Usages in wwPDB of concept: c_0200
nUsages: 206; SSE string: HHHHEEHHHHH
3e94:A   (VAL232) to   (ILE442)  CRYSTAL STRUCTURE OF RXRALPHA LIGAND BINDING DOMAIN IN COMPLEX WITH TRIBUTYLTIN AND A COACTIVATOR FRAGMENT  |   PROTEIN-LIGAND COMPLEX, DNA-BINDING, HOST-VIRUS INTERACTION, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, UBL CONJUGATION, ZINC, ZINC-FINGER, ACTIVATOR, PHOSPHOPROTEIN 
1nde:A   (PRO265) to   (ASN478)  ESTROGEN RECEPTOR BETA WITH SELECTIVE TRIAZINE MODULATOR  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER, ERB, TRIAZINE, ESTROGEN, ESTRADIOL, OESTROGEN, TRANSCRIPTION 
2p1u:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF THE LIGAND BINDING DOMAIN OF THE RETINOID X RECEPTOR ALPHA IN COMPLEX WITH 3-(2'-ETHOXY)- TETRAHYDRONAPHTYL CINNAMIC ACID AND A FRAGMENT OF THE COACTIVATOR TIF-2  |   PROTEIN-LIGAND COMPLEX, HORMONE RECEPTOR 
2p1v:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF THE LIGAND BINDING DOMAIN OF THE RETINOID X RECEPTOR ALPHA IN COMPLEX WITH 3-(2'-PROPOXY)- TETRAHYDRONAPHTYL CINNAMIC ACID AND A FRAGMENT OF THE COACTIVATOR TIF-2  |   PROTEIN-LIGAND COMPLEX, HORMONE RECEPTOR 
2p7g:A   (LYS236) to   (GLY442)  X-RAY STRUCTURE OF ESTROGEN RELATED RECEPTOR G IN COMPLEX WITH BISPHENOL A.  |   THREE LAYERED ALPHA HELICAL SANDWICH, HORMONE RECEPTOR 
2p7z:A   (LYS236) to   (LYS439)  ESTROGEN RELATED RECEPTOR GAMMA IN COMPLEX WITH 4-HYDROXY- TAMOXIFEN  |   THREE LAYERED ALPHA HELICAL SANDWICH, HORMONE RECEPTOR 
2bj4:A   (THR311) to   (MET528)  ESTROGEN RECEPTOR ALPHA LBD IN COMPLEX WITH A PHAGE-DISPLAY DERIVED PEPTIDE ANTAGONIST  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, PEPTIDE ANTAGONIST, LIGAND-BINDING DOMAIN (LBD), DNA-BINDING, NUCLEAR PROTEIN STEROID-BINDING 
1bsx:A   (THR215) to   (GLU445)  STRUCTURE AND SPECIFICITY OF NUCLEAR RECEPTOR-COACTIVATOR INTERACTIONS  |   NUCLEAR RECEPTORS, COACTIVATORS, GRIP1, SPECIFICITY INTERACTION SITE, HORMONE/GROWTH FACTOR COMPLEX 
1bsx:B   (THR215) to   (GLU445)  STRUCTURE AND SPECIFICITY OF NUCLEAR RECEPTOR-COACTIVATOR INTERACTIONS  |   NUCLEAR RECEPTORS, COACTIVATORS, GRIP1, SPECIFICITY INTERACTION SITE, HORMONE/GROWTH FACTOR COMPLEX 
3fal:A   (VAL232) to   (CYS432)  HUMANRXR ALPHA & MOUSE LXR ALPHA COMPLEXED WITH RETENOIC ACID AND GSK2186  |   NUCLEAR HORMONE RECEPTOR NONSTEROIDAL LXR AGONIST CHOLOESTOROL METABOLISM, DNA-BINDING, HOST-VIRUS INTERACTION, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, UBL CONJUGATION, ZINC, ZINC-FINGER, SIGNALING PROTEIN 
3fal:C   (VAL232) to   (LEU433)  HUMANRXR ALPHA & MOUSE LXR ALPHA COMPLEXED WITH RETENOIC ACID AND GSK2186  |   NUCLEAR HORMONE RECEPTOR NONSTEROIDAL LXR AGONIST CHOLOESTOROL METABOLISM, DNA-BINDING, HOST-VIRUS INTERACTION, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, UBL CONJUGATION, ZINC, ZINC-FINGER, SIGNALING PROTEIN 
3fc6:A   (VAL232) to   (LEU433)  HRXRALPHA & MLXRALPHA WITH AN INDOLE PHARMACOPHORE, SB786875  |   LIVER X RECEPTOR, NUCLEAR HORMONE RECEPTORS, AGONISTS, EPOXYCHOLESTEROL, DNA-BINDING, HOST-VIRUS INTERACTION, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, UBL CONJUGATION, ZINC, ZINC-FINGER 
3fc6:C   (VAL232) to   (GLU434)  HRXRALPHA & MLXRALPHA WITH AN INDOLE PHARMACOPHORE, SB786875  |   LIVER X RECEPTOR, NUCLEAR HORMONE RECEPTORS, AGONISTS, EPOXYCHOLESTEROL, DNA-BINDING, HOST-VIRUS INTERACTION, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, UBL CONJUGATION, ZINC, ZINC-FINGER 
1ovl:A   (SER363) to   (ASP580)  CRYSTAL STRUCTURE OF NURR1 LBD  |   NUUR1, LBD, TRANSCRIPTION 
2q6j:B   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR ALPHA COMPLEXED TO A B-N SUBSTITUTED LIGAND  |   PROTEIN-LIGAND COMPLEX, TRANSCRIPTION 
2qab:A   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN MUTANT 537S COMPLEXED WITH AN ETHYL INDAZOLE COMPOUND  |   PROTEIN-LIGAND COMPLEX, TRANSCRIPTION 
2qab:B   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN MUTANT 537S COMPLEXED WITH AN ETHYL INDAZOLE COMPOUND  |   PROTEIN-LIGAND COMPLEX, TRANSCRIPTION 
2qgt:B   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED TO AN ETHER ESTRADIOL COMPOUND  |   PROTEIN-LIGAND COMPLEX, TRANSCRIPTION 
2qgw:A   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED WITH A CHLORO-INDAZOLE COMPOUND  |   PROTEIN-LIGAND COMPLEX, TRANSCRIPTION 
2qgw:B   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED WITH A CHLORO-INDAZOLE COMPOUND  |   PROTEIN-LIGAND COMPLEX, TRANSCRIPTION 
1dkf:A   (PRO236) to   (PHE443)  CRYSTAL STRUCTURE OF A HETERODIMERIC COMPLEX OF RAR AND RXR LIGAND-BINDING DOMAINS  |   HELICAL SANDWICH, HETERODIMER, PROTEIN-LIGAND COMPLEX, HORMONE/GROWTH FACTOR RECEPTOR, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS 
1dkf:B   (PRO182) to   (ILE402)  CRYSTAL STRUCTURE OF A HETERODIMERIC COMPLEX OF RAR AND RXR LIGAND-BINDING DOMAINS  |   HELICAL SANDWICH, HETERODIMER, PROTEIN-LIGAND COMPLEX, HORMONE/GROWTH FACTOR RECEPTOR, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS 
4iu7:A   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH CONSTRAINED WAY-DERIVATIVE, 2B  |   NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, NUCLEUS, TRANSCRIPTION 
4iv2:A   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DYNAMIC WAY-DERIVATIVE, 5A  |   NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION 
4iw8:B   (THR311) to   (LYS531)  CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DYNAMIC WAY-DERIVATIVE, 9A  |   NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION 
1pq6:A   (THR221) to   (ASP446)  HUMAN LXR BETA HORMONE RECEPTOR / GW3965 COMPLEX  |   LXRB+KB043546/WAY207380/GW3965, TRANSCRIPTION REGULATION 
1pq6:D   (ALA222) to   (LEU444)  HUMAN LXR BETA HORMONE RECEPTOR / GW3965 COMPLEX  |   LXRB+KB043546/WAY207380/GW3965, TRANSCRIPTION REGULATION 
1pq9:C   (THR221) to   (ARG411)  HUMAN LXR BETA HORMONE RECEPTOR COMPLEXED WITH T0901317 COMPLEX  |   LXRB+T0901317 SPLIT, TRANSCRIPTION REGULATION 
2qtu:A   (PRO265) to   (MET479)  ESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN COMPLEXED TO A BENZOPYRAN LIGAND  |   NUCLEAR RECEPTOR, LIGAND-BINDING DOMAIN, ALTERNATIVE SPLICING, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, TRANSCRIPTION REGULATOR 
2qtu:B   (SER264) to   (MET479)  ESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN COMPLEXED TO A BENZOPYRAN LIGAND  |   NUCLEAR RECEPTOR, LIGAND-BINDING DOMAIN, ALTERNATIVE SPLICING, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, TRANSCRIPTION REGULATOR 
4j24:A   (SER264) to   (ASN483)  ESTROGEN RECEPTOR IN COMPLEX WITH PROLINE-FLANKED LXXLL PEPTIDES  |   ESTROGEN RECEPTOR, PROLINE, LXXLL, ALPHA-HELIX, STRUCTURE STABILIZATION, HORMONE RECEPTOR-PEPTIDE COMPLEX 
4j24:B   (PRO265) to   (ASN483)  ESTROGEN RECEPTOR IN COMPLEX WITH PROLINE-FLANKED LXXLL PEPTIDES  |   ESTROGEN RECEPTOR, PROLINE, LXXLL, ALPHA-HELIX, STRUCTURE STABILIZATION, HORMONE RECEPTOR-PEPTIDE COMPLEX 
4j24:C   (SER264) to   (ASN483)  ESTROGEN RECEPTOR IN COMPLEX WITH PROLINE-FLANKED LXXLL PEPTIDES  |   ESTROGEN RECEPTOR, PROLINE, LXXLL, ALPHA-HELIX, STRUCTURE STABILIZATION, HORMONE RECEPTOR-PEPTIDE COMPLEX 
4j24:D   (PRO265) to   (ASN483)  ESTROGEN RECEPTOR IN COMPLEX WITH PROLINE-FLANKED LXXLL PEPTIDES  |   ESTROGEN RECEPTOR, PROLINE, LXXLL, ALPHA-HELIX, STRUCTURE STABILIZATION, HORMONE RECEPTOR-PEPTIDE COMPLEX 
4j5w:D   (GLU233) to   (GLY443)  CRYSTAL STRUCTURE OF THE APO-PXR/RXRALPHA LBD HETEROTETRAMER COMPLEX  |   PREGNANE X RECEPTOR, RETINOID X RECEPTOR ALPHA, LIGAND BINDING DOMAIN, NUCLEAR RECEPTOR, ALPHA HELICAL SANDWICH, UNIQUE INTERMOLECULAR BETA-SHEET DIMERIZATION, XENOBIOTIC SENSING, UPREGULATION OF DRUG METABOLISM ENZYMES, RETINOIC ACID-BINDING PROTEIN 
4j5x:D   (GLU233) to   (GLY443)  CRYSTAL STRUCTURE OF THE SR12813-BOUND PXR/RXRALPHA LBD HETEROTETRAMER COMPLEX  |   PREGNANE X RECEPTOR, RETINOID X RECEPTOR ALPHA, LIGAND BINDING DOMAIN, NUCLEAR RECEPTOR, SR12813, ALPHA HELICAL SANDWICH, UNIQUE INTERMOLECULAR BETA-SHEET DIMERIZATION, XENOBIOTIC SENSING, UPREGULATION OF DRUG METABOLISM ENZYMES, RETINOIC ACID-BINDING PROTEIN 
3h0a:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA (PPARG) AND RETINOIC ACID RECEPTOR ALPHA (RXRA) IN COMPLEX WITH 9-CIS RETINOIC ACID, CO-ACTIVATOR PEPTIDE, AND A PARTIAL AGONIST  |   PPAR, TRANSCRIPTION, NUCLEAR RECEPTOR FOLD, TRANSCRIPTION REGULATION, HORMONE, GROWTH FACTOR RECEPTOR, COMPLEX, DNA-BINDING, HOST-VIRUS INTERACTION, ISOPEPTIDE BOND, METAL-BINDING, NUCLEUS, RECEPTOR, ZINC-FINGER, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, OBESITY, PHOSPHOPROTEIN, ACYLTRANSFERASE, PROTO-ONCOGENE, TRANSFERASE 
1qkm:A   (PRO265) to   (MET479)  HUMAN OESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN IN COMPLEX WITH PARTIAL AGONIST GENISTEIN  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, PHYTO-OESTROGEN, PARTIAL AGONIST 
2e2r:A   (LYS236) to   (GLY442)  CRYSTAL STRUCTURE OF HUMAN ESTROGEN-RELATED RECEPTOR GAMMA LIGAND BINDING DOMAIN COMPLEX WITH BISPHENOL A  |   ERR GAMMA, BPA, NUCLEAR RECEPTOR, TRANSCRIPTION 
1r1k:A   (SER209) to   (HIS439)  CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE HETERODIMER ECR/USP BOUND TO PONASTERONE A  |   NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, HETERODIMER, ALPHA-HELICAL SANDWICH, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX 
1fby:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF THE HUMAN RXR ALPHA LIGAND BINDING DOMAIN BOUND TO 9-CIS RETINOIC ACID  |   NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, RETINOID RECEPTOR, TRANSCRIPTION 
1r20:A   (SER209) to   (HIS439)  CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE HETERODIMER ECR/USP BOUND TO THE SYNTHETIC AGONIST BYI06830  |   NUCLEAR RECEPTOR, HETERODIMER, ALPHA-HELICAL SANDWICH, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX 
4jyg:A   (GLU172) to   (PRO396)  CRYSTAL STRUCTURE OF RARBETA LBD IN COMPLEX WITH AGONIST BMS411 [4- {[(5,5-DIMETHYL-8-PHENYL-5,6-DIHYDRONAPHTHALEN-2-YL) CARBONYL]AMINO}BENZOIC ACID]  |   LIGAND BINDING DOMAIN, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION- AGONIST COMPLEX 
4jyh:A   (GLU172) to   (LYS392)  CRYSTAL STRUCTURE OF RARBETA LBD IN COMPLEX WITH SELECTIVE AGONIST BMS948 [4-{[(8-PHENYLNAPHTHALEN-2-YL)CARBONYL]AMINO}BENZOIC ACID]  |   LIGAND BINDING DOMAIN, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION- AGONIST COMPLEX 
4jyi:B   (GLU176) to   (ILE395)  CRYSTAL STRUCTURE OF RARBETA LBD IN COMPLEX WITH SELECTIVE PARTIAL AGONIST BMS641 [3-CHLORO-4-[(E)-2-(5,5-DIMETHYL-8-PHENYL-5,6- DIHYDRONAPHTHALEN-2-YL)ETHENYL]BENZOIC ACID]  |   LIGAND BINDING DOMAIN, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION- AGONIST COMPLEX 
1fm9:A   (VAL232) to   (GLY443)  THE 2.1 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE HETERODIMER OF THE HUMAN RXRALPHA AND PPARGAMMA LIGAND BINDING DOMAINS RESPECTIVELY BOUND WITH 9-CIS RETINOIC ACID AND GI262570 AND CO-ACTIVATOR PEPTIDES.  |   THE HETERODIMER OF THE NUCLEAR RECEPTOR LIGAND BINDING DOMAINS OF RXRALPHA AND PPARGAMMA BOUND RESPECTIVELY WITH 9-CIS RETINOIC ACID AND GI262570 AND CO-ACTIVATOR PEPTIDES, TRANSCRIPTION 
2ewp:C   (ASN235) to   (LYS439)  CRYSTAL STRUCTURE OF ESTROGEN RELATED RECEPTOR-3 (ERR-GAMMA) LIGAND BINDING DOMAIND WITH TAMOXIFEN ANALOG GSK5182  |   TAMOXIFEN, ERR, ESTROGEN RELATED RECEPTOR, ORPHAN RECEPTOR, TRANSCRIPTION 
2ewp:D   (ILE237) to   (MET419)  CRYSTAL STRUCTURE OF ESTROGEN RELATED RECEPTOR-3 (ERR-GAMMA) LIGAND BINDING DOMAIND WITH TAMOXIFEN ANALOG GSK5182  |   TAMOXIFEN, ERR, ESTROGEN RELATED RECEPTOR, ORPHAN RECEPTOR, TRANSCRIPTION 
2ewp:E   (ILE237) to   (LYS439)  CRYSTAL STRUCTURE OF ESTROGEN RELATED RECEPTOR-3 (ERR-GAMMA) LIGAND BINDING DOMAIND WITH TAMOXIFEN ANALOG GSK5182  |   TAMOXIFEN, ERR, ESTROGEN RELATED RECEPTOR, ORPHAN RECEPTOR, TRANSCRIPTION 
4k6i:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF HUMAN RETINOID X RECEPTOR ALPHA-LIGAND BINDING DOMAIN COMPLEX WITH TARGRETIN AND THE COACTIVATOR PEPTIDE GRIP-1  |   LIGAND BINDING DOMAIN, CANCER, TARGRETIN (BEXAROTENE), TRANSCRIPTION 
1rdt:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF A NEW REXINOID BOUND TO THE RXRALPHA LIGAND BINDING DOAMIN IN THE RXRALPHA/PPARGAMMA HETERODIMER  |   HORMONE, RECEPTOR, POLYMORPHISM, HORMONE/GROWTH FACTOR COMPLEX 
1g2n:A   (ILE210) to   (PHE438)  CRYSTAL STRUCTURE OF THE LIGAND BINDING DOMAIN OF THE ULTRASPIRACLE PROTEIN USP, THE ORTHOLOG OF RXRS IN INSECTS  |   ANTIPARALLEL ALPHA-HELICAL SANDWICH, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS, GENE REGULATION 
1g50:A   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF A WILD TYPE HER ALPHA LBD AT 2.9 ANGSTROM RESOLUTION  |   ALPHA HELICES, ESTRADIOL, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS, DNA BINDING PROTEIN 
3uu7:A   (THR311) to   (LYS531)  CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BISPHENOL-A  |   LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR 
2fsz:A   (PRO265) to   (MET479)  A SECOND BINDING SITE FOR HYDROXYTAMOXIFEN WITHIN THE COACTIVATOR-BINDING GROOVE OF ESTROGEN RECEPTOR BETA  |   NUCLEAR HORMONE BINDING DOMAIN, HORMONE/GROWTH FACTOR COMPLEX 
2fsz:B   (PRO265) to   (MET479)  A SECOND BINDING SITE FOR HYDROXYTAMOXIFEN WITHIN THE COACTIVATOR-BINDING GROOVE OF ESTROGEN RECEPTOR BETA  |   NUCLEAR HORMONE BINDING DOMAIN, HORMONE/GROWTH FACTOR COMPLEX 
4zi1:A   (SER264) to   (ASN483)  HUMAN ESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN IN COMPLEX WITH KB095285 AND CIA12 COACTIVATOR PEPTIDE  |   ESTROGEN RECEPTOR BETA, BETA SELECTIVE, ERB, SIGNALING PROTEIN 
1gwr:B   (THR311) to   (ASN532)  HUMAN OESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH 17BETA-OESTRADIOL AND TIF2 NRBOX3 PEPTIDE  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, TRANSACTIVATION, AGONIST, AF2 COACTIVATOR , RECEPTOR, ACTIVATOR, TRANSCRIPTI REGULATION, DNA-BINDING, NUCLEAR PROTEIN, ZINC FINGER, STER BINDING, PHOSPHORYLATION, POLYMORPHISM, ALTERNATIVE SPLICING 
4kzi:B   (ASN363) to   (ASP580)  CRYSTAL STRUCTURE OF TR3 LBD IN COMPLEX WITH DPDO  |   ORPHAN NUCLEAR RECEPTOR, TRANSCRIPTION 
2giu:A   (PRO265) to   (LEU476)  HUMAN ESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN IN COMPLEX WITH COMPOUND 45  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ER-BETA, AGONIST, TRANSCRIPTION REGULATOR 
4zn9:B   (THR311) to   (SER527)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH OXABICYCLIC HEPTENE SULFONATE (OBHS)  |   PROTEIN LIGAND COMPLEX, TRANSCRIPTION 
4zns:A   (THR311) to   (LYS529)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH A 3-FLUORO-SUBSTITUTED OBHS DERIVATIVE  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
2gp7:A   (ILE237) to   (GLY442)  ESTROGEN RELATED RECEPTOR-GAMMA LIGAND BINDING DOMAIN  |   ESTROGEN RELATED RECEPTOR, ERR, ERRG, ESRRG, NUCLEAR RECEPTOR, STEROID RECEPTOR, TRANSCRIPTION 
2gp7:B   (ILE237) to   (GLY442)  ESTROGEN RELATED RECEPTOR-GAMMA LIGAND BINDING DOMAIN  |   ESTROGEN RELATED RECEPTOR, ERR, ERRG, ESRRG, NUCLEAR RECEPTOR, STEROID RECEPTOR, TRANSCRIPTION 
2gp7:C   (ILE237) to   (GLY442)  ESTROGEN RELATED RECEPTOR-GAMMA LIGAND BINDING DOMAIN  |   ESTROGEN RELATED RECEPTOR, ERR, ERRG, ESRRG, NUCLEAR RECEPTOR, STEROID RECEPTOR, TRANSCRIPTION 
1h9u:A   (VAL301) to   (ILE513)  THE STRUCTURE OF THE HUMAN RETINOID-X-RECEPTOR BETA LIGAND BINDING DOMAIN IN COMPLEX WITH THE SPECIFIC SYNTHETIC AGONIST LG100268  |   NUCLEAR RECEPTOR, RXR, TRANSCRIPTION FACTOR 
1h9u:B   (VAL301) to   (ILE513)  THE STRUCTURE OF THE HUMAN RETINOID-X-RECEPTOR BETA LIGAND BINDING DOMAIN IN COMPLEX WITH THE SPECIFIC SYNTHETIC AGONIST LG100268  |   NUCLEAR RECEPTOR, RXR, TRANSCRIPTION FACTOR 
1h9u:C   (ASP302) to   (ILE513)  THE STRUCTURE OF THE HUMAN RETINOID-X-RECEPTOR BETA LIGAND BINDING DOMAIN IN COMPLEX WITH THE SPECIFIC SYNTHETIC AGONIST LG100268  |   NUCLEAR RECEPTOR, RXR, TRANSCRIPTION FACTOR 
1h9u:D   (VAL301) to   (ILE513)  THE STRUCTURE OF THE HUMAN RETINOID-X-RECEPTOR BETA LIGAND BINDING DOMAIN IN COMPLEX WITH THE SPECIFIC SYNTHETIC AGONIST LG100268  |   NUCLEAR RECEPTOR, RXR, TRANSCRIPTION FACTOR 
4zsh:A   (VAL232) to   (LEU441)  RXR LBD IN COMPLEX WITH 9-CIS-13,14-DIHYDRORETINOIC ACID  |   TRANSCRIPTION, NUCLEAR RECEPTOR, RXR 
3ips:A   (SER207) to   (ASP432)  X-RAY STRUCTURE OF BENZISOXAZOLE SYNTHETIC AGONIST BOUND TO THE LXR- ALPHA  |   NUCLEAR RECEPTOR, LXR HOMODIMER, LXR SIGNALING, ALTERNATIVE SPLICING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ACTIVATOR, ISOPEPTIDE BOND, PROTO-ONCOGENE, CHOLESTEROL, ABCA1, HETERODIMER, RXR, LIGAND COMPLEX 
1hj1:A   (SER219) to   (MET434)  RAT OESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN IN COMPLEX WITH PURE ANTIOESTROGEN ICI164,384  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, OESTROGEN, ANTAGONIST 
1u3q:A   (PRO265) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH CL-272  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1u3q:B   (SER264) to   (LYS482)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH CL-272  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1u3q:C   (SER264) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH CL-272  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1u3q:D   (SER264) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH CL-272  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1u3r:A   (SER264) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-338  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1u3r:B   (SER264) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-338  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1u9e:A   (SER264) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-397  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1u9e:B   (SER264) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-397  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
2i0g:A   (PRO265) to   (MET479)  BENZOPYRANS ARE SELECTIVE ESTROGEN RECEPTOR BETA AGONISTS (SERBAS) WITH NOVEL ACTIVITY IN MODELS OF BENIGN PROSTATIC HYPERPLASIA  |   NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, TRANSCRIPTION 
2i0g:B   (SER264) to   (MET479)  BENZOPYRANS ARE SELECTIVE ESTROGEN RECEPTOR BETA AGONISTS (SERBAS) WITH NOVEL ACTIVITY IN MODELS OF BENIGN PROSTATIC HYPERPLASIA  |   NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, TRANSCRIPTION 
1uhl:A   (VAL301) to   (GLY514)  CRYSTAL STRUCTURE OF THE LXRALFA-RXRBETA LBD HETERODIMER  |   LIGAND-BINDING DOMAIN, DNA BINDING PROTEIN 
4m8e:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF HUMAN RETINOID X RECEPTOR ALPHA-LIGAND BINDING DOMAIN COMPLEX WITH (S) 4-METHYL 9CUAB30 COACTIVATOR PEPTIDE GRIP-1  |   ANTIPARALLEL SANDWICH, LIGAND BINDING, COACTIVATOR BINDING, DIMERIZATION, ACTIVATION FUNCTION, TRANSCRIPTION, NUCLEAR RECEPTORS, LIGAND BINDING DOMIAN, LIGAND BINDING POCKET, COACTIVATOR BINDING SITE, CANCER, 4-METHYL 9CUAB30 ((2E,4E,6Z,8E)-8-[(4'S)METHYL-3',4'- DIHYDRO-1'(2'H)-NAPHTHALEN-1'-YLIDENE]-3,7-DIMETHYL-2,4,6- OCTATRIENOIC ACID) 
4mga:B   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH 4-TERT- OCTYLPHENOL  |   LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR 
2j7y:A   (SER219) to   (ASN438)  STRUCTURE OF 17-EPIESTRIOL-BOUND ESTROGEN RECEPTOR BETA LBD IN COMPLEX WITH LXXLL MOTIF FROM NCOA5  |   RECEPTOR, ACTIVATOR, REPRESSOR, ZINC-FINGER, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, NUCLEAR PROTEIN, PHOSPHORYLATION, STEROID-BINDING, COACTIVATOR, COREPRESSOR, DNA-BINDING, GLYCOPROTEIN, TRANSCRIPTION REGULATION, TRANSCRIPTION, METAL-BINDING, LIPID-BINDING 
4n1y:A   (GLN248) to   (GLY458)  CRYSTAL STRUCTURE OF THE PACIFIC OYSTER ESTROGEN RECEPTOR LIGAND BINDING DOMAIN  |   ESTROGEN, NUCLEAR HORMONE RECEPTOR, ENDOCRINE SIGNALING, TRANSCRIPTION 
4n1y:B   (GLN248) to   (GLY458)  CRYSTAL STRUCTURE OF THE PACIFIC OYSTER ESTROGEN RECEPTOR LIGAND BINDING DOMAIN  |   ESTROGEN, NUCLEAR HORMONE RECEPTOR, ENDOCRINE SIGNALING, TRANSCRIPTION 
1k74:A   (VAL232) to   (GLY443)  THE 2.3 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE HETERODIMER OF THE HUMAN PPARGAMMA AND RXRALPHA LIGAND BINDING DOMAINS RESPECTIVELY BOUND WITH GW409544 AND 9-CIS RETINOIC ACID AND CO-ACTIVATOR PEPTIDES.  |   THE HETERODIMER OF THE NUCLEAR RECEPTOR LIGAND BINDING DOMAINS OF RXRALPHA AND PPARGAMMA BOUND RESPECTIVELY WITH 9-CIS RETINOIC ACID AND GW409544 AND COACTIVATOR PEPTIDES, TRANSCRIPTION 
1x7b:B   (SER264) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH ERB-041  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1x78:A   (PRO265) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-244  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1x78:B   (PRO265) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-244  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1x7e:B   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR ALPHA COMPLEXED WITH WAY-244  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN RECEPTOR ALPHA, ER-ALPHA, ESTROGEN, NUCLEAR RECEPT TRANSCRIPTION FACTOR, AGONIST 
1l2j:A   (PRO265) to   (LEU476)  HUMAN ESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN IN COMPLEX WITH (R, R)-5,11-CIS-DIETHYL-5,6,11,12-TETRAHYDROCHRYSENE-2,8-DIOL  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ESTROGEN, ANTAGONIST, TRANSCRIPTION RECEPTOR 
1l2j:B   (PRO265) to   (MET479)  HUMAN ESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN IN COMPLEX WITH (R, R)-5,11-CIS-DIETHYL-5,6,11,12-TETRAHYDROCHRYSENE-2,8-DIOL  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ESTROGEN, ANTAGONIST, TRANSCRIPTION RECEPTOR 
3jzc:A   (THR215) to   (GLU445)  CRYSTAL STRUCTURE OF TR-BETA BOUND TO THE SELECTIVE THYROMIMETIC TRIAC  |   TR, TRIAC, ENTROPY, DEAFNESS, DISEASE MUTATION, DNA-BINDING, METAL- BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER 
4oc7:A   (VAL232) to   (GLY443)  RETINOIC ACID RECEPTOR ALPHA IN COMPLEX WITH (E)-3-(3'-ALLYL-6- HYDROXY-[1,1'-BIPHENYL]-3-YL)ACRYLIC ACID AND A FRAGMENT OF THE COACTIVATOR TIF2  |   LIGAND BINDING DOMAIN, TRANSCRIPTION 
2nxx:E   (SER333) to   (ASN532)  CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE T.CASTANEUM (COLEOPTERA) HETERODIMER ECRUSP BOUND TO PONASTERONE A  |   HORMONE RECEPTOR, APO AND HOLO LIGAND BINDING POCKET, HORMONE/GROWTH FACTOR COMPLEX 
2nxx:F   (SER333) to   (ASN532)  CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE T.CASTANEUM (COLEOPTERA) HETERODIMER ECRUSP BOUND TO PONASTERONE A  |   HORMONE RECEPTOR, APO AND HOLO LIGAND BINDING POCKET, HORMONE/GROWTH FACTOR COMPLEX 
2nxx:G   (SER333) to   (ASN532)  CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE T.CASTANEUM (COLEOPTERA) HETERODIMER ECRUSP BOUND TO PONASTERONE A  |   HORMONE RECEPTOR, APO AND HOLO LIGAND BINDING POCKET, HORMONE/GROWTH FACTOR COMPLEX 
2nxx:H   (SER333) to   (ASN532)  CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE T.CASTANEUM (COLEOPTERA) HETERODIMER ECRUSP BOUND TO PONASTERONE A  |   HORMONE RECEPTOR, APO AND HOLO LIGAND BINDING POCKET, HORMONE/GROWTH FACTOR COMPLEX 
2z4b:A   (PRO265) to   (MET479)  ESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN COMPLEXED TO A BENZOPYRAN LIGAND  |   NUCLEAR RECEPTOR LIGAND BINDING DOMAIN, TRANSCRIPTION 
2z4b:B   (SER264) to   (MET479)  ESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN COMPLEXED TO A BENZOPYRAN LIGAND  |   NUCLEAR RECEPTOR LIGAND BINDING DOMAIN, TRANSCRIPTION 
1xiu:A   (VAL214) to   (ASP418)  CRYSTAL STRUCTURE OF THE AGONIST-BOUND LIGAND-BINDING DOMAIN OF BIOMPHALARIA GLABRATA RXR  |   NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, RETINOID RECEPTOR, TRANSCRIPTION-TRANSFERASE COMPLEX 
1xiu:B   (VAL214) to   (GLY417)  CRYSTAL STRUCTURE OF THE AGONIST-BOUND LIGAND-BINDING DOMAIN OF BIOMPHALARIA GLABRATA RXR  |   NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, RETINOID RECEPTOR, TRANSCRIPTION-TRANSFERASE COMPLEX 
2zas:A   (LYS236) to   (GLY442)  CRYSTAL STRUCTURE OF HUMAN ESTROGEN-RELATED RECEPTOR GAMMA LIGAND BINDING DOMAIN COMPLEX WITH 4-ALPHA-CUMYLPHENOL, A BISPHENOL A DERIVATIVE  |   ERR GAMMA, BPA, 4-ALPHA-CUMYLPHENOL, NUCLEAR RECEPTOR, TRANSCRIPTION, ACTIVATOR, DNA-BINDING, METAL-BINDING, NUCLEUS, TRANSCRIPTION REGULATION, ZINC-FINGER 
2zkc:A   (LYS236) to   (GLY442)  CRYSTAL STRUCTURE OF HUMAN ESTROGEN-RELATED RECEPTOR GAMMA LIGAND BINDING DOMAIN COMPLEX WITH BISPHENOL Z  |   ERR GAMMA, BPA, NUCLEAR RECEPTOR, TRANSCRIPTION, ACTIVATOR, DNA- BINDING, METAL-BINDING, NUCLEUS, TRANSCRIPTION REGULATION, ZINC- FINGER 
1xv9:A   (VAL232) to   (ILE442)  CRYSTAL STRUCTURE OF CAR/RXR HETERODIMER BOUND WITH SRC1 PEPTIDE, FATTY ACID, AND 5B-PREGNANE-3,20-DIONE.  |   CAR, RXR, SRC1, PREGNANEDIONE, DNA BINDING PROTEIN 
2zxz:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF THE HUMAN RXR ALPHA LIGAND BINDING DOMAIN BOUND TO A SYNTHETIC AGONIST COMPOUND AND A COACTIVATOR PEPTIDE  |   TRANSCRIPTION REGULATION, NUCLEAR RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM FOR RESEARCH ON GENE EXPRESSION, SGCGES 
2zy0:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF THE HUMAN RXR ALPHA LIGAND BINDING DOMAIN BOUND TO A SYNTHETIC AGONIST COMPOUND AND A COACTIVATOR PEPTIDE  |   TRANSCRIPTION REGULATION, NUCLEAR RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM FOR RESEARCH ON GENE EXPRESSION, SGCGES 
2zy0:C   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF THE HUMAN RXR ALPHA LIGAND BINDING DOMAIN BOUND TO A SYNTHETIC AGONIST COMPOUND AND A COACTIVATOR PEPTIDE  |   TRANSCRIPTION REGULATION, NUCLEAR RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM FOR RESEARCH ON GENE EXPRESSION, SGCGES 
3kmr:A   (PRO182) to   (GLU401)  CRYSTAL STRUCTURE OF RARALPHA LIGAND BINDING DOMAIN IN COMPLEX WITH AN AGONIST LIGAND (AM580) AND A COACTIVATOR FRAGMENT  |   NUCLEAR RECEPTOR TRANSCRIPTION FACTOR LIGAND BINDING DOMAIN, DNA- BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER, ACTIVATOR, ACYLTRANSFERASE, ISOPEPTIDE BOND, TRANSFERASE 
1mv9:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF THE HUMAN RXR ALPHA LIGAND BINDING DOMAIN BOUND TO THE EICOSANOID DHA (DOCOSA HEXAENOIC ACID) AND A COACTIVATOR PEPTIDE  |   TRANSCRIPTION REGULATION, NUCLEAR PROTEIN 
1mzn:C  (VAL1232) to  (ILE1442)  CRYSTAL STRUCTURE AT 1.9 ANGSTROEMS RESOLUTION OF THE HOMODIMER OF HUMAN RXR ALPHA LIGAND BINDING DOMAIN BOUND TO THE SYNTHETIC AGONIST COMPOUND BMS 649 AND A COACTIVATOR PEPTIDE  |   TRANSCRIPTION, NUCLEAR RECEPTOR, RETINOIC ACID RECEPTORS, AGONIST 
1mzn:G  (VAL3232) to  (LEU3441)  CRYSTAL STRUCTURE AT 1.9 ANGSTROEMS RESOLUTION OF THE HOMODIMER OF HUMAN RXR ALPHA LIGAND BINDING DOMAIN BOUND TO THE SYNTHETIC AGONIST COMPOUND BMS 649 AND A COACTIVATOR PEPTIDE  |   TRANSCRIPTION, NUCLEAR RECEPTOR, RETINOIC ACID RECEPTORS, AGONIST 
5die:A   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A TRIFLUORO-SUBSTITUTED A-CD RING ESTROGEN DERIVATIVE (1S,3AR, 5S,7AS)-7A-METHYL-5-(2,3,5-TRIFLUORO-4-HYDROXYPHENYL)OCTAHYDRO-1H- INDEN-1-OL  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
5dmf:B   (THR311) to   (LYS531)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 4-FLUOROPHENYLAMINO-SUBSTITUTED, METHYL TRIARYL-ETHYLENE DERIVATIVE 4,4'-(2-{3-[(4-FLUOROPHENYL)AMINO]PHENYL}PROP-1-ENE-1,1- DIYL)DIPHENOL  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
4poh:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF HUMAN RETINOID X RECEPTOR ALPHA-LIGAND BINDING DOMAIN COMPLEX WITH 8-METHYL UAB30 AND THE COACTIVATOR PEPTIDE GRIP-1  |   LIGAND BINDING DOMAIN, NUCLEAR RECEPTOR, CANCER, METHYL SUBSTITUTED REXINOID, 8-METHYL UAB30, TRANSCRIPTION 
4poj:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF HUMAN RETINOID X RECEPTOR ALPHA-LIGAND BINDING DOMAIN COMPLEX WITH 7-METHYL UAB30 AND THE COACTIVATOR PEPTIDE GRIP-1  |   LIGAND BINDING DOMAIN, NUCLEAR RECEPTOR, CANCER, LIPID TOXICITY, REXINOID, 7-METHYL UAB30, TRANSCRIPTION 
4pp3:A   (VAL232) to   (LEU441)  CRYSTAL STRUCTURE OF HUMAN RETINOID X RECEPTOR ALPHA-LIGAND BINDING DOMAIN COMPLEX WITH 6-METHYL UAB30 AND THE COACTIVATOR PEPTIDE GRIP-1  |   LIGAND BINDING DOMAIN, 6-METHYL UAB30, REXINOID, CANCER, LIPID TOXICITY, TRANSCRIPTION 
4pp5:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF HUMAN RETINOID X RECEPTOR ALPHA-LIGAND BINDING DOMAIN COMPLEX WITH 5-METHYL UAB30 AND THE COACTIVATOR PEPTIDE GRIP-1  |   LIGAND BINDING DOMAIN. 6-METHYL UAB30, REXINOID, CANCER, LIPID TOXICITY, LIGAND BINDING DOMAIN, 6-METHYL UAB30, TRANSCRIPTION 
4pp6:A   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH RESVERATROL  |   NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, NUCLEUS, PROTEIN BINDING 
1zaf:A   (SER264) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH 3-BROMO-6-HYDROXY-2-(4-HYDROXY-PHENYL)-INDEN-1-ONE  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST, TRANSCRIPTION/TRANSFERASE COMPLEX 
1zaf:B   (PRO265) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH 3-BROMO-6-HYDROXY-2-(4-HYDROXY-PHENYL)-INDEN-1-ONE  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST, TRANSCRIPTION/TRANSFERASE COMPLEX 
5dtv:A   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DIMETHYL-SUBSTITUTED, 3,4-DIARYLTHIOPHENE DIOXIDE CORE LIGAND  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
5du5:A   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DICHLORO-SUBSTITUTED, 3,4-DIARYLTHIOPHENE DIOXIDE CORE LIGAND  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
5dwg:A   (ALA312) to   (ASN532)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE TRIARYL-SUBSTITUTED IMINE ANALOG, 4-{(E)-(4-HYDROXYPHENYL) [(2-METHYLPHENYL)IMINO]METHYL}BENZENE-1,3-DIOL  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
5dxm:B   (THR311) to   (LYS531)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 3-[(E)-(1S,5S)-BICYCLO[3.3.1]NON-9- YLIDENE(4-HYDROXYPHENYL)METHYL]PHENOL  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
5dyd:A   (ALA312) to   (LYS531)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-{[(3S)-3-(METHYLSULFANYL) CYCLOHEXYLIDENE]METHANEDIYL}DIPHENOL  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
4q50:C   (THR311) to   (TYR526)  THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN D538G MUTANT IN COMPLEX WITH 4-HYDROXYTAMOXIFEN  |   ACQUIRED SERM-RESISTANCE, BREAST CANCER, ACTIVATING MUTATION, SERM-ER STRUCTURE, ALPHA HELIX, NUCLEAR HORMONE RECEPTOR, HORMONE BINDING PROTEIN 
5e19:A   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE METHYL {4-[BIS(4-HYDROXYPHENYL) METHYLIDENE]CYCLOHEXYL}ACETATE  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
5ei1:A   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH THE IMIDAZOPYRIDINE DERIVATIVE 2-(4-HYDROXYPHENYL)-3- IODANYL-IMIDAZO[1,2-A]PYRIDIN-6-OL  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
5ei1:B   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH THE IMIDAZOPYRIDINE DERIVATIVE 2-(4-HYDROXYPHENYL)-3- IODANYL-IMIDAZO[1,2-A]PYRIDIN-6-OL  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
2acl:A   (VAL232) to   (GLU434)  LIVER X-RECEPTOR ALPHA LIGAND BINDING DOMAIN WITH SB313987  |   NUCLEAR HORMONE RECEPTOR LIGAND BINDING DOMAIN TRANSCRIPTION FACTOR THREE LAYERED A-HELIX FOLD 
2acl:C   (VAL232) to   (GLU434)  LIVER X-RECEPTOR ALPHA LIGAND BINDING DOMAIN WITH SB313987  |   NUCLEAR HORMONE RECEPTOR LIGAND BINDING DOMAIN TRANSCRIPTION FACTOR THREE LAYERED A-HELIX FOLD 
2acl:E   (VAL232) to   (GLU434)  LIVER X-RECEPTOR ALPHA LIGAND BINDING DOMAIN WITH SB313987  |   NUCLEAR HORMONE RECEPTOR LIGAND BINDING DOMAIN TRANSCRIPTION FACTOR THREE LAYERED A-HELIX FOLD 
2acl:H   (PHE227) to   (ASP430)  LIVER X-RECEPTOR ALPHA LIGAND BINDING DOMAIN WITH SB313987  |   NUCLEAR HORMONE RECEPTOR LIGAND BINDING DOMAIN TRANSCRIPTION FACTOR THREE LAYERED A-HELIX FOLD 
5eit:A   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH THE IMIDAZOPYRIDINE DERIVATIVE 2-(4-HYDROXYPHENYL)-3- (TRIFLUOROMETHYL)IMIDAZO[1,2-A]PYRIDIN-6-OL  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
5eit:B   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH THE IMIDAZOPYRIDINE DERIVATIVE 2-(4-HYDROXYPHENYL)-3- (TRIFLUOROMETHYL)IMIDAZO[1,2-A]PYRIDIN-6-OL  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
4ree:B    (ALA31) to   (ASP249)  CRYSTAL STRUCTURE OF TR3 LBD IN COMPLEX WITH MOLECULE 6  |   LBD, TRANSCRIPTION 
4rfw:A   (VAL232) to   (ILE442)  CRYSTAL STRUCTURE OF HUMAN RETINOID X RECEPTOR ALPHA-LIGAND BINDING DOMAIN COMPLEX WITH 9CUAB70 AND THE COACTIVATOR PEPTIDE GRIP-1  |   LIGAND BINDING DOMAIN, CANCER PREVENTION, COACTIVATOR PEPTIDE, CONFORMATIONALLY CONSTRAINED RETINOIDS, TRANSCRIPTION 
4rmc:A   (VAL232) to   (LEU420)  CRYSTAL STRUCTURE OF HUMAN RETINOID X RECEPTOR ALPHA-LIGAND BINDING DOMAIN COMPLEX WITH 9CUAB76 AND THE COACTIVATOR PEPTIDE GRIP-1  |   LIGAND BINDING DOMAIN, CANCER PREVENTION, TRANSCRIPTION 
4rmd:A   (VAL232) to   (LEU441)  CRYSTAL STRUCTURE OF HUMAN RETINOID X RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEX WITH 9CUAB110 AND COACTIVATOR PEPTIDE GRIP-1  |   CANCER PREVENTION, LIGAND BINDING DOMAIN, TRANSCRIPTION 
3oap:A   (VAL232) to   (LEU420)  CRYSTAL STRUCTURE OF HUMAN RETINOID X RECEPTOR ALPHA-LIGAND BINDING DOMAIN COMPLEX WITH 9-CIS RETINOIC ACID AND THE COACTIVATOR PEPTIDE GRIP-1  |   ANTIPARALLEL SANDWICH, LIGAND BINDING, COACTIVATOR BINDING, DIMERIZATION, ACTIVATION FUNCTION, TRANSCRIPTION 
3oll:A   (PRO265) to   (ASN483)  CRYSTAL STRUCTURE OF PHOSPHORYLATED ESTROGEN RECEPTOR BETA LIGAND BINDING DOMAIN  |   STEROID BINDING, PHOSPHORYLATION, HORMONE RECEPTOR-ACTIVATOR COMPLEX 
3oll:B   (PRO265) to   (ASN483)  CRYSTAL STRUCTURE OF PHOSPHORYLATED ESTROGEN RECEPTOR BETA LIGAND BINDING DOMAIN  |   STEROID BINDING, PHOSPHORYLATION, HORMONE RECEPTOR-ACTIVATOR COMPLEX 
3omo:A   (PRO265) to   (ASN483)  FRAGMENT-BASED DESIGN OF NOVEL ESTROGEN RECEPTOR LIGANDS  |   STEROID BINDING, PROTEIN BINDING 
3omo:B   (PRO265) to   (ASN483)  FRAGMENT-BASED DESIGN OF NOVEL ESTROGEN RECEPTOR LIGANDS  |   STEROID BINDING, PROTEIN BINDING 
3omp:A   (PRO265) to   (ASN483)  FRAGMENT-BASED DESIGN OF NOVEL ESTROGEN RECEPTOR LIGANDS  |   STEROID BINDING, PROTEIN BINDING 
3omp:B   (PRO265) to   (ASN483)  FRAGMENT-BASED DESIGN OF NOVEL ESTROGEN RECEPTOR LIGANDS  |   STEROID BINDING, PROTEIN BINDING 
3omq:A   (PRO265) to   (ASN483)  FRAGMENT-BASED DESIGN OF NOVEL ESTROGEN RECEPTOR LIGANDS  |   STEROID BINDING, PROTEIN BINDING 
3omq:B   (PRO265) to   (ASN483)  FRAGMENT-BASED DESIGN OF NOVEL ESTROGEN RECEPTOR LIGANDS  |   STEROID BINDING, PROTEIN BINDING 
3ozj:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF HUMAN RETINOIC X RECEPTOR ALPHA COMPLEXED WITH BIGELOVIN AND COACTIVATOR SRC-1  |   NUCLEAR RECEPTOR LIGAND-BINDING DOMAIN, LIGAND-BINDING AND TRANSACTIVATION, TRANSCRIPTION 
3ozj:C   (GLU233) to   (GLY443)  CRYSTAL STRUCTURE OF HUMAN RETINOIC X RECEPTOR ALPHA COMPLEXED WITH BIGELOVIN AND COACTIVATOR SRC-1  |   NUCLEAR RECEPTOR LIGAND-BINDING DOMAIN, LIGAND-BINDING AND TRANSACTIVATION, TRANSCRIPTION 
5hjp:C   (VAL301) to   (GLY514)  IDENTIFICATION OF LXRBETA SELECTIVE AGONISTS FOR THE TREATMENT OF ALZHEIMER'S DISEASE  |   AGONIST, ALZHEIMER'S, SIGNALING PROTEIN 
4dk7:A   (THR221) to   (ASP446)  CRYSTAL STRUCTURE OF LXR LIGAND BINDING DOMAIN IN COMPLEX WITH FULL AGONIST 1  |   LIGAND BINDING DOMAIN, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION- PEPTIDE-AGONIST COMPLEX 
4dk8:A   (THR221) to   (ASP446)  CRYSTAL STRUCTURE OF LXR LIGAND BINDING DOMAIN IN COMPLEX WITH PARTIAL AGONIST 5  |   LIGAND BINDING DOMAIN, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION- PEPTIDE-AGONIST COMPLEX 
5hjs:A    (SER43) to   (ASP268)  IDENTIFICATION OF LXRBETA SELECTIVE AGONISTS FOR THE TREATMENT OF ALZHEIMER'S DISEASE  |   AGONIST, ALZHEIMER'S, SIGNALING PROTEIN 
4dm8:B  (TYR1180) to  (ILE1404)  CRYSTAL STRUCTURE OF RARB LBD IN COMPLEX WITH 9CIS RETINOIC ACID  |   NUCLEAR RECEPTOR, RARB, 9CIS RETINOIC ACID, ALPHA HELICAL SANDWICH, TRANSCRIPTION FACTOR, RETINOIC ACID, TRANSCRIPTION-PROTEIN BINDING COMPLEX 
5hyr:A   (THR311) to   (ASN532)  ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN Y537S MUTANT IN COMPLEX WITH STAPLED PEPTIDE SRC2-SP2 AND ESTRADIOL  |   BREAST CANCER, ESTROGEN RECEPTOR, SYNTHETIC PEPTIDE, STAPLED PEPTIDE, ENDOCRINE, HORMONE, GENE REGULATION 
5i4v:B   (VAL301) to   (ILE513)  DISCOVERY OF NOVEL, ORALLY EFFICACIOUS LIVER X RECEPTOR (LXR) BETA AGONISTS  |   LXRBETA-LBD, RXRBETA-LBD, HETERODIMER, AGONIST, DNA BINDING PROTEIN 
5i4v:F   (VAL301) to   (ILE513)  DISCOVERY OF NOVEL, ORALLY EFFICACIOUS LIVER X RECEPTOR (LXR) BETA AGONISTS  |   LXRBETA-LBD, RXRBETA-LBD, HETERODIMER, AGONIST, DNA BINDING PROTEIN 
3q95:A   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF HUMAN ESTROGEN RECEPTOR ALPHA LBD IN COMPLEX WITH GRIP PEPTIDE AND ESTRIOL  |   TRANSCRIPTIONAL REGULATOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATOR 
3r5m:A   (ASN227) to   (ILE442)  CRYSTAL STRUCTURE OF RXRALPHALBD COMPLEXED WITH THE AGONIST MAGNOLOL  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, TRANSCRIPTION-TRANSCRIPTION AGONIST COMPLEX 
5jy3:B   (ALA222) to   (GLN445)  CRYSTAL STRUCTURE OF LXRBETA (NUCLEAR RECEPTOR SUBFAMILY 1, GROUP H, MEMBER 2) COMPLEXED WITH BMS-852927  |   NHR, NR1H2, LXR-B, LXRB, UNR, NER-I, RIP15, NER, TRANSCRIPTION 
5jy3:D   (THR221) to   (GLN445)  CRYSTAL STRUCTURE OF LXRBETA (NUCLEAR RECEPTOR SUBFAMILY 1, GROUP H, MEMBER 2) COMPLEXED WITH BMS-852927  |   NHR, NR1H2, LXR-B, LXRB, UNR, NER-I, RIP15, NER, TRANSCRIPTION 
5kcc:B   (ALA312) to   (LYS529)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH OXABICYCLIC HEPTENE SULFONAMIDE (OBHS-N)  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
5kct:A   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-ETHYL, 4-CHLOROBENZYL OBHS-N DERIVATIVE  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
5kyj:B   (VAL301) to   (LEU512)  BRAIN PENETRANT LIVER X RECEPTOR (LXR) MODULATORS BASED ON A 2,4,5,6- TETRAHYDROPYRROLO[3,4-C]PYRAZOLE CORE  |   DNA BINDING PROTEIN, NUCLEAR RECEPTORS, LIVER X RECEPTOR, RETINOIC ACID X RECEPTOR, LXRBETA-LBD/RXRBETA-LBD HETERODIMER, CHEMICAL MODULATORS 
5kyj:F   (VAL301) to   (ILE513)  BRAIN PENETRANT LIVER X RECEPTOR (LXR) MODULATORS BASED ON A 2,4,5,6- TETRAHYDROPYRROLO[3,4-C]PYRAZOLE CORE  |   DNA BINDING PROTEIN, NUCLEAR RECEPTORS, LIVER X RECEPTOR, RETINOIC ACID X RECEPTOR, LXRBETA-LBD/RXRBETA-LBD HETERODIMER, CHEMICAL MODULATORS 
1a52:B   (THR311) to   (LYS531)  ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN COMPLEXED TO ESTRADIOL  |   RECEPTOR, ESTROGEN, LIGAND, TRANSCRIPTION REGULATION 
4whg:B    (ASN32) to   (ASP249)  CRYSTAL STRUCTURE OF TR3 LBD IN COMPLEX WITH MOLECULE 3  |   LBD, TRANSCRIPTION 
2p1t:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF THE LIGAND BINDING DOMAIN OF THE RETINOID X RECEPTOR ALPHA IN COMPLEX WITH 3-(2'-METHOXY)- TETRAHYDRONAPHTYL CINNAMIC ACID AND A FRAGMENT OF THE COACTIVATOR TIF-2  |   PROTEIN-LIGAND COMPLEX, HORMONE RECEPTOR 
3fug:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF THE RETINOID X RECEPTOR LIGAND BINDING DOMAIN BOUND TO THE SYNTHETIC AGONIST 3-[4-HYDROXY-3-(3,5, 5,8,8-PENTAMETHYL-5,6,7,8-TETRAHYDRONAPHTHALEN-2-YL)- PHENYL]ACRYLIC ACID  |   PROTEIN-LIGAND COMPLEX, HORMONE RECEPTOR, DNA-BINDING, HOST- VIRUS INTERACTION, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, UBL CONJUGATION, ZINC, ZINC-FINGER, ACTIVATOR, PHOSPHOPROTEIN, TRANSCRIPTION/TRANSCRIPTION REGULATOR COMPLEX 
2q70:A   (THR311) to   (MET528)  ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN COMPLXED TO A BENZOPYRAN LIGAND  |   TRANSCRIPTION FACTOR, ESTROGEN RECEPTOR 
1pqc:C   (ALA222) to   (ASP446)  HUMAN LXR BETA HORMONE RECEPTOR COMPLEXED WITH T0901317  |   LXRB+T0901317, TRANSCRIPTION REGULATION 
1pqc:D   (THR221) to   (ARG443)  HUMAN LXR BETA HORMONE RECEPTOR COMPLEXED WITH T0901317  |   LXRB+T0901317, TRANSCRIPTION REGULATION 
4j26:A   (PRO265) to   (ASN483)  ESTROGEN RECEPTOR IN COMPLEX WITH PROLINE-FLANKED LXXLL PEPTIDES  |   ESTROGEN RECEPTOR, PROLINE, LXXLL, ALPHA-HELIX, STRUCTURE STABILIZATION, HORMONE RECEPTOR-PEPTIDE COMPLEX 
4j26:B   (PRO265) to   (ASN483)  ESTROGEN RECEPTOR IN COMPLEX WITH PROLINE-FLANKED LXXLL PEPTIDES  |   ESTROGEN RECEPTOR, PROLINE, LXXLL, ALPHA-HELIX, STRUCTURE STABILIZATION, HORMONE RECEPTOR-PEPTIDE COMPLEX 
4k4j:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF HUMAN RETINOID X RECEPTOR ALPHA-LIGAND BINDING DOMAIN COMPLEX WITH 9CUAB30 AND THE COACTIVATOR PEPTIDE GRIP-1  |   LIGAND BINDING DOMAIN, CANCER, 9-CIS-UAB30, TRANSCRIPTION 
4znu:B   (THR311) to   (MET528)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH A 2-METHYL-SUBSTITUTED OBHS DERIVATIVE  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
1u3s:A   (PRO265) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-797  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1u3s:B   (PRO265) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-797  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1uom:A   (PRO336) to   (LEU525)  THE STRUCTURE OF ESTROGEN RECEPTOR IN COMPLEX WITH A SELECTIVE AND POTENT TETRAHYDROISOCHIOLIN LIGAND.  |   SELECTIVE ESTROGEN RECEPTOR MODULATORS, SERM, RECEPTOR, TRANSCRIPTION REGULATION, DNA-BINDING, NUCLEAR PROTEIN, ZINC-FINGER, STEROID-BINDING, PHOSPHORYLATION, POLYMORPHISM 3D-STRUCTURE, ALTERNATIVE SPLICING 
2jj3:A   (PRO265) to   (MET479)  ESTROGEN RECEPTOR BETA LIGAND BINDING DOMAIN IN COMPLEX WITH A BENZOPYRAN AGONIST  |   PHOSPHORYLATION, STEROID-BINDING, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, ALTERNATIVE SPLICING, LIGAND BINDING DOMAIN, ZINC, NUCLEUS, RECEPTOR, ZINC-FINGER, DNA-BINDING, TRANSCRIPTION, METAL-BINDING, LIPID-BINDING 
2jj3:B   (SER264) to   (MET479)  ESTROGEN RECEPTOR BETA LIGAND BINDING DOMAIN IN COMPLEX WITH A BENZOPYRAN AGONIST  |   PHOSPHORYLATION, STEROID-BINDING, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, ALTERNATIVE SPLICING, LIGAND BINDING DOMAIN, ZINC, NUCLEUS, RECEPTOR, ZINC-FINGER, DNA-BINDING, TRANSCRIPTION, METAL-BINDING, LIPID-BINDING 
1x76:B   (PRO265) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-697  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1x7j:A   (SER264) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH GENISTEIN  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1x7j:B   (SER264) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH GENISTEIN  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1xdk:A   (ALA231) to   (GLY448)  CRYSTAL STRUCTURE OF THE RARBETA/RXRALPHA LIGAND BINDING DOMAIN HETERODIMER IN COMPLEX WITH 9-CIS RETINOIC ACID AND A FRAGMENT OF THE TRAP220 COACTIVATOR  |   NUCLEAR RECEPTOR, COACTIVATOR, LIGAND, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX 
1xdk:E   (ALA231) to   (GLY448)  CRYSTAL STRUCTURE OF THE RARBETA/RXRALPHA LIGAND BINDING DOMAIN HETERODIMER IN COMPLEX WITH 9-CIS RETINOIC ACID AND A FRAGMENT OF THE TRAP220 COACTIVATOR  |   NUCLEAR RECEPTOR, COACTIVATOR, LIGAND, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX 
2yly:B   (PRO265) to   (MET479)  SULFONAMIDES AS SELECTIVE ESTROGEN RECEPTOR BETA AGONISTS.  |   RECEPTOR 
1mvc:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF THE HUMAN RXR ALPHA LIGAND BINDING DOMAIN BOUND TO THE SYNTHETIC AGONIST COMPOUND BMS 649 AND A COACTIVATOR PEPTIDE  |   NUCLEAR RECEPTOR, RETINOIC ACID, AGONIST RECOGNITION, TRANSCRIPTION FACTOR 
3kwy:A   (VAL232) to   (GLY443)  CRYSTAL STRUCTURE OF RXRALPHA LIGAND BINDING DOMAIN IN COMPLEX WITH TRIPHENYLTIN AND A COACTIVATOR FRAGMENT  |   NUCLEAR RECEPTOR TRANSCRIPTION ORGANOTIN, DNA-BINDING, HOST-VIRUS INTERACTION, ISOPEPTIDE BOND, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER, ACTIVATOR, PHOSPHOPROTEIN 
5dkb:B   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 3-METHYLPHENYLAMINO-SUBSTITUTED ETHYL TRIARYL-ETHYLENE DERIVATIVE 4,4'-(2-{3-[(3-METHYLPHENYL)AMINO]PHENYL}BUT-1-ENE-1,1- DIYL)DIPHENOL  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
1yy4:A   (SER264) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH 1-CHLORO-6-(4-HYDROXY-PHENYL)-NAPHTHALEN-2-OL  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1yy4:B   (SER264) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH 1-CHLORO-6-(4-HYDROXY-PHENYL)-NAPHTHALEN-2-OL  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
1yye:B   (SER264) to   (LYS482)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-202196  |   ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST 
5dx3:B   (THR311) to   (ASN532)  ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN Y537S MUTANT IN COMPLEX WITH STAPLED PEPTIDE SRC2-P3 AND ESTRADIOL  |   SYNTHETIC PEPTIDE, STAPLED PEPTIDE, ESTROGEN RECEPTOR ALPHA, SOMATIC MUTATION, PEPTIDE MIMETIC, AF-2 BINDING, HORMONE RECEPTOR-PEPTIDE COMPLEX 
5egv:B   (THR311) to   (ASN532)  CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX THE 3,4-DIARYL-FURAN DERIVATIVE 3-CHLORANYL-4-[4-(2- CHLORANYL-4-OXIDANYL-PHENYL)FURAN-3-YL]PHENOL  |   NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION 
4rme:A   (VAL232) to   (LEU420)  CRYSTAL STRUCTURE OF HUMAN RETINOID X RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEX WITH 9CUAB111 AND COACTIVATOR PEPTIDE GRIP-1  |   LIGAND BINDING DOMAIN, CANCER PREVENTION, TRANSCRIPTION 
3ols:A   (PRO265) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA LIGAND BINDING DOMAIN  |   STEROID BINDING, HORMONE RECEPTOR-ACTIVATOR COMPLEX 
3ols:B   (PRO265) to   (ASN483)  CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA LIGAND BINDING DOMAIN  |   STEROID BINDING, HORMONE RECEPTOR-ACTIVATOR COMPLEX 
4dm6:B  (TYR1180) to  (ILE1404)  CRYSTAL STRUCTURE OF RARB LBD HOMODIMER IN COMPLEX WITH TTNPB  |   TRANSCRIPTION, NUCLEAR RECEPTOR, RETINOIC ACID, ALPHA HELICAL SANDWICH, TRANSCRIPTION REGULATOR, RETINOIC ACID BINDING, NUCLEUS - CYTOPLASM, TRANSCRIPTION-PROTEIN BINDING COMPLEX 
5kya:B   (VAL301) to   (ILE513)  BRAIN PENETRANT LIVER X RECEPTOR (LXR) MODULATORS BASED ON A 2,4,5,6- TETRAHYDROPYRROLO[3,4-C]PYRAZOLE CORE  |   NUCLEAR RECEPTOR, LIVER X RECEPTOR, LXRBETA-LBD/RXRBETA-LBD HETERODIMER, CHEMICAL MODULATORS, DNA BINDING PROTEIN 
5kya:F   (VAL301) to   (ILE513)  BRAIN PENETRANT LIVER X RECEPTOR (LXR) MODULATORS BASED ON A 2,4,5,6- TETRAHYDROPYRROLO[3,4-C]PYRAZOLE CORE  |   NUCLEAR RECEPTOR, LIVER X RECEPTOR, LXRBETA-LBD/RXRBETA-LBD HETERODIMER, CHEMICAL MODULATORS, DNA BINDING PROTEIN