Usages in wwPDB of concept: c_0288
nUsages: 438; SSE string: EEEHEHEHE
2oag:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) WITH PYRROLIDINE-CONSTRAINED PHENETHYLAMINE 29G  |   SERINE-PEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
2oag:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) WITH PYRROLIDINE-CONSTRAINED PHENETHYLAMINE 29G  |   SERINE-PEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
2aj8:A   (SER511) to   (VAL653)  PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH 7-BENZYL-1,3- DIMETHYL-8-PIPERAZIN-1-YL-3,7-DIHYDRO-PURINE-2,6-DIONE (BDPX)  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE 
2aj8:B   (SER511) to   (VAL653)  PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH 7-BENZYL-1,3- DIMETHYL-8-PIPERAZIN-1-YL-3,7-DIHYDRO-PURINE-2,6-DIONE (BDPX)  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE 
2aj8:C   (SER511) to   (VAL653)  PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH 7-BENZYL-1,3- DIMETHYL-8-PIPERAZIN-1-YL-3,7-DIHYDRO-PURINE-2,6-DIONE (BDPX)  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE 
2aj8:D   (SER511) to   (VAL653)  PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH 7-BENZYL-1,3- DIMETHYL-8-PIPERAZIN-1-YL-3,7-DIHYDRO-PURINE-2,6-DIONE (BDPX)  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE 
2ajc:C   (SER511) to   (VAL653)  PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH 4-(2- AMINOETHYL)-BENZENE SULPHONYL FLUORIDE (AEBSF)  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
2ajc:D   (SER511) to   (VAL653)  PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH 4-(2- AMINOETHYL)-BENZENE SULPHONYL FLUORIDE (AEBSF)  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
2ajl:J   (SER511) to   (VAL653)  X-RAY STRUCTURE OF NOVEL BIARYL-BASED DIPEPTIDYL PEPTIDASE IV INHIBITOR  |   AMINOPEPTIDASE, HYDROLASE, PROTEASE, SERINE PROTEASE 
2og1:A    (GLY19) to   (MET135)  CRYSTAL STRUCTURE OF BPHD, A C-C HYDROLASE FROM BURKHOLDERIA XENOVORANS LB400  |   BPHD, ALPHA/BETA HYDROLASE, PCB DEGRADATION, META CLEAVAGE PRODUCT HYDROLASE, MCP HYDROLASE, 2-HYDROXY-6-OXO-6-PHENYLHEXA-2, 4-DIENOATE HYDROLASE, HYDROLASE 
2og1:B    (GLY19) to   (MET135)  CRYSTAL STRUCTURE OF BPHD, A C-C HYDROLASE FROM BURKHOLDERIA XENOVORANS LB400  |   BPHD, ALPHA/BETA HYDROLASE, PCB DEGRADATION, META CLEAVAGE PRODUCT HYDROLASE, MCP HYDROLASE, 2-HYDROXY-6-OXO-6-PHENYLHEXA-2, 4-DIENOATE HYDROLASE, HYDROLASE 
2ogz:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DPP-IV COMPLEXED WITH LILLY ARYL KETONE INHIBITOR  |   DIPEPTIDYL PEPTIDASE IV, CD26, DPIV, DPP-IV, DPP4, SERINE PROTEASE, INHIBITOR, HYDROLASE 
2ogz:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DPP-IV COMPLEXED WITH LILLY ARYL KETONE INHIBITOR  |   DIPEPTIDYL PEPTIDASE IV, CD26, DPIV, DPP-IV, DPP4, SERINE PROTEASE, INHIBITOR, HYDROLASE 
3ebl:C    (VAL63) to   (LEU224)  CRYSTAL STRUCTURE OF RICE GID1 COMPLEXED WITH GA4  |   ALPHA/BETA HYDROLASE, LIPASE, GIBBERELLIN SIGNALING PATHWAY, HYDROLASE, NUCLEUS, RECEPTOR, HYDROLASE RECEPTOR 
3ebl:F    (VAL63) to   (LEU224)  CRYSTAL STRUCTURE OF RICE GID1 COMPLEXED WITH GA4  |   ALPHA/BETA HYDROLASE, LIPASE, GIBBERELLIN SIGNALING PATHWAY, HYDROLASE, NUCLEUS, RECEPTOR, HYDROLASE RECEPTOR 
1ni4:D   (VAL178) to   (THR296)  HUMAN PYRUVATE DEHYDROGENASE  |   THIAMIN PYROPHOSPHATE, PYRUVATE, ALPHA-KETO ACID DEHYDROGENASE, PYRUVATE DEHYDROGENASE, OXIDOREDUCTASE 
4wjl:A   (LYS532) to   (VAL674)  STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE 10 (DPPY): A MODULATOR OF NEURONAL KV4 CHANNELS  |   INACTIVE DIPEPTIDYL PEPTIDASE 10, DPP4 STRUCTURE HOMOLOGUE, ALPHA/BETA HYDROLASE, BETA-PROPELLER, MEMBRANE PROTEIN 
4wjl:B   (LYS532) to   (VAL674)  STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE 10 (DPPY): A MODULATOR OF NEURONAL KV4 CHANNELS  |   INACTIVE DIPEPTIDYL PEPTIDASE 10, DPP4 STRUCTURE HOMOLOGUE, ALPHA/BETA HYDROLASE, BETA-PROPELLER, MEMBRANE PROTEIN 
2onc:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-4  |   DPP4 PROTEIN-INHIBITOR COMPLEX, HYDROLASE 
2onc:B   (PRO510) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-4  |   DPP4 PROTEIN-INHIBITOR COMPLEX, HYDROLASE 
2onc:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-4  |   DPP4 PROTEIN-INHIBITOR COMPLEX, HYDROLASE 
2onc:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-4  |   DPP4 PROTEIN-INHIBITOR COMPLEX, HYDROLASE 
4h0c:A     (MSE1) to   (THR129)  CRYSTAL STRUCTURE OF PHOSPHOLIPASE/CARBOXYLESTERASE FROM DYADOBACTER FERMENTANS DSM 18053  |   PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, PHOSPHOLIPASE/CARBOXYLESTERASE, HYDROLASE 
2oqv:A   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV (DPP4) WITH PIPERIDINE- CONSTRAINED PHENETHYLAMINE  |   SERINE-PEPTIDASE, INHIBITOR, HYDROLASE 
2oqv:B   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV (DPP4) WITH PIPERIDINE- CONSTRAINED PHENETHYLAMINE  |   SERINE-PEPTIDASE, INHIBITOR, HYDROLASE 
3eio:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE ANALYSIS OF DPPIV INHIBITOR  |   PROTEIN-INHIBITOR COMPLEX, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
3eio:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE ANALYSIS OF DPPIV INHIBITOR  |   PROTEIN-INHIBITOR COMPLEX, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
2oxe:A    (GLY26) to   (LEU194)  STRUCTURE OF THE HUMAN PANCREATIC LIPASE-RELATED PROTEIN 2  |   GLYCOPROTEIN, HYDROLASE, LIPID DEGRADATION, PANCREATIC LIPASE, STRUCTURAL GENOMICS CONSORTIUM, SGC 
1nu8:A   (SER511) to   (ALA654)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPP-IV) IN COMPLEX WITH DIPROTIN A (IPI)  |   B-BARREL, ALPHA/BETA HYDROLASE FOLD, EXOPEPTIDASE, DIPROTIN A, HYDROLASE 
1nu8:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPP-IV) IN COMPLEX WITH DIPROTIN A (IPI)  |   B-BARREL, ALPHA/BETA HYDROLASE FOLD, EXOPEPTIDASE, DIPROTIN A, HYDROLASE 
2ozl:D   (GLY177) to   (THR296)  HUMAN PYRUVATE DEHYDROGENASE S264E VARIANT  |   PYRUVATE_DEHYDROGENASE_COMPLEX; HUMAN; E1; MULTIENZYME_COMPLEX_COMPONENT; THIAMINE_PYROPHOSPHATE; THIAMIN_DIPHOSPHATE; HETEROTETRAMERIC; LIPOYL_SUBSTRATE; PYRUVATE; DIHYDROLIPOAMIDE_ACETYLTRANSFERASE; DIHYDROLIPOAMIDE_DEHYDROGENASE;, OXIDOREDUCTASE 
2bgn:D   (SER511) to   (VAL653)  HIV-1 TAT PROTEIN DERIVED N-TERMINAL NONAPEPTIDE TRP2-TAT (1-9) BOUND TO THE ACTIVE SITE OF DIPEPTIDYL PEPTIDASE IV (CD26)  |   HYDROLASE, HYDROLASE/COMPLEX, DIPETIDYL PEPTIDASE IV, DPPIV, CD26, ALPHA/BETA-HYDROLASE FOLD, BETA-PROPELLER FOLD, PROTEIN-PROTEIN COMPLEX, ADENOSINE DEAMINASE, ADA, SERINE PROTEASE, AMINOPEPTIDASE, HIV-1 TAT PROTEIN 
2bgr:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HIV-1 TAT DERIVED NONAPEPTIDES TAT(1-9) BOUND TO THE ACTIVE SITE OF DIPEPTIDYL PEPTIDASE IV (CD26)  |   HYDROLASE, HYDROLASE/COMPLEX, DPPIV, ALPHA/BETA-HYDROLASE FOLD, BETA-PROPELLER FOLD 
2bgr:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HIV-1 TAT DERIVED NONAPEPTIDES TAT(1-9) BOUND TO THE ACTIVE SITE OF DIPEPTIDYL PEPTIDASE IV (CD26)  |   HYDROLASE, HYDROLASE/COMPLEX, DPPIV, ALPHA/BETA-HYDROLASE FOLD, BETA-PROPELLER FOLD 
3exg:F   (GLY177) to   (THR296)  CRYSTAL STRUCTURE OF THE PYRUVATE DEHYDROGENASE (E1P) COMPONENT OF HUMAN PYRUVATE DEHYDROGENASE COMPLEX  |   HETEROTETRAMER; THIAMINE DIPHOSPHATE-DEPENDENT ENZYME; DISEASE MUTATION; GLYCOLYSIS; LEIGH SYNDROME; MITOCHONDRION; OXIDOREDUCTASE; PHOSPHOPROTEIN; ALTERNATIVE SPLICING; POLYMORPHISM; PYRUVATE; THIAMINE PYROPHOSPHATE; TRANSIT PEPTIDE, OXIDOREDUCTASE 
3exg:L   (GLY177) to   (THR296)  CRYSTAL STRUCTURE OF THE PYRUVATE DEHYDROGENASE (E1P) COMPONENT OF HUMAN PYRUVATE DEHYDROGENASE COMPLEX  |   HETEROTETRAMER; THIAMINE DIPHOSPHATE-DEPENDENT ENZYME; DISEASE MUTATION; GLYCOLYSIS; LEIGH SYNDROME; MITOCHONDRION; OXIDOREDUCTASE; PHOSPHOPROTEIN; ALTERNATIVE SPLICING; POLYMORPHISM; PYRUVATE; THIAMINE PYROPHOSPHATE; TRANSIT PEPTIDE, OXIDOREDUCTASE 
3exg:2   (VAL178) to   (THR296)  CRYSTAL STRUCTURE OF THE PYRUVATE DEHYDROGENASE (E1P) COMPONENT OF HUMAN PYRUVATE DEHYDROGENASE COMPLEX  |   HETEROTETRAMER; THIAMINE DIPHOSPHATE-DEPENDENT ENZYME; DISEASE MUTATION; GLYCOLYSIS; LEIGH SYNDROME; MITOCHONDRION; OXIDOREDUCTASE; PHOSPHOPROTEIN; ALTERNATIVE SPLICING; POLYMORPHISM; PYRUVATE; THIAMINE PYROPHOSPHATE; TRANSIT PEPTIDE, OXIDOREDUCTASE 
3s2z:A     (GLY0) to   (ALA130)  CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536 S106A MUTANT IN COMPLEX WITH CAFFEIC ACID  |   ALPHA/BETA HYDROLASE FOLD, ESTERASE, HYDROLASE, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES 
3s2z:B     (GLY0) to   (ALA130)  CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536 S106A MUTANT IN COMPLEX WITH CAFFEIC ACID  |   ALPHA/BETA HYDROLASE FOLD, ESTERASE, HYDROLASE, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES 
3fak:A    (ASP43) to   (ILE171)  STRUCTURAL AND FUNCTIONAL ANALYSIS OF A HORMONE-SENSITIVE LIPASE LIKE ESTE5 FROM A METAGENOME LIBRARY  |   HSL, ESTE5, ESTERASE, LIPASE, HYDROLASE 
2bua:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A LOW MOLECULAR WEIGHT INHIBITOR.  |   HYDROLASE/INHIBITOR, DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX (HYDROLASE/INHIBITOR) 
2bua:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A LOW MOLECULAR WEIGHT INHIBITOR.  |   HYDROLASE/INHIBITOR, DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX (HYDROLASE/INHIBITOR) 
2bua:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A LOW MOLECULAR WEIGHT INHIBITOR.  |   HYDROLASE/INHIBITOR, DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX (HYDROLASE/INHIBITOR) 
2bua:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A LOW MOLECULAR WEIGHT INHIBITOR.  |   HYDROLASE/INHIBITOR, DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX (HYDROLASE/INHIBITOR) 
2bub:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A REVERSED AMIDE INHIBITOR  |   HYDROLASE/INHIBITOR, COMPLEX (HYDROLASE/INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX 
4hxe:B   (GLU350) to   (ASN489)  PYROCOCCUS HORIKOSHII ACYLAMINOACYL PEPTIDASE (UNCOMPLEXED)  |   SELF-COMPARTMENTALIZATION, BETA-PROPELLER, ALPHA/BETA HYRDOLASE FOLD, HYDROLASE 
