3eaw:X (GLN200) to (GLY300) REPLACEMENT OF VAL3 IN HUMAN THYMIDYLATE SYNTHASE AFFECTS ITS KINETIC PROPERTIES AND INTRACELLULAR STABILITY | TRANSFERASE, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS
1nje:A (LEU201) to (ASN303) THYMIDYLATE SYNTHASE WITH 2'-DEOXYCYTIDINE 5'-MONOPHOSPHATE (DCMP) | TRANSFERASE, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE (METHYLTRANSFERASE)
3ehi:X (GLN200) to (GLY300) CRYSTAL STRUCTURE OF HUMAN THYMIDYALTE SYNTHASE M190K WITH LOOP 181- 197 STABILIZED IN THE INACTIVE CONFORMATION | METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
1ajm:A (ALA148) to (GLY251) CRYSTAL STRUCTURE OF THYMIDYLATE SYNTHASE R126E MUTANT | TRANSFERASE, METHYLTRANSFERASE, DUMP
4h0r:A (LEU151) to (GLY253) CRYSTAL STRUCTURE OF THYMIDYLATE SYNTHASE FROM CORYNEBACTERIUM GLUTAMICUM | NUCLEOTIDE, DUMP, TRANSFERASE
4h0r:B (LEU151) to (GLY253) CRYSTAL STRUCTURE OF THYMIDYLATE SYNTHASE FROM CORYNEBACTERIUM GLUTAMICUM | NUCLEOTIDE, DUMP, TRANSFERASE
4h0u:A (LEU152) to (GLY253) CRYSTAL STRUCTURE OF THYMIDYLATE SYNTHASE FROM CORYNEBACTERIUM GLUTAMICUM IN COMPLEX WITH DUMP | NUCLEOTIDE,DUMP, TRANSFERASE
4h0u:B (LEU152) to (GLY253) CRYSTAL STRUCTURE OF THYMIDYLATE SYNTHASE FROM CORYNEBACTERIUM GLUTAMICUM IN COMPLEX WITH DUMP | NUCLEOTIDE,DUMP, TRANSFERASE
4h0u:C (LEU152) to (GLY253) CRYSTAL STRUCTURE OF THYMIDYLATE SYNTHASE FROM CORYNEBACTERIUM GLUTAMICUM IN COMPLEX WITH DUMP | NUCLEOTIDE,DUMP, TRANSFERASE
4h0u:D (LEU151) to (GLY253) CRYSTAL STRUCTURE OF THYMIDYLATE SYNTHASE FROM CORYNEBACTERIUM GLUTAMICUM IN COMPLEX WITH DUMP | NUCLEOTIDE,DUMP, TRANSFERASE
4h1i:A (LEU198) to (GLY300) STRUCTURE OF HUMAN THYMIDYLATE SYNTHASE AT LOW SALT CONDITIONS | NUCLEOTIDE METABOLISM, CANCER CHEMOTHERAPY TARGET, METHYL TRANSFERASE, TRANSFERASE
1aob:A (ALA148) to (GLY251) E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH DDURD | TRANSFERASE (METHYLTRANSFERASE), SUBSTRATE MODULES
1bid:A (PHE149) to (GLY251) E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH DUMP | TRANSFERASE (METHYLTRANSFERASE), SUBSTRATE MODULES, METHYLTRANSFERASE
1bko:B (TYR163) to (ASN266) THERMOSTABLE THYMIDYLATE SYNTHASE A FROM BACILLUS SUBTILIS | METHYLTRANSFERASE, DTMP SYNTHASE
1bkp:A (TYR163) to (ASN266) THERMOSTABLE THYMIDYLATE SYNTHASE A FROM BACILLUS SUBTILIS | METHYLTRANSFERASE, DTMP SYNTHASE
1bq1:A (PHE149) to (GLY251) E. COLI THYMIDYLATE SYNTHASE MUTANT N177A IN COMPLEX WITH CB3717 AND 2'-DEOXYURIDINE 5'-MONOPHOSPHATE (DUMP) | TRANSFERASE, ACTIVE SITE MUTANT, REACTION INTERMEDIATE
1bsf:A (TYR163) to (ASN266) THERMOSTABLE THYMIDYLATE SYNTHASE A FROM BACILLUS SUBTILIS | METHYLTRANSFERASE, DTMP SYNTHASE
1bsf:B (TYR163) to (ASN266) THERMOSTABLE THYMIDYLATE SYNTHASE A FROM BACILLUS SUBTILIS | METHYLTRANSFERASE, DTMP SYNTHASE
1bsp:A (TYR163) to (GLY270) THERMOSTABLE THYMIDYLATE SYNTHASE A FROM BACILLUS SUBTILIS | METHYLTRANSFERASE, DTMP SYNTHASE
1bsp:B (TYR163) to (ASN266) THERMOSTABLE THYMIDYLATE SYNTHASE A FROM BACILLUS SUBTILIS | METHYLTRANSFERASE, DTMP SYNTHASE
1ddu:A (PHE149) to (GLY251) E. COLI THYMIDYLATE SYNTHASE IN COMPLEX WITH CB3717 AND 2', 5'-DIDEOXYURIDINE (DDURD) | TRANSFERASE (METHYLTRANSFERASE), SUBSTRATE MODULES
1ddu:B (ALA148) to (GLY251) E. COLI THYMIDYLATE SYNTHASE IN COMPLEX WITH CB3717 AND 2', 5'-DIDEOXYURIDINE (DDURD) | TRANSFERASE (METHYLTRANSFERASE), SUBSTRATE MODULES
4xsc:A (LEU186) to (GLY288) COMPLEX STRUCTURE OF THYMIDYLATE SYNTHASE FROM VARICELLA ZOSTER VIRUS WITH A PHOSPHORYLATED BVDU | VZV, THYMIDYLATE SYNTHASE, HERPESVIRUS, TRANSFERASE
4xsc:C (LEU186) to (GLY288) COMPLEX STRUCTURE OF THYMIDYLATE SYNTHASE FROM VARICELLA ZOSTER VIRUS WITH A PHOSPHORYLATED BVDU | VZV, THYMIDYLATE SYNTHASE, HERPESVIRUS, TRANSFERASE
4xse:B (LEU186) to (GLY288) COMPLEX STRUCTURE OF THYMIDYLATE SYNTHASE FROM VARICELLA ZOSTER VIRUS | THYMIDYLATE SYNTHASE, HERPESVIRUS, VARICELLA ZOSTER VIRUS, VZV, VIRAL PROTEIN
3gg5:D (ALA197) to (GLY300) REPLACEMENT OF VAL3 IN HUMAN THYMIDYLATE SYNTHASE AFFECTS ITS KINETIC PROPERTIES AND INTRACELLULAR STABILITY | METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
4jef:A (HIS196) to (GLY300) CRYSTAL STRUCTURE OF HUMAN THYMIDYLATE SYNTHASE Y202A IN INACTIVE CONFORMATION. | INACTIVE FORM OF HUMAN THYMIDYLATE SYNTHASE, HOT SPOT RESIDUE, TRANSFERASE
1f4b:A (ALA148) to (GLY251) CRYSTAL STRUCTURE OF ESCHERICHIA COLI THYMIDYLATE SYNTHASE | E. COLI THYMIDYLATE SYNTHASE, TRANSFERASE
1f4c:A (ALA148) to (GLY251) CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COVALENTLY MODIFIED AT C146 WITH N-[TOSYL-D-PROLINYL]AMINO-ETHANETHIOL | E. COLI THYMIDYLATE SYNTHASE MODIFIED AT CYSTEINE 146, TRANSFERASE
1f4c:B (PHE149) to (GLY251) CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COVALENTLY MODIFIED AT C146 WITH N-[TOSYL-D-PROLINYL]AMINO-ETHANETHIOL | E. COLI THYMIDYLATE SYNTHASE MODIFIED AT CYSTEINE 146, TRANSFERASE
1f4d:B (PHE149) to (GLY251) CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE C146S, L143C COVALENTLY MODIFIED AT C143 WITH N-[TOSYL-D-PROLINYL]AMINO- ETHANETHIOL | CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE C146S, L143C COVALENTLY MODIFIED AT C143 WITH N-[TOSYL-D-PROLINYL]AMINO- ETHANETHIOL, TRANSFERASE
1f4e:A (ALA148) to (GLY251) CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH TOSYL-D-PROLINE | CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH TOSYL-D-PROLINE, TRANSFERASE
1f4f:A (ALA148) to (GLY251) CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH SP- 722 | CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH SP- 722, TRANSFERASE
1f4f:B (ALA148) to (GLY251) CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH SP- 722 | CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH SP- 722, TRANSFERASE
1f4g:A (ALA148) to (GLY251) CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH SP- 876 | CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH SP- 876, TRANSFERASE
1f4g:B (ALA148) to (GLY251) CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH SP- 876 | CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH SP- 876, TRANSFERASE
1ffl:A (ALA148) to (GLY251) CRYSTAL STRUCTURE OF THE APO-THYMIDYLATE SYNTHASE R166Q MUTANT | TRANSFERASE, METHYLTRANSFERASE
3um5:B (LEU493) to (ASN595) DOUBLE MUTANT (A16V+S108T) PLASMODIUM FALCIPARUM DIHYDROFOLATE REDUCTASE-THYMIDYLATE SYNTHASE (PFDHFR-TS-T9/94) COMPLEXED WITH PYRIMETHAMINE, NADPH, AND DUMP | MALARIAL DHFR-TS, PYRIMETHAMINE, ANTIFOLATE, NAPDH, DUMP, OXIDOREDUCTASE, TRANSFERASE-INHIBITOR COMPLEX
3um6:B (LEU493) to (ASN595) DOUBLE MUTANT (A16V+S108T) PLASMODIUM FALCIPARUM DHFR-TS (T9/94) COMPLEXED WITH CYCLOGUANIL, NADPH AND DUMP | MALARIAL DHFR-TS, CYCLOGUANIL, ANTIFOLATE, NAPDH, DUMP, OXIDOREDUCTASE, TRANSFERASE-INHIBITOR COMPLEX
3uwl:A (MET200) to (GLY302) CRYSTAL STRUCTURE OF ENTEROCCOCUS FAECALIS THYMIDYLATE SYNTHASE (EFTS) IN COMPLEX WITH 5-FORMYL TETRAHYDROFOLATE | METHYLTRANSFERASE, TRANSFERASE
3uwl:C (MET200) to (GLY302) CRYSTAL STRUCTURE OF ENTEROCCOCUS FAECALIS THYMIDYLATE SYNTHASE (EFTS) IN COMPLEX WITH 5-FORMYL TETRAHYDROFOLATE | METHYLTRANSFERASE, TRANSFERASE
2fto:X (ALA148) to (GLY251) Y94F MUTANT OF THYMIDYLATE SYNTHASE BOUND TO THYMIDINE-5'-PHOSPHATE AND 10-PROPARGYL-5,8-DIDEAZAFOLID ACID | METHYLTRANSFERASE, TRANSFERASE
2ftq:A (PHE149) to (GLY251) E. COLI THYMIDYLATE SYNTHASE AT 1.8 A RESOLUTION | METHYLTRANSFERASE, TRANSFERASE
4knz:A (ALA148) to (GLY251) THYMIDYLATE SYNTHASE TERNARY COMPLEX WITH DUMP AND CB3717 | ALPHA/BETA PROTEIN, METHYLTRANSFERASE, METHYLENETETRAHYDROFOLATE, ANTIFOLATE, TRANSFERASE
4knz:B (ALA148) to (GLY251) THYMIDYLATE SYNTHASE TERNARY COMPLEX WITH DUMP AND CB3717 | ALPHA/BETA PROTEIN, METHYLTRANSFERASE, METHYLENETETRAHYDROFOLATE, ANTIFOLATE, TRANSFERASE
3i3r:A (PHE396) to (ASP498) X-RAY STRUCTURE DIHYDROFOLATE REDUCTASE/THYMIDYLATE SYNTHASE FROM BABESIA BOVIS AT 2.35A RESOLUTION | SSGCID, BABESIA BOVIS, DIHYDROFOLATE REDUCTASE, THYMIDYLATE SYNTHASE, METHYLTRANSFERASE, TRANSFERASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE
3i3r:B (PHE396) to (ASP498) X-RAY STRUCTURE DIHYDROFOLATE REDUCTASE/THYMIDYLATE SYNTHASE FROM BABESIA BOVIS AT 2.35A RESOLUTION | SSGCID, BABESIA BOVIS, DIHYDROFOLATE REDUCTASE, THYMIDYLATE SYNTHASE, METHYLTRANSFERASE, TRANSFERASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE
2g8x:A (ALA148) to (GLY251) ESCHERICHIA COLI Y209W APOPROTEIN | BETA SHEET, ALPHA/BETA PROTEIN, DTT, TRANSFERASE
1syn:A (ALA148) to (GLY251) E. COLI THYMIDYLATE SYNTHASE IN COMPLEX WITH BW1843U89 AND 2'-DEOXYURIDINE 5'-MONOPHOSPHATE (DUMP) | TRANSFERASE (METHYLTRANSFERASE)
3ihi:A (LEU192) to (HIS298) CRYSTAL STRUCTURE OF MOUSE THYMIDYLATE SYNTHASE | PROTEIN-LIGAND COMPLEX, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
3ihi:B (LEU192) to (GLY294) CRYSTAL STRUCTURE OF MOUSE THYMIDYLATE SYNTHASE | PROTEIN-LIGAND COMPLEX, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
3ijz:A (THR200) to (ASN303) LACTOBACILLUS CASEI THYMIDYLATE SYNTHASE TERNARY COMPLEX WITH DUMP AND PTHALIMIDIC DERIVATIVE 15C | TRANSFERASE, NUCLEOTIDE SYNTHASE, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS
3ik0:A (LEU201) to (ASN303) LACTOBACILLUS CASEI THYMIDYLATE SYNTHASE IN TERNARY COMPLEX WITH DUMP AND THE PHTALIMIDIC DERIVATIVE 7C1 | TRANSFERASE, NUCLEOTIDE SYNTHASE, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS
3ik1:A (LEU201) to (ASN303) LACTOBACILLUS CASEI THYMIDYLATE SYNTHASE IN TERNARY COMPLEX WITH DUMP AND THE PHTALIMIDIC DERIVATIVE 20C | TRANSFERASE, NUCLEOTIDE SYNTHASE, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS
1tdu:A (ALA148) to (GLY251) E. COLI THYMIDYLATE SYNTHASE IN COMPLEX WITH CB3717 AND 2'- DEOXYURIDINE (DURD) | TRANSFERASE (METHYLTRANSFERASE), SUBSTRATE MODULES
1tsn:A (ALA148) to (GLY251) THYMIDYLATE SYNTHASE TERNARY COMPLEX WITH FDUMP AND METHYLENETETRAHYDROFOLATE | TRANSFERASE, METHYLTRANSFERASE
1tys:A (ALA148) to (GLY251) WATER-MEDIATED SUBSTRATE(SLASH)PRODUCT DISCRIMINATION: THE PRODUCT COMPLEX OF THYMIDYLATE SYNTHASE AT 1.83 ANGSTROMS | TRANSFERASE, METHYLTRANSFERASE
1i00:A (LEU198) to (GLY300) CRYSTAL STRUCTURE OF HUMAN THYMIDYLATE SYNTHASE, TERNARY COMPLEX WITH DUMP AND TOMUDEX | THYMIDYLATE SYNTHASE, HUMAN, TERNARY COMPLEX, DUMP, TOMUDEX, OPEN CONFORMATION, TRANSFERASE
4lrr:A (PHE149) to (GLY251) TERNARY COMPLEX BETWEEN E. COLI THYMIDYLATE SYNTHASE, DUMP, AND F9 | THYMIDINE MONOPHOSPHATE SYNTHESIS, N-TERMINAL ACETYLATED METHIONINE, BETA-MERCAPTOETHANOL MODIFIED CYSTEINE, TRANSFERASE
1j3i:C (LEU493) to (HIS599) WILD-TYPE PLASMODIUM FALCIPARUM DIHYDROFOLATE REDUCTASE- THYMIDYLATE SYNTHASE (PFDHFR-TS) COMPLEXED WITH WR99210, NADPH, AND DUMP | BIFUNCTIONAL, OXIDOREDUCTASE, TRANSFERASE
1j3j:D (LEU493) to (HIS599) DOUBLE MUTANT (C59R+S108N) PLASMODIUM FALCIPARUM DIHYDROFOLATE REDUCTASE-THYMIDYLATE SYNTHASE (PFDHFR-TS) COMPLEXED WITH PYRIMETHAMINE, NADPH, AND DUMP | BIFUNCTIONAL, OXIDOREDUCTASE, TRANSFERASE
1jg0:A (ALA148) to (GLY251) CRYSTAL STRUCTURE OF ESCHERICHIA COLI THYMIDYLATE SYNTHASE COMPLEXED WITH 2'-DEOXYURIDINE-5'-MONOPHOSPHATE AND N,O-DIDANSYL-L-TYROSINE | THYMIDYLATE SYNTHASE, DIDANSYL TYROSINE, TRANSFERASE
1jg0:B (PHE149) to (GLY251) CRYSTAL STRUCTURE OF ESCHERICHIA COLI THYMIDYLATE SYNTHASE COMPLEXED WITH 2'-DEOXYURIDINE-5'-MONOPHOSPHATE AND N,O-DIDANSYL-L-TYROSINE | THYMIDYLATE SYNTHASE, DIDANSYL TYROSINE, TRANSFERASE
1vzd:A (THR200) to (ASN303) L. CASEI THYMIDYLATE SYNTHASE MUTANT E60Q TERNARY COMPLEX WITH FDUMP AND CB3717 | METHYLTRANSFERASE, NUCLEOTIDE SYNTHASE
5by6:D (CYS191) to (ASN294) CRYSTAL STRUCTURE OF TRICHINELLA SPIRALIS THYMIDYLATE SYNTHASE COMPLEXED WITH DUMP | TRICHINELLA SPIRALIS, PARASITIC NEMATODE, PROTEIN-LIGAND COMPLEX, METHYLTRANSFERASE, TRANSFERASE
4o1x:A (SER195) to (GLY300) CRYSTAL STRUCTURE OF HUMAN THYMIDYLATE SYNTHASE DOUBLE MUTANT C195S- Y202C | DIMER-DIMER INTERFACE MODIFICATION, ACTIVE CONFORMATION, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
4o1x:B (SER195) to (GLY300) CRYSTAL STRUCTURE OF HUMAN THYMIDYLATE SYNTHASE DOUBLE MUTANT C195S- Y202C | DIMER-DIMER INTERFACE MODIFICATION, ACTIVE CONFORMATION, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
4o7u:C (THR199) to (GLY302) ETHEROCOMPLEX OF ENTEROCCOCUS FAECALIS THYMIDYLATE SYNTHASE WITH 5- HYDROXYMETHILENE-6-HYDROFOLIC ACID AND THE PHTALIMIDIC INHIBITOR SS7 | TRANSFERASE, FOLATE BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3k2h:B (CYS395) to (ASP498) CO-CRYSTAL STRUCTURE OF DIHYDROFOLATE REDUCTASE/THYMIDYLATE SYNTHASE FROM BABESIA BOVIS WITH DUMP, PEMETREXED AND NADP | NIAID, SSGCID, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, ALIMTA, FOLIC ACID ANALOG, THYA, FOLATE ANTIMETABOLITES, TIC-BORNE PARASITIC PROTOZOAN, BABESIOSIS, MALARIA-LIKE DISEASE, METHYLTRANSFERASE, TRANSFERASE
3kjr:A (CYS395) to (ASP498) CRYSTAL STRUCTURE OF DIHYDROFOLATE REDUCTASE/THYMIDYLATE SYNTHASE FROM BABESIA BOVIS DETERMINED USING SLIPCHIP BASED MICROFLUIDICS | MICROFLUIDICS, SLIPCHIP,STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, ACCELERATED TECHNOLOGIES CENTER FOR GENE TO 3D STRUCTURE, ATCG3D, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, METHYLTRANSFERASE, TRANSFERASE, SSGCID
3kjr:B (CYS395) to (ASP498) CRYSTAL STRUCTURE OF DIHYDROFOLATE REDUCTASE/THYMIDYLATE SYNTHASE FROM BABESIA BOVIS DETERMINED USING SLIPCHIP BASED MICROFLUIDICS | MICROFLUIDICS, SLIPCHIP,STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, ACCELERATED TECHNOLOGIES CENTER FOR GENE TO 3D STRUCTURE, ATCG3D, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, METHYLTRANSFERASE, TRANSFERASE, SSGCID
2a9w:A (ALA148) to (GLY251) E. COLI TS COMPLEXED WITH DUMP AND INHIBITOR GA9 | PROTEIN-INHIBITOR COMPLEX, TRANSFERASE
2a9w:C (ALA148) to (GLY251) E. COLI TS COMPLEXED WITH DUMP AND INHIBITOR GA9 | PROTEIN-INHIBITOR COMPLEX, TRANSFERASE
2a9w:D (PHE149) to (GLY251) E. COLI TS COMPLEXED WITH DUMP AND INHIBITOR GA9 | PROTEIN-INHIBITOR COMPLEX, TRANSFERASE
3bfi:A (ALA148) to (GLY251) E. COLI THYMIDYLATE SYNTHASE Y209M MUTANT COMPLEXED WITH 5-NITRO-DUMP | METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, REPRESSOR, RNA-BINDING, TRANSLATION REGULATION, TRANSFERASE
3bhl:A (ALA148) to (GLY251) E.COLI THYMIDYLATE SYNTHASE COMPLEXES WITH 5-NO2DUMP AND TETRAHYDROFOLATE AT 1.4 A RESOLUTION | METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, REPRESSOR, RNA-BINDING, TRANSLATION REGULATION, TRANSFERASE
3bhl:B (ALA148) to (GLY251) E.COLI THYMIDYLATE SYNTHASE COMPLEXES WITH 5-NO2DUMP AND TETRAHYDROFOLATE AT 1.4 A RESOLUTION | METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, REPRESSOR, RNA-BINDING, TRANSLATION REGULATION, TRANSFERASE
3bhr:A (ALA148) to (GLY251) E. COLI TS COMPLEXED WITH 5-NO2DUMP AND TETRAHYDROFOLATE AT 1.9 A RESOLUTION (SPACE GROUP 152) | METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, REPRESSOR, RNA-BINDING, TRANSLATION REGULATION, TRANSFERASE
3byx:A (LEU201) to (ASN303) LACTOBACILLUS CASEI THYMIDYLATE SYNTHASE TERNARY COMPLEX WITH DUMP AND THE PHTALIMIDIC DERIVATIVE C00 IN MULTIPLE BINDING MODES | STRUCTURE BASED DRUG DESIGN, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
3c0a:A (THR200) to (ASN303) LACTOBACILLUS CASEI THYMIDYLATE SYNTHASE TERNARY COMPLEX WITH DUMP AND THE PHTALIMIDIC DERIVATIVE 14C IN MULTIPLE BINDING MODES-MODE 2 | METHYLTRANSFERASE, STRUCTURE-BASED DRUG DESIGN, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
5fct:A (LEU192) to (GLY294) MOUSE THYMIDYLATE SYNTHASE IN TERNARY COMPLEX WITH FDUMP AND METHYLENETETRAHYDROFOLATE. | COMPLEX, ENZYME, INHIBITOR, COFACTOR, TRANSFERASE
5fct:B (LEU192) to (GLY294) MOUSE THYMIDYLATE SYNTHASE IN TERNARY COMPLEX WITH FDUMP AND METHYLENETETRAHYDROFOLATE. | COMPLEX, ENZYME, INHIBITOR, COFACTOR, TRANSFERASE
3n5e:A (HIS208) to (GLY312) CRYSTAL STRUCTURE OF HUMAN THYMIDYLATE SYNTHASE BOUND TO A PEPTIDE INHIBITOR | PEPTIDE INHIBITOR, PROTEIN-PEPTIDE COMPLEX, INTERFACE INHIBITOR, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3n5e:B (HIS208) to (GLY312) CRYSTAL STRUCTURE OF HUMAN THYMIDYLATE SYNTHASE BOUND TO A PEPTIDE INHIBITOR | PEPTIDE INHIBITOR, PROTEIN-PEPTIDE COMPLEX, INTERFACE INHIBITOR, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3n5g:A (GLN212) to (GLY312) CRYSTAL STRUCTURE OF HISTIDINE-TAGGED HUMAN THYMIDYLATE SYNTHASE | PEPTIDE INHIBITOR, PROTEIN-PEPTIDE COMPLEX, INTERFACE INHIBITOR, TRANSFERASE
3cl9:A (LEU405) to (PHE495) STRUCTURE OF BIFUNCTIONAL TCDHFR-TS IN COMPLEX WITH MTX | BIFUNCTIONAL ENZYME IN COMPLEX WITH NADP, MTX AND DUMP, METHYLTRANSFERASE, MULTIFUNCTIONAL ENZYME, NUCLEOTIDE BIOSYNTHESIS, ONE-CARBON METABOLISM, OXIDOREDUCTASE, TRANSFERASE, OXIDOREDUCTASE- TRANSFERASE COMPLEX
3nrr:A (CYS395) to (ASP498) CO-CRYSTAL STRUCTURE OF DIHYDROFOLATE REDUCTASE-THYMIDYLATE SYNTHASE FROM BABESIA BOVIS WITH DUMP, RALTITREXED AND NADP | STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, SSGCID, NIAID, DIHYDROFOLATE REDUCTASE, THYMIDYLATE SYNTHASE, DHFR, TS, THYA, OXIDOREDUCTASE, METHYLTRANSFERASE, BABESIOSIS, DUMP, NADP, RALTITREXED, TOMUDEX, TRANSFERASE
3nrr:B (CYS395) to (ASP498) CO-CRYSTAL STRUCTURE OF DIHYDROFOLATE REDUCTASE-THYMIDYLATE SYNTHASE FROM BABESIA BOVIS WITH DUMP, RALTITREXED AND NADP | STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, SSGCID, NIAID, DIHYDROFOLATE REDUCTASE, THYMIDYLATE SYNTHASE, DHFR, TS, THYA, OXIDOREDUCTASE, METHYLTRANSFERASE, BABESIOSIS, DUMP, NADP, RALTITREXED, TOMUDEX, TRANSFERASE
3ob7:C (ALA197) to (HIS304) HUMAN THYMIDYLATE SYNTHASE R163K WITH CYS 195 COVALENTLY MODIFIED BY GLUTATHIONE | METHYLTRANSFERASE, TRANSFERASE
5hs3:B (LEU198) to (GLY300) HUMAN THYMIDYLATE SYNTHASE COMPLEXED WITH DUMP AND 3-AMINO-2-BENZOYL- 4-METHYLTHIENO[2,3-B]PYRIDIN-6-OL | NHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hs3:F (LEU198) to (GLY300) HUMAN THYMIDYLATE SYNTHASE COMPLEXED WITH DUMP AND 3-AMINO-2-BENZOYL- 4-METHYLTHIENO[2,3-B]PYRIDIN-6-OL | NHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4dq1:B (MET204) to (ASP305) THYMIDYLATE SYNTHASE FROM STAPHYLOCOCCUS AUREUS. | STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, STRUCTURES OF MTB PROTEINS CONFERRING SUSCEPTIBILITY TO KNOWN MTB INHIBITORS, MTBI, THYMIDYLATE SYNTHASE, TRANSFERASE
4e28:A (HIS196) to (GLY300) STRUCTURE OF HUMAN THYMIDYLATE SYNTHASE IN INACTIVE CONFORMATION WITH A NOVEL NON-PEPTIDIC INHIBITOR | HUMAN THYMIDYLATE SYNTHASE (HTS) INACTIVE CONFORMATION, HTS-INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e5o:A (LEU192) to (HIS298) CRYSTAL STRUCTURE OF MOUSE THYMIDYLATE SYNTHASE IN COMPLEX WITH DUMP | PROTEIN-LIGAND COMPLEX, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
4e5o:B (LEU192) to (GLY294) CRYSTAL STRUCTURE OF MOUSE THYMIDYLATE SYNTHASE IN COMPLEX WITH DUMP | PROTEIN-LIGAND COMPLEX, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
4e5o:C (LEU192) to (HIS298) CRYSTAL STRUCTURE OF MOUSE THYMIDYLATE SYNTHASE IN COMPLEX WITH DUMP | PROTEIN-LIGAND COMPLEX, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
4e5o:D (LEU192) to (HIS298) CRYSTAL STRUCTURE OF MOUSE THYMIDYLATE SYNTHASE IN COMPLEX WITH DUMP | PROTEIN-LIGAND COMPLEX, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
4e5o:F (LEU192) to (GLY294) CRYSTAL STRUCTURE OF MOUSE THYMIDYLATE SYNTHASE IN COMPLEX WITH DUMP | PROTEIN-LIGAND COMPLEX, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
4eb4:B (LEU192) to (GLY294) CRYSTAL STRUCTURE OF MOUSE THYMIDYLATE SYNTHASE IN TERNARY COMPLEX WITH DUMP AND TOMUDEX | TERNARY COMPLEX, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
4eb4:D (LEU192) to (ARG277) CRYSTAL STRUCTURE OF MOUSE THYMIDYLATE SYNTHASE IN TERNARY COMPLEX WITH DUMP AND TOMUDEX | TERNARY COMPLEX, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
4ein:B (LEU192) to (HIS298) CRYSTAL STRUCTURE OF MOUSE THYMIDYLATE SYNTHASE IN BINARY COMPLEX WITH A SUBSTRATE ANALOGUE AND STRONG INHIBITOR, N(4)-HYDROXY-2'- DEOXYCYTIDINE-5'-MONOPHOSPHATE | METHYLTRANSFERASE, BINDING SITE, CATALYSIS, DIMERIZATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ez8:A (LEU192) to (GLY294) CRYSTAL STRUCTURE OF MOUSE THYMIDYLATE SYTHASE IN TERNARY COMPLEX WITH N(4)-HYDROXY-2'-DEOXYCYTIDINE-5'-MONOPHOSPHATE AND THE COFACTOR PRODUCT, DIHYDROFOLATE | METHYLTRANSFERASE, TERNARY COMPLEX, DIHYDROFOLIC ACID, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4f2v:A (ALA148) to (GLY251) CRYSTAL STRUCTURE OF DE NOVO DESIGNED SERINE HYDROLASE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM (NESG) TARGET OR165 | STRUCTURAL GENOMICS, PSI-BIOLOGY, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, NESG, DE NOVO DESIGN, DE NOVO PROTEIN
3qgt:A (LEU493) to (HIS599) CRYSTAL STRUCTURE OF WILD-TYPE PFDHFR-TS COMPLEXED WITH NADPH, DUMP AND PYRIMETHAMINE | MALARIAL DHFR-TS ANTIFOLATE COMPLEX, ROSSMANN FOLD, REDUCTASE, DIHYDROFOLATE BINDING, DUMP BINDING, NADPH BINDING, OXIDOREDUCTASE, TRANSFERASE-INHIBITOR COMPLEX
3qgt:B (LEU493) to (ASN595) CRYSTAL STRUCTURE OF WILD-TYPE PFDHFR-TS COMPLEXED WITH NADPH, DUMP AND PYRIMETHAMINE | MALARIAL DHFR-TS ANTIFOLATE COMPLEX, ROSSMANN FOLD, REDUCTASE, DIHYDROFOLATE BINDING, DUMP BINDING, NADPH BINDING, OXIDOREDUCTASE, TRANSFERASE-INHIBITOR COMPLEX
3qj7:B (PHE149) to (ASN250) CRYSTAL STRUCTURE OF THE MYCOBACTERIUM TUBERCULOSIS THYMIDYLATE SYNTHASE (THYA) BOUND TO DUMP | THYMIDILATE SYNTHASE, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, TRANSFERASE
5j7w:A (MET200) to (GLY302) ENTEROCOCCUS FAECALIS THYMIDYLATE SYNTHASE COMPLEX WITH METHOTREXATE | ENTEROCOCCUS FAECALIS, THYMIDYLATE SYNTHASE, METHOTREXATE, COMPLEX, TRANSFERASE
4fgt:A (GLN200) to (GLY300) ALLOSTERIC PEPTIDIC INHIBITOR OF HUMAN THYMIDYLATE SYNTHASE THAT STABILIZES INACTIVE CONFORMATION OF THE ENZYME. | DIMER, MUTANT K47A OF HTS, INACTIVE HTS CONFORMATION, HTS COMPLEX WITH PEPTIDIC INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gd7:A (HIS196) to (GLY300) WILD-TYPE HUMAN THYMIDYLATE SYNTHASE WITH BOUND PURPUROGALLIN | METHYLTRANSFERASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ebu:A (HIS196) to (GLY300) REPLACEMENT OF VAL3 IN HUMAN THYMIDYLATE SYNTHASE AFFECTS ITS KINETIC PROPERTIES AND INTRACELLULAR STABILITY | TRANSFERASE, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS
4gyh:A (HIS196) to (GLY300) STRUCTURE OF HUMAN THYMIDYLATE SYNTHASE AT HIGH SALT CONDITIONS | METHYL TRANSFERASE, TRANSFERASE
1aiq:A (ALA148) to (GLY251) CRYSTAL STRUCTURE OF THYMIDYLATE SYNTHASE R126E MUTANT | TRANSFERASE, METHYLTRANSFERASE
1an5:A (PHE149) to (GLY251) E. COLI THYMIDYLATE SYNTHASE IN COMPLEX WITH CB3717 | TRANSFERASE (METHYLTRANSFERASE), SUBSTRATE MODULES
4isk:A (ALA148) to (GLY251) CRYSTAL STRUCTURE OF E.COLI THYMIDYLATE SYNTHASE WITH DUMP AND THE BGC 945 INHIBITOR | ALPHA/BETA PROTEIN, METHYLASE, METHYLTRANSFERASE, DUMP SUBTRATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4isk:D (ALA148) to (GLY251) CRYSTAL STRUCTURE OF E.COLI THYMIDYLATE SYNTHASE WITH DUMP AND THE BGC 945 INHIBITOR | ALPHA/BETA PROTEIN, METHYLASE, METHYLTRANSFERASE, DUMP SUBTRATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4isk:E (ALA148) to (GLY251) CRYSTAL STRUCTURE OF E.COLI THYMIDYLATE SYNTHASE WITH DUMP AND THE BGC 945 INHIBITOR | ALPHA/BETA PROTEIN, METHYLASE, METHYLTRANSFERASE, DUMP SUBTRATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4isk:F (ALA148) to (GLY251) CRYSTAL STRUCTURE OF E.COLI THYMIDYLATE SYNTHASE WITH DUMP AND THE BGC 945 INHIBITOR | ALPHA/BETA PROTEIN, METHYLASE, METHYLTRANSFERASE, DUMP SUBTRATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4isk:H (ALA148) to (GLY251) CRYSTAL STRUCTURE OF E.COLI THYMIDYLATE SYNTHASE WITH DUMP AND THE BGC 945 INHIBITOR | ALPHA/BETA PROTEIN, METHYLASE, METHYLTRANSFERASE, DUMP SUBTRATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1evg:A (ALA148) to (GLY251) CRYSTAL STRUCTURE ANALYSIS OF CYS167 MUTANT OF ESCHERICHIA COLI WITH UNMODIFIED CATALYTIC CYSTEINE | THR167 E. COLI THYMIDYLATE SYNTHASE WITH UNMODIFIED CATALYTIC CYSTEINE, TRANSFERASE
2ftn:A (ALA148) to (GLY251) E. COLI THYMIDYLATE SYNTHASE Y94F MUTANT | METHYLTRANSFERASE, TRANSFERASE
4kpw:A (GLN200) to (GLY300) CRYSTAL STRUCTURE OF HIS-TAGGED HUMAN THYMIDYLATE SYNTHASE R175A MUTANT | INTERFACE HOT SPOT, TRANSFERASE, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS
1kzi:A (ALA148) to (GLY251) CRYSTAL STRUCTURE OF ECTS/DUMP/THF COMPLEX | ENZYME SUBSTRATE COMPLEX, TRANSFERASE
1kzi:B (ALA148) to (GLY251) CRYSTAL STRUCTURE OF ECTS/DUMP/THF COMPLEX | ENZYME SUBSTRATE COMPLEX, TRANSFERASE
1kzj:A (ALA148) to (GLY251) CRYSTAL STRUCTURE OF ECTS W80G/DUMP/CB3717 COMPLEX | ENZYME SUBSTRATE COFACTOR ANALOG COMPLEX, TRANSFERASE
1kzj:B (ALA148) to (GLY251) CRYSTAL STRUCTURE OF ECTS W80G/DUMP/CB3717 COMPLEX | ENZYME SUBSTRATE COFACTOR ANALOG COMPLEX, TRANSFERASE
1kzj:F (ALA148) to (GLY251) CRYSTAL STRUCTURE OF ECTS W80G/DUMP/CB3717 COMPLEX | ENZYME SUBSTRATE COFACTOR ANALOG COMPLEX, TRANSFERASE
3bz0:A (THR200) to (ASN303) LACTOBACILLUS CASEI THYMIDYLATE SYNTHASE TERNARY COMPLEX WITH DUMP AND THE PHTALIMIDIC DERIVATIVE C00 | NUCLEOTIDE SYNTHASE, STRUCTURE BASED DRUG DESIGN, METHYLTRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TRANSFERASE
3qg2:B (LEU493) to (ASN595) PLASMODIUM FALCIPARUM DHFR-TS QRADRUPLE MUTANT (N51I+C59R+S108N+I164L, V1/S) PYRIMETHAMINE COMPLEX | PYRIMETHAMINE, ANTIFOLATE RESISTANCE, PLASMODIUM FALCIPARUM, DIHYDROFOLATE REDUCTASE, OXIDOREDUCTASE, TRANSFERASE, TRANSFERASE- INHIBITOR COMPLEX
4gev:B (ALA148) to (GLY251) E. COLI THYMIDYLATE SYNTHASE Y209W VARIANT IN COMPLEX WITH SUBSTRATE AND A COFACTOR ANALOG | BETA SHEET, ALPHA/BETA PROTEIN, METHYLASE, TRANSFERASE