3rjw:A (LEU1013) to (THR1146) CRYSTAL STRUCTURE OF HISTONE LYSINE METHYLTRANSFERASE G9A WITH AN INHIBITOR | CHEMICAL PROBE, METHYLTRANSFERASE INHIBITOR, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3rjw:B (LEU1013) to (THR1146) CRYSTAL STRUCTURE OF HISTONE LYSINE METHYLTRANSFERASE G9A WITH AN INHIBITOR | CHEMICAL PROBE, METHYLTRANSFERASE INHIBITOR, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3fpd:A (LEU1070) to (ALA1203) G9A-LIKE PROTEIN LYSINE METHYLTRANSFERASE INHIBITION BY BIX- 01294 | EPIGENETICS, HISTONE LYSINE METHYLATION, CATALYTIC SET DOMAIN, INHIBITION BY BIX-01294, ALTERNATIVE SPLICING, ANK REPEAT, CHROMATIN REGULATOR, METAL-BINDING, METHYLTRANSFERASE, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, S- ADENOSYL-L-METHIONINE, TRANSFERASE, ZINC
3fpd:B (LEU1070) to (ALA1203) G9A-LIKE PROTEIN LYSINE METHYLTRANSFERASE INHIBITION BY BIX- 01294 | EPIGENETICS, HISTONE LYSINE METHYLATION, CATALYTIC SET DOMAIN, INHIBITION BY BIX-01294, ALTERNATIVE SPLICING, ANK REPEAT, CHROMATIN REGULATOR, METAL-BINDING, METHYLTRANSFERASE, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, S- ADENOSYL-L-METHIONINE, TRANSFERASE, ZINC
3swc:A (LEU1070) to (ALA1203) GLP (G9A-LIKE PROTEIN) SET DOMAIN IN COMPLEX WITH DNMT3AK44ME2 PEPTIDE | EPIGENETICS, NON-HISTONE LYSINE METHYLATION, SET DOMAIN, PROTEIN LYSINE METHYLTRANSFERASE, TRANSFERASE
3swc:B (LEU1070) to (ALA1203) GLP (G9A-LIKE PROTEIN) SET DOMAIN IN COMPLEX WITH DNMT3AK44ME2 PEPTIDE | EPIGENETICS, NON-HISTONE LYSINE METHYLATION, SET DOMAIN, PROTEIN LYSINE METHYLTRANSFERASE, TRANSFERASE
2r3a:A (PRO114) to (ALA253) METHYLTRANSFERASE DOMAIN OF HUMAN SUPPRESSOR OF VARIEGATION 3-9 HOMOLOG 2 | HISTONE H3-K9 METHYLTRANSFERASE 2, HISTONE-LYSINE N- METHYLTRANSFERASE, H3 LYSINE-9 SPECIFIC 2, ALTERNATIVE SPLICING, CELL CYCLE, CHROMATIN REGULATOR, CHROMOSOMAL PROTEIN, DIFFERENTIATION, NUCLEUS, REPRESSOR, S-ADENOSYL-L- METHIONINE, TELOMERE, TRANSCRIPTION, TRANSCRIPTION REGULATION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
4ypa:B (PHE2114) to (ALA2247) ASH1L SET DOMAIN Q2265A MUTANT IN COMPLEX WITH S-ADENOSYL METHIONINE (SAM) | HISTONE METHYLATION, SET DOMAIN, TRANSFERASE
4ypa:D (PHE2114) to (ALA2247) ASH1L SET DOMAIN Q2265A MUTANT IN COMPLEX WITH S-ADENOSYL METHIONINE (SAM) | HISTONE METHYLATION, SET DOMAIN, TRANSFERASE
3hna:A (LEU1070) to (ALA1203) CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF HUMAN EUCHROMATIC HISTONE METHYLTRANSFERASE 1 IN COMPLEX WITH SAH AND MONO-METHYLATED H3K9 PEPTIDE | EHMT1, STRUCTURAL GENOMICS, SGC, STRUCTURAL GENOMICS CONSORTIUM, ANK REPEAT, CHROMATIN REGULATOR, METAL-BINDING, METHYLTRANSFERASE, NUCLEUS, PHOSPHOPROTEIN, S-ADENOSYL-L-METHIONINE, TRANSFERASE, HYDROLASE-HYDROLASE REGULATOR COMPLEX
3hna:B (LEU1070) to (ALA1203) CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF HUMAN EUCHROMATIC HISTONE METHYLTRANSFERASE 1 IN COMPLEX WITH SAH AND MONO-METHYLATED H3K9 PEPTIDE | EHMT1, STRUCTURAL GENOMICS, SGC, STRUCTURAL GENOMICS CONSORTIUM, ANK REPEAT, CHROMATIN REGULATOR, METAL-BINDING, METHYLTRANSFERASE, NUCLEUS, PHOSPHOPROTEIN, S-ADENOSYL-L-METHIONINE, TRANSFERASE, HYDROLASE-HYDROLASE REGULATOR COMPLEX
2igq:A (LEU1070) to (ALA1203) HUMAN EUCHROMATIC HISTONE METHYLTRANSFERASE 1 | EUCHROMATIC HISTONE METHYLTRANSFERASE 1, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
2igq:B (LEU1070) to (ALA1203) HUMAN EUCHROMATIC HISTONE METHYLTRANSFERASE 1 | EUCHROMATIC HISTONE METHYLTRANSFERASE 1, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
4nvq:A (LEU1013) to (THR1146) HUMAN G9A IN COMPLEX WITH INHIBITOR A-366 | LYSINE METHYL TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4nvq:B (LEU1013) to (THR1146) HUMAN G9A IN COMPLEX WITH INHIBITOR A-366 | LYSINE METHYL TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3k5k:A (LEU1013) to (THR1146) DISCOVERY OF A 2,4-DIAMINO-7-AMINOALKOXY-QUINAZOLINE AS A POTENT INHIBITOR OF HISTONE LYSINE METHYLTRANSFERASE, G9A | HISTONE LYSINE METHYLTRANSFERASE, G9A, ANK REPEAT, CHROMATIN REGULATOR, METAL-BINDING, METHYLTRANSFERASE, NUCLEUS, PHOSPHOPROTEIN, S-ADENOSYL-L-METHIONINE, TRANSFERASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
3k5k:B (LEU1013) to (THR1146) DISCOVERY OF A 2,4-DIAMINO-7-AMINOALKOXY-QUINAZOLINE AS A POTENT INHIBITOR OF HISTONE LYSINE METHYLTRANSFERASE, G9A | HISTONE LYSINE METHYLTRANSFERASE, G9A, ANK REPEAT, CHROMATIN REGULATOR, METAL-BINDING, METHYLTRANSFERASE, NUCLEUS, PHOSPHOPROTEIN, S-ADENOSYL-L-METHIONINE, TRANSFERASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
1mvh:A (ALA302) to (PRO443) STRUCTURE OF THE SET DOMAIN HISTONE LYSINE METHYLTRANSFERASE CLR4 | LYSINE METHYLTRANSFERASE, CLR4, SET-DOMAIN
3mo0:A (LEU1070) to (ALA1203) HUMAN G9A-LIKE (GLP, ALSO KNOWN AS EHMT1) IN COMPLEX WITH INHIBITOR E11 | EPIGENETICS, HISTONE LYSINE METHYLATION, ENZYMATIC INHIBITION, LYSINE MIMICS, TRANSFERASE
3mo0:B (PRO1069) to (ALA1203) HUMAN G9A-LIKE (GLP, ALSO KNOWN AS EHMT1) IN COMPLEX WITH INHIBITOR E11 | EPIGENETICS, HISTONE LYSINE METHYLATION, ENZYMATIC INHIBITION, LYSINE MIMICS, TRANSFERASE
3mo2:A (LEU1070) to (ALA1203) HUMAN G9A-LIKE (GLP, ALSO KNOWN AS EHMT1) IN COMPLEX WITH INHIBITOR E67 | EPIGENETICS, HISTONE LYSINE METHYLATION, ENZYMATIC INHIBITION, LYSINE MIMICS, TRANSFERASE
3mo2:B (LEU1070) to (ALA1203) HUMAN G9A-LIKE (GLP, ALSO KNOWN AS EHMT1) IN COMPLEX WITH INHIBITOR E67 | EPIGENETICS, HISTONE LYSINE METHYLATION, ENZYMATIC INHIBITION, LYSINE MIMICS, TRANSFERASE
3mo2:C (LEU1070) to (ALA1203) HUMAN G9A-LIKE (GLP, ALSO KNOWN AS EHMT1) IN COMPLEX WITH INHIBITOR E67 | EPIGENETICS, HISTONE LYSINE METHYLATION, ENZYMATIC INHIBITION, LYSINE MIMICS, TRANSFERASE
3mo2:D (LEU1070) to (ALA1203) HUMAN G9A-LIKE (GLP, ALSO KNOWN AS EHMT1) IN COMPLEX WITH INHIBITOR E67 | EPIGENETICS, HISTONE LYSINE METHYLATION, ENZYMATIC INHIBITION, LYSINE MIMICS, TRANSFERASE
3mo5:A (LEU1070) to (ALA1203) HUMAN G9A-LIKE (GLP, ALSO KNOWN AS EHMT1) IN COMPLEX WITH INHIBITOR E72 | EPIGENETICS, HISTONE LYSINE METHYLATION, ENZYMATIC INHIBITION, LYSINE MIMICS, TRANSFERASE
3mo5:B (LEU1070) to (ALA1203) HUMAN G9A-LIKE (GLP, ALSO KNOWN AS EHMT1) IN COMPLEX WITH INHIBITOR E72 | EPIGENETICS, HISTONE LYSINE METHYLATION, ENZYMATIC INHIBITION, LYSINE MIMICS, TRANSFERASE
3mo5:C (LEU1070) to (ALA1203) HUMAN G9A-LIKE (GLP, ALSO KNOWN AS EHMT1) IN COMPLEX WITH INHIBITOR E72 | EPIGENETICS, HISTONE LYSINE METHYLATION, ENZYMATIC INHIBITION, LYSINE MIMICS, TRANSFERASE
3mo5:D (LEU1070) to (ALA1203) HUMAN G9A-LIKE (GLP, ALSO KNOWN AS EHMT1) IN COMPLEX WITH INHIBITOR E72 | EPIGENETICS, HISTONE LYSINE METHYLATION, ENZYMATIC INHIBITION, LYSINE MIMICS, TRANSFERASE
3bo5:A (PRO100) to (PRO240) CRYSTAL STRUCTURE OF METHYLTRANSFERASE DOMAIN OF HUMAN HISTONE-LYSINE N-METHYLTRANSFERASE SETMAR | TRANSFERASE, SET DOMAIN, METHYLTRANSFERASE, SETMAR, CHROMATIN REGULATOR, DNA DAMAGE, DNA REPAIR, DNA-BINDING, NUCLEUS, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
5jin:A (LEU1013) to (THR1146) STRUCTURE OF G9A SET-DOMAIN WITH HISTONE H3K9M MUTANT PEPTIDE AND BOUND S-ADENOSYLMETHIONINE | SET-DOMAIN, HISTONE METHYL TRANSFERASE, HISTONE PEPTIDE, TRANSFERASE
5jin:B (LEU1013) to (THR1146) STRUCTURE OF G9A SET-DOMAIN WITH HISTONE H3K9M MUTANT PEPTIDE AND BOUND S-ADENOSYLMETHIONINE | SET-DOMAIN, HISTONE METHYL TRANSFERASE, HISTONE PEPTIDE, TRANSFERASE
5jiy:A (LEU1013) to (THR1146) STRUCTURE OF G9A SET-DOMAIN WITH HISTONE H3K9NORLEUCINE MUTANT PEPTIDE AND BOUND S-ADENOSYLMETHIONINE | SET-DOMAIN, HISTONE METHYL TRANSFERASE, HISTONE PEPTIDE, TRANSFERASE
5jiy:B (LEU1013) to (THR1146) STRUCTURE OF G9A SET-DOMAIN WITH HISTONE H3K9NORLEUCINE MUTANT PEPTIDE AND BOUND S-ADENOSYLMETHIONINE | SET-DOMAIN, HISTONE METHYL TRANSFERASE, HISTONE PEPTIDE, TRANSFERASE
5jj0:A (LEU1013) to (THR1146) STRUCTURE OF G9A SET-DOMAIN WITH HISTONE H3K9M PEPTIDE AND EXCESS SAH | SET-DOMAIN, HISTONE METHYL TRANSFERASE, HISTONE PEPTIDE, TRANSFERASE
5jj0:B (LEU1013) to (THR1146) STRUCTURE OF G9A SET-DOMAIN WITH HISTONE H3K9M PEPTIDE AND EXCESS SAH | SET-DOMAIN, HISTONE METHYL TRANSFERASE, HISTONE PEPTIDE, TRANSFERASE
5lt6:A (MET1526) to (SER1658) STRUCTURE OF THE EPIGENETIC ONCOGENE MMSET AND INHIBITION BY N-ALKYL SINEFUNGIN DERIVATIVES | LYSINE METHYLTRANSFERASE SETD2 SET DOMAIN, SETD2#1, TRANSFERASE
5lt7:A (MET1526) to (SER1658) STRUCTURE OF THE EPIGENETIC ONCOGENE MMSET AND INHIBITION BY N-ALKYL SINEFUNGIN DERIVATIVES | LYSINE METHYLTRANSFERASE SETD2 SET DOMAIN, TRANSFERASE
5t0k:A (LEU1013) to (THR1146) STRUCTURE OF G9A SET-DOMAIN WITH H3K9M MUTANT PEPTIDE AND SAM | HISTONE METHYLTRANSFERASE, SET DOMAIN, TRANSFERASE
5t0k:B (LEU1013) to (THR1146) STRUCTURE OF G9A SET-DOMAIN WITH H3K9M MUTANT PEPTIDE AND SAM | HISTONE METHYLTRANSFERASE, SET DOMAIN, TRANSFERASE
2o8j:A (LEU1013) to (THR1146) HUMAN EUCHROMATIC HISTONE METHYLTRANSFERASE 2 | HLA-B-ASSOCIATED TRANSCRIPT 8, BAT8, G9A, NG36/G9A, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
2o8j:B (LEU1013) to (THR1146) HUMAN EUCHROMATIC HISTONE METHYLTRANSFERASE 2 | HLA-B-ASSOCIATED TRANSCRIPT 8, BAT8, G9A, NG36/G9A, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
2o8j:C (LEU1013) to (THR1146) HUMAN EUCHROMATIC HISTONE METHYLTRANSFERASE 2 | HLA-B-ASSOCIATED TRANSCRIPT 8, BAT8, G9A, NG36/G9A, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
2o8j:D (LEU1013) to (THR1146) HUMAN EUCHROMATIC HISTONE METHYLTRANSFERASE 2 | HLA-B-ASSOCIATED TRANSCRIPT 8, BAT8, G9A, NG36/G9A, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
2rfi:A (LEU1070) to (ALA1203) CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF HUMAN EUCHROMATIC HISTONE METHYLTRANSFERASE 1 IN COMPLEX WITH SAH AND DIMETHYLATED H3K9 PEPTIDE | EUCHROMATIC HISTONE METHYLTRANSFERASE 1, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ALTERNATIVE SPLICING, ANK REPEAT, CHROMATIN REGULATOR, NUCLEUS, PHOSPHORYLATION, POLYMORPHISM, S-ADENOSYL-L-METHIONINE, ACETYLATION, CHROMOSOMAL PROTEIN, DNA DAMAGE, DNA REPAIR, DNA-BINDING, METHYLATION, NUCLEOSOME CORE, TRANSFERASE
2rfi:B (LEU1070) to (ALA1203) CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF HUMAN EUCHROMATIC HISTONE METHYLTRANSFERASE 1 IN COMPLEX WITH SAH AND DIMETHYLATED H3K9 PEPTIDE | EUCHROMATIC HISTONE METHYLTRANSFERASE 1, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ALTERNATIVE SPLICING, ANK REPEAT, CHROMATIN REGULATOR, NUCLEUS, PHOSPHORYLATION, POLYMORPHISM, S-ADENOSYL-L-METHIONINE, ACETYLATION, CHROMOSOMAL PROTEIN, DNA DAMAGE, DNA REPAIR, DNA-BINDING, METHYLATION, NUCLEOSOME CORE, TRANSFERASE
4ype:B (PHE2114) to (ALA2247) ASH1L SET DOMAIN H2193F MUTANT IN COMPLEX WITH S-ADENOSYL METHIONINE (SAM) | HISTONE METHYLATION, SET DOMAIN, TRANSFERASE
5jhn:A (LEU1013) to (THR1146) STRUCTURE OF G9A SET-DOMAIN WITH HISTONE H3K9ALA MUTANT PEPTIDE AND BOUND S-ADENOSYLMETHIONINE | SET-DOMAIN, HISTONE METHYL TRANSFERASE, HISTONE PEPTIDE, TRANSFERASE
5jhn:B (LEU1013) to (THR1146) STRUCTURE OF G9A SET-DOMAIN WITH HISTONE H3K9ALA MUTANT PEPTIDE AND BOUND S-ADENOSYLMETHIONINE | SET-DOMAIN, HISTONE METHYL TRANSFERASE, HISTONE PEPTIDE, TRANSFERASE
5jjy:A (MET1526) to (SER1658) CRYSTAL STRUCTURE OF SETD2 BOUND TO HISTONE H3.3 K36M PEPTIDE | SET DOMAIN, TRANSFERASE
5t0m:A (LEU1013) to (THR1146) A HISTONE H3K9M MUTATION TRAPS HISTONE METHYLTRANSFERASE CLR4 TO PREVENT HETEROCHROMATIN SPREADING | HISTONE METHYLTRANSFERASE, SET DOMAIN, TRANSFERASE
5t0m:B (LEU1013) to (THR1146) A HISTONE H3K9M MUTATION TRAPS HISTONE METHYLTRANSFERASE CLR4 TO PREVENT HETEROCHROMATIN SPREADING | HISTONE METHYLTRANSFERASE, SET DOMAIN, TRANSFERASE