4hxf:B   (GLU350) to   (ASN489)  ACYLAMINOACYL PEPTIDASE IN COMPLEX WITH Z-GLY-GLY-PHE-CHLOROMETHYL KETONE  |   SELF-COMPARTMENTALIZATION, BETA-PROPELLER, ALPHA/BETA HYRDOLASE FOLD, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4hxg:A   (GLU350) to   (ASN489)  PYROCOCCUS HORIKOSHII ACYLAMINOACYL PEPTIDASE (ORTHORHOMBIC CRYSTAL FORM)  |   SELF-COMPARTMENTALIZATION, BETA-PROPELLER, ALPHA/BETA HYRDOLASE FOLD, HYDROLASE 
4hxg:B   (GLU350) to   (ASN489)  PYROCOCCUS HORIKOSHII ACYLAMINOACYL PEPTIDASE (ORTHORHOMBIC CRYSTAL FORM)  |   SELF-COMPARTMENTALIZATION, BETA-PROPELLER, ALPHA/BETA HYRDOLASE FOLD, HYDROLASE 
4hxg:G   (GLU350) to   (ASN489)  PYROCOCCUS HORIKOSHII ACYLAMINOACYL PEPTIDASE (ORTHORHOMBIC CRYSTAL FORM)  |   SELF-COMPARTMENTALIZATION, BETA-PROPELLER, ALPHA/BETA HYRDOLASE FOLD, HYDROLASE 
4hxg:H   (PHE354) to   (ASN489)  PYROCOCCUS HORIKOSHII ACYLAMINOACYL PEPTIDASE (ORTHORHOMBIC CRYSTAL FORM)  |   SELF-COMPARTMENTALIZATION, BETA-PROPELLER, ALPHA/BETA HYRDOLASE FOLD, HYDROLASE 
4hxg:J   (GLU350) to   (ASN489)  PYROCOCCUS HORIKOSHII ACYLAMINOACYL PEPTIDASE (ORTHORHOMBIC CRYSTAL FORM)  |   SELF-COMPARTMENTALIZATION, BETA-PROPELLER, ALPHA/BETA HYRDOLASE FOLD, HYDROLASE 
4i19:A    (TYR65) to   (ASN197)  THE CRYSTAL STRUCTURE OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS.  |   STRUCTURAL GENOMICS, PSI-BIOLOGY, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESI, NATPRO, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, HYDROLASE 
2pu5:A    (SER10) to   (MET135)  CRYSTAL STRUCTURE OF A C-C BOND HYDROLASE, BPHD, FROM BURKHOLDERIA XENOVORANS LB400  |   C-C BOND HYDROLASE, HYDROLASE 
2pu5:B    (GLY19) to   (GLY136)  CRYSTAL STRUCTURE OF A C-C BOND HYDROLASE, BPHD, FROM BURKHOLDERIA XENOVORANS LB400  |   C-C BOND HYDROLASE, HYDROLASE 
2puh:A    (GLY19) to   (MET135)  CRYSTAL STRUCTURE OF THE S112A MUTANT OF A C-C HYDROLASE, BPHD FROM BURKHOLDERIA XENOVORANS LB400, IN COMPLEX WITH ITS SUBSTRATE HOPDA  |   C-C BOND HYDROLASE, HYDROLASE 
1orv:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26)  |   SERINE PROTEASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, HYDROLASE 
1orv:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26)  |   SERINE PROTEASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, HYDROLASE 
2q0x:A    (HIS16) to   (GLY142)  ALPHA/BETA HYDROLASE FOLD PROTEIN OF UNKNOWN FUNCTION  |   ALPHA/BETA HYDROLASE FOLD, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA CONSORTIUM, SGPP, PSI, PROTEIN STRUCTURE INITIATIVE, UNKNOWN FUNCTION 
2q0x:B    (HIS16) to   (GLY142)  ALPHA/BETA HYDROLASE FOLD PROTEIN OF UNKNOWN FUNCTION  |   ALPHA/BETA HYDROLASE FOLD, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA CONSORTIUM, SGPP, PSI, PROTEIN STRUCTURE INITIATIVE, UNKNOWN FUNCTION 
3fvr:A    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvr:B    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvr:C    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvr:D    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvr:E    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvr:F    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvr:G    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvr:H    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvr:I    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvr:L    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvr:M    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvr:N    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3sww:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH SA-(+)-3- (AMINOMETHYL)-4-(2,4-DICHLOROPHENYL)-6-(2-METHOXYPHENYL)- 2-METHYL- 5H-PYRROLO[3,4-B]PYRIDIN-7(6H)-ONE  |   EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3sww:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH SA-(+)-3- (AMINOMETHYL)-4-(2,4-DICHLOROPHENYL)-6-(2-METHOXYPHENYL)- 2-METHYL- 5H-PYRROLO[3,4-B]PYRIDIN-7(6H)-ONE  |   EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0b:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH TAK-322  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0b:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH TAK-322  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0b:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH TAK-322  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0b:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH TAK-322  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3sx4:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH SA-(+)-3- (AMINOMETHYL)-4-(2,4-DICHLOROPHENYL)-6-(2-METHOXYPHENYL)- 2-METHYL- 5H-PYRROLO[3,4-B]PYRIDIN-7(6H)-ONE  |   EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3sx4:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH SA-(+)-3- (AMINOMETHYL)-4-(2,4-DICHLOROPHENYL)-6-(2-METHOXYPHENYL)- 2-METHYL- 5H-PYRROLO[3,4-B]PYRIDIN-7(6H)-ONE  |   EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0d:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 2  |   DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0d:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 2  |   DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0d:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 2  |   DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0d:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 2  |   DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0g:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINONE INHIBITOR 3  |   DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0g:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINONE INHIBITOR 3  |   DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0g:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINONE INHIBITOR 3  |   DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0g:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINONE INHIBITOR 3  |   DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
2qky:A   (SER511) to   (VAL653)  COMPLEX STRUCTURE OF DIPEPTIDYL PEPTIDASE IV AND A OXADIAZOLYL KETONE  |   BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
2qky:C   (SER511) to   (VAL653)  COMPLEX STRUCTURE OF DIPEPTIDYL PEPTIDASE IV AND A OXADIAZOLYL KETONE  |   BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
2qky:D   (SER511) to   (VAL653)  COMPLEX STRUCTURE OF DIPEPTIDYL PEPTIDASE IV AND A OXADIAZOLYL KETONE  |   BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
3g9u:A    (ASP43) to   (ILE171)  CRYSTAL STRUCTURE OF ESTE5, WAS SOAKED BY P-NITROPHENYL BUTYRATE FOR 5MIN  |   HSL, ESTE5, ESTERASE, LIPASE, HYDROLASE 
2qoe:A   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A TRIAZOLOPIPERAZINE- BASED BETA AMINO ACID INHIBITOR  |   ALPHA/BETA INHIBITORS, BETA-PROPELLER,DIMER, DIABETES, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
2qoe:B   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A TRIAZOLOPIPERAZINE- BASED BETA AMINO ACID INHIBITOR  |   ALPHA/BETA INHIBITORS, BETA-PROPELLER,DIMER, DIABETES, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
2qr5:A   (GLY332) to   (ALA469)  AEROPYRUM PERNIX ACYLAMINOACYL PEPTIDASE, H367A MUTANT  |   ACYLAMINOACYL PEPTIDASE, THERMOPHILIC ENZYME, OXYANION BINDING SITE, CATALYTIC ACTIVITY, HYDROLASE 
2qr5:B   (GLY332) to   (ALA469)  AEROPYRUM PERNIX ACYLAMINOACYL PEPTIDASE, H367A MUTANT  |   ACYLAMINOACYL PEPTIDASE, THERMOPHILIC ENZYME, OXYANION BINDING SITE, CATALYTIC ACTIVITY, HYDROLASE 
2qru:A     (ASN5) to   (PHE128)  CRYSTAL STRUCTURE OF AN ALPHA/BETA HYDROLASE SUPERFAMILY PROTEIN FROM ENTEROCOCCUS FAECALIS  |   ENTEROCOCCUS FAECALIS, ALPHA/BETA-HYDROLASE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, UNKNOWN FUNCTION 
2qt9:A   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A 4-ARYL CYCLOHEXYLALANINE INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE 
2qt9:B   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A 4-ARYL CYCLOHEXYLALANINE INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE 
2qtb:A   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A 4-ARYL CYCLOHEXYLALANINE INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE 
2qtb:B   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A 4-ARYL CYCLOHEXYLALANINE INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE 
2qzp:A   (VAL336) to   (ALA469)  CRYSTAL STRUCTURE OF MUTATION OF AN ACYLPTIDE HYDROLASE/ESTERASE FROM AEROPYRUM PERNIX K1  |   CRYSTAL STRUCTURE, TRUNCATED, ACYLPEPTIDE HYDROLASE, AEROPYRUM PERNIX K1, CYTOPLASM 
2qzp:B   (GLY332) to   (ALA469)  CRYSTAL STRUCTURE OF MUTATION OF AN ACYLPTIDE HYDROLASE/ESTERASE FROM AEROPYRUM PERNIX K1  |   CRYSTAL STRUCTURE, TRUNCATED, ACYLPEPTIDE HYDROLASE, AEROPYRUM PERNIX K1, CYTOPLASM 
2d5l:A   (GLU480) to   (GLY627)  CRYSTAL STRUCTURE OF PROLYL TRIPEPTIDYL AMINOPEPTIDASE FROM PORPHYROMONAS GINGIVALIS  |   PEPTIDASE FAMILY S9, SERINE PEPTIDASE, PROLYL OLIGOPEPTIDASE FAMILY, HYDROLASE 
4j3j:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DPP-IV WITH COMPOUND C3  |   INHIBITOR COMPLEX, SERINE EXOPEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
2dcm:A   (GLU480) to   (GLY627)  THE CRYSTAL STRUCTURE OF S603A MUTATED PROLYL TRIPEPTIDYL AMINOPEPTIDASE COMPLEXED WITH SUBSTRATE  |   PEPTIDASE FAMILY S9, SERINE PEPTIDASE, PROLYL OLIGOPEPTIDASE FAMILY, SITE-DIRECTED MUTANGENESIS, HYDROLASE 
4y9s:A     (LYS3) to   (LEU128)  STRUCTURE OF AN H300N MUTANT OF POTATO EPOXIDE HYDROLASE, STEH1  |   MUTATION OF CATALYTIC RESIDUE, HYDROLASE 
2dst:A     (ARG3) to   (GLU108)  CRYSTAL STRUCTURE ANALYSIS OF TT1977  |   CONSERVED HYPOTHETICAL PROTEIN, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, UNKNOWN FUNCTION 
4jh0:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL-PEPTIDASE 4 (CD26, ADENOSINE DEAMINASE COMPLEXING PROTEIN 2) (DPP-IV-WT) COMPLEX WITH BMS-767778 AKA 2-(3- (AMINOMETHYL)-4-(2,4- DICHLOROPHENYL)-2-METHYL-5-OXO-5,7-DIHYDRO-6H- PYRROLO[3,4- B]PYRIDIN-6-YL)-N,N-DIMETHYLACETAMIDE  |   EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP-IV, DIMER, HYDROLASE 
4jh0:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL-PEPTIDASE 4 (CD26, ADENOSINE DEAMINASE COMPLEXING PROTEIN 2) (DPP-IV-WT) COMPLEX WITH BMS-767778 AKA 2-(3- (AMINOMETHYL)-4-(2,4- DICHLOROPHENYL)-2-METHYL-5-OXO-5,7-DIHYDRO-6H- PYRROLO[3,4- B]PYRIDIN-6-YL)-N,N-DIMETHYLACETAMIDE  |   EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP-IV, DIMER, HYDROLASE 
3h04:A     (ILE4) to   (TYR126)  THE CRYSTAL STRUCTURE OF THE PROTEIN WITH UNKNOWN FUNCTION FROM STAPHYLOCOCCUS AUREUS SUBSP. AUREUS MU50  |   PROTEIN WITH UNKNOWN FUNCTION, STRUCTURAL GENOMICS, MCSG, PSI, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, UNKNOWN FUNCTION 
3h0c:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A REVERSED AMIDE INHIBITOR  |   COMPLEX (HYDROLASE-INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, CELL MEMBRANE, DISULFIDE BOND, MEMBRANE, SECRETED 
3h0c:B   (SER511) to   (ALA654)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A REVERSED AMIDE INHIBITOR  |   COMPLEX (HYDROLASE-INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, CELL MEMBRANE, DISULFIDE BOND, MEMBRANE, SECRETED 
2rgu:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF COMPLEX OF HUMAN DPP4 AND INHIBITOR  |   PEPTIDASE, INHIBITOR, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
2rgu:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF COMPLEX OF HUMAN DPP4 AND INHIBITOR  |   PEPTIDASE, INHIBITOR, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
2rip:A   (SER511) to   (VAL653)  STRUCTURE OF DPPIV IN COMPLEX WITH AN INHIBITOR  |   DPPIV, DIABETES, DRUG DESIGN, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE 
3h19:A    (ASP43) to   (ILE171)  CRYSTAL STRUCTURE OF ESTE5, WAS SOAKED BY METHYL ALCOHOL  |   HSL, ESTE5, ESTERASE, LIPASE, HYDROLASE 
1evq:A    (ALA46) to   (TYR183)  THE CRYSTAL STRUCTURE OF THE THERMOPHILIC CARBOXYLESTERASE EST2 FROM ALICYCLOBACILLUS ACIDOCALDARIUS  |   ALPHA/BETA HYDROLASE FOLD 
1qtr:A    (TYR14) to   (GLY137)  CRYSTAL STRUCTURE ANALYSIS OF THE PROLYL AMINOPEPTIDASE FROM SERRATIA MARCESCENS  |   ALPHA BETA HYDROLASE FOLD, PROLINE, PROLYL AMINOPEPTIDASE, SERRATIA, IMINOPEPTIDASE 
1qz3:A    (ALA46) to   (TYR183)  CRYSTAL STRUCTURE OF MUTANT M211S/R215L OF CARBOXYLESTERASE EST2 COMPLEXED WITH HEXADECANESULFONATE  |   ALPHA/BETA HYDROLASE FOLD, HYDROLASE 
2ecf:A   (PRO486) to   (ALA634)  CRYSTAL STRUCTURE OF DIPEPTIDYL AMINOPEPTIDASE IV FROM STENOTROPHOMONAS MALTOPHILIA  |   PROLYL OLIGOPEPTIDASE FAMILY, PEPTIDASE FAMILY S9, DIPEPTIDYL PEPTIDASE IV, HYDROLASE 
2eep:A   (GLU480) to   (GLY626)  PROLYL TRIPEPTIDYL AMINOPEPTIDASE COMPLEXED WITH AN INHIBITOR  |   PEPTIDASE FAMILY S9, PROLYL OLIGOPEPTIDASE FAMILY, SERINE PEPTIDASE, INHIBITOR COMPLEX, HYDROLASE 
3hea:B     (SER1) to   (GLY119)  THE L29P/L124I MUTATION OF PSEUDOMONAS FLUORESCENS ESTERASE  |   ALPHA/BETA HYDROLASE, ESTERASE, COVALENT ADDUCT, TETRAHEDRAL INTERMEDIATE, HYDROLASE, OXIDOREDUCTASE, PEROXIDASE 
3hea:C     (SER1) to   (GLY119)  THE L29P/L124I MUTATION OF PSEUDOMONAS FLUORESCENS ESTERASE  |   ALPHA/BETA HYDROLASE, ESTERASE, COVALENT ADDUCT, TETRAHEDRAL INTERMEDIATE, HYDROLASE, OXIDOREDUCTASE, PEROXIDASE 
1r9m:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV AT 2.1 ANG. RESOLUTION.  |   AMINOPEPTIDASE, SERINE PROTEASE, GLYCOPROTEIN, HYDROLASE 
1r9m:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV AT 2.1 ANG. RESOLUTION.  |   AMINOPEPTIDASE, SERINE PROTEASE, GLYCOPROTEIN, HYDROLASE 
1r9m:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV AT 2.1 ANG. RESOLUTION.  |   AMINOPEPTIDASE, SERINE PROTEASE, GLYCOPROTEIN, HYDROLASE 
1r9m:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV AT 2.1 ANG. RESOLUTION.  |   AMINOPEPTIDASE, SERINE PROTEASE, GLYCOPROTEIN, HYDROLASE 
2fjp:A   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH AN INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, HYDROLASE 
2fjp:B   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH AN INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, HYDROLASE 
4z8z:A    (LYS63) to   (ASN210)  CRYSTAL STRUCTURE OF THE HYPOTHETICAL PROTEIN FROM RUMINICLOSTRIDIUM THERMOCELLUM ATCC 27405  |   STRUCTURAL GENOMICS, HUMAN MICROBIOME, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, PSI-BIOLOGY 
3v1k:A    (GLY19) to   (MET135)  CRYSTAL STRUCTURE OF THE H265Q MUTANT OF A C-C HYDROLASE, BPHD FROM BURKHOLDERIA XENOVORANS LB400.  |   C-C BOND HYDROLASE, ALPHA/BETA HYDROLASE FOLD, BPHD, ALPHA/BETA HYDROLASE, PCB DEGRADATION, META CLEAVAGE PRODUCT HYDROLASE, MCP HYDROLASE, 2-HYDROXY-6-OXO-6-PHENYL-HEXA-2,4-DIENOATE HYDROLASE, HYDROLASE 
3v1k:B    (GLY19) to   (MET135)  CRYSTAL STRUCTURE OF THE H265Q MUTANT OF A C-C HYDROLASE, BPHD FROM BURKHOLDERIA XENOVORANS LB400.  |   C-C BOND HYDROLASE, ALPHA/BETA HYDROLASE FOLD, BPHD, ALPHA/BETA HYDROLASE, PCB DEGRADATION, META CLEAVAGE PRODUCT HYDROLASE, MCP HYDROLASE, 2-HYDROXY-6-OXO-6-PHENYL-HEXA-2,4-DIENOATE HYDROLASE, HYDROLASE 
2fx5:A    (THR24) to   (ILE147)  PSEUDOMONAS MENDOCINA LIPASE  |   ALPHA-BETA HYDROLASE 
4kr0:A   (SER511) to   (VAL653)  COMPLEX STRUCTURE OF MERS-COV SPIKE RBD BOUND TO CD26  |   8-BLADED BETA-PROPELLER DOMAIN, ALPHA/BETA HYDROLASE DOMAIN, BLADES IV AND V, CD26 BETA-PROPELLER, HYDROLASE-VIRAL PROTEIN COMPLEX 
4kry:A    (ALA59) to   (TYR195)  STRUCTURE OF AES FROM E. COLI IN COVALENT COMPLEX WITH PMS  |   ALPHA/BETA-HYDROLASE, HORMONE-SENSITIVE-LIPASE FAMILY, INHIBITION OF MALT, ACYL ESTERASE, PHENYLMETHYLSULFONYL-SERINE, HYDROLASE 
3v9a:A    (ASP43) to   (ILE171)  CRYSTAL STRUCTURE OF ESTERASE/LIPASE FROM UNCULTURED BACTERIUM  |   ESTERASE, LIPASE, HYDROLASE ACTIVATOR 
2g5p:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) COMPLEXED WITH CYANOPYRROLIDINE (C5-PRO-PRO) INHIBITOR 21AC  |   SERINE PEPTIDASE, BETA-PROPELLER, HYDROLASE 
2g5p:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) COMPLEXED WITH CYANOPYRROLIDINE (C5-PRO-PRO) INHIBITOR 21AC  |   SERINE PEPTIDASE, BETA-PROPELLER, HYDROLASE 
2g5t:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) COMPLEXED WITH CYANOPYRROLIDINE (C5-PRO-PRO) INHIBITOR 21AG  |   SERINE PEPTIDASE, BETA-PROPELLER, HYDROLASE 
2g63:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) COMPLEXED WITH CYANOPYRROLIDINE (C5-PRO-PRO) INHIBITOR 24B  |   SERINE PEPTIDASE, BETA-PROPELLER, HYDROLASE 
2g63:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) COMPLEXED WITH CYANOPYRROLIDINE (C5-PRO-PRO) INHIBITOR 24B  |   SERINE PEPTIDASE, BETA-PROPELLER, HYDROLASE 
2gbf:A   (SER512) to   (VAL654)  RAT DPP-IV WITH ALKYNYL CYANOPYRROLIDINE #1  |   SERINE PEPTIDASE BETA PROPELLER, HYDROLASE 
2gbf:B   (SER512) to   (VAL654)  RAT DPP-IV WITH ALKYNYL CYANOPYRROLIDINE #1  |   SERINE PEPTIDASE BETA PROPELLER, HYDROLASE 
2gbg:A   (VAL508) to   (VAL654)  RAT DPP-IV WITH ALKYNYL CYANOPYRROLIDINE #2  |   SERINE PEPTIDASE BETA PROPELLER, HYDROLASE 
2gbg:B   (VAL508) to   (VAL654)  RAT DPP-IV WITH ALKYNYL CYANOPYRROLIDINE #2  |   SERINE PEPTIDASE BETA PROPELLER, HYDROLASE 
2gbi:A   (SER512) to   (VAL654)  RAT DPP-IV WITH XANTHINE INHIBITOR 4  |   SERINE PEPTIDASE BETA PROPELLER, HYDROLASE 
2gbi:B   (SER512) to   (VAL654)  RAT DPP-IV WITH XANTHINE INHIBITOR 4  |   SERINE PEPTIDASE BETA PROPELLER, HYDROLASE 
3ia2:B     (SER1) to   (GLY119)  PSEUDOMONAS FLUORESCENS ESTERASE COMPLEXED TO THE R-ENANTIOMER OF A SULFONATE TRANSITION STATE ANALOG  |   ALPHA-BETA HYDROLASE FOLD, TRANSITION STATE ANALOG, HYDROLASE, OXIDOREDUCTASE, PEROXIDASE 
3ia2:D     (SER1) to   (GLY119)  PSEUDOMONAS FLUORESCENS ESTERASE COMPLEXED TO THE R-ENANTIOMER OF A SULFONATE TRANSITION STATE ANALOG  |   ALPHA-BETA HYDROLASE FOLD, TRANSITION STATE ANALOG, HYDROLASE, OXIDOREDUCTASE, PEROXIDASE 
3ia2:E     (SER1) to   (GLY119)  PSEUDOMONAS FLUORESCENS ESTERASE COMPLEXED TO THE R-ENANTIOMER OF A SULFONATE TRANSITION STATE ANALOG  |   ALPHA-BETA HYDROLASE FOLD, TRANSITION STATE ANALOG, HYDROLASE, OXIDOREDUCTASE, PEROXIDASE 
3ib3:B    (GLY44) to   (TRP192)  CRYSTAL STRUCTURE OF SACOL2612 - COCE/NOND FAMILY HYDROLASE FROM STAPHYLOCOCCUS AUREUS  |   STRUCTURAL GENOMICS, HYDROLASE, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID 
3vjk:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DEPIPTIDYL PEPTIDASE IV (DPP-4) IN COMPLEX WITH MP-513  |   ALPHA/BETA, BETA-PROPELLER, AMINOPEPTIDASE, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, DIABETES, GLYCOPROTEIN, CELL MEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3vjl:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DEPIPTIDYL PEPTIDASE IV (DPP-4) IN COMPLEX WITH A PROLYLTHIAZOLIDINE INHIBITOR #2  |   ALPHA/BETA, BETA-PROPELLER, AMINOPEPTIDASE, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, DIABETES, GLYCOPROTEIN, CELL MEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3vjm:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DEPIPTIDYL PEPTIDASE IV (DPP-4) IN COMPLEX WITH A PROLYLTHIAZOLIDINE INHIBITOR #1  |   ALPHA/BETA, BETA-PROPELLER, AMINOPEPTIDASE, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, DIABETES, GLYCOPROTEIN, CELL MEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3vjm:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DEPIPTIDYL PEPTIDASE IV (DPP-4) IN COMPLEX WITH A PROLYLTHIAZOLIDINE INHIBITOR #1  |   ALPHA/BETA, BETA-PROPELLER, AMINOPEPTIDASE, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, DIABETES, GLYCOPROTEIN, CELL MEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4l72:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF MERS-COV COMPLEXED WITH HUMAN DPP4  |   ALPHA/BETA HYDROLASE BETA-PROPELLER, GLYCOLATION, VIRUS RECEPTOR- BINDING DOMAIN, HYDROLASE-VIRAL PROTEIN COMPLEX 
4l9a:A     (ALA3) to   (LEU124)  CRYSTAL STRUCTURE OF SMU.1393C FROM CARIOGENIC PATHOGEN STREPTOCOCCUS MUTANS  |   ALPHA/BETA HYDROLASE, CARBOXYLESTERASE, HYDROLASE 
4l9a:B     (ALA3) to   (LEU124)  CRYSTAL STRUCTURE OF SMU.1393C FROM CARIOGENIC PATHOGEN STREPTOCOCCUS MUTANS  |   ALPHA/BETA HYDROLASE, CARBOXYLESTERASE, HYDROLASE 
1hde:A    (PRO22) to   (MET147)  HALOALKANE DEHALOGENASE MUTANT WITH PHE 172 REPLACED WITH TRP  |   DEHALOGENASE, HYDROLASE, DETOXIFICATION 
1hde:B    (PRO22) to   (MET147)  HALOALKANE DEHALOGENASE MUTANT WITH PHE 172 REPLACED WITH TRP  |   DEHALOGENASE, HYDROLASE, DETOXIFICATION 
4zwn:A    (LEU15) to   (SER148)  CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF THE MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE  |   MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, SERINE HYDROLASE, ALPHA/BETA HYDROLASE, HYDROLASE 
4zwn:B    (GLU14) to   (SER148)  CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF THE MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE  |   MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, SERINE HYDROLASE, ALPHA/BETA HYDROLASE, HYDROLASE 
4zwn:C    (GLU14) to   (SER148)  CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF THE MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE  |   MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, SERINE HYDROLASE, ALPHA/BETA HYDROLASE, HYDROLASE 
4zwn:D    (GLN16) to   (SER148)  CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF THE MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE  |   MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, SERINE HYDROLASE, ALPHA/BETA HYDROLASE, HYDROLASE 
4lko:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH BMS-744891  |   EXOPEPTIDASE, BETA BARREL, ALPHA/BETA HYDROLASE FOLD, HYDROLASE 
2hm7:A    (ALA46) to   (ILE182)  CRYSTAL STRUCTURE ANALYSIS OF THE G84S EST2 MUTANT  |   ALPHA/BETA HYDROLASE FOLD, HYDROLASE 
2wj6:A     (LEU6) to   (MET125)  CRYSTAL STRUCTURE OF THE COFACTOR-DEVOID 1-H-3-HYDROXY-4- OXOQUINALDINE 2,4-DIOXYGENASE (HOD) FROM ARTHROBACTER NITROGUAJACOLICUS RU61A COMPLEXED WITH ITS NATURAL PRODUCT N-ACETYLANTHRANILATE  |   OXIDOREDUCTASE, ALPHA/BETA HYDROLASE 
1u2e:A     (SER8) to   (GLY134)  CRYSTAL STRUCTURE OF THE C-C BOND HYDROLASE MHPC  |   ALPHA/BETA HYDROLASE FOLD 
1u2e:B  (SER1008) to  (GLY1134)  CRYSTAL STRUCTURE OF THE C-C BOND HYDROLASE MHPC  |   ALPHA/BETA HYDROLASE FOLD 
1u4n:A    (ALA46) to   (ILE182)  CRYSTAL STRUCTURE ANALYSIS OF THE M211S/R215L EST2 MUTANT  |   ALPHA/BETA HYDROLASE FOLD, HYDROLASE 
2hu5:A   (VAL336) to   (ALA469)  BINDING OF INHIBITORS BY ACYLAMINOACYL-PEPTIDASE  |   ALPHA/BETA HYDROLASE, BETA-PROPELLER, ENZYME-INHIBITOR COMPLEX, HYDROLASE 
2hu5:B   (GLY332) to   (ALA469)  BINDING OF INHIBITORS BY ACYLAMINOACYL-PEPTIDASE  |   ALPHA/BETA HYDROLASE, BETA-PROPELLER, ENZYME-INHIBITOR COMPLEX, HYDROLASE 
2hu7:A   (VAL336) to   (ALA469)  BINDING OF INHIBITORS BY ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE, BETA-PROPELLER, ENZYME-INHIBITOR COMPLEX, HYDROLASE 
2hu8:A   (VAL336) to   (ALA469)  BINDING OF INHIBITORS BY ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE, BETA-PROPELLER, ENZYME-INHIBITOR COMPLEX, HYDROLASE 
2hu8:B   (VAL336) to   (ALA469)  BINDING OF INHIBITORS BY ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE, BETA-PROPELLER, ENZYME-INHIBITOR COMPLEX, HYDROLASE 
3w2t:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DEPIPTIDYL PEPTIDASE IV (DPP-4) IN COMPLEX WITH VILDAGLIPTIN  |   ALPHA/BETA, BETA-PROPELLER, HYDROLASE, AMINOPEPTIDASE, SERINE PROTEASE, SECRETED, SIGNAL-ANCHOR, TRANSMEMBRANE, DIABETES, GLYCOPROTEIN, CELL MEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3w2t:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DEPIPTIDYL PEPTIDASE IV (DPP-4) IN COMPLEX WITH VILDAGLIPTIN  |   ALPHA/BETA, BETA-PROPELLER, HYDROLASE, AMINOPEPTIDASE, SERINE PROTEASE, SECRETED, SIGNAL-ANCHOR, TRANSMEMBRANE, DIABETES, GLYCOPROTEIN, CELL MEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
1u8e:A   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 MUTANT Y547F  |   ALPHA/BETA HYDROLASE, BETA-PROPELLER, HOMODIMER, HYDROLASE 
1u8e:B   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 MUTANT Y547F  |   ALPHA/BETA HYDROLASE, BETA-PROPELLER, HOMODIMER, HYDROLASE 
2wtm:B    (GLY-1) to   (SER129)  EST1E FROM BUTYRIVIBRIO PROTEOCLASTICUS  |   ESTERASE, HYDROLASE, FERULIC ACID ESTERASE 
2wtm:D    (GLY-1) to   (SER129)  EST1E FROM BUTYRIVIBRIO PROTEOCLASTICUS  |   ESTERASE, HYDROLASE, FERULIC ACID ESTERASE 
1ufo:B     (ARG2) to   (ILE136)  CRYSTAL STRUCTURE OF TT1662 FROM THERMUS THERMOPHILUS  |   ALPHA-BETA FOLD, HYDROLASE, STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI 
1ufo:C     (MSE1) to   (ILE136)  CRYSTAL STRUCTURE OF TT1662 FROM THERMUS THERMOPHILUS  |   ALPHA-BETA FOLD, HYDROLASE, STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI 
1ufo:E     (MSE1) to   (ILE136)  CRYSTAL STRUCTURE OF TT1662 FROM THERMUS THERMOPHILUS  |   ALPHA-BETA FOLD, HYDROLASE, STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI 
2i3d:A     (PRO2) to   (ILE130)  CRYSTAL STRUCTURE OF PROTEIN OF UNKNOWN FUNCTION ATU1826, A PUTATIVE ALPHA/BETA HYDROLASE FROM AGROBACTERIUM TUMEFACIENS  |   STRUCTURAL GENOMICS, APC5865, HYDROLASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, UNKNOWN FUNCTION 
2i3d:B     (GLU3) to   (ILE130)  CRYSTAL STRUCTURE OF PROTEIN OF UNKNOWN FUNCTION ATU1826, A PUTATIVE ALPHA/BETA HYDROLASE FROM AGROBACTERIUM TUMEFACIENS  |   STRUCTURAL GENOMICS, APC5865, HYDROLASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, UNKNOWN FUNCTION 
2i3z:A   (SER512) to   (VAL654)  RAT DPP-IV WITH XANTHINE MIMETIC INHIBITOR #7  |   ENZYME, PEPTIDASE, INHIBITOR, HYDROLASE 
2i3z:B   (SER512) to   (VAL654)  RAT DPP-IV WITH XANTHINE MIMETIC INHIBITOR #7  |   ENZYME, PEPTIDASE, INHIBITOR, HYDROLASE 
1ik6:A   (GLU186) to   (ALA294)  3D STRUCTURE OF THE E1BETA SUBUNIT OF PYRUVATE DEHYDROGENASE FROM THE ARCHEON PYROBACULUM AEROPHILUM  |   E1BETA, PYRUVATE DEHYDROGENASE, TETRAMER, GXXXG, OXIDOREDUCTASE 
2i78:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPP IV) COMPLEXED WITH ABT-341, A CYCLOHEXENE-CONSTRAINED PHENETHYLAMINE INHIBITOR  |   SERINE PEPTIDASE,, HYDROLASE 
2i78:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPP IV) COMPLEXED WITH ABT-341, A CYCLOHEXENE-CONSTRAINED PHENETHYLAMINE INHIBITOR  |   SERINE PEPTIDASE,, HYDROLASE 
2i78:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPP IV) COMPLEXED WITH ABT-341, A CYCLOHEXENE-CONSTRAINED PHENETHYLAMINE INHIBITOR  |   SERINE PEPTIDASE,, HYDROLASE 
1j2e:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE IV, CD26, PROLYL OLIGOPEPTIDASE, BETA-PROPELLER STRUCTURE, HYDROLASE 
1j2e:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE IV, CD26, PROLYL OLIGOPEPTIDASE, BETA-PROPELLER STRUCTURE, HYDROLASE 
2iu4:A    (GLN24) to   (ASP132)  DIHYDROXYACETONE KINASE OPERON CO-ACTIVATOR DHA-DHAQ  |   TRANSFERASE, LACTOCOCCUS LACTIS, DIHYDROXYACETONE, CO-ACTIVATOR, KINASE 
2iu4:B    (GLN24) to   (ASP133)  DIHYDROXYACETONE KINASE OPERON CO-ACTIVATOR DHA-DHAQ  |   TRANSFERASE, LACTOCOCCUS LACTIS, DIHYDROXYACETONE, CO-ACTIVATOR, KINASE 
2iu6:A    (GLN24) to   (ASP133)  REGULATION OF THE DHA OPERON OF LACTOCOCCUS LACTIS  |   KINASE, DIHYDROXYACETONE KINASE TRANSFERASE, TRANSFERASE 
2iu6:B    (GLN24) to   (ASP133)  REGULATION OF THE DHA OPERON OF LACTOCOCCUS LACTIS  |   KINASE, DIHYDROXYACETONE KINASE TRANSFERASE, TRANSFERASE 
1va4:A     (SER1) to   (GLY119)  PSEUDOMONAS FLUORESCENS ARYL ESTERASE  |   ALPHA/BETA HYDROLASE, ESTERASE, NON-COFACTOR DEPENDENT HALOPEROXIDASE, HYDROLASE 
1va4:C     (SER1) to   (GLY119)  PSEUDOMONAS FLUORESCENS ARYL ESTERASE  |   ALPHA/BETA HYDROLASE, ESTERASE, NON-COFACTOR DEPENDENT HALOPEROXIDASE, HYDROLASE 
1va4:E     (SER1) to   (GLY119)  PSEUDOMONAS FLUORESCENS ARYL ESTERASE  |   ALPHA/BETA HYDROLASE, ESTERASE, NON-COFACTOR DEPENDENT HALOPEROXIDASE, HYDROLASE 
1jfr:A    (SER26) to   (THR154)  CRYSTAL STRUCTURE OF THE STREPTOMYCES EXFOLIATUS LIPASE AT 1.9A RESOLUTION: A MODEL FOR A FAMILY OF PLATELET- ACTIVATING FACTOR ACETYLHYDROLASES  |   SERINE HYDROLASE, LIPASE 
1jfr:B    (SER26) to   (THR154)  CRYSTAL STRUCTURE OF THE STREPTOMYCES EXFOLIATUS LIPASE AT 1.9A RESOLUTION: A MODEL FOR A FAMILY OF PLATELET- ACTIVATING FACTOR ACETYLHYDROLASES  |   SERINE HYDROLASE, LIPASE 
1ve6:A   (VAL336) to   (ALA469)  CRYSTAL STRUCTURE OF AN ACYLPEPTIDE HYDROLASE/ESTERASE FROM AEROPYRUM PERNIX K1  |   BETA PROPELLER DOMAIN, ALPHA/BETA HYDROLASE DOMAIN, HYDROLASE 
1ve6:B   (GLY332) to   (ALA469)  CRYSTAL STRUCTURE OF AN ACYLPEPTIDE HYDROLASE/ESTERASE FROM AEROPYRUM PERNIX K1  |   BETA PROPELLER DOMAIN, ALPHA/BETA HYDROLASE DOMAIN, HYDROLASE 
1ve7:A   (VAL336) to   (ALA469)  CRYSTAL STRUCTURE OF AN ACYLPEPTIDE HYDROLASE/ESTERASE FROM AEROPYRUM PERNIX K1 IN COMPLEX WITH P-NITROPHENYL PHOSPHATE  |   BETA PROPELLER DOMAIN, ALPHA/BETA HYDROLASE DOMAIN, HYDROLASE 
1ve7:B   (ARG334) to   (ALA469)  CRYSTAL STRUCTURE OF AN ACYLPEPTIDE HYDROLASE/ESTERASE FROM AEROPYRUM PERNIX K1 IN COMPLEX WITH P-NITROPHENYL PHOSPHATE  |   BETA PROPELLER DOMAIN, ALPHA/BETA HYDROLASE DOMAIN, HYDROLASE 
3wqh:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH ANAGLIPTIN  |   DIABETES, BETA-PROPELLER, AMINOPEPTIDASE, MEMBRANE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX 
3wqh:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH ANAGLIPTIN  |   DIABETES, BETA-PROPELLER, AMINOPEPTIDASE, MEMBRANE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX 
1w1i:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV (DPPIV OR CD26) IN COMPLEX WITH ADENOSINE DEAMINASE  |   HYDROLASE, HYDROLASE/COMPLEX, DIPETIDYL PEPTIDASE IV, DPPIV, CD26, ALPHA/BETA-HYDROLASE FOLD, BETA-PROPELLER FOLD, PROTEIN-PROTEIN COMPLEX, ADENOSINE DEAMINASE, ADA, SERINE PROTEASE, AMINOPEPTIDASE 
2jgd:B   (ASN796) to   (TYR901)  E. COLI 2-OXOGLUTARATE DEHYDROGENASE (E1O)  |   2-OXOGLUTARATE DEHYDROGENASE, FLAVOPROTEIN, OXIDOREDUCTASE, THIAMINE DIPHOSPHATE, THIAMINE PYROPHOSPHATE, ADENOSINE MONOPHOSPHATE, E1O, KGDH, OGDH, GLYCOLYSIS, OXALOACETATE 
4n8d:A   (SER511) to   (VAL653)  DPP4 COMPLEXED WITH SYN-7AA  |   HYDROLASE 
4n8d:B   (SER511) to   (VAL653)  DPP4 COMPLEXED WITH SYN-7AA  |   HYDROLASE 
4n8e:A   (SER511) to   (VAL653)  DPP4 COMPLEXED WITH COMPOUND 12A  |   HYDROLASE 
4n8e:B   (SER511) to   (VAL653)  DPP4 COMPLEXED WITH COMPOUND 12A  |   HYDROLASE 
2jid:A   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH 1-(3,4- DIMETHOXY-PHENYL)-3-M-TOLYL-PIPERIDINE-4-YLAMINE  |   HYDROLASE, DIABETES TYPE II, DIPEPTIDYL PEPTIDASE, PROTEASE, MEMBRANE, B-PROPELLER, STRUCTURE BASED DESIGN, GLYCOPROTEIN, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE FOLD, AMINOPEPTIDASE, SERINE PROTEASE 
3jw8:A    (PRO30) to   (ILE155)  CRYSTAL STRUCTURE OF HUMAN MONO-GLYCERIDE LIPASE  |   ALPHA-BETA HYDROLASE, HYDROLASE 
3jw8:B    (PRO30) to   (ILE155)  CRYSTAL STRUCTURE OF HUMAN MONO-GLYCERIDE LIPASE  |   ALPHA-BETA HYDROLASE, HYDROLASE 
3jwe:B    (PRO30) to   (ILE155)  CRYSTAL STRUCTURE OF HUMAN MONO-GLYCERIDE LIPASE IN COMPLEX WITH SAR629  |   ALPHA-BETA HYDROLASE, HYDROLASE 
2z3z:A   (GLU480) to   (GLY627)  PROLYL TRIPEPTIDYL AMINOPEPTIDASE MUTANT E636A COMPLEXD WITH AN INHIBITOR  |   PEPTIDASE FAMILY S9, PROLYL OLIGOPEPTIDASE FAMILY, SERINE PROTEASE, PROLINE-SPECIFIC PEPTIDASE, HYDROLASE 
2z3w:A   (GLU480) to   (GLY627)  PROLYL TRIPEPTIDYL AMINOPEPTIDASE MUTANT E636A  |   PROLYL OLIGOPEPTIDASE FAMILY, PEPTIDASE FAMILY S9, SERINE PROTEASE, PROLINE-SPECIFIC PEPTIDASE, HYDROLASE 
3kwj:A   (SER511) to   (VAL653)  STRUCUTRE OF HUMAN DPP-IV WITH (2S,3S,11BS)-3-(3-FLUOROMETHYL-PHENYL)- 9,10-DIMETHOXY-1,3,4,6,7,11B-HEXAHYDRO-2H-PYRIDO[2,1-A]ISOQUINOLIN-2- YLAMINE  |   DIABETES TYPE II, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
3l1h:A    (ASP43) to   (ILE171)  CRYSTAL STRUCTURE OF ESTE5, WAS SOAKED BY FECL3  |   HSL, ESTE5, ESTERASE, LIPASE, HYDROLASE 
3l1i:A    (ASP43) to   (ILE171)  CRYSTAL STRUCTURE OF ESTE5, WAS SOAKED BY CUSO4  |   HSL, ESTE5, ESTERASE, LIPASE, HYDROLASE 
4pnz:A   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH THE LONG-ACTING INHIBITOR OMARIGLIPTIN (MK-3102)  |   ALPHA/BETA, BETA-PROPELLER, DIMER, DIABETES, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4pnz:B   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH THE LONG-ACTING INHIBITOR OMARIGLIPTIN (MK-3102)  |   ALPHA/BETA, BETA-PROPELLER, DIMER, DIABETES, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4pv7:A   (SER511) to   (VAL653)  COCRYSTAL STRUCTURE OF DIPEPTIDYL-PEPTIDASE 4 WITH AN INDOLE SCAFFOLD INHIBITOR  |   BETA-PROPELLER, HYDROLASE, EXTROCELLULAR SIDE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4pw0:A    (THR13) to   (GLY131)  ALPHA/BETA HYDROLASE FOLD PROTEIN FROM CHITINOPHAGA PINENSIS  |   STRUCTURAL GENOMICS, APC103277, ALPHA/BETA HYDROLASE FOLD PROTEIN, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, HYDROLASE 
4q3k:A     (MET1) to   (GLY136)  CRYSTAL STRUCTURE OF MGS-M1, AN ALPHA/BETA HYDROLASE ENZYME FROM A MEDEE BASIN DEEP-SEA METAGENOME LIBRARY  |   METAGENOME, METAGENOMIC LIBRARY, ALPHA AND BETA PROTEINS, ALPHA/BETA HYDROLASE SUPERFAMILY, ESTERASE/LIPASE FOLD, HYDROLASE 
4q3l:A     (SER2) to   (ASN121)  CRYSTAL STRUCTURE OF MGS-M2, AN ALPHA/BETA HYDROLASE ENZYME FROM A MEDEE BASIN DEEP-SEA METAGENOME LIBRARY  |   METAGENOME, METAGENOMIC LIBRARY, ALPHA AND BETA PROTEINS, ALPHA/BETA HYDROLASE SUPERFAMILY, ESTERASE/LIPASE FOLD, HYDROLASE 
4q3l:C     (SER2) to   (ASN121)  CRYSTAL STRUCTURE OF MGS-M2, AN ALPHA/BETA HYDROLASE ENZYME FROM A MEDEE BASIN DEEP-SEA METAGENOME LIBRARY  |   METAGENOME, METAGENOMIC LIBRARY, ALPHA AND BETA PROTEINS, ALPHA/BETA HYDROLASE SUPERFAMILY, ESTERASE/LIPASE FOLD, HYDROLASE 
4q3l:D     (SER2) to   (ASN121)  CRYSTAL STRUCTURE OF MGS-M2, AN ALPHA/BETA HYDROLASE ENZYME FROM A MEDEE BASIN DEEP-SEA METAGENOME LIBRARY  |   METAGENOME, METAGENOMIC LIBRARY, ALPHA AND BETA PROTEINS, ALPHA/BETA HYDROLASE SUPERFAMILY, ESTERASE/LIPASE FOLD, HYDROLASE 
4q3l:H     (SER2) to   (ASN121)  CRYSTAL STRUCTURE OF MGS-M2, AN ALPHA/BETA HYDROLASE ENZYME FROM A MEDEE BASIN DEEP-SEA METAGENOME LIBRARY  |   METAGENOME, METAGENOMIC LIBRARY, ALPHA AND BETA PROTEINS, ALPHA/BETA HYDROLASE SUPERFAMILY, ESTERASE/LIPASE FOLD, HYDROLASE 
4q3o:F    (VAL92) to   (GLY221)  CRYSTAL STRUCTURE OF MGS-MT1, AN ALPHA/BETA HYDROLASE ENZYME FROM A LAKE MATAPAN DEEP-SEA METAGENOME LIBRARY  |   METAGENOME, METAGENOMIC LIBRARY, ALPHA AND BETA PROTEINS, ALPHA/BETA HYDROLASE SUPERFAMILY, ESTERASE/LIPASE FOLD, HYDROLASE 
4qa9:A    (TYR65) to   (ASN197)  ENSEMBLE REFINEMENT OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS.  |   STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, EPOXIDE HYDROLASE, PSI-BIOLOGY, HYDROLASE 
3b5e:B    (PRO10) to   (LEU141)  CRYSTAL STRUCTURE OF CARBOXYLESTERASE (NP_108484.1) FROM MESORHIZOBIUM LOTI AT 1.75 A RESOLUTION  |   NP_108484.1, CARBOXYLESTERASE, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, HYDROLASE 
5f4z:A    (PRO67) to   (ASN198)  THE CRYSTAL STRUCTURE OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS  |   EPOXIDE HYDROLASE, STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, HYDROLASE 
5f4z:B    (PRO67) to   (ASN198)  THE CRYSTAL STRUCTURE OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS  |   EPOXIDE HYDROLASE, STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, HYDROLASE 
5f4z:C    (PRO67) to   (ASN198)  THE CRYSTAL STRUCTURE OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS  |   EPOXIDE HYDROLASE, STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, HYDROLASE 
5f4z:D    (VAL66) to   (ASN198)  THE CRYSTAL STRUCTURE OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS  |   EPOXIDE HYDROLASE, STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, HYDROLASE 
5f4z:E    (PRO67) to   (ASN198)  THE CRYSTAL STRUCTURE OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS  |   EPOXIDE HYDROLASE, STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, HYDROLASE 
4qzv:A   (SER511) to   (VAL653)  BAT-DERIVED CORONAVIRUS HKU4 USES MERS-COV RECEPTOR HUMAN CD26 FOR CELL ENTRY  |   8-BLADED BETA-PROPELLER DOMAIN, ALPHA/BETA HYDROLASE DOMAIN, BLADES IV AND V, CD26 BETA-PROPELLER, HYDROLASE-VIRAL PROTEIN COMPLEX 
4qzv:C   (VAL507) to   (VAL653)  BAT-DERIVED CORONAVIRUS HKU4 USES MERS-COV RECEPTOR HUMAN CD26 FOR CELL ENTRY  |   8-BLADED BETA-PROPELLER DOMAIN, ALPHA/BETA HYDROLASE DOMAIN, BLADES IV AND V, CD26 BETA-PROPELLER, HYDROLASE-VIRAL PROTEIN COMPLEX 
3c43:A   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A FLOUROOLEFIN INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE 
3c43:B   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A FLOUROOLEFIN INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE 
3c45:A   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A FLUOROOLEFIN INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE 
3c45:B   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A FLUOROOLEFIN INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE 
3ccb:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A BENZIMIDAZOLE DERIVATIVE  |   STRUCTURE-BASED DESIGN, DENZIMIDAZOLE DERIVATIVES, PEPTIDASE, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
3ccb:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A BENZIMIDAZOLE DERIVATIVE  |   STRUCTURE-BASED DESIGN, DENZIMIDAZOLE DERIVATIVES, PEPTIDASE, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
3ccb:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A BENZIMIDAZOLE DERIVATIVE  |   STRUCTURE-BASED DESIGN, DENZIMIDAZOLE DERIVATIVES, PEPTIDASE, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
3ccc:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A BENZIMIDAZOLE DERIVATIVE  |   STRUCTURE-BASED DESIGN, DENZIMIDAZOLE DERIVATIVES, PEPTIDASE, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
3ccc:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A BENZIMIDAZOLE DERIVATIVE  |   STRUCTURE-BASED DESIGN, DENZIMIDAZOLE DERIVATIVES, PEPTIDASE, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
3ccc:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A BENZIMIDAZOLE DERIVATIVE  |   STRUCTURE-BASED DESIGN, DENZIMIDAZOLE DERIVATIVES, PEPTIDASE, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
3ccc:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A BENZIMIDAZOLE DERIVATIVE  |   STRUCTURE-BASED DESIGN, DENZIMIDAZOLE DERIVATIVES, PEPTIDASE, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
4re5:A   (VAL336) to   (ALA469)  ACYLAMINOACYL PEPTIDASE COMPLEXED WITH A CHLOROMETHYLKETONE INHIBITOR  |   BETA-PROPELLER, ALPHA-BETA-HYDROLASE FOLD, CHLOROMETHYL-KETONE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4re5:B   (VAL336) to   (ALA469)  ACYLAMINOACYL PEPTIDASE COMPLEXED WITH A CHLOROMETHYLKETONE INHIBITOR  |   BETA-PROPELLER, ALPHA-BETA-HYDROLASE FOLD, CHLOROMETHYL-KETONE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4re6:A   (GLY332) to   (ALA469)  ACYLAMINOACYL PEPTIDASE COMPLEXED WITH A CHLOROMETHYLKETONE INHIBITOR  |   BETA-PROPELLER, ALPHA-BETA-HYDROLASE FOLD, CHLOROMETHYL-KETONE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4re6:B   (GLY332) to   (ALA469)  ACYLAMINOACYL PEPTIDASE COMPLEXED WITH A CHLOROMETHYLKETONE INHIBITOR  |   BETA-PROPELLER, ALPHA-BETA-HYDROLASE FOLD, CHLOROMETHYL-KETONE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4re6:C   (GLY332) to   (ALA469)  ACYLAMINOACYL PEPTIDASE COMPLEXED WITH A CHLOROMETHYLKETONE INHIBITOR  |   BETA-PROPELLER, ALPHA-BETA-HYDROLASE FOLD, CHLOROMETHYL-KETONE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4re6:D   (GLY332) to   (ALA469)  ACYLAMINOACYL PEPTIDASE COMPLEXED WITH A CHLOROMETHYLKETONE INHIBITOR  |   BETA-PROPELLER, ALPHA-BETA-HYDROLASE FOLD, CHLOROMETHYL-KETONE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4c88:B    (ARG76) to   (LEU201)  ESTERASE LPEST1 FROM LACTOBACILLUS PLANTARUM: NATIVE STRUCTURE  |   HYDROLASE 
4c88:C    (ARG76) to   (LEU201)  ESTERASE LPEST1 FROM LACTOBACILLUS PLANTARUM: NATIVE STRUCTURE  |   HYDROLASE 
4c89:B    (ARG76) to   (LEU201)  CRYSTAL STRUCTURE OF CARBOXYLESTERASE LPEST1 FROM LACTOBACILLUS PLANTARUM: HIGH RESOLUTION MODEL  |   HYDROLASE 
4c89:C    (ARG76) to   (LEU201)  CRYSTAL STRUCTURE OF CARBOXYLESTERASE LPEST1 FROM LACTOBACILLUS PLANTARUM: HIGH RESOLUTION MODEL  |   HYDROLASE 
3nox:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH SA-(+)-(6- (AMINOMETHYL)-5-(2,4-DICHLOROPHENYL)-7-METHYLIMIDAZO[1,2-A]PYRIMIDIN- 2-YL)(MORPHOLINO)METHANONE  |   EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE 
3nox:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH SA-(+)-(6- (AMINOMETHYL)-5-(2,4-DICHLOROPHENYL)-7-METHYLIMIDAZO[1,2-A]PYRIMIDIN- 2-YL)(MORPHOLINO)METHANONE  |   EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE 
3cxu:A     (LYS3) to   (LEU128)  STRUCTURE OF A Y149F MUTANT OF EPOXIDE HYDROLASE FROM SOLANUM TUBEROSUM  |   EPOXIDE HYDROLASE, ALPHA/BETA HYDROLASE FOLD, Y149F, PROTON WIRE 
3o4h:A   (VAL336) to   (ALA469)  STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY 
3o4h:B   (VAL336) to   (ALA469)  STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY 
3o4h:C   (VAL336) to   (ALA469)  STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY 
3o4h:D   (VAL336) to   (ALA469)  STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY 
3o4j:A   (GLY332) to   (ALA469)  STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY 
3o4j:B   (GLY332) to   (ALA469)  STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY 
3o4j:C   (GLY332) to   (ALA469)  STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY 
3o4j:D   (GLY332) to   (ALA469)  STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY 
3o95:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-100  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX 
3o95:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-100  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX 
3o95:C   (SER511) to   (ALA654)  CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-100  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX 
3o95:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-100  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX 
3d4l:A   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A NOVEL INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE 
3d4l:B   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A NOVEL INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE 
3o9v:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-986  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX 
3o9v:B   (SER511) to   (ALA654)  CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-986  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX 
3o9v:C   (SER511) to   (ALA654)  CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-986  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX 
3o9v:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-986  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX 
3doi:A   (PHE162) to   (CYS310)  CRYSTAL STRUCTURE OF A THERMOSTABLE ESTERASE COMPLEX WITH PARAOXON  |   ALPHA-BETA HYDROLASE, BETA SHEET 
3opm:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-294  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE-HYDROLASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3opm:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-294  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE-HYDROLASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3opm:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-294  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE-HYDROLASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3opm:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-294  |   PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE-HYDROLASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3e3a:A   (LEU-11) to   (ALA111)  THE STRUCTURE OF RV0554 FROM MYCOBACTERIUM TUBERCULOSIS  |   ALPHA/BETA HYDROLASE, OXIDOREDUCTASE, PEROXIDASE 
3e3a:B   (GLU-13) to   (ALA111)  THE STRUCTURE OF RV0554 FROM MYCOBACTERIUM TUBERCULOSIS  |   ALPHA/BETA HYDROLASE, OXIDOREDUCTASE, PEROXIDASE 
4dsz:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DPP-IV WITH COMPOUND C2  |   INHIBITOR COMPLEX, SERINE EXOPEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4dsz:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DPP-IV WITH COMPOUND C2  |   INHIBITOR COMPLEX, SERINE EXOPEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4dtc:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DPP-IV WITH COMPOUND C5  |   INHIBITOR COMPLEX, SERINE EXOPEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4dtc:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DPP-IV WITH COMPOUND C5  |   INHIBITOR COMPLEX, SERINE EXOPEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3pf8:A     (GLY0) to   (ALA130)  CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536  |   ALPHA/BETA HYDROLASE FOLD, ESTERASE, HYDROLASE, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES, EXTRACELLULAR 
3pf8:B     (ALA2) to   (ALA130)  CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536  |   ALPHA/BETA HYDROLASE FOLD, ESTERASE, HYDROLASE, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES, EXTRACELLULAR 
3pf9:A     (GLY0) to   (ALA130)  CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536 S106A MUTANT  |   ALPHA/BETA HYDROLASE FOLD, ESTERASE, HYDROLASE, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES, EXTRACELLULAR 
3pfb:A     (GLY0) to   (LEU129)  CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536 S106A MUTANT IN COMPLEX WITH ETHYLFERULATE  |   ALPHA/BETA HYDROLASE FOLD, ESTERASE, HYDROLASE, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES, EXTRACELLULAR 
3pfc:A     (GLY0) to   (ALA130)  CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536 S106A MUTANT IN COMPLEX WITH FERULIC ACID  |   ALPHA/BETA HYDROLASE FOLD, ESTERASE, HYDROLASE, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES, EXTRACELLULAR 
4ufn:B     (LYS3) to   (LEU128)  LABORATORY EVOLVED VARIANT R-C1B1 OF POTATO EPOXIDE HYDROLASE STEH1  |   HYDROLASE, EPOXIDE HYDROLYSIS, ALPHA/BETA-HYDROLASE, DIRECTED EVOLUTION, ASYMMETRIC SYNTHESES 
4ufo:B     (LYS3) to   (LEU128)  LABORATORY EVOLVED VARIANT R-C1B1D33E6 OF POTATO EPOXIDE HYDROLASE STEH1  |   HYDROLASE, EPOXIDE HYDROLYSIS, ALPHA/BETA-HYDROLASE, DIRECTED EVOLUTION, ASYMMETRIC SYNTHESES 
4ufp:A     (LYS3) to   (LEU128)  LABORATORY EVOLVED VARIANT R-C1B1D33 OF POTATO EPOXIDE HYDROLASE STEH1  |   HYDROLASE, EPOXIDE HYDROLYSIS, ALPHA/BETA-HYDROLASE, DIRECTED EVOLUTION, ASYMMETRIC SYNTHESES 
4ufp:B     (LYS3) to   (LEU128)  LABORATORY EVOLVED VARIANT R-C1B1D33 OF POTATO EPOXIDE HYDROLASE STEH1  |   HYDROLASE, EPOXIDE HYDROLYSIS, ALPHA/BETA-HYDROLASE, DIRECTED EVOLUTION, ASYMMETRIC SYNTHESES 
3q0t:A   (SER511) to   (ALA654)  CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITHSA-(+)- METHYL2-(3- (AMINOMETHYL)-4-(2,4-DICHLOROPHENYL)-2-METHYL- 7-OXO-5H-PYRROLO[3,4- B]PYRIDIN-6(7H)-YL)ACETATE  |   EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3q0t:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITHSA-(+)- METHYL2-(3- (AMINOMETHYL)-4-(2,4-DICHLOROPHENYL)-2-METHYL- 7-OXO-5H-PYRROLO[3,4- B]PYRIDIN-6(7H)-YL)ACETATE  |   EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5ivi:A    (CYS89) to   (SER244)  THE ALPHA-ESTERASE-7 CARBOXYLESTERASE, E3, FROM THE BLOWFLY LUCILIA CUPRINA: PHOSPHORYLATED ENZYME QFIT MULTI-CONFORMER MODEL  |   CARBOXYLESTERASE, ORGANOPHOSPHATE, PROTEIN DYNAMICS, ACETYLCHOLINESTERASE, HYDROLASE 
3qm1:A     (GLY0) to   (ALA130)  CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536 S106A MUTANT IN COMPLEX WITH ETHYLFERULATE, FORM II  |   ALPHA/BETA HYDROLASE FOLD, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES, HYDROLASE 
4w1p:A    (CYS89) to   (SER244)  KINETIC CRYSTALLOGRAPHY OF ALPHA_E7-CARBOXYLESTERSE FROM LUCILLA CUPRINA - ABSORBED X-RAY DOSE 5.54 MGY TEMP 150K  |   ALPHA/BETA HYDROLASE FOLD, CARBOXYLESTERASE, HYDROLASE 
4w1r:A    (CYS89) to   (SER244)  KINETIC CRYSTALLOGRAPHY OF ALPHA_E7-CARBOXYLESTERSE FROM LUCILLA CUPRINA - ABSORBED X-RAY DOSE 9.24 MGY TEMP 150K  |   ALPHA/BETA HYDROLASE FOLD, CARBOXYLESTERASE, HYDROLASE 
3r3u:A    (GLY10) to   (LEU133)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - WT/APO  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r3u:B    (GLY10) to   (LEU133)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - WT/APO  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r3v:B    (GLY10) to   (LEU133)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - ASP110ASN/FLUOROACETATE  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r3w:A    (GLY10) to   (LEU133)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - ASP110ASN/CHLOROACETATE  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r3w:B    (GLY10) to   (LEU133)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - ASP110ASN/CHLOROACETATE  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r3x:A    (GLY12) to   (LEU133)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - ASP110ASN/BROMOACETATE  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r3x:B    (GLY10) to   (LEU133)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - ASP110ASN/BROMOACETATE  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r3y:A    (GLY12) to   (ASP134)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - HIS280ASN/FLUOROACETATE  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r3y:B    (GLY10) to   (ASP134)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - HIS280ASN/FLUOROACETATE  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r3z:A    (GLY10) to   (LEU133)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - WT/GLYCOLATE  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r3z:B    (GLY10) to   (LEU133)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - WT/GLYCOLATE  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r3z:C    (GLY10) to   (ASP134)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - WT/GLYCOLATE  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r3z:D    (GLY10) to   (LEU133)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - WT/GLYCOLATE  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r40:A    (GLY10) to   (LEU133)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - ASP110ASN/APO  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r40:B    (GLY10) to   (LEU133)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - ASP110ASN/APO  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r41:A    (GLY10) to   (ASP134)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - HIS280ASN/APO  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
3r41:B    (GLY10) to   (ASP134)  CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - HIS280ASN/APO  |   FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE 
4g1f:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIDOPYRIMIDINEDIONE ANALOGUE  |   PROTEASE, 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, SECRETED, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4g1f:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIDOPYRIMIDINEDIONE ANALOGUE  |   PROTEASE, 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, SECRETED, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4g1f:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIDOPYRIMIDINEDIONE ANALOGUE  |   PROTEASE, 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, SECRETED, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4g1f:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIDOPYRIMIDINEDIONE ANALOGUE  |   PROTEASE, 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, SECRETED, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5l8s:A   (MET341) to   (PHE482)  THE CRYSTAL STRUCTURE OF A COLD-ADAPTED ACYLAMINOACYL PEPTIDASE REVEALS A NOVEL QUATERNARY ARCHITECTURE BASED ON THE ARM-EXCHANGE MECHANISM  |   ACYL AMINOACYL PEPTIDASE, ALPHA/BETA HYDROLASE DOMAIN, ARM EXCHANGE, BETA-PROPELLER DOMAIN, COLD ADAPTATION, DIMERIZATION, PROLINE HINGE, SPOROSARCINA PSYCHROPHILA, HYDROLASE 
5l8s:B   (MET341) to   (PHE482)  THE CRYSTAL STRUCTURE OF A COLD-ADAPTED ACYLAMINOACYL PEPTIDASE REVEALS A NOVEL QUATERNARY ARCHITECTURE BASED ON THE ARM-EXCHANGE MECHANISM  |   ACYL AMINOACYL PEPTIDASE, ALPHA/BETA HYDROLASE DOMAIN, ARM EXCHANGE, BETA-PROPELLER DOMAIN, COLD ADAPTATION, DIMERIZATION, PROLINE HINGE, SPOROSARCINA PSYCHROPHILA, HYDROLASE 
5t4b:A   (SER511) to   (VAL653)  HUMAN DPP4 IN COMPLEX WITH A LIGAND 34A  |   STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5t4b:B   (SER511) to   (VAL653)  HUMAN DPP4 IN COMPLEX WITH A LIGAND 34A  |   STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5t4e:A   (SER511) to   (VAL653)  HUMAN DPP4 IN COMPLEX WITH LIGAND 19A  |   STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5t4e:B   (SER511) to   (VAL653)  HUMAN DPP4 IN COMPLEX WITH LIGAND 19A  |   STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5t4f:A   (SER511) to   (VAL653)  HUMAN DPP4 IN COMPLEX WITH LIGAND 34P  |   STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5t4f:B   (SER511) to   (VAL653)  HUMAN DPP4 IN COMPLEX WITH LIGAND 34P  |   STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5t4h:A   (SER511) to   (VAL653)  HUMAN DPP4 IN COMPLEX WITH LIGAND 34N  |   STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5t4h:B   (SER511) to   (VAL653)  HUMAN DPP4 IN COMPLEX WITH LIGAND 34N  |   STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
2ajb:B   (SER511) to   (ALA654)  PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH THE TRIPEPTIDE TERT-BUTYL-GLY-L-PRO-L-ILE (TBU-GPI)  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
2ajb:C   (SER511) to   (VAL653)  PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH THE TRIPEPTIDE TERT-BUTYL-GLY-L-PRO-L-ILE (TBU-GPI)  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
2ajb:D   (SER511) to   (VAL653)  PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH THE TRIPEPTIDE TERT-BUTYL-GLY-L-PRO-L-ILE (TBU-GPI)  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
2ajd:B   (SER511) to   (VAL653)  PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH L-PRO-BORO-L- PRO (BOROPRO)  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE 
2ajd:C   (SER511) to   (ALA654)  PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH L-PRO-BORO-L- PRO (BOROPRO)  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE 
2ajd:D   (SER511) to   (VAL653)  PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH L-PRO-BORO-L- PRO (BOROPRO)  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE 
3ed1:C    (VAL63) to   (LEU224)  CRYSTAL STRUCTURE OF RICE GID1 COMPLEXED WITH GA3  |   ALPHA/BETA HYDROLASE, LIPASE, GIBBERELLIN SIGNALING PATHWAY, HYDROLASE, NUCLEUS, RECEPTOR, HYDROLASE RECEPTOR 
3ed1:E    (VAL63) to   (LEU224)  CRYSTAL STRUCTURE OF RICE GID1 COMPLEXED WITH GA3  |   ALPHA/BETA HYDROLASE, LIPASE, GIBBERELLIN SIGNALING PATHWAY, HYDROLASE, NUCLEUS, RECEPTOR, HYDROLASE RECEPTOR 
3ed1:F    (VAL63) to   (LEU224)  CRYSTAL STRUCTURE OF RICE GID1 COMPLEXED WITH GA3  |   ALPHA/BETA HYDROLASE, LIPASE, GIBBERELLIN SIGNALING PATHWAY, HYDROLASE, NUCLEUS, RECEPTOR, HYDROLASE RECEPTOR 
2oph:A   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH AN ALPHA AMINO ACID INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, TYPE 2 DIABETES, SELECTIVE INHIBITOR, HYDROLASE 
2oph:B   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH AN ALPHA AMINO ACID INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, TYPE 2 DIABETES, SELECTIVE INHIBITOR, HYDROLASE 
2p8s:A   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A CYCLOHEXALAMINE INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, STRUCTURE-BASED DESIGN, HYDROLASE 
2p8s:B   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A CYCLOHEXALAMINE INHIBITOR  |   ALPHA/BETA, BETA-PROPELLER, DIMER, STRUCTURE-BASED DESIGN, HYDROLASE 
1bn6:A    (ASP22) to   (MET140)  HALOALKANE DEHALOGENASE FROM A RHODOCOCCUS SPECIES  |   DEHALOGENASE, ALPHA/BETA-HYDROLASE, DHLA, CRYSTAL STRUCTURE 
2buc:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A TETRAHYDROISOQUINOLINE INHIBITOR  |   HYDROLASE/INHIBITOR, COMPLEX (HYDROLASE/INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX 
2buc:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A TETRAHYDROISOQUINOLINE INHIBITOR  |   HYDROLASE/INHIBITOR, COMPLEX (HYDROLASE/INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX 
2buc:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A TETRAHYDROISOQUINOLINE INHIBITOR  |   HYDROLASE/INHIBITOR, COMPLEX (HYDROLASE/INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX 
2buc:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A TETRAHYDROISOQUINOLINE INHIBITOR  |   HYDROLASE/INHIBITOR, COMPLEX (HYDROLASE/INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX 
1orw:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A PEPTIDOMIMETIC INHIBITOR  |   SERINE PROTEASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, HYDROLASE 
1orw:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A PEPTIDOMIMETIC INHIBITOR  |   SERINE PROTEASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, HYDROLASE 
2q2e:A   (GLY178) to   (GLY289)  CRYSTAL STRUCTURE OF THE TOPOISOMERASE VI HOLOENZYME FROM METHANOSARCINA MAZEI  |   TOPOISOMERASE, DNA-BINDING, SPO11, ATPASE, ISOMERASE 
3fvt:B    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM II  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvt:F    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM II  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvt:I    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM II  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvt:L    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM II  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3fvt:M    (GLY53) to   (ASP203)  CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM II  |   ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE 
3g0c:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 1  |   DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0c:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 1  |   DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0c:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 1  |   DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3g0c:D   (VAL507) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 1  |   DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
2qjr:A   (SER511) to   (VAL653)  DIPEPDYL PEPTIDASE IV IN COMPLEX WITH INHIBITOR PZF  |   PROTEIN-INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
2qjr:B   (SER511) to   (VAL653)  DIPEPDYL PEPTIDASE IV IN COMPLEX WITH INHIBITOR PZF  |   PROTEIN-INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
3t4u:A     (SER1) to   (GLY119)  L29I MUTATION IN AN ARYL ESTERASE FROM PSEUDOMONAS FLUORESCENS LEADS TO UNIQUE PEPTIDE FLIP AND INCREASED ACTIVITY  |   OXIDOREDUCTASE, HYDRLOASE 
3t4u:B     (SER1) to   (GLY119)  L29I MUTATION IN AN ARYL ESTERASE FROM PSEUDOMONAS FLUORESCENS LEADS TO UNIQUE PEPTIDE FLIP AND INCREASED ACTIVITY  |   OXIDOREDUCTASE, HYDRLOASE 
3t4u:C     (SER1) to   (GLY119)  L29I MUTATION IN AN ARYL ESTERASE FROM PSEUDOMONAS FLUORESCENS LEADS TO UNIQUE PEPTIDE FLIP AND INCREASED ACTIVITY  |   OXIDOREDUCTASE, HYDRLOASE 
3t4u:D     (SER1) to   (GLY119)  L29I MUTATION IN AN ARYL ESTERASE FROM PSEUDOMONAS FLUORESCENS LEADS TO UNIQUE PEPTIDE FLIP AND INCREASED ACTIVITY  |   OXIDOREDUCTASE, HYDRLOASE 
3t4u:E     (SER1) to   (GLY119)  L29I MUTATION IN AN ARYL ESTERASE FROM PSEUDOMONAS FLUORESCENS LEADS TO UNIQUE PEPTIDE FLIP AND INCREASED ACTIVITY  |   OXIDOREDUCTASE, HYDRLOASE 
3t4u:F     (SER1) to   (GLY119)  L29I MUTATION IN AN ARYL ESTERASE FROM PSEUDOMONAS FLUORESCENS LEADS TO UNIQUE PEPTIDE FLIP AND INCREASED ACTIVITY  |   OXIDOREDUCTASE, HYDRLOASE 
3h17:A    (ASP43) to   (ILE171)  CRYSTAL STRUCTURE OF ESTE5-PMSF (I)  |   HSL, ESTE5, ESTERASE, LIPASE, HYDROLASE, PMSF, PHENYLMETHYLSULFONYL FLUORIDE 
3hab:A   (SER511) to   (VAL653)  THE STRUCTURE OF DPP4 IN COMPLEX WITH PIPERIDINE FUSED BENZIMIDAZOLE 25  |   ALPHA/BETA, BETA-PROPELLER, DIMER, HYDROLASE, DIABETES, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3hab:B   (SER511) to   (VAL653)  THE STRUCTURE OF DPP4 IN COMPLEX WITH PIPERIDINE FUSED BENZIMIDAZOLE 25  |   ALPHA/BETA, BETA-PROPELLER, DIMER, HYDROLASE, DIABETES, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3hac:A   (SER511) to   (VAL653)  THE STRUCTURE OF DPP-4 IN COMPLEX WITH PIPERIDINE FUSED IMIDAZOPYRIDINE 34  |   ALPHA/BETA, BETA-PROPELLER, DIMER, HYDROLASE, DIABETES, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3hac:B   (SER511) to   (VAL653)  THE STRUCTURE OF DPP-4 IN COMPLEX WITH PIPERIDINE FUSED IMIDAZOPYRIDINE 34  |   ALPHA/BETA, BETA-PROPELLER, DIMER, HYDROLASE, DIABETES, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3hju:A    (PRO20) to   (ILE145)  CRYSTAL STRUCTURE OF HUMAN MONOGLYCERIDE LIPASE  |   ALPHA/BETA HYDROLASE, HYDROLASE, SERINE ESTERASE 
2fuk:A    (LEU13) to   (ALA141)  CRYSTAL STRUCTURE OF XC6422 FROM XANTHOMONAS CAMPESTRIS: A MEMBER OF A/B SERINE HYDROLASE WITHOUT LID AT 1.6 RESOLUTION  |   A/B HYDROLASE, XANTHOMONAS CAMPESTRIS, STRUCTURAL GENOMICS, X-RAY DIFFRACTION 
1sfr:A     (PRO7) to   (MET149)  CRYSTAL STRUCTURE OF THE MYCOBACTERIUM TUBERCULOSIS ANTIGEN 85A PROTEIN  |   ALPHA/BETA HYDROLASE, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, TRANSFERASE 
2gbc:A   (SER512) to   (VAL654)  NATIVE DPP-IV (CD26) FROM RAT  |   BETA PROPELLER, HYDROLASE 
2gbc:B   (SER512) to   (VAL654)  NATIVE DPP-IV (CD26) FROM RAT  |   BETA PROPELLER, HYDROLASE 
1tht:A     (LYS6) to   (ALA135)  STRUCTURE OF A MYRISTOYL-ACP-SPECIFIC THIOESTERASE FROM VIBRIO HARVEYI  |   THIOESTERASE 
1tht:B     (LYS6) to   (VAL136)  STRUCTURE OF A MYRISTOYL-ACP-SPECIFIC THIOESTERASE FROM VIBRIO HARVEYI  |   THIOESTERASE 
1tk3:A   (SER511) to   (ALA654)  CRYSTAL STRUCTURE OF HUMAN APO DIPEPTIDYL PEPTIDASE IV/CD26  |   ALPHA/BETA HYDROLASE, BETA-PROPELLER, HOMODIMER, HYDROLASE 
1tk3:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN APO DIPEPTIDYL PEPTIDASE IV/CD26  |   ALPHA/BETA HYDROLASE, BETA-PROPELLER, HOMODIMER, HYDROLASE 
1tkr:B   (SER511) to   (ALA654)  HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 INHIBITED WITH DIISOPROPYL FLUOROPHOSPHATE  |   ALPHA/BETA HYDROLASE, BETA-PROPELLER, HOMODIMER, HYDROLASE 
4zxf:A    (GLU14) to   (SER148)  CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE IN COMPLEX WITH A SUBSTRATE ANALOG  |   HYDROLASE, MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, COMPLEX, SUBSTRATE ANALOG 
4zxf:B    (GLU14) to   (GLY149)  CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE IN COMPLEX WITH A SUBSTRATE ANALOG  |   HYDROLASE, MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, COMPLEX, SUBSTRATE ANALOG 
4zxf:C    (GLU14) to   (SER148)  CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE IN COMPLEX WITH A SUBSTRATE ANALOG  |   HYDROLASE, MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, COMPLEX, SUBSTRATE ANALOG 
4zxf:D    (PRO13) to   (GLY149)  CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE IN COMPLEX WITH A SUBSTRATE ANALOG  |   HYDROLASE, MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, COMPLEX, SUBSTRATE ANALOG 
2hha:A   (SER511) to   (VAL653)  THE STRUCTURE OF DPP4 IN COMPLEX WITH AN OXADIAZOLE INHIBITOR  |   HYDROLASE, ALPHA/BETA, BETA-PROPELLER, DIMER 
2hha:B   (SER511) to   (VAL653)  THE STRUCTURE OF DPP4 IN COMPLEX WITH AN OXADIAZOLE INHIBITOR  |   HYDROLASE, ALPHA/BETA, BETA-PROPELLER, DIMER 
2i03:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE 4 (DPP IV) WITH POTENT ALKYNYL CYANOPYRROLIDINE (ABT-279)  |   ENZYME, SERINE PEPTIDASE, HYDROLASE 
2iit:A   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE 4 IN COMPLEX WITH A DIAZEPAN-2-ONE INHIBITOR  |   HYDROLASE; ALPHA/BETA; BETA-PROPELLER; DIMER, HYDROLASE 
2iit:B   (SER511) to   (VAL653)  HUMAN DIPEPTIDYL PEPTIDASE 4 IN COMPLEX WITH A DIAZEPAN-2-ONE INHIBITOR  |   HYDROLASE; ALPHA/BETA; BETA-PROPELLER; DIMER, HYDROLASE 
1wcy:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) COMPLEX WITH DIPROTIN A  |   SERINE PROTEASE, DIPEPTIDYL PEPTIDASE IV, CD26, PROLYL OLIGOPEPTIDASE, BETA-PROPELLER STRUCTURE, DIPROTIN A, HYDROLASE 
4a5s:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A NOVAL HETEROCYCLIC DPP4 INHIBITOR  |   HYDROLASE, TYPE 2 DIABETES, NOVARTIS COMPOUND NVP-BIV988 
4a5s:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A NOVAL HETEROCYCLIC DPP4 INHIBITOR  |   HYDROLASE, TYPE 2 DIABETES, NOVARTIS COMPOUND NVP-BIV988 
3kwf:B   (SER511) to   (VAL653)  HUMAN DPP-IV WITH CARMEGLIPTIN (S)-1-((2S,3S,11BS)-2-AMINO- 9,10-DIMETHOXY-1,3,4,6,7,11B-HEXAHYDRO-2H-PYRIDO[2,1- A]ISOQUINOLIN-3-YL)-4-FLUOROMETHYL-PYRROLIDIN-2-ONE  |   DIABETES TYPE II, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE 
1z68:A   (ASN500) to   (VAL647)  CRYSTAL STRUCTURE OF HUMAN FIBROBLAST ACTIVATION PROTEIN ALPHA  |   SEPRASE, FIBROBLAST ACTIVATION PROTEIN ALPHA,FAPALPHA, DIPEPTIDYLPEPTIDASE,S9B, INTEGRAL MEMBRANE SERINE PROTEASE, LYASE 
1z68:B   (PRO504) to   (VAL647)  CRYSTAL STRUCTURE OF HUMAN FIBROBLAST ACTIVATION PROTEIN ALPHA  |   SEPRASE, FIBROBLAST ACTIVATION PROTEIN ALPHA,FAPALPHA, DIPEPTIDYLPEPTIDASE,S9B, INTEGRAL MEMBRANE SERINE PROTEASE, LYASE 
4q1v:A   (TYR476) to   (GLY626)  CRYSTAL STRUCTURE OF A PUTATIVE DIPEPTIDYL AMINOPEPTIDASE IV (BACOVA_01349) FROM BACTEROIDES OVATUS ATCC 8483 AT 2.48 A RESOLUTION  |   TWO DOMAIN PROTEIN, DIPEPTIDYL-PEPTIDASE IV FAMILY (PF00930), PROLYL OLIGOPEPTIDASE FAMILY (PF00326), STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI- BIOLOGY, HYDROLASE 
4q1v:B   (TYR476) to   (GLY627)  CRYSTAL STRUCTURE OF A PUTATIVE DIPEPTIDYL AMINOPEPTIDASE IV (BACOVA_01349) FROM BACTEROIDES OVATUS ATCC 8483 AT 2.48 A RESOLUTION  |   TWO DOMAIN PROTEIN, DIPEPTIDYL-PEPTIDASE IV FAMILY (PF00930), PROLYL OLIGOPEPTIDASE FAMILY (PF00326), STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI- BIOLOGY, HYDROLASE 
3bjm:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH (1S,3S, 5S)-2-[(2S)- 2-AMINO-2-(3-HYDROXYTRICYCLO[3.3.1.13,7]DEC-1- YL)ACETYL]-2- AZABICYCLO[3.1.0]HEXANE-3-CARBONITRILE (CAS), (1S,3S,5S)-2-((2S)-2- AMINO-2-(3-HYDROXYADAMANTAN-1- YL)ACETYL)-2-AZABICYCLO[3.1.0]HEXANE- 3-CARBONITRILE (IUPAC), OR BMS-477118  |   EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE 
3bjm:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH (1S,3S, 5S)-2-[(2S)- 2-AMINO-2-(3-HYDROXYTRICYCLO[3.3.1.13,7]DEC-1- YL)ACETYL]-2- AZABICYCLO[3.1.0]HEXANE-3-CARBONITRILE (CAS), (1S,3S,5S)-2-((2S)-2- AMINO-2-(3-HYDROXYADAMANTAN-1- YL)ACETYL)-2-AZABICYCLO[3.1.0]HEXANE- 3-CARBONITRILE (IUPAC), OR BMS-477118  |   EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE 
4c87:C    (ARG76) to   (LEU201)  ESTERASE LPEST1 FROM LACTOBACILLUS PLANTARUM WCFS1  |   HYDROLASE 
3o4g:A   (GLY332) to   (ALA469)  STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY 
3o4g:B   (VAL336) to   (ALA469)  STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY 
3o4g:C   (GLY332) to   (ALA469)  STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY 
3o4g:D   (VAL336) to   (ALA469)  STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY 
3o4i:A   (VAL336) to   (ALA469)  STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY 
3o4i:B   (VAL336) to   (ALA469)  STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE  |   ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY 
3our:C   (TYR166) to   (GLY296)  CRYSTAL STRUCTURE OF COMPLEX BETWEEN EIIA AND A NOVEL PYRUVATE DECARBOXYLASE  |   EXHIBIT NO HYDROLASE ACTIVITY1, LYASE-TRANSFERASE COMPLEX 
5i7u:A   (SER511) to   (VAL653)  HUMAN DPP4 IN COMPLEX WITH A NOVEL TRICYCLIC HETERO-CYCLE INHIBITOR  |   STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5i7u:B   (SER511) to   (VAL653)  HUMAN DPP4 IN COMPLEX WITH A NOVEL TRICYCLIC HETERO-CYCLE INHIBITOR  |   STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
4uuq:A    (PRO30) to   (ILE155)  CRYSTAL STRUCTURE OF HUMAN MONO-GLYCERIDE LIPASE IN COMPLEX WITH SAR127303  |   HYDROLASE 
5ism:A   (SER511) to   (VAL653)  HUMAN DPP4 IN COMPLEX WITH A NOVEL 5,5,6-TRICYCLIC PYRROLIDINE INHIBITOR  |   STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5ism:B   (SER511) to   (VAL653)  HUMAN DPP4 IN COMPLEX WITH A NOVEL 5,5,6-TRICYCLIC PYRROLIDINE INHIBITOR  |   STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3qbj:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH INHIBITOR  |   DIABETES MELLITUS, DIPEPTIDYL-PEPTIDASE IV INHIBITOR, HYPOGLYCEMIC AGENT, PYRROLIDINES, SPRAGUE-DAWLEY, STRUCTURE-ACTIVITY RELATIONSHIP, HYDROLASE, GLYCOSYLATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
3qbj:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH INHIBITOR  |   DIABETES MELLITUS, DIPEPTIDYL-PEPTIDASE IV INHIBITOR, HYPOGLYCEMIC AGENT, PYRROLIDINES, SPRAGUE-DAWLEY, STRUCTURE-ACTIVITY RELATIONSHIP, HYDROLASE, GLYCOSYLATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5kby:A   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH SYR-472  |   PEPTIDASE, GLP-1, METABOLIC DISEASE, CO-COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5kby:B   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH SYR-472  |   PEPTIDASE, GLP-1, METABOLIC DISEASE, CO-COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5kby:C   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH SYR-472  |   PEPTIDASE, GLP-1, METABOLIC DISEASE, CO-COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5kby:D   (SER511) to   (VAL653)  CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH SYR-472  |   PEPTIDASE, GLP-1, METABOLIC DISEASE, CO-COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX 
5lls:A   (SER511) to   (VAL653)  PORCINE DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH 8-(3-AMINOPIPERIDIN-1- YL)-7-[(2-BROMOPHENYL)METHYL]-1,3-DIMETHