2o8y:A (GLY198) to (SER336) APO IRAK4 KINASE DOMAIN | PROTEIN KINASE, IMMUNODEFICIENCY, INFLAMMATION, TRANSFERASE
2o8y:B (GLY198) to (SER336) APO IRAK4 KINASE DOMAIN | PROTEIN KINASE, IMMUNODEFICIENCY, INFLAMMATION, TRANSFERASE
3e62:A (GLY861) to (GLN1003) FRAGMENT BASED DISCOVERY OF JAK-2 INHIBITORS | DRUG DISCOVERY, JAK2, FRAGMENT BASED, ATP-BINDING, DISEASE MUTATION, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
1na7:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF THE CATALYTIC SUBUNIT OF HUMAN PROTEIN KINASE CK2 | CK2, PROTEIN KINASE, MICROCRYSTALS, THIN-FILM NANOTECHNOLOGY, MICROFOCUS ESRF, TRANSFERASE
4gub:A (SER51) to (PHE181) CASEIN KINASE II BOUND TO INHIBITOR | KINASE, TRANSFERASE, CYTOSOL, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gva:A (GLY35) to (VAL171) ADP-BOUND FORM OF THE ERK2 KINASE | MITOGEN-ACTIVATED PROTEIN KINASE, TRANSFERASE
4gvj:A (GLY909) to (GLU1050) TYK2 (JH1) IN COMPLEX WITH ADENOSINE DI-PHOSPHATE | KINASE, HYDROLASE
2oid:B (GLY198) to (ALA335) CRYSTAL STRUCTURE OF IRAK4 KINASE DOMAIN COMPLEXED WITH AMPPNP | KINASE, TRANSFERASE
2ojj:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH (S)-N-(1-(3- CHLORO-4-FLUOROPHENYL)-2-HYDROXYETHYL)-4-(4-(3- CHLOROPHENYL)-1H-PYRAZOL-3-YL)-1H-PYRROLE-2-CARBOXAMIDE | KINASE INHIBITOR, TRANSFERASE
4wno:A (ALA28) to (GLN173) STRUCTURE OF ULK1 BOUND TO AN INHIBITOR | KINASE, AUTOPHAGY, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3eid:A (GLY16) to (GLY153) CDK2/CYCLINA COMPLEXED WITH A PYRAZOLOPYRIDAZINE INHIBITOR | CDK2, CYCLIN, ATP-BINDING, CELL CYCLE, CELL DIVISION, KINASE, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE, NUCLEUS, TRANSFERASE-CELL CYCLE COMPLEX
3eid:C (GLY16) to (GLY153) CDK2/CYCLINA COMPLEXED WITH A PYRAZOLOPYRIDAZINE INHIBITOR | CDK2, CYCLIN, ATP-BINDING, CELL CYCLE, CELL DIVISION, KINASE, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE, NUCLEUS, TRANSFERASE-CELL CYCLE COMPLEX
3ej1:A (GLY16) to (GLY153) CDK2/CYCLINA COMPLEXED WITH A PYRAZOLOPYRIDAZINE INHIBITOR | CDK, CYCLIN, KINASE, ATP-BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, NUCLEUS, TRANSFERASE-CELL CYCLE COMPLEX
4h3p:A (GLY37) to (VAL173) CRYSTAL STRUCTURE OF HUMAN ERK2 COMPLEXED WITH A MAPK DOCKING PEPTIDE | KINASE DOMAIN, SIGNALING, LINEAR MOTIF, SURFACE MUTATION, TRANSFERASE
4h3q:A (GLY37) to (ALA174) CRYSTAL STRUCTURE OF HUMAN ERK2 COMPLEXED WITH A MAPK DOCKING PEPTIDE | KINASE DOMAIN, SIGNALING, LINEAR MOTIF, SURFACE MUTATION, TRANSFERASE
2ow3:A (GLY68) to (GLN206) GLYCOGEN SYNTHASE KINASE-3 BETA IN COMPLEX WITH BIS- (INDOLE)MALEIMIDE PYRIDINOPHANE INHIBITOR | KINASE-INHIBITOR COMPLEX, TRANSFERASE
2oxd:A (SER51) to (PHE181) PROTEIN KINASE CK2 IN COMPLEX WITH TETRABROMOBENZOIMIDAZOLE K17, K22 AND K32 INHIBITORS | KINASE, INHIBITOR COMPLEX, TRANSFERASE
2oxy:A (GLU55) to (PHE181) PROTEIN KINASE CK2 IN COMPLEX WITH TETRABROMOBENZOIMIDAZOLE DERIVATIVES K17, K22 AND K32 | PROTEIN KINASE CK2, INHIBITORS, TETRABROMOBENZOIMIDAZOLE DERIVATIVES, TRANSFERASE
2oxy:B (SER51) to (PHE181) PROTEIN KINASE CK2 IN COMPLEX WITH TETRABROMOBENZOIMIDAZOLE DERIVATIVES K17, K22 AND K32 | PROTEIN KINASE CK2, INHIBITORS, TETRABROMOBENZOIMIDAZOLE DERIVATIVES, TRANSFERASE
2b7a:A (GLY861) to (GLN1003) THE STRUCTURAL BASIS OF JANUS KINASE 2 INHIBITION BY A POTENT AND SPECIFIC PAN-JANUS KINASE INHIBITOR | KINASE, TRANSFERASE
2b7a:B (GLY861) to (GLN1003) THE STRUCTURAL BASIS OF JANUS KINASE 2 INHIBITION BY A POTENT AND SPECIFIC PAN-JANUS KINASE INHIBITOR | KINASE, TRANSFERASE
3eoc:A (GLY16) to (GLY153) CDK2/CYCLINA COMPLEXED WITH A IMIDAZO TRIAZIN-2-AMINE | CDK, CYCLIN, ATP-BINDING, CELL CYCLE, CELL DIVISION, KINASE, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, NUCLEUS, TRANSFERASE-CELL CYCLE COMPLEX
2b9f:A (GLY25) to (ILE161) CRYSTAL STRUCTURE OF NON-PHOSPHORYLATED FUS3 | TRANSFERASE
2b9j:A (GLY25) to (ILE162) CRYSTAL STRUCTURE OF FUS3 WITH A DOCKING MOTIF FROM FAR1 | TRANSFERASE
1ny3:A (LEU79) to (THR215) CRYSTAL STRUCTURE OF ADP BOUND TO MAP KAP KINASE 2 | MAP KAP KINASE 2, MK2, ADP, KINASE, SER/THR KINASE, TRANSFERASE
4ww5:A (ILE29) to (SER189) CRYSTAL STRUCTURE OF BINARY COMPLEX BUD32-CGI121 IN COMPLEX WITH AMPP | KEOPS, BINARY COMPLEX, BUD32-CGI121, TRNA T6A, TRANSFERASE
4ww9:A (ILE29) to (SER189) CRYSTAL STRUCTURE OF BINARY COMPLEX BUD32-CGI121 IN COMPLEX WITH ADP | KEOPS, BINARY COMPLEX, BUD32-CGI121, TRNA T6A, TRANSCRIPTION
4wwa:A (ILE29) to (VAL188) CRYSTAL STRUCTURE OF BINARY COMPLEX BUD32-CGI121 | KEOPS, BINARY COMPLEX, BUD32-CGI121, TRNA T6A, TRANSFERASE, HYDROLASE
3erk:A (GLY35) to (VAL171) THE COMPLEX STRUCTURE OF THE MAP KINASE ERK2/SB220025 | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, MAP KINASE, ERK2
4hge:A (GLY861) to (GLN1003) JAK2 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 8 | PROTEIN KINASE, PHOSPHOTRANSFER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4hge:B (GLY861) to (GLN1003) JAK2 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 8 | PROTEIN KINASE, PHOSPHOTRANSFER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3eyg:A (LEU891) to (THR1030) CRYSTAL STRUCTURES OF JAK1 AND JAK2 INHIBITOR COMPLEXES | JAK KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
2bkz:A (GLY16) to (GLY153) STRUCTURE OF CDK2-CYCLIN A WITH PHA-404611 | TRANSFERASE/COMPLEX, PROTEIN KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, PHOSPHORYLATION, CELL DIVISION, CYCLIN, ATP-BINDING, CELL CYCLE, MITOSIS, POLYMORPHISM
2bkz:C (GLY16) to (GLY153) STRUCTURE OF CDK2-CYCLIN A WITH PHA-404611 | TRANSFERASE/COMPLEX, PROTEIN KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, PHOSPHORYLATION, CELL DIVISION, CYCLIN, ATP-BINDING, CELL CYCLE, MITOSIS, POLYMORPHISM
2bpm:C (GLY16) to (PHE152) STRUCTURE OF CDK2-CYCLIN A WITH PHA-630529 | PROTEIN KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, PHOSPHORYLATION, CELL DIVISION, CYCLIN
3f5x:A (GLY16) to (GLY153) CDK-2-CYCLIN COMPLEX WITH INDAZOLE INHIBITOR 9 BOUND AT ITS ACTIVE SITE | KINASE, PKC, PROTEIN KINASE, INHIBITOR, ATP-BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, CYCLIN, NUCLEUS, TRANSFERASE-CELL CYCLE COMPLEX
3f5x:C (GLY16) to (GLY153) CDK-2-CYCLIN COMPLEX WITH INDAZOLE INHIBITOR 9 BOUND AT ITS ACTIVE SITE | KINASE, PKC, PROTEIN KINASE, INHIBITOR, ATP-BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, CYCLIN, NUCLEUS, TRANSFERASE-CELL CYCLE COMPLEX
3s95:B (GLY351) to (VAL486) CRYSTAL STRUCTURE OF THE HUMAN LIMK1 KINASE DOMAIN IN COMPLEX WITH STAUROSPORINE | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, LIM DOMAIN KINASE, TRANSFERASE-ANTIBIOTIC COMPLEX
3sa0:A (GLY37) to (VAL173) COMPLEX OF ERK2 WITH NORATHYRIOL | NORATHYRIOL COMPLEX, SIGNAL-REGULATED KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2bva:B (VAL335) to (VAL465) CRYSTAL STRUCTURE OF THE HUMAN P21-ACTIVATED KINASE 4 | PROTEIN KINASE, STE20, PAK4, ATP-BINDING, TRANSFERASE
2phk:A (ARG35) to (PRO176) THE CRYSTAL STRUCTURE OF A PHOSPHORYLASE KINASE PEPTIDE SUBSTRATE COMPLEX: KINASE SUBSTRATE RECOGNITION | CATALYTIC MECHANISM, DIMERIZATION, PHOSPHORYLASE KINASE, REVERSIBLE PHOSPHORYLISATION, SUBSTRATE RECOGNITION, COMPLEX (TRANSFERASE- PEPTIDE), COMPLEX (TRANSFERASE-PEPTIDE) COMPLEX
4hvg:A (GLY834) to (LEU976) JAK3 KINASE DOMAIN IN COMPLEX WITH 2-CYCLOPROPYL-5H-PYRROLO[2,3- B]PYRAZINE-7-CARBOXYLIC ACID ((S)-2-HYDROXY-1,2-DIMETHYL-PROPYL)- AMIDE | KINASE-INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2pmi:C (THR20) to (GLY159) STRUCTURE OF THE PHO85-PHO80 CDK-CYCLIN COMPLEX OF THE PHOSPHATE- RESPONSIVE SIGNAL TRANSDUCTION PATHWAY WITH BOUND ATP-GAMMA-S | CYCLIN-DEPENDENT KINASE, CYCLIN, SIGNALING PROTEIN,TRANSFERASE-CELL CYCLE COMPLEX
1oiu:A (VAL17) to (ALA151) STRUCTURE OF HUMAN THR160-PHOSPHO CDK2/CYCLIN A COMPLEXED WITH A 6-CYCLOHEXYLMETHYLOXY-2-ANILINO-PURINE INHIBITOR | KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP- BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, PHOSPHORYLATION
1okv:A (GLY16) to (GLY153) CYCLIN A BINDING GROOVE INHIBITOR H-ARG-ARG-LEU-ILE-PHE-NH2 | KINASE-CYCLIN COMPLEX, CYCLIN A, INHIBITOR, LIGAND EXCHANGE, DRUG DESIGN, PEPTIDOMIMETICS, CELL CYCLE, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3fl5:A (SER51) to (PHE181) PROTEIN KINASE CK2 IN COMPLEX WITH THE INHIBITOR QUINALIZARIN | PROTEIN KINASE CK2-INHIBITOR COMPLEX, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
1ol2:C (VAL17) to (GLY153) CYCLIN A BINDING GROOVE INHIBITOR H-ARG-ARG-LEU-ASN-(P-F-PHE)-NH2 | CELL CYCLE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, CYCLIN A, LIGAND EXCHANGE, PEPTIDOMIMETICS, KINASE
1om1:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF MAIZE CK2 ALPHA IN COMPLEX WITH IQA | CK2, IQA, INHIBITOR, ZEA MAYS, TRANSFERASE
2pvh:A (GLU55) to (PHE181) STRUCTURE-BASED DESIGN OF PYRAZOLO[1,5-A][1,3,5]TRIAZINE DERIVATIVES AS POTENT INHIBITORS OF PROTEIN KINASE CK2 | STRUCTURE-BASED DRUG DESIGN, ENZYME-INHIBITOR COMPLEX, CASEIN KINASE II, PROTEIN KINASE CK2, TRANSFERASE
2pvj:A (GLU52) to (PHE181) STRUCTURE-BASED DESIGN OF PYRAZOLO[1,5-A][1,3,5]TRIAZINE DERIVATIVES AS POTENT INHIBITORS OF PROTEIN KINASE CK2 | STRUCTURE-BASED DRUG DESIGN, ENZYME-INHIBITOR COMPLEX, CASEIN KINASE II, PROTEIN KINASE CK2, TRANSFERASE
2pvk:A (GLU55) to (PHE181) STRUCTURE-BASED DESIGN OF PYRAZOLO[1,5-A][1,3,5]TRIAZINE DERIVATIVES AS POTENT INHIBITORS OF PROTEIN KINASE CK2 | STRUCTURE-BASED DRUG DESIGN, ENZYME-INHIBITOR COMPLEX, CASEIN KINASE II, PROTEIN KINASE CK2, TRANSFERASE
2pvn:A (SER51) to (PHE181) STRUCTURE-BASED DESIGN OF PYRAZOLO[1,5-A][1,3,5]TRIAZINE DERIVATIVES AS POTENT INHIBITORS OF PROTEIN KINASE CK2 | STRUCTURE-BASED DRUG DESIGN, ENZYME-INHIBITOR COMPLEX, CASEIN KINASE II, PROTEIN KINASE CK2, TRANSFERASE
4i5c:B (GLY887) to (THR1030) THE JAK1 KINASE DOMAIN IN COMPLEX WITH INHIBITOR | KINASE, TRANSFERASE
1opk:A (GLU274) to (MET407) STRUCTURAL BASIS FOR THE AUTO-INHIBITION OF C-ABL TYROSINE KINASE | TRANSFERASE
1opl:A (GLU274) to (MET407) STRUCTURAL BASIS FOR THE AUTO-INHIBITION OF C-ABL TYROSINE KINASE | TRANSFERASE
3fpm:A (LEU79) to (THR215) CRYSTAL STRUCTURE OF A SQUARATE INHIBITOR BOUND TO MAPKAP KINASE-2 | 3D-STRUCTURE, ATP-BINDING, ALTERNATIVE SPLICING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2c5o:A (GLY16) to (GLY153) DIFFERENTIAL BINDING OF INHIBITORS TO ACTIVE AND INACTIVE CDK2 PROVIDES INSIGHTS FOR DRUG DESIGN | DIFFERENTIAL INHIBITION, TRANSFERASE, CDK2, ATP-BINDING, CELL CYCLE, CELL DIVISION, POLYMORPHISM, PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN, KINASE, MITOSIS, CYCLIN
2c5n:C (GLY16) to (GLY153) DIFFERENTIAL BINDING OF INHIBITORS TO ACTIVE AND INACTIVE CDK2 PROVIDES INSIGHTS FOR DRUG DESIGN | DIFFERENTIAL INHIBITION, TRANSFERASE, CDK2, ATP-BINDING, CELL CYCLE, CELL DIVISION, POLYMORPHISM, PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN, KINASE, MITOSIS, CYCLIN
2c5x:C (GLY16) to (GLY153) DIFFERENTIAL BINDING OF INHIBITORS TO ACTIVE AND INACTIVE CDK2 PROVIDES INSIGHTS FOR DRUG DESIGN | TRANSFERASE/INHIBITOR, INHIBITION, ACTIVE, INACTIVE, CDK2, CELL CYCLE, CELL DIVISION, KINASE, MITOSIS, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, COMPLEX (TRANSFERASE/INHIBITOR)
2pzy:C (GLY76) to (THR215) STRUCTURE OF MK2 COMPLEXED WITH COMPOUND 76 | MK2, PROTEIN KINASE, TRANSFERASE
4ib5:A (GLU55) to (PHE181) STRUCTURE OF HUMAN PROTEIN KINASE CK2 CATALYTIC SUBUNIT IN COMPLEX WITH A CK2BETA-COMPETITIVE CYCLIC PEPTIDE | PROTEIN KINASE FOLD, PROTEIN PHOSPHORYLATION, BINDING OF CK2BETA, PHOSPHORYLATION, NUCLEUS, TRANSFERASE
4ib5:B (SER51) to (PHE181) STRUCTURE OF HUMAN PROTEIN KINASE CK2 CATALYTIC SUBUNIT IN COMPLEX WITH A CK2BETA-COMPETITIVE CYCLIC PEPTIDE | PROTEIN KINASE FOLD, PROTEIN PHOSPHORYLATION, BINDING OF CK2BETA, PHOSPHORYLATION, NUCLEUS, TRANSFERASE
4ib5:C (SER51) to (PHE181) STRUCTURE OF HUMAN PROTEIN KINASE CK2 CATALYTIC SUBUNIT IN COMPLEX WITH A CK2BETA-COMPETITIVE CYCLIC PEPTIDE | PROTEIN KINASE FOLD, PROTEIN PHOSPHORYLATION, BINDING OF CK2BETA, PHOSPHORYLATION, NUCLEUS, TRANSFERASE
4idt:A (GLY412) to (LEU541) CRYSTAL STRUCTURE OF NIK WITH 11-BROMO-5,6,7,8-TETRAHYDROPYRIMIDO[4', 5':3,4]CYCLOHEPTA[1,2-B]INDOL-2-AMINE (T28) | NIK, NUCLEAR FACTOR (NF)-KB, P100 PROCESSING, 2-AMINOPYRIMIDINE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4idv:C (HIS415) to (PRO543) CRYSTAL STRUCTURE OF NIK WITH COMPOUND 4-{3-[2-AMINO-5-(2- METHOXYETHOXY)PYRIMIDIN-4-YL]-1H-INDOL-5-YL}-2-METHYLBUT-3-YN-2-OL (13V) | NIK, NUCLEAR FACTOR (NF)-KB, P100 PROCESSING, 2-AMINOPYRIMIDINE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3fyj:X (ASN75) to (GLU213) CRYSTAL STRUCTURE OF AN OPTIMZIED BENZOTHIOPHENE INHIBITOR BOUND TO MAPKAP KINASE-2 (MK-2) | MK-2, MK2, MAPKAP-2, SER/THR KINASE, MAP KINASE, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4xne:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH AN INHIBITOR | SERINE THREONINE KINASE INHIBITOR, TRANSFERASE
2cdz:A (GLY333) to (SER466) CRYSTAL STRUCTURE OF THE HUMAN P21-ACTIVATED KINASE 4 IN COMPLEX WITH CGP74514A | TRANSFERASE, PROTEIN KINASE, STE20, PAK4, ATP-BINDING
4xoy:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH AN INHIBITOR | SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4xoz:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH AN INHIBITOR | SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4xp0:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH AN INHIBITOR | SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4xp3:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH AN INHIBITOR | SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2qg5:B (GLY40) to (ARG175) CRYPTOSPORIDIUM PARVUM CALCIUM DEPENDENT PROTEIN KINASE CGD7_1840 | MALARIA, CALCIUM DEPENDENT KINASE, SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSFERASE
4xrj:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH AN INHIBITOR | SERINE THREONINE KINASE INHIBITOR, APOPTOSIS
4xrl:A (GLY35) to (VAL171) CRYSTAL STRUCTURE AT ROOM TEMPERATURE OF ERK2 IN COMPLEX WITH AN INHIBITOR | SERINE THREONINE KINASE INHIBITOR, TRANSFERASE
2qkr:A (VAL36) to (PHE169) CRYPTOSPORIDIUM PARVUM CYCLIN-DEPENDENT KINASE CGD5_2510 WITH INDIRUBIN 3'-MONOXIME BOUND | CP-SPECIFIC CYCLIN-DEPENDENT KINASE, MALARIA, CRYPTOSPORIDIUM PARVUM, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3gb2:A (VAL69) to (GLN206) GSK3BETA INHIBITOR COMPLEX | PROTEIN KINASE, INHIBITOR, COMPLEX, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY, CDM
1pjk:A (SER51) to (TYR182) CRYSTAL STRUCTURE OF A C-TERMINAL DELETION MUTANT OF HUMAN PROTEIN KINASE CK2 CATALYTIC SUBUNIT | EUKARYOTIC PROTEIN KINASE FOLD, TRANSFERASE
4iva:A (GLY861) to (GLN1003) JAK2 KINASE (JH1 DOMAIN) IN COMPLEX WITH THE INHIBITOR TRANS-4-[(8AS)- 2-[(1R)-1-HYDROXYETHYL]IMIDAZO[4,5-D]PYRROLO[2,3-B]PYRIDIN-1(8AH)- YL]CYCLOHEXANECARBONITRILE | PROTEIN KINASE, PHOSPHOTRANSFER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ivb:A (GLY887) to (THR1030) JAK1 KINASE (JH1 DOMAIN) IN COMPLEX WITH THE INHIBITOR TRANS-4-{2- [(1R)-1-HYDROXYETHYL]IMIDAZO[4,5-D]PYRROLO[2,3-B]PYRIDIN-1(6H)- YL}CYCLOHEXANECARBONITRILE | PROTEIN KINASE, PHOSPHOTRANSFER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4iz5:A (GLY37) to (VAL173) STRUCTURE OF THE COMPLEX BETWEEN ERK2 PHOSPHOMIMETIC MUTANT AND PEA-15 | MAP KINASE, DEATH EFFECTOR DOMAIN, TRANSFERASE
4iz5:B (GLY37) to (VAL173) STRUCTURE OF THE COMPLEX BETWEEN ERK2 PHOSPHOMIMETIC MUTANT AND PEA-15 | MAP KINASE, DEATH EFFECTOR DOMAIN, TRANSFERASE
4iz5:C (GLY37) to (VAL173) STRUCTURE OF THE COMPLEX BETWEEN ERK2 PHOSPHOMIMETIC MUTANT AND PEA-15 | MAP KINASE, DEATH EFFECTOR DOMAIN, TRANSFERASE
4iz5:D (GLY37) to (VAL173) STRUCTURE OF THE COMPLEX BETWEEN ERK2 PHOSPHOMIMETIC MUTANT AND PEA-15 | MAP KINASE, DEATH EFFECTOR DOMAIN, TRANSFERASE
4iz7:C (GLY37) to (VAL173) STRUCTURE OF NON-PHOSPHORYLATED ERK2 BOUND TO THE PEA-15 DEATH EFFECTOR DOMAIN | MAP KINASE, DEATH EFFECTOR DOMAIN, TRANSFERASE
4iz7:A (GLY37) to (VAL173) STRUCTURE OF NON-PHOSPHORYLATED ERK2 BOUND TO THE PEA-15 DEATH EFFECTOR DOMAIN | MAP KINASE, DEATH EFFECTOR DOMAIN, TRANSFERASE
4iza:A (GLY37) to (VAL173) STRUCTURE OF DUALLY PHOSPHORYLATED ERK2 BOUND TO THE PEA-15 DEATH EFFECTOR DOMAIN | MAP KINASE, DEATH EFFECTOR DOMAIN, TRANSFERASE
4iza:C (GLY37) to (VAL173) STRUCTURE OF DUALLY PHOSPHORYLATED ERK2 BOUND TO THE PEA-15 DEATH EFFECTOR DOMAIN | MAP KINASE, DEATH EFFECTOR DOMAIN, TRANSFERASE
3gok:A (LEU79) to (THR215) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:B (LEU79) to (THR215) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:C (LEU79) to (THR215) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:D (LEU79) to (THR214) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:E (LEU79) to (THR215) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:F (LEU79) to (THR215) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:G (LEU79) to (THR215) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:H (LEU79) to (THR215) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:I (LEU79) to (THR215) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:J (LEU79) to (THR214) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:K (LEU79) to (THR215) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:L (LEU79) to (THR215) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
1pyx:A (GLY68) to (GLN206) GSK-3 BETA COMPLEXED WITH AMP-PNP | KINASE, INSULIN PATHWAY, TRANSFERASE
4y73:A (GLY198) to (SER336) CRYSTAL STRUCTURE OF IRAK4 KINASE DOMAIN WITH INHIBITOR | KINASE, INHIBITOR
4y73:C (GLY198) to (SER336) CRYSTAL STRUCTURE OF IRAK4 KINASE DOMAIN WITH INHIBITOR | KINASE, INHIBITOR
4y73:D (GLY198) to (SER336) CRYSTAL STRUCTURE OF IRAK4 KINASE DOMAIN WITH INHIBITOR | KINASE, INHIBITOR
3tei:A (TYR36) to (ALA174) CRYSTAL STRUCTURE OF HUMAN ERK2 COMPLEXED WITH A MAPK DOCKING PEPTIDE | TRANSFERASE
2r7i:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF CATALYTIC SUBUNIT OF PROTEIN KINASE CK2 | CATALYTIC SUBUNIT, KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
2r7i:B (TYR50) to (PHE181) CRYSTAL STRUCTURE OF CATALYTIC SUBUNIT OF PROTEIN KINASE CK2 | CATALYTIC SUBUNIT, KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
2r7i:C (GLU52) to (PHE181) CRYSTAL STRUCTURE OF CATALYTIC SUBUNIT OF PROTEIN KINASE CK2 | CATALYTIC SUBUNIT, KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
2r7i:D (SER51) to (PHE181) CRYSTAL STRUCTURE OF CATALYTIC SUBUNIT OF PROTEIN KINASE CK2 | CATALYTIC SUBUNIT, KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
1q3d:A (GLY68) to (GLN206) GSK-3 BETA COMPLEXED WITH STAUROSPORINE | KINASE, INSULIN PATHWAY, TRANSFERASE
4y83:A (PHE149) to (GLN276) CRYSTAL STRUCTURE OF COT KINASE DOMAIN IN COMPLEX WITH 5-(2-AMINO-5- (QUINOLIN-3-YL)PYRIDIN-3-YL)-1,3,4-OXADIAZOLE-2(3H)-THIONE | COT, TPL-2, MAP3K8, KINASE, INHIBITOR, COMPLEX, TRANSFERASE
4y83:B (PHE149) to (MET277) CRYSTAL STRUCTURE OF COT KINASE DOMAIN IN COMPLEX WITH 5-(2-AMINO-5- (QUINOLIN-3-YL)PYRIDIN-3-YL)-1,3,4-OXADIAZOLE-2(3H)-THIONE | COT, TPL-2, MAP3K8, KINASE, INHIBITOR, COMPLEX, TRANSFERASE
3tjc:A (PHE860) to (GLN1003) CO-CRYSTAL STRUCTURE OF JAK2 WITH THIENOPYRIDINE 8 | JAK2, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3tjc:B (GLY861) to (GLN1003) CO-CRYSTAL STRUCTURE OF JAK2 WITH THIENOPYRIDINE 8 | JAK2, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3tjd:A (GLY861) to (GLN1003) CO-CRYSTAL STRUCTURE OF JAK2 WITH THIENOPYRIDINE 19 | JAK2, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3tjd:B (GLY861) to (GLN1003) CO-CRYSTAL STRUCTURE OF JAK2 WITH THIENOPYRIDINE 19 | JAK2, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3tnh:A (GLY31) to (ALA173) CDK9/CYCLIN T IN COMPLEX WITH CAN508 | KINASE, CYCLIN, PHOSPHTRANSFER, CYCLIN T, PHOSPHORYLATED ON THREONINE 186, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3tni:A (GLU32) to (ALA173) STRUCTURE OF CDK9/CYCLIN T F241L | CYCLIN DEPENDENT KINASE, KINASE ,CYCLIN, PHOSPHOTRANSFER, CDK-CYCLIN COMPLEX, PHOSPHORYLATED ON THREONINE 186, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jg8:A (SER434) to (LEU568) STRUCTURE OF RSK2 T493M CTD MUTANT BOUND TO 2-CYANO-N-(1-HYDROXY-2- METHYLPROPAN-2-YL)-3-(3-(3,4,5-TRIMETHOXYPHENYL)-1H-INDAZOL-5-YL) ACRYLAMIDE | PROTEIN KINASE, PHOSPHORYLATION, COVALENT INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4ji9:A (PHE860) to (GLN1003) JAK2 KINASE (JH1 DOMAIN) IN COMPLEX WITH TG101209 | PROTEIN KINASE, PHOSPHO-TRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ji9:B (GLY861) to (GLN1003) JAK2 KINASE (JH1 DOMAIN) IN COMPLEX WITH TG101209 | PROTEIN KINASE, PHOSPHO-TRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1ql6:A (SER31) to (GLN173) THE CATALYTIC MECHANISM OF PHOSPHORYLASE KINASE PROBED BY MUTATIONAL STUDIES | KINASE (GLYCOGEN METABOLISM), GLYCOGEN METABOLISM, TRANSFERASE, SERINE/THREONINE-PROTEIN, KINASE, ATP-BINDING, CALMODULIN-BINDING
3h30:B (SER51) to (PHE181) CRYSTAL STRUCTURE OF THE CATALYTIC SUBUNIT OF HUMAN PROTEIN KINASE CK2 WITH 5,6-DICHLORO-1-BETA-D- RIBOFURANOSYLBENZIMIDAZOLE | PROTEIN KINASE CK2, CASEIN KINASE 2, CASEIN KINASE II, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
1f0q:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF THE ALPHA SUBUNIT OF PROTEIN KINASE CK2 IN COMPLEX WITH THE NUCLEOTIDE COMPETITIVE INHIBITOR EMODIN | PROTEIN KINASE-INHIBITOR COMPLEX, TRANSFERASE
4ylj:A (GLN172) to (GLN313) CRYSTAL STRUCTURE OF DYRK1A IN COMPLEX WITH 10-IODO-SUBSTITUTED 11H- INDOLO[3,2-C]QUINOLINE-6-CARBOXYLIC ACID INHIBITOR 5J | HALOGEN, INHIBITOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ylj:B (GLY171) to (GLN313) CRYSTAL STRUCTURE OF DYRK1A IN COMPLEX WITH 10-IODO-SUBSTITUTED 11H- INDOLO[3,2-C]QUINOLINE-6-CARBOXYLIC ACID INHIBITOR 5J | HALOGEN, INHIBITOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ylj:C (GLY171) to (GLN313) CRYSTAL STRUCTURE OF DYRK1A IN COMPLEX WITH 10-IODO-SUBSTITUTED 11H- INDOLO[3,2-C]QUINOLINE-6-CARBOXYLIC ACID INHIBITOR 5J | HALOGEN, INHIBITOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ylj:D (GLY171) to (GLN313) CRYSTAL STRUCTURE OF DYRK1A IN COMPLEX WITH 10-IODO-SUBSTITUTED 11H- INDOLO[3,2-C]QUINOLINE-6-CARBOXYLIC ACID INHIBITOR 5J | HALOGEN, INHIBITOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ylk:A (GLY171) to (GLN313) CRYSTAL STRUCTURE OF DYRK1A IN COMPLEX WITH 10-CHLORO-SUBSTITUTED 11H- INDOLO[3,2-C]QUINOLONE-6-CARBOXYLIC ACID INHIBITOR 5S | HALOGEN, INHIBITOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yll:A (GLN172) to (GLN313) CRYSTAL STRUCTURE OF DYRK1AA IN COMPLEX WITH 10-BROMO-SUBSTITUTED 11H- INDOLO[3,2-C]QUINOLONE-6-CARBOXYLIC ACID INHIBITOR 5T | HALOGEN, INHIBITOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1r0e:B (GLY68) to (GLN206) GLYCOGEN SYNTHASE KINASE-3 BETA IN COMPLEX WITH 3-INDOLYL-4- ARYLMALEIMIDE INHIBITOR | SER/THR PROTEIN KINASE, TRANSFERASE
3u87:A (SER51) to (PHE181) STRUCTURE OF A CHIMERIC CONSTRUCT OF HUMAN CK2ALPHA AND HUMAN CK2ALPHA' IN COMPLEX WITH A NON-HYDROLYSABLE ATP-ANALOGUE | PROTEIN KINASE CK2 CASEIN KINASE 2, PROTEIN KINASE FOLD, EUKARYOTIC PROTEIN KINASE, TRANSFERASE
3u87:B (SER51) to (PHE181) STRUCTURE OF A CHIMERIC CONSTRUCT OF HUMAN CK2ALPHA AND HUMAN CK2ALPHA' IN COMPLEX WITH A NON-HYDROLYSABLE ATP-ANALOGUE | PROTEIN KINASE CK2 CASEIN KINASE 2, PROTEIN KINASE FOLD, EUKARYOTIC PROTEIN KINASE, TRANSFERASE
3u8w:A (GLY36) to (THR175) CRYSTAL STRUCTURE OF P38A MITOGEN-ACTIVATED PROTEIN KINASE IN COMPLEX WITH A TRIAZOLOPYRIDAZINONE INHIBITOR | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2uzd:C (GLY16) to (ALA151) CRYSTAL STRUCTURE OF HUMAN CDK2 COMPLEXED WITH A THIAZOLIDINONE INHIBITOR | TRANSFERASE, ATP-BINDING, PHOSPHORYLATION, CDK2, KINASE, CYCLIN, MITOSIS, CELL CYCLE, CELL DIVISION, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, THIAZOLIDINONE LIGAND
4yo6:C (GLY198) to (SER336) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yo6:D (GLY198) to (SER336) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yp8:A (GLY198) to (SER336) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yp8:C (GLY198) to (SER336) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yp8:D (GLY198) to (SER336) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2v22:A (GLY16) to (GLY153) REPLACE: A STRATEGY FOR ITERATIVE DESIGN OF CYCLIN BINDING GROOVE INHIBITORS | POLYMORPHISM, CYCLIN GROOVE, CELL DIVISION, CDK2, KINASE, CYCLIN, ACTIVE, MITOSIS, INHIBITION, PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE, NONPEPTIDE, TRANSFERASE, ATP-BINDING
1fin:C (GLY16) to (GLY153) CYCLIN A-CYCLIN-DEPENDENT KINASE 2 COMPLEX | COMPLEX (TRANSFERASE/CYCLIN), CYCLIN, CDK, PHOSPHORYLATION
2erk:A (MET36) to (ASP175) PHOSPHORYLATED MAP KINASE ERK2 | PHOSPHOTRANSFERASE, KINASE, SERINE/THREONINE-PROTEIN KINASE
4ytf:A (GLY861) to (GLN1003) DISCOVERY OF VX-509 (DECERNOTINIB): A POTENT AND SELECTIVE JANUS KINASE (JAK) 3 INHIBITOR FOR THE TREATMENT OF AUTOIMMUNE DISEASES | JANUS KINASE, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1fq1:B (GLY16) to (PHE152) CRYSTAL STRUCTURE OF KINASE ASSOCIATED PHOSPHATASE (KAP) IN COMPLEX WITH PHOSPHO-CDK2 | PHOSPHO-PROTEIN/PROTEIN COMPLEX, HYDROLASE/TRANSFERASE COMPLEX
2v7o:A (PHE25) to (GLN165) CRYSTAL STRUCTURE OF HUMAN CALCIUM-CALMODULIN-DEPENDENT PROTEIN KINASE II GAMMA | KINASE, S/T KINASE, TRANSFERASE, ATP-BINDING, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, CALMODULIN-BINDING
4k6z:A (LEU891) to (THR1030) THE JAK1 KINASE DOMAIN IN COMPLEX WITH COMPOUND 37 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4k77:A (GLY887) to (THR1030) JAK1 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 6 | PROTEIN KINASE, PHOSPHOTRANSFER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1fvv:C (GLY16) to (GLY153) THE STRUCTURE OF CDK2/CYCLIN A IN COMPLEX WITH AN OXINDOLE INHIBITOR | CYCLIN-DEPENDENT KINASE, CYCLIN A, TRANSFERASE, CELL CYCLE
2f49:A (GLY25) to (ILE161) CRYSTAL STRUCTURE OF FUS3 IN COMPLEX WITH A STE5 PEPTIDE | PROTEIN-PETIDE COMPLEX, TRANSFERASE
2f57:A (GLY461) to (SER594) CRYSTAL STRUCTURE OF THE HUMAN P21-ACTIVATED KINASE 5 | PAK5, KINASE DOMAINS, GROUPII PAKS, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
2fa2:B (GLY25) to (ILE161) CRYSTAL STRUCTURE OF FUS3 WITHOUT A PEPTIDE FROM STE5 | MAP KINASE, TRANSFERASE
1gng:A (GLY68) to (GLN206) GLYCOGEN SYNTHASE KINASE-3 BETA (GSK3) COMPLEX WITH FRATTIDE PEPTIDE | TRANSFERASE, PROTEIN KINASE, GSK3/FRATTIDE COMPLEX, PHOSPHORYLATED, ACTIVE
2fys:B (MET36) to (ASP173) CRYSTAL STRUCTURE OF ERK2 COMPLEX WITH KIM PEPTIDE DERIVED FROM MKP3 | MAP KINASE, MKP3, KIM, TRANSFERASE
2fys:A (GLY35) to (ALA172) CRYSTAL STRUCTURE OF ERK2 COMPLEX WITH KIM PEPTIDE DERIVED FROM MKP3 | MAP KINASE, MKP3, KIM, TRANSFERASE
2vn9:A (SER26) to (GLN165) CRYSTAL STRUCTURE OF HUMAN CALCIUM CALMODULIN DEPENDENT PROTEIN KINASE II DELTA ISOFORM 1, CAMKD | SERINE/THREONINE-PROTEIN KINASE, SERINE-THREONINE KINASE, CELLULAR DIFFERENTIATION, VASCULAR SMOOTH MUSCLE, KINASE, TRANSFERASE, ATP-BINDING, PHOSPHOPROTEIN, CALMODULIN-BINDING, NUCLEOTIDE-BINDING
2vn9:B (SER26) to (GLN165) CRYSTAL STRUCTURE OF HUMAN CALCIUM CALMODULIN DEPENDENT PROTEIN KINASE II DELTA ISOFORM 1, CAMKD | SERINE/THREONINE-PROTEIN KINASE, SERINE-THREONINE KINASE, CELLULAR DIFFERENTIATION, VASCULAR SMOOTH MUSCLE, KINASE, TRANSFERASE, ATP-BINDING, PHOSPHOPROTEIN, CALMODULIN-BINDING, NUCLEOTIDE-BINDING
1gol:A (GLY35) to (ALA172) COORDINATES OF RAT MAP KINASE ERK2 WITH AN ARGININE MUTATION AT POSITION 52 | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, CELL CYCLE, PHOSPHORYLATION
4krc:A (THR20) to (GLY159) CRYSTAL STRUCTURE OF PHO85-PCL10-ATP-GAMMA-S COMPLEX | GLYCOGEN SYNTHESIS, GLYCOGEN SYNTHESIS REGULATION, TRANSFERASE- SIGNALING PROTEIN COMPLEX
4ks7:A (ILE420) to (SER552) PAK6 KINASE DOMAIN IN COMPLEX WITH PF-3758309 | PROTEIN KINASE, PHOSPHOTRANSFER, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4ks8:A (GLY419) to (SER552) PAK6 KINASE DOMAIN IN COMPLEX WITH SUNITINIB | PROTEIN KINASE, PHOSPHOTRANSFER, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4zim:A (GLY861) to (GLN1003) CRYSTAL STRUCTURE OF JANUS KINASE 2 IN COMPLEX WITH A 9H-CARBAZOLE-1- CARBOXAMIDE INHIBITOR | KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4zim:B (GLY861) to (GLN1003) CRYSTAL STRUCTURE OF JANUS KINASE 2 IN COMPLEX WITH A 9H-CARBAZOLE-1- CARBOXAMIDE INHIBITOR | KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4kwp:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF HUMAN CK2-ALPHA IN COMPLEX WITH A BENZIMIDAZOLE INHIBITOR (K164) AT 1.25 A RESOLUTION | KINASE, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3i5z:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK2 BOUND TO (S)-N-(2-HYDROXY-1-PHENYLETHYL)-4- (5-METHYL-2-(PHENYLAMINO)PYRIMIDIN-4-YL)-1H-PYRROLE-2-CARBOXAMIDE | KINASE, INHIBITOR, ATP-BINDING, CELL CYCLE, HOST-VIRUS INTERACTION, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4zji:A (GLY282) to (ILE414) PAK1 IN COMPLEX WITH 2-CHLORO-5-ETHYL-8-FLUORO-11-(4-METHYLPIPERAZIN- 1-YL)-DIBENZODIAZEPINE | INHIBITOR, KINASE, PAK1, ALLOSTERIC, TRANSFERASE
4zji:B (GLY282) to (ILE414) PAK1 IN COMPLEX WITH 2-CHLORO-5-ETHYL-8-FLUORO-11-(4-METHYLPIPERAZIN- 1-YL)-DIBENZODIAZEPINE | INHIBITOR, KINASE, PAK1, ALLOSTERIC, TRANSFERASE
4zjj:A (GLY282) to (ILE414) PAK1 IN COMPLEX WITH (S)-N-(TERT-BUTYL)-3-((2-CHLORO-5-ETHYL-8-FLUORO- DIBENZODIAZEPIN-11-YL)AMINO)PYRROLIDINE-1-CARBOXAMIDE | PAK1, INHIBITOR, KINASE, ALLOSTERIC, TRANSFERASE
1h26:A (VAL17) to (ALA151) CDK2/CYCLIN A IN COMPLEX WITH AN 11-RESIDUE RECRUITMENT PEPTIDE FROM P53 | CELL CYCLE, PROTEIN KINASE, CYCLIN, CDK2, RECRUITMENT, PEPTIDE SPECIFICITY
1h27:A (VAL17) to (ALA151) CDK2/CYCLIN A IN COMPLEX WITH AN 11-RESIDUE RECRUITMENT PEPTIDE FROM P27 | CELL CYCLE, PROTEIN KINASE, CYCLIN, CDK2, RECRUITMENT, PEPTIDE SPECIFICITY, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, CELL DIVISION, MITOSIS, PHOSPHORYLATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1h4l:B (GLY16) to (GLY152) STRUCTURE AND REGULATION OF THE CDK5-P25(NCK5A) COMPLEX | KINASE/KINASE ACTIVATOR, COMPLEX(CYCLINS/CDK), CYCLINS, CYCLIN-DEPENDENT KINASES, CDK5, P35, P25, TRANSFERASE, ATP-BINDING, CELL CYCLE, CELL DIVISION, PHOSPHORYLATION
2w1i:A (GLY861) to (LEU1001) STRUCTURE DETERMINATION OF AURORA KINASE IN COMPLEX WITH INHIBITOR | CHROMOSOMAL REARRANGEMENT, NUCLEOTIDE-BINDING, TYROSINE-PROTEIN KINASE, PROTO-ONCOGENE, PHOSPHOPROTEIN, DISEASE MUTATION, SH2 DOMAIN, TRANSFERASE, ATP-BINDING, POLYMORPHISM, KINASE, CANCER, AURORA, MEMBRANE, INHIBITOR
2w1i:B (GLY861) to (GLN1003) STRUCTURE DETERMINATION OF AURORA KINASE IN COMPLEX WITH INHIBITOR | CHROMOSOMAL REARRANGEMENT, NUCLEOTIDE-BINDING, TYROSINE-PROTEIN KINASE, PROTO-ONCOGENE, PHOSPHOPROTEIN, DISEASE MUTATION, SH2 DOMAIN, TRANSFERASE, ATP-BINDING, POLYMORPHISM, KINASE, CANCER, AURORA, MEMBRANE, INHIBITOR
4ztm:C (GLY198) to (SER336) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ztm:D (GLY198) to (SER336) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ztn:C (VAL199) to (SER336) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ztn:D (GLY198) to (SER336) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3io7:A (GLY861) to (GLN1003) 2-AMINOPYRAZOLO[1,5-A]PYRIMIDINES AS POTENT AND SELECTIVE INHIBITORS OF JAK2 | KINASE, INHIBITOR, JAK2, JANUS KINASE, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO- ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
4zxt:A (GLY37) to (VAL173) COMPLEX OF ERK2 WITH CATECHOL | CATECHOL COMPLEX, MITOGEN-ACTIVATED PROTEIN KINASE, SIGNAL-REGULATED KINASE, TRANSFERASE
2wel:A (SER26) to (GLN165) CRYSTAL STRUCTURE OF SU6656-BOUND CALCIUM/CALMODULIN- DEPENDENT PROTEIN KINASE II DELTA IN COMPLEX WITH CALMODULIN | CELLULAR DIFFERENTIATION, SERINE/THREONINE-PROTEIN KINASE, PHOSPHOPROTEIN, CALMODULIN-BINDING, CALMODULIN BINDING, KINASE, TRANSFERASE, ATP-BINDING, NUCLEOTIDE-BINDING, VASCULAR SMOOTH MUSCLE, SERINE-THREONINE KINASE
4ll0:A (LYS737) to (LEU862) EGFR L858R/T790M IN COMPLEX WITH PD168393 | KINASE, PD168393, 34-JAB, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2wfy:A (GLY16) to (GLY153) TRUNCATION AND OPTIMISATION OF PEPTIDE INHIBITORS OF CDK2, CYCLIN A THROUGH STRUCTURE GUIDED DESIGN | CDK2, KINASE, CYCLIN, ACTIVE, NUCLEUS, MITOSIS, SERINE/THREONINE-PROTEIN KINASE, CYTOPLASM, INHIBITION, CELL CYCLE, ATP-BINDING, CELL DIVISION, PHOSPHOPROTEIN, NUCLEOTIDE-BINDING, TRANSFERASE, POLYMORPHISM, BETA-PEPTIDE, CYCLIN GROOVE
4zzm:A (GLY37) to (VAL173) HUMAN ERK2 IN COMPLEX WITH AN IRREVERSIBLE INHIBITOR | TRANSFERASE
4zzn:A (GLY35) to (VAL171) HUMAN ERK2 IN COMPLEX WITH AN INHIBITOR | TRANSFERASE
4zzo:A (GLY37) to (VAL173) HUMAN ERK2 IN COMPLEX WITH AN IRREVERSIBLE INHIBITOR | TRANSFERASE
2whb:A (VAL17) to (GLY153) TRUNCATION AND OPTIMISATION OF PEPTIDE INHIBITORS OF CDK2, CYCLIN A THROUGH STRUCTURE GUIDED DESIGN | CDK2, KINASE, CYCLIN, ACTIVE, NUCLEUS, MITOSIS, SERINE/THREONINE-PROTEIN KINASE, CYTOPLASM, INHIBITION, CELL CYCLE, ATP-BINDING, CELL DIVISION, PHOSPHOPROTEIN, NUCLEOTIDE-BINDING, TRANSFERASE, POLYMORPHISM, BETA-PEPTIDE, CYCLIN GROOVE
2wih:A (GLY16) to (GLY153) STRUCTURE OF CDK2-CYCLIN A WITH PHA-848125 | CELL CYCLE, ATP-BINDING, TRANSFERASE, POLYMORPHISM, PHOSPHORYLATION, NUCLEOTIDE-BINDING, CELL DIVISION, SERINE/THREONINE-PROTEIN 2 KINASE, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, MITOSIS
2wih:C (GLY16) to (GLY153) STRUCTURE OF CDK2-CYCLIN A WITH PHA-848125 | CELL CYCLE, ATP-BINDING, TRANSFERASE, POLYMORPHISM, PHOSPHORYLATION, NUCLEOTIDE-BINDING, CELL DIVISION, SERINE/THREONINE-PROTEIN 2 KINASE, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, MITOSIS
1u5q:B (ALA41) to (MET176) CRYSTAL STRUCTURE OF THE TAO2 KINASE DOMAIN: ACTIVATION AND SPECIFITY OF A STE20P MAP3K | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE
3w8l:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF HUMAN CK2 IN COMPLEX WITH INOSITOL HEXAKISPHOSPHATE | PROTEIN KINASE CK2, APOPTOSIS
3w8l:B (GLU55) to (PHE181) CRYSTAL STRUCTURE OF HUMAN CK2 IN COMPLEX WITH INOSITOL HEXAKISPHOSPHATE | PROTEIN KINASE CK2, APOPTOSIS
1ung:A (GLY16) to (GLY152) STRUCTURAL MECHANISM FOR THE INHIBITION OF CDK5-P25 BY ROSCOVITINE, ALOISINE AND INDIRUBIN. | CELL CYCLE, COMPLEX(KINASE/ACTIVATOR), INHIBITORS, NEURODEGENERATIVE DISEASES
1ung:B (THR17) to (GLY152) STRUCTURAL MECHANISM FOR THE INHIBITION OF CDK5-P25 BY ROSCOVITINE, ALOISINE AND INDIRUBIN. | CELL CYCLE, COMPLEX(KINASE/ACTIVATOR), INHIBITORS, NEURODEGENERATIVE DISEASES
1unh:A (GLY16) to (GLY152) STRUCTURAL MECHANISM FOR THE INHIBITION OF CDK5-P25 BY ROSCOVITINE, ALOISINE AND INDIRUBIN. | CELL CYCLE, NEURODEGENERATIVE DISEASES, INDIRUBIN
1unh:B (GLY16) to (GLY152) STRUCTURAL MECHANISM FOR THE INHIBITION OF CDK5-P25 BY ROSCOVITINE, ALOISINE AND INDIRUBIN. | CELL CYCLE, NEURODEGENERATIVE DISEASES, INDIRUBIN
1unl:A (GLY16) to (GLY152) STRUCTURAL MECHANISM FOR THE INHIBITION OF CD5-P25 FROM THE ROSCOVITINE, ALOISINE AND INDIRUBIN. | CYCLIN DEPENDENT KINASE, INHIBITOR, ATP-ANALOGUE, NEURODEGENERATIVE DISEASES
1unl:B (GLY16) to (GLY152) STRUCTURAL MECHANISM FOR THE INHIBITION OF CD5-P25 FROM THE ROSCOVITINE, ALOISINE AND INDIRUBIN. | CYCLIN DEPENDENT KINASE, INHIBITOR, ATP-ANALOGUE, NEURODEGENERATIVE DISEASES
1urc:C (GLY16) to (GLY153) CYCLIN A BINDING GROOVE INHIBITOR ACE-ARG-LYS-LEU-PHE-GLY | TRANSFERASE-INHIBITOR COMPLEX, INHIBITOR, LIGAND EXCHANGE, DRUG DESIGN, PEPTIDOMIMETICS
4md8:E (SER51) to (PHE181) CRYSTAL STRUCTURE OF FULL-LENGTH SYMMETRIC CK2 HOLOENZYME WITH MUTATED ALPHA SUBUNIT (F121E) | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
4md8:F (SER51) to (PHE181) CRYSTAL STRUCTURE OF FULL-LENGTH SYMMETRIC CK2 HOLOENZYME WITH MUTATED ALPHA SUBUNIT (F121E) | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
3wi6:D (LEU79) to (THR215) CRYSTAL STRUCTURE OF MAPKAP KINASE-2 (MK2) IN COMPLEX WITH NON- SELECTIVE INHIBITOR | GLY-RICH LOOP FORMED, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3wik:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF THE CK2ALPHA/COMPOUND10 COMPLEX | TRANSFERASE
1v0o:B (GLY16) to (PHE150) STRUCTURE OF P. FALCIPARUM PFPK5-INDIRUBIN-5-SULPHONATE LIGAND COMPLEX | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, CDK
5air:A (GLY68) to (GLN206) STRUCTURAL ANALYSIS OF MOUSE GSK3BETA FUSED WITH LRP6 PEPTIDE. | TRANSFERASE, LRP6, GSK3 BETA
1j91:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF Z. MAYS CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE ATP-COMPETITIVE INHIBITOR 4,5,6,7- TETRABROMOBENZOTRIAZOLE | CK2, CASEIN KINASE 2, INHIBITORS, TETRABROMO-BENZOTRIAZOLE, TRANSFERASE
1j91:B (SER51) to (PHE181) CRYSTAL STRUCTURE OF Z. MAYS CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE ATP-COMPETITIVE INHIBITOR 4,5,6,7- TETRABROMOBENZOTRIAZOLE | CK2, CASEIN KINASE 2, INHIBITORS, TETRABROMO-BENZOTRIAZOLE, TRANSFERASE
2xa4:A (PHE860) to (GLN1003) INHIBITORS OF JAK2 KINASE DOMAIN | KINASE, MEMBRANE, TRANSFERASE, ATP-BINDING, PROTO-ONCOGENE, PHOSPHOPROTEIN
2j0i:A (GLY333) to (SER466) CRYSTAL STRUCTURE OF THE HUMAN P21-ACTIVATED KINASE 4 | PROTEIN KINASE, PHOSPHORYLATION, NUCLEOTIDE-BINDING, PAK4, STE20, KINASE, TRANSFERASE, ATP-BINDING, ALTERNATIVE SPLICING, SERINE/THREONINE-PROTEIN KINASE
4mwh:A (GLU53) to (PHE220) CRYSTAL STRUCTURE OF SCCK2 ALPHA IN COMPLEX WITH ATP | PROTEIN KINASE, PROTEIN PHOSPHORYLATION, TRANSFERASE
1jwh:B (SER51) to (PHE181) CRYSTAL STRUCTURE OF HUMAN PROTEIN KINASE CK2 HOLOENZYME | CASEIN KINASE 2, CK2 HOLOENZYME, PROTEIN KINASE CK2, TRANSFERASE
4n0s:A (GLY37) to (VAL173) COMPLEX OF ERK2 WITH CAFFEIC ACID | CAFFEIC ACID COMPLEX, MITOGEN-ACTIVATED PROTEIN KINASE, SIGNAL- REGULATED KINASE, TRANSFERASE
5b0x:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF THE CK2A/BENZOIC ACID DERIVATIVE COMPLEX | INHIBITOR, COMPLEX, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2jbo:A (LEU79) to (THR215) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-1, SOAKING) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, MK2, KINASE, ATP SITE, TRANSFERASE, ATP-BINDING, SERINE/THREONINE-PROTEIN KINASE, SMALL MOLECULE INHIBITOR, NUCLEOTIDE-BINDING
2jbp:A (LEU79) to (THR214) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:B (LYS77) to (THR214) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:E (LEU79) to (THR215) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:F (GLY76) to (THR215) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:G (GLY76) to (THR215) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:K (LYS77) to (THR214) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:L (LYS77) to (THR215) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
3zc6:B (GLY834) to (LEU974) CRYSTAL STRUCTURE OF JAK3 KINASE DOMAIN IN COMPLEX WITH AN INDAZOLE SUBSTITUTED PYRROLOPYRAZINE INHIBITOR | TRANSFERASE, SCID, SEVERE COMBINED IMMUNODEFICIENCY, STAT5, STAT6, INTERLEUKIN-2, COMMON-GAMMA CHAIN, ATP SITE KINASE INHIBITOR, CANCER
2jfm:A (GLY46) to (THR181) CRYSTAL STRUCTURE OF HUMAN STE20-LIKE KINASE (UNLIGANDED FORM) | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, MUSCLE DEVELOPMENT, KINASE, APOPTOSIS, GERMINAL CENTRE KINASE, SERINE- THREONINE KINASE 2, NUCLEOTIDE-BINDING, SERINE-THREONINE-PROTEIN KINASE
5bms:A (ILE334) to (SER466) CRYSTAL STRUCTURE OF P21-ACTIVATED KINASE 4 IN COMPLEX WITH AN INHIBITOR COMPOUND 29 | KINASE, INHIBITOR, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2jii:B (GLY178) to (CYS334) STRUCTURE OF VACCINIA RELATED KINASE 3 | TRANSFERASE, PSEUDO KINASE DOMAIN, VACCINIA RELATED KINASE, SERINE/THREONINE-PROTEIN KINASE, VRK3, KINASE, ATP-BINDING, NUCLEOTIDE-BINDING
4nct:B (GLN172) to (LEU314) HUMAN DYRK1A IN COMPLEX WITH PKC412 | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5bui:A (GLY35) to (VAL171) ERK2 COMPLEXED WITH 2-PYRIDIYL TETRAHYDROAZAINDAZOLE | ERK2, MITOGEN-ACTIVATED PROTEIN KINASE 1, ATP-INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5buj:A (GLY35) to (ALA172) ERK2 COMPLEXED WITH A N-H TETRAHYDROAZAINDAZOLE | ERK2, MITOGEN-ACTIVATED PROTEIN KINASE 1, ATP INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5bve:A (GLY35) to (VAL171) TETRAHYDROPYRROLO-DIAZEPENONES AS INHIBITORS OF ERK2 KINASE | INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4nh1:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF A HETEROTETRAMERIC CK2 HOLOENZYME COMPLEX CARRYING THE ANDANTE-MUTATION IN CK2BETA AND CONSISTENT WITH PROPOSED MODELS OF AUTOINHIBITION AND TRANS-AUTOPHOSPHORYLATION | EUKARYOTIC PROTEIN KINASE FOLD, PHOSPHOTRANSFERASE (KINASE), PHOSPHORYLATION, TRANSFERASE
4nh1:B (SER51) to (PHE181) CRYSTAL STRUCTURE OF A HETEROTETRAMERIC CK2 HOLOENZYME COMPLEX CARRYING THE ANDANTE-MUTATION IN CK2BETA AND CONSISTENT WITH PROPOSED MODELS OF AUTOINHIBITION AND TRANS-AUTOPHOSPHORYLATION | EUKARYOTIC PROTEIN KINASE FOLD, PHOSPHOTRANSFERASE (KINASE), PHOSPHORYLATION, TRANSFERASE
4nif:B (GLY37) to (ALA174) HETERODIMERIC STRUCTURE OF ERK2 AND RSK1 | KINASE DOMAIN, SIGNALING, SUBSTRATE KINASE BINDING, TRANSFERASE
4nif:E (GLY37) to (VAL173) HETERODIMERIC STRUCTURE OF ERK2 AND RSK1 | KINASE DOMAIN, SIGNALING, SUBSTRATE KINASE BINDING, TRANSFERASE
4njd:A (GLY333) to (SER466) STRUCTURE OF P21-ACTIVATED KINASE 4 WITH A NOVEL INHIBITOR KY-04031 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2y9q:A (GLY37) to (ALA174) CRYSTAL STRUCTURE OF HUMAN ERK2 COMPLEXED WITH A MAPK DOCKING PEPTIDE | TRANSFERASE, SIGNALING, PROTEIN-PROTEIN INTERACTION
3zu7:A (MET36) to (VAL171) CRYSTAL STRUCTURE OF A DESIGNED SELECTED ANKYRIN REPEAT PROTEIN IN COMPLEX WITH THE MAP KINASE ERK2 | TRANSFERASE-DE NOVO PROTEIN COMPLEX, TRANSFERASE, SELECTED BINDER, PROTEIN DESIGN
3zuv:A (GLY35) to (ASP175) CRYSTAL STRUCTURE OF A DESIGNED SELECTED ANKYRIN REPEAT PROTEIN IN COMPLEX WITH THE PHOSPHORYLATED MAP KINASE ERK2 | DE NOVO PROTEIN-TRANSFERASE COMPLEX, ANKYRIN REPEAT PROTEIN, SELECTED BINDER, PROTEIN DESIGN
4nu1:A (GLY68) to (GLN206) CRYSTAL STRUCTURE OF A TRANSITION STATE MIMIC OF THE GSK-3/AXIN COMPLEX BOUND TO PHOSPHORYLATED N-TERMINAL AUTO-INHIBITORY PS9 PEPTIDE | WNT, LRP6, GSK-3, AXIN, KINASE, PRIMED SUBSTRATE, TRANSITION STATE, PHOSPHORYLATED N-TERMINAL AUTO-INHIBITORY PS9 PEPTIDE, TRANSFERASE- PEPTIDE COMPLEX
4o0y:A (ILE334) to (SER466) BACK POCKET FLEXIBILITY PROVIDES GROUP-II PAK SELECTIVITY FOR TYPE 1 KINASE INHIBITORS | PAK4, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2nru:B (VAL199) to (GLU337) CRYSTAL STRUCTURE OF IRAK-4 | KINASE, INHIBITOR, IRAK, TRANSFERASE
2nru:D (VAL199) to (GLU337) CRYSTAL STRUCTURE OF IRAK-4 | KINASE, INHIBITOR, IRAK, TRANSFERASE
2nry:B (GLY198) to (SER336) CRYSTAL STRUCTURE OF IRAK-4 | KINASE, INHIBITOR, STAUROSPORINE, TRANSFERASE
2nry:C (GLY198) to (SER336) CRYSTAL STRUCTURE OF IRAK-4 | KINASE, INHIBITOR, STAUROSPORINE, TRANSFERASE
3juh:B (SER51) to (PHE181) CRYSTAL STRUCTURE OF A MUTANT OF HUMAN PROTEIN KINASE CK2ALPHA WITH ALTERED COSUBSTRATE SPECIFICITY | EUKARYOTIC PROTEIN KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
4o6e:A (GLY37) to (VAL173) DISCOVERY OF 5,6,7,8-TETRAHYDROPYRIDO[3,4-D]PYRIMIDINE INHIBITORS OF ERK2 | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5cf4:A (GLY861) to (GLN1003) CRYSTAL STRUCTURE OF JANUS KINASE 2 IN COMPLEX WITH N,N-DICYCLOPROPYL- 10-ETHYL-7-[(3-METHOXYPROPYL)AMINO] -3-METHYL-3,5,8,10- TETRAAZATRICYCLO[7.3.0.0,6] DODECA-1(9),2(6),4,7,11-PENTAENE-11- CARBOXAMIDE | KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5cf4:B (GLY861) to (GLN1003) CRYSTAL STRUCTURE OF JANUS KINASE 2 IN COMPLEX WITH N,N-DICYCLOPROPYL- 10-ETHYL-7-[(3-METHOXYPROPYL)AMINO] -3-METHYL-3,5,8,10- TETRAAZATRICYCLO[7.3.0.0,6] DODECA-1(9),2(6),4,7,11-PENTAENE-11- CARBOXAMIDE | KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5cf5:A (GLY861) to (GLN1003) CRYSTAL STRUCTURE OF JANUS KINASE 2 IN COMPLEX WITH N,N-DICYCLOPROPYL- 7-[(DIMETHYL-1,3-THIAZOL-2-YL)AMINO]-10-ETHYL-3-METHYL-3,5,8,10- TETRAAZATRICYCLO[7.3.0.02,6] DODECA-1(9),2(6),4,7,11-PENTAENE-11- CARBOXAMIDE | KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5cf5:B (GLY861) to (GLN1003) CRYSTAL STRUCTURE OF JANUS KINASE 2 IN COMPLEX WITH N,N-DICYCLOPROPYL- 7-[(DIMETHYL-1,3-THIAZOL-2-YL)AMINO]-10-ETHYL-3-METHYL-3,5,8,10- TETRAAZATRICYCLO[7.3.0.02,6] DODECA-1(9),2(6),4,7,11-PENTAENE-11- CARBOXAMIDE | KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5cf6:A (GLY861) to (GLN1003) CRYSTAL STRUCTURE OF JANUS KINASE 2 IN COMPLEX WITH N,N-DICYCLOPROPYL- 10-[(2S)-2,3-DIHYDROXYPROPYL]-3-METHYL-7-(METHYLAMINO)-3,5,8,10- TETRAAZATRICYCLO [7.3.0.02,6]DODECA-1(9),2(6),4,7,11-PENTAENE-11- CARBOXAMIDE | KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5cf6:B (GLY861) to (GLN1003) CRYSTAL STRUCTURE OF JANUS KINASE 2 IN COMPLEX WITH N,N-DICYCLOPROPYL- 10-[(2S)-2,3-DIHYDROXYPROPYL]-3-METHYL-7-(METHYLAMINO)-3,5,8,10- TETRAAZATRICYCLO [7.3.0.02,6]DODECA-1(9),2(6),4,7,11-PENTAENE-11- CARBOXAMIDE | KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3jy9:A (GLY861) to (GLN1003) JANUS KINASE 2 INHIBITORS | KINASE, INHIBITOR, JAK2, JANUS KINASE, ATP-BINDING, DISEASE MUTATION, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3k2l:A (GLY161) to (TYR301) CRYSTAL STRUCTURE OF DUAL-SPECIFICITY TYROSINE PHOSPHORYLATION REGULATED KINASE 2 (DYRK2) | DYRK2, DUAL-SPECIFICITY TYROSINE-(Y)-PHOSPHORYLATION REGULATED KINASE 2, PSK-H2, KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, APOPTOSIS, ATP-BINDING, MAGNESIUM, MANGANESE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE
4ogr:E (GLU32) to (ALA173) CRYSTAL STRUCTURE OF P-TEFB COMPLEX WITH AFF4 AND TAT | P-TEFB, CYCLIN-DEPENDENT KINASE 9, CYCLIN FOLD, INTRINSICALLY UNSTRUCTURED AFF4, TRANSCRIPTIONAL REGULATION AT HIV PROMOTER, BINDS TAR, N-TERMINAL ACETYLATION OF TAT, TRANSFERASE-VIRAL PROTEIN COMPLEX
5clp:B (SER51) to (PHE181) CRYSTAL STRUCTURE OF CK2ALPHA WITH 3,4-DICHLOROPHENETHYLAMINE BOUND | TRANSFERASE, CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION
4oh4:A (GLY895) to (SER1035) CRYSTAL STRUCTURE OF BRI1 IN COMPLEX WITH BKI1 | KINASE DOMAIN, TRANSFERASE, ATP BINDING, PHOSPHORYLATION, MEMBRANE, TRANSFERASE-SIGNALING PROTEIN COMPLEX
1lpu:A (SER51) to (PHE181) LOW TEMPERATURE CRYSTAL STRUCTURE OF THE APO-FORM OF THE CATALYTIC SUBUNIT OF PROTEIN KINASE CK2 FROM ZEA MAYS | PROTEIN KINASE, CK2, CASEIN KINASE 2, DUAL-COSUBSTRATE SPECIFICITY, TRANSFERASE
5cqw:A (SER51) to (PHE181) TETRAGONAL COMPLEX STRUCTURE OF PROTEIN KINASE CK2 CATALYTIC SUBUNIT WITH A BENZOTRIAZOLE-BASED INHIBITOR GENERATED BY CLICK-CHEMISTRY | TRANSFERASE, ATP-COMPETITIVE INHIBITOR, PROTEIN KINASE CK2, CASEIN KINASE 2
5cqw:B (SER51) to (PHE181) TETRAGONAL COMPLEX STRUCTURE OF PROTEIN KINASE CK2 CATALYTIC SUBUNIT WITH A BENZOTRIAZOLE-BASED INHIBITOR GENERATED BY CLICK-CHEMISTRY | TRANSFERASE, ATP-COMPETITIVE INHIBITOR, PROTEIN KINASE CK2, CASEIN KINASE 2
1xo2:B (LYS26) to (TYR170) CRYSTAL STRUCTURE OF A HUMAN CYCLIN-DEPENDENT KINASE 6 COMPLEX WITH A FLAVONOL INHIBITOR, FISETIN | CRYSTAL STRUCTURE,HUMAN CYCLIN-DEPENDENT KINASE 6, FISETIN, CELL CYCLE-TRANSFERASE COMPLEX
1m2p:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF 1,8-DI-HYDROXY-4-NITRO- ANTHRAQUINONE/CK2 KINASE COMPLEX | KINASE, INHIBITOR-ENZYME COMPLEX, TRANSFERASE
1m2q:A (TYR50) to (PHE181) CRYSTAL STRUCTURE OF 1,8-DI-HYDROXY-4-NITRO-XANTEN-9- ONE/CK2 KINASE COMPLEX | KINASE, INHIBITOR-ENZYME COMPLEX, TRANSFERASE
5ct0:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF CK2ALPHA WITH 3-(3-CHLORO-4-(PHENYL)BENZYLAMINO) PROPAN-1-OL BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
3kcf:B (GLY217) to (ASP359) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A PYRAZOLONE INHIBITOR | KINASE, TGFBETARI, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, AORTIC ANEURYSM, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3kck:A (GLY861) to (LEU1001) A NOVEL CHEMOTYPE OF KINASE INHIBITORS | KINASE, INHIBITOR, JAK2, JANUS KINASE, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO- ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
5cu2:B (SER51) to (PHE181) CRYSTAL STRUCTURE OF CK2ALPHA WITH 2-HYDROXY-5-METHYLBENZOIC ACID AND (METHYL 4-((3-(3-CHLORO-4-(PHENYL)BENZYLAMINO)PROPYL)AMINO)-4- OXOBUTANOAT BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
5cu3:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF CK2ALPHA WITH COMPOUND 10 BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
5cu3:B (GLU55) to (PHE181) CRYSTAL STRUCTURE OF CK2ALPHA WITH COMPOUND 10 BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
2zjw:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF HUMAN CK2 ALPHA COMPLEXED WITH ELLAGIC ACID | PROTEIN-INHIBITOR COMPLEX, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
5cvf:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF CK2ALPHA WITH COMPOUND 5 BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
5cvh:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF CK2ALPHA | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
5cvh:B (SER51) to (PHE181) CRYSTAL STRUCTURE OF CK2ALPHA | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
4or5:A (GLU32) to (ALA173) CRYSTAL STRUCTURE OF HIV-1 TAT COMPLEXED WITH HUMAN P-TEFB AND AFF4 | CDK9, TAT, AFF4, ZINC FINGER, TRANSCRIPTION, RNA BINDING, PHOSPHORYLATION, TRANSFERASE-TRANSCRIPTION COMPLEX
5cx9:B (SER51) to (PHE181) CRYSTAL STRUCTURE OF CK2ALPHA WITH (METHYL 4-((3-(3-CHLORO-4-(PHENYL) BENZYLAMINO)PROPYL)AMINO)-4-OXOBUTANOATE BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
2zoq:A (GLY54) to (ALA191) STRUCTURAL DISSECTION OF HUMAN MITOGEN-ACTIVATED KINASE ERK1 | SERINE/THREONINE KINASE, ERK1, ACETYLATION, ATP-BINDING, CELL CYCLE, HOST-VIRUS INTERACTION, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kga:A (ASN75) to (THR214) CRYSTAL STRUCTURE OF MAPKAP KINASE 2 (MK2) COMPLEXED WITH A POTENT 3-AMINOPYRAZOLE ATP SITE INHIBITOR | SMALL MOLECULE INHIBITOR, 3-AMINOPYRAZOLE SCAFFOLD, SCAFFOLD HOPING, ATP-SITE KINASE INHIBITOR, INDUCED FIT, NOVEL HYDROPHOBIC POCKET, ACTIVATION LOOP DELETION, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kl8:C (SER25) to (VAL163) CAMKIINTIDE INHIBITOR COMPLEX | CAMKII, CAMKIINTIDE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL JUNCTION, CELL MEMBRANE, MEMBRANE, POSTSYNAPTIC CELL MEMBRANE, PROTEIN KINASE INHIBITOR, SYNAPSE, SYNAPTOSOME, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3kl8:E (SER25) to (VAL163) CAMKIINTIDE INHIBITOR COMPLEX | CAMKII, CAMKIINTIDE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL JUNCTION, CELL MEMBRANE, MEMBRANE, POSTSYNAPTIC CELL MEMBRANE, PROTEIN KINASE INHIBITOR, SYNAPSE, SYNAPTOSOME, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3kl8:G (SER25) to (VAL163) CAMKIINTIDE INHIBITOR COMPLEX | CAMKII, CAMKIINTIDE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL JUNCTION, CELL MEMBRANE, MEMBRANE, POSTSYNAPTIC CELL MEMBRANE, PROTEIN KINASE INHIBITOR, SYNAPSE, SYNAPTOSOME, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3kl8:I (SER25) to (VAL163) CAMKIINTIDE INHIBITOR COMPLEX | CAMKII, CAMKIINTIDE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL JUNCTION, CELL MEMBRANE, MEMBRANE, POSTSYNAPTIC CELL MEMBRANE, PROTEIN KINASE INHIBITOR, SYNAPSE, SYNAPTOSOME, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4p7e:A (GLY861) to (GLN1003) TRIAZOLOPYRIDINE COMPOUNDS AS SELECTIVE JAK1 INHIBITORS: FROM HIT IDENTIFICATION TO GLPG0634 | TRANSFERASE, JAK1 INHIBITOR, TRIAZOLOPYRIDINE
4p7e:B (GLY861) to (GLN1003) TRIAZOLOPYRIDINE COMPOUNDS AS SELECTIVE JAK1 INHIBITORS: FROM HIT IDENTIFICATION TO GLPG0634 | TRANSFERASE, JAK1 INHIBITOR, TRIAZOLOPYRIDINE
4p90:A (GLY282) to (ILE414) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN PAK1 IN COMPLEX WITH COMPOUND 15 | INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4pdp:A (ALA210) to (GLN346) CRYSTAL STRUCTURE OF RAD53 KINASE DOMAIN AND SCD2 | SER/THR KINASE DOMAIN, N-LOBE, C-LOBE, ACTIVATION SEGMENT EXCHANGE, TRANSFERASE
4pdp:B (LYS213) to (GLN346) CRYSTAL STRUCTURE OF RAD53 KINASE DOMAIN AND SCD2 | SER/THR KINASE DOMAIN, N-LOBE, C-LOBE, ACTIVATION SEGMENT EXCHANGE, TRANSFERASE
3a7g:B (LYS40) to (THR170) HUMAN MST3 KINASE | TWO-LOBE PROTEIN KINASE FOLD, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, TRANSFERASE
3kxg:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF Z. MAYS CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE INHIBITOR 3,4,5,6,7-PENTABROMO-1H-INDAZOLE (K64) | PROTEIN KINASE CK2-INHIBITOR COMPLEX, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3kxh:A (SER51) to (TYR182) CRYSTAL STRUCTURE OF Z. MAYS CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE INHIBITOR (2-DYMETHYLAMMINO-4,5,6,7-TETRABROMOBENZOIMIDAZOL-1YL- ACETIC ACID (K66) | PROTEIN KINASE CK2-INHIBITOR COMPLEX, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3kxm:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF Z. MAYS CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE INHIBITOR K74 | PROTEIN KINASE CK2-INHIBITOR COMPLEX, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3kxn:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF Z. MAYS CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE INHIBITOR TETRAIODOBENZIMIDAZOLE (K88) | PROTEIN KINASE CK2-INHIBITOR COMPLEX, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5dew:A (GLY282) to (THR415) CRYSTAL STRUCTURE OF PAK1 IN COMPLEX WITH AN INHIBITOR COMPOUND 5 | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1yvj:A (GLY834) to (LEU974) CRYSTAL STRUCTURE OF THE JAK3 KINASE DOMAIN IN COMPLEX WITH A STAUROSPORINE ANALOGUE | TYROSINE KINASE; SCID; SEVERE COMBINED IMMUNODEFICIENCY; STAT5; STAT6; INTERLEUKIN-2; COMMON-GAMMA CHAIN, TRANSFERASE
4anm:A (SER51) to (PHE181) COMPLEX OF CK2 WITH A CDC7 INHIBITOR | TRANSFERASE
3amy:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF HUMAN CK2 ALPHA COMPLEXED WITH APIGENIN | TRANSFERASE, ATP-BINDING
4py1:A (GLY909) to (GLU1050) CRYSTAL STRUCTURE OF TYK2 IN COMPLEX WITH COMPOUND 15, 6-((2,5- DIMETHOXYPHENYL)THIO)-3-(1-METHYL-1H-PYRAZOL-4-YL)-[1,2,4]TRIAZOLO[4, 3-B]PYRIDAZINE | KINASE, TRANSFERASE
3lpb:A (PHE860) to (GLN1003) CRYSTAL STRUCTURE OF JAK2 COMPLEXED WITH A POTENT 2,8-DIARYL- QUINOXALINE INHIBITOR | SMALL MOLECULE INHIBITOR, ATP SITE KINASE INHIBITOR, NOVARTIS PRODUCT NVP-BLU040, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE
3lpb:B (GLY861) to (GLN1003) CRYSTAL STRUCTURE OF JAK2 COMPLEXED WITH A POTENT 2,8-DIARYL- QUINOXALINE INHIBITOR | SMALL MOLECULE INHIBITOR, ATP SITE KINASE INHIBITOR, NOVARTIS PRODUCT NVP-BLU040, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE
1zog:A (GLU52) to (PHE181) CRYSTAL STRUCTURE OF PROTEIN KINASE CK2 IN COMPLEX WITH TBB- DERIVATIVES | PROTEIN KINASE CK2, TBB, TETRABROMO-BENZIMIDAZOLE, INHIBITORS, PHARMACOPHORE, TRANSFERASE
1zoh:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF PROTEIN KINASE CK2 IN COMPLEX WITH TBB- DERIVATIVES INHIBITORS | PROTEIN KINASE CK2, TETRABROMO-BENZIMIDAZOLE, TBB, INHIBITORS, PHARMACOPHORE, TRANSFERASE
4au8:A (GLY16) to (PHE151) CRYSTAL STRUCTURE OF COMPOUND 4A IN COMPLEX WITH CDK5, SHOWING AN UNUSUAL BINDING MODE TO THE HINGE REGION VIA A WATER MOLECULE | TRANSFERASE, CDK2, ALZHEIMER DISEASE
4au8:B (GLY16) to (PHE151) CRYSTAL STRUCTURE OF COMPOUND 4A IN COMPLEX WITH CDK5, SHOWING AN UNUSUAL BINDING MODE TO THE HINGE REGION VIA A WATER MOLECULE | TRANSFERASE, CDK2, ALZHEIMER DISEASE
5e1e:B (PHE886) to (THR1030) HUMAN JAK1 KINASE IN COMPLEX WITH COMPOUND 30 AT 2.30 ANGSTROMS RESOLUTION | KINASE, TRANSFERASE
3lxl:A (GLY834) to (LEU976) STRUCTURAL AND THERMODYNAMIC CHARACTERIZATION OF THE TYK2 AND JAK3 KINASE DOMAINS IN COMPLEX WITH CP-690550 AND CMP-6 | TYK2, JAK3, INFLAMMATION, CANCER, PAN INHIBITOR, ATP-BINDING, DISEASE MUTATION, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SCID, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3lxn:A (GLY909) to (GLU1050) STRUCTURAL AND THERMODYNAMIC CHARACTERIZATION OF THE TYK2 AND JAK3 KINASE DOMAINS IN COMPLEX WITH CP-690550 AND CMP-6 | TYK2, JAK3, INFLAMMATION, CANCER, PAN INHIBITOR, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3lxp:A (LEU913) to (GLU1050) STRUCTURAL AND THERMODYNAMIC CHARACTERIZATION OF THE TYK2 AND JAK3 KINASE DOMAINS IN COMPLEX WITH CP-690550 AND CMP-6 | TYK2, JAK3, INFLAMMATION, CANCER, PAN INHIBITOR, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
2a1a:B (GLY279) to (LEU439) PKR KINASE DOMAIN-EIF2ALPHA COMPLEX | TRANSFERASE, KINASE, PROTEIN BIOSYNTHESIS, PROTEIN SYNTHESIS- TRANSFERASE COMPLEX
5e8v:A (ALA256) to (LEU404) TGF-BETA RECEPTOR TYPE 2 KINASE DOMAIN (E431A,R433A,E485A,K488A,R493A, R495A) | KINASE DOMAIN, TRANSFERASE
5e91:A (ALA256) to (LEU404) TGF-BETA RECEPTOR TYPE 2 KINASE DOMAIN (E431A,R433A,E485A,K488A,R493A, R495A) IN COMPLEX WITH 3-AMINO-6-[4-(2- HYDROXYETHYL)PHENYL]-N-[4- (MORPHOLIN-4-YL)PYRIDIN-3-YL] PYRAZINE-2-CARBOXAMIDE | KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5e92:A (ALA256) to (PRO406) TGF-BETA RECEPTOR TYPE 2 KINASE DOMAIN (E431A,R433A,E485A,K488A,R493A, R495A) IN COMPLEX WITH AMPPNP | KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3m2w:A (GLY76) to (THR214) CRYSTAL STRUCTURE OF MAPKAK KINASE 2 (MK2) COMPLEXED WITH A SPIROAZETIDINE-TETRACYCLIC ATP SITE INHIBITOR | SMALL MOLECULE INHIBITOR, SPIROAZETIDINE-TETRACYCLE, ATP-SITE KINASE INHIBITOR, NOVARTIS COMPOUND NVP-BXS169, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3axw:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF HUMAN CK2ALPHA COMPLEXED WITH A POTENT INHIBITOR | KINASE DOMAIN, SERINE/THREONINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ebz:C (ASN28) to (VAL172) HUMAN KINASE | KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ebz:F (ASN28) to (VAL172) HUMAN KINASE | KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ebz:G (ASN28) to (VAL172) HUMAN KINASE | KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ebz:H (ASN28) to (VAL172) HUMAN KINASE | KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ebz:I (ASN28) to (VAL172) HUMAN KINASE | KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ebz:K (ASN28) to (VAL172) HUMAN KINASE | KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ebz:L (ASN28) to (VAL172) HUMAN KINASE | KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3mb6:A (SER51) to (PHE181) HUMAN CK2 CATALYTIC DOMAIN IN COMPLEX WITH A DIFURANE DERIVATIVE INHIBITOR (CPA) | KINASES, DIFURANE, INHIBITOR, CK2, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4qmw:A (GLY36) to (THR170) MST3 IN COMPLEX WITH PP-121, 1-CYCLOPENTYL-3-(1H-PYRROLO[2,3- B]PYRIDIN-5-YL)-1H-PYRAZOLO[3,4-D]PYRIMIDIN-4-AMINE | PROTEIN KINASE, MST3, STK24, STERILE 20-LIKE KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4bcp:A (VAL17) to (ALA151) STRUCTURE OF CDK2 IN COMPLEX WITH CYCLIN A AND A 2-AMINO-4- HETEROARYL-PYRIMIDINE INHIBITOR | TRANSFERASE-CELL CYCLE COMPLEX, CDK-CYCLIN COMPLEX, CYCLIN-INHIBITOR, STRUCTURE-BASED DRUG DESIGN
4qp1:A (GLY37) to (VAL173) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH N-CYCLOHEXYL-9H-PURIN-6- AMINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qp1:B (GLY37) to (VAL173) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH N-CYCLOHEXYL-9H-PURIN-6- AMINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qp2:A (GLY37) to (VAL173) CRYSTAL STRUCTURE OF ERKS IN COMPLEX WITH 5-CHLOROBENZO[D]OXAZOL-2- AMINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qp3:A (MET38) to (ALA174) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH (S)-2-((9H-PURIN-6-YL) AMINO)-3-PHENYLPROPAN-1-OL | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qp3:B (GLY37) to (VAL173) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH (S)-2-((9H-PURIN-6-YL) AMINO)-3-PHENYLPROPAN-1-OL | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qp4:A (GLY37) to (VAL173) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH N-CYCLOHEXYL-9H-PURIN-6- AMINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qp4:B (GLY37) to (VAL173) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH N-CYCLOHEXYL-9H-PURIN-6- AMINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qp6:A (GLY37) to (VAL173) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH 5H-PYRROLO[2,3-B]PYRAZINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qp6:B (GLY37) to (VAL173) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH 5H-PYRROLO[2,3-B]PYRAZINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qp8:A (GLY37) to (ALA174) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH 2-(1H-PYRAZOL-4-YL)-7- (PYRIDIN-3-YL)-5H-PYRROLO[2,3-B]PYRAZINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qp8:B (GLY37) to (ALA174) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH 2-(1H-PYRAZOL-4-YL)-7- (PYRIDIN-3-YL)-5H-PYRROLO[2,3-B]PYRAZINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qp9:A (GLY37) to (VAL173) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH 7-(1-PROPYL-1H-PYRAZOL-4- YL)-2-(PYRIDIN-4-YL)-5H-PYRROLO[2,3-B]PYRAZINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qpa:B (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH 7-(1-BENZYL-1H-PYRAZOL-4- YL)-2-(PYRIDIN-4-YL)-5H-PYRROLO[2,3-B]PYRAZINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3mi9:A (GLU32) to (ALA173) CRYSTAL STRUCTURE OF HIV-1 TAT COMPLEXED WITH HUMAN P-TEFB | P-TEFB, TAT, HIV-1, PROTEIN BINDING
3mia:A (GLU32) to (ALA173) CRYSTAL STRUCTURE OF HIV-1 TAT COMPLEXED WITH ATP-BOUND HUMAN P-TEFB | P-TEFB, CDK9, CYCLIN T1, HIV-1, TAT, PROTEIN BINDING
4qps:C (GLY834) to (LEU976) CRYSTAL STRUCTURE OF JAK3 COMPLEXED TO N-[3-(6-PHENYLAMINO-PYRAZIN-2- YL)-3H-BENZOIMIDAZOL-5-YL]-ACRYLAMIDE | KINASE CATALYTIC DOMAIN, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4bid:B (GLY692) to (ARG828) CRYSTAL STRUCTURES OF ASK1-INHIBITOR COMPLEXES | TRANSFERASE
4qta:A (GLY37) to (ALA174) STRUCTURE OF HUMAN ERK2 IN COMPLEX WITH SCH772984 REVEALING A NOVEL INHIBITOR-INDUCED BINDING POCKET | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE, KINASE, MAPK, SIGNALLING, INHIBITOR, ALLOSTERIC, STRUCTURAL GENOMICS CONSORTIUM (SGC), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qtb:A (GLY54) to (ALA191) STRUCTURE OF HUMAN ERK1 IN COMPLEX WITH SCH772984 REVEALING A NOVEL INHIBITOR-INDUCED BINDING POCKET | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE, KINASE, MAPK, SIGNALLING, INHIBITOR, ALLOSTERIC, STRUCTURAL GENOMICS CONSORTIUM (SGC), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qtb:B (GLY54) to (ALA191) STRUCTURE OF HUMAN ERK1 IN COMPLEX WITH SCH772984 REVEALING A NOVEL INHIBITOR-INDUCED BINDING POCKET | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE, KINASE, MAPK, SIGNALLING, INHIBITOR, ALLOSTERIC, STRUCTURAL GENOMICS CONSORTIUM (SGC), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3blq:A (GLY31) to (ALA173) CRYSTAL STRUCTURE OF HUMAN CDK9/CYCLINT1 IN COMPLEX WITH ATP | TRANSCRIPTIONAL CDK/CYCLIN COMPLEX, PHOSPHORYLATED, IN COMPLEX WITH ATP, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSCRIPTION REGULATION, TRANSFERASE, ACETYLATION, CELL CYCLE, CELL DIVISION, COILED COIL, HOST-VIRUS INTERACTION
5f1z:A (LYS910) to (GLU1050) STRUCTURE OF TYK2 WITH INHIBITOR 16: 3-AZANYL-5-[(2~{S})-3- METHYLBUTAN-2-YL]-7-[1-METHYL-5-(2-OXIDANYLPROPAN-2-YL)PYRAZOL-3-YL]- 1~{H}-PYRAZOLO[4,3-C]PYRIDIN-4-ONE | KINASE, COMPLEX, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5f20:A (LYS910) to (VAL1048) STRUCTURE OF TYK2 WITH INHIBITOR 4: 3-AZANYL-5-(2-METHYLPHENYL)-7-(1- METHYLPYRAZOL-3-YL)-1~{H}-PYRAZOLO[4,3-C]PYRIDIN-4-ONE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3my0:U (GLY214) to (SER356) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3nga:A (GLU55) to (PHE181) HUMAN CK2 CATALYTIC DOMAIN IN COMPLEX WITH CX-4945 | KINASE, CK2, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3nga:B (SER51) to (PHE181) HUMAN CK2 CATALYTIC DOMAIN IN COMPLEX WITH CX-4945 | KINASE, CK2, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3niz:A (GLY35) to (PHE169) CRYPTOSPORIDIUM PARVUM CYCLIN-DEPENDENT KINASE CGD5_2510 WITH ADP BOUND. | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, PHOSPHOTRANSFERASE, CYCLIN DEPENDENT KINASE, TRANSFERASE
4c61:A (SER862) to (GLN1003) INHIBITORS OF JAK2 KINASE DOMAIN | KINASE, TRANSFERASE
4c62:A (GLY861) to (GLN1003) INHIBITORS OF JAK2 KINASE DOMAIN | TRANSFERASE
4rlk:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF Z. MAYS CK2ALPHA IN COMPLEX WITH THE ATP- COMPETITIVE INHIBITOR 4-[(E)-(FLUOREN-9-YLIDENEHYDRAZINYLIDENE)- METHYL] BENZOATE | TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4rmz:A (VAL199) to (ALA335) CRYSTAL STRUCTURE OF IRAK-4 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3nsz:A (GLU55) to (PHE181) HUMAN CK2 CATALYTIC DOMAIN IN COMPLEX WITH AMPPN | KINASE, CK2, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3com:A (SER43) to (THR175) CRYSTAL STRUCTURE OF MST1 KINASE | KINASE, MST1, SERINE/THREONINE-PROTEIN KINASE 4, STE20-LIKE KINASE, PSI, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ALTERNATIVE SPLICING, APOPTOSIS, ATP- BINDING, COILED COIL, CYTOPLASM, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE
4ci6:B (HIS144) to (ARG292) MECHANISMS OF CRIPPLING ACTIN-DEPENDENT PHAGOCYTOSIS BY YOPO | TRANSFERASE-STRUCTURAL PROTEIN COMPLEX, BUBONIC PLAGUE
3nyx:A (GLY909) to (GLU1050) NON-PHOSPHORYLATED TYK2 JH1 DOMAIN WITH QUINOLINE-THIADIAZOLE- THIOPHENE INHIBITOR | PROTEIN KINASE, TYROSINE PHOSPHORYLATION, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3nz0:A (LEU913) to (VAL1048) NON-PHOSPHORYLATED TYK2 KINASE WITH CMP6 | PROTEIN KINASE, TYROSINE PHOSPHORYLATION, TRANSFERASE
3o0g:A (GLY16) to (GLY152) CRYSTAL STRUCTURE OF CDK5:P25 IN COMPLEX WITH AN ATP ANALOGUE | KINASE, KINASE ACTIVATOR COMPLEX, KINASE INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE ACTIVATOR COMPLEX
4s2z:A (GLY35) to (VAL171) ERK2 INTRINSICALLY ACTIVE MUTANT R65S | SIGNAL TRANSDUCTION, PHOSPHORYLATION, KINASE, TRANSFERASE
4s31:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF MITOGEN-ACTIVATED PROTEIN KINASE 1 WTERK2 AT 1.45A | SIGNAL TRANSDUCTION, PHOSPHORYLATION, TRANSFERASE
4s30:A (GLY35) to (VAL171) ERK2 INTRINSICALLY ACTIVE MUTANT (I84A) | SIGNAL TRANSDUCTION, PHOSPHORYLATION, TRANSFERASE
4s32:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK2 AMP-PNP COMPLEX | SIGNAL TRANSDUCTION, PHOSPHORYLATION, TRANSFERASE
4s34:A (GLY35) to (VAL171) ERK2 (I84A) IN COMPLEX WITH AMP-PNP | SIGNAL TRANSDUCTION, PHOSPHORYLATION, TRANSFERASE
3d4q:B (THR470) to (VAL600) PYRAZOLE-BASED INHIBITORS OF B-RAF KINASE | KINASE, ATP-BINDING, CARDIOMYOPATHY, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ZINC-FINGER
3d7z:A (SER37) to (THR175) CRYSTAL STRUCTURE OF P38 KINASE IN COMPLEX WITH A BIPHENYL AMIDE INHIBITOR | P38, SERINE/THREONINE PROTEIN KINASE, MAP KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
3dls:A (TRP1014) to (ARG1155) CRYSTAL STRUCTURE OF HUMAN PAS KINASE BOUND TO ADP | PAS KINASE, PASK, PROTEIN KINASE, DRUG DISCOVERY, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
3dls:E (TRP1014) to (ARG1155) CRYSTAL STRUCTURE OF HUMAN PAS KINASE BOUND TO ADP | PAS KINASE, PASK, PROTEIN KINASE, DRUG DISCOVERY, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
5h8b:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF CK2 WITH COMPOUND 2 | KINASE, INHIBITOR, CK2, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5h8b:B (SER51) to (PHE181) CRYSTAL STRUCTURE OF CK2 WITH COMPOUND 2 | KINASE, INHIBITOR, CK2, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5h8e:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF CK2 WITH COMPOUND 7H | KINASE, INHIBITOR, CK2, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5h8e:B (SER51) to (PHE181) CRYSTAL STRUCTURE OF CK2 WITH COMPOUND 7H | KINASE, INHIBITOR, CK2, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5h8g:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF CK2 WITH COMPOUND 7B | KINASE, INHIBITOR, CK2, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3owl:A (SER51) to (PHE181) HUMAN CK2 CATALYTIC DOMAIN IN COMPLEX WITH A BENZOPYRIDOINDOLE DERIVATIVE INHIBITOR | SERINE/THREONINE-PROTEIN KINASE, CK2, INHIBITOR, PYRIDOCARBAZOL, ELLIPTICINE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4dgl:D (SER51) to (PHE181) CRYSTAL STRUCTURE OF THE CK2 TETRAMERIC HOLOENZYME | PROTEIN KINASE, TRANSFERASE
4dgm:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF MAIZE CK2 IN COMPLEX WITH THE INHIBITOR APIGENIN | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4dgo:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF MAIZE CK2 IN COMPLEX WITH TYRPHOSTIN AG99 | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4dn5:A (GLY412) to (GLN542) CRYSTAL STRUCTURE OF NF-KB-INDUCING KINASE (NIK) | NON-RD KINASE, PROTEIN SERINE/THREONINE KINASE, TRANSFERASE, ATP BINDING
4ub7:A (GLU52) to (PHE181) HIGH-SALT STRUCTURE OF PROTEIN KINASE CK2 CATALYTIC SUBUNIT WITH 4'- CARBOXY-6,8-BROMO-FLAVONOL (FLC26) SHOWING AN EXTREME DISTORTION OF THE ATP-BINDING LOOP COMBINED WITH A PI-HALOGEN BOND | PROTEIN KINASE CK2, ATP-COMPETITIVE INHIBITORS, HALOGEN BOND, 4'- CARBOXY-6, 8-BROMO-FLAVONOL, TRANSFERASE
4uba:A (SER51) to (PHE181) LOW-SALT STRUCTURE OF PROTEIN KINASE CK2 CATALYTIC SUBUNIT WITH 4'- CARBOXY-6,8-BROMO-FLAVONOL (FLC26) | PROTEIN KINASE CK2, ATP-COMPETITIVE INHIBITORS, HALOGEN BOND, 4'- CARBOXY-6, 8-BROMO-FLAVONOL, TRANSFERASE
4uba:B (SER51) to (PHE181) LOW-SALT STRUCTURE OF PROTEIN KINASE CK2 CATALYTIC SUBUNIT WITH 4'- CARBOXY-6,8-BROMO-FLAVONOL (FLC26) | PROTEIN KINASE CK2, ATP-COMPETITIVE INHIBITORS, HALOGEN BOND, 4'- CARBOXY-6, 8-BROMO-FLAVONOL, TRANSFERASE
3e3p:B (THR33) to (LYS176) GLYCOGEN SYNTHASE KINASE FROM LEISHMANIA MAJOR | GLYCOGEN SYNTHASE KINASE, LEISHMANIASIS, KINASE, TRANSFERASE
5hvj:A (GLY351) to (MET485) CRYSTAL STRUCTURE OF LIMK1 D460N MUTANT IN COMPLEX WITH AMP-PNP | KINASE ATP ANALOG ACTIN-REMODELING, TRANSFERASE
5hvj:B (PHE350) to (LEU484) CRYSTAL STRUCTURE OF LIMK1 D460N MUTANT IN COMPLEX WITH AMP-PNP | KINASE ATP ANALOG ACTIN-REMODELING, TRANSFERASE
5hx8:A (PHE886) to (THR1030) JAK1 COMPLEX WITH 4-[(4-AMINOCYCLOHEXYL)AMINO]-3-(1H-BENZIMIDAZOL-2- YL)-1H-PYRIDIN-2-ONE | KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3pe1:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF HUMAN PROTEIN KINASE CK2 ALPHA SUBUNIT IN COMPLEX WITH THE INHIBITOR CX-4945 | KINASE, CK2-INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3pe2:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF HUMAN PROTEIN KINASE CK2 IN COMPLEX WITH THE INHIBITOR CX-5011 | KINASE, CK2-INHIBITOR COMPLEX, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3pjc:A (GLY834) to (LEU976) CRYSTAL STRUCTURE OF JAK3 COMPLEXED WITH A POTENT ATP SITE INHIBITOR SHOWING HIGH SELECTIVITY WITHIN THE JANUS KINASE FAMILY | SMALL MOLECULE INHIBITOR, ATP SITE KINASE INHIBITOR, ATP-BINDING, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e1z:A (GLY905) to (GLU1046) STRUCTURE OF MOUSE TYK-2 COMPLEXED TO A 3-AMINOINDAZOLE INHIBITOR | KINASE CATALYTIC DOMAIN, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e20:A (GLY905) to (GLU1046) STRUCTURE OF MOUSE TYK-2 COMPLEXED TO A 3-AMINOINDAZOLE INHIBITOR | KINASE CATALYTIC DOMAIN, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ppk:A (LYS473) to (VAL600) HUMAN B-RAF KINASE IN COMPLEX WITH A NON-OXIME FUROPYRIDINE INHIBITOR | PROTEIN KINASE, B-RAF ATP-COMPETITIVE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4e4l:B (LEU891) to (THR1030) JAK1 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 30 | O-PHOSPHOTYROSINE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e4m:E (GLY861) to (LEU1001) JAK2 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 30 | O-PHOSPHOTYROSINE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e4n:A (GLY887) to (THR1030) JAK1 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 49 | O-PHOSPHOTYROSINE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e5w:A (GLY887) to (THR1030) JAK1 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 26 | JAK1, KINASE DOMAIN, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e5w:B (LEU891) to (ILE1028) JAK1 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 26 | JAK1, KINASE DOMAIN, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3pvg:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF Z. MAYS CK2 ALPHA SUBUNIT IN COMPLEX WITH THE INHIBITOR 4,5,6,7-TETRABROMO-1-CARBOXYMETHYLBENZIMIDAZOLE (K68) | PROTEIN KINASE CK2-INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ehz:A (GLY887) to (THR1030) THE JAK1 KINASE DOMAIN IN COMPLEX WITH INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3pwd:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF MAIZE CK2 IN COMPLEX WITH NBC (Z1) | PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3py3:A (GLY36) to (THR175) CRYSTAL STRUCTURE OF PHOSPHORYLATED P38ALPHA MAP KINASE | KINASE, TRANSFERASE, PHOSPHORYLATION
3pzh:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF MAIZE CK2 ALPHA IN COMPLEX WITH EMODIN AT 1.92 A RESOLUTION | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3q32:A (MET865) to (GLN1003) STRUCTURE OF JANUS KINASE 2 WITH A PYRROLOTRIAZINE INHIBITOR | ATP-BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3q32:B (GLY861) to (GLN1003) STRUCTURE OF JANUS KINASE 2 WITH A PYRROLOTRIAZINE INHIBITOR | ATP-BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4eoj:C (GLY16) to (ALA151) THR 160 PHOSPHORYLATED CDK2 H84S, Q85M, K89D - HUMAN CYCLIN A3 COMPLEX WITH ATP | PROTEIN KINASE, CELL CYCLE, COMPLEX, PHOSPHORYLATION, TRANSFERASE
4eom:A (GLY16) to (ALA151) THR 160 PHOSPHORYLATED CDK2 H84S, Q85M, Q131E - HUMAN CYCLIN A3 COMPLEX WITH ATP | PROTEIN KINASE, CELL CYCLE, COMPLEX, PHOSPHORYLATION, TRANSFERASE
4eop:A (GLY16) to (ALA151) THR 160 PHOSPHORYLATED CDK2 Q131E - HUMAN CYCLIN A3 COMPLEX WITH THE INHIBITOR RO3306 | PROTEIN KINASE, CELL CYCLE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4eor:A (GLY16) to (ALA151) THR 160 PHOSPHORYLATED CDK2 WT - HUMAN CYCLIN A3 COMPLEX WITH THE INHIBITOR NU6102 | PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4eos:C (GLY16) to (ALA151) THR 160 PHOSPHORYLATED CDK2 WT - HUMAN CYCLIN A3 COMPLEX WITH THE INHIBITOR RO3306 | PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3q4z:A (GLY282) to (THR415) STRUCTURE OF UNPHOSPHORYLATED PAK1 KINASE DOMAIN | KINASE DOMAIN, SIGNALLING PATHWAY, TRANSFERASE
3q53:A (GLY282) to (THR415) STRUCTURE OF PHOSPHORYLATED PAK1 KINASE DOMAIN IN COMPLEX WITH ATP | KINASE DOMAIN, SIGNALLING PATHWAY, TRANSFERASE
5iu2:A (GLY150) to (GLN276) DISCOVERY OF IMIDAZOQUINOLINES AS A NOVEL CLASS OF POTENT, SELECTIVE AND IN VIVO EFFICACIOUS COT KINASE INHIBITORS | COT, TPL-2, MAP3K8, KINASE, INHIBITOR, COMPLEX, TRANSFERASE
5iu2:B (GLY150) to (GLN276) DISCOVERY OF IMIDAZOQUINOLINES AS A NOVEL CLASS OF POTENT, SELECTIVE AND IN VIVO EFFICACIOUS COT KINASE INHIBITORS | COT, TPL-2, MAP3K8, KINASE, INHIBITOR, COMPLEX, TRANSFERASE
4erk:A (GLY35) to (VAL171) THE COMPLEX STRUCTURE OF THE MAP KINASE ERK2/OLOMOUCINE | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, MAP KINASE, ERK2
3q9y:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF HUMAN CK2 ALPHA IN COMPLEX WITH QUINALIZARIN AT PH 8.5 | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3q9z:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF HUMAN CK2 ALPHA IN COMPLEX WITH QUINALIZARIN AT PH 6.5 | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qa0:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF THE APO-FORM OF HUMAN CK2 ALPHA AT PH 6.5 | PROTEIN KINASE, APO-FORM, TRANSFERASE
4f08:A (GLY861) to (GLN1003) DISCOVERY AND OPTIMIZATION OF C-2 METHYL IMIDAZO-PYRROLOPYRIDINES AS POTENT AND ORALLY BIOAVAILABLE JAK1 INHIBITORS WITH SELECTIVITY OVER JAK2 | JAK2, KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4f08:B (GLY861) to (GLN1003) DISCOVERY AND OPTIMIZATION OF C-2 METHYL IMIDAZO-PYRROLOPYRIDINES AS POTENT AND ORALLY BIOAVAILABLE JAK1 INHIBITORS WITH SELECTIVITY OVER JAK2 | JAK2, KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4f09:A (GLY861) to (GLN1003) DISCOVERY AND OPTIMIZATION OF C-2 METHYL IMIDAZO-PYRROLOPYRIDINES AS POTENT AND ORALLY BIOAVAILABLE JAK1 INHIBITORS WITH SELECTIVITY OVER JAK2 | JAK2, KINASE DOMAIN, JH1 DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4f99:A (SER70) to (GLY202) HUMAN CDC7 KINASE IN COMPLEX WITH DBF4 AND NUCLEOTIDE | SER/THR PROTEIN KINASE, TRANSFERASE, PHOSPHORYLATION, CELL CYCLE, CELL DIVISION, MITOSIS, S PHASE, SERINE/THREONINE-PROTEIN KINASE, DBF4-DEPENDENT KINASE, DDK, ATP-BINDING, NUCLEOTIDE-BINDING, ZINC- BINDING, NUCLEUS
4f9a:A (SER70) to (GLY202) HUMAN CDC7 KINASE IN COMPLEX WITH DBF4 AND NUCLEOTIDE | SER/THR PROTEIN KINASE, TRANSFERASE, PHOSPHORYLATION, CELL CYCLE, CELL DIVISION, MITOSIS, S PHASE, SERINE/THREONINE-PROTEIN KINASE, DBF4-DEPENDENT KINASE, DDK, ATP-BINDING, NUCLEOTIDE-BINDING, ZINC- BINDING, NUCLEUS
4f9a:C (SER70) to (GLY202) HUMAN CDC7 KINASE IN COMPLEX WITH DBF4 AND NUCLEOTIDE | SER/THR PROTEIN KINASE, TRANSFERASE, PHOSPHORYLATION, CELL CYCLE, CELL DIVISION, MITOSIS, S PHASE, SERINE/THREONINE-PROTEIN KINASE, DBF4-DEPENDENT KINASE, DDK, ATP-BINDING, NUCLEOTIDE-BINDING, ZINC- BINDING, NUCLEUS
4v0g:A (GLY834) to (LEU974) JAK3 IN COMPLEX WITH A COVALENT EGFR INHIBITOR | TRANSFERASE, EGFR MUTANT, T790M
4fbx:A (SER51) to (PHE181) COMPLEX STRUCTURE OF HUMAN PROTEIN KINASE CK2 CATALYTIC SUBUNIT CRYSTALLIZED IN THE PRESENCE OF A BISUBSTRATE INHIBITOR | PROTEIN KINASE FOLD, PROTEIN PHOSPHORYLATION, BISUBSTRATE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qyw:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH AN INHIBITOR | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING CELL CYCLE, PHOSPHORYLATION, PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qyz:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH AN INHIBITOR | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING CELL CYCLE, PHOSPHORYLATION, PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fi1:A (SER52) to (PHE220) CRYSTAL STRUCTURE OF SCCK2 ALPHA IN COMPLEX WITH ATP | PROTEIN-ATP COMPLEX, PROTEIN KINASE, PHOSPHORYLATION, TRANSFERASE
4fie:A (CYS336) to (SER466) FULL-LENGTH HUMAN PAK4 | SERINE/THREONINE-PROTEIN KINASE PAK4, KINASE DOMAIN, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
4fie:B (CYS336) to (SER466) FULL-LENGTH HUMAN PAK4 | SERINE/THREONINE-PROTEIN KINASE PAK4, KINASE DOMAIN, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
4w7p:B (GLY88) to (ASN224) CRYSTAL STRUCTURE OF ROCK 1 BOUND TO YB-15-QD37 | INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fk6:A (LEU891) to (THR1030) JAK1 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 72 | PROTEIN KINASE, PHOSPHO TRANSFER, PHOSPHO TYROSINE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4fmq:A (GLY37) to (ALA174) CRYSTAL STRUCTURE OF HUMAN ERK2 COMPLEXED WITH A MAPK DOCKING PEPTIDE | TRANSFERASE, SIGNALING, PROTEIN-PROTEIN INTERACTION, TRANSFERASE- SIGNALING PROTEIN COMPLEX
4fv0:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF THE ERK2 COMPLEXED WITH EK3 | TRANSFERASE
4fv2:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF THE ERK2 COMPLEXED WITH EK5 | TRANSFERASE
4fv4:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF THE ERK2 COMPLEXED WITH EK7 | TRANSFERASE
4fv6:A (GLY35) to (ALA172) CRYSTAL STRUCTURE OF THE ERK2 COMPLEXED WITH E57 | TRANSFERASE
4fv8:A (GLY35) to (ALA172) CRYSTAL STRUCTURE OF THE ERK2 COMPLEXED WITH E63 | TRANSFERASE
4fv9:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF THE ERK2 COMPLEXED WITH E71 | TRANSFERASE
4g3c:B (HIS417) to (GLN544) CRYSTAL STRUCTURE OF APO MURINE NF-KAPPAB INDUCING KINASE (NIK) | NON-RD KINASE, PROTEIN SERINE/THREONINE KINASE, NF-KAPPAB, MAP3K14, TRANSFERASE
4g3d:A (GLU413) to (PRO543) CRYSTAL STRUCTURE OF HUMAN NF-KAPPAB INDUCING KINASE (NIK) | NON-RD KINASE, PROTEIN SERINE/THREONINE KINASE, NF-KAPPAB, MAP3K14, TRANSFERASE
4g3d:B (HIS415) to (LEU541) CRYSTAL STRUCTURE OF HUMAN NF-KAPPAB INDUCING KINASE (NIK) | NON-RD KINASE, PROTEIN SERINE/THREONINE KINASE, NF-KAPPAB, MAP3K14, TRANSFERASE
4g3d:E (HIS415) to (GLN542) CRYSTAL STRUCTURE OF HUMAN NF-KAPPAB INDUCING KINASE (NIK) | NON-RD KINASE, PROTEIN SERINE/THREONINE KINASE, NF-KAPPAB, MAP3K14, TRANSFERASE
4g3e:A (HIS417) to (CYS542) CRYSTAL STRUCTURE OF MURINE NF-KAPPAB INDUCING KINASE (NIK) BOUND TO A 6-ALKYNYLINDOLINE (CMP1) | NON-RD KINASE, PROTEIN SERINE/THREONINE KINASE, NF-KAPPAB,STRUCTURE- BASED DRUG DESIGN, MAP3K14, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4g3e:B (HIS417) to (GLN544) CRYSTAL STRUCTURE OF MURINE NF-KAPPAB INDUCING KINASE (NIK) BOUND TO A 6-ALKYNYLINDOLINE (CMP1) | NON-RD KINASE, PROTEIN SERINE/THREONINE KINASE, NF-KAPPAB,STRUCTURE- BASED DRUG DESIGN, MAP3K14, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4g6o:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF THE ERK2 | TRANSFERASE
5k5n:A (GLY68) to (GLN206) CRYSTAL STRUCTURE OF GSK-3BETA COMPLEXED WITH PF-04802367, A HIGHLY SELECTIVE BRAIN-PENETRANT KINASE INHIBITOR | PROTEIN KINASE, ALZHIMER'S DISEASE, TAU KINASE, TRANSFERASE
5k5n:B (GLY68) to (GLN206) CRYSTAL STRUCTURE OF GSK-3BETA COMPLEXED WITH PF-04802367, A HIGHLY SELECTIVE BRAIN-PENETRANT KINASE INHIBITOR | PROTEIN KINASE, ALZHIMER'S DISEASE, TAU KINASE, TRANSFERASE
4gfo:A (GLY909) to (GLU1050) TYK2 KINASE (JH1 DOMAIN) WITH 2,6-DICHLORO-N-(2-OXO-2,5- DIHYDROPYRIDIN-4-YL)BENZAMIDE | PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gih:A (GLY909) to (PRO1049) TYK2 (JH1) IN COMPLEX WITH 2,6-DICHLORO-N-{2-[(CYCLOPROPYLCARBONYL) AMINO]PYRIDIN-4-YL}BENZAMIDE | TYROSINE KINASE, KINASE, ATP BINDING, INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4gii:A (GLY909) to (PRO1049) TYK2 (JH1) IN COMPLEX WITH 2,6-DICHLORO-4-CYANO-N-{2- [(CYCLOPROPYLCARBONYL)AMINO]PYRIDIN-4-YL}BENZAMIDE | AMINOPYRIDINE, BENZAMIDE, KINASE, ENZYME INHIBITOR, TYROSINE KINASE, ATP BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gj2:A (GLY909) to (PRO1049) TYK2 (JH1) IN COMPLEX WITH 2,6-DICHLORO-N-[2-({[(1R,2R)-2- FLUOROCYCLOPROPYL]CARBONYL}AMINO)PYRIDIN-4-YL]BENZAMIDE | KINASE, ATP BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5khw:A (GLY887) to (THR1030) CRYSTAL STRUCTURE OF JAK1 IN COMPLEX WITH ADP | JAK1, KINASE, INHIBITOR, COMPLEX, TRANSFERASE
5khw:B (GLY887) to (THR1030) CRYSTAL STRUCTURE OF JAK1 IN COMPLEX WITH ADP | JAK1, KINASE, INHIBITOR, COMPLEX, TRANSFERASE
4gl9:A (MET865) to (GLN1003) CRYSTAL STRUCTURE OF INHIBITORY PROTEIN SOCS3 IN COMPLEX WITH JAK2 KINASE DOMAIN AND FRAGMENT OF GP130 INTRACELLULAR DOMAIN | KINASE INHIBITOR RECEPTOR CYTOKINE SIGNALLING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gl9:C (MET865) to (GLN1003) CRYSTAL STRUCTURE OF INHIBITORY PROTEIN SOCS3 IN COMPLEX WITH JAK2 KINASE DOMAIN AND FRAGMENT OF GP130 INTRACELLULAR DOMAIN | KINASE INHIBITOR RECEPTOR CYTOKINE SIGNALLING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gl9:D (MET865) to (GLN1003) CRYSTAL STRUCTURE OF INHIBITORY PROTEIN SOCS3 IN COMPLEX WITH JAK2 KINASE DOMAIN AND FRAGMENT OF GP130 INTRACELLULAR DOMAIN | KINASE INHIBITOR RECEPTOR CYTOKINE SIGNALLING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4grb:A (GLU55) to (PHE181) CASEIN KINASE 2 (CK2) BOUND TO INHIBITOR | KINASE, PROTEIN KINASE, CYTOSOL, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5kx8:C (GLY198) to (SER336) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5kx8:D (GLY198) to (SER336) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5l3a:A (GLY861) to (GLN1003) FRAGMENT-BASED DISCOVERY OF 6-ARYLINDAZOLE JAK INHIBITORS | DOUBLE F MUTANT, TRANSFERASE
5l6w:L (PHE350) to (MET485) STRUCTURE OF THE LIMK1-ATPGAMMAS-CFL1 COMPLEX | KINASE COMPLEX, TRANSFERASE
5lcj:A (GLY37) to (VAL173) IN-GEL ACTIVITY-BASED PROTEIN PROFILING OF A CLICKABLE COVALENT ERK 1/2 INHIBITOR | ERK1/2 COVALENT INHIBITOR, TRANSFERASE
5lpy:A (GLY895) to (SER1035) CRYSTAL STRUCTURE OF THE BRI1 KINASE DOMAIN (865-1160) IN COMPLEX WITH ATP FROM ARABIDOPSIS THALIANA | BRASSINOSTEROID RECEPTOR, KINASE DOMAIN, DUAL-SPECIFICIFY KINASE, MEMBRANE RECEPTOR KINASE, PLASMA MEMBRANE, TRANSFERASE
5lpz:A (GLY895) to (SER1035) CRYSTAL STRUCTURE OF THE BRI1 KINASE DOMAIN (865-1196) IN COMPLEX WITH ADP FROM ARABIDOPSIS THALIANA | BRASSINOSTEROID RECEPTOR, KINASE DOMAIN, DUAL-SPECIFICIFY KINASE, MEMBRANE RECEPTOR KINASE, PLASMA MEMBRANE, TRANSFERASE
5lwm:A (GLY834) to (LEU976) CRYSTAL STRUCTURE OF JAK3 IN COMPLEX WITH COMPOUND 4 (FM381) | TRANSFERASE, KINASE, JAK3, COVALENT INHIBITOR, REVERSIBLE COVALENT INHIBITOR, INDUCED POCKET, ARGININE POCKET, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
5toz:A (PHE833) to (LEU976) JAK3 WITH COVALENT INHIBITOR PF-06651600 | JAK3 COVALENT KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3eb0:A (PHE20) to (LYS191) CRYSTAL STRUCTURE OF CGD4_240 FROM CRYPTOSPORIDIUM PARVUM IN COMPLEX WITH INDIRUBIN E804 | KINASE CRYPTOSPORIDIUM PARVUM, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, UNKNOWN FUNCTION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
3eb0:C (PHE20) to (LYS191) CRYSTAL STRUCTURE OF CGD4_240 FROM CRYPTOSPORIDIUM PARVUM IN COMPLEX WITH INDIRUBIN E804 | KINASE CRYPTOSPORIDIUM PARVUM, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, UNKNOWN FUNCTION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
2oib:A (GLY198) to (GLU337) CRYSTAL STRUCTURE OF IRAK4 KINASE DOMAIN APO FORM | KINASE, HELIC C, TRANSFERASE
2oib:B (GLY198) to (SER336) CRYSTAL STRUCTURE OF IRAK4 KINASE DOMAIN APO FORM | KINASE, HELIC C, TRANSFERASE
2oib:D (GLY198) to (GLU337) CRYSTAL STRUCTURE OF IRAK4 KINASE DOMAIN APO FORM | KINASE, HELIC C, TRANSFERASE
3rvg:A (GLY861) to (GLN1003) CRYSTALS STRUCTURE OF JAK2 WITH A 1-AMINO-5H-PYRIDO[4,3-B]INDOL-4- CARBOXAMIDE INHIBITOR | TYROSINE KINASE, JANUS KINASE 2, ENZYME INHIBITORS, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
2oxx:A (SER51) to (PHE181) PROTEIN KINASE CK2 IN COMPLEX WITH TETRABROMOBENZOIMIDAZOLE DERIVATIVES K17, K22 AND K32 | PROTEIN KINASE CK2, INHIBITORS, TETRABROMOBENZOIMIDAZOLE DERIVATIVES, TRANSFERASE
1nxk:A (LEU79) to (THR215) CRYSTAL STRUCTURE OF STAUROSPORINE BOUND TO MAP KAP KINASE 2 | PROTEIN KINASE, MK2, PHOSPHORYLATION, STAUROSPORINE, TRANSFERASE
1nxk:B (LEU79) to (THR215) CRYSTAL STRUCTURE OF STAUROSPORINE BOUND TO MAP KAP KINASE 2 | PROTEIN KINASE, MK2, PHOSPHORYLATION, STAUROSPORINE, TRANSFERASE
3eyh:A (LEU891) to (THR1030) CRYSTAL STRUCTURES OF JAK1 AND JAK2 INHIBITOR COMPLEXES | JAK KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
2pk9:A (ALA19) to (GLY159) STRUCTURE OF THE PHO85-PHO80 CDK-CYCLIN COMPLEX OF THE PHOSPHATE-RESPONSIVE SIGNAL TRANSDUCTION PATHWAY | CYCLIN-DEPENDENT KINASE, CYCLIN, SIGNALING PROTEIN, TRANSFERASE/ CELL CYCLE COMPLEX, SIGNALING PROTEIN, TRANSFERASE/CELL CYCLE COMPLEX
2pk9:C (THR20) to (GLY159) STRUCTURE OF THE PHO85-PHO80 CDK-CYCLIN COMPLEX OF THE PHOSPHATE-RESPONSIVE SIGNAL TRANSDUCTION PATHWAY | CYCLIN-DEPENDENT KINASE, CYCLIN, SIGNALING PROTEIN, TRANSFERASE/ CELL CYCLE COMPLEX, SIGNALING PROTEIN, TRANSFERASE/CELL CYCLE COMPLEX
2pvm:A (SER51) to (PHE181) STRUCTURE-BASED DESIGN OF PYRAZOLO[1,5-A][1,3,5]TRIAZINE DERIVATIVES AS POTENT INHIBITORS OF PROTEIN KINASE CK2 | STRUCTURE-BASED DRUG DESIGN, ENZYME-INHIBITOR COMPLEX, CASEIN KINASE II, PROTEIN KINASE CK2, TRANSFERASE
3fup:A (GLY861) to (GLN1003) CRYSTAL STRUCTURES OF JAK1 AND JAK2 INHIBITOR COMPLEXES | KINASE, PTK DOMAIN, PROTEIN-INHIBITOR COMPLEX, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO- ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3fup:B (THR875) to (GLN1003) CRYSTAL STRUCTURES OF JAK1 AND JAK2 INHIBITOR COMPLEXES | KINASE, PTK DOMAIN, PROTEIN-INHIBITOR COMPLEX, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO- ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3fyk:X (LEU79) to (THR215) CRYSTAL STRUCTURE OF A BENZTHIOPHENE LEAD BOUND TO MAPKAP KINASE-2 (MK-2) | MK-2, MK2, MAPKAP-2, SER/THR KINASE, MAP KINASE, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4xp2:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH AN INHIBITOR | SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4xs2:A (PHE197) to (SER336) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4xs2:D (GLY198) to (SER336) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4imy:C (GLU32) to (ALA173) THE AFF4 SCAFFOLD BINDS HUMAN P-TEFB ADJACENT TO HIV TAT | TRANSCRIPTIONAL CDK9-CYCT1 COMPLEX, PHOSPHORYLATED, INTRINSICALLY DISORDERED AFF4, REGULATION OF TRANSCRIPTION ELONGATION, SER/THR KINASE, PHOSPHORYLATION OF POLII-CTD, DSIF, AND NELF, HIV-1 TAT, HOST-VIRUS INTERACTION, PHOSPHOPROTEIN, NUCLEUS, TRANSFERASE
1phk:A (ARG35) to (GLN173) TWO STRUCTURES OF THE CATALYTIC DOMAIN OF PHOSPHORYLASE, KINASE: AN ACTIVE PROTEIN KINASE COMPLEXED WITH NUCLEOTIDE, SUBSTRATE-ANALOGUE AND PRODUCT | GLYCOGEN METABOLISM, TRANSFERASE, SERINE/THREONINE-PROTEIN, KINASE, ATP-BINDING, CALMODULIN-BINDING
4ivc:A (GLY887) to (THR1030) JAK1 KINASE (JH1 DOMAIN) IN COMPLEX WITH THE INHIBITOR (TRANS-4-{2- [(1R)-1-HYDROXYETHYL]IMIDAZO[4,5-D]PYRROLO[2,3-B]PYRIDIN-1(6H)- YL}CYCLOHEXYL)ACETONITRILE | PROTEIN KINASE, PHOSPHO TRANSFER, PHOSPHO TYROSINE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jia:A (GLY861) to (PRO1002) JAK2 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 9 | PROTEIN KINASE, PHOSPHOTRANSFER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3u4u:A (SER51) to (PHE181) CASEIN KINASE 2 IN COMPLEX WITH AZ-INHIBITOR | KINASE, TRANSFERASE, INHIBITOR BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3u9c:A (SER51) to (PHE181) STRUCTURE OF A C-TERMINAL DELETION MUTANT OF HUMAN PROTEIN KINASE CK2 CATALYTIC SUBUNIT WITH THE ATP-COMPETITIVE INHIBITOR RESORUFIN | PROTEIN KINASE CK2 CASEIN KINASE 2, EUKARYOTIC PROTEIN KINASE FOLD, ATP:PROTEIN PHOSPHOTRANSFERASE, PROTEIN KINASE, ATP CK2BETA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3u9c:B (SER51) to (PHE181) STRUCTURE OF A C-TERMINAL DELETION MUTANT OF HUMAN PROTEIN KINASE CK2 CATALYTIC SUBUNIT WITH THE ATP-COMPETITIVE INHIBITOR RESORUFIN | PROTEIN KINASE CK2 CASEIN KINASE 2, EUKARYOTIC PROTEIN KINASE FOLD, ATP:PROTEIN PHOSPHOTRANSFERASE, PROTEIN KINASE, ATP CK2BETA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2eu9:A (GLY168) to (ASP327) CRYSTAL STRUCTURE OF CLK3 | KINASE DOMAIN, TRANSFERASE
4yti:A (PHE860) to (GLN1003) DISCOVERY OF VX-509 (DECERNOTINIB): A POTENT AND SELECTIVE JANUS KINASE (JAK) 3 INHIBITOR FOR THE TREATMENT OF AUTOIMMUNE DISEASE | JANUS KINASE, JAK2, JAK3, KINASE, INHIBITOR, AUTOIMMUNE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
2f9g:A (GLY25) to (ILE161) CRYSTAL STRUCTURE OF FUS3 PHOSPHORYLATED ON TYR182 | MAP KINASE, TRANSFERASE
3i60:A (GLY35) to (ALA172) CRYSTAL STRUCTURE OF ERK2 BOUND TO (S)-4-(2-(2-CHLOROPHENYLAMINO)-5- METHYLPYRIMIDIN-4-YL)-N-(2-HYDROXY-1-PHENYLETHYL)-1H-PYRROLE-2- CARBOXAMIDE | KINASE, INHIBITOR, ATP-BINDING, CELL CYCLE, HOST-VIRUS INTERACTION, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2vx3:C (GLY171) to (GLN313) CRYSTAL STRUCTURE OF THE HUMAN DUAL SPECIFICITY TYROSINE- PHOSPHORYLATION-REGULATED KINASE 1A | SERINE/THREONINE-PROTEIN KINASE, MINIBRAIN HOMOLOG, NUCLEOTIDE-BINDING, TRANSFERASE, PHOSPHOPROTEIN, TYROSINE-PROTEIN KINASE, CASP8, KINASE
2gph:A (GLY35) to (VAL171) DOCKING MOTIF INTERACTIONS IN THE MAP KINASE ERK2 | ERK2, DOCKING INTERACTION, D-MOTIF, ALLOSTERY, CD-SITE, PHOSPHATASE-DERIVED PEPTIDE, PROCESSING CONFORMATION, TRANSFERASE
3iok:A (GLY861) to (GLN1003) 2-AMINOPYRAZOLO[1,5-A]PYRIMIDINES AS POTENT AND SELECTIVE INHIBITORS OF JAK2 | KINASE, INHIBITOR, JAK2, JANUS KINASE, ATP-BINDING, DISEASE MUTATION, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
2wip:A (GLY27) to (GLY153) STRUCTURE OF CDK2-CYCLIN A COMPLEXED WITH 8-ANILINO-1- METHYL-4,5-DIHYDRO-1H-PYRAZOLO[4,3-H] QUINAZOLINE-3- CARBOXYLIC ACID | CELL CYCLE, ATP-BINDING, TRANSFERASE, POLYMORPHISM, PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN 2 KINASE, SERINE/THREONINE-PROTEIN KINASE, CELL DIVISION, PHOSPHOPROTEIN, PROTEIN KINASE, KINASE, CYCLIN, NUCLEUS, MITOSIS, CYTOPLASM
2wip:C (VAL17) to (GLY153) STRUCTURE OF CDK2-CYCLIN A COMPLEXED WITH 8-ANILINO-1- METHYL-4,5-DIHYDRO-1H-PYRAZOLO[4,3-H] QUINAZOLINE-3- CARBOXYLIC ACID | CELL CYCLE, ATP-BINDING, TRANSFERASE, POLYMORPHISM, PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN 2 KINASE, SERINE/THREONINE-PROTEIN KINASE, CELL DIVISION, PHOSPHOPROTEIN, PROTEIN KINASE, KINASE, CYCLIN, NUCLEUS, MITOSIS, CYTOPLASM
5a4l:B (GLY171) to (LEU314) DYRK1A IN COMPLEX WITH FLUORO BENZOTHIAZOLE FRAGMENT | TRANSFERASE
4md9:E (SER51) to (PHE181) CRYSTAL STRUCTURE OF SYMMETRIC CK2 HOLOENZYME WITH MUTATED ALPHA SUBUNIT (F121E TRUNCATED AT AA 336) | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
4md9:F (GLU55) to (PHE181) CRYSTAL STRUCTURE OF SYMMETRIC CK2 HOLOENZYME WITH MUTATED ALPHA SUBUNIT (F121E TRUNCATED AT AA 336) | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
4md9:H (SER51) to (PHE181) CRYSTAL STRUCTURE OF SYMMETRIC CK2 HOLOENZYME WITH MUTATED ALPHA SUBUNIT (F121E TRUNCATED AT AA 336) | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
4md9:L (SER51) to (PHE181) CRYSTAL STRUCTURE OF SYMMETRIC CK2 HOLOENZYME WITH MUTATED ALPHA SUBUNIT (F121E TRUNCATED AT AA 336) | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
4md9:P (GLU55) to (PHE181) CRYSTAL STRUCTURE OF SYMMETRIC CK2 HOLOENZYME WITH MUTATED ALPHA SUBUNIT (F121E TRUNCATED AT AA 336) | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
4n4s:A (GLY35) to (ALA172) A DOUBLE MUTANT RAT ERK2 IN COMPLEX WITH A PYRAZOLO[3,4-D]PYRIMIDINE INHIBITOR | SERINE/THREONINE KINASE, MAP KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4n4s:B (GLY35) to (ALA172) A DOUBLE MUTANT RAT ERK2 IN COMPLEX WITH A PYRAZOLO[3,4-D]PYRIMIDINE INHIBITOR | SERINE/THREONINE KINASE, MAP KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3zep:A (SER835) to (LEU976) CRYSTAL STRUCTURE OF JAK3 KINASE DOMAIN IN COMPLEX WITH A PYRROLOPYRAZINE-2-PHENYL ETHER INHIBITOR | TRANSFERASE, STAT5, STAT6, INTERLEUKIN-2, COMMON-GAMMA CHAIN, ATP SITE KINASE INHIBITOR, CANCER, SCID, SEVERE COMBINED IMMUNODEFICIENCY
3zep:D (SER835) to (LEU976) CRYSTAL STRUCTURE OF JAK3 KINASE DOMAIN IN COMPLEX WITH A PYRROLOPYRAZINE-2-PHENYL ETHER INHIBITOR | TRANSFERASE, STAT5, STAT6, INTERLEUKIN-2, COMMON-GAMMA CHAIN, ATP SITE KINASE INHIBITOR, CANCER, SCID, SEVERE COMBINED IMMUNODEFICIENCY
5bue:A (GLY35) to (ALA172) ERK2 COMPLEXED WITH N-BENZYLPYRIDONE TETRAHYDROAZAINDAZOLE | ERK KINASE, ATP INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3kc3:B (ASN75) to (THR215) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:D (ASN75) to (THR214) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:E (LYS77) to (THR215) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:F (LYS77) to (THR214) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:H (LEU79) to (THR215) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:J (LYS77) to (THR215) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:L (GLY76) to (THR214) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
5ctp:A (GLU55) to (PHE181) CRYSTAL STRUCTURE OF CK2ALPHA WITH N-(3-(3-CHLORO-4-(PHENYL) BENZYLAMINO)PROPYL)ACETAMIDE BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
5cu0:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF CK2ALPHA WITH 2-HYDROXY-5-METHYLBENZOIC ACID AND N-(3-(3-CHLORO-4-(PHENYL)BENZYLAMINO)PROPYL)ACETAMIDE BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
5cu0:B (SER51) to (PHE181) CRYSTAL STRUCTURE OF CK2ALPHA WITH 2-HYDROXY-5-METHYLBENZOIC ACID AND N-(3-(3-CHLORO-4-(PHENYL)BENZYLAMINO)PROPYL)ACETAMIDE BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
3a2c:A (LEU79) to (THR215) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:B (LEU79) to (THR215) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:C (LEU79) to (THR215) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:F (LEU79) to (THR215) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:I (LEU79) to (THR215) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:J (LEU79) to (THR215) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:L (LEU79) to (THR215) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4app:A (GLY333) to (SER466) CRYSTAL STRUCTURE OF THE HUMAN P21-ACTIVATED KINASE 4 IN COMPLEX WITH (S)-N-(5-(3-BENZYL-1-METHYLPIPERAZINE-4- CARBONYL)-6,6-DIMETHYL-1,4,5,6-TETRAHYDROPYRROLO(3,4-C) PYRAZOL-3-YL)-3-PHENOXYBENZAMIDE | TRANSFERASE, PROTEIN KINASE
4aqc:A (PHE860) to (GLN1003) TRIAZOLOPYRIDINE-BASED INHIBITOR OF JANUS KINASE 2 | TRANSFERASE, ATP-BINDING
4azf:A (GLN162) to (TYR301) HUMAN DYRK2 IN COMPLEX WITH LEUCETTINE L41 | TRANSFERASE
3lxk:A (GLY834) to (LEU976) STRUCTURAL AND THERMODYNAMIC CHARACTERIZATION OF THE TYK2 AND JAK3 KINASE DOMAINS IN COMPLEX WITH CP-690550 AND CMP-6 | TYK2, JAK3, INFLAMMATION, CANCER, PAN INHIBITOR, ATP-BINDING, DISEASE MUTATION, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SCID, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
4b7t:A (GLY68) to (GLN206) GLYCOGEN SYNTHASE KINASE 3 BETA COMPLEXED WITH AXIN PEPTIDE AND LEUCETTINE L4 | TRANSFERASE-PEPTIDE COMPLEX, TRANSFERASE, INSULIN PATHWAY, WNT SIGNALING PATHWAY, INHIBITOR
3mb7:A (SER51) to (PHE181) HUMAN CK2 CATALYTIC DOMAIN IN COMPLEX WITH A DIFURANE DERIVATIVE INHIBITOR (AMR) | KINASES, DIFURANE, INHIBITOR, CK2, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4bbf:A (GLY861) to (LEU1001) AMINOALKYLPYRIMIDINE INHIBITOR COMPLEXES WITH JAK2 | TRANSFERASE, INHIBITOR
4bbf:B (GLY861) to (GLN1003) AMINOALKYLPYRIMIDINE INHIBITOR COMPLEXES WITH JAK2 | TRANSFERASE, INHIBITOR
4bbf:C (GLY861) to (GLN1003) AMINOALKYLPYRIMIDINE INHIBITOR COMPLEXES WITH JAK2 | TRANSFERASE, INHIBITOR
4bbf:D (GLY861) to (LEU1001) AMINOALKYLPYRIMIDINE INHIBITOR COMPLEXES WITH JAK2 | TRANSFERASE, INHIBITOR
4qmt:A (GLY36) to (THR170) MST3 IN COMPLEX WITH HESPERADIN | PROTEIN KINASE, MST3, STK24, STERILE 20-LIKE KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4bco:A (VAL17) to (ALA151) STRUCTURE OF CDK2 IN COMPLEX WITH CYCLIN A AND A 2-AMINO-4- HETEROARYL-PYRIMIDINE INHIBITOR | TRANSFERASE-CELL CYCLE COMPLEX, CDK-CYCLIN COMPLEX, CYCLIN-INHIBITOR, STRUCTURE-BASED DRUG DESIGN
4qp7:B (GLY37) to (VAL173) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH 2-(1H-PYRAZOL-4-YL)-5H- PYRROLO[2,3-B]PYRAZINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3be9:A (GLU55) to (PHE181) STRUCTURE-BASED DESIGN AND SYNTHESIS OF NOVEL MACROCYCLIC PYRAZOLO[1,5-A] [1,3,5]TRIAZINE COMPOUNDS AS POTENT INHIBITORS OF PROTEIN KINASE CK2 AND THEIR ANTICANCER ACTIVITIES | STRUCTURE-BASED DRUG DESIGN, ENZYME-INHIBITOR COMPLEX, CASEIN KINASE II, PROTEIN KINASE CK2, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4bgq:A (GLY25) to (SER161) CRYSTAL STRUCTURE OF THE HUMAN CDKL5 KINASE DOMAIN | TRANSFERASE, PHOSPHO-MIMETIC, KINASE
3c9w:A (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK-2 WITH HYPOTHEMYCIN COVALENTLY BOUND | ERK, ACETYLATION, ATP-BINDING, CELL CYCLE, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
3c9w:B (GLY35) to (VAL171) CRYSTAL STRUCTURE OF ERK-2 WITH HYPOTHEMYCIN COVALENTLY BOUND | ERK, ACETYLATION, ATP-BINDING, CELL CYCLE, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
4rio:A (GLY834) to (LEU976) CRYSTAL STRUCTURE OF JAK3 KINASE DOMAIN IN COMPLEX WITH A PYRROLOPYRIDAZINE CARBOXAMIDE INHIBITOR | TRANSFERASE, TRANSFERASE-INHIBITOR COMPLEX
3o71:A (GLY35) to (ALA172) CRYSTAL STRUCTURE OF ERK2/DCC PEPTIDE COMPLEX | PROTEIN-PEPTIDE COMPLEX, KINASE, DCC, TRANSFERASE-PROTEIN BINDING COMPLEX
4d1s:A (PHE860) to (GLN1003) PYRROLE-3-CARBOXAMIDES AS POTENT AND SELECTIVE JAK2 INHIBITORS | TRANSFERASE, KINASE, JAK2, DRUG DISCOVERY, PROTEIN KINASE INHIBITORS, STRUCTURE-ACTIVITY RELATIONSHIP, POLYCYTHEMIA VERA, TUMOUR CELL PROLIFERATION INHIBITION, ANTI-CANCER AGENTS
5hez:A (MET865) to (GLN1003) JAK2 KINASE (JH1 DOMAIN) MUTANT P1057A IN COMPLEX WITH TG101209 | PROTEIN KINASE, INHIBITOR, MUTATION, TYK2, SURROGATE, P1104A, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hez:B (GLY861) to (GLN1003) JAK2 KINASE (JH1 DOMAIN) MUTANT P1057A IN COMPLEX WITH TG101209 | PROTEIN KINASE, INHIBITOR, MUTATION, TYK2, SURROGATE, P1104A, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hez:C (GLY861) to (GLN1003) JAK2 KINASE (JH1 DOMAIN) MUTANT P1057A IN COMPLEX WITH TG101209 | PROTEIN KINASE, INHIBITOR, MUTATION, TYK2, SURROGATE, P1104A, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hez:D (GLY861) to (GLN1003) JAK2 KINASE (JH1 DOMAIN) MUTANT P1057A IN COMPLEX WITH TG101209 | PROTEIN KINASE, INHIBITOR, MUTATION, TYK2, SURROGATE, P1104A, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3oz6:A (ILE24) to (VAL160) CRYSTAL STRUCTURE OF MAPK FROM CRYPTOSPORIDIUM PARVUM, CGD2_1960 | STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE
3oz6:B (GLY23) to (VAL160) CRYSTAL STRUCTURE OF MAPK FROM CRYPTOSPORIDIUM PARVUM, CGD2_1960 | STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE
4dgn:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF MAIZE CK2 IN COMPLEX WITH THE INHIBITOR LUTEOLIN | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e6d:A (GLY861) to (GLN1003) JAK2 KINASE (JH1 DOMAIN) TRIPLE MUTANT IN COMPLEX WITH COMPOUND 7 | JAK2, KINASE, TRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e6d:B (GLY861) to (GLN1003) JAK2 KINASE (JH1 DOMAIN) TRIPLE MUTANT IN COMPLEX WITH COMPOUND 7 | JAK2, KINASE, TRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e6q:A (GLY861) to (PRO1002) JAK2 KINASE (JH1 DOMAIN) TRIPLE MUTANT IN COMPLEX WITH COMPOUND 12 | JAK2, KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e6q:B (GLY861) to (GLN1003) JAK2 KINASE (JH1 DOMAIN) TRIPLE MUTANT IN COMPLEX WITH COMPOUND 12 | JAK2, KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3q9x:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF HUMAN CK2 ALPHA IN COMPLEX WITH EMODIN AT PH 6.5 | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4f9b:A (SER70) to (GLY202) HUMAN CDC7 KINASE IN COMPLEX WITH DBF4 AND PHA767491 | SER/THR PROTEIN KINASE, TRANSFERASE, PHOSPHORYLATION, CELL CYCLE, CELL DIVISION, MITOSIS, S PHASE, SERINE/THREONINE-PROTEIN KINASE, DBF4-DEPENDENT KINASE, DDK, ATP-BINDING, NUCLEOTIDE-BINDING, ZINC- BINDING, NUCLEUS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4f9b:C (SER70) to (THR203) HUMAN CDC7 KINASE IN COMPLEX WITH DBF4 AND PHA767491 | SER/THR PROTEIN KINASE, TRANSFERASE, PHOSPHORYLATION, CELL CYCLE, CELL DIVISION, MITOSIS, S PHASE, SERINE/THREONINE-PROTEIN KINASE, DBF4-DEPENDENT KINASE, DDK, ATP-BINDING, NUCLEOTIDE-BINDING, ZINC- BINDING, NUCLEUS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4f9c:A (SER70) to (GLY202) HUMAN CDC7 KINASE IN COMPLEX WITH DBF4 AND XL413 | SER/THR PROTEIN KINASE, TRANSFERASE, PHOSPHORYLATION, CELL CYCLE, CELL DIVISION, MITOSIS, S PHASE, SERINE/THREONINE-PROTEIN KINASE, DBF4-DEPENDENT KINASE, DDK, ATP-BINDING, NUCLEOTIDE-BINDING, ZINC- BINDING, NUCLEUS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r0t:A (SER51) to (PHE181) CRYSTAL STRUCTURE OF HUMAN PROTEIN KINASE CK2 ALPHA SUBUNIT IN COMPLEX WITH THE INHIBITOR CX-5279 | KINASE, CK2-INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:A (LEU79) to (THR215) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:B (LEU79) to (THR215) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:D (LEU79) to (THR215) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:F (LEU79) to (THR215) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:I (LEU79) to (THR215) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:J (LYS77) to (THR215) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:K (LEU79) to (THR215) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:L (LYS77) to (THR215) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fv5:A (GLY35) to (ALA172) CRYSTAL STRUCTURE OF THE ERK2 COMPLEXED WITH EK9 | TRANSFERASE
5k4i:A (GLY37) to (ALA174) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH COMPOUND 22 | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gj3:A (GLY909) to (PRO1049) TYK2 (JH1) IN COMPLEX WITH 2,6-DICHLORO-4-CYANO-N-[2-({[(1R,2R)-2- FLUOROCYCLOPROPYL]CARBONYL}AMINO)PYRIDIN-4-YL]BENZAMIDE | KINASE, ATP BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5khx:A (LYS888) to (THR1030) CRYSTAL STRUCTURE OF JAK1 IN COMPLEX WITH PF-4950736 | JAK1, KINASE, INHIBITOR, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5kx7:B (GLY198) to (SER336) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5lck:A (GLY37) to (VAL173) A CLICKABLE COVALENT ERK 1/2 INHIBITOR | ERK2 COVALENT INHIBITOR, TRANSFERASE
5lwn:A (GLY834) to (LEU976) CRYSTAL STRUCTURE OF JAK3 IN COMPLEX WITH COMPOUND 5 (FM409) | TRANSFERASE, JAK3, COVALENT INHIBITOR, REVERSIBLE COVALENT INHIBITOR, INDUCED POCKET, ARGININE POCKET, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC