLOTINIB RESISTANT EGFR KINASE DOMAIN L858R+T790M | KINASE DOMAIN, PHOSPHOTRANSFER, ATP BINDING, TRANSFERASE
4i21:A (GLY779) to (ARG973) CRYSTAL STRUCTURE OF L858R + T790M EGFR KINASE DOMAIN IN COMPLEX WITH MIG6 PEPTIDE | EGFR KINASE DOMAIN, PHOSPHOTRANSFER, MIG6 PEPTIDE, ATP BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4i21:B (GLY779) to (ARG973) CRYSTAL STRUCTURE OF L858R + T790M EGFR KINASE DOMAIN IN COMPLEX WITH MIG6 PEPTIDE | EGFR KINASE DOMAIN, PHOSPHOTRANSFER, MIG6 PEPTIDE, ATP BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4i23:A (GLY779) to (ARG973) CRYSTAL STRUCTURE OF THE WILD-TYPE EGFR KINASE DOMAIN IN COMPLEX WITH DACOMITINIB (SOAKED) | KINASE DOMAIN, PHOSPHOTRANSFER, ATP BINDING, TRANSFERASE
2pvy:A (LEU551) to (LEU763) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC K659N MUTATION RESPONSIBLE FOR AN UNCLASSIFIED CRANIOSYNOSTOSIS SYNDROME. | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, TRANSFERASE
2pvy:D (LEU551) to (THR764) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC K659N MUTATION RESPONSIBLE FOR AN UNCLASSIFIED CRANIOSYNOSTOSIS SYNDROME. | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, TRANSFERASE
4xli:A (LEU348) to (SER546) CRYSTAL STRUCTURE OF ABL2/ARG KINASE IN COMPLEX WITH DASATINIB | TRANSFERASE, INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4xli:B (LEU348) to (SER546) CRYSTAL STRUCTURE OF ABL2/ARG KINASE IN COMPLEX WITH DASATINIB | TRANSFERASE, INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1opl:B (LEU321) to (GLU518) STRUCTURAL BASIS FOR THE AUTO-INHIBITION OF C-ABL TYROSINE KINASE | TRANSFERASE
3fqe:A (GLY437) to (HIS639) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH YM193306 | SYK, SPLEEN TYPROSINE KINASE, KINASE INHIBITOR, PYRIMIDINE-5- CARBOXAMIDE, ATP-BINDING, HOST-VIRUS INTERACTION, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
4id7:A (GLY194) to (GLN389) ACK1 KINASE IN COMPLEX WITH THE INHIBITOR CIS-3-[8-AMINO-1-(4- PHENOXYPHENYL)IMIDAZO[1,5-A]PYRAZIN-3-YL]CYCLOBUTANOL | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3srv:A (GLY437) to (VAL633) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE (SYK) IN COMPLEX WITH A DIAMINOPYRIMIDINE CARBOXAMIDE INHIBITOR | SK363, SYK, NON-RECEPTOR TYROSINE KINASE, SPLEEN TYROSINE KINASE, TRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3srv:B (GLY437) to (ASP632) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE (SYK) IN COMPLEX WITH A DIAMINOPYRIMIDINE CARBOXAMIDE INHIBITOR | SK363, SYK, NON-RECEPTOR TYROSINE KINASE, SPLEEN TYROSINE KINASE, TRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4xlv:A (GLY1064) to (LEU1262) CRYSTAL STRUCTURE OF THE ACTIVATED INSULIN RECEPTOR TYROSINE KINASE DIMER | TYROSINE KINASE, SIGNAL TRANSDUCTION, PHOSPHORYL TRANSFER, TRANSFERASE
3sxr:A (TYR476) to (ARG670) CRYSTAL STRUCTURE OF BMX NON-RECEPTOR TYROSINE KINASE COMPLEX WITH DASATINIB | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3sxr:B (TYR476) to (ARG670) CRYSTAL STRUCTURE OF BMX NON-RECEPTOR TYROSINE KINASE COMPLEX WITH DASATINIB | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3sxs:A (TYR476) to (ARG670) CRYSTAL STRUCTURE OF BMX NON-RECEPTOR TYROSINE KINASE COMPLEXED WITH PP2 | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4iwd:A (GLY1144) to (HIS1321) STRUCTURE OF DUALLY PHOSPHORYLATED C-MET RECEPTOR KINASE IN COMPLEX WITH AN MK-8033 ANALOG | PROTEIN KINASE, TYROSINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3gqi:A (ILE544) to (LEU760) CRYSTAL STRUCTURE OF ACTIVATED RECEPTOR TYROSINE KINASE IN COMPLEX WITH SUBSTRATES | PHOSPHORYLATED KINASE, PY-RECOGNITION, TANDEM SH2 DOMAINS, ATP ANALOG, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, DWARFISM, GLYCOPROTEIN, HEPARIN-BINDING, HYPOGONADOTROPIC HYPOGONADISM, IMMUNOGLOBULIN DOMAIN, KALLMANN SYNDROME, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, HYDROLASE, LIPID DEGRADATION, SH2 DOMAIN, SH3 DOMAIN, TRANSDUCER, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4j95:B (LEU551) to (THR762) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC K659N MUTATION RESPONSIBLE FOR AN UNCLASSIFIED CRANIOSYNOSTOSIS SYNDROME IN SPACE GROUP C2. | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, RECEPTOR TYROSINE KINASE, ATP BINDING, TRANSFERASE
4j95:C (LEU551) to (THR764) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC K659N MUTATION RESPONSIBLE FOR AN UNCLASSIFIED CRANIOSYNOSTOSIS SYNDROME IN SPACE GROUP C2. | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, RECEPTOR TYROSINE KINASE, ATP BINDING, TRANSFERASE
4j96:A (LEU551) to (ASN766) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC GAIN-OF-FUNCTION K659M MUTATION IDENTIFIED IN CERVICAL CANCER. | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, RECEPTOR TYROSINE KINASE, ATP BINDING, TRANSFERASE
4j97:A (LEU551) to (LEU763) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC GAIN-OF-FUNCTION K659E MUTATION IDENTIFIED IN ENDOMETRIAL CANCER. | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, RECEPTOR TYROSINE KINASE, ATP BINDING, TRANSFERASE
4j97:C (ILE547) to (LEU763) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC GAIN-OF-FUNCTION K659E MUTATION IDENTIFIED IN ENDOMETRIAL CANCER. | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, RECEPTOR TYROSINE KINASE, ATP BINDING, TRANSFERASE
4j97:D (GLY552) to (THR764) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC GAIN-OF-FUNCTION K659E MUTATION IDENTIFIED IN ENDOMETRIAL CANCER. | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, RECEPTOR TYROSINE KINASE, ATP BINDING, TRANSFERASE
4j99:B (LEU551) to (THR764) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE GAIN-OF-FUNCTION K659T MUTATION. | BILOBATE PROTEIN KINASE FOLD, RECEPTOR TYROSINE KINASE, ATP BINDING, TRANSFERASE
4j99:C (GLY552) to (THR764) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE GAIN-OF-FUNCTION K659T MUTATION. | BILOBATE PROTEIN KINASE FOLD, RECEPTOR TYROSINE KINASE, ATP BINDING, TRANSFERASE
2dq7:X (TYR70) to (ASP262) CRYSTAL STRUCTURE OF FYN KINASE DOMAIN COMPLEXED WITH STAUROSPORINE | SRC FAMILY, KINASE DOMAIN, STAUROSPORINE, TRANSFERASE
2rf9:A (LEU754) to (ARG949) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN THE EGFR KINASE DOMAIN AND A MIG6 PEPTIDE | KINASE DOMAIN, INHIBITION, DIMER, PEPTIDE, ALTERNATIVE SPLICING, ANTI-ONCOGENE, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, UBL CONJUGATION, CYTOPLASM
4jq7:A (GLY755) to (ARG949) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN IN COMPLEX WITH COMPOUND 2A | TRANSFERASE, TYROSINE KINASE DOMAIN, ATP-BINDING DOMAIN, AUTOPHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jq8:A (GLY755) to (ARG949) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN IN COMPLEX WITH COMPOUND 4B | TRANSFERASE, TYROSINE KINASE DOMAIN, ATP-BINDING DOMAIN, AUTOPHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jr3:A (GLY755) to (ARG949) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN IN COMPLEX WITH COMPOUND 3G | TRANSFERASE, TYROSINE KINASE DOMAIN, ATP-BINDING DOMAIN, AUTOPHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jrv:A (GLY755) to (ARG949) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN IN COMPLEX WITH COMPOUND 4C | TRANSFERASE, TYROSINE KINASE DOMAIN, ATP-BINDING DOMAIN, AUTOPHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yjo:A (GLY437) to (TYR630) THE KINASE DOMAIN OF HUMAN SPLEEN TYROSINE (SYK) IN COMPLEX WITH GTC000222 | SYK, NON-RECEPTOR TYROSINE KINASE, SPLEEN TYROSINE KINASE, TRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yjp:A (VAL433) to (ASP632) THE KINASE DOMAIN OF HUMAN SPLEEN TYROSINE (SYK) IN COMPLEX WITH GTC000223 | SYK, NON-RECEPTOR TYROSINE KINASE, SPLEEN TYROSINE KINASE, TRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yjq:A (GLY437) to (ARG627) SYK KINASE DOMAIN IN COMPLEX WITH INHIBITOR GTC000224 | SYK, NON-RECEPTOR TYROSINE KINASE, SPLEEN TYROSINE KINASE, TRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yjr:A (GLY437) to (ARG627) SYK KINASE DOMAIN IN COMPLEX WITH INHIBITOR GTC000225 | SYK, NON-RECEPTOR TYROSINE KINASE, SPLEEN TYROSINE KINASE, TRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yjs:A (GLY437) to (ASP632) THE KINASE DOMAIN OF HUMAN SPLEEN TYROSINE (SYK) IN COMPLEX WITH GTC000226 | SYK, NON-RECEPTOR TYROSINE KINASE, SPLEEN TYROSINE KINASE, TRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yjt:A (GLY437) to (ARG627) THE KINASE DOMAIN OF HUMAN SPLEEN TYROSINE (SYK) IN COMPLEX WITH GTC000233 | SYK, NON-RECEPTOR TYROSINE KINASE, SPLEEN TYROSINE KINASE, TRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yju:A (GLY437) to (TYR630) THE KINASE DOMAIN OF HUMAN SPLEEN TYROSINE (SYK) IN COMPLEX WITH GTC000249 | SYK, NON-RECEPTOR TYROSINE KINASE, SPLEEN TYROSINE KINASE, TRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yjv:A (GLY437) to (ARG627) THE KINASE DOMAIN OF HUMAN SPLEEN TYROSINE (SYK) IN COMPLEX WITH GTC000250 | SYK, NON-RECEPTOR TYROSINE KINASE, SPLEEN TYROSINE KINASE, TRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2eb2:A (GLY779) to (ARG973) CRYSTAL STRUCTURE OF MUTATED EGFR KINASE DOMAIN (G719S) | KINASE, TYROSINE-PROTEIN KINASE, RECEPTOR, TRANSFERASE, PHOSPHORYLATION, ATP-BINDING, DISEASE MUTATION, TRANSMEMBRANE, CELL CYCLE, EC 2.7.10.1, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
4k33:A (LEU551) to (THR755) CRYSTAL STRUCURE OF FGF RECEPTOR 3 (FGFR3) KINASE DOMAIN HARBORING THE K650E MUTATION, A GAIN-OF-FUNCTION MUTATION RESPONSIBLE FOR THANATOPHORIC DYSPLASIA TYPE II AND SPERMATOCYTIC SEMINOMA | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, RECEPTOR TYROSINE KINASE, TRANSFERASE
3ug1:A (GLY779) to (ARG973) CRYSTAL STRUCTURE OF THE MUTATED EGFR KINASE DOMAIN (G719S/T790M) IN THE APO FORM | KINASE, TYROSINE-PROTEIN KINASE, TRANSFERASE, ATP BINDING, PHOSPHORYLATION, TRANSMEMBRANE, RECEPTOR, DISEASE MUTATION, CELL CYCLE, DRUG RESISTANCE
3ug2:A (GLY779) to (PRO975) CRYSTAL STRUCTURE OF THE MUTATED EGFR KINASE DOMAIN (G719S/T790M) IN COMPLEX WITH GEFITINIB | KINASE, TYROSINE-PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSMEMBRANE, RECEPTOR, DISEASE MUTATION, CELL CYCLE, DRUG RESISTANCE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2fo0:A (LEU317) to (THR514) ORGANIZATION OF THE SH3-SH2 UNIT IN ACTIVE AND INACTIVE FORMS OF THE C-ABL TYROSINE KINASE | N-TERMINAL CAP, AUTOINHIBITION, MYRISTOYLATION, SH3-SH2 CLAMP, PHOSPHOSERINE, TRANSFERASE
4zau:A (GLY779) to (ARG973) AZD9291 COMPLEX WITH WILD TYPE EGFR | TRANSFERASE, KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3vf9:A (GLY437) to (VAL634) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE SYK CATALYTIC DOMAIN WITH THIENOPYRAZOLYLINDOLE INHIBITOR 027 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3vf8:A (GLY437) to (ASN635) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE SYK CATALYTIC DOMAIN WITH PYRAZOLYLBENZIMIDAZOLE INHIBITOR 416 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1h24:A (ASP68) to (GLN287) CDK2/CYCLIN A IN COMPLEX WITH A 9 RESIDUE RECRUITMENT PEPTIDE FROM E2F | TRANSFERASE, CELL CYCLE, PROTEIN KINASE, CYCLIN, CDK2, RECRUITMENT, PEPTIDE SPECIFICITY, SERINE/THREONINE-PROTEIN KINASE, ATP- BINDING, CELL DIVISION, MITOSIS, PHOSPHORYLATION
2gs2:A (GLY755) to (ARG949) CRYSTAL STRUCTURE OF THE ACTIVE EGFR KINASE DOMAIN | EGFR, KINASE, ACTIVE, TRANSFERASE
2gs6:A (GLY755) to (ARG949) CRYSTAL STRUCTURE OF THE ACTIVE EGFR KINASE DOMAIN IN COMPLEX WITH AN ATP ANALOG-PEPTIDE CONJUGATE | EGFR, KINASE,ACTIVE, ATP-ANALOG PEPTIDE CONJUGATE, TRANSFERASE
2w4j:A (GLU81) to (GLN271) X-RAY STRUCTURE OF A DAP-KINASE 2-277 | POLYMORPHISM, PHOSPHOPROTEIN, CALMODULIN-BINDING, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, ALTERNATIVE SPLICING, DAPK, KINASE, COMPLEX, APOPTOSIS, CYTOPLASM, ANK REPEAT, CALMODULIN, TRANSFERASE, ATP-BINDING
4li5:A (GLY779) to (ARG973) EGFR-K IN COMPLEX WITH N-[3-[[5-CHLORO-4-(1H-INDOL-3-YL)PYRIMIDIN-2- YL]AMINO]-4-METHOXY-PHENYL] PROP-2-ENAMIDE | EGF RECEPTOR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4lrm:B (GLY782) to (ARG976) EGFR D770_N771INSNPG IN COMPLEX WITH PD168393 | EGFR, KINASE, PD168393, 34-JAB, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4lrm:C (GLY782) to (ARG976) EGFR D770_N771INSNPG IN COMPLEX WITH PD168393 | EGFR, KINASE, PD168393, 34-JAB, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4lrm:E (GLY782) to (ARG976) EGFR D770_N771INSNPG IN COMPLEX WITH PD168393 | EGFR, KINASE, PD168393, 34-JAB, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1u4d:A (GLY194) to (GLN389) STRUCTURE OF THE ACK1 KINASE DOMAIN BOUND TO DEBROMOHYMENIALDISINE | TYROSINE KINASE, TRANSFERASE
1u4d:B (GLY194) to (ALA388) STRUCTURE OF THE ACK1 KINASE DOMAIN BOUND TO DEBROMOHYMENIALDISINE | TYROSINE KINASE, TRANSFERASE
1u54:A (GLY194) to (ALA388) CRYSTAL STRUCTURES OF THE PHOSPHORYLATED AND UNPHOSPHORYLATED KINASE DOMAINS OF THE CDC42-ASSOCIATED TYROSINE KINASE ACK1 BOUND TO AMP-PCP | TYROSINE KINASE, TRANSFERASE
1u54:B (GLY194) to (ALA388) CRYSTAL STRUCTURES OF THE PHOSPHORYLATED AND UNPHOSPHORYLATED KINASE DOMAINS OF THE CDC42-ASSOCIATED TYROSINE KINASE ACK1 BOUND TO AMP-PCP | TYROSINE KINASE, TRANSFERASE
3w2o:A (GLY779) to (ARG973) EGFR KINASE DOMAIN T790M/L858R MUTANT WITH TAK-285 | ANTI-ONCOGENE, CELL CYCLE, DISEASE MUTATION, KINASE DOMAIN, RECEPTOR, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3w2p:A (GLY779) to (ARG973) EGFR KINASE DOMAIN T790M/L858R MUTANT WITH COMPOUND 2 | ANTI-ONCOGENE, CELL CYCLE, DISEASE MUTATION, KINASE DOMAIN, RECEPTOR, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3w2q:A (GLY779) to (ARG973) EGFR KINASE DOMAIN T790M/L858R MUTANT WITH HKI-272 | ANTI-ONCOGENE, CELL CYCLE, DISEASE MUTATION, KINASE DOMAIN, RECEPTOR, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2hz4:B (LEU302) to (GLN498) ABL KINASE DOMAIN UNLIGATED AND IN COMPLEX WITH TETRAHYDROSTAUROSPORINE | TYROSINE KINASE, TRANSFERASE
2x2l:A (TYR791) to (MET1009) CRYSTAL STRUCTURE OF PHOSPHORYLATED RET TYROSINE KINASE DOMAIN WITH INHIBITOR | HIRSCHSPRUNG DISEASE, GDNF RECEPTOR, TRANSMEMBRANE, PROTO-ONCOGENE, PHOSPHOPROTEIN, DISEASE MUTATION, PHOSPHOTRANSFERASE, RET, KINASE, MEMBRANE, TRANSFERASE
2x2m:A (TYR791) to (ARG1013) CRYSTAL STRUCTURE OF PHOSPHORYLATED RET TYROSINE KINASE DOMAIN WITH INHIBITOR | HIRSCHSPRUNG DISEASE, GDNF RECEPTOR, TRANSMEMBRANE, PROTO-ONCOGENE, PHOSPHOPROTEIN, DISEASE MUTATION, PHOSPHOTRANSFERASE, RET, KINASE, MEMBRANE, TRANSFERASE
2x2m:B (ILE788) to (LYS1011) CRYSTAL STRUCTURE OF PHOSPHORYLATED RET TYROSINE KINASE DOMAIN WITH INHIBITOR | HIRSCHSPRUNG DISEASE, GDNF RECEPTOR, TRANSMEMBRANE, PROTO-ONCOGENE, PHOSPHOPROTEIN, DISEASE MUTATION, PHOSPHOTRANSFERASE, RET, KINASE, MEMBRANE, TRANSFERASE
2itp:A (GLY779) to (ARG973) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN G719S MUTATION IN COMPLEX WITH AEE788 | RECEPTOR, CELL CYCLE, ATP-BINDING, TRANSFERASE, TRANSMEMBRANE, PHOSPHORYLATION, DISEASE MUTATION, POLYMORPHISM, GLYCOPROTEIN, ANTI-ONCOGENE, NUCLEOTIDE- BINDING, ALTERNATIVE SPLICING, AEE788, EGFR, G719S, KINASE, MEMBRANE, TYROSINE-PROTEIN KINASE, EPIDERMAL GROWTH FACTOR
2itq:A (GLY779) to (ARG973) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN G719S MUTATION IN COMPLEX WITH AFN941 | RECEPTOR, CELL CYCLE, ATP-BINDING, TRANSFERASE, TRANSMEMBRANE, PHOSPHORYLATION, DISEASE MUTATION, POLYMORPHISM, GLYCOPROTEIN, ANTI-ONCOGENE, NUCLEOTIDE- BINDING, ALTERNATIVE SPLICING, AFN941, EGFR, G719S, STAUROSPORINE, MEMBRANE, TYROSINE-PROTEIN KINASE, EPIDERMAL GROWTH FACTOR
2ivs:A (VAL787) to (ARG1012) CRYSTAL STRUCTURE OF NON-PHOSPHORYLATED RET TYROSINE KINASE DOMAIN | NUCLEOTIDE-BINDING, HIRSCHSPRUNG DISEASE, PHOSPHORYLATION, DISEASE MUTATION, PHOSPHOTRANSFERASE, TYROSINE-PROTEIN KINASE, CHROMOSOMAL TRANSLOCATION, POLYMORPHISM, GDNF RECEPTOR, TRANSMEMBRANE, PROTO-ONCOGENE, TYROSINE KINASE, RET, KINASE, MEMBRANE, ATP-BINDING, TRANSFERASE
2ivt:A (VAL787) to (ARG1012) CRYSTAL STRUCTURE OF PHOSPHORYLATED RET TYROSINE KINASE DOMAIN | NUCLEOTIDE-BINDING, HIRSCHSPRUNG DISEASE, PHOSPHORYLATION, DISEASE MUTATION, PHOSPHOTRANSFERASE, TYROSINE-PROTEIN KINASE, CHROMOSOMAL TRANSLOCATION, POLYMORPHISM, GDNF RECEPTOR, TRANSMEMBRANE, PROTO-ONCOGENE, TYROSINE KINASE, RET, KINASE, MEMBRANE, ATP-BINDING, TRANSFERASE
2ivu:A (GLY792) to (ARG1012) CRYSTAL STRUCTURE OF PHOSPHORYLATED RET TYROSINE KINASE DOMAIN COMPLEXED WITH THE INHIBITOR ZD6474 | NUCLEOTIDE-BINDING, HIRSCHSPRUNG DISEASE, PHOSPHORYLATION, DISEASE MUTATION, PHOSPHOTRANSFERASE, TYROSINE-PROTEIN KINASE, CHROMOSOMAL TRANSLOCATION, POLYMORPHISM, GDNF RECEPTOR, TRANSMEMBRANE, PROTO-ONCOGENE, TYROSINE KINASE, RET, KINASE, MEMBRANE, ATP-BINDING, TRANSFERASE
2ivv:A (TYR791) to (LYS1011) CRYSTAL STRUCTURE OF PHOSPHORYLATED RET TYROSINE KINASE DOMAIN COMPLEXED WITH THE INHIBITOR PP1 | NUCLEOTIDE-BINDING, HIRSCHSPRUNG DISEASE, PHOSPHORYLATION, DISEASE MUTATION, PHOSPHOTRANSFERASE, TYROSINE-PROTEIN KINASE, CHROMOSOMAL TRANSLOCATION, POLYMORPHISM, GDNF RECEPTOR, TRANSMEMBRANE, PROTO-ONCOGENE, TYROSINE KINASE, RET, KINASE, MEMBRANE, ATP-BINDING, TRANSFERASE
5amn:A (GLY792) to (VAL1010) THE DISCOVERY OF 2-SUBSTITUTED PHENOL QUINAZOLINES AS POTENT AND SELECTIVE RET KINASE INHIBITORS | TRANSFERASE, RET, ONCOGENE, RECEPTOR TYROSINE KINASE, CHEMICAL INHIBITOR, CANCER
2j5e:A (GLY779) to (ARG973) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN IN COMPLEX WITH AN IRREVERSIBLE INHIBITOR 13-JAB | CELL CYCLE, ATP-BINDING, TRANSFERASE, POLYMORPHISM, IRREVERSIBLE INHIBITOR, TYROSINE-PROTEIN KINASE, EGFR, KINASE, 13-JAB, MEMBRANE, RECEPTOR, WILD-TYPE, EPIDERMAL GROWTH FACTOR, ANTI-ONCOGENE, TRANSMEMBRANE, NUCLEOTIDE- BINDING, ALTERNATIVE SPLICING, UBL CONJUGATION, PHOSPHORYLATION, DISEASE MUTATION, GLYCOPROTEIN
3zew:A (GLU680) to (ASN880) CRYSTAL STRUCTURE OF EPHB4 IN COMPLEX WITH STAUROSPORINE | TRANSFERASE, INHIBITOR
2jit:A (GLY779) to (ARG973) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN T790M MUTATION | EGFR, T790M, KINASE, RECEPTOR, CELL CYCLE, PHOSPHORYLATION, DISEASE MUTATION, NUCLEOTIDE-BINDING, TYROSINE-PROTEIN KINASE, ANTI-ONCOGENE, EPIDERMAL GROWTH FACTOR, ATP-BINDING, TRANSFERASE
2jiu:A (GLY779) to (ARG973) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN T790M MUTATION IN COMPLEX WITH AEE788 | CELL CYCLE, ATP-BINDING, TRANSFERASE, NUCLEOTIDE-BINDING, ALTERNATIVE SPLICING, EGFR, T790M, KINASE, AEE788, RECEPTOR, TYROSINE-PROTEIN KINASE, EPIDERMAL GROWTH FACTOR, PHOSPHORYLATION, DISEASE MUTATION, ANTI-ONCOGENE, TRANSMEMBRANE
2jiu:B (GLY779) to (ARG973) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN T790M MUTATION IN COMPLEX WITH AEE788 | CELL CYCLE, ATP-BINDING, TRANSFERASE, NUCLEOTIDE-BINDING, ALTERNATIVE SPLICING, EGFR, T790M, KINASE, AEE788, RECEPTOR, TYROSINE-PROTEIN KINASE, EPIDERMAL GROWTH FACTOR, PHOSPHORYLATION, DISEASE MUTATION, ANTI-ONCOGENE, TRANSMEMBRANE
5c26:A (GLY437) to (HIS636) CRYSTAL STRUCTURE OF SYK IN COMPLEX WITH COMPOUND 1 | SPLEEN TYROSINE KINASE, INHIBITOR, TRANSFERASE-INHIBITOR COMPLEX
5c27:A (GLY437) to (ASN635) CRYSTAL STRUCTURE OF SYK IN COMPLEX WITH COMPOUND 2 | SPLEEN TYROSINE KINASE, INHIBITOR, TRANSFERASE-INHIBITOR COMPLEX
1xba:A (GLY437) to (GLU636) CRYSTAL STRUCTURE OF APO SYK TYROSINE KINASE DOMAIN | SPLEEN TYPROSINE KINASE, ACTIVE CONFORMATION, STRUCTURAL GENOMICS, STRUCTURAL GENOMIX, TRANSFERASE
1xbb:A (GLY437) to (HIS639) CRYSTAL STRUCTURE OF THE SYK TYROSINE KINASE DOMAIN WITH GLEEVEC | GLEEVEC, STI-571, IMATINIB, SYK, SPLEEN TYPROSINE KINASE, ACTIVE CONFORMATION, STRUCTURAL GENOMICS, STRUCTURAL GENOMIX, TRANSFERASE
1xbc:A (GLY437) to (GLU636) CRYSTAL STRUCTURE OF THE SYK TYROSINE KINASE DOMAIN WITH STAUROSPORIN | STAUROSPORINE, SYK, SPLEEN TYPROSINE KINASE, ACTIVE CONFORMATION, STRUCTURAL GENOMICS, STRUCTURAL GENOMIX, TRANSFERASE
5cav:A (GLY779) to (ARG973) EGFR KINASE DOMAIN WITH COMPOUND 41A | PROTEIN KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1m14:A (GLY755) to (ARG949) TYROSINE KINASE DOMAIN FROM EPIDERMAL GROWTH FACTOR RECEPTOR | TRANSFERASE, TYROSINE KINASE DOMAIN
1m17:A (GLY755) to (ARG949) EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE DOMAIN WITH 4-ANILINOQUINAZOLINE INHIBITOR ERLOTINIB | TRANSFERASE, TYROSINE KINASE DOMAIN
5cxh:A (GLY437) to (HIS639) SYK CATALYTIC DOMAIN COMPLEXED WITH A POTENT ORALLY BIOAVAILABLE THIAZOLE INHIBITOR | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5cxz:A (GLY437) to (HIS636) SYK CATALYTIC DOMAIN COMPLEXED WITH NAPHTHYRIDINE INHIBITOR | TRANSFERASE/TRANSFERASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5cy3:A (GLY437) to (GLY637) SYK CATALYTIC DOMAIN COMPLEXED WITH A POTENT AND ORALLY BIOAVAILABLE BENZISOTHIAZOLE INHIBITOR | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5czh:A (GLY779) to (ARG973) EGFR L858R MUTANT IN COMPLEX WITH AN OPTIMAL PEPTIDE SUBSTRATE | EGFR, L858R, KINASE, EGF, TRANSFERASE
5czi:A (GLY779) to (ARG973) EGFR L858R MUTANT IN COMPLEX WITH A SHC PEPTIDE SUBSTRATE | EGFR, L858R, KINASE, EGF, TRANSFERASE
3krr:A (VAL916) to (ASN1107) CRYSTAL STRUCTURE OF JAK2 COMPLEXED WITH A POTENT QUINOXALINE ATP SITE INHIBITOR | SMALL MOLECULE INHIBITOR, ATP SITE KINASE INHIBITOR, ATP-BINDING, DISEASE MUTATION, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE
3kul:B (GLY701) to (PRO899) KINASE DOMAIN OF HUMAN EPHRIN TYPE-A RECEPTOR 8 (EPHA8) | ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, RECEPTOR, TRANSFERASE, PHOSPHORYLATION, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, GLYCOPROTEIN, MEMBRANE, PHOSPHOPROTEIN
3kxx:C (GLY549) to (LEU760) STRUCTURE OF THE MUTANT FIBROBLAST GROWTH FACTOR RECEPTOR 1 | KINASE, RTK, INTERFACE, PHOSPHORYLATION, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, DWARFISM, GLYCOPROTEIN, HEPARIN-BINDING, HYPOGONADOTROPIC HYPOGONADISM, IMMUNOGLOBULIN DOMAIN, KALLMANN SYNDROME, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3kxx:D (GLY549) to (SER762) STRUCTURE OF THE MUTANT FIBROBLAST GROWTH FACTOR RECEPTOR 1 | KINASE, RTK, INTERFACE, PHOSPHORYLATION, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, DWARFISM, GLYCOPROTEIN, HEPARIN-BINDING, HYPOGONADOTROPIC HYPOGONADISM, IMMUNOGLOBULIN DOMAIN, KALLMANN SYNDROME, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3lcd:A (LEU650) to (GLN913) INHIBITOR BOUND TO A DFG-IN STRUCTURE OF THE KINASE DOMAIN OF CSF-1R | KINASE CFMS CSF-1R CSF TYROSINE-KINASE COLONY STIMULATING FACTOR 1 RECEPTOR, ATP-BINDING, DISULFIDE BOND, GLYCOPROTEIN, IMMUNOGLOBULIN DOMAIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
4puz:A (GLY437) to (VAL633) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE (SYK) IN COMPLEX WITH GS- 9973 | SYK, SPLEEN TYROSINE KINASE, KINASE INHIBITOR, PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4puz:B (GLY437) to (VAL634) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE (SYK) IN COMPLEX WITH GS- 9973 | SYK, SPLEEN TYROSINE KINASE, KINASE INHIBITOR, PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4pv0:A (GLY437) to (GLU636) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE (SYK) IN COMPLEX WITH AN IMIDAZOPYRAZINE INHIBITOR | SYK, SPLEEN TYROSINE KINASE, KINASE INHIBITOR, PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4px6:A (GLY437) to (ASN635) SYK CATALYTIC DOMAIN IN COMPLEX WITH A POTENT PYRIDOPYRIMIDINONE INHIBITOR | KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5eg3:A (LEU551) to (GLU767) CRYSTAL STRUCURE OF THE ACTIVATED FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN IN COMPLEX WITH THE CSH2 DOMAIN OF PHOSPHOLIPASE C GAMMA (PLCGAMMA) | SIGNALING COMPLEX, TYROSINE KINASE DOMAIN, SH2 DOMAIN, RECRUITMENT, PHOSPHORYLATION, TRANSFERASE-HYDROLASE COMPLEX
5em8:A (GLY779) to (ARG973) EGFR KINASE DOMAIN WITH PYRIDONE COMPOUND 13: 4-[(2-METHOXYPHENYL) AMINO]-~{N}-[4-(4-METHYLPIPERAZIN-1-YL)PHENYL]-2-OXIDANYLIDENE-1~{H}- PYRIDINE-3-CARBOXAMIDE | PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3bce:A (GLY760) to (PRO956) CRYSTAL STRUCTURE OF THE ERBB4 KINASE | ACTIVE CONFORMATION, ATP-BINDING, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3bce:B (GLY760) to (ARG954) CRYSTAL STRUCTURE OF THE ERBB4 KINASE | ACTIVE CONFORMATION, ATP-BINDING, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3bce:C (GLY760) to (PRO956) CRYSTAL STRUCTURE OF THE ERBB4 KINASE | ACTIVE CONFORMATION, ATP-BINDING, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3bu3:A (LEU1063) to (LEU1263) CRYSTAL STRUCTURE OF THE INSULIN RECEPTOR KINASE IN COMPLEX WITH IRS2 KRLB PEPTIDE | IRK, KRLB, IRS2, INSULIN RECEPTOR, PEPTIDE, SUBSTRATE, ALTERNATIVE SPLICING, ATP-BINDING, CARBOHYDRATE METABOLISM, CLEAVAGE ON PAIR OF BASIC RESIDUES, DIABETES MELLITUS, DISEASE MUTATION, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, TRANSDUCER
3c0g:B (GLU79) to (HIS273) CASK CAM-KINASE DOMAIN- 3'-AMP COMPLEX, P1 FORM | CASK, NEUREXIN, CA2+/CALMODULIN DEPENDENT PROTEIN KINASE, MG2+, SYNAPTIC PLASTICITY, PSEUDOKINASE, MAGUK, MEMBRANE-ASSOCIATED GUANYLATE KINASE, ATP-BINDING, CALMODULIN-BINDING, MAGNESIUM, METAL- BINDING, NUCLEOTIDE-BINDING, NUCLEUS, SERINE/THREONINE-PROTEIN KINASE, SH3 DOMAIN, TRANSFERASE
5fed:A (GLY779) to (ARG973) EGFR KINASE DOMAIN IN COMPLEX WITH A COVALENT AMINOBENZIMIDAZOLE INHIBITOR. | KINASE, INHIBITOR, COVALENTLY-BOUND, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4r3p:A (GLY779) to (ARG973) CRYSTAL STRUCTURES OF EGFR IN COMPLEX WITH MIG6 | KINASE, MIG6, PHOSPHORYLATION, TRANSFERASE
4r3r:A (GLY779) to (ARG973) CRYSTAL STRUCTURES OF EGFR IN COMPLEX WITH MIG6 | KINASE, PHOPHORYLATION, ATP HYDROLYSIS, MIG6, PHOSPHORYLATION, TRANSFERASE
5flf:A (LEU548) to (THR761) DISEASE LINKED MUTATION IN FGFR | TRANSFERASE, AUTO-ACTIVATING, CANCER, GROWTH FACTOR, RECEPTOR, MUTATION;
5flf:B (LEU548) to (LEU760) DISEASE LINKED MUTATION IN FGFR | TRANSFERASE, AUTO-ACTIVATING, CANCER, GROWTH FACTOR, RECEPTOR, MUTATION;
5flf:C (LEU548) to (LEU760) DISEASE LINKED MUTATION IN FGFR | TRANSFERASE, AUTO-ACTIVATING, CANCER, GROWTH FACTOR, RECEPTOR, MUTATION;
5flf:D (LEU548) to (LEU760) DISEASE LINKED MUTATION IN FGFR | TRANSFERASE, AUTO-ACTIVATING, CANCER, GROWTH FACTOR, RECEPTOR, MUTATION;
3cly:A (LEU1551) to (GLU1768) CRYSTAL STRUCTURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAINS TRAPPED IN TRANS-PHOSPHORYLATION REACTION | KINASE DOMAIN, TRANS-PHOSPHORYLATION, ATP-BINDING, DISEASE MUTATION, ECTODERMAL DYSPLASIA, GLYCOPROTEIN, HEPARIN-BINDING, IMMUNOGLOBULIN DOMAIN, LACRIMO-AURICULO-DENTO-DIGITAL SYNDROME, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
4riw:B (GLY755) to (ALA948) CRYSTAL STRUCTURE OF AN EGFR/HER3 KINASE DOMAIN HETERODIMER | RECEPTOR TYROSINE KINASE, PSEUDOKINASE, KINASE, ATP BINDING, MEMBRANE, TRANSFERASE
4riw:D (GLY755) to (ARG949) CRYSTAL STRUCTURE OF AN EGFR/HER3 KINASE DOMAIN HETERODIMER | RECEPTOR TYROSINE KINASE, PSEUDOKINASE, KINASE, ATP BINDING, MEMBRANE, TRANSFERASE
4rix:B (GLY755) to (ARG949) CRYSTAL STRUCTURE OF AN EGFR/HER3 KINASE DOMAIN HETERODIMER CONTAINING THE CANCER-ASSOCIATED HER3-Q790R MUTATION | RECEPTOR TYROSINE KINASE, PSEUDOKINASE, KINASE, ATP BINDING, MEMBRANE, TRANSFERASE
4riy:B (GLY755) to (ALA948) CRYSTAL STRUCTURE OF AN EGFR/HER3 KINASE DOMAIN HETERODIMER CONTAINING THE CANCER-ASSOCIATED HER3-E909G MUTATION | RECEPTOR TYROSINE KINASE, PSEUDOKINASE, KINASE, ATP BINDING, MEMBRANE, TRANSFERASE
4riy:D (GLY755) to (ALA948) CRYSTAL STRUCTURE OF AN EGFR/HER3 KINASE DOMAIN HETERODIMER CONTAINING THE CANCER-ASSOCIATED HER3-E909G MUTATION | RECEPTOR TYROSINE KINASE, PSEUDOKINASE, KINASE, ATP BINDING, MEMBRANE, TRANSFERASE
4rss:A (GLY437) to (VAL633) CRYSTAL STRUCTURE OF TYROSINE-PROTEIN KINASE SYK WITH AN INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4cki:A (VAL787) to (ARG1013) CRYSTAL STRUCTURE OF ONCOGENIC RET TYROSINE KINASE M918T BOUND TO ADENOSINE | TRANSFERASE
4ckj:A (TYR791) to (ARG1013) CRYSTAL STRUCTURE OF RET TYROSINE KINASE DOMAIN BOUND TO ADENOSINE | TRANSFERASE
4rx7:A (GLY437) to (HIS637) SYK CATALYTIC DOMAIN COMPLEXED WITH A POTENT TRIAZINE INHIBITOR | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4rx8:A (GLY437) to (HIS638) SYK CATALYTIC DOMAIN COMPLEXED WITH A POTENT TRIAZINE INHIBITOR2 | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4rx9:A (GLY437) to (HIS639) SYK CATALYTIC DOMAIN COMPLEXED WITH A POTENT PYRIMIDINE INHIBITOR | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4tks:A (GLY779) to (ARG973) NATIVE-SAD PHASING FOR HUMAN EGFR KINASE DOMAIN. | EGFR KINASE DOMAIN, NATIVE-SAD PHASING, MULTIPLE CRYSTALS, LOW ENERGY
4trl:A (GLU679) to (ILE875) STRUCTURE OF EPHRIN TYPE-A RECEPTOR 2 | ACTIVE STATE, PHOSPHORYLATED
5ghv:A (GLY437) to (ASN635) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5ghv:B (GLY437) to (ASN635) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3dqw:C (TYR326) to (TYR519) C-SRC KINASE DOMAIN THR338ILE MUTANT IN COMPLEX WITH ATPGS | SRC, KINASE, ACTIVE, GATEKEEPER, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
4dfl:A (GLY437) to (GLU636) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH A SULFONAMIDOPYRAZINE PIPERIDINE INHIBITOR | SYK, TRANSFERASE, KINASE, INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4dfn:A (GLY437) to (VAL634) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH AN ADAMANTYLPYRAZINE INHIBITOR | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hg5:A (GLY779) to (ARG973) EGFR (L858R, T790M, V948R) IN COMPLEX WITH N-{3-[(2-{[4-(4- METHYLPIPERAZIN-1-YL)PHENYL]AMINO}-7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL) OXY]PHENYL}PROP-2-ENAMIDE | EGFR, INHIBITOR, COMPLEX, LUNG CANCER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hg8:A (GLY779) to (ARG973) EGFR (L858R, T790M, V948R) IN COMPLEX WITH N-[3-({2-[(1-METHYL-1H- PYRAZOL-4-YL)AMINO]-7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL}OXY)PHENYL]PROP- 2-ENAMIDE | EGFR, KINASE, INHIBITOR, LUNG CANCER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hg9:A (GLY779) to (ARG973) EGFR (L858R, T790M, V948R) IN COMPLEX WITH 1-[(3R,4R)-3-[({2-[(1- METHYL-1H-PYRAZOL-4-YL)AMINO]-7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL}OXY) METHYL]-4-(TRIFLUOROMETHYL)PYRROLIDIN-1-YL]PROP-2-EN-1-ONE | EGFR, KINASE, INHIBITOR, LUNG CANCER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hib:A (GLY779) to (ARG973) EGFR KINASE DOMAIN MUTANT "TMLR" WITH A PYRAZOLOPYRIMIDINE INHIBITOR | PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3pp0:A (GLY787) to (ARG981) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN HER2 (ERBB2). | KINASE DOMAIN, ANTI-ONCOGENE, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, TYROSINE KINASE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3pp0:B (GLY787) to (ASP982) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN HER2 (ERBB2). | KINASE DOMAIN, ANTI-ONCOGENE, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, TYROSINE KINASE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4ewh:A (GLY194) to (ALA388) CO-CRYSTAL STRUCTURE OF ACK1 WITH INHIBITOR | DRUG DESIGN, ENZYME INHIBITORS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4f4p:A (GLY437) to (GLY637) SYK IN COMPLEX WITH LIGAND LASW836 | TYROSINE-PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fk6:B (ILE937) to (GLU1133) JAK1 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 72 | PROTEIN KINASE, PHOSPHO TRANSFER, PHOSPHO TYROSINE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4fl1:A (GLY437) to (ASN635) STRUCTURAL AND BIOPHYSICAL CHARACTERIZATION OF THE SYK ACTIVATION SWITCH | TRANSFERASE, PROTEIN KINASE
5j9y:A (GLY779) to (ARG973) EGFR-T790M IN COMPLEX WITH PYRAZOLOPYRIMIDINE INHIBITOR 1B | TYROSINE KINASE, COVALENT INHIBITOR, DRUG RESISTANCE, TRANSFERASE
4fyn:A (GLY437) to (HIS639) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH 3-(8-{4- [ETHYL-(2-HYDROXY-ETHYL)-AMINO]-PHENYLAMINO}-IMIDAZO[1,2-A]PYRAZIN-5- YL)-PHENOL | KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fyo:A (GLY437) to (HIS639) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH N-{(S)-1- [7-(3,4-DIMETHOXY-PHENYLAMINO)-THIAZOLO[5,4-D]PYRIMIDIN-5-YL]- PYRROLIDIN-3-YL}-TEREPHTHALAMIC ACID | KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fz6:A (GLY437) to (HIS639) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH [6-((S)-2- METHYL-PYRROLIDIN-1-YL)-PYRIDIN-2-YL]-(6-PHENYL-IMIDAZO[1,2- B]PYRIDAZIN-8-YL)-AMINE | KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fz7:A (GLY437) to (HIS639) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH 6-((1R,2S)- 2-AMINO-CYCLOHEXYLAMINO)-4-(6-ETHYL-PYRIDIN-2-YLAMINO)-PYRIDAZINE-3- CARBOXYLIC ACID AMIDE | KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4g5j:A (GLY779) to (ARG973) CRYSTAL STRUCTURE OF EGFR KINASE IN COMPLEX WITH BIBW2992 | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4g5p:A (GLY779) to (PRO975) CRYSTAL STRUCTURE OF EGFR KINASE T790M IN COMPLEX WITH BIBW2992 | EGF RECEPTOR KINASE MUTANT T790M, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4g5p:B (VAL774) to (ARG973) CRYSTAL STRUCTURE OF EGFR KINASE T790M IN COMPLEX WITH BIBW2992 | EGF RECEPTOR KINASE MUTANT T790M, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gfm:A (VAL916) to (ASN1107) JAK2 KINASE (JH1 DOMAIN) WITH 2,6-DICHLORO-N-(2-OXO-2,5- DIHYDROPYRIDIN-4-YL)BENZAMIDE | O-PHOSPHOTYROSINE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5lma:A (GLY437) to (ASP632) HUMAN SPLEEN TYROSINE KINASE KINASE DOMAIN IN COMPLEX WITH AZANAPHTHYRIDINE INHIBITOR | INHIBITOR, COMPLEX, KINASE, TRANSFERASE
5lmb:A (GLY437) to (VAL634) HUMAN SPLEEN TYROSINE KINASE KINASE DOMAIN IN COMPLEX WITH AZANAPHTHYRIDINE INHIBITOR | INHIBITOR, COMPLEX, KINASE, TRANSFERASE
5lmb:B (GLY437) to (TYR630) HUMAN SPLEEN TYROSINE KINASE KINASE DOMAIN IN COMPLEX WITH AZANAPHTHYRIDINE INHIBITOR | INHIBITOR, COMPLEX, KINASE, TRANSFERASE
5t68:A (GLY437) to (GLU636) CRYSTAL STRUCTURE OF SYK CATALYTIC DOMAIN IN COMPLEX WITH A FURO[3,2- D]PYRIMIDINE | SPLEEN TYROSINE KINASE SYK CATALYTIC DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5t68:B (GLY437) to (ASN635) CRYSTAL STRUCTURE OF SYK CATALYTIC DOMAIN IN COMPLEX WITH A FURO[3,2- D]PYRIMIDINE | SPLEEN TYROSINE KINASE SYK CATALYTIC DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5tr6:A (GLY437) to (HIS639) DISCOVERY OF TAK-659, AN ORALLY AVAILABLE INVESTIGATIONAL INHIBITOR OF SPLEEN TYROSINE KINASE (SYK) | INHIBITOR, KINASE, LEUKEMIA, LYMPHOMA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5tt7:A (GLY437) to (HIS639) DISCOVERY OF TAK-659, AN ORALLY AVAILABLE INVESTIGATIONAL INHIBITOR OF SPLEEN TYROSINE KINASE (SYK) | INHIBITOR, KINASE, LEUKEMIA, LYMPHOMA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4wnm:A (GLY437) to (VAL633) SYK CATALYTIC DOMAIN IN COMPLEX WITH A POTENT TRIAZOLOPYRIDINE INHIBITOR | SYK CATALYTIC DOMAIN IN COMPLEX WITH A POTENT TRIAZOLOPYRIDINE BASED INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3fqh:A (GLY437) to (VAL634) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH A 2-SUBSTITUTED 7-AZAINDOLE | SYK, SPLEEN TYPROSINE KINASE, KINASE INHIBITOR, 7-AZAINDOLE, ALTERNATIVE SPLICING, ATP-BINDING, HOST-VIRUS INTERACTION, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, UBL CONJUGATION
3fqh:B (GLY437) to (VAL633) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH A 2-SUBSTITUTED 7-AZAINDOLE | SYK, SPLEEN TYPROSINE KINASE, KINASE INHIBITOR, 7-AZAINDOLE, ALTERNATIVE SPLICING, ATP-BINDING, HOST-VIRUS INTERACTION, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, UBL CONJUGATION
3fqs:A (GLY437) to (HIS639) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH R406 | SYK, SPLEEN TYPROSINE KINASE, KINASE INHIBITOR, R406, R788, AMINO- PYRIMIDINE, ATP-BINDING, HOST-VIRUS INTERACTION, KINASE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
2qoh:B (LEU302) to (LEU510) CRYSTAL STRUCTURE OF ABL KINASE BOUND WITH PPY-A | ABL, KINASE, INHIBITOR, TRANSFERASE
4j98:A (LEU551) to (THR764) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE GAIN-OF-FUNCTION K659Q MUTATION. | FGF RECEPTOR, RECEPTOR TYROSINE KINASE, GAIN-OF-FUNCTION MUTATION, ATP BINDING, TRANSFERASE
4j98:B (LEU551) to (THR764) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE GAIN-OF-FUNCTION K659Q MUTATION. | FGF RECEPTOR, RECEPTOR TYROSINE KINASE, GAIN-OF-FUNCTION MUTATION, ATP BINDING, TRANSFERASE
2g2f:A (LEU302) to (VAL506) A SRC-LIKE INACTIVE CONFORMATION IN THE ABL TYROSINE KINASE DOMAIN | PROTEIN KINASE, TRANSFERASE
4zjv:A (HIS773) to (ARG973) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN IN COMPLEX WITH MITOGEN- INDUCIBLE GENE 6 PROTEIN | EPIDERMAL GROWTH FACTOR RECEPTOR (EGFR), ERBB RECEPTOR FEEDBACK INHIBITOR 1, MITOGEN-INDUCIBLE GENE 6 PROTEIN(MIG6), TRANSFERASE- INHIBITOR COMPLEX
4zjv:B (GLY779) to (ARG973) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN IN COMPLEX WITH MITOGEN- INDUCIBLE GENE 6 PROTEIN | EPIDERMAL GROWTH FACTOR RECEPTOR (EGFR), ERBB RECEPTOR FEEDBACK INHIBITOR 1, MITOGEN-INDUCIBLE GENE 6 PROTEIN(MIG6), TRANSFERASE- INHIBITOR COMPLEX
3vjn:A (GLY779) to (ARG973) CRYSTAL STRUCTURE OF THE MUTATED EGFR KINASE DOMAIN (G719S/T790M) IN COMPLEX WITH AMPPNP. | RECEPTOR, DISEASE MUTATION, CELL CYCLE, DRUG RESISTANCE, KINASE, TYROSINE-PROTEIN KINASE, TRANSFERASE, ATP BINDING, PHOSPHORYLATION, TRANSMEMBRANE
3vjo:A (GLY779) to (ARG973) CRYSTAL STRUCTURE OF THE WILD-TYPE EGFR KINASE DOMAIN IN COMPLEX WITH AMPPNP. | RECEPTOR, DISEASE MUTATION, CELL CYCLE, DRUG RESISTANCE, KINASE, TYROSINE-PROTEIN KINASE, TRANSFERASE, ATP BINDING, PHOSPHORYLATION, TRANSMEMBRANE
3ika:A (GLY779) to (PRO975) CRYSTAL STRUCTURE OF EGFR 696-1022 T790M MUTANT COVALENTLY BINDING TO WZ4002 | EGFR, T790M, WZ4002, WZ-4002, ALTERNATIVE SPLICING, ATP- BINDING, CELL MEMBRANE, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, ISOPEPTIDE BOND, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TUMOR SUPPRESSOR, TYROSINE-PROTEIN KINASE, UBL CONJUGATION
3ika:B (GLY779) to (ASP974) CRYSTAL STRUCTURE OF EGFR 696-1022 T790M MUTANT COVALENTLY BINDING TO WZ4002 | EGFR, T790M, WZ4002, WZ-4002, ALTERNATIVE SPLICING, ATP- BINDING, CELL MEMBRANE, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, ISOPEPTIDE BOND, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TUMOR SUPPRESSOR, TYROSINE-PROTEIN KINASE, UBL CONJUGATION
1u46:A (GLY194) to (GLN389) CRYSTAL STRUCTURE OF THE UNPHOSPHORYLATED KINASE DOMAIN OF THE TYROSINE KINASE ACK1 | TYROSINE KINASE, TRANSFERASE
1u46:B (GLY194) to (ALA388) CRYSTAL STRUCTURE OF THE UNPHOSPHORYLATED KINASE DOMAIN OF THE TYROSINE KINASE ACK1 | TYROSINE KINASE, TRANSFERASE
1ir3:A (GLY1064) to (LEU1262) PHOSPHORYLATED INSULIN RECEPTOR TYROSINE KINASE IN COMPLEX WITH PEPTIDE SUBSTRATE AND ATP ANALOG | TYROSINE KINASE, SIGNAL TRANSDUCTION, PHOSPHOTRANSFERASE, COMPLEX (KINASE/PEPTIDE SUBSTRATE/ATP ANALOG), ENZYME, COMPLEX (TRANSFERASE/SUBSTRATE)
2x2k:A (TYR791) to (ARG1013) CRYSTAL STRUCTURE OF PHOSPHORYLATED RET TYROSINE KINASE DOMAIN WITH INHIBITOR | TYROSINE KINASE, HIRSCHSPRUNG DISEASE, TYROSINE-PROTEIN KINASE, PROTO-ONCOGENE, PHOSPHOPROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE
3bu5:A (GLY1064) to (LEU1263) CRYSTAL STRUCTURE OF THE INSULIN RECEPTOR KINASE IN COMPLEX WITH IRS2 KRLB PEPTIDE AND ATP | IRK, KRLB, IRS2, ATP, INSULIN RECEPTOR, PEPTIDE, SUBSTRATE, ALTERNATIVE SPLICING, ATP-BINDING, CARBOHYDRATE METABOLISM, CLEAVAGE ON PAIR OF BASIC RESIDUES, DIABETES MELLITUS, DISEASE MUTATION, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, TRANSDUCER
3c0h:A (GLU79) to (HIS273) CASK CAM-KINASE DOMAIN- AMPPNP COMPLEX, P1 FORM | CASK, NEUREXIN, CA2+/CALMODULIN DEPENDENT PROTEIN KINASE, MG2+, SYNAPTIC PLASTICITY, PSEUDOKINASE, MAGUK, MEMBRANE-ASSOCIATED GUANYLATE KINASE, ATP-BINDING, CALMODULIN-BINDING, MAGNESIUM, METAL- BINDING, NUCLEOTIDE-BINDING, NUCLEUS, SERINE/THREONINE-PROTEIN KINASE, SH3 DOMAIN, TRANSFERASE
3c0h:B (GLU79) to (LEU257) CASK CAM-KINASE DOMAIN- AMPPNP COMPLEX, P1 FORM | CASK, NEUREXIN, CA2+/CALMODULIN DEPENDENT PROTEIN KINASE, MG2+, SYNAPTIC PLASTICITY, PSEUDOKINASE, MAGUK, MEMBRANE-ASSOCIATED GUANYLATE KINASE, ATP-BINDING, CALMODULIN-BINDING, MAGNESIUM, METAL- BINDING, NUCLEOTIDE-BINDING, NUCLEUS, SERINE/THREONINE-PROTEIN KINASE, SH3 DOMAIN, TRANSFERASE
5hg7:A (GLY779) to (ARG973) EGFR (L858R, T790M, V948R) IN COMPLEX WITH 1-{(3R,4R)-3-[5-CHLORO-2- (1-METHYL-1H-PYRAZOL-4-YLAMINO)-7H-PYRROLO[2,3-D]PYRIMIDIN-4- YLOXYMETHYL]-4-METHOXY-PYRROLIDIN-1-YL}PROPENONE (PF-06459988) | EGFR, INHIBITOR, COMPLEX, LUNG CANCER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gfg:A (GLY437) to (GLY637) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH R9021 | SYK, SPLEEN TYPROSINE KINASE, PYRIMIDINE-5-CARBOXAMIDE, ATP-BINDING, HOST-VIRUS INTERACTION, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX