3rkb:A    (SER46) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR RC-2-73  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4wb6:B    (GLN84) to   (HIS294)  CRYSTAL STRUCTURE OF A L205R MUTANT OF HUMAN CAMP-DEPENDENT PROTEIN KINASE A (CATALYTIC ALPHA SUBUNIT)  |   CUSHING'S SYNDROME, PROTEIN KINASE, PHOSPHORYLATION, MUTANT, ADENOSINE TRIPHOSPHATE, CATALYSIS 
4wb7:A   (ILE140) to   (HIS349)  CRYSTAL STRUCTURE OF A CHIMERIC FUSION OF HUMAN DNAJ (HSP40) AND CAMP- DEPENDENT PROTEIN KINASE A (CATALYTIC ALPHA SUBUNIT)  |   CHAPERONE, CATALYSIS, PROTEIN KINASE, ADENOSINE TRIPHOSPHATE, PHOSPHORYLATION, CHIMERA, FUSION, FIBROLAMELLAR HEPATOCELLULAR CARINOMA 
4wb7:B   (ILE140) to   (HIS349)  CRYSTAL STRUCTURE OF A CHIMERIC FUSION OF HUMAN DNAJ (HSP40) AND CAMP- DEPENDENT PROTEIN KINASE A (CATALYTIC ALPHA SUBUNIT)  |   CHAPERONE, CATALYSIS, PROTEIN KINASE, ADENOSINE TRIPHOSPHATE, PHOSPHORYLATION, CHIMERA, FUSION, FIBROLAMELLAR HEPATOCELLULAR CARINOMA 
3e8c:D    (ILE85) to   (HIS294)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, PROTEIN KINASE INHIBITOR 
3e8c:F    (GLN84) to   (HIS294)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, PROTEIN KINASE INHIBITOR 
3e8e:E    (GLN84) to   (HIS294)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
4gu6:B   (ASP462) to   (GLN686)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH N-{3-[(5-CYANO- 2-PHENYL-1H-PYRROLO[2,3-B]PYRIDIN-4-YLAMINO)- METHYL]-PYRIDIN-2-YL}- N-METHYL-METHANESULFONAMIDE  |   PROTEIN TYROSINE KINASE, ATP BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4gu9:A   (ASP462) to   (ALA685)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH (2-FLUORO- PHENYL)-(1H-PYRAZOLO[3,4-D]PYRIMIDIN-4-YL)-AMINE  |   PROTEIN TYROSINE KINASE, TRANSFERASE, ATP BINDING 
4gu9:B   (ASP462) to   (GLU683)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH (2-FLUORO- PHENYL)-(1H-PYRAZOLO[3,4-D]PYRIMIDIN-4-YL)-AMINE  |   PROTEIN TYROSINE KINASE, TRANSFERASE, ATP BINDING 
2oh4:A   (THR873) to  (GLN1167)  CRYSTAL STRUCTURE OF VEGFR2 WITH A BENZIMIDAZOLE-UREA INHIBITOR  |   VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2 TYROSINE-PROTEIN KINASE 3D-STRUCTURE VEGFR2 ANGIOGENESIS ATP-BINDING PHOSPHORYLATION EC 2.7.1.112 VEGFR-2 KINASE INSERT DOMAIN RECEPTOR PROTEIN-TYROSINE KINASE RECEPTOR FLK-1, TRANSFERASE 
2oiq:A   (SER303) to   (TYR519)  CRYSTAL STRUCTURE OF CHICKEN C-SRC KINASE DOMAIN IN COMPLEX WITH THE CANCER DRUG IMATINIB.  |   SRC,KINASE,IMATINIB,INACTIVE, TRANSFERASE 
3efj:A  (ILE1118) to  (SER1342)  STRUCTURE OF C-MET WITH PYRIMIDONE INHIBITOR 7  |   C-MET, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3efk:B  (ILE1118) to  (SER1342)  STRUCTURE OF C-MET WITH PYRIMIDONE INHIBITOR 50  |   C-MET, KINASE INHIBITOR PYRIMIDONE, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3efl:A   (THR875) to  (HIS1178)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH MOTESANIB  |   ANGIOGENESIS, MOTESANIB, NICOTINAMIDE, RECEPTOR TYROSINE KINASE, TRANSFERASE 
3efl:B   (HIS876) to  (GLN1165)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH MOTESANIB  |   ANGIOGENESIS, MOTESANIB, NICOTINAMIDE, RECEPTOR TYROSINE KINASE, TRANSFERASE 
1agw:A   (GLU522) to   (THR761)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF FIBROBLAST GROWTH FACTOR RECEPTOR 1 IN COMPLEX WITH SU4984 INHIBITOR  |   PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE, ATP- BINDING, PHOSPHORYLATION, INHIBITOR 
1agw:B   (GLU522) to   (THR761)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF FIBROBLAST GROWTH FACTOR RECEPTOR 1 IN COMPLEX WITH SU4984 INHIBITOR  |   PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE, ATP- BINDING, PHOSPHORYLATION, INHIBITOR 
4h1j:A   (THR464) to   (ALA690)  CRYSTAL STRUCTURE OF PYK2 WITH THE PYRAZOLE 13A  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3rzb:A    (THR47) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR RC-2-23  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2b53:A    (PRO45) to   (HIS283)  HUMAN CYCLIN DEPENDENT KINASE 2 (CDK2) COMPLEXED WITH DIN- 234325  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION, TRANSFERASE 
2b55:A    (PRO45) to   (HIS283)  HUMAN CYCLIN DEPENDENT KINASE 2 (CDK2) COMPLEXED WITH INDENOPYRAXOLE DIN-101312  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION, TRANSFERASE 
3en4:A   (SER303) to   (TYR519)  TARGETED POLYPHARMACOLOGY: CRYSTAL STRUCTURE OF THE C-SRC KINASE DOMAIN IN COMPLEX WITH PP121, A MULTITARGETED KINASE INHIBITOR  |   SRC, TYROSINE, KINASE, POLYPHARMACOLOGY, INHIBITOR, MULTITARGET, PHOSPHOINOSITIDE, TRANSFERASE, SIGNALING, PYRAZOLOPYRIMIDINE, KINASE-INHIBITOR COMPLEX, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TYROSINE-PROTEIN KINASE 
3en4:B   (SER303) to   (TYR519)  TARGETED POLYPHARMACOLOGY: CRYSTAL STRUCTURE OF THE C-SRC KINASE DOMAIN IN COMPLEX WITH PP121, A MULTITARGETED KINASE INHIBITOR  |   SRC, TYROSINE, KINASE, POLYPHARMACOLOGY, INHIBITOR, MULTITARGET, PHOSPHOINOSITIDE, TRANSFERASE, SIGNALING, PYRAZOLOPYRIMIDINE, KINASE-INHIBITOR COMPLEX, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TYROSINE-PROTEIN KINASE 
3en5:B   (SER303) to   (TYR519)  TARGETED POLYPHARMACOLOGY: CRYSTAL STRUCTURE OF THE C-SRC KINASE DOMAIN IN COMPLEX WITH PP494, A MULTITARGETED KINASE INHIBITOR  |   SRC, TYROSINE, KINASE, POLYPHARMACOLOGY, INHIBITOR, MULTITARGET, PHOSPHOINOSITIDE, TRANSFERASE, SIGNALING, PYRAZOLOPYRIMIDINE, KINASE-INHIBITOR COMPLEX, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TYROSINE-PROTEIN KINASE 
3en7:A   (PHE307) to   (TYR519)  TARGETED POLYPHARMACOLOGY: CRYSTAL STRUCTURE OF THE C-SRC KINASE DOMAIN IN COMPLEX WITH S1, A MULTITARGETED KINASE INHIBITOR  |   SRC, TYROSINE, KINASE, POLYPHARMACOLOGY, INHIBITOR, MULTITARGET, PHOSPHOINOSITIDE, TRANSFERASE, SIGNALING, PYRAZOLOPYRIMIDINE, KINASE-INHIBITOR COMPLEX, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TYROSINE-PROTEIN KINASE 
3enm:A    (ASN89) to   (HIS311)  THE STRUCTURE OF THE MAP2K MEK6 REVEALS AN AUTOINHIBITORY DIMER  |   MEK6, AUTOINHIBITED DIMER, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3enm:C    (GLN91) to   (HIS311)  THE STRUCTURE OF THE MAP2K MEK6 REVEALS AN AUTOINHIBITORY DIMER  |   MEK6, AUTOINHIBITED DIMER, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE 
4wun:A   (THR521) to   (LEU760)  STRUCTURE OF FGFR1 IN COMPLEX WITH AZD4547 (N-{3-[2-(3,5- DIMETHOXYPHENYL)ETHYL]-1H-PYRAZOL-5-YL}-4-[(3R,5S)-3,5- DIMETHYLPIPERAZIN-1-YL]BENZAMIDE) AT 1.65 ANGSTROM  |   TRANSFERASE; TRANSFERASE INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2p2i:A   (THR875) to  (HIS1177)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A NICOTINAMIDE INHIBITOR  |   RECEPTOR TYROSINE KINASE, KDR, TRANSFERASE 
4hct:A   (GLU406) to   (SER618)  CRYSTAL STRUCTURE OF ITK IN COMPLEX WITH COMPOUND 52  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4hcu:A   (GLU406) to   (SER618)  CRYSTAL STRUCTURE OF ITK IN COMPLEXT WITH COMPOUND 40  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4hcv:A   (ALA407) to   (SER618)  CRYSTAL STRUCTURE OF ITK IN COMPLEX WITH COMPOUND 53  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ewh:A   (THR875) to  (GLN1170)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A PYRIDYL-PYRIMIDINE BENZIMIDAZOLE INHIBITOR  |   ANGIOGENESIS, RECEPTOR TYROSINE KINASE, DFG-OUT, TRANSFERASE 
3s2p:A    (PRO45) to   (GLN287)  CRYSTAL STRUCTURE OF CDK2 WITH A 2-AMINOPYRIMIDINE COMPOUND  |   PROTEIN KINASE, TRANSFERASE, CELL DIVISION PROTEIN KINASE 2, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1blx:A    (ILE59) to   (HIS297)  P19INK4D/CDK6 COMPLEX  |   INHIBITOR PROTEIN, CYCLIN-DEPENDENT KINASE, CELL CYCLE CONTROL, ALPHA/BETA, COMPLEX (INHIBITOR PROTEIN/KINASE) 
3f3u:A   (SER303) to   (TYR519)  KINASE DOMAIN OF CSRC IN COMPLEX WITH INHIBITOR RL37 (TYPE III)  |   ALLOSTERIC, TYPE III, DFG-OUT, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3f3u:B   (SER303) to   (TYR519)  KINASE DOMAIN OF CSRC IN COMPLEX WITH INHIBITOR RL37 (TYPE III)  |   ALLOSTERIC, TYPE III, DFG-OUT, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3f3v:A   (SER303) to   (TYR519)  KINASE DOMAIN OF CSRC IN COMPLEX WITH INHIBITOR RL45 (TYPE II)  |   ALLOSTERIC, TYPE II, DFG-OUT, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3f3v:B   (SER303) to   (TYR519)  KINASE DOMAIN OF CSRC IN COMPLEX WITH INHIBITOR RL45 (TYPE II)  |   ALLOSTERIC, TYPE II, DFG-OUT, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3f3w:B   (SER303) to   (TYR519)  DRUG RESISTANT CSRC KINASE DOMAIN IN COMPLEX WITH INHIBITOR RL45 (TYPE II)  |   ALLOSTERIC, TYPE II, DFG-OUT, DRUG RESISTANCE MUTATION, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE 
3f5u:A    (ARG58) to   (HIS272)  CRYSTAL STRUCTURE OF THE DEATH ASSOCIATED PROTEIN KINASE IN COMPLEX WITH AMPPNP AND MG2+  |   KINASE-AMPPNP COMPLEX, ALTERNATIVE SPLICING, ANK REPEAT, APOPTOSIS, ATP-BINDING, CALMODULIN-BINDING, CYTOPLASM, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3f66:A  (ASP1117) to  (THR1343)  HUMAN C-MET KINASE IN COMPLEX WITH QUINOXALINE INHIBITOR  |   C-MET, PROTEIN KINASE, QUINOXALINE, ALTERNATIVE SPLICING; ATP-BINDING; CHROMOSOMAL REARRANGEMENT; DISEASE MUTATION; GLYCOPROTEIN; KINASE; MEMBRANE; NUCLEOTIDE-BINDING; PHOSPHOPROTEIN; POLYMORPHISM; PROTO-ONCOGENE; RECEPTOR; REPEAT; SIGNAL; TRANSFERASE; TRANSMEMBRANE; TYROSINE- PROTEIN KINASE. 
4x6q:C    (GLU86) to   (ALA298)  AN ISOFORM-SPECIFIC MYRISTYLATION SWITCH TARGETS RIIB PKA HOLOENZYMES TO MEMBRANES  |   PKA, MEMBRANE BINDING, MOLECULAR SWITCH, TRANSFERASE 
4x6r:A    (ILE85) to   (ALA298)  AN ISOFORM-SPECIFIC MYRISTYLATION SWITCH TARGETS RIIB PKA HOLOENZYMES TO MEMBRANES  |   PKA, MEMBRANE BINDING, MOLECULAR SWITCH, TRANSFERASE 
3f82:A  (GLY1119) to  (PHE1344)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF THE HEPATOCYTE GROWTH FACTOR RECEPTOR C-MET IN COMPLEX WITH N- (4-(2-AMINO-3-CHLOROPYRIDIN-4-YLOXY)-3-FLUOROPHENYL)-4- ETHOXY-1-(4-FLUOROPHENYL)-2-OXO-1,2-DIHYDROPYRIDINE-3- CARBOXAMIDE  |   ALTERNATIVE SPLICING, RECEPTOR TYROSINE KINASE, SIGNAL TRANSDUCTION, GRB2, SHC, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
2btr:A    (ALA48) to   (GLN287)  STRUCTURE OF CDK2 COMPLEXED WITH PNU-198873  |   PROTEIN KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN 2 KINASE, PHOSPHORYLATION, CELL DIVISION 
2bts:A    (THR47) to   (GLN287)  STRUCTURE OF CDK2 COMPLEXED WITH PNU-230032  |   PROTEIN KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN 2 KINASE, PHOSPHORYLATION, CELL DIVISION, ATP-BINDING, CELL CYCLE, MITOSIS, POLYMORPHISM 
3fc1:X    (SER61) to   (SER261)  CRYSTAL STRUCTURE OF P38 KINASE BOUND TO PYRIMIDO-PYRIDAZINONE INHIBITOR  |   KINASE INHIBITOR, ATP-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
4hzs:A   (GLN167) to   (ALA388)  CRYSTAL STRUCTURE OF ACK1 KINASE DOMAIN WITH C-TERMINAL SH3 DOMAIN  |   INACTIVE STATE, ALLOSTERY, DIMERIZATION, OLIGOMERIZATION, NEGATIVE REGULATION, ACTIVATION, PHOSPHOTRANSFER, TRANSFERASE 
4hzs:B   (GLN167) to   (ALA388)  CRYSTAL STRUCTURE OF ACK1 KINASE DOMAIN WITH C-TERMINAL SH3 DOMAIN  |   INACTIVE STATE, ALLOSTERY, DIMERIZATION, OLIGOMERIZATION, NEGATIVE REGULATION, ACTIVATION, PHOSPHOTRANSFER, TRANSFERASE 
4hzs:C   (GLN167) to   (ALA388)  CRYSTAL STRUCTURE OF ACK1 KINASE DOMAIN WITH C-TERMINAL SH3 DOMAIN  |   INACTIVE STATE, ALLOSTERY, DIMERIZATION, OLIGOMERIZATION, NEGATIVE REGULATION, ACTIVATION, PHOSPHOTRANSFER, TRANSFERASE 
4hzs:D   (GLN167) to   (ALA388)  CRYSTAL STRUCTURE OF ACK1 KINASE DOMAIN WITH C-TERMINAL SH3 DOMAIN  |   INACTIVE STATE, ALLOSTERY, DIMERIZATION, OLIGOMERIZATION, NEGATIVE REGULATION, ACTIVATION, PHOSPHOTRANSFER, TRANSFERASE 
4i22:A   (ALA755) to   (ARG973)  STRUCTURE OF THE MONOMERIC (V948R)GEFITINIB/ERLOTINIB RESISTANT DOUBLE MUTANT (L858R+T790M) EGFR KINASE DOMAIN CO-CRYSTALLIZED WITH GEFITINIB  |   KINASE DOMAIN, PHOSPHOTRASFER, ATP BINDING, TRANSFERASE 
4i24:A   (ASN756) to   (ARG973)  STRUCTURE OF T790M EGFR KINASE DOMAIN CO-CRYSTALLIZED WITH DACOMITINIB  |   KINASE DOMAIN, PHOSPHOTRASFER, ATP BINDING, TRANSFERASE 
4i24:B   (ASN756) to   (ARG973)  STRUCTURE OF T790M EGFR KINASE DOMAIN CO-CRYSTALLIZED WITH DACOMITINIB  |   KINASE DOMAIN, PHOSPHOTRASFER, ATP BINDING, TRANSFERASE 
1oi9:C    (PRO45) to   (GLN287)  STRUCTURE OF HUMAN THR160-PHOSPHO CDK2/CYCLIN A COMPLEXED WITH A 6-CYCLOHEXYLMETHYLOXY-2-ANILINO-PURINE INHIBITOR  |   KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP- BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, PHOSPHORYLATION 
1oiq:A    (THR47) to   (HIS283)  IMIDAZOPYRIDINES: A POTENT AND SELECTIVE CLASS OF CYCLIN-DEPENDENT KINASE INHIBITORS IDENTIFIED THROUGH STRUCTURE-BASED HYBRIDISATION  |   KINASE, PROTEIN KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, PHOSPHORYLATION, 
1oit:A    (ALA48) to   (HIS283)  IMIDAZOPYRIDINES: A POTENT AND SELECTIVE CLASS OF CYCLIN-DEPENDENT KINASE INHIBITORS IDENTIFIED THROUGH STRUCTURE-BASED HYBRIDISATION  |   KINASE, PROTEIN KINASE 
1oiy:C    (PRO45) to   (GLN287)  STRUCTURE OF HUMAN THR160-PHOSPHO CDK2/CYCLIN A COMPLEXED WITH A 6-CYCLOHEXYLMETHYLOXY-2-ANILINO-PURINE INHIBITOR  |   KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP- BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, PHOSPHORYLATION 
1cdk:A    (ILE85) to   (HIS294)  CAMP-DEPENDENT PROTEIN KINASE CATALYTIC SUBUNIT (E.C.2.7.1.37) (PROTEIN KINASE A) COMPLEXED WITH PROTEIN KINASE INHIBITOR PEPTIDE FRAGMENT 5-24 (PKI(5-24) ISOELECTRIC VARIANT CA) AND MN2+ ADENYLYL IMIDODIPHOSPHATE (MNAMP-PNP) AT PH 5.6 AND 7C AND 4C  |   COMPLEX (TRANSFERASE-INHIBITOR), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1ol6:A   (HIS176) to   (HIS380)  STRUCTURE OF UNPHOSPHORYLATED D274N MUTANT OF AURORA-A  |   TRANSFERASE, CELL CYCLE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION 
4i4e:A   (ARG465) to   (GLN686)  STRUCTURE OF FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH HINGE BINDING PYRAZOLOBENZOTHIAZINE COMPOUND.  |   PHOSPHORYLATED ON TYROSINES, TRANSFERASE, CYTOPLASMIC; LOCALIZED TO FOCAL ADHESIONS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1ckp:A    (SER46) to   (GLN287)  HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR PURVALANOL B  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION, HORMONE-GROWTH FACTOR COMPLEX 
2pzr:B   (THR524) to   (ASN766)  CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC K641R MUTATION RESPONSIBLE FOR PFEIFFER SYNDROME  |   KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, TRANSFERASE 
2c5y:A    (SER46) to   (GLN287)  DIFFERENTIAL BINDING OF INHIBITORS TO ACTIVE AND INACTIVE CDK2 PROVIDES INSIGHTS FOR DRUG DESIGN  |   CDK2, DRUG DESIGN, ATP-BINDING, CELL CYCLE, CELL DIVISION, KINASE, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
2c68:A    (SER46) to   (GLN287)  CRYSTAL STRUCTURE OF THE HUMAN CDK2 COMPLEXED WITH THE TRIAZOLOPYRIMIDINE INHIBITOR  |   TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, CDK2, ATP-BINDING, CELL CYCLE, MITOSIS, PHOSPHORYLATION, TRIAZOLOPYRIMIDINE INHIBITOR, CELL DIVISION, KINASE, POLYMORPHISM, NUCLEOTIDE-BINDING 
2c69:A    (SER46) to   (GLN287)  CRYSTAL STRUCTURE OF THE HUMAN CDK2 COMPLEXED WITH THE TRIAZOLOPYRIMIDINE INHIBITOR  |   TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, CDK2, ATP-BINDING, CELL CYCLE, MITOSIS, PHOSPHORYLATION, TRIAZOLOPYRIMIDINE INHIBITOR, CELL DIVISION, KINASE, POLYMORPHISM, NUCLEOTIDE-BINDING 
2q0b:A   (THR524) to   (THR765)  CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC E565A MUTATION RESPONSIBLE FOR PFEIFFER SYNDROME  |   KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, TRANSFERASE 
2c6k:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF THE HUMAN CDK2 COMPLEXED WITH THE TRIAZOLOPYRIMIDINE INHIBITOR  |   TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, CDK2, ATP-BINDING, CELL CYCLE, MITOSIS, PHOSPHORYLATION, TRIAZOLOPYRIMIDINE INHIBITOR, CELL DIVISION, KINASE, POLYMORPHISM, NUCLEOTIDE-BINDING 
2c6m:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF THE HUMAN CDK2 COMPLEXED WITH THE TRIAZOLOPYRIMIDINE INHIBITOR  |   TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, CDK2, ATP-BINDING, CELL CYCLE, MITOSIS, PHOSPHORYLATION, TRIAZOLOPYRIMIDINE INHIBITOR, CELL DIVISION, KINASE, POLYMORPHISM, NUCLEOTIDE-BINDING 
2c6o:A    (THR47) to   (GLN287)  CRYSTAL STRUCTURE OF THE HUMAN CDK2 COMPLEXED WITH THE TRIAZOLOPYRIMIDINE INHIBITOR  |   SERINE/THREONINE PROTEIN KINASE, CDK2, ATP-BINDING, CELL CYCLE, MITOSIS, PHOSPHORYLATION, TRIAZOLOPYRIMIDINE INHIBITOR, CELL DIVISION, KINASE, TRANSFERASE, NUCLEOTIDE- BINDING 
1ouk:A    (SER61) to   (LEU262)  THE STRUCTURE OF P38 ALPHA IN COMPLEX WITH A PYRIDINYLIMIDAZOLE INHIBITOR  |   MAP KINASE, HYDROPHOBIC POCKET, KINASE DOMAIN, ATP BINDING DOMAIN, TRANSFERASE 
3fxx:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE AND JUXTAMEMBRANE REGION BOUND TO SUBSTRATE KQWDNYE[PTYR]IW  |   RECEPTOR TYROSINE KINASE, JUXTAMEMBRANE SEGMENT, STRUCTURAL GENOMICS, PEPTIDE CO-CRYSTAL STRUCTURE, SUBSTRATE COMPLEX, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, CELL MEMBRANE, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3svv:B   (SER303) to   (TYR519)  CRYSTAL STRUCTURE OF T338C C-SRC COVALENTLY BOUND TO VINYLSULFONAMIDE- PYRAZOLOPYRIMIDINE 9  |   COVALENTLY BOUND LIGAND, CYSTEINE GATEKEEPER, SRC, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
2cch:C    (PRO45) to   (GLN287)  THE CRYSTAL STRUCTURE OF CDK2 CYCLIN A IN COMPLEX WITH A SUBSTRATE PEPTIDE DERIVED FROM CDC MODIFIED WITH A GAMMA- LINKED ATP ANALOGUE  |   COMPLEX(TRANSFERASE/CELL DIVISION), ATP-BINDING, CDK2, CELL CYCLE, CELL DIVISION, CYCLIN, MITOSIS, NUCLEAR PROTEIN, PEPTIDE SPECIFICITY, PHOSPHORYLATION, POLYMORPHISM, PROTEIN KINASE, RECRUITMENT, SERINE-THREONINE-PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
2cci:A    (PRO45) to   (HIS283)  CRYSTAL STRUCTURE OF PHOSPHO-CDK2 CYCLIN A IN COMPLEX WITH A PEPTIDE CONTAINING BOTH THE SUBSTRATE AND RECRUITMENT SITES OF CDC6  |   COMPLEX (TRANSFERASE/CELL DIVISION), PROTEIN KINASES, CELL CYCLE, RECRUITMENT, SUBSTRATE RECOGNITION, ATP-BINDING, CELL DIVISION, KINASE, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE, CYCLIN, DNA REPLICATION, NUCLEAR PROTEIN, COMPLEX 
3fzp:A   (ASP466) to   (GLU692)  CRYSTAL STRUCTURE OF PYK2 COMPLEXED WITH ATPGS  |   KINASE, ATPGS, DFG, ALTERNATIVE SPLICING, ATP-BINDING, CELL MEMBRANE, CYTOPLASM, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3fzr:A   (ASP466) to   (ALA690)  CRYSTAL STRUCTURE OF PYK2 COMPLEXED WITH PF-431396  |   PYK2, KINASE, DFG, ALTERNATIVE SPLICING, ATP-BINDING, CELL MEMBRANE, CYTOPLASM, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3fzt:A   (THR464) to   (ALA690)  CRYSTAL STRUCTURE OF PYK2 COMPLEXED WITH PF-4618433  |   PYK2, KINASE, DFG, ALTERNATIVE SPLICING, ATP-BINDING, CELL MEMBRANE, CYTOPLASM, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3g0f:B   (HIS630) to   (GLN927)  KIT KINASE DOMAIN MUTANT D816H IN COMPLEX WITH SUNITINIB  |   KIT KINASE DOMAIN, SUTENT BINDING, DRUG RESISTANCE, ATP- BINDING, DISEASE MUTATION, GLYCOPROTEIN, IMMUNOGLOBULIN DOMAIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, RECEPTOR, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, TRANSFERASE 
2cjm:C    (PRO45) to   (GLN287)  MECHANISM OF CDK INHIBITION BY ACTIVE SITE PHOSPHORYLATION: CDK2 Y15P T160P IN COMPLEX WITH CYCLIN A STRUCTURE  |   PHOSPHORYLATION, NUCLEOTIDE-BINDING, MITOSIS, CELL CYCLE, REGULATION, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, TRANSFERASE, CELL DIVISION, CYCLIN-DEPENDENT KINASE, COMPLEX (TRANSFERASE/CELL DIVISION) 
1di8:A    (SER46) to   (HIS283)  THE STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 (CDK2) IN COMPLEX WITH 4-[3-HYDROXYANILINO]-6,7-DIMETHOXYQUINAZOLINE  |   SERINE/THREONINE PROTEIN KINASE, CELL CYCLE, ATP-BINDING, TRANSFERASE 
3gc9:B    (SER61) to   (MET288)  THE STRUCTURE OF P38BETA C119S, C162S IN COMPLEX WITH A DIHYDROQUINAZOLINONE INHIBITOR  |   SERINE/THREONINE KINASE, DRUG DESIGN, SELECTIVITY, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
1dm2:A    (PRO45) to   (HIS283)  HUMAN CYCLIN-DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR HYMENIALDISINE  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION 
4xuf:B   (SER652) to   (GLN946)  CRYSTAL STRUCTURE OF THE FLT3 KINASE DOMAIN BOUND TO THE INHIBITOR QUIZARTINIB (AC220)  |   FLT3, RECEPTOR TYROSINE KINASE, AC220, QUIZARTINIB, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3gcu:A    (SER61) to   (LEU262)  HUMAN P38 MAP KINASE IN COMPLEX WITH RL48  |   DFG-OUT, TYPE II, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3gcu:B    (SER61) to   (LEU262)  HUMAN P38 MAP KINASE IN COMPLEX WITH RL48  |   DFG-OUT, TYPE II, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
4xv1:A   (THR491) to   (GLU716)  B-RAF KINASE V600E ONCOGENIC MUTANT IN COMPLEX WITH PLX7904  |   B-RAF, BRAF, PROTO-ONCOGENE, V600E, KINASE, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
2qo2:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE AND JUXTAMEMBRANE REGION, DEPHOSPHORYLATED, APO STRUCTURE  |   RECEPTOR TYROSINE KINASE, JUXTAMEMBRANE SEGMENT, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
2qob:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE DOMAIN, BASE STRUCTURE  |   RECEPTOR TYROSINE KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, MEMBRANE, NUCLEOTIDE- BINDING, PHOSPHORYLATION, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
2qoc:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE DOMAIN, PHOSPHORYLATED, AMP-PNP BOUND STRUCTURE  |   RECEPTOR TYROSINE KINASE, STRUCTURAL GENOMICS, AMP-PNP, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
2qod:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE AND JUXTAMEMBRANE REGION, Y602F MUTANT  |   RECEPTOR TYROSINE KINASE, JUXTAMEMBRANE SEGMENT, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
2qoi:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE AND JUXTAMEMBRANE REGION, Y596F:Y602F DOUBLE MUTANT  |   RECEPTOR TYROSINE KINASE, JUXTAMEMBRANE SEGMENT, STRUCTURAL GENOMICS, MUTANTS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP- BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
2qof:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE AND JUXTAMEMBRANE REGION, Y596F MUTANT  |   RECEPTOR TYROSINE KINASE, JUXTAMEMBRANE SEGMENT, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
2qol:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE AND JUXTAMEMBRANE REGION, Y596:Y602:S768G TRIPLE MUTANT  |   RECEPTOR TYROSINE KINASE, JUXTAMEMBRANE SEGMENT, STRUCTURAL GENOMICS, MUTANT, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP- BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
2qon:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE AND JUXTAMEMBRANE REGION, Y596F:Y602F:Y742A TRIPLE MUTANT  |   RECEPTOR TYROSINE KINASE, JUXTAMEMBRANE SEGMENT, STRUCTURAL GENOMICS, MUTANT, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
2qoo:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE AND JUXTAMEMBRANE REGION, Y596F:Y602F:Y742F TRIPLE MUTANT  |   RECEPTOR TYROSINE KINASE, JUXTAMEMBRANE SEGMENT, STRUCTURAL GENOMICS, MUTANT, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP- BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
2qoq:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE AND JUXTAMEMBRANE REGION, BASE, AMP-PNP BOUND STRUCTURE  |   RECEPTOR TYROSINE KINASE, STRUCTURAL GENOMICS, JUXTAMEMBRANE SEGMENT, AMP-PNP, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE 
1pkg:B   (LEU631) to   (ILE928)  STRUCTURE OF A C-KIT KINASE PRODUCT COMPLEX  |   KINASE, AUTOPHOSPHORYLATION, TRANSACTIVATION, TRANSFERASE ACTIVATOR 
3gen:A   (GLU439) to   (GLU657)  THE 1.6 A CRYSTAL STRUCTURE OF HUMAN BRUTON'S TYROSINE KINASE BOUND TO A PYRROLOPYRIMIDINE-CONTAINING COMPOUND  |   BRUTON'S TYROSINE KINASE, 4-AMINO-5-(4-PHENOXYPHENYL)-5H- PYRROLO[3, 2-D]PYRIMIDIN-7-YL-CYCLOPENTANE, TEC-FAMILY, COMPLEX, ACETYLATION, ATP-BINDING, CYTOPLASM, DISEASE MUTATION, KINASE, MEMBRANE, METAL-BINDING, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, ZINC, ZINC-FINGER 
2qu6:A   (THR875) to  (HIS1178)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A BENZOXAZOLE INHIBITOR  |   RECEPTOR TYROSINE KINASE, KDR, ANGIOGENESIS, ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST- VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
2qu6:B   (HIS876) to  (GLN1165)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A BENZOXAZOLE INHIBITOR  |   RECEPTOR TYROSINE KINASE, KDR, ANGIOGENESIS, ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST- VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3t9t:A   (GLU406) to   (SER618)  CRYSTAL STRUCTURE OF BTK MUTANT (F435T,K596R) COMPLEXED WITH IMIDAZO[1,5-A]QUINOXALINE  |   KINASE DOMAIN, ALPHA/BETA, ATP BINDING, PHOSPHORYLATION, INTRACELLULAR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1e1v:A    (SER46) to   (HIS283)  HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR NU2058  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION 
1e1x:A    (SER46) to   (HIS283)  HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR NU6027  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION 
3gop:A   (ASN732) to   (ARG949)  CRYSTAL STRUCTURE OF THE EGF RECEPTOR JUXTAMEMBRANE AND KINASE DOMAINS  |   KINASE, JUXTAMEMBRANE, EGFR, ANTI-ONCOGENE, ATP-BINDING, CELL CYCLE, CELL MEMBRANE, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, ISOPEPTIDE BOND, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3gql:B   (LYS523) to   (THR761)  CRYSTAL STRUCTURE OF ACTIVATED RECEPTOR TYROSINE KINASE IN COMPLEX WITH SUBSTRATES  |   PHOSPHORYLATED KINASE, ACTIVATION, ATP ANALOG, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, DWARFISM, GLYCOPROTEIN, HEPARIN-BINDING, HYPOGONADOTROPIC HYPOGONADISM, IMMUNOGLOBULIN DOMAIN, KALLMANN SYNDROME, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3gql:C   (LYS523) to   (SER762)  CRYSTAL STRUCTURE OF ACTIVATED RECEPTOR TYROSINE KINASE IN COMPLEX WITH SUBSTRATES  |   PHOSPHORYLATED KINASE, ACTIVATION, ATP ANALOG, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, DWARFISM, GLYCOPROTEIN, HEPARIN-BINDING, HYPOGONADOTROPIC HYPOGONADISM, IMMUNOGLOBULIN DOMAIN, KALLMANN SYNDROME, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1pxj:A    (SER46) to   (HIS283)  HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR 4-(2,4-DIMETHYL-THIAZOL-5-YL)-PYRIMIDIN-2-YLAMINE  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, 3D-STRUCTURE. 
1pxk:A    (SER46) to   (HIS283)  HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR N-[4-(2,4-DIMETHYL-THIAZOL-5-YL)PYRIMIDIN-2-YL]- N'-HYDROXYIMINOFORMAMIDE  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, 3D-STRUCTURE. 
1pxo:A    (PRO45) to   (GLN287)  HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR [4-(2-AMINO-4-METHYL-THIAZOL-5-YL)-PYRIMIDIN-2- YL]-(3-NITRO-PHENYL)-AMINE  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, 3D-STRUCTURE. 
2r3h:A    (PRO45) to   (HIS283)  CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE, INHIBITION, CYCLIN-DEPENDENT KINASE, CANCER, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE 
2r3i:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE, INHIBITION, CYCLIN-DEPENDENT KINASE, CANCER, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE 
2r3j:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE, INHIBITION, CYCLIN-DEPENDENT KINASE, CANCER, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE 
2r3l:A    (PRO45) to   (HIS283)  CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE, INHIBITION, CYCLIN-DEPENDENT KINASE, CANCER, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE 
2r3m:A    (SER46) to   (GLN287)  CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE, INHIBITION, CYCLIN-DEPENDENT KINASE, CANCER, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE 
2r3o:A    (SER46) to   (GLN287)  CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE, INHIBITION, CYCLIN-DEPENDENT KINASE, CANCER, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE 
2r3p:A    (SER46) to   (GLN287)  CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE, INHIBITION, CYCLIN-DEPENDENT KINASE, CANCER, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE 
3gt8:A   (ALA731) to   (ARG949)  CRYSTAL STRUCTURE OF THE INACTIVE EGFR KINASE DOMAIN IN COMPLEX WITH AMP-PNP  |   INACTIVE KINASE, DIMER, ALTERNATIVE SPLICING, ANTI-ONCOGENE, ATP-BINDING, CELL CYCLE, CELL MEMBRANE, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, ISOPEPTIDE BOND, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE, UBL CONJUGATION 
3gt8:B   (PRO729) to   (ARG949)  CRYSTAL STRUCTURE OF THE INACTIVE EGFR KINASE DOMAIN IN COMPLEX WITH AMP-PNP  |   INACTIVE KINASE, DIMER, ALTERNATIVE SPLICING, ANTI-ONCOGENE, ATP-BINDING, CELL CYCLE, CELL MEMBRANE, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, ISOPEPTIDE BOND, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE, UBL CONJUGATION 
2r64:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF A 3-AMINOINDAZOLE COMPOUND WITH CDK2  |   PROTEIN KINASE, INHIBITOR, CELL DIVISION, ATP-BINDING, CELL CYCLE, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
1q24:A    (ILE85) to   (ALA298)  PKA DOUBLE MUTANT MODEL OF PKB IN COMPLEX WITH MGATP  |   Q181 SWITCH, MG-ATP BINDING, PKB-MODEL, TRANSFERASE/TRANSFERASE INHIBITOR COMPLEX 
1e9h:A    (PRO45) to   (GLN287)  THR 160 PHOSPHORYLATED CDK2 - HUMAN CYCLIN A3 COMPLEX WITH THE INHIBITOR INDIRUBIN-5-SULPHONATE BOUND  |   CELL CYCLE, COMPLEX (PROTEIN KINASE/CYCLIN), KINASES, INHIBITOR, CYCLIN, COMPLEX, PHOSPHORYLATION 
4jai:A   (VAL174) to   (HIS380)  CRYSTAL STRUCTURE OF AURORA KINASE A IN COMPLEX WITH N-{4-[(6-OXO-5,6- DIHYDROBENZO[C][1,8]NAPHTHYRIDIN-1-YL)AMINO]PHENYL}BENZAMIDE  |   KINASE INHIBITOR COMPLEX, ATP-BINDING, CELL CYCLE,CYTOPLASM, CYTOSKELETON, KINASE, NUCLEOTIDE-BINDING,PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, PROTEIN KINASE-LIKE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ti1:A    (PRO45) to   (GLN287)  CDK2 IN COMPLEX WITH SUNITINIB  |   PROTEIN KINASE, ALLOSTERIC LIGAND, SUNITINIB, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4y93:A   (ALA446) to   (GLU657)  CRYSTAL STRUCTURE OF THE PH-TH-KINASE CONSTRUCT OF BRUTON'S TYROSINE KINASE (BTK)  |   PH-TH, BTK, TYROSINE KINASE 
4y95:A   (GLU445) to   (GLU657)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF BRUTON'S TYROSINE KINASE WITH MUTATIONS IN THE ACTIVATION LOOP  |   BTK, KINASE DOMAIN, TRANSFERASE 
4y95:B   (GLU445) to   (GLU657)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF BRUTON'S TYROSINE KINASE WITH MUTATIONS IN THE ACTIVATION LOOP  |   BTK, KINASE DOMAIN, TRANSFERASE 
4y95:C   (GLU439) to   (GLU657)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF BRUTON'S TYROSINE KINASE WITH MUTATIONS IN THE ACTIVATION LOOP  |   BTK, KINASE DOMAIN, TRANSFERASE 
4y95:D   (GLU445) to   (GLU657)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF BRUTON'S TYROSINE KINASE WITH MUTATIONS IN THE ACTIVATION LOOP  |   BTK, KINASE DOMAIN, TRANSFERASE 
2ds1:A    (SER46) to   (HIS283)  HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE CDK4 INHIBITOR  |   PROTEIN KINASE, CELL CYCLE, INHIBITION, TRANSFERASE 
3tnq:B    (GLN84) to   (ALA298)  STRUCTURE AND ALLOSTERY OF THE PKA RIIB TETRAMERIC HOLOENZYME  |   PKA RIIB TETRAMERIC HOLOENZYME, TRANSFERASE 
3tnw:A    (PRO45) to   (GLN287)  STRUCTURE OF CDK2/CYCLIN A IN COMPLEX WITH CAN508  |   CYCLIN DEPENDENT KINASE, KINASE CYCLIN, PHOSPHOTRANSFERASE, CYCLIN A, PHOSPHORYLATION AT CDK2 THREONINE 160, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ybj:A   (SER303) to   (TYR519)  TYPE II DASATINIB ANALOG CRYSTALLIZED WITH C-SRC KINASE  |   PROTEIN KINASE, INACTIVE CONFORMATION, TRANSFERASE 
4ybj:B   (SER303) to   (TYR519)  TYPE II DASATINIB ANALOG CRYSTALLIZED WITH C-SRC KINASE  |   PROTEIN KINASE, INACTIVE CONFORMATION, TRANSFERASE 
4ybk:A   (PRO304) to   (TYR519)  C-HELIX-OUT DASATINIB ANALOG CRYSTALLIZED WITH C-SRC KINASE  |   PROTEIN KINASE, C-HELIX-OUT, TRANSFERASE 
4yc6:A    (THR47) to   (HIS284)  CDK1/CKS1  |   CDK1, CYCLIN B1, CKS2, CELL CYCLE 
4yc6:C    (THR47) to   (HIS284)  CDK1/CKS1  |   CDK1, CYCLIN B1, CKS2, CELL CYCLE 
4yc6:E    (THR47) to   (HIS284)  CDK1/CKS1  |   CDK1, CYCLIN B1, CKS2, CELL CYCLE 
4yc6:G    (THR47) to   (HIS284)  CDK1/CKS1  |   CDK1, CYCLIN B1, CKS2, CELL CYCLE 
2duv:A    (ILE49) to   (HIS283)  STRUCTURE OF CDK2 WITH A 3-HYDROXYCHROMONES  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE, CELL DIVISION, TRANSFERASE 
3tt0:A   (THR521) to   (LEU760)  CO-STRUCTURE OF FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN WITH 3-(2,6-DICHLORO-3,5-DIMETHOXY-PHENYL)-1-{6-[4-(4-ETHYL-PIPERAZIN-1- YL)-PHENYLAMINO]-PYRIMIDIN-4-YL}-1-METHYL-UREA (BGJ398)  |   KINASE DOMAIN, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2rfe:A   (ALA731) to   (ASP950)  CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN THE EGFR KINASE DOMAIN AND A MIG6 PEPTIDE  |   KINASE DOMAIN, INHIBITION, DIMER, PEPTIDE, ALTERNATIVE SPLICING, ANTI-ONCOGENE, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, UBL CONJUGATION, CYTOPLASM 
2rfe:C   (ASN732) to   (ARG949)  CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN THE EGFR KINASE DOMAIN AND A MIG6 PEPTIDE  |   KINASE DOMAIN, INHIBITION, DIMER, PEPTIDE, ALTERNATIVE SPLICING, ANTI-ONCOGENE, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, UBL CONJUGATION, CYTOPLASM 
2rfe:D   (ASN732) to   (ARG949)  CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN THE EGFR KINASE DOMAIN AND A MIG6 PEPTIDE  |   KINASE DOMAIN, INHIBITION, DIMER, PEPTIDE, ALTERNATIVE SPLICING, ANTI-ONCOGENE, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, UBL CONJUGATION, CYTOPLASM 
3h0y:A   (VAL174) to   (HIS380)  AURORA A IN COMPLEX WITH A BISANILINOPYRIMIDINE  |   PROTEIN:INHIBITOR COMPLEX AURORA-A, CELL CYCLE, SERINE/THREONINE, PROTEIN KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3h10:D   (VAL174) to   (HIS380)  AURORA A INHIBITOR COMPLEX  |   PROTEIN:INHIBITOR COMPLEX AURORA-A, CELL CYCLE, SERINE/THREONINE, PROTEIN KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3tud:A   (ALA412) to   (ASP632)  CRYSTAL STRUCTURE OF SYK KINASE DOMAIN WITH N-(4-METHYL-3-(8-METHYL-7- OXO-2-(PHENYLAMINO)-7,8-DIHYDROPYRIDO[2,3-D]PYRIMIDIN-6-YL)PHENYL)-3- (TRIFLUOROMETHYL)BENZAMIDE  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3tuc:A   (LEU413) to   (VAL633)  CRYSTAL STRUCTURE OF SYK KINASE DOMAIN WITH 1-BENZYL-N-(5-(6,7- DIMETHOXYQUINOLIN-4-YLOXY)PYRIDIN-2-YL)-2-OXO-1,2-DIHYDROPYRIDINE-3- CARBOXAMIDE  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3h3c:A   (THR464) to   (GLU692)  CRYSTAL STRUCTURE OF PYK2 IN COMPLEX WITH SULFOXIMINE- SUBSTITUTED TRIFLUOROMETHYLPYRIMIDINE ANALOG  |   PYK2, KINASE, ALTERNATIVE SPLICING, ATP-BINDING, CELL MEMBRANE, CYTOPLASM, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TYROSINE-PROTEIN KINASE 
2src:A   (SER303) to   (TYR519)  CRYSTAL STRUCTURE OF HUMAN TYROSINE-PROTEIN KINASE C-SRC, IN COMPLEX WITH AMP-PNP  |   SRC, TYROSINE-PROTEIN KINASE, PHOSPHORYLATION, SH2, SH3, PHOSPHOTYROSINE, PROTO-ONCOGENE, PHOSPHOTRANSFERASE 
4yhf:A   (ALA446) to   (GLU658)  BRUTON'S TYROSINE KINASE IN COMPLEX WITH A T-BUTYL CYANOACRYLAMIDE INHIBITOR  |   COVALENT INHIBITOR, CYANOACRYLAMIDE, CYSTEINE, TRANSFERASE 
4yhf:B   (GLU439) to   (GLU658)  BRUTON'S TYROSINE KINASE IN COMPLEX WITH A T-BUTYL CYANOACRYLAMIDE INHIBITOR  |   COVALENT INHIBITOR, CYANOACRYLAMIDE, CYSTEINE, TRANSFERASE 
3tz7:A   (SER303) to   (TYR519)  KINASE DOMAIN OF CSRC IN COMPLEX WITH RL103  |   TYPE II, ALLOSTERIC, DFG-OUT, DRUG RESISTANCE MUTATIONS, TYROSIN- PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3tz8:A   (SER303) to   (TYR519)  KINASE DOMAIN OF CSRC IN COMPLEX WITH RL104  |   TYPE II, ALLOSTERIC, DFG-OUT, DRUG RESISTANCE MUTATIONS, TYROSIN- PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3tz8:B   (PRO304) to   (TYR519)  KINASE DOMAIN OF CSRC IN COMPLEX WITH RL104  |   TYPE II, ALLOSTERIC, DFG-OUT, DRUG RESISTANCE MUTATIONS, TYROSIN- PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3tz9:A   (PRO304) to   (TYR519)  KINASE DOMAIN OF CSRC IN COMPLEX WITH RL130  |   TYPE II, ALLOSTERIC, DFG-OUT, DRUG RESISTANCE MUTATIONS, TYROSIN- PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3tz9:B   (SER303) to   (TYR519)  KINASE DOMAIN OF CSRC IN COMPLEX WITH RL130  |   TYPE II, ALLOSTERIC, DFG-OUT, DRUG RESISTANCE MUTATIONS, TYROSIN- PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ha8:A    (SER61) to   (LEU262)  THE COMPLEX STRUCTURE OF THE MAP KINASE P38/COMPOUND 14B  |   TRANSFERASE, INHIBITOR, MAP KINASE, SERINE/ THREONINE-PROTEIN KINASE, P38, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE 
2eb3:A   (LYS754) to   (ARG973)  CRYSTAL STRUCTURE OF MUTATED EGFR KINASE DOMAIN (L858R) IN COMPLEX WITH AMPPNP  |   KINASE, TYROSINE-PROTEIN KINASE, RECEPTOR, TRANSFERASE, PHOSPHORYLATION, ATP-BINDING, DISEASE MUTATION, TRANSMEMBRANE, CELL CYCLE, EC 2.7.10.1, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI 
3u51:A   (PRO304) to   (TYR519)  SRC IN COMPLEX WITH DNA-TEMPLATED MACROCYCLIC INHIBITOR MC1  |   PROTEIN KINASE, SRC-LIKE INACTIVE CONFORMATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3u51:B   (PRO304) to   (TYR519)  SRC IN COMPLEX WITH DNA-TEMPLATED MACROCYCLIC INHIBITOR MC1  |   PROTEIN KINASE, SRC-LIKE INACTIVE CONFORMATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
2uvx:A    (ILE85) to   (ALA298)  STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH 7-AZAINDOLE  |   TRANSFERASE/INHIBITOR, CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE/INHIBITOR COMPLEX, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP- BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION 
2uvy:A    (ILE85) to   (ALA298)  STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH METHYL-(4-(9H- PURIN-6-YL)-BENZYL)-AMINE  |   TRANSFERASE/INHIBITOR, CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION, TRANSFERASE/INHIBITOR COMPLEX 
2uvz:A    (ILE85) to   (ALA298)  STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH C-PHENYL-C-(4-( 9H-PURIN-6-YL)-PHENYL)-METHYLAMINE  |   TRANSFERASE/INHIBITOR, CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION, TRANSFERASE/INHIBITOR COMPLEX 
1r0p:A  (ILE1118) to  (PHE1344)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF THE HEPATOCYTE GROWTH FACTOR RECEPTOR C-MET IN COMPLEX WITH THE MICROBIAL ALKALOID K-252A  |   RECEPTOR TYROSINE KINASE, SIGNAL TRANSDUCTION, GRB2, SHC, TRANSFERASE 
2uw4:A    (ILE85) to   (HIS294)  STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH 2-(4-(5-METHYL- 1H-PYRAZOL-4-YL)-PHENYL)-ETHYLAMINE  |   CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION 
2uw5:A    (ILE85) to   (ALA298)  STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH  (R)-2-(4- CHLORO-PHENYL)-2-(4-1H-PYRAZOL-4-YL)-PHENYL)-ETHYLAMINE  |   TRANSFERASE/INHIBITOR, CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION, TRANSFERASE/INHIBITOR COMPLEX 
3u6i:A  (ILE1118) to  (PHE1344)  CRYSTAL STRUCTURE OF C-MET IN COMPLEX WITH PYRAZOLONE INHIBITOR 58A  |   KINASE DOMAIN, PHOSPHOTRANSFERASE, CANCER, HEPATOCYTE GROWTH FACTOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3u6j:A   (HIS876) to  (ARG1172)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A PYRAZOLONE INHIBITOR  |   KDR, FLK-1, ANGIOGENESIS, PHOSPHOTRANSFERASE, CANCER, VASCULAR ENDOTHELIAL GROWTH FACTOR, TRANSFERASE/TRANSFERASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4jxf:A    (MET53) to   (HIS262)  CRYSTAL STRUCTURE OF PLK4 KINASE WITH AN INHIBITOR: 400631 ((1R,2S)-2- {3-[(E)-2-{4-[(DIMETHYLAMINO)METHYL]PHENYL}ETHENYL]-2H-INDAZOL-6-YL}- 5'-METHOXYSPIRO[CYCLOPROPANE-1,3'-INDOL]-2'(1'H)-ONE)  |   SERINE/THREONINE KINASE, POLO-LIKE KINASE 4, INHIBITOR, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2uzb:C    (PRO45) to   (GLN287)  CRYSTAL STRUCTURE OF HUMAN CDK2 COMPLEXED WITH A THIAZOLIDINONE INHIBITOR  |   TRANSFERASE, ATP-BINDING, PHOSPHORYLATION, CDK2, KINASE, CYCLIN, MITOSIS, CELL CYCLE, CELL DIVISION, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, THIAZOLIDINONE LIGAND 
2uzl:C    (PRO45) to   (GLN287)  CRYSTAL STRUCTURE OF HUMAN CDK2 COMPLEXED WITH A THIAZOLIDINONE INHIBITOR  |   TRANSFERASE, ATP-BINDING, PHOSPHORYLATION, CDK2, KINASE, CYCLIN, MITOSIS, CELL CYCLE, CELL DIVISION, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, THIAZOLIDINONE LIGAND 
2uzn:A    (THR47) to   (GLN287)  CRYSTAL STRUCTURE OF HUMAN CDK2 COMPLEXED WITH A THIAZOLIDINONE INHIBITOR  |   TRANSFERASE, ATP-BINDING, PHOSPHORYLATION, CDK2, KINASE, CYCLIN, MITOSIS, CELL CYCLE, CELL DIVISION, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, THIAZOLIDINONE LIGAND 
1fgi:A   (GLU522) to   (THR761)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF FIBROBLAST GROWTH FACTOR RECEPTOR 1 IN COMPLEX WITH SU5402 INHIBITOR  |   PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE, ATP- BINDING, PHOSPHORYLATION, INHIBITOR 
1fgi:B   (GLU522) to   (THR761)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF FIBROBLAST GROWTH FACTOR RECEPTOR 1 IN COMPLEX WITH SU5402 INHIBITOR  |   PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE, ATP- BINDING, PHOSPHORYLATION, INHIBITOR 
1fgk:A   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF FIBROBLAST GROWTH FACTOR RECEPTOR 1  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, RECEPTOR, PHOSPHOTRANSFERASE 
1fgk:B   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF FIBROBLAST GROWTH FACTOR RECEPTOR 1  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, RECEPTOR, PHOSPHOTRANSFERASE 
3uc4:B    (ARG64) to   (HIS274)  THE CRYSTAL STRUCTURE OF SNF1-RELATED KINASE 2.6  |   SNRK2.6, KINASE, ABA SIGNALING, TRANSFERASE 
1r78:A    (ALA48) to   (GLN287)  CDK2 COMPLEX WITH A 4-ALKYNYL OXINDOLE INHIBITOR  |   CYCLIN DEPENDENT KINASE, SERINE/THREONINE PROTEIN KINASE, OXINDOLE, TRANSFERASE 
2etm:A   (GLN470) to   (GLN686)  CRYSTAL STRUCTURE OF FOCAL ADHESION KINASE DOMAIN COMPLEXED WITH 7H-PYRROLO [2,3-D] PYRIMIDINE DERIVATIVE  |   KINASE CATALYTIC DOMAIN, TRANSFERASE 
2etm:B   (LEU469) to   (GLU689)  CRYSTAL STRUCTURE OF FOCAL ADHESION KINASE DOMAIN COMPLEXED WITH 7H-PYRROLO [2,3-D] PYRIMIDINE DERIVATIVE  |   KINASE CATALYTIC DOMAIN, TRANSFERASE 
1fmk:A   (GLU305) to   (TYR519)  CRYSTAL STRUCTURE OF HUMAN TYROSINE-PROTEIN KINASE C-SRC  |   SRC, TYROSINE KINASE, PHOSPHORYLATION, SH2, SH3, PHOSPHOTYROSINE, PROTO-ONCOGENE, PHOSPHOTRANSFERASE 
4k8a:A   (SER461) to   (GLU683)  FRAGMENT-BASED DISCOVERY OF FOCAL ADHESION KINASE INHIBITORS  |   TYROSINE PROTEIN KINASE, TRANSFERASE, ATP BINDING, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4k8a:B   (LEU469) to   (GLU682)  FRAGMENT-BASED DISCOVERY OF FOCAL ADHESION KINASE INHIBITORS  |   TYROSINE PROTEIN KINASE, TRANSFERASE, ATP BINDING, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
1fvt:A    (THR47) to   (GLN287)  THE STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 (CDK2) IN COMPLEX WITH AN OXINDOLE INHIBITOR  |   CYCLIN-DEPENDENT KINASE, OXINDOLE, TRANSFERASE, CELL CYCLE 
4kab:A   (ASP462) to   (GLN686)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH 3-METHYL-1,4- DIHYDRO-PYRAZOLO[4,5-C]PYRAZOLE  |   TYROSINE PROTEIN KINASE, TRANSFERASE, ATP BINDING, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4kab:B   (LEU469) to   (GLU682)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH 3-METHYL-1,4- DIHYDRO-PYRAZOLO[4,5-C]PYRAZOLE  |   TYROSINE PROTEIN KINASE, TRANSFERASE, ATP BINDING, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4kao:A   (LEU469) to   (GLN686)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH 1-(5-TERT- BUTYL-2-P-TOLYL-2H-PYRAZOL-3-YL)-3-(4-PYRIDIN-3- YL-PHENYL)-UREA  |   TYROSINE PROTEIN KINASE, TRANSFERASE,ATP BINDING, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4kao:B   (ASP462) to   (GLN686)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH 1-(5-TERT- BUTYL-2-P-TOLYL-2H-PYRAZOL-3-YL)-3-(4-PYRIDIN-3- YL-PHENYL)-UREA  |   TYROSINE PROTEIN KINASE, TRANSFERASE,ATP BINDING, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4yzb:B    (GLN66) to   (HIS282)  CDPK1 FROM EIMERIA TENELLA IN COMPLEX WITH INHIBITOR UW1521  |   SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4yzm:A  (THR1066) to  (LEU1292)  HUMANIZED ROCO4 BOUND TO LRRK2-IN1  |   ROCO-PROTEIN, KINASE, LRRK2, INHIBITOR, TRANSFERASE 
4yzm:B  (GLU1067) to  (LEU1292)  HUMANIZED ROCO4 BOUND TO LRRK2-IN1  |   ROCO-PROTEIN, KINASE, LRRK2, INHIBITOR, TRANSFERASE 
2f7z:E    (GLN84) to   (HIS294)  PROTEIN KINASE A BOUND TO (R)-1-(1H-INDOL-3-YLMETHYL)-2-(2- PYRIDIN-4-YL-[1,7]NAPHTYRIDIN-5-YLOXY)-EHYLAMINE  |   PROTEIN KINASE A, AKT INHIBITORS, TRANSFERASE 
3unj:A    (ALA48) to   (GLN287)  CDK2 IN COMPLEX WITH INHIBITOR YL1-038-31  |   PROTEIN KINASE, ALLOSTERIC LIGAND, ANS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2fgi:A   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF FGF RECEPTOR 1 IN COMPLEX WITH INHIBITOR PD173074  |   PROTEIN KINASE, TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, INHIBITOR, TRANSFERASE 
2fgi:B   (THR521) to   (THR761)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF FGF RECEPTOR 1 IN COMPLEX WITH INHIBITOR PD173074  |   PROTEIN KINASE, TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, INHIBITOR, TRANSFERASE 
3uqf:A   (SER303) to   (TYR519)  C-SRC KINASE DOMAIN IN COMPLEX WITH BKI RM-1-89  |   TYROSINE PROTEIN KINASE, ATP-BINDING, KINASE DOMAIN, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3uqf:B   (PRO304) to   (TYR519)  C-SRC KINASE DOMAIN IN COMPLEX WITH BKI RM-1-89  |   TYROSINE PROTEIN KINASE, ATP-BINDING, KINASE DOMAIN, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4kio:B   (ASP402) to   (SER618)  KINASE DOMAIN MUTANT OF HUMAN ITK IN COMPLEX WITH A COVALENTLY-BINDING INHIBITOR  |   KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4kio:C   (GLU401) to   (ALA616)  KINASE DOMAIN MUTANT OF HUMAN ITK IN COMPLEX WITH A COVALENTLY-BINDING INHIBITOR  |   KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4kio:D   (GLU401) to   (SER618)  KINASE DOMAIN MUTANT OF HUMAN ITK IN COMPLEX WITH A COVALENTLY-BINDING INHIBITOR  |   KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4z83:E    (ILE85) to   (HIS294)  PKAB3 IN COMPLEX WITH PYRROLIDINE INHIBITOR 47A  |   INHIBITOR, PROTEIN KINASE, STRUCTURE-GUIDED, TRANSFERASE 
3huc:A    (SER61) to   (LEU262)  HUMAN P38 MAP KINASE IN COMPLEX WITH RL40  |   DFG-OUT, GLYCINE-RICH LOOP, ALTERNATIVE SPLICING, ATP-BINDING, CYTOPLASM, KINASE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3hv3:A    (SER61) to   (LEU262)  HUMAN P38 MAP KINASE IN COMPLEX WITH RL49  |   DFG-OUT, TYPE II, RL49, QUINOLINE-PYRAZOLOUREA, HYBRID, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3hv4:B    (SER61) to   (SER261)  HUMAN P38 MAP KINASE IN COMPLEX WITH RL51  |   DFG-OUT, TYPE II, RL51, QUINOLINE-PYRAZOLOUREA, HYBRID, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3hv5:A    (SER61) to   (GLN260)  HUMAN P38 MAP KINASE IN COMPLEX WITH RL24  |   DFG-OUT, TYPE II, RL24, QUINOLINE-PYRAZOLOUREA, HYBRID, ALTERNATIVE SPLICING, ATP-BINDING, CYTOPLASM, KINASE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
1gih:A    (PRO45) to   (GLN287)  HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE CDK4 INHIBITOR  |   PROTEIN KINASE, CELL CYCLE, INHIBITION, TRANSFERASE 
1gij:A    (ALA48) to   (GLN287)  HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE CDK4 INHIBITOR  |   PROTEIN KINASE, CELL CYCLE, INHIBITION, TRANSFERASE 
4knb:D  (ILE1118) to  (ARG1336)  C-MET IN COMPLEX WITH OSI LIGAND  |   PROTEIN KINASE, TRANSFERASE 
3v5j:A   (SER399) to   (SER618)  CRYSTAL STRUCTURE OF INTERLEUKIN-2 INDUCIBLE T-CELL KINASE ITK CATALYTIC DOMAIN WITH THIENOPYRAZOLYLINDOLE INHIBITOR 090  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3v5j:B   (SER399) to   (SER618)  CRYSTAL STRUCTURE OF INTERLEUKIN-2 INDUCIBLE T-CELL KINASE ITK CATALYTIC DOMAIN WITH THIENOPYRAZOLYLINDOLE INHIBITOR 090  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2vny:A    (ILE85) to   (HIS294)  STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH (1-(9H-PURIN-6- YL)PIPERIDIN-4-YL)AMINE  |   TRANSFERASE, LIPOPROTEIN, ATP-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, CAMP, KINASE, NUCLEUS, MYRISTATE, CYTOPLASM 
3v8t:A   (SER399) to   (SER618)  CRYSTAL STRUCTURE OF INTERLEUKIN-2 INDUCIBLE T-CELL KINASE ITK CATALYTIC DOMAIN WITH THIENOPYRAZOLYLINDOLE INHIBITOR 477  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3v8w:A   (SER399) to   (SER618)  CRYSTAL STRUCTURE OF INTERLEUKIN-2 INDUCIBLE T-CELL KINASE ITK CATALYTIC DOMAIN WITH THIENOPYRAZOLYLINDOLE INHIBITOR 469  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3v8w:B   (SER399) to   (SER618)  CRYSTAL STRUCTURE OF INTERLEUKIN-2 INDUCIBLE T-CELL KINASE ITK CATALYTIC DOMAIN WITH THIENOPYRAZOLYLINDOLE INHIBITOR 469  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1snu:A   (SER399) to   (GLU617)  CRYSTAL STRUCTURE OF THE UNPHOSPHORYLATED INTERLEUKIN-2 TYROSINE KINASE CATALYTIC DOMAIN  |   PROTEIN KINASE, IMMUNOLOGY, TRANSFERASE 
2vtj:A    (SER46) to   (GLN287)  IDENTIFICATION OF N-(4-PIPERIDINYL)-4-(2,6- DICHLOROBENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXAMIDE (AT7519), A NOVEL CYCLIN DEPENDENT KINASE INHIBITOR USING FRAGMENT- BASED X-RAY CRYSTALLOGRAPHY AND STRUCTURE BASED DRUG DESIGN.  |   TRANSFERASE, MITOSIS, CELL CYCLE, SERINE/THREONINE PROTEIN KINASE 
2vtl:A    (PRO45) to   (GLN287)  IDENTIFICATION OF N-(4-PIPERIDINYL)-4-(2,6- DICHLOROBENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXAMIDE (AT7519), A NOVEL CYCLIN DEPENDENT KINASE INHIBITOR USING FRAGMENT- BASED X-RAY CRYSTALLOGRAPHY AND STRUCTURE BASED DRUG DESIGN.  |   TRANSFERASE, MITOSIS, CELL CYCLE, SERINE/THREONINE PROTEIN KINASE 
2vtm:A    (PRO45) to   (GLN287)  IDENTIFICATION OF N-(4-PIPERIDINYL)-4-(2,6- DICHLOROBENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXAMIDE (AT7519), A NOVEL CYCLIN DEPENDENT KINASE INHIBITOR USING FRAGMENT- BASED X-RAY CRYSTALLOGRAPHY AND STRUCTURE BASED DRUG DESIGN.  |   TRANSFERASE, MITOSIS, CELL CYCLE, SERINE/THREONINE PROTEIN KINASE 
2vtn:A    (SER46) to   (GLN287)  IDENTIFICATION OF N-(4-PIPERIDINYL)-4-(2,6- DICHLOROBENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXAMIDE (AT7519), A NOVEL CYCLIN DEPENDENT KINASE INHIBITOR USING FRAGMENT- BASED X-RAY CRYSTALLOGRAPHY AND STRUCTURE BASED DRUG DESIGN.  |   TRANSFERASE, MITOSIS, CELL CYCLE, SERINE/THREONINE PROTEIN KINASE 
2vts:A    (SER46) to   (GLN287)  IDENTIFICATION OF N-(4-PIPERIDINYL)-4-(2,6- DICHLOROBENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXAMIDE (AT7519), A NOVEL CYCLIN DEPENDENT KINASE INHIBITOR USING FRAGMENT- BASED X-RAY CRYSTALLOGRAPHY AND STRUCTURE BASED DRUG DESIGN.  |   TRANSFERASE, MITOSIS, CELL CYCLE, SERINE/THREONINE PROTEIN KINASE 
2vtt:A    (THR47) to   (GLN287)  IDENTIFICATION OF N-(4-PIPERIDINYL)-4-(2,6- DICHLOROBENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXAMIDE (AT7519), A NOVEL CYCLIN DEPENDENT KINASE INHIBITOR USING FRAGMENT- BASED X-RAY CRYSTALLOGRAPHY AND STRUCTURE BASED DRUG DESIGN.  |   TRANSFERASE, MITOSIS, CELL CYCLE, SERINE/THREONINE PROTEIN KINASE 
2vu3:A    (THR47) to   (GLN287)  IDENTIFICATION OF N-(4-PIPERIDINYL)-4-(2,6- DICHLOROBENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXAMIDE (AT7519), A NOVEL CYCLIN DEPENDENT KINASE INHIBITOR USING FRAGMENT- BASED X-RAY CRYSTALLOGRAPHY AND STRUCTURE BASED DRUG DESIGN.  |   TRANSFERASE, MITOSIS, CELL CYCLE, SERINE/THREONINE PROTEIN KINASE 
2g9x:A    (PRO45) to   (GLN287)  STRUCTURE OF THR 160 PHOSPHORYLATED CDK2/CYCLIN A IN COMPLEX WITH THE INHIBITOR NU6271  |   TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, ATP-BINDING, CELL CYCLE, PHOSPHORYLATION, TRANSFERASE-CELL CYCLE COMPLEX 
2vwu:A   (THR654) to   (ILE878)  EPHB4 KINASE DOMAIN INHIBITOR COMPLEX  |   TYROSINE-PROTEIN KINASE, RECEPTOR TYROSINE KINASE, KINASE, MUTANT, MEMBRANE, RECEPTOR, TRANSFERASE, ATP-BINDING, POLYMORPHISM, GLYCOPROTEIN, TRANSMEMBRANE, PHOSPHOPROTEIN, UNPHOSPHORYLATED, NUCLEOTIDE-BINDING 
2vwv:A   (THR654) to   (ASN880)  EPHB4 KINASE DOMAIN INHIBITOR COMPLEX  |   TYROSINE-PROTEIN KINASE, RECEPTOR TYROSINE KINASE, KINASE, MUTANT, MEMBRANE, RECEPTOR, TRANSFERASE, ATP-BINDING, POLYMORPHISM, GLYCOPROTEIN, TRANSMEMBRANE, PHOSPHOPROTEIN, UNPHOSPHORYLATED, NUCLEOTIDE-BINDING 
2vww:A   (THR654) to   (ASN880)  EPHB4 KINASE DOMAIN INHIBITOR COMPLEX  |   TYROSINE-PROTEIN KINASE, RECEPTOR TYROSINE KINASE, KINASE, MUTANT, MEMBRANE, RECEPTOR, TRANSFERASE, ATP-BINDING, POLYMORPHISM, GLYCOPROTEIN, TRANSMEMBRANE, PHOSPHOPROTEIN, UNPHOSPHORYLATED, NUCLEOTIDE-BINDING 
2vwx:A   (SER663) to   (ILE878)  EPHB4 KINASE DOMAIN INHIBITOR COMPLEX  |   TYROSINE-PROTEIN KINASE, RECEPTOR TYROSINE KINASE, KINASE, MUTANT, MEMBRANE, RECEPTOR, TRANSFERASE, ATP-BINDING, POLYMORPHISM, GLYCOPROTEIN, TRANSMEMBRANE, PHOSPHOPROTEIN, UNPHOSPHORYLATED, NUCLEOTIDE-BINDING 
2vwy:A   (THR654) to   (ASN880)  EPHB4 KINASE DOMAIN INHIBITOR COMPLEX  |   TYROSINE-PROTEIN KINASE, RECEPTOR TYROSINE KINASE, KINASE, MUTANT, MEMBRANE, RECEPTOR, TRANSFERASE, ATP-BINDING, POLYMORPHISM, GLYCOPROTEIN, TRANSMEMBRANE, PHOSPHOPROTEIN, UNPHOSPHORYLATED, NUCLEOTIDE-BINDING 
2vwz:A   (THR654) to   (ASN880)  EPHB4 KINASE DOMAIN INHIBITOR COMPLEX  |   TYROSINE-PROTEIN KINASE, RECEPTOR TYROSINE KINASE, KINASE, MUTANT, MEMBRANE, RECEPTOR, TRANSFERASE, ATP-BINDING, POLYMORPHISM, GLYCOPROTEIN, TRANSMEMBRANE, PHOSPHOPROTEIN, UNPHOSPHORYLATED, NUCLEOTIDE-BINDING 
2vx0:A   (SER663) to   (ASN880)  EPHB4 KINASE DOMAIN INHIBITOR COMPLEX MUTANT, MEMBRANE, TRANSFERASE, ATP-BINDING, POLYMORPHISM, GLYCOPROTEIN, TRANSMEMBRANE, PHOSPHOPROTEIN, UNPHOSPHORYLATED, NUCLEOTIDE-BINDING  |    
2vx1:A   (SER663) to   (ASN880)  EPHB4 KINASE DOMAIN INHIBITOR COMPLEX  |   TYROSINE-PROTEIN KINASE, RECEPTOR TYROSINE KINASE, KINASE, MUTANT, MEMBRANE, RECEPTOR, TRANSFERASE, ATP-BINDING, POLYMORPHISM, GLYCOPROTEIN, TRANSMEMBRANE, PHOSPHOPROTEIN, UNPHOSPHORYLATED, NUCLEOTIDE-BINDING 
1svg:A    (ILE85) to   (HIS294)  CRYSTAL STRUCTURE OF PROTEIN KINASE A IN COMPLEX WITH AZEPANE DERIVATIVE 4  |   KINASE-INHIBITOR-COMPLEX, SERINE/THREONINE-PROTEIN KINASE, BALANOL DERIVATIVE, TRANSFERASE 
1h00:A    (SER46) to   (HIS283)  CDK2 IN COMPLEX WITH A DISUBSTITUTED 4, 6-BIS ANILINO PYRIMIDINE CDK4 INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, MITOSIS, TRANSFERASE 
1h01:A    (SER46) to   (HIS283)  CDK2 IN COMPLEX WITH A DISUBSTITUTED 2, 4-BIS ANILINO PYRIMIDINE CDK4 INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, MITOSIS, TRANSFERASE 
1h07:A    (SER46) to   (HIS283)  CDK2 IN COMPLEX WITH A DISUBSTITUTED 4, 6-BIS ANILINO PYRIMIDINE CDK4 INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, MITOSIS, TRANSFERASE 
1h08:A    (SER46) to   (GLN287)  CDK2 IN COMPLEX WITH A DISUBSTITUTED 2, 4-BIS ANILINO PYRIMIDINE CDK4 INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, MITOSIS, TRANSFERASE 
1h0v:A    (SER46) to   (HIS283)  HUMAN CYCLIN DEPENDENT PROTEIN KINASE 2 IN COMPLEX WITH THE INHIBITOR 2-AMINO-6-[(R)-PYRROLIDINO-5'-YL]METHOXYPURINE  |   TRANSFERASE, DRUG METABOLISM, MYCOBACTERIA, ISONIAZID, ARYLAMINE N-ACETYLTRANSFERASE, NAT, SERINE/THREONINE - PROTEIN KINASE, ATP-BINDING, CELL CYCLE, CELL DIVISION, MITOSIS 
1h0w:A    (SER46) to   (GLN287)  HUMAN CYCLIN DEPENDENT PROTEIN KINASE 2 IN COMPLEX WITH THE INHIBITOR 2-AMINO-6-[CYCLOHEX-3-ENYL]METHOXYPURINE  |   TRANSFERASE, PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION 
1h1p:C    (PRO45) to   (GLN287)  STRUCTURE OF HUMAN THR160-PHOSPHO CDK2/CYCLIN A COMPLEXED WITH THE INHIBITOR NU2058  |   KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP- BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, PHOSPHORYLATION 
3vhe:A   (HIS876) to  (ASN1167)  CRYSTAL STRUCTURE OF HUMAN VEGFR2 KINASE DOMAIN WITH A NOVEL PYRROLOPYRIMIDINE INHIBITOR.  |   KINASE DOMAIN, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1h1q:A    (PRO45) to   (GLN287)  STRUCTURE OF HUMAN THR160-PHOSPHO CDK2/CYCLIN A COMPLEXED WITH THE INHIBITOR NU6094  |   KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP- BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, PHOSPHORYLATION 
1h1r:A    (PRO45) to   (GLN287)  STRUCTURE OF HUMAN THR160-PHOSPHO CDK2/CYCLIN A COMPLEXED WITH THE INHIBITOR NU6086  |   KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP- BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, PHOSPHORYLATION 
3vhk:A   (HIS876) to  (ALA1168)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A BACK POCKET BINDER  |   VEGFR2, KINASE DOMAIN, COMPLEX, TRANSFERASE 
1h1s:C    (PRO45) to   (GLN287)  STRUCTURE OF HUMAN THR160-PHOSPHO CDK2/CYCLIN A COMPLEXED WITH THE INHIBITOR NU6102  |   KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP- BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, PHOSPHORYLATION 
1h25:A    (PRO45) to   (GLN287)  CDK2/CYCLIN A IN COMPLEX WITH AN 11-RESIDUE RECRUITMENT PEPTIDE FROM RETINOBLASTOMA-ASSOCIATED PROTEIN  |   TRANSFERASE, CELL CYCLE, PROTEIN KINASE, CYCLIN, CDK2, RECRUITMENT, PEPTIDE SPECIFICITY 
1h28:A    (PRO45) to   (GLN287)  CDK2/CYCLIN A IN COMPLEX WITH AN 11-RESIDUE RECRUITMENT PEPTIDE FROM P107  |   CELL CYCLE, PROTEIN KINASE, CYCLIN, CDK2, RECRUITMENT, PEPTIDE SPECIFICITY, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, CELL DIVISION, MITOSIS, PHOSPHORYLATION, CELL CYCLE-TRANSFERASE SUBSTRATE, CELL CYCLE-TRANSFERASE SUBSTRATE COMPLEX 
1h28:C    (SER46) to   (GLN287)  CDK2/CYCLIN A IN COMPLEX WITH AN 11-RESIDUE RECRUITMENT PEPTIDE FROM P107  |   CELL CYCLE, PROTEIN KINASE, CYCLIN, CDK2, RECRUITMENT, PEPTIDE SPECIFICITY, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, CELL DIVISION, MITOSIS, PHOSPHORYLATION, CELL CYCLE-TRANSFERASE SUBSTRATE, CELL CYCLE-TRANSFERASE SUBSTRATE COMPLEX 
3vid:A   (HIS876) to  (ASN1167)  CRYSTAL STRUCTURE OF HUMAN VEGFR2 KINASE DOMAIN WITH COMPOUND A.  |   KINASE, TRANSFERASE, PHOSPHORYLATION 
2w05:A    (ALA48) to   (GLN287)  STRUCTURE OF CDK2 IN COMPLEX WITH AN IMIDAZOLYL PYRIMIDINE, COMPOUND 5B  |   KINASE, MITOSIS, CELL CYCLE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, POLYMORPHISM, CELL DIVISION, PHOSPHOPROTEIN, PHOSPHORYLATION, NUCLEOTIDE-BINDING 
2w06:A    (SER46) to   (HIS283)  STRUCTURE OF CDK2 IN COMPLEX WITH AN IMIDAZOLYL PYRIMIDINE, COMPOUND 5C  |   KINASE, MITOSIS, CELL CYCLE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, POLYMORPHISM, CELL DIVISION, PHOSPHOPROTEIN, PHOSPHORYLATION, NUCLEOTIDE-BINDING 
2gnf:A    (ILE85) to   (ALA298)  PROTEIN KINASE A FIVEFOLD MUTANT MODEL OF RHO-KINASE WITH Y- 27632  |   PKA, RHO-KINASE, SURROGATE, Y-27632, TRANSFERASE/TRANSFERASE INHIBITOR COMPLEX 
2gnh:A    (ILE85) to   (ALA298)  PKA FIVE FOLD MUTANT MODEL OF RHO-KINASE WITH H1152P  |   PKA, SURROGATE, RHO-KINASE, H1152P, INHIBITOR, TRANSFERASE/TRANSFERASE INHIBITOR COMPLEX 
2gnj:A    (ILE85) to   (HIS294)  PKA THREE FOLD MUTANT MODEL OF RHO-KINASE WITH Y-27632  |   PKA, SURROGATE, RHO-KINASE, H1152P, INHIBITOR, TRANSFERASE/TRANSFERASE INHIBITOR COMPLEX 
2w17:A    (THR47) to   (GLN287)  CDK2 IN COMPLEX WITH THE IMIDAZOLE PYRIMIDINE AMIDE, COMPOUND (S)-8B  |   KINASE, MITOSIS, CELL CYCLE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, CELL DIVISION, PHOSPHOPROTEIN, PHOSPHORYLATION, NUCLEOTIDE-BINDING 
2w1h:A    (SER46) to   (GLN287)  FRAGMENT-BASED DISCOVERY OF THE PYRAZOL-4-YL UREA (AT9283), A MULTI-TARGETED KINASE INHIBITOR WITH POTENT AURORA KINASE ACTIVITY  |   STRUCTURE BASED DRUG DESIGN, KINASE, MITOSIS, CELL CYCLE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, POLYMORPHISM, CELL DIVISION, PHOSPHOPROTEIN, FRAGMENT SCREENING, NUCLEOTIDE-BINDING 
3ig7:A    (SER46) to   (HIS283)  NOVEL CDK-5 INHIBITORS - CRYSTAL STRUCTURE OF INHIBITOR EFP WITH CDK-2  |   PROTEIN KINASE, TRANSFERASE,SERINE/THREONINE PROTEIN KINASE, ATP-BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, 4- AMINOIMIDAZOLE, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE 
3igg:A    (SER46) to   (HIS283)  NOVEL CDK-5 INHIBITORS - CRYSTAL STRUCTURE OF INHIBITOR EFQ WITH CDK-2  |   PROTEIN KINASE, TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, INHIBITOR, ATP-BINDING, CELL CYCLE, CELL DIVISION, KINASE, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE 
4l7s:A   (GLU400) to   (SER618)  KINASE DOMAIN MUTANT OF HUMAN ITK IN COMPLEX WITH AN AMINOBENZOTHIAZOLE INHIBITOR  |   KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4l7s:B   (SER399) to   (SER618)  KINASE DOMAIN MUTANT OF HUMAN ITK IN COMPLEX WITH AN AMINOBENZOTHIAZOLE INHIBITOR  |   KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4zsa:A   (THR521) to   (LEU760)  CRYSTAL STRUCTURE OF FGFR1 KINASE DOMAIN IN COMPLEX WITH 7N  |   FGFR1 INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4zsa:B   (THR521) to   (LEU760)  CRYSTAL STRUCTURE OF FGFR1 KINASE DOMAIN IN COMPLEX WITH 7N  |   FGFR1 INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4zse:A   (SER752) to   (ARG973)  CRYSTAL STRUCTURE OF EGFR 696-1022 T790M/V948R, CRYSTAL FORM II  |   EGFR, T790M, V948R, TRANSFERASE 
4zse:C   (SER752) to   (ARG973)  CRYSTAL STRUCTURE OF EGFR 696-1022 T790M/V948R, CRYSTAL FORM II  |   EGFR, T790M, V948R, TRANSFERASE 
4zse:D   (ASN756) to   (ALA972)  CRYSTAL STRUCTURE OF EGFR 696-1022 T790M/V948R, CRYSTAL FORM II  |   EGFR, T790M, V948R, TRANSFERASE 
1hck:A    (SER46) to   (GLN287)  HUMAN CYCLIN-DEPENDENT KINASE 2  |   TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, ATP-BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, PHOSPHORYLATION 
1hcl:A    (SER46) to   (HIS283)  HUMAN CYCLIN-DEPENDENT KINASE 2  |   TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, ATP-BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, PHOSPHORYLATION 
4lgg:B   (SER303) to   (TYR519)  STRUCTURE OF 3MB-PP1 BOUND TO ANALOG-SENSITIVE SRC KINASE  |   KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2h34:A    (THR59) to   (ALA274)  APOENZYME CRYSTAL STRUCTURE OF THE TUBERCULOSIS SERINE/THREONINE KINASE, PKNE  |   APOENZYME, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE 
3vo3:A   (HIS876) to  (ASN1167)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN VEGFR2 WITH IMIDAZO[1, 2-B]PYRIDAZINE DERIVATIVE  |   VEGFR2, KINASE DOMAIN, TYROSIN-PROTEIN KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
2hen:A   (THR668) to   (ASN894)  CRYSTAL STRUCTURE OF THE EPHB2 RECEPTOR KINASE DOMAIN IN COMPLEX WITH ADP  |   EPH KINASE DOMAIN, ACTIVATION, TRANSFERASE 
2hen:B   (THR668) to   (ASN894)  CRYSTAL STRUCTURE OF THE EPHB2 RECEPTOR KINASE DOMAIN IN COMPLEX WITH ADP  |   EPH KINASE DOMAIN, ACTIVATION, TRANSFERASE 
2hen:C   (THR668) to   (ASN894)  CRYSTAL STRUCTURE OF THE EPHB2 RECEPTOR KINASE DOMAIN IN COMPLEX WITH ADP  |   EPH KINASE DOMAIN, ACTIVATION, TRANSFERASE 
2hen:D   (THR668) to   (ASN894)  CRYSTAL STRUCTURE OF THE EPHB2 RECEPTOR KINASE DOMAIN IN COMPLEX WITH ADP  |   EPH KINASE DOMAIN, ACTIVATION, TRANSFERASE 
5a14:A    (ALA48) to   (GLN287)  HUMAN CDK2 WITH TYPE II INHIBITOR  |   TRANSFERASE, CDK2, CYCLIN, KINASE, TYPE II, INHIBITOR 
4lqm:A   (THR751) to   (ARG973)  EGFR L858R IN COMPLEX WITH PD168393  |   EGFR, KINASE, PD168393, 34-JAB, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2wmb:A    (PRO45) to   (GLN287)  STRUCTURAL AND THERMODYNAMIC CONSEQUENCES OF CYCLIZATION OF PEPTIDE LIGANDS FOR THE RECRUITMENT SITE OF CYCLIN A  |   CELL CYCLE, CELL DIVISION, ANTI-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, PHOSPHORYLATION, NUCLEOTIDE-BINDING, TRANSCRIPTION REGULATION, CHROMATIN REGULATOR, RECRUITMENT, TRANSCRIPTION, NUCLEUS, MITOSIS, ATP-BINDING, TRANSFERASE 
3w18:A   (GLU181) to   (HIS380)  STRUCTURE OF AURORA KINASE A COMPLEXED TO BENZOIMIDAZOLE-INDAZOLE INHIBITOR XIII  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3w2s:A   (SER752) to   (ARG973)  EGFR KINASE DOMAIN WITH COMPOUND4  |   ANTI-ONCOGENE, CELL CYCLE, DISEASE MUTATION, KINASE DOMAIN, RECEPTOR, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3w33:A   (ASN756) to   (ARG973)  EGFR KINASE DOMAIN COMPLEXED WITH COMPOUND 19B  |   ANTI-ONCOGENE, CELL CYCLE, DISEASE MUTATION, KINASE DOMAIN, RECEPTOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2hwp:A   (ALA311) to   (TYR519)  CRYSTAL STRUCTURE OF SRC KINASE DOMAIN IN COMPLEX WITH COVALENT INHIBITOR PD168393  |   KINASE, COVALENT, QUINAZOLINE, MODIFICATION, TRANSFERASE 
5a46:A   (THR521) to   (LEU760)  FGFR1 IN COMPLEX WITH DOVITINIB  |   TRANSFERASE, KINASE 
5a46:B   (GLU522) to   (THR761)  FGFR1 IN COMPLEX WITH DOVITINIB  |   TRANSFERASE, KINASE 
5a4c:A   (THR521) to   (LEU760)  FGFR1 LIGAND COMPLEX  |   TRANSFERASE, KINASE 
5a4c:B   (GLU522) to   (LEU760)  FGFR1 LIGAND COMPLEX  |   TRANSFERASE, KINASE 
4lyn:A    (PRO45) to   (GLN287)  CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 (CDK2-WT) COMPLEX WITH (2S)-N-(5-(((5-TERT-BUTYL-1,3-OXAZOL-2-YL)METHYL)SULFANYL)-1,3- THIAZOL-2-YL)-2-PHENYLPROPANAMIDE  |   KINASE, MITOSIS, CELL CYCLE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2hz0:B   (VAL280) to   (MET496)  ABL KINASE DOMAIN IN COMPLEX WITH NVP-AEG082  |   TYROSINE KINASE, TRANSFERASE 
4m12:A   (ALA407) to   (SER618)  CRYSTAL STRUCTURE OF ITK IN COMPLEX WITH COMPOUND 7 [4- (CARBAMOYLAMINO)-1-(7-ETHOXYNAPHTHALEN-1-YL)-1H-PYRAZOLE-3- CARBOXAMIDE]  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3wbl:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF CDK2 IN COMPLEX WITH PYRAZOLOPYRIMIDINE INHIBITOR  |   BINDING SITES, TUMOR, CYCLIN-DEPENDENT KINASE 2, DRUG DESIGN, MAP KINASE KINASE 2, MK2, PROTEIN KINASE INHIBITORS, PYRAZOLES, PYRIMIDINES, STRUCTURE-ACTIVITY RELATIONSHIP, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
2wzj:C    (SER91) to   (ASP301)  CATALYTIC AND UBA DOMAIN OF KINASE MARK2/(PAR-1) K82R, T208E DOUBLE MUTANT  |   UBA DOMAIN, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, SIGNALING PROTEIN, S/T PROTEIN KINASE, DIFFERENTIATION, DEVELOPMENTAL PROTEIN 
1urw:A    (ALA48) to   (GLN287)  CDK2 IN COMPLEX WITH AN IMIDAZO[1,2-B]PYRIDAZINE  |   SERINE/THREONINE-PROTEIN KINASE, MITOSIS, TRANSFERASE 
3we4:A   (LYS135) to   (HIS349)  CRYSTAL STRUCTURE OF S6K1 KINASE DOMAIN IN COMPLEX WITH A PYRIMIDINE DERIVATIVE PF-4708671 2-{[4-(5-ETHYLPYRIMIDIN-4-YL)PIPERAZIN-1- YL]METHYL}-5-(TRIFLUOROMETHYL)-1H-BENZIMIDAZOLE  |   SERINE/THREONINE PROTEIN KINASE DOMAIN, TRANSFERASE, PHOSPHORYLATION, ATP-BINDING, ZINC-BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4mcv:A   (ALA306) to   (TYR519)  STAR 12 BOUND TO ANALOG-SENSITIVE SRC KINASE  |   KINASE DOMAIN, TYROSINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4mcv:B   (GLU305) to   (TYR519)  STAR 12 BOUND TO ANALOG-SENSITIVE SRC KINASE  |   KINASE DOMAIN, TYROSINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3wf5:A   (THR140) to   (HIS349)  CRYSTAL STRUCTURE OF S6K1 KINASE DOMAIN IN COMPLEX WITH A PYRAZOLOPYRIMIDINE DERIVATIVE 4-[4-(1H-BENZIMIDAZOL-2-YL)PIPERIDIN-1- YL]-1H-PYRAZOLO[3,4-D]PYRIMIDINE  |   SERINE/THREONINE PROTEIN KINASE DOMAIN, TRANSFERASE, PHOSPHORYLATION, ATP-BINDING, ZINC-BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2ijm:A   (LEU469) to   (GLN686)  CRYSTAL STRUCTURE OF FOCAL ADHESION KINASE DOMAIN WITH 2 MOLECULES IN THE ASYMMETRIC UNIT COMPLEXED WITH ADP AND ATP  |   KINASE CATALYTIC DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
2ijm:B   (ASP462) to   (GLU689)  CRYSTAL STRUCTURE OF FOCAL ADHESION KINASE DOMAIN WITH 2 MOLECULES IN THE ASYMMETRIC UNIT COMPLEXED WITH ADP AND ATP  |   KINASE CATALYTIC DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
3wf7:A   (THR137) to   (HIS349)  CRYSTAL STRUCTURE OF S6K1 KINASE DOMAIN IN COMPLEX WITH A PURINE DERIVATIVE 1-(9H-PURIN-6-YL)-N-[3-(TRIFLUOROMETHYL)PHENYL]PIPERIDINE- 4-CARBOXAMIDE  |   SERINE/THREONINE PROTEIN KINASE DOMAIN, TRANSFERASE, PHOSPHORYLATION, ATP-BINDING, ZINC-BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1v1k:A    (THR47) to   (HIS283)  CDK2 IN COMPLEX WITH A DISUBSTITUTED 4, 6-BIS ANILINO PYRIMIDINE CDK4 INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, MITOSIS, TRANSFERASE 
2x9f:A   (THR654) to   (ASN880)  EPHB4 KINASE DOMAIN INHIBITOR COMPLEX  |   TRANSFERASE, ATP-BINDING, GLYCOPROTEIN, TRANSMEMBRANE 
5am6:B   (THR521) to   (LEU760)  NATIVE FGFR1 WITH AN INHIBITOR  |   TRANSFERASE, FGFR, GROWTH FACTOR, CANCER, DOVITINIB, TKI258, KINASE 
2iw6:A    (PRO45) to   (GLN287)  STRUCTURE OF HUMAN THR160-PHOSPHO CDK2-CYCLIN A COMPLEXED WITH A BISANILINOPYRIMIDINE INHIBITOR  |   PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE COMPLEX, KINASE, MITOSIS, CELL CYCLE, TRANSFERASE, ATP-BINDING 
2iw8:C    (PRO45) to   (GLN287)  STRUCTURE OF HUMAN THR160-PHOSPHO CDK2-CYCLIN A F82H-L83V- H84D MUTANT WITH AN O6-CYCLOHEXYLMETHYLGUANINE INHIBITOR  |   PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE COMPLEX, KINASE, MITOSIS, CELL CYCLE, TRANSFERASE 
2iw9:A    (PRO45) to   (GLN287)  STRUCTURE OF HUMAN THR160-PHOSPHO CDK2-CYCLIN A COMPLEXED WITH A BISANILINOPYRIMIDINE INHIBITOR  |   PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE COMPLEX, KINASE, MITOSIS, CELL CYCLE, TRANSFERASE 
2iw9:C    (PRO45) to   (GLN287)  STRUCTURE OF HUMAN THR160-PHOSPHO CDK2-CYCLIN A COMPLEXED WITH A BISANILINOPYRIMIDINE INHIBITOR  |   PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE COMPLEX, KINASE, MITOSIS, CELL CYCLE, TRANSFERASE 
2xb7:A  (SER1157) to  (ASP1389)  STRUCTURE OF HUMAN ANAPLASTIC LYMPHOMA KINASE IN COMPLEX WITH NVP- TAE684  |   ATP-BINDING, RECEPTOR, TRANSFERASE 
5and:A    (PRO45) to   (GLN287)  CRYSTAL STRUCTURE OF CDK2 IN COMPLEX WITH 2-IMIDAZOL-1-YL-1H- BENZIMIDAZOLE PROCESSED WITH THE CRYSTALDIRECT AUTOMATED MOUNTING AND CRYO-COOLING TECHNOLOGY  |   TRANSFERASE, PROTEIN KINASE, INHIBITOR, AUTOMATED CRYSTAL HARVESTING, AUTOMATED CRYO-COOLING, CRYSTALDIRECT 
5ang:A    (SER46) to   (GLN287)  CRYSTAL STRUCTURE OF CDK2 IN COMPLEX WITH 7-HYDROXY-4-( MORPHOLINOMETHYL)CHROMEN-2-ONE PROCESSED WITH THE CRYSTALDIRECT AUTOMATED MOUNTING AND CRYO-COOLING TECHNOLOGY  |   TRANSFERASE, PROTEIN KINASE, INHIBITOR, AUTOMATED CRYSTAL HARVESTING, AUTOMATED CRYO-COOLING, CRYSTALDIRECT 
5ank:A    (SER46) to   (GLN287)  CRYSTAL STRUCTURE OF CDK2 IN COMPLEX WITH 2,4,6-TRIOXO-1- PHENYL-HEXAHYDROPYRIMIDINE-5-CARBOXAMIDE PROCESSED WITH THE CRYSTALDIRECT AUTOMATED MOUNTING AND CRYO-COOLING TECHNOLOGY  |   TRANSFERASE, PROTEIN KINASE, INHIBITOR, AUTOMATED CRYSTAL HARVESTING, AUTOMATED CRYO-COOLING, CRYSTALDIRECT 
5ano:A    (SER46) to   (GLN287)  CRYSTAL STRUCTURE OF CDK2 PROCESSED WITH THE CRYSTALDIRECT AUTOMATED MOUNTING AND CRYO-COOLING TECHNOLOGY  |   TRANSFERASE, PROTEIN KINASE, AUTOMATED CRYSTAL HARVESTING, AUTOMATED CRYO-COOLING, CRYSTALDIRECT 
2j0j:A   (SER461) to   (GLN686)  CRYSTAL STRUCTURE OF A FRAGMENT OF FOCAL ADHESION KINASE CONTAINING THE FERM AND KINASE DOMAINS.  |   CELL MIGRATION, FERM, TRANSFERASE, INTEGRIN SIGNALING 
2j0k:A   (ASP462) to   (GLN686)  CRYSTAL STRUCTURE OF A FRAGMENT OF FOCAL ADHESION KINASE CONTAINING THE FERM AND KINASE DOMAINS.  |   CELL MIGRATION, TRANSFERASE, INTEGRIN SIGNALING 
2j0k:B   (SER461) to   (GLN686)  CRYSTAL STRUCTURE OF A FRAGMENT OF FOCAL ADHESION KINASE CONTAINING THE FERM AND KINASE DOMAINS.  |   CELL MIGRATION, TRANSFERASE, INTEGRIN SIGNALING 
2j0m:B   (ASP462) to   (LYS684)  CRYSTAL STRUCTURE A TWO-CHAIN COMPLEX BETWEEN THE FERM AND KINASE DOMAINS OF FOCAL ADHESION KINASE.  |   FOCAL ADHESION, CELL MIGRATION, PHOSPHORYLATION, FERM, KINASE, TRANSFERASE, ATP-BINDING, INTEGRIN SIGNALING, NUCLEOTIDE-BINDING, TYROSINE-PROTEIN KINASE 
2xk3:A    (THR45) to   (ASN268)  STRUCTURE OF NEK2 BOUND TO AMINOPYRAZINE COMPOUND 35  |   TRANSFERASE, CENTROSOME, MITOSIS 
2xk4:A    (THR45) to   (GLU267)  STRUCTURE OF NEK2 BOUND TO AMINOPYRAZINE COMPOUND 17  |   TRANSFERASE, CENTROSOME, MITOSIS 
2xk6:A    (THR45) to   (GLU267)  STRUCTURE OF NEK2 BOUND TO AMINOPYRAZINE COMPOUND 36  |   TRANSFERASE, CENTROSOME, MITOSIS 
2xk7:A    (THR45) to   (GLU267)  STRUCTURE OF NEK2 BOUND TO AMINOPYRAZINE COMPOUND 23  |   TRANSFERASE, CENTROSOME, MITOSIS 
2xk8:A    (THR45) to   (ASN268)  STRUCTURE OF NEK2 BOUND TO AMINOPYRAZINE COMPOUND 15  |   TRANSFERASE, CENTROSOME, MITOSIS 
2xkc:A    (THR45) to   (ASN268)  STRUCTURE OF NEK2 BOUND TO AMINOPYRAZINE COMPOUND 14  |   TRANSFERASE, CENTROSOME, MITOSIS 
2xke:A    (THR45) to   (GLU267)  STRUCTURE OF NEK2 BOUND TO AMINIPYRAZINE COMPOUND 5  |   TRANSFERASE, CENTROSOME, MITOSIS 
2xkf:A    (THR45) to   (GLU267)  STRUCTURE OF NEK2 BOUND TO AMINOPYRAZINE COMPOUND 2  |   TRANSFERASE, CENTROSOME, MITOSIS 
1vr2:A   (THR875) to  (ASN1167)  HUMAN VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2 (KDR) KINASE DOMAIN  |   TYROSINE KINASE, TRANSFERASE 
4mxx:B   (SER303) to   (TYR519)  HUMAN SRC A403T MUTANT BOUND TO KINASE INHIBITOR BOSUTINIB  |   KINASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4mxz:A   (GLU310) to   (TYR519)  SRC M314L T338M DOUBLE MUTANT BOUND TO KINASE INHIBITOR BOSUTINIB  |   KINASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1jsv:A    (THR47) to   (HIS283)  THE STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 (CDK2) IN COMPLEX WITH 4-[(6-AMINO-4-PYRIMIDINYL) AMINO]BENZENESULFONAMIDE  |   CDK2, SERINE/THREONINE PROTEIN KINASE, CELL CYCLE, ATP- BINDING, TRANSFERASE 
2xmy:A    (SER46) to   (GLN287)  DISCOVERY AND CHARACTERISATION OF 2-ANILINO-4-(THIAZOL-5-YL) PYRIMIDINE TRANSCRIPTIONAL CDK INHIBITORS AS ANTICANCER AGENTS  |   CELL CYCLE, TRANSFERASE, CDK9 INHIBITOR 
1jvp:P    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF HUMAN CDK2 (UNPHOSPHORYLATED) IN COMPLEX WITH PKF049-365  |   PROTEIN KINASE, CELL DIVISION, CELL CYCLE, ENZYME INHIBITORS, DRUG DESIGN, TRANSFERASE 
2xnb:A    (PRO45) to   (GLN287)  DISCOVERY AND CHARACTERISATION OF 2-ANILINO-4-(THIAZOL-5-YL) PYRIMIDINE TRANSCRIPTIONAL CDK INHIBITORS AS ANTICANCER AGENTS  |   CELL CYCLE, TRANSFERASE, CDK9 INHIBITOR 
2xnn:A    (THR45) to   (GLU267)  STRUCTURE OF NEK2 BOUND TO CCT242430  |   TRANSFERASE, CENTROSOME, MITOSIS, CELL CYCLE 
2xnp:A    (GLU46) to   (ASN268)  STRUCTURE OF NEK2 BOUND TO CCT244858  |   TRANSFERASE, CENTROSOME, MITOSIS, CELL CYCLE 
3wzd:A   (THR875) to  (ASN1167)  KDR IN COMPLEX WITH LIGAND LENVATINIB  |   KDR RECEPTOR KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3wze:A   (HIS876) to  (ASN1167)  KDR IN COMPLEX WITH LIGAND SORAFENIB  |   KDR RECEPTOR KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3x2u:A    (ILE85) to   (HIS294)  MICHAELIS-LIKE INITIAL COMPLEX OF CAMP-DEPENDENT PROTEIN KINASE CATALYTIC SUBUNIT.  |   MICHAELIS-LIKE COMPLEX, PROTEIN-SUBSTRATE, PKAC-ATPMG2 TERNARY, SER/THR KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-PEPTIDE COMPLEX 
5b2l:A   (LYS173) to   (HIS393)  A CRUCIAL ROLE OF CYS218 IN THE STABILIZATION OF AN UNPRECEDENTED AUTO-INHIBITION FORM OF MAP2K7  |   PROTEIN KINASE, MUTATION, APO STRUCTURE, TRANSFERASE 
5b7v:B   (LYS523) to   (LEU760)  HUMAN FGFR1 KINASE IN COMPLEX WITH CH5183284  |   PROTEIN KINASE, ATP-BINDING, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3zew:B   (THR654) to   (ASN880)  CRYSTAL STRUCTURE OF EPHB4 IN COMPLEX WITH STAUROSPORINE  |   TRANSFERASE, INHIBITOR 
3zfm:A   (GLU661) to   (ASN886)  CRYSTAL STRUCTURE OF EPHB2  |   TRANSFERASE 
3zfx:C   (SER658) to   (ASN884)  CRYSTAL STRUCTURE OF EPHB1  |   TRANSFERASE 
2xvd:A   (THR654) to   (ASN880)  EPHB4 KINASE DOMAIN INHIBITOR COMPLEX  |   TRANSFERASE, NUCLEOTIDE-BINDING 
3zfy:A   (THR672) to   (ASN898)  CRYSTAL STRUCTURE OF EPHB3  |   TRANSFERASE 
3zfy:B   (ARG674) to   (ASN898)  CRYSTAL STRUCTURE OF EPHB3  |   TRANSFERASE 
1w8c:A    (SER46) to   (HIS283)  CO-CRYSTAL STRUCTURE OF 6-CYCLOHEXYLMETHOXY-8-ISOPROPYL-9H- PURIN-2-YLAMINE AND MONOMERIC CDK2  |   TRANSFERASE, CELL CYCLE, PHOSPHORYLATION, MITOSIS, INHIBITION, CELL DIVISION 
2jiv:A   (GLU758) to   (ALA972)  CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN T790M MUTATION IN COMPEX WITH HKI-272  |   HKI272, HKI-272, RECEPTOR, CELL CYCLE, ATP-BINDING, TRANSFERASE, TYROSINE-PROTEIN KINASE, TRANSMEMBRANE, PHOSPHORYLATION, DISEASE MUTATION, NUCLEOTIDE-BINDING, ANTI-ONCOGENE, EPIDERMAL GROWTH FACTOR 
2jkm:A   (SER463) to   (GLN686)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH BIS- ANILINO PYRIMIDINE INHIBITOR  |   TYROSINE-PROTEIN KINASE, TYROSINE- PROTEIN KINASE, KINASE, MEMBRANE, TRANSFERASE, ATP-BINDING, INTEGRIN SIGNALING, NUCLEOTIDE-BINDING, FOCAL ADHESION, CELL MIGRATION, KINASE INHIBITOR, CELL JUNCTION, CELL MEMBRANE, PHOSPHOPROTEIN 
2jko:A   (ASP462) to   (GLN686)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH BIS- ANILINO PYRIMIDINE INHIBITOR  |   TYROSINE-PROTEIN KINASE, TYROSINE- PROTEIN KINASE, KINASE, MEMBRANE, TRANSFERASE, ATP-BINDING, INTEGRIN SIGNALING, NUCLEOTIDE-BINDING, FOCAL ADHESION, CELL MIGRATION, KINASE INHIBITOR, CELL JUNCTION, CELL MEMBRANE, PHOSPHOPROTEIN 
2jkq:A   (ASP462) to   (GLN686)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH BIS- ANILINO PYRIMIDINE INHIBITOR  |   TRANSFERASE, NUCLEOTIDE-BINDING, TYROSINE-PROTEIN KINASE, KINASE INHIBITOR, INTEGRIN SIGNALING, KINASE, ATP-BINDING, CELL MIGRATION, FOCAL ADHESION 
1wcc:A    (SER46) to   (HIS283)  SCREENING FOR FRAGMENT BINDING BY X-RAY CRYSTALLOGRAPHY  |   CDK2, KINASE, CELL CYCLE, FRAGMENT SCREENING, TRANSFERASE 
2xyu:A   (ASP661) to   (ILE882)  CRYSTAL STRUCTURE OF EPHA4 KINASE DOMAIN IN COMPLEX WITH VUF 12058  |   SIGNALING PROTEIN, TRANSFERASE 
5bvn:A   (THR662) to   (ALA909)  FRAGMENT-BASED DISCOVERY OF POTENT AND SELECTIVE DDR1/2 INHIBITORS  |   DDR1, FRAGMENTS, TRANSFERASE 
5bvo:A   (THR662) to   (LEU905)  FRAGMENT-BASED DISCOVERY OF POTENT AND SELECTIVE DDR1/2 INHIBITORS  |   DDR1, FRAGMENTS, TRANSFERASE 
4neu:B    (ASN52) to   (GLU269)  X-RAY STRUCTURE OF RECEPTOR INTERACTING PROTEIN 1 (RIP1)KINASE DOMAIN WITH A 1-AMINOISOQUINOLINE INHIBITOR  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE 
4nk9:A   (THR521) to   (LEU760)  CRYSTAL STRUCTURE OF HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN IN COMPLEX WITH PYRAZOLAMINOPYRIMIDINE 1  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANS-MEMBRANE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4nk9:B   (THR521) to   (LEU760)  CRYSTAL STRUCTURE OF HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN IN COMPLEX WITH PYRAZOLAMINOPYRIMIDINE 1  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANS-MEMBRANE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4nka:A   (LYS523) to   (LEU760)  CRYSTAL STRUCTURE OF HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN IN COMPLEX WITH PYRAZOLAMINOPYRIMIDINE 2  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANS-MEMBRANE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4nka:B   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN IN COMPLEX WITH PYRAZOLAMINOPYRIMIDINE 2  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANS-MEMBRANE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4nks:A   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN IN COMPLEX WITH PYRAZOLAMINOPYRIMIDINE 3  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANS-MEMBRANE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4nks:B   (THR521) to   (LEU760)  CRYSTAL STRUCTURE OF HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN IN COMPLEX WITH PYRAZOLAMINOPYRIMIDINE 3  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANS-MEMBRANE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
1ke5:A    (PRO45) to   (HIS283)  CDK2 COMPLEXED WITH N-METHYL-4-{[(2-OXO-1,2-DIHYDRO-3H- INDOL-3-YLIDENE)METHYL]AMINO}BENZENESULFONAMIDE  |   CYCLIN KINASE, TRANSFERASE 
1ke7:A    (SER46) to   (GLN287)  CYCLIN-DEPENDENT KINASE 2 (CDK2) COMPLEXED WITH 3-{[(2,2- DIOXIDO-1,3-DIHYDRO-2-BENZOTHIEN-5-YL)AMINO]METHYLENE}-5- (1,3-OXAZOL-5-YL)-1,3-DIHYDRO-2H-INDOL-2-ONE  |   CYCLIN, KINASE, TRANSFERASE 
1ke8:A    (SER46) to   (GLN287)  CYCLIN-DEPENDENT KINASE 2 (CDK2) COMPLEXED WITH 4-{[(2-OXO- 1,2-DIHYDRO-3H-INDOL-3-YLIDENE)METHYL]AMINO}-N-(1,3- THIAZOL-2-YL)BENZENESULFONAMIDE  |   CYCLIN KINASE, TRANSFERASE 
1ke9:A    (SER46) to   (HIS283)  CYCLIN-DEPENDENT KINASE 2 (CDK2) COMPLEXED WITH 3-{[4- ({[AMINO(IMINO)METHYL]AMINOSULFONYL)ANILINO]METHYLENE}-2- OXO-2,3-DIHYDRO-1H-INDOLE  |   CYCLIN, KINASE, TRANSFERASE 
2y4p:C    (SER57) to   (HIS272)  DIMERIC STRUCTURE OF DAPK-1 CATALYTIC DOMAIN  |   CALMODULIN-BINDING, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, APOPTOSIS, TRANSFERASE, ATP-BINDING 
3zos:A   (LYS663) to   (LEU905)  STRUCTURE OF THE DDR1 KINASE DOMAIN IN COMPLEX WITH PONATINIB  |   TRANSFERASE, RTK, COLLAGEN, DISCOIDIN DOMAIN 
2y6m:A   (THR660) to   (ILE882)  CRYSTAL STRUCTURE OF EPHA4 KINASE DOMAIN  |   TRANSFERASE 
2y6o:A   (LEU668) to   (ILE882)  CRYSTAL STRUCTURE OF EPHA4 KINASE DOMAIN IN COMPLEX WITH DASATINIB.  |   SIGNALLING PROTEIN, TRANSFERASE 
2yak:A    (SER57) to   (HIS272)  STRUCTURE OF DEATH-ASSOCIATED PROTEIN KINASE 1 (DAPK1) IN COMPLEX WITH A RUTHENIUM OCTASPORINE LIGAND (OSV)  |   TRANSFERASE, OCTAHEDRAL RUTHENIUM INHIBITORY COMPLEX, KINASE INHIBITOR 
3zut:B    (GLU60) to   (HIS274)  THE STRUCTURE OF OST1 (D160A) KINASE  |   TRANSFERASE, KINASE REGULATION, PLANT ABIOTIC STRESS, SIGNALING 
4nwm:A   (GLU439) to   (GLU657)  CRYSTAL STRUCTURE OF BRUTON AGAMMAGLOBULINEMIA TYROSINE KINASE COMPLEXED WITH BMS-809959 AKA 4-TERT-BUTYL-N-[2-ME THYL-3-(6-{[4- (MORPHOLINE-4-CARBONYL)PHENYL]AMINO}-9H- PURIN-2-YL)PHENYL]BENZAMIDE  |   KINASE, BTK, ATK, XLA, PSCTK1, AGMX1, AT, IMD1, MGC126261, MGC126262 BPK, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4nwm:B   (ALA446) to   (GLU657)  CRYSTAL STRUCTURE OF BRUTON AGAMMAGLOBULINEMIA TYROSINE KINASE COMPLEXED WITH BMS-809959 AKA 4-TERT-BUTYL-N-[2-ME THYL-3-(6-{[4- (MORPHOLINE-4-CARBONYL)PHENYL]AMINO}-9H- PURIN-2-YL)PHENYL]BENZAMIDE  |   KINASE, BTK, ATK, XLA, PSCTK1, AGMX1, AT, IMD1, MGC126261, MGC126262 BPK, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5c8k:A   (SER752) to   (ARG973)  EGFR KINASE DOMAIN MUTANT "TMLR" WITH COMPOUND 1  |   PROTEIN KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5c8m:A   (SER752) to   (ARG973)  EGFR KINASE DOMAIN MUTANT "TMLR" WITH COMPOUND 17  |   PROTEIN KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5c8n:A   (SER752) to   (ARG973)  EGFR KINASE DOMAIN MUTANT "TMLR" WITH COMPOUND 23  |   PROTEIN KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5cal:A   (SER752) to   (ARG973)  EGFR KINASE DOMAIN MUTANT "TMLR" WITH COMPOUND 24  |   PROTEIN KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5caq:A   (SER752) to   (ARG973)  EGFR KINASE DOMAIN MUTANT "TMLR" WITH COMPOUND 33  |   PROTEIN KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5can:A   (SER752) to   (ARG973)  EGFR KINASE DOMAIN MUTANT "TMLR" WITH COMPOUND 27  |   PROTEIN KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5cao:A   (SER752) to   (ARG973)  EGFR KINASE DOMAIN MUTANT "TMLR" WITH COMPOUND 29  |   PHOSPHOTRANSFER, INHIBITOR, PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5cap:A   (SER752) to   (ARG973)  EGFR KINASE DOMAIN MUTANT "TMLR" WITH COMPOUND 30  |   PROTEIN KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2yjr:A  (GLU1158) to  (ASP1389)  STRUCTURE OF F1174L MUTANT ANAPLASTIC LYMPHOMA KINASE  |   TRANSFERASE, CRIZOTINIB 
2yn8:A   (SER663) to   (ASN880)  EPHB4 KINASE DOMAIN INHIBITOR COMPLEX  |   TRANSFERASE, UNPHOSPHORYLATED 
2yn8:B   (SER663) to   (ASN880)  EPHB4 KINASE DOMAIN INHIBITOR COMPLEX  |   TRANSFERASE, UNPHOSPHORYLATED 
1xh6:A    (ILE85) to   (HIS294)  CRYSTAL STRUCTURES OF PROTEIN KINASE B SELECTIVE INHIBITORS IN COMPLEX WITH PROTEIN KINASE A AND MUTANTS  |   PKA, KINASE-INHIBITOR-COMPLEX, SERINE/THREONINE-PROTEIN KINASE, BALANOL DERIVATIVE, TRANSFERASE/TRANSFERASE INHIBITOR COMPLEX 
5cnn:A   (ASN732) to   (ARG949)  CRYSTAL STRUCTURE OF THE EGFR KINASE DOMAIN MUTANT I682Q  |   KINASE EGFR, TRANSFERASE 
5cno:A   (ALA731) to   (ARG949)  CRYSTAL STRUCTURE OF THE EGFR KINASE DOMAIN MUTANT V924R  |   KINASE EGFR, TRANSFERASE 
5cno:B   (ASN732) to   (ARG949)  CRYSTAL STRUCTURE OF THE EGFR KINASE DOMAIN MUTANT V924R  |   KINASE EGFR, TRANSFERASE 
3k54:A   (GLU444) to   (GLU658)  STRUCTURES OF HUMAN BRUTON'S TYROSINE KINASE IN ACTIVE AND INACTIVE CONFORMATIONS SUGGESTS A MECHANISM OF ACTIVATION FOR TEC FAMILY KINASES.  |   BRUTON'S TYROSINE KINASE, BTK, DASATINIB, ATP-BINDING, DISEASE MUTATION, KINASE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
4a4x:A    (GLU46) to   (ASN268)  NEK2-EDE BOUND TO CCT248662  |   TRANSFERASE, PROTEIN KINASE, MITOSIS 
1xkk:A   (ASN756) to   (ARG973)  EGFR KINASE DOMAIN COMPLEXED WITH A QUINAZOLINE INHIBITOR- GW572016  |   EGFR, EPIDERMAL GROWTH FACTOR RECEPTOR, KINASE, TRANSFERASE 
5cyi:A    (PRO45) to   (GLN287)  CDK2/CYCLIN A COVALENT COMPLEX WITH 6-(CYCLOHEXYLMETHOXY)-N-(4- (VINYLSULFONYL)PHENYL)-9H-PURIN-2-AMINE (NU6300)  |   CDK2 CYCLIN A COVALENT INHIBITOR VINYLSULPHONE, TRANSFERASE 
5cyi:C    (PRO45) to   (GLN287)  CDK2/CYCLIN A COVALENT COMPLEX WITH 6-(CYCLOHEXYLMETHOXY)-N-(4- (VINYLSULFONYL)PHENYL)-9H-PURIN-2-AMINE (NU6300)  |   CDK2 CYCLIN A COVALENT INHIBITOR VINYLSULPHONE, TRANSFERASE 
4ot5:A   (GLU439) to   (GLU657)  CRYSTAL STRUCTURE OF BTK KINASE DOMAIN COMPLEXED WITH 4-TERT-BUTYL-N- (3-{8-[4-(4-METHYL-PIPERAZINE-1-CARBONYL)-PHENYLAMINO]-IMIDAZO[1,2- A]PYRAZIN-6-YL}-PHENYL)-BENZAMIDE  |   TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4otf:A   (GLU439) to   (ASN658)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF BRUTON'S TYROSINE KINASE WITH GDC0834  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4otq:A   (GLU445) to   (GLU657)  CRYSTAL STRUCTURE OF BTK KINASE DOMAIN COMPLEXED WITH 1-[5-[3-(7-TERT- BUTYL-4-OXO-QUINAZOLIN-3-YL)-2-METHYL-PHENYL]-1-METHYL-2-OXO-3- PYRIDYL]-3-METHYL-UREA  |   TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4acm:A    (SER46) to   (GLN287)  CDK2 IN COMPLEX WITH 3-AMINO-6-(4-{[2-(DIMETHYLAMINO)ETHYL] SULFAMOYL}-PHENYL)-N-PYRIDIN-3-YLPYRAZINE-2-CARBOXAMIDE  |   MITOSIS, CELL CYCLE, TRANSFERASE, SERINE/THREONINE- PROTEIN KINASE, ATP-BINDING, CELL DIVISION, NUCLEOTIDE-BINDING 
5d1j:A    (ARG50) to   (GLN287)  CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 (CDK2-WT) COMPLEX WITH N-[5-[[[5-(1,1-DIMETHYLETHYL)-2-OXAZOLYL] METHYL]THIO]-2-THIAZOLYL]- 4-PIPERIDINECARBOXAMIDE (BMS-387032)  |   KINASE, MITOSIS, CELL CYCLE, TRANSFERASE-TRANSFERASE INHIBIT COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4afe:A    (GLU46) to   (GLU267)  NEK2 BOUND TO HYBRID COMPOUND 21  |   TRANSFERASE, MITOSIS 
4agc:A   (HIS876) to  (ALA1168)  CRYSTAL STRUCTURE OF VEGFR2 (JUXTAMEMBRANE AND KINASE DOMAINS) IN COMPLEX WITH AXITINIB (AG-013736) (N-METHYL-2-( 3-((E)-2-PYRIDIN-2-YL-VINYL)-1H-INDAZOL-6-YLSULFANYL)- BENZAMIDE)  |   TRANSFERASE, ANGIOGENESIS, NUCLEOTIDE-BINDING, INHIBITOR, PHOSPHORYLATION, TRANSMEMBRANE 
4p2k:A   (THR653) to   (ILE875)  STRUCTURE OF EPHRIN TYPE-A RECEPTOR 2  |   EPHA2, TRANSFERASE 
1y6a:A   (THR873) to  (ASN1165)  CRYSTAL STRUCTURE OF VEGFR2 IN COMPLEX WITH A 2-ANILINO-5-ARYL-OXAZOLE INHIBITOR  |   TRANSFERASE 
1y6b:A   (THR873) to  (ALA1166)  CRYSTAL STRUCTURE OF VEGFR2 IN COMPLEX WITH A 2-ANILINO-5-ARYL-OXAZOLE INHIBITOR  |   TRANSFERASE 
4p4c:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE DOMAIN IN COMPLEX WITH QUINOXALINE DERIVATIVES  |   TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4p5z:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE DOMAIN IN COMPLEX WITH QUINOXALINE DERIVATIVES  |   TRANSFERASE, TRANSFERASE INHIBITOR 
1mp8:A   (ARG465) to   (GLN686)  CRYSTAL STRUCTURE OF FOCAL ADHESION KINASE (FAK)  |   TYROSINE PROTEIN KINASE, TRANSFERASE 
1y8y:A    (SER46) to   (GLN287)  CRYSTAL STRUCTURE OF HUMAN CDK2 COMPLEXED WITH A PYRAZOLO[1, 5-A]PYRIMIDINE INHIBITOR  |   SERINE/THREONINE PROTEIN KINASE, CDK2, ATP-BINDING, CELL CYCLE, MITOSIS, PHOSPHORYLATION, PYRAZOLOPYRIMIDINE INHIBITOR, TRANSFERASE 
1mqb:A   (THR653) to   (ALA877)  CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE  |   TYROSINE PROTEIN KINASE, TRANSFERASE 
1mqb:B   (THR653) to   (ALA877)  CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE  |   TYROSINE PROTEIN KINASE, TRANSFERASE 
3a4p:A  (ASP1117) to  (ARG1336)  HUMAN C-MET KINASE DOMAIN COMPLEXED WITH 6-BENZYLOXYQUINOLINE INHIBITOR  |   C-MET, TYROSINE-PROTEIN KINASE, HEPATOCYTE GROWTH FACTOR RECEPTOR, TRANSFERASE 
4pdo:A   (THR653) to   (ILE875)  STRUCTURE OF EPHRIN TYPE-A RECEPTOR 2  |   EPHA2, TRANSFERASE 
4pdo:B   (THR653) to   (ILE875)  STRUCTURE OF EPHRIN TYPE-A RECEPTOR 2  |   EPHA2, TRANSFERASE 
3ky2:A   (THR521) to   (LEU760)  CRYSTAL STRUCTURE OF FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN  |   KINASE, RTK, PHOSPHORYLATION, INTERFACE, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, DWARFISM, GLYCOPROTEIN, HEPARIN-BINDING, HYPOGONADOTROPIC HYPOGONADISM, IMMUNOGLOBULIN DOMAIN, KALLMANN SYNDROME, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3ky2:B   (THR521) to   (LEU760)  CRYSTAL STRUCTURE OF FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN  |   KINASE, RTK, PHOSPHORYLATION, INTERFACE, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, DWARFISM, GLYCOPROTEIN, HEPARIN-BINDING, HYPOGONADOTROPIC HYPOGONADISM, IMMUNOGLOBULIN DOMAIN, KALLMANN SYNDROME, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
5dg5:A  (ILE1118) to  (PHE1344)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF THE HEPATOCYTE GROWTH FACTOR RECEPTOR C-MET IN COMPLEX WITH ALTIRATINIB ANALOG DP- 4157  |   TYROSINE KINASE DOMAIN, HEPATOCYTE GROWTH FACTOR RECEPTOR C-MET, C- MET, ALTIRATINIB ANALOG, DP-4157, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1yqj:A    (SER61) to   (SER261)  CRYSTAL STRUCTURE OF P38 ALPHA IN COMPLEX WITH A SELECTIVE PYRIDAZINE INHIBITOR  |   TRANSFERASE 
1ywn:A   (THR873) to  (GLN1167)  VEGFR2 IN COMPLEX WITH A NOVEL 4-AMINO-FURO[2,3-D]PYRIMIDINE  |   TRANSFERASE 
4pmt:A   (ARG559) to   (HIS788)  THE STRUCTURE OF TRKA KINASE BOUND TO THE INHIBITOR N~4~-(4-MORPHOLIN- 4-YLPHENYL)-N~6~-(PYRIDIN-3-YLMETHYL)PYRIDO[3,2-D]PYRIMIDINE-4,6- DIAMINE  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3l8v:A  (GLY1119) to  (PHE1344)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF THE HEPATOCYTE GROWTH FACTOR RECEPTOR C-MET IN COMPLEX WITH A BIARYLAMINE BASED INHIBITOR  |   RECEPTOR TYROSINE KINASE, SIGNAL TRANSDUCTION, GRB2, SHC, ATP- BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, ALTERNATIVE SPLICING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, DISULFIDE BOND, KINASE, POLYMORPHISM, RECEPTOR 
4pp9:A   (SER399) to   (SER618)  ITK KINASE DOMAIN WITH COMPOUND 1 (N-[1-(3-CYANOBENZYL)-1H-PYRAZOL-4- YL]-2H-INDAZOLE-3-CARBOXAMIDE)  |   PROTEIN KINASE, PHOSPHO-TRANSFER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4pp9:B   (SER399) to   (SER618)  ITK KINASE DOMAIN WITH COMPOUND 1 (N-[1-(3-CYANOBENZYL)-1H-PYRAZOL-4- YL]-2H-INDAZOLE-3-CARBOXAMIDE)  |   PROTEIN KINASE, PHOSPHO-TRANSFER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ppa:A   (PHE403) to   (GLU617)  ITK KINASE DOMAIN WITH COMPOUND 11 (N-[1-(3-CYANOBENZYL)-1H-PYRAZOL-4- YL]-6-(1H-PYRAZOL-4-YL)-1H-INDAZOLE-3-CARBOXAMIDE)  |   PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ppb:B   (GLU401) to   (ALA616)  ITK KINASE DOMAIN WITH COMPOUND 28 (N-{1-[(1S)-3-(DIMETHYLAMINO)-1- PHENYLPROPYL]-1H-PYRAZOL-4-YL}-6-(1H-PYRAZOL-4-YL)-1H-INDAZOLE-3- CARBOXAMIDE)  |   PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4pqn:A   (GLU400) to   (ILE615)  ITK KINASE DOMAIN WITH COMPOUND GNE-9822  |   PROTEIN KINASE, PHOSPHO-TRANSFER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3lfq:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF CDK2 WITH SAR60, AN AMINOINDAZOLE TYPE INHIBITOR  |   PROTEIN KINASE FOLD, ACETYLATION, ATP-BINDING, CELL CYCLE, CELL DIVISION, KINASE, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3lfs:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF CDK2 WITH SAR37, AN AMINOINDAZOLE TYPE INHIBITOR  |   PROTEIN KINASE FOLD, ACETYLATION, ATP-BINDING, CELL CYCLE, CELL DIVISION, KINASE, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
5dr6:A   (VAL174) to   (HIS380)  AURORA A KINASE IN COMPLEX WITH AA30 AND JNJ-7706621 IN SPACE GROUP P6122  |   AURORA A KINASE, MITOTIC KINASE, PPI, TRANSFERASE 
4aoj:A   (GLU551) to   (ALA787)  HUMAN TRKA IN COMPLEX WITH THE INHIBITOR AZ-23  |   TRANSFERASE, INHIBITOR 
4aoj:B   (GLU551) to   (ALA787)  HUMAN TRKA IN COMPLEX WITH THE INHIBITOR AZ-23  |   TRANSFERASE, INHIBITOR 
4aoj:C   (SER550) to   (ALA787)  HUMAN TRKA IN COMPLEX WITH THE INHIBITOR AZ-23  |   TRANSFERASE, INHIBITOR 
3lmg:B   (ASP739) to   (PRO953)  CRYSTAL STRUCTURE OF THE ERBB3 KINASE DOMAIN IN COMPLEX WITH AMP-PNP  |   ERBB3, HER3, TYROSINE KINASE DOMAIN, AMP-PNP, NUCLEOTIDE BINDING, TRANSFERASE 
3lq8:A  (ILE1118) to  (THR1343)  STRUCTURE OF THE KINASE DOMAIN OF C-MET BOUND TO XL880 (GSK1363089)  |   KINASE DOMAIN, XL880, GSK1363089, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
4aw5:A   (THR130) to   (PRO357)  COMPLEX OF THE EPHB4 KINASE DOMAIN WITH AN OXINDOLE INHIBITOR  |   TRANSFERASE 
1zy4:A   (THR633) to   (SER978)  CRYSTAL STRUCTURE OF EIF2ALPHA PROTEIN KINASE GCN2: R794G HYPERACTIVATING MUTANT IN APO FORM.  |   TRANSLATION REGULATOR, PROTEIN KINASE, SIGNAL TRANSDUCTION, AMINO- ACID STARVATION, STARVATION STRESS RESPONSE, EIF2ALPHA KINASE, TRANSFERASE 
1zy5:A   (THR633) to   (SER978)  CRYSTAL STRUCTURE OF EIF2ALPHA PROTEIN KINASE GCN2: R794G HYPERACTIVATING MUTANT COMPLEXED WITH AMPPNP.  |   TRANSLATION REGULATOR, PROTEIN KINASE, SIGNAL TRANSDUCTION, AMINO-ACID STARVATION, STARVATION STRESS RESPONSE, EIF2ALPHA KINASE, TRANSFERASE 
2a0c:X    (SER46) to   (GLN287)  HUMAN CDK2 IN COMPLEX WITH OLOMOUCINE II, A NOVEL 2,6,9- TRISUBSTITUTED PURINE CYCLIN-DEPENDENT KINASE INHIBITOR  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, 3D-STRUCTURE 
2a4l:A    (ALA48) to   (GLN287)  HUMAN CYCLIN-DEPENDENT KINASE 2 IN COMPLEX WITH ROSCOVITINE  |   TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, ATP-BINDING, CELL CYCLE, CELL DIVISION, ROSCOVITINE, PHOSPHORYLATION 
4qd6:A   (PHE403) to   (SER618)  ITK KINASE DOMAIN IN COMPLEX WITH INHIBITOR COMPOUND  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5edp:A   (SER752) to   (ARG973)  EGFR KINASE (T790M/L858R) APO  |   PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5edq:A   (SER752) to   (ARG973)  EGFR KINASE (T790M/L858R) WITH INHIBITOR COMPOUND 15: ~{N}-(7- CHLORANYL-1~{H}-INDAZOL-3-YL)-7,7-DIMETHYL-2-(1~{H}-PYRAZOL-4-YL)- 5~{H}-FURO[3,4-D]PYRIMIDIN-4-AMINE  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5edr:A   (SER752) to   (ARG973)  EGFR KINASE (T790M/L858R) WITH INHIBITOR COMPOUND 27: ~{N}-(1~{H}- INDAZOL-3-YL)-7,7-DIMETHYL-2-(2-METHYLPYRAZOL-3-YL)-5~{H}-FURO[3,4- D]PYRIMIDIN-4-AMINE  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4bb4:A   (THR654) to   (ASN880)  EPHB4 KINASE DOMAIN INHIBITOR COMPLEX  |   TRANSFERASE, UNPHOSPHORYLATED 
3b8q:A   (SER877) to  (HIS1178)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A NAPHTHAMIDE INHIBITOR  |   RECEPTOR TYROSINE KINASE, ANGIOGENESIS, ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST- VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3b8r:A   (HIS876) to  (HIS1178)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A NAPHTHAMIDE INHIBITOR  |   RECEPTOR TYROSINE KINASE, ANGIOGENESIS, ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST- VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3b8r:B   (THR875) to  (ALA1166)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A NAPHTHAMIDE INHIBITOR  |   RECEPTOR TYROSINE KINASE, ANGIOGENESIS, ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST- VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
4bci:A    (ILE61) to   (SER317)  STRUCTURE OF CDK9 IN COMPLEX WITH CYCLIN T AND A 2-AMINO-4- HETEROARYL-PYRIMIDINE INHIBITOR  |   TRANSFERASE-CELL CYCLE COMPLEX, CDK-CYCLIN COMPLEX, TRANSCRIPTION-PROTEIN BINDING, STRUCTURE-BASED DRUG DESIGN 
4bck:A    (PRO45) to   (GLN287)  STRUCTURE OF CDK2 IN COMPLEX WITH CYCLIN A AND A 2-AMINO-4- HETEROARYL-PYRIMIDINE INHIBITOR  |   TRANSFERASE-CELL CYCLE COMPLEX, CDK-CYCLIN COMPLEX, STRUCTURE-BASED DRUG DESIGN 
4bck:C    (PRO45) to   (GLN287)  STRUCTURE OF CDK2 IN COMPLEX WITH CYCLIN A AND A 2-AMINO-4- HETEROARYL-PYRIMIDINE INHIBITOR  |   TRANSFERASE-CELL CYCLE COMPLEX, CDK-CYCLIN COMPLEX, STRUCTURE-BASED DRUG DESIGN 
5ek7:B   (THR653) to   (ILE875)  STRUCTURE OF THE AUTOINHIBITED EPHA2 JMS-KD  |   EPHA2, KINASE, AUTOINHIBITION, TRANSFERASE 
4bcn:A    (PRO45) to   (GLN287)  STRUCTURE OF CDK2 IN COMPLEX WITH CYCLIN A AND A 2-AMINO-4- HETEROARYL-PYRIMIDINE INHIBITOR  |   TRANSFERASE-CELL CYCLE COMPLEX, CDK-CYCLIN COMPLEX, CYCLIN-INHIBITOR, STRUCTURE-BASED DRUG DESIGN 
4bcq:C    (PRO45) to   (HIS283)  STRUCTURE OF CDK2 IN COMPLEX WITH CYCLIN A AND A 2-AMINO-4- HETEROARYL-PYRIMIDINE INHIBITOR  |   TRANSFERASE-CELL CYCLE COMPLEX, CDK-CYCLIN COMPLEX, CYCLIN A, CYCLIN- DEPENDENT KINASE 2, STRUCTURE-BASED DRUG DESIGN 
5em5:A   (SER752) to   (ARG973)  EGFR KINASE DOMAIN MUTANT "TMLR" WITH PYRIDONE COMPOUND 2: 4-[2-(4- CHLOROPHENYL)ETHYLAMINO]-~{N}-[4-(4-METHYLPIPERAZIN-1-YL)PHENYL]-2- OXIDANYLIDENE-1~{H}-PYRIDINE-3-CARBOXAMIDE  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5em6:A   (PRO753) to   (ARG973)  EGFR KINASE DOMAIN MUTANT "TMLR" WITH PYRIDONE COMPOUND 19: 4-[(2- AZANYLPYRIMIDIN-4-YL)AMINO]-~{N}-[4-(4-METHYLPIPERAZIN-1-YL)PHENYL]- 2-OXIDANYLIDENE-1~{H}-PYRIDINE-3-CARBOXAMIDE  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5em7:A   (SER752) to   (ARG973)  EGFR KINASE DOMAIN MUTANT "TMLR" WITH PYRIDONE COMPOUND 13: 4-[(2- METHOXYPHENYL)AMINO]-~{N}-[4-(4-METHYLPIPERAZIN-1-YL)PHENYL]-2- OXIDANYLIDENE-1~{H}-PYRIDINE-3-CARBOXAMIDE  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3bbt:B   (ASN737) to   (PRO956)  CRYSTAL STRUCTURE OF THE ERBB4 KINASE IN COMPLEX WITH LAPATINIB  |   INACTIVE KINASE CONFORMATION, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3bbt:D   (VAL738) to   (ARG954)  CRYSTAL STRUCTURE OF THE ERBB4 KINASE IN COMPLEX WITH LAPATINIB  |   INACTIVE KINASE CONFORMATION, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3mj2:A   (GLU406) to   (ILE615)  X-RAY CRYSTAL STRUCTURE OF ITK COMPLEXED WITH INHIBITOR BMS-509744  |   HELIX C-OUT, SUBSTRATE BLOCKING ACTIVATION LOOP CONFORMATION, TRANSFERASE 
4bi0:A   (ASP561) to   (HIS788)  SCAFFOLD FOCUSED VIRTUAL SCREENING: PROSPECTIVE APPLICATION TO THE DISCOVERY OF TTK INHIBITOR  |   TRANSFERASE, PROTEIN KINASE, MITOSIS 
4bie:B   (LEU722) to   (ASP935)  CRYSTAL STRUCTURES OF ASK1-INHIBITOR COMPLEXES  |   TRANSFERASE, STRUCTURE BASED DESGIN 
5etc:A    (SER61) to   (SER261)  STRUCTURE OF INACTIVE MAPK14 WITH ORDERED ACTIVATION LOOP  |   MAPK14, INACTIVE KINASE, ACTIVATION LOOP, MAPK, TRANSFERASE 
4bkj:A   (THR662) to   (VAL913)  CRYSTAL STRUCTURE OF THE HUMAN DDR1 KINASE DOMAIN IN COMPLEX WITH IMATINIB  |   TRANSFERASE, RECEPTOR, RTK, COLLAGEN, DISCOIDIN DOMAIN, RECEPTOR TYROSINE KINASE 
4bkj:B   (THR662) to   (VAL913)  CRYSTAL STRUCTURE OF THE HUMAN DDR1 KINASE DOMAIN IN COMPLEX WITH IMATINIB  |   TRANSFERASE, RECEPTOR, RTK, COLLAGEN, DISCOIDIN DOMAIN, RECEPTOR TYROSINE KINASE 
5ew8:A   (GLU522) to   (LEU760)  FIBROBLAST GROWTH FACTOR RECEPTOR 1 IN COMPLEX WITH JNJ-4275693  |   FGFR1 KINASE INHIBITOR COMPLEX, KINASE, TRANSFERASE 
5ew8:B   (GLU522) to   (LEU760)  FIBROBLAST GROWTH FACTOR RECEPTOR 1 IN COMPLEX WITH JNJ-4275693  |   FGFR1 KINASE INHIBITOR COMPLEX, KINASE, TRANSFERASE 
5eyk:B   (GLU135) to   (HIS340)  CRYSTAL STRUCTURE OF AURORA B IN COMPLEX WITH BI 847325  |   KINASE, INHIBITOR, TRANSFERASE 
3my1:A    (PRO60) to   (SER317)  STRUCTURE OF CDK9/CYCLINT1 IN COMPLEX WITH DRB  |   CDK-CYCLIN COMPLEX, PHOSPHORYLATED, TRANSCRIPTION-PROTEIN BINDING- INHIBITOR COMPLEX 
4brx:A   (ASP462) to   (LYS684)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH A DIARYLAMINO-1,3,5-TRIAZINE INHIBITOR  |   TRANSFERASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
3bwj:A    (ILE85) to   (HIS294)  COMPLEX OF PKA WITH THE BISUBSTRATE PROTEIN KINASE INHIBITOR LEAD COMPOUND ARC-1034  |   BISUBSTRATE INHIBITOR, PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, CAMP, PHOSPHOPROTEIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3bz3:A   (SER463) to   (GLU688)  CRYSTAL STRUCTURE ANALYSIS OF FOCAL ADHESION KINASE WITH A METHANESULFONAMIDE DIAMINOPYRIMIDINE INHIBITOR  |   KINASE, DFG-HELIX, ACETYLATION, ALTERNATIVE SPLICING, ATP- BINDING, CELL JUNCTION, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3c1x:A  (ILE1118) to  (PHE1344)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF THE HEPATOCYTE GROWTH FACTOR RECEPTOR C-MET IN COMPLEX WITH A PYRROLOTRIAZINE BASED INHIBITOR  |   RECEPTOR TYROSINE KINASE, SIGNAL TRANSDUCTION, GRB2, SHC, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
5fbn:D   (GLU439) to   (GLU657)  BTK KINASE DOMAIN WITH INHIBITOR 1  |   KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, TRANSFERASE 
5fbo:A   (GLU441) to   (GLU657)  BTK-INHIBITOR CO-STRUCTURE  |   KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3c7q:A   (THR875) to  (GLN1169)  STRUCTURE OF VEGFR2 KINASE DOMAIN IN COMPLEX WITH BIBF1120  |   ALPHA BETA, ANGIOGENESIS, ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST-VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE 
4r7i:A   (ALA624) to   (ALA914)  CRYSTAL STRUCTURE OF FMS KINASE DOMAIN WITH A SMALL MOLECULAR INHIBITOR, GLEEVEC  |   CSF-1-R, FMS PROTO-ONCOGENE, C-FMS, CD115 ANTIGEN, KINASE, ATP- BINDING, GLEEVEC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3cc6:A   (LEU465) to   (GLU692)  CRYSTAL STRUCTURE OF KINASE DOMAIN OF PROTEIN TYROSINE KINASE 2 BETA (PTK2B)  |   FOCAL ADHESION KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3cjf:A   (THR873) to  (ASN1165)  CRYSTAL STRUCTURE OF VEGFR2 IN COMPLEX WITH A 3,4,5-TRIMETHOXY ANILINE CONTAINING PYRIMIDINE  |   VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2. VEGFR-2, KINASE INSERT DOMAIN RECEPTOR, PROTEIN-TYROSINE KINASE RECEPTOR FLK-1, ANGIOGENESIS, ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST-VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
4c7t:A   (SER463) to   (LYS684)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH A DIARYLAMINO-1,3,5-TRIAZINE INHIBITOR  |   TRANSFERASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
5fp5:A    (THR47) to   (GLN287)  STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH SMALL-MOLECULE LIGAND 4-FLUOROBENZOIC ACID (AT222) IN AN ALTERNATE BINDING SITE.  |   TRANSFERASE, KINASE, MITOSIS, CELL CYCLE, FRAGMENT SCREENING, ALTERNATE BINDING SITE. 
5fp6:A    (PRO45) to   (HIS283)  STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH SMALL-MOLECULE LIGAND 3-(4,7-DICHLORO-1H-INDOL-3-YL)PROP-2-YN-1-OL (AT17833) IN AN ALTERNATE BINDING SITE.  |   TRANSFERASE, KINASE, MITOSIS, CELL CYCLE, FRAGMENT SCREENING, ALTERNATE BINDING SITE. 
4riw:A   (ASP739) to   (ARG951)  CRYSTAL STRUCTURE OF AN EGFR/HER3 KINASE DOMAIN HETERODIMER  |   RECEPTOR TYROSINE KINASE, PSEUDOKINASE, KINASE, ATP BINDING, MEMBRANE, TRANSFERASE 
4rix:A   (HIS740) to   (ARG951)  CRYSTAL STRUCTURE OF AN EGFR/HER3 KINASE DOMAIN HETERODIMER CONTAINING THE CANCER-ASSOCIATED HER3-Q790R MUTATION  |   RECEPTOR TYROSINE KINASE, PSEUDOKINASE, KINASE, ATP BINDING, MEMBRANE, TRANSFERASE 
4riy:A   (THR738) to   (ARG951)  CRYSTAL STRUCTURE OF AN EGFR/HER3 KINASE DOMAIN HETERODIMER CONTAINING THE CANCER-ASSOCIATED HER3-E909G MUTATION  |   RECEPTOR TYROSINE KINASE, PSEUDOKINASE, KINASE, ATP BINDING, MEMBRANE, TRANSFERASE 
4rj4:A   (SER752) to   (ARG973)  EGFR KINASE (T790M/L858R) WITH INHIBITOR COMPOUND 6  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4rj5:A   (SER752) to   (ARG973)  EGFR KINASE (T790M/L858R) WITH INHIBITOR COMPOUND 5  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4rj6:A   (SER752) to   (ARG973)  EGFR KINASE (T790M/L858R) WITH INHIBITOR COMPOUND 4  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4rj8:A   (PRO753) to   (ARG973)  EGFR KINASE (T790M/L858R) WITH INHIBITOR COMPOUND 8  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ns9:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF CDK2 IN COMPLEX WITH INHIBITOR BS-194  |   PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3cp9:A   (THR875) to  (HIS1178)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A PYRIDONE INHIBITOR  |   RECEPTOR TYROSINE KINASE, ANGIOGENESIS, ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST- VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3cp9:B   (HIS876) to  (LEU1164)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A PYRIDONE INHIBITOR  |   RECEPTOR TYROSINE KINASE, ANGIOGENESIS, ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST- VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3cpb:A   (THR875) to  (HIS1178)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A BISAMIDE INHIBITOR  |   RECEPTOR TYROSINE KINASE, ANGIOGENESIS, ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST- VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3cpb:B   (SER877) to  (LEU1164)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A BISAMIDE INHIBITOR  |   RECEPTOR TYROSINE KINASE, ANGIOGENESIS, ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST- VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3cpc:A   (THR875) to  (HIS1178)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A PYRIDONE INHIBITOR  |   RECEPTOR TYROSINE KINASE, ANGIOGENESIS, ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST-VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
4cfm:A    (PRO45) to   (GLN287)  STRUCTURE-BASED DESIGN OF C8-SUBSTITUTED O6- CYCLOHEXYLMETHOXYGUANINE CDK1 AND 2 INHIBITORS.  |   CELL CYCLE, CYCLIN DEPENDENT KINASES, STRUCTURE-BASED DRUG DESIGN, CONFORMATIONAL RESTRAINT, REVERSED BINDING MODE 
4cfm:C    (PRO45) to   (GLN287)  STRUCTURE-BASED DESIGN OF C8-SUBSTITUTED O6- CYCLOHEXYLMETHOXYGUANINE CDK1 AND 2 INHIBITORS.  |   CELL CYCLE, CYCLIN DEPENDENT KINASES, STRUCTURE-BASED DRUG DESIGN, CONFORMATIONAL RESTRAINT, REVERSED BINDING MODE 
4cfn:A    (PRO45) to   (GLN287)  STRUCTURE-BASED DESIGN OF C8-SUBSTITUTED O6-CYCLOHEXYLMETHOXYGUANINE CDK1 AND 2 INHIBITORS.  |   CELL CYCLE, CYCLIN DEPENDENT KINASES, STRUCTURE-BASED DRUG DESIGN, CONFORMATIONAL RESTRAINT, REVERSED BINDING MODE 
4cfn:C    (PRO45) to   (GLN287)  STRUCTURE-BASED DESIGN OF C8-SUBSTITUTED O6-CYCLOHEXYLMETHOXYGUANINE CDK1 AND 2 INHIBITORS.  |   CELL CYCLE, CYCLIN DEPENDENT KINASES, STRUCTURE-BASED DRUG DESIGN, CONFORMATIONAL RESTRAINT, REVERSED BINDING MODE 
4cfv:C    (PRO45) to   (GLN287)  STRUCTURE-BASED DESIGN OF C8-SUBSTITUTED O6- CYCLOHEXYLMETHOXYGUANINE CDK1 AND 2 INHIBITORS.  |   TRANSFERASE, CYCLIN DEPENDENT KINASES, STRUCTURE-BASED DRUG DESIGN, CONFORMATIONAL RESTRAINT, REVERSED BINDING MODE 
4cfw:C    (PRO45) to   (GLN287)  STRUCTURE-BASED DESIGN OF C8-SUBSTITUTED O6- CYCLOHEXYLMETHOXYGUANINE CDK1 AND 2 INHIBITORS.  |   CELL CYCLE, STRUCTURE-BASED DRUG DESIGN, CONFORMATIONAL RESTRAINT, REVERSED BINDING MODE 
4cfx:A    (PRO45) to   (GLN287)  STRUCTURE-BASED DESIGN OF C8-SUBSTITUTED O6-CYCLOHEXYLMETHOXYGUANINE CDK1 AND 2 INHIBITORS.  |   CELL CYCLE, STRUCTURE-BASED DRUG DESIGN, CONFORMATIONAL RESTRAINT, REVERSED BINDING MODE 
3cs9:B   (THR277) to   (SER500)  HUMAN ABL KINASE IN COMPLEX WITH NILOTINIB  |   NILOTINIB, AMN107, KINASE, ABL, ALTERNATIVE SPLICING, ATP- BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, ABL KINASE WT IN COMPLEX WITH NVP-AMN107 
3cs9:D   (GLU279) to   (SER500)  HUMAN ABL KINASE IN COMPLEX WITH NILOTINIB  |   NILOTINIB, AMN107, KINASE, ABL, ALTERNATIVE SPLICING, ATP- BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, ABL KINASE WT IN COMPLEX WITH NVP-AMN107 
3ctj:A  (GLY1119) to  (PHE1344)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF THE HEPATOCYTE GROWTH FACTOR RECEPTOR C-MET IN COMPLEX WITH A AMINOPYRIDINE BASED INHIBITOR  |   RECEPTOR TYROSINE KINASE, SIGNAL TRANSDUCTION, GRB2, SHC, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
4rt7:A   (SER652) to   (ASP949)  CRYSTAL STRUCTURE OF FLT3 WITH A SMALL MOLECULE INHIBITOR  |   KINASE, TRANSFERASE, TRANSFERASE INHIBITOR, COMPLEX, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4rwi:A   (THR521) to   (LEU760)  CRYSTAL STRUCTURE OF V561M FGFR1 GATEKEEPER MUTATION (C488A, C584S, V561M), APO  |   RECEPTOR TYROSINE KINASE, GATEKEEPER MUTATION, PROTO-ONCOGENE, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4rwi:B   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF V561M FGFR1 GATEKEEPER MUTATION (C488A, C584S, V561M), APO  |   RECEPTOR TYROSINE KINASE, GATEKEEPER MUTATION, PROTO-ONCOGENE, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4rwj:A   (THR521) to   (LEU760)  CRYSTAL STRUCTURE OF FGFR1 (C488A, C584S) IN COMPLEX WITH AZD4547 (N- {3-[2-(3,5-DIMETHOXYPHENYL)ETHYL]-1H-PYRAZOL-5-YL}-4-[(3R,5S)-3,5- DIMETHYLPIPERAZIN-1-YL]BENZAMIDE)  |   RECEPTOR TYROSINE KINASE, KINASE, PROTO-ONCOGENE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4rwj:B   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF FGFR1 (C488A, C584S) IN COMPLEX WITH AZD4547 (N- {3-[2-(3,5-DIMETHOXYPHENYL)ETHYL]-1H-PYRAZOL-5-YL}-4-[(3R,5S)-3,5- DIMETHYLPIPERAZIN-1-YL]BENZAMIDE)  |   RECEPTOR TYROSINE KINASE, KINASE, PROTO-ONCOGENE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4rwk:A   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF V561M FGFR1 GATEKEEPER MUTATION (C488A, C584S, V561M) IN COMPLEX WITH N-{3-[2-(3,5-DIMETHOXYPHENYL)ETHYL]-1H- PYRAZOL-5-YL}-4-[(3R,5S)-3,5-DIMETHYLPIPERAZIN-1-YL]BENZAMIDE (AZD4547)  |   RECEPTOR TYROSINE KINASE, GATEKEEPER MUTATION, PROTO-ONCOGENE, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4rwk:B   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF V561M FGFR1 GATEKEEPER MUTATION (C488A, C584S, V561M) IN COMPLEX WITH N-{3-[2-(3,5-DIMETHOXYPHENYL)ETHYL]-1H- PYRAZOL-5-YL}-4-[(3R,5S)-3,5-DIMETHYLPIPERAZIN-1-YL]BENZAMIDE (AZD4547)  |   RECEPTOR TYROSINE KINASE, GATEKEEPER MUTATION, PROTO-ONCOGENE, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4rwl:A   (THR521) to   (LEU760)  CRYSTAL STRUCTURE OF FGFR1 (C488A, C584C) IN COMPLEX WITH 6-(7-((1- AMINOCYCLOPROPYL) METHOXY)-6-METHOXYQUINOLIN-4-YLOXY)-N-METHYL-1- NAPHTHAMIDE (E3810)  |   RECEPTOR TYROSINE KINASE, GATEKEEPER MUTATION, PROTO-ONCOGENE, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4rwl:B   (GLU522) to   (THR761)  CRYSTAL STRUCTURE OF FGFR1 (C488A, C584C) IN COMPLEX WITH 6-(7-((1- AMINOCYCLOPROPYL) METHOXY)-6-METHOXYQUINOLIN-4-YLOXY)-N-METHYL-1- NAPHTHAMIDE (E3810)  |   RECEPTOR TYROSINE KINASE, GATEKEEPER MUTATION, PROTO-ONCOGENE, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3o51:A   (VAL174) to   (HIS380)  CRYSTAL STRUCTURE OF ANTHRANILAMIDE 10 BOUND TO AURORAA  |   AURORAA, KINASE DOMAIN, TRANSFERASE 
4csv:A    (SER45) to   (MET262)  TYROSINE KINASE AS - A COMMON ANCESTOR OF SRC AND ABL BOUND TO GLEEVEC  |   TRANSFERASE, DFG 
4ctc:A  (GLN1159) to  (ASP1389)  STRUCTURE OF THE HUMAN ANAPLASTIC LYMPHOMA KINASE IN COMPLEX WITH THE INHIBITOR 7-AMINO-3-CYCLOPROPYL-12-FLUORO- 1,10,16-TRIMETHYL-16,17-DIHYDRO-1H-8,4-(METHENO)PYRAZOLO(4, 3-H)(2,5,11)BENZOXADIAZACYCLOTETRADECIN-15(10H)-ONE  |   TRANSFERASE, INHIBITOR 
4cv9:A   (ASP561) to   (HIS788)  MPS1 KINASE WITH 3-AMINOPYRIDIN-2-ONE INHIBITORS  |   TRANSFERASE, INHIBITOR 
3ocb:A   (VAL192) to   (HIS405)  AKT1 KINASE DOMAIN WITH PYRROLOPYRIMIDINE INHIBITOR  |   SERINE-THREONINE KINASE, TRANSFERASE 
3oez:B   (SER303) to   (TYR519)  CRYSTAL STRUCTURE OF THE L317I MUTANT OF THE CHICKEN C-SRC TYROSINE KINASE DOMAIN COMPLEXED WITH IMATINIB  |   C-SRC L317I MUTANT, TYROSINE KINASE, IMATINIB, TRANSFERASE 
4tth:B    (PRO55) to   (GLN301)  CRYSTAL STRUCTURE OF A CDK6/VCYCLIN COMPLEX WITH INHIBITOR BOUND  |   KINASE, TRANSFERASE-CELL CYCLE-INHIBITOR COMPLEX 
3dj6:A   (VAL187) to   (HIS393)  CRYSTAL STRUCTURE OF THE MOUSE AURORA-A CATALYTIC DOMAIN (ASN186->GLY, LYS240->ARG, MET302->LEU) IN COMPLEX WITH COMPOUND 823.  |   AURORA A, SMALL-MOLECULE INHIBITOR, FRAGMENT-BASED DRUG DISCOVERY, KINASE, TRANSFERASE 
4d1z:A    (ARG50) to   (HIS283)  CDK2 IN COMPLEX WITH A LUCIFERIN DERIVATE  |   TRANSFERASE, CDK2, KINASE 
3dkf:A  (ILE1118) to  (ARG1336)  STRUCTURE OF MET RECEPTOR TYROSINE KINASE IN COMPLEX WITH INHIBITOR SGX-523  |   DRUG DISCOVERY, C-MET KINASE, FRAGMENT BASED, MEMBRANE, RECEPTOR, TRANSMEMBRANE, ONCOPROTEIN 
3dkg:A  (ILE1118) to  (ARG1336)  STRUCTURE OF MUTANT(Y1248L) MET RECEPTOR TYROSINE KINASE IN COMPLEX WITH INHIBITOR SGX-523  |   DRUG DISCOVERY, C-MET KINASE, FRAGMENT BASED, MEMBRANE, RECEPTOR, TRANSMEMBRANE, ONCOPROTEIN 
3dko:A   (THR672) to   (ASN896)  COMPLEX BETWEEN THE KINASE DOMAIN OF HUMAN EPHRIN TYPE-A RECEPTOR 7 (EPHA7) AND INHIBITOR ALW-II-49-7  |   ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, RECEPTOR, SIGNAL, TRANSFERASE, PHOSPHORYLATION, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE, ALTERNATIVE SPLICING, GLYCOPROTEIN, INHIBITOR, STRUCTURAL GENOMICS CONSORTIUM, SGC, MEMBRANE, PHOSPHOPROTEIN, POLYMORPHISM, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES 
4twn:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE DOMAIN IN COMPLEX WITH BIRB796  |   TRANSFERASE/TRANSFERASE INHIBITOR, TRANSFERASE 
4two:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE DOMAIN IN COMPLEX WITH COMPOUND 164  |   TRANSFERASE/TRANSFERASE INHIBITOR, TRANSFERASE 
4d4r:A   (ASP462) to   (LEU685)  FOCAL ADHESION KINASE CATALYTIC DOMAIN  |   TRANSFERASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
4d4r:B   (ASP462) to   (LYS684)  FOCAL ADHESION KINASE CATALYTIC DOMAIN  |   TRANSFERASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
4d4s:A   (SER461) to   (GLN686)  FOCAL ADHESION KINASE CATALYTIC DOMAIN  |   TRANSFERASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
4d4s:B   (SER461) to   (GLN686)  FOCAL ADHESION KINASE CATALYTIC DOMAIN  |   TRANSFERASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
4d4y:A   (SER461) to   (GLN686)  FOCAL ADHESION KINASE CATALYTIC DOMAIN  |   TRANSFERASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
4d4y:B   (SER461) to   (LEU685)  FOCAL ADHESION KINASE CATALYTIC DOMAIN  |   TRANSFERASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
4d58:A   (SER461) to   (GLN686)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH BIS- ANILINO PYRIMIDINE INHIBITOR  |   TRANSFERASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
4d58:B   (SER461) to   (LEU685)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH BIS- ANILINO PYRIMIDINE INHIBITOR  |   TRANSFERASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
3dnd:A    (ILE85) to   (HIS294)  CAMP-DEPENDENT PROTEIN KINASE PKA CATALYTIC SUBUNIT WITH PKI-5-24  |   ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, CAMP, PROTEIN KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4d5h:A   (ARG465) to   (GLN686)  FOCAL ADHESION KINASE CATALYTIC DOMAIN  |   TRANSFERASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
4d5h:B   (SER461) to   (LEU685)  FOCAL ADHESION KINASE CATALYTIC DOMAIN  |   TRANSFERASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
4d5k:A   (SER461) to   (LEU685)  FOCAL ADHESION KINASE CATALYTIC DOMAIN  |   TRANSFERASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
4d5k:B   (SER461) to   (LEU685)  FOCAL ADHESION KINASE CATALYTIC DOMAIN  |   TRANSFERASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
3dog:A    (PRO45) to   (GLN287)  STRUCTURE OF THR 160 PHOSPHORYLATED CDK2/CYCLIN A IN COMPLEX WITH THE INHIBITOR N-&-N1  |   SER/THR PROTEIN KINASE; TRANSFERASE; PHOSPHORYLATION; CELL CYCLE, ATP-BINDING, CELL CYCLE, CELL DIVISION, KINASE, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, CYCLIN, CYTOPLASM, NUCLEUS 
4tye:A   (SER510) to   (GLU752)  STRUCTURAL ANALYSIS OF THE HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 4 KINASE  |   FIBROBLAST GROWTH FACTOR RECEPTOR, KINASE, TRANSFERASE, DOVITINIB, PONATINB, PROTEROS BIOSTRUCTURES GMBH 
4tyi:A   (SER510) to   (VAL750)  STRUCTURAL ANALYSIS OF THE HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 4  |   FIBROBLAST GROWTH FACTOR RECEPTOR, KINASE, TRANSFERASE, DOVITINIB, PONATINB, PROTEROS BIOSTRUCTURES GMBH 
3dtc:A   (THR184) to   (THR405)  CRYSTAL STRUCTURE OF MIXED-LINEAGE KINASE MLK1 COMPLEXED WITH COMPOUND 16  |   MIXED-LINEAGE KINASE, MLK FAMILY, MLK1 AND MLK3 SUBTYPE SELECTIVE INHIBITORS, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, SH3 DOMAIN, TRANSFERASE 
3dtw:A   (SER877) to  (HIS1178)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A BENZISOXAZOLE INHIBITOR  |   ANGIOGENESIS, RECEPTOR TYROSINE KINASE, TRANSFERASE 
3dtw:B   (THR875) to  (LEU1164)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A BENZISOXAZOLE INHIBITOR  |   ANGIOGENESIS, RECEPTOR TYROSINE KINASE, TRANSFERASE 
3orm:A    (PRO50) to   (ASN278)  MYCOBACTERIUM TUBERCULOSIS PKNB KINASE DOMAIN D76A MUTANT  |   STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, KINASE DOMAIN, SIGNAL TRANSDUCTION, TRANSFERASE 
4dce:A  (SER1157) to  (ASP1389)  CRYSTAL STRUCTURE OF HUMAN ANAPLASTIC LYMPHOMA KINASE IN COMPLEX WITH A PIPERIDINE-CARBOXAMIDE INHIBITOR  |   RECEPTOR TYROSINE KINASE, INHIBITOR, NPM-ALK, EML4-ALK, TRANSFERASE- INHIBITOR COMPLEX 
4dce:B  (SER1157) to  (ASP1389)  CRYSTAL STRUCTURE OF HUMAN ANAPLASTIC LYMPHOMA KINASE IN COMPLEX WITH A PIPERIDINE-CARBOXAMIDE INHIBITOR  |   RECEPTOR TYROSINE KINASE, INHIBITOR, NPM-ALK, EML4-ALK, TRANSFERASE- INHIBITOR COMPLEX 
5hcx:A   (SER752) to   (ARG973)  EGFR KINASE DOMAIN MUTANT "TMLR" WITH AZABENZIMIDAZOLE COMPOUND 7  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5hcz:A   (SER752) to   (ARG973)  EGFR KINASE DOMAIN MUTANT "TMLR" WITH 3-AZETIDINYL AZAINDAZOLE COMPOUND 21  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4dg2:E    (ILE85) to   (HIS294)  CRYSTAL STRUCTURE OF MYRISTOYLATED WT CATALYTIC SUBUNIT OF CAMP- DEPENDENT PROTEIN KINASE IN COMPLEX WITH SP20  |   PROTEIN KINASE, MYRISTOYLATED, PHOSPHOTRANSFERASE OF SER/THR, MG, PKI, PKA REGULATORY SUBUNITS, PHOSPHORYLATED ON S139, T197, S338, MYRISTOYLATED ON G1, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4dgg:A   (SER303) to   (TYR519)  C-SRC KINASE DOMAIN IN COMPLEX WITH RM-1-176  |   TYROSINE PROTEIN KINASE, ATP-BINDING, KINASE DOMAIN, TRANSFERASE 
4dgg:B   (PHE307) to   (TYR519)  C-SRC KINASE DOMAIN IN COMPLEX WITH RM-1-176  |   TYROSINE PROTEIN KINASE, ATP-BINDING, KINASE DOMAIN, TRANSFERASE 
4dh3:A    (GLN84) to   (HIS294)  LOW TEMPERATURE X-RAY STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A CATALYTIC SUBUNIT WITH HIGH MG2+, ATP AND IP20  |   PROTEIN, PHOSPHORYLATION, ATP AND PEPTIDIC INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3dzq:A   (THR660) to   (ILE882)  HUMAN EPHA3 KINASE DOMAIN IN COMPLEX WITH INHIBITOR AWL-II- 38.3  |   RECEPTOR TYROSINE KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, MEMBRANE, NUCLEOTIDE BINDING, PHOSPHORYLATION, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE, INHIBITOR-COMPLEX, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN 
5hni:X  (VAL1121) to  (PHE1344)  CRYSTAL STRUCTURE OF CMET WT WITH COMPOUND 3  |   TRANSFERASE 
5hni:Y  (VAL1121) to  (PHE1344)  CRYSTAL STRUCTURE OF CMET WT WITH COMPOUND 3  |   TRANSFERASE 
5hor:A  (VAL1121) to  (PHE1344)  CRYSTAL STRUCTURE OF C-MET-M1250T IN COMPLEX WITH SAR125844.  |   TRANSFERASE, INHIBITOR 
5hzn:C  (MET1038) to  (ILE1263)  STRUCTURE OF NVP-AEW541 IN COMPLEX WITH IGF-1R KINASE  |   INHIBITOR, KINASE, TRANSFERASE 
5hzn:G  (MET1038) to  (ILE1263)  STRUCTURE OF NVP-AEW541 IN COMPLEX WITH IGF-1R KINASE  |   INHIBITOR, KINASE, TRANSFERASE 
4uj9:A    (ILE85) to   (HIS294)  PROTEIN KINASE A IN COMPLEX WITH AN INHIBITOR  |   TRANSFERASE, PKA 
3pj1:A   (GLU439) to   (GLU657)  CRYSTAL STRUCTURE OF BTK KINASE DOMAIN COMPLEXED WITH 3-(2,6-DICHLORO- PHENYL)-7-[4-(2-DIETHYLAMINO-ETHOXY)-PHENYLAMINO]-1-METHYL-3,4- DIHYDRO-1H-PYRIMIDO[4,5-D]PYRIMIDIN-2-ONE  |   HELIX C-IN, DFG-IN, TRANSFERASE, TRANSFERASE-INHIBITOR COMPLEX 
3pj8:A    (PRO45) to   (HIS283)  STRUCTURE OF CDK2 IN COMPLEX WITH A PYRAZOLO[4,3-D]PYRIMIDINE BIOISOSTERE OF ROSCOVITINE.  |   PHOSPHORYLATION, CELL DIVISION, MITOSIS, CYCLIN, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
5i9x:A   (THR653) to   (ALA877)  CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE WITH BOSUTINIB (SKI-606)  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, RECEPTOR, ATP-BINDING 
5i9y:A   (THR653) to   (ALA877)  CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE WITH DASATINIB  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, RECEPTOR, ATP-BINDING 
5i9z:A   (THR653) to   (ALA877)  CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE WITH DANUSERTIB (PHA739358)  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, RECEPTOR, ATP-BINDING 
5ia0:A   (THR653) to   (ALA877)  CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE WITH ALISERTIB (MLN8237)  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, RECEPTOR, ATP-BINDING 
5ia0:B   (THR653) to   (ALA877)  CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE WITH ALISERTIB (MLN8237)  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, RECEPTOR, ATP-BINDING 
5ia0:C   (GLU654) to   (ALA877)  CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE WITH ALISERTIB (MLN8237)  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, RECEPTOR, ATP-BINDING 
5ia1:A   (THR653) to   (ALA877)  CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE WITH MLN8054  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, RECEPTOR, ATP-BINDING 
5ia2:A   (THR653) to   (ALA877)  CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE WITH COMPOUND 66  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, RECEPTOR, ATP-BINDING 
5ia4:A   (THR653) to   (ALA877)  CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE WITH FORETINIB (XL880)  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, RECEPTOR, ATP-BINDING 
5ia5:A   (THR653) to   (ALA877)  CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE WITH GOLVATINIB (E7050)  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, RECEPTOR, ATP-BINDING 
4ebv:A   (ASP462) to   (GLN686)  STRUCTURE OF FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH NOVEL ALLOSTERIC INHIBITOR  |   KINASE DOMAIN, ALLOSTERIC INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ebw:A   (ASP462) to   (GLN686)  STRUCTURE OF FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH NOVEL ALLOSTERIC INHIBITOR  |   KINASE DOMAIN, ALLOSTERIC INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ec8:A    (ILE61) to   (SER317)  STRUCTURE OF FULL LENGTH CDK9 IN COMPLEX WITH CYCLINT AND DRB  |   CYCLIN DEPENDEND KINASE, CYCLIN, TRANSFERASE-PROTEIN BINDING COMPLEX 
3pxf:A    (PRO45) to   (GLN287)  CDK2 IN COMPLEX WITH TWO MOLECULES OF 8-ANILINO-1-NAPHTHALENE SULFONATE  |   PROTEIN KINASE, ALLOSTERIC LIGAND, TRANSFERASE 
3pxk:A   (LEU469) to   (GLN687)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH PYRROLO[2,3- D]THIAZOLE  |   TYROSINE PROTEIN KINASE, TRANSFERASE, ATP BINDING 
3pxk:B   (SER461) to   (GLN687)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH PYRROLO[2,3- D]THIAZOLE  |   TYROSINE PROTEIN KINASE, TRANSFERASE, ATP BINDING 
4ek3:A    (SER46) to   (GLN287)  CRYSTAL STRUCTURE OF APO CDK2  |   ALPHA AND BETA PROTEIN (A+B), TRANSFERASE 
4ek6:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH AMINOPYRAZOLE INHIBITOR  |   ALPHA AND BETA PROTEIN (A+B), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ek8:A    (SER46) to   (GLN287)  CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH THIAZOLYLPYRIMIDINE INHIBITOR  |   ALPHA AND BETA PROTEIN (A+B), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4eok:C    (PRO45) to   (GLN287)  THR 160 PHOSPHORYLATED CDK2 H84S, Q85M, K89D - HUMAN CYCLIN A3 COMPLEX WITH THE INHIBITOR NU6102  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4eor:C    (PRO45) to   (GLN287)  THR 160 PHOSPHORYLATED CDK2 WT - HUMAN CYCLIN A3 COMPLEX WITH THE INHIBITOR NU6102  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4eos:A    (PRO45) to   (HIS283)  THR 160 PHOSPHORYLATED CDK2 WT - HUMAN CYCLIN A3 COMPLEX WITH THE INHIBITOR RO3306  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4eqm:A    (GLU50) to   (VAL270)  STRUCTURAL ANALYSIS OF STAPHYLOCOCCUS AUREUS SERINE/THREONINE KINASE PKNB  |   KINASE, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE 
4eqm:B    (GLU49) to   (VAL270)  STRUCTURAL ANALYSIS OF STAPHYLOCOCCUS AUREUS SERINE/THREONINE KINASE PKNB  |   KINASE, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE 
4eqm:C    (GLU50) to   (VAL270)  STRUCTURAL ANALYSIS OF STAPHYLOCOCCUS AUREUS SERINE/THREONINE KINASE PKNB  |   KINASE, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE 
3q6u:A  (ILE1118) to  (THR1343)  STRUCTURE OF THE APO MET RECEPTOR KINASE IN THE DUALLY-PHOSPHORYLATED, ACTIVATED STATE  |   TYROSINE KINASE, TRANSFERASE 
4uwb:B   (GLU522) to   (LEU760)  FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE IN COMPLEX WITH JK-P5  |   TRANSFERASE 
4uwc:A   (THR521) to   (LEU760)  FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE IN COMPLEX WITH JK-P3  |   TRANSFERASE, RECEPTOR TYROSINE KINASE, TRANSFERASE INHIBITOR 
4uwc:B   (GLU522) to   (LEU760)  FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE IN COMPLEX WITH JK-P3  |   TRANSFERASE, RECEPTOR TYROSINE KINASE, TRANSFERASE INHIBITOR 
5iug:A  (SER1157) to  (ASP1389)  CRYSTAL STRUCTURE OF ANAPLASTIC LYMPHOMA KINASE (ALK) IN COMPLEX WITH 5A  |   CATALYTIC DOMAIN, TRANSFERASE 
5iuh:A  (GLU1158) to  (ASP1389)  CRYSTAL STRUCTURE OF THE ANAPLASTIC LYMPHOMA KINASE (ALK) IN COMPLEX WITH 5D  |   CATALYTIC DOMAIN, TRANSFERASE 
4f0i:A   (SER551) to   (ALA786)  CRYSTAL STRUCTURE OF APO TRKA  |   TYROSINE KINASE, ROSSMANN FOLD, TRANSFERASE 
5izf:A    (GLN84) to   (ALA298)  COMPLEX OF PKA WITH THE BISUBSTRATE PROTEIN KINASE INHIBITOR ARC-1408  |   PROTEIN KINASE, INHIBITOR, BISUBSTRATE, OLIGOARGININE, PKA, TRANSFERASE 
5izj:A    (GLN84) to   (HIS294)  COMPLEX OF PKA WITH THE BISUBSTRATE PROTEIN KINASE INHIBITOR ARC-1411  |   PROTEIN KINASE, INHIBITOR, BISUBSTRATE, OLIGOARGININE, PKA, TRANSFERASE 
5izj:B    (GLN84) to   (HIS294)  COMPLEX OF PKA WITH THE BISUBSTRATE PROTEIN KINASE INHIBITOR ARC-1411  |   PROTEIN KINASE, INHIBITOR, BISUBSTRATE, OLIGOARGININE, PKA, TRANSFERASE 
5j5s:A   (SER303) to   (TYR519)  SRC KINASE IN COMPLEX WITH A SULFONAMIDE INHIBITOR  |   PROTEIN KINASE, INACTIVE KINASE, SULFONAMIDE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4f63:A   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN IN COMPLEX WITH COMPOUND 1  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANS-MEMBRANE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4f63:B   (THR521) to   (LEU760)  CRYSTAL STRUCTURE OF HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN IN COMPLEX WITH COMPOUND 1  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANS-MEMBRANE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4f64:A   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN IN COMPLEX WITH COMPOUND 6  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANS-MEMBRANE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4f64:B   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN IN COMPLEX WITH COMPOUND 6  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANS-MEMBRANE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4f65:A   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN IN COMPLEX WITH COMPOUND 8  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANS-MEMBRANE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4f65:B   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN IN COMPLEX WITH COMPOUND 8  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANS-MEMBRANE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
5j7h:A  (SER1157) to  (ASP1389)  CRYSTAL STRUCTURE OF ANAPLASTIC LYMPHOMA KINASE (ALK) BOUND BY BRIGATINIB  |   RECEPTOR TYROSINE KINASE, SMALL MOLECULE INHIBITOR, TARGETED THERAPY, CANCER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qlg:A   (SER303) to   (TYR519)  CRYSTAL STRUCTURE OF THE L317I MUTANT OF THE C-SRC TYROSINE KINASE DOMAIN COMPLEXED WITH DASATINIB  |   C-SRC L317I MUTANT, TYROSINE KINASE, TRANSFERASE, DASATINIB 
3qlg:B   (SER303) to   (TYR519)  CRYSTAL STRUCTURE OF THE L317I MUTANT OF THE C-SRC TYROSINE KINASE DOMAIN COMPLEXED WITH DASATINIB  |   C-SRC L317I MUTANT, TYROSINE KINASE, TRANSFERASE, DASATINIB 
4uwy:A   (THR521) to   (LEU760)  FGFR1 APO STRUCTURE  |   TRANSFERASE, INHIBITOR, DRUG, CANCER, FGF, RECEPTORS, GROWTH FACTORS, SIGNALLING 
4uwy:B   (THR521) to   (LEU760)  FGFR1 APO STRUCTURE  |   TRANSFERASE, INHIBITOR, DRUG, CANCER, FGF, RECEPTORS, GROWTH FACTORS, SIGNALLING 
4uxq:A   (LYS512) to   (VAL750)  FGFR4 IN COMPLEX WITH PONATINIB  |   TRANSFERASE, KINASE DFG-OUT FGFR INHIBITOR COMPLEX 
4v01:A   (THR521) to   (LEU760)  FGFR1 IN COMPLEX WITH PONATINIB (CO-CRYSTALLISATION).  |   TRANSFERASE 
4v01:B   (GLU522) to   (LEU760)  FGFR1 IN COMPLEX WITH PONATINIB (CO-CRYSTALLISATION).  |   TRANSFERASE 
4v05:A   (THR521) to   (LEU760)  FGFR1 IN COMPLEX WITH AZD4547.  |   TRANSFERASE 
4v05:B   (LYS523) to   (LEU760)  FGFR1 IN COMPLEX WITH AZD4547.  |   TRANSFERASE 
3qqf:A    (SER46) to   (GLN287)  CDK2 IN COMPLEX WITH INHIBITOR L1  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qqh:A    (PRO45) to   (GLN287)  CDK2 IN COMPLEX WITH INHIBITOR L2-2  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qqj:A    (PRO45) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR L2  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qqk:A    (PRO45) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR L4  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qrj:A   (VAL280) to   (MET496)  THE CRYSTAL STRUCTURE OF HUMAN ABL1 KINASE DOMAIN T315I MUTANT IN COMPLEX WITH DCC-2036  |   ABL1, KINASE, KINASE DOMAIN, T315I, GATEKEEPER MUTATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3qrj:B   (VAL280) to   (THR495)  THE CRYSTAL STRUCTURE OF HUMAN ABL1 KINASE DOMAIN T315I MUTANT IN COMPLEX WITH DCC-2036  |   ABL1, KINASE, KINASE DOMAIN, T315I, GATEKEEPER MUTATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3qti:A  (ASP1117) to  (PHE1344)  C-MET KINASE IN COMPLEX WITH NVP-BVU972  |   KINASE, TRANSERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qti:B  (ILE1118) to  (PHE1344)  C-MET KINASE IN COMPLEX WITH NVP-BVU972  |   KINASE, TRANSERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qtq:A    (SER46) to   (GLN287)  CDK2 IN COMPLEX WITH INHIBITOR RC-1-137  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qtr:A    (ALA48) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR RC-1-148  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qwj:A    (PRO45) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR KVR-1-142  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qx2:A    (SER46) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR KVR-1-190  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qx4:A    (PRO45) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR KVR-1-78  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fic:A   (ALA311) to   (TYR519)  KINASE DOMAIN OF CSRC IN COMPLEX WITH A HINGE REGION-BINDING FRAGMENT  |   HINGE BINDING FRAGMENT, TYPE I, DFG-IN, TYROSINE-PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qzf:A    (PRO45) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR JWS-6-52  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3r1y:A    (SER46) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR KVR-1-134  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fkg:A    (SER46) to   (GLN287)  CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH AMINOPYRAZOLE INHIBITOR  |   ALPHA AND BETA PROTEIN (A+B), TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fki:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH AMINOPYRAZOLE INHIBITOR  |   ALPHA AND BETA PROTEIN (A+B), TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fkl:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH THIAZOLYLPYRIMIDINE INHIBITOR  |   ALPHA AND BETA PROTEIN (A+B), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fkq:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH OXINDOLE INHIBITOR  |   ALPHA AND BETA PROTEIN (A+B), TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fkw:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH OXINDOLE INHIBITOR  |   ALPHA AND BETA PROTEIN (A+B), TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5j9z:A   (SER752) to   (ARG973)  EGFR-T790M IN COMPLEX WITH PYRAZOLOPYRIMIDINE INHIBITOR 1A  |   TYROSINE KINASE, COVALENT INHIBITOR, DRUG RESISTANCE, TRANSFERASE 
3r71:A    (SER46) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR KVR-1-162  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3r7i:A    (SER46) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR KVR-1-74  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3r7y:A    (PRO45) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR KVR-2-88  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3r83:A    (SER46) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR KVR-2-92  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3r8m:A    (ILE49) to   (GLN287)  CDK2 IN COMPLEX WITH INHIBITOR L3-3  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3r8p:A    (SER46) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR NSK-MC1-6  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3r8z:A    (SER46) to   (GLN287)  CDK2 IN COMPLEX WITH INHIBITOR RC-1-136  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3r9o:A    (SER46) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR RC-2-143  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fnx:A  (SER1157) to  (ASP1389)  CRYSTAL STRUCTURE OF THE APO R1275Q ANAPLASTIC LYMPHOMA KINASE CATALYTIC DOMAIN  |   RECEPTOR TYROSINE KINASE, INHIBITOR, CRIZOTINIB, NEUROBLASTOMA, CD246, PHOSPHOTRANSFERASE, NPM-ALK, EML4-ALK, TRANSFERASE 
4fny:A  (SER1157) to  (ASP1389)  CRYSTAL STRUCTURE OF THE R1275Q ANAPLASTIC LYMPHOMA KINASE CATALYTIC DOMAIN IN COMPLEX WITH A BENZOXAZOLE INHIBITOR  |   RECEPTOR TYROSINE KINASE, INHIBITOR, CRIZOTINIB, NEUROBLASTOMA, CD246, PHOSPHOTRANSFERASE, NPM-ALK, EML4-ALK, TRANSFERASE-INHIBITOR COMPLEX 
4fnz:A  (GLN1159) to  (ASP1389)  CRYSTAL STRUCTURE OF HUMAN ANAPLASTIC LYMPHOMA KINASE IN COMPLEX WITH PIPERIDINE-CARBOXAMIDE INHIBITOR 2  |   RECEPTOR TYROSINE KINASE, INHIBITOR, CRIZOTINIB, NEUROBLASTOMA, CD246, PHOSPHOTRANSFERASE, NPM-ALK, EML4-ALK, TRANSFERASE-INHIBITOR COMPLEX 
3rcd:A   (LYS762) to   (PRO983)  HER2 KINASE DOMAIN COMPLEXED WITH TAK-285  |   KINASE DOMAIN, RECEPTOR, TRANSFERASE, TYROSINE-PROTEIN KINASE, TYROSINE KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, ANTI-ONCOGENE, CELL CYCLE, DISEASE, MUTATION, ATP-BINDING, NUCLEOTIDE-BINDING, GLYCOPROTEIN, PHOSPHOPROTEIN, MEMBRANE, SECRETED 
3rcd:B   (LYS762) to   (PRO983)  HER2 KINASE DOMAIN COMPLEXED WITH TAK-285  |   KINASE DOMAIN, RECEPTOR, TRANSFERASE, TYROSINE-PROTEIN KINASE, TYROSINE KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, ANTI-ONCOGENE, CELL CYCLE, DISEASE, MUTATION, ATP-BINDING, NUCLEOTIDE-BINDING, GLYCOPROTEIN, PHOSPHOPROTEIN, MEMBRANE, SECRETED 
3rcd:D   (LYS762) to   (PRO983)  HER2 KINASE DOMAIN COMPLEXED WITH TAK-285  |   KINASE DOMAIN, RECEPTOR, TRANSFERASE, TYROSINE-PROTEIN KINASE, TYROSINE KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, ANTI-ONCOGENE, CELL CYCLE, DISEASE, MUTATION, ATP-BINDING, NUCLEOTIDE-BINDING, GLYCOPROTEIN, PHOSPHOPROTEIN, MEMBRANE, SECRETED 
5jkg:A   (ASP513) to   (LEU748)  THE CRYSTAL STRUCTURE OF FGFR4 KINASE DOMAIN IN COMPLEX WITH LY2874455  |   KINASE, SMALL-MOLECULE INHIBITOR, ATP BINDING POCKET, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3rhx:B   (LYS523) to   (LEU760)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF FGFR1 KINASE IN COMPLEX WITH ARQ 069  |   FGFR1 KINASE, FGFR2 KINASE, INACTIVE CONFORMATION, KINASE-INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3rhx:A   (GLU522) to   (LEU760)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF FGFR1 KINASE IN COMPLEX WITH ARQ 069  |   FGFR1 KINASE, FGFR2 KINASE, INACTIVE CONFORMATION, KINASE-INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ri1:A   (THR524) to   (THR765)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF FGFR2 KINASE IN COMPLEX WITH ARQ 069  |   FGFR1 KINASE, FGFR2 KINASE, INACTIVE CONFORMATION, KINASE-INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ri1:B   (THR524) to   (ASN766)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF FGFR2 KINASE IN COMPLEX WITH ARQ 069  |   FGFR1 KINASE, FGFR2 KINASE, INACTIVE CONFORMATION, KINASE-INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5jrs:A   (GLU439) to   (ASP656)  CRYSTAL STRUCTURE OF BRUTON AGAMMAGLOBULINEMIA TYROSINE KINASE COMPLEXED WITH 4-[2-FLUORO-3-(4-OXO -3,4-DIHYDROQUINAZOLIN-3-YL) PHENYL]-7-(2-HYDROXYPROPAN-2-Y L)-9H-CARBAZOLE-1-CARBOXAMIDE  |   KINASE, BTK, PROTEIN INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5jsm:D   (THR491) to   (LEU721)  BRAFV600E KINASE DOMAIN IN COMPLEX WITH CHEMICALLY LINKED VEMURAFENIB INHIBITOR VEM-3-VEM  |   KINASE, DIMER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4g2f:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE DOMAIN IN COMPLEX WITH COMPOUND 7  |   RECEPTOR TYROSINE KINASE, ATP BINDING, PHOSPHORYLATION, MEMBRANE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5k4j:A    (SER46) to   (GLN287)  CRYSTAL STRUCTURE OF CDK2 IN COMPLEX WITH COMPOUND 22  |   PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4gk2:A   (THR660) to   (ARG883)  HUMAN EPHA3 KINASE DOMAIN IN COMPLEX WITH LIGAND 66  |   RECEPTOR TYROSINE KINASE, ATP-BINDING, PHOSPHORYLATION, MEMBRANE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4gk3:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE DOMAIN IN COMPLEX WITH LIGAND 87  |   RECEPTOR TYROSINE KINASE, ATP-BINDING, PHOSPHORYLATION, MEMBRANE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4gk4:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE DOMAIN IN COMPLEX WITH LIGAND 90  |   RECEPTOR TYROSINE KINASE, ATP-BINDING, PHOSPHORYLATION, MEMBRANE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5l6o:A   (THR672) to   (ASN898)  EPHB3 KINASE DOMAIN COVALENTLY BOUND TO AN IRREVERSIBLE INHIBITOR (COMPOUND 3)  |   KINASE, IRREVERSIBLE INHIBITOR, QUINAZOLINE, SIGNALING, TRANSFERASE 
5l6p:A   (THR672) to   (ASN898)  EPHB3 KINASE DOMAIN COVALENTLY BOUND TO AN IRREVERSIBLE INHIBITOR (COMPOUND 6)  |   KINASE, IRREVERSIBLE INHIBITOR, QUINAZOLINE, SIGNALING, TRANSFERASE 
5loh:B    (LYS65) to   (HIS832)  KINASE DOMAIN OF HUMAN GREATWALL  |   KINASE DOMAIN, INHIBITOR, TRANSFERASE 
5t3q:A  (ILE1118) to  (ARG1336)  CRYSTAL STRUCTURE OF THE C-MET KINASE DOMAIN IN COMPLEX WITH A PYRAZOLONE INHIBITOR  |   PHOSPHOTRANSFERASE, CANCER, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3rpo:A    (PRO45) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR KVR-1-156  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2ojf:E    (ILE85) to   (ALA298)  CRYSTAL STRUCTURE OF PROTEIN KINASE A IN COMPLEX WITH PYRIDINE-PYRAZOLOPYRIDINE BASED INHIBITORS  |   PROTEIN KINASE A, AKT, TRANSFERASE 
3el7:A   (SER303) to   (TYR519)  CRYSTAL STRUCTURE OF C-SRC IN COMPLEX WITH PYRAZOLOPYRIMIDINE 3  |   KINASE, C-SRC, PYRAZOLOPYRIMIDINE, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
2p0c:B   (SER636) to   (LEU861)  CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE-PROTEIN KINASE MER  |   ATP-BINDING, DISEASE MUTATION, GLYCOPROTEIN, KINASE, NUCLEOTIDE- BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, RECEPTOR, RETINITIS PIGMENTOSA, SENSORY TRANSDUCTION, TRANSFERASE, TYROSINE-PROTEIN KINASE, VISION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC 
2p2h:A   (THR875) to  (ASP1171)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A PYRIDINYL-TRIAZINE INHIBITOR  |   RECEPTOR TYROSINE KINASE, KDR, TRANSFERASE 
1b39:A    (PRO45) to   (HIS283)  HUMAN CYCLIN-DEPENDENT KINASE 2 PHOSPHORYLATED ON THR 160  |   PROTEIN KINASE, TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, ATP-BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, PHOSPHORYLATION 
2bdf:A   (SER303) to   (TYR519)  SRC KINASE IN COMPLEX WITH INHIBITOR AP23451  |   SRC KINASE INHIBITOR, TRANSFERASE 
4hw7:A   (ALA624) to   (ALA914)  CRYSTAL STRUCTURE OF FMS KINASE DOMAIN WITH A SMALL MOLECULAR INHIBITOR, PLX647-OME  |   CSF-1-R, FMS PROTO-ONCOGENE, C-FMS, CD115 ANTIGEN, KINASE, ATP- BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4xcu:A   (SER510) to   (ALA749)  CRYSTAL STRUCTURE OF FGFR4 WITH AN IRREVERSIBLE INHIBITOR  |   RECEPTOR TYROSINE KINASE, HEPATOCELLULAR CARCINOMA, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
1ogu:A    (PRO45) to   (GLN287)  STRUCTURE OF HUMAN THR160-PHOSPHO CDK2/CYCLIN A COMPLEXED WITH A 2-ARYLAMINO-4-CYCLOHEXYLMETHYL-5-NITROSO-6-AMINOPYRIMIDINE INHIBITOR  |   KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP- BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, PHOSPHORYLATION 
3fhr:A    (SER78) to   (HIS301)  HIGH RESOLUTION CRYSTAL STRUCTURE OF MITOGEN-ACTIVATED PROTEIN KINASE- ACTIVATED PROTEIN KINASE 3 (MK3)-INHIBITOR COMPLEX  |   KINASE-INHIBITOR COMPLEX, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
1oir:A    (THR47) to   (GLN287)  IMIDAZOPYRIDINES: A POTENT AND SELECTIVE CLASS OF CYCLIN-DEPENDENT KINASE INHIBITORS IDENTIFIED THROUGH STRUCTURE-BASED HYBRIDISATION  |   KINASE, PROTEIN KINASE 
2psq:B   (THR524) to   (ASN766)  CRYSTAL STRUCTURE OF UNPHOSPHORYLATED UNACTIVATED WILD TYPE FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN  |   KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, TRANSFERASE 
2ptk:A   (PHE307) to   (TYR519)  CHICKEN SRC TYROSINE KINASE  |   TYROSINE-PROTEIN KINASE, SRC, SH2, SH3 
2c6i:A    (PRO45) to   (GLN287)  CRYSTAL STRUCTURE OF THE HUMAN CDK2 COMPLEXED WITH THE TRIAZOLOPYRIMIDINE INHIBITOR  |   TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, CDK2, ATP-BINDING, CELL CYCLE, MITOSIS, PHOSPHORYLATION, TRIAZOLOPYRIMIDINE INHIBITOR, CELL DIVISION, KINASE, POLYMORPHISM, NUCLEOTIDE-BINDING 
3fy2:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE AND JUXTAMEMBRANE REGION BOUND TO SUBSTRATE KQWDNYEFIW  |   RECEPTOR TYROSINE KINASE, JUXTAMEMBRANE SEGMENT, STRUCTURAL GENOMICS, PEPTIDE CO-CRYSTAL STRUCTURE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, CELL MEMBRANE, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3fzo:A   (THR464) to   (MET691)  CRYSTAL STRUCTURE OF PYK2-APO, PROLINE-RICH TYROSINE KINASE  |   TYROSINE KINASE, DFG-OUT, ALTERNATIVE SPLICING, ATP-BINDING, CELL MEMBRANE, CYTOPLASM, KINASE, MEMBRANE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TYROSINE-PROTEIN KINASE 
2qi8:B   (GLU310) to   (TYR519)  CRYSTAL STRUCTURE OF DRUG RESISTANT SRC KINASE DOMAIN  |   SRC KINASE DOMAIN; DRUG RESISTANCE, SIGNALING PROTEIN, TRANSFERASE 
2qo7:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE AND JUXTAMEMBRANE REGION, DEPHOSPHORYLATED, AMP-PNP BOUND  |   RECEPTOR TYROSINE KINASE, JUXTAMEMBRANE SEGMENT, STRUCTURAL GENOMICS, AMP-PNP, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
2qo9:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE AND JUXTAMEMBRANE REGION, PHOSPHORYLATED, AMP-PNP BOUND  |   RECEPTOR TYROSINE KINASE, JUXTAMEMBRANE SEGMENT, STRUCTURAL GENOMICS, AMP-PNP, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP- BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
4ith:A    (ALA59) to   (GLU269)  CRYSTAL STRUCTURE OF RIP1 KINASE IN COMPLEX WITH NECROSTATIN-1 ANALOG  |   ALPHA/BETA, RIP1 KINASE, NECROPTOSIS, NECROSTATINS, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ith:B    (ASN57) to   (LYS284)  CRYSTAL STRUCTURE OF RIP1 KINASE IN COMPLEX WITH NECROSTATIN-1 ANALOG  |   ALPHA/BETA, RIP1 KINASE, NECROPTOSIS, NECROSTATINS, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2qu5:A   (THR875) to  (GLN1170)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A BENZIMIDAZOLE INHIBITOR  |   RECEPTOR TYROSINSE KINASE, KDR, ANGIOGENESIS, ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST- VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
1pw2:A    (SER46) to   (HIS283)  APO STRUCTURE OF HUMAN CYCLIN-DEPENDENT KINASE 2  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, 3D-STRUCTURE. 
2r3k:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE, INHIBITION, CYCLIN-DEPENDENT KINASE, CANCER, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE 
2r3n:A    (PRO45) to   (HIS283)  CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE, INHIBITION, CYCLIN-DEPENDENT KINASE, CANCER, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE 
1pye:A    (ALA48) to   (GLN287)  CRYSTAL STRUCTURE OF CDK2 WITH INHIBITOR  |   CDK, CYCLIN-DEPENDENT KINASE 2, TRANSFERASE 
1q8t:A    (ILE85) to   (ALA298)  THE CATALYTIC SUBUNIT OF CAMP-DEPENDENT PROTEIN KINASE (PKA) IN COMPLEX WITH RHO-KINASE INHIBITOR Y-27632  |   KINASE-INHIBITOR-COMPLEX, PHOSPHOTRANSFERASE/INHIBITOR, CAMP, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, ATP- BINDING, PKA, RHO-KINASE, TRANSFERASE/TRANSFERASE INHIBITOR COMPLEX 
2rfd:A   (ALA731) to   (ARG949)  CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN THE EGFR KINASE DOMAIN AND A MIG6 PEPTIDE  |   KINASE DOMAIN, INHIBITION, DIMER, PEPTIDE, ALTERNATIVE SPLICING, ANTI-ONCOGENE, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, UBL CONJUGATION, CYTOPLASM 
2rfd:B   (ALA731) to   (ARG949)  CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN THE EGFR KINASE DOMAIN AND A MIG6 PEPTIDE  |   KINASE DOMAIN, INHIBITION, DIMER, PEPTIDE, ALTERNATIVE SPLICING, ANTI-ONCOGENE, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, UBL CONJUGATION, CYTOPLASM 
3tub:A   (ALA412) to   (VAL633)  CRYSTAL STRUCTURE OF SYK KINASE DOMAIN WITH 1-(5-(6,7- DIMETHOXYQUINOLIN-4-YLOXY)PYRIDIN-2-YL)-3-((1R,2S)-2- PHENYLCYCLOPROPYL)UREA  |   KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2rl5:A   (THR875) to  (ARG1172)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A 2,3-DIHYDRO-1,4-BENZOXAZINE INHIBITOR  |   RECEPTOR TYROSINE KINASE, ANGIOGENESIS, , ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST- VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3u6h:A  (ILE1118) to  (ARG1336)  CRYSTAL STRUCTURE OF C-MET IN COMPLEX WITH PYRAZOLONE INHIBITOR 26  |   KINASE DOMAIN, PHOSPHOTRANSFERASE, CANCER, HEPATOCYTE GROWTH FACTOR, HGF, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1r1w:A  (ILE1118) to  (ARG1336)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF THE HEPATOCYTE GROWTH FACTOR RECEPTOR C-MET  |   RECEPTOR TYROSINE KINASE, SIGNAL TRANSDUCTION, GRB2, SHC, TRANSFERASE 
2v0d:A    (PRO45) to   (GLN287)  CRYSTAL STRUCTURE OF HUMAN CDK2 COMPLEXED WITH A THIAZOLIDINONE INHIBITOR  |   PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE, ATP-BINDING, CELL DIVISION, NUCLEOTIDE- BINDING, THIAZOLIDINONE LIGAND, CDK2, KINASE, CYCLIN, MITOSIS, CELL CYCLE 
2exm:A    (SER46) to   (GLN287)  HUMAN CDK2 IN COMPLEX WITH ISOPENTENYLADENINE  |   TYPICAL PROTEIN KINASE FOLD, LIGAND BINDING POCKET BETWEEN N-TERMINAL AND C-TERMINAL DOMAIN, TRANSFERASE 
3uvr:A    (SER61) to   (GLN260)  HUMAN P38 MAP KINASE IN COMPLEX WITH KM064  |   PROTEIN KINASE, SELECTIVE P38 INHIBITOR, SAR, ANNULEN DERIVATIVE, PYRAZOLO UREA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3v5l:A   (ASP402) to   (ALA616)  CRYSTAL STRUCTURE OF INTERLEUKIN-2 INDUCIBLE T-CELL KINASE ITK CATALYTIC DOMAIN WITH THIENOPYRAZOLYLINDOLE INHIBITOR 542  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3v5l:B   (GLU400) to   (SER618)  CRYSTAL STRUCTURE OF INTERLEUKIN-2 INDUCIBLE T-CELL KINASE ITK CATALYTIC DOMAIN WITH THIENOPYRAZOLYLINDOLE INHIBITOR 542  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3v5l:C   (SER399) to   (ALA616)  CRYSTAL STRUCTURE OF INTERLEUKIN-2 INDUCIBLE T-CELL KINASE ITK CATALYTIC DOMAIN WITH THIENOPYRAZOLYLINDOLE INHIBITOR 542  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3v5l:D   (SER399) to   (SER618)  CRYSTAL STRUCTURE OF INTERLEUKIN-2 INDUCIBLE T-CELL KINASE ITK CATALYTIC DOMAIN WITH THIENOPYRAZOLYLINDOLE INHIBITOR 542  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3v5q:A   (THR578) to   (THR831)  DISCOVERY OF A SELECTIVE TRK INHIBITOR WITH EFFICACY IN RODENT CANCER TUMOR MODELS  |   KINASE DOMAIN, KINASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2vto:A    (SER46) to   (GLN287)  IDENTIFICATION OF N-(4-PIPERIDINYL)-4-(2,6- DICHLOROBENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXAMIDE (AT7519), A NOVEL CYCLIN DEPENDENT KINASE INHIBITOR USING FRAGMENT- BASED X-RAY CRYSTALLOGRAPHY AND STRUCTURE BASED DRUG DESIGN.  |   TRANSFERASE, MITOSIS, CELL CYCLE, SERINE/THREONINE PROTEIN KINASE 
2vtp:A    (SER46) to   (HIS283)  IDENTIFICATION OF N-(4-PIPERIDINYL)-4-(2,6- DICHLOROBENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXAMIDE (AT7519), A NOVEL CYCLIN DEPENDENT KINASE INHIBITOR USING FRAGMENT- BASED X-RAY CRYSTALLOGRAPHY AND STRUCTURE BASED DRUG DESIGN.  |   TRANSFERASE, MITOSIS, CELL CYCLE, SERINE/THREONINE PROTEIN KINASE 
2vtq:A    (SER46) to   (GLN287)  IDENTIFICATION OF N-(4-PIPERIDINYL)-4-(2,6- DICHLOROBENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXAMIDE (AT7519), A NOVEL CYCLIN DEPENDENT KINASE INHIBITOR USING FRAGMENT- BASED X-RAY CRYSTALLOGRAPHY AND STRUCTURE BASED DRUG DESIGN.  |   TRANSFERASE, MITOSIS, CELL CYCLE, SERINE/THREONINE PROTEIN KINASE 
1gy3:C    (PRO45) to   (GLN287)  PCDK2/CYCLIN A IN COMPLEX WITH MGADP, NITRATE AND PEPTIDE SUBSTRATE  |   TRANSFERASE-TRANSFERASE SUBSTRATE COMPLEX, CELL CYCLE REGULATORY PROTEIN KINASE, THR160-PHOSPHO-CYCLIN DEPENDENT PROTEIN KINASE 2 IN ASSOCIATION WITH CYCLIN A, TRANSFERASE- TRANSFERASE SUBSTRATE COMPLEX 
1t46:A   (LEU631) to   (SER931)  STRUCTURAL BASIS FOR THE AUTOINHIBITION AND STI-571 INHIBITION OF C-KIT TYROSINE KINASE  |   KINASE, STRUCTURE, INHIBITOR, STI-571, GLEEVEC, TRANSFERASE ACTIVATOR 
2gnl:A    (ILE85) to   (HIS294)  PKA THREEFOLD MUTANT MODEL OF RHO-KINASE WITH INHIBITOR H- 1152P  |   PKA, MUTANT, RHO-KINASE, SURROGATE, INHIBITOR, H-1152P, TRANSFERASE/TRANSFERASE INHIBITOR COMPLEX 
2w1g:A   (VAL174) to   (HIS380)  STRUCTURE DETERMINATION OF AURORA KINASE IN COMPLEX WITH INHIBITOR  |   CANCER, AURORA, KINASE, INHIBITOR, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, POLYMORPHISM, PHOSPHOPROTEIN, CELL CYCLE 
2gu8:A    (GLN84) to   (ALA298)  DISCOVERY OF 2-PYRIMIDYL-5-AMIDOTHIOPHENES AS NOVEL AND POTENT INHIBITORS FOR AKT: SYNTHESIS AND SAR STUDIES  |   CAMP-DEPENDENT PROTEIN KINASE, PKA, AKT, KINASE, DRUG DESIGN, TERNARY COMPLEX, SIGNALING PROTEIN, TRANSFERASE/INHIBITOR COMPLEX 
4lg4:E    (LEU64) to   (HIS275)  STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5  |   HIPPO, MST AUTOACTIVATION, DIMERIZATION, SIGNALING PROTEIN 
3vnt:A   (HIS876) to  (ALA1168)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN VEGFR2 WITH A [1, 3]THIAZOLO[5,4-B]PYRIDINE DERIVATIVE  |   VEGFR2, KINASE DOMAIN, TYROSIN-PROTEIN KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
5am7:A   (LYS523) to   (LEU760)  FGFR1 MUTANT WITH AN INHIBITOR  |   TRANSFERASE, FGFR, CANCER, DOVITINIB, TKI258, GATEKEEPER, GATE KEEPER 
5am7:B   (GLU522) to   (LEU760)  FGFR1 MUTANT WITH AN INHIBITOR  |   TRANSFERASE, FGFR, CANCER, DOVITINIB, TKI258, GATEKEEPER, GATE KEEPER 
1jpa:A   (THR668) to   (ASN894)  CRYSTAL STRUCTURE OF UNPHOSPHORYLATED EPHB2 RECEPTOR TYROSINE KINASE AND JUXTAMEMBRANE REGION  |   RECEPTOR TYROSINE KINASE, AUTOINHIBITED, UNPHOSPHORYLATED, JUXTAMEMBRANE, TRANSFERASE 
1jpa:B   (THR668) to   (ASN894)  CRYSTAL STRUCTURE OF UNPHOSPHORYLATED EPHB2 RECEPTOR TYROSINE KINASE AND JUXTAMEMBRANE REGION  |   RECEPTOR TYROSINE KINASE, AUTOINHIBITED, UNPHOSPHORYLATED, JUXTAMEMBRANE, TRANSFERASE 
2xir:A   (HIS876) to  (ALA1168)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH PF-00337210 (N,2-DIMETHYL-6-(7-(2-MORPHOLINOETHOXY) QUINOLIN-4-YLOXY)BENZOFURAN-3-CARBOXAMIDE)  |   ANGIOGENESIS, NUCLEOTIDE-BINDING, INHIBITOR, PHOSPHORYLATION, RECEPTOR, TRANSFERASE, TRANSMEMBRANE 
5ax9:B    (GLU64) to   (HIS286)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN TRAF2 AND NCK- INTERACTING PROTEIN KINASE IN COMPLEX WITH COMPUND 9  |   INHIBITOR, KINASE, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4mxy:A   (GLU310) to   (TYR519)  SRC M314L T338M DOUBLE MUTANT BOUND TO KINASE INHIBITOR BOSUTINIB  |   KINASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1w0x:C    (PRO45) to   (HIS283)  CRYSTAL STRUCTURE OF HUMAN CDK2 IN COMPLEX WITH THE INHIBITOR OLOMOUCINE.  |   PROTEIN KINASE INHIBITORS, CYCLIN-DEPENDENT KINASE, CELL CYCLE REGULATION, CANCER, TRANSFERASE, SERINE/THREONINE - PROTEIN KINASE, ATP-BINDING 
3zbx:A  (ASP1117) to  (THR1343)  X-RAY STRUCTURE OF C-MET KINASE IN COMPLEX WITH INHIBITOR 6- ((6-(4-FLUOROPHENYL)-(1,2,4)TRIAZOLO(4,3-B)(1,2,4)TRIAZIN- 3-YL)METHYL)QUINOLINE.  |   TRANSFERASE, INHIBITOR 
2jkk:A   (SER463) to   (GLU683)  FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH BIS- ANILINO PYRIMIDINE INHIBITOR  |   TYROSINE-PROTEIN KINASE, TYROSINE- PROTEIN KINASE, KINASE, MEMBRANE, TRANSFERASE, ATP-BINDING, INTEGRIN SIGNALING, NUCLEOTIDE-BINDING, FOCAL ADHESION, CELL MIGRATION, KINASE INHIBITOR, CELL JUNCTION, CELL MEMBRANE, PHOSPHOPROTEIN 
1ke6:A    (SER46) to   (GLN287)  CYCLIN-DEPENDENT KINASE 2 (CDK2) COMPLEXED WITH N-METHYL-{4- [2-(7-OXO-6,7-DIHYDRO-8H-[1,3]THIAZOLO[5,4-E]INDOL-8- YLIDENE)HYDRAZINO]PHENYL}METHANESULFONAMIDE  |   CYCLIN, KINASE, TRANSFERASE 
3js2:A   (THR521) to   (LEU760)  CRYSTAL STRUCTURE OF MINIMAL KINASE DOMAIN OF FIBROBLAST GROWTH FACTOR RECEPTOR 1 IN COMPLEX WITH 5-(2-THIENYL) NICOTINIC ACID  |   FIBROBLAST GROWTH FACTOR, RECEPTOR TYROSINE KINASE, INHIBITOR, THIENYL NICOTINIC ACID, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, DWARFISM, GLYCOPROTEIN, HEPARIN-BINDING, HYPOGONADOTROPIC HYPOGONADISM, IMMUNOGLOBULIN DOMAIN, KALLMANN SYNDROME, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3js2:B   (LYS523) to   (THR761)  CRYSTAL STRUCTURE OF MINIMAL KINASE DOMAIN OF FIBROBLAST GROWTH FACTOR RECEPTOR 1 IN COMPLEX WITH 5-(2-THIENYL) NICOTINIC ACID  |   FIBROBLAST GROWTH FACTOR, RECEPTOR TYROSINE KINASE, INHIBITOR, THIENYL NICOTINIC ACID, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, DWARFISM, GLYCOPROTEIN, HEPARIN-BINDING, HYPOGONADOTROPIC HYPOGONADISM, IMMUNOGLOBULIN DOMAIN, KALLMANN SYNDROME, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
1xh5:A    (ILE85) to   (ALA298)  CRYSTAL STRUCTURES OF PROTEIN KINASE B SELECTIVE INHIBITORS IN COMPLEX WITH PROTEIN KINASE A AND MUTANTS  |   PKA, KINASE-INHIBITOR-COMPLEX, SERINE/THREONINE-PROTEIN KINASE, BALANOL DERIVATIVE, TRANSFERASE/TRANSFERASE INHIBITOR COMPLEX 
5clr:B   (ALA110) to   (GLN315)  CRYSTAL STRUCTURE OF LEGK4_APO KINASE  |   LEGIONELLA, BACTERIAL EFFECTORS, SERINE/THREONINE KINASE, TYPE IV SECRETION SYSTEM, TRANSFERASE 
5cwz:A    (GLU62) to   (HIS286)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN TRAF2 AND NCK- INTERACTING PROTEIN KINASE  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5d41:A   (SER752) to   (ARG973)  EGFR KINASE DOMAIN IN COMPLEX WITH MUTANT SELECTIVE ALLOSTERIC INHIBITOR  |   ALLOSTERIC INHIBITOR, EGFR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5d41:B   (SER752) to   (ARG973)  EGFR KINASE DOMAIN IN COMPLEX WITH MUTANT SELECTIVE ALLOSTERIC INHIBITOR  |   ALLOSTERIC INHIBITOR, EGFR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4p5q:A   (THR660) to   (ASN884)  HUMAN EPHA3 KINASE DOMAIN IN COMPLEX WITH QUINOXALINE DERIVATIVES  |   TRANSFERASE, TRANSFERASE INHIBITOR 
1mq4:A   (HIS176) to   (ASN386)  CRYSTAL STRUCTURE OF AURORA-A PROTEIN KINASE  |   PROTEIN KINASE STRUCTURE, TRANSFERASE 
5d7a:B    (GLU62) to   (HIS286)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF TRAF2 AND NCK-INTERACTING PROTEIN KINASE WITH NCB-0846  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3krl:A   (ASP625) to   (GLU912)  CFMS TYROSINE KINASE IN COMPLEX WITH 5-CYANO-FURAN-2-CARBOXYLIC ACID [4-(4-METHYL-PIPERAZIN-1-YL)-2-PIPERIDIN-1-YL-PHENYL]-AMIDE  |   KINASE, INHIBITOR, CHIMERA, ATP-BINDING, DISULFIDE BOND, GLYCOPROTEIN, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3l9n:A    (GLN84) to   (ALA298)  CRYSTAL STRUCTURE OF PKAB3 (PKA TRIPLE MUTANT V123A, L173M, Q181K) WITH COMPOUND 27  |   PKB, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4asd:A   (HIS876) to  (ASN1167)  CRYSTAL STRUCTURE OF VEGFR2 (JUXTAMEMBRANE AND KINASE DOMAINS) IN COMPLEX WITH SORAFENIB (BAY 43-9006)  |   ANGIOGENESIS, NUCLEOTIDE-BINDING, INHIBITOR, PHOSPHORYLATION, RECEPTOR, TRANSFERASE, KDR 
4q9s:A   (ARG465) to   (GLN686)  CRYSTAL STRUCTURE OF HUMAN FOCAL ADHESION KINASE (FAK) BOUND TO COMPOUND1 (3,5-DIHYDRO[1,2,4]TRIAZINO[3,4-C][1,4]BENZOXAZIN-2(1H)- ONE)  |   KINASE CATALYTIC DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3m11:A   (VAL174) to   (HIS380)  CRYSTAL STRUCTURE OF AURORA A KINASE COMPLEXED WITH INHIBITOR  |   AURORA KINASE INHIBITOR, X-RAY CO-CRYSTAL ANALYSIS, STRUCTURE-BASED DRUG DESIGN, ATP-BINDING, CELL CYCLE, CYTOSKELETON, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4bcf:A    (PRO60) to   (SER317)  STRUCTURE OF CDK9 IN COMPLEX WITH CYCLIN T AND A 2-AMINO-4- HETEROARYL-PYRIMIDINE INHIBITOR  |   TRANSFERASE-CELL CYCLE COMPLEX, CDK-CYCLIN COMPLEX, TRANSCRIPTION-PROTEIN BINDING, STRUCTURE-BASED DRUG DESIGN 
4bcm:A    (PRO45) to   (GLN287)  STRUCTURE OF CDK2 IN COMPLEX WITH CYCLIN A AND A 2-AMINO-4- HETEROARYL-PYRIMIDINE INHIBITOR  |   TRANSFERASE-CELL CYCLE COMPLEX, CDK-CYCLIN COMPLEX, STRUCTURE-BASED DRUG DESIGN 
4bcm:C    (PRO45) to   (GLN287)  STRUCTURE OF CDK2 IN COMPLEX WITH CYCLIN A AND A 2-AMINO-4- HETEROARYL-PYRIMIDINE INHIBITOR  |   TRANSFERASE-CELL CYCLE COMPLEX, CDK-CYCLIN COMPLEX, STRUCTURE-BASED DRUG DESIGN 
3miy:B   (SER399) to   (GLY619)  X-RAY CRYSTAL STRUCTURE OF ITK COMPLEXED WITH SUNITINIB  |   HELIX C-IN, TRANSFERASE 
3be2:A   (THR875) to  (GLN1170)  CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH A BENZAMIDE INHIBITOR  |   ANGIOGENESIS, RECEPTOR TYROSINE KINASE, ATP-BINDING, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, GLYCOPROTEIN, HOST- VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
4bgh:A    (SER46) to   (HIS283)  CRYSTAL STRUCTURE OF CDK2 IN COMPLEX WITH PAN-CDK INHIBITOR  |   TRANSFERASE 
3bhu:C    (PRO45) to   (GLN287)  STRUCTURE OF PHOSPHORYLATED THR160 CDK2/CYCLIN A IN COMPLEX WITH THE INHIBITOR MERIOLIN 5  |   SER/THR PROTEIN KINASE, TRANSFERASE, PHOSPHORYLATION, CELL CYCLE, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, CYCLIN 
3bhv:C    (PRO45) to   (GLN287)  STRUCTURE OF PHOSPHORYLATED THR160 CDK2/CYCLIN A IN COMPLEX WITH THE INHIBITOR VARIOLIN B  |   SER/THR PROTEIN KINASE, TRANSFERASE, PHOSPHORYLATION, CELL CYCLE, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE- PROTEIN KINASE, CYCLIN 
3bhy:A    (SER57) to   (HIS272)  CRYSTAL STRUCTURE OF HUMAN DEATH ASSOCIATED PROTEIN KINASE 3 (DAPK3) IN COMPLEX WITH A BETA-CARBOLINE LIGAND  |   DEATH ASSOCIATED KINASE, DAPK3, ZIP KINASE, ZIPK, DAP KINASE 3, DAP LIKE KINASE, DLK, STRUCTURAL GENOMICS CONSORTIUM, SGC, APOPTOSIS, ATP-BINDING, CHROMATIN REGULATOR, NUCLEOTIDE-BINDING, NUCLEUS, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
5ew3:A   (THR875) to  (ALA1168)  HUMAN VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2 (KDR) KINASE DOMAIN IN COMPLEX WITH AAL993  |   KDR, KINASE DOMAIN, ATP-BINDING SITE, VEGFR2 INHIBITORS, TRANSFERASE 
5ew3:B   (THR875) to  (LEU1164)  HUMAN VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2 (KDR) KINASE DOMAIN IN COMPLEX WITH AAL993  |   KDR, KINASE DOMAIN, ATP-BINDING SITE, VEGFR2 INHIBITORS, TRANSFERASE 
3c4f:A   (GLU522) to   (LEU760)  FGFR TYROSINE KINASE DOMAIN IN COMPLEX WITH 3-(3- METHOXYBENZYL)-7-AZAINDOLE  |   FIBROBLAST GROWTH FACTOR RECEPTOR, TYROSINE KINASE DOMAIN, RECEPTOR TYROSINE KINASE, FGFR1, FGFR, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, DWARFISM, GLYCOPROTEIN, HEPARIN-BINDING, IMMUNOGLOBULIN DOMAIN, KALLMANN SYNDROME, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3c4f:B   (GLU522) to   (LEU760)  FGFR TYROSINE KINASE DOMAIN IN COMPLEX WITH 3-(3- METHOXYBENZYL)-7-AZAINDOLE  |   FIBROBLAST GROWTH FACTOR RECEPTOR, TYROSINE KINASE DOMAIN, RECEPTOR TYROSINE KINASE, FGFR1, FGFR, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, DWARFISM, GLYCOPROTEIN, HEPARIN-BINDING, IMMUNOGLOBULIN DOMAIN, KALLMANN SYNDROME, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
4rj3:A    (SER46) to   (HIS283)  CDK2 WITH EGFR INHIBITOR COMPOUND 8  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, LYSINE ACETYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3cqw:A   (VAL192) to   (HIS405)  CRYSTAL STRUCTURE OF AKT-1 COMPLEXED WITH SUBSTRATE PEPTIDE AND INHIBITOR  |   KINASE, APOPTOSIS, ATP-BINDING, CARBOHYDRATE METABOLISM, CYTOPLASM, GLUCOSE METABOLISM, GLYCOGEN BIOSYNTHESIS, GLYCOGEN METABOLISM, MEMBRANE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, SUGAR TRANSPORT, TRANSFERASE, TRANSLATION REGULATION, TRANSPORT, ALTERNATIVE SPLICING, WNT SIGNALING PATHWAY 
4cfu:C    (PRO45) to   (GLN287)  STRUCTURE-BASED DESIGN OF C8-SUBSTITUTED O6- CYCLOHEXYLMETHOXYGUANINE CDK1 AND 2 INHIBITORS.  |   TRANSFERASE, STRUCTURE-BASED DRUG DESIGN, CONFORMATIONAL RESTRAINT, REVERSED BINDING MODE 
4rvt:A    (LEU68) to   (HIS286)  MAP4K4 IN COMPLEX WITH A PYRIDIN-2(1H)-ONE DERIVATIVE  |   PYRIDIN-2(1H)-ONE LIGAND, TYPE I, DFG-IN, SERINE/THREONINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ckr:A   (THR662) to   (VAL913)  CRYSTAL STRUCTURE OF THE HUMAN DDR1 KINASE DOMAIN IN COMPLEX WITH DDR1-IN-1  |   TRANSFERASE, COLLAGEN, DISCOIDIN DOMAIN 
4rx5:A   (GLU439) to   (ASN658)  BRUTON'S TYROSINE KINASE (BTK) WITH PYRIDAZINONE COMPOUND 23  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE 
3oct:A   (SER438) to   (MET655)  CRYSTAL STRUCTURE OF BRUTON'S TYROSINE KINASE MUTANT V555R IN COMPLEX WITH DASATINIB  |   TYROSINE KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ddp:A    (PRO45) to   (GLN287)  STRUCTURE OF PHOSPHORYLATED THR160 CDK2/CYCLIN A IN COMPLEX WITH THE INHIBITOR CR8  |   SER/THR PROTEIN KINASE; PHOSPHORYLATION; CELL CYCLE, ATP- BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, CYCLIN, CYTOPLASM, NUCLEUS, TRANSFERASE/CELL CYCLE COMPLEX 
4d4v:A   (ARG465) to   (LEU685)  FOCAL ADHESION KINASE CATALYTIC DOMAIN  |   TRANSFERASE, FOCAL ADHESION KINASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
4d4v:B   (SER461) to   (LEU685)  FOCAL ADHESION KINASE CATALYTIC DOMAIN  |   TRANSFERASE, FOCAL ADHESION KINASE, KINASE INHIBITOR, ATP-BINDING, INTEGRIN SIGNALING 
4tyj:A   (ASP511) to   (SER751)  STRUCTURAL ANALYSIS OF THE HUMAN FIBROBLAST GROWTH FACTOR RECEPTOR 4 KINASE  |   FIBROBLAST GROWTH FACTOR RECEPTOR, KINASE, TRANSFERASE, DOVITINIB, PONATINB, PROTEROS BIOSTRUCTURES GMBH 
4u0i:A   (LEU631) to   (THR932)  CRYSTAL STRUCTURE OF KIT IN COMPLEX WITH PONATINIB  |   KIT, RECEPTOR TYROSINE KINASE, INHIBITOR, PONATINIB, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3ori:C    (PRO50) to   (GLY279)  MYCOBACTERIUM TUBERCULOSIS PKNB KINASE DOMAIN L33D MUTANT (CRYSTAL FORM 1)  |   STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, KINASE, SIGNAL TRANSDUCTION, TRANSFERASE 
5hx6:A    (ILE54) to   (GLU269)  CRYSTAL STRUCTURE OF RIP1 KINASE WITH A BENZO[B][1,4]OXAZEPIN-4-ONE  |   KINASE, INHIBITOR COMPLEX, NON-HINGE BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3poo:A    (ILE85) to   (ALA298)  HUMAN CAMP-DEPENDENT PROTEIN KINASE IN COMPLEX WITH AN INHIBITOR  |   ATP BINDING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5i9w:A   (THR653) to   (ALA877)  CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE WITH ANP  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, RECEPTOR, ATP-BINDING 
5ia3:A   (THR653) to   (ALA877)  CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE WITH PD173955  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, RECEPTOR, ATP-BINDING 
4eev:A  (GLY1119) to  (THR1343)  CRYSTAL STRUCTURE OF C-MET IN COMPLEX WITH LY2801653  |   PROTEIN TYROSINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ez7:A    (SER46) to   (GLN287)  CDK2 IN COMPLEX WITH STAUROSPORINE AND 2 MOLECULES OF 8-ANILINO-1- NAPHTHALENE SULFONIC ACID  |   PROTEIN KINASE, ANS, TRANSFERASE-ANTIBIOTIC COMPLEX 
3qgy:A   (SER399) to   (ALA616)  CRYSTAL STRUCTURE OF ITK INHIBITOR COMPLEX  |   PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qgy:B   (GLU400) to   (ALA616)  CRYSTAL STRUCTURE OF ITK INHIBITOR COMPLEX  |   PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qlf:B   (GLU305) to   (TYR519)  CRYSTAL STRUCTURE OF THE L317I MUTANT OF THE C-SRC TYROSINE KINASE DOMAIN COMPLEXED WITH PYRAZOLOPYRIMIDINE 5  |   C-SRC L317I MUTANT, TYROSINE KINASE, TRANSFERASE, PYRAZOLOPYRIMIDINE 5 
4v04:A   (GLU522) to   (LEU760)  FGFR1 IN COMPLEX WITH PONATINIB.  |   TRANSFERASE 
4v04:B   (GLU522) to   (LEU760)  FGFR1 IN COMPLEX WITH PONATINIB.  |   TRANSFERASE 
3qu0:A    (PRO45) to   (HIS283)  CDK2 IN COMPLEX WITH INHIBITOR RC-2-38  |   PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fkj:A    (SER46) to   (GLN287)  CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH AMINOPYRAZOLE INHIBITOR  |   ALPHA AND BETA PROTEIN (A+B), TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5l2s:A    (LEU56) to   (GLN301)  THE X-RAY CO-CRYSTAL STRUCTURE OF HUMAN CDK6 AND ABEMACICLIB.  |   CYCLIN-DEPENDENT KINASE, KINASE INHIBITOR, KINASE SELECTIVITY, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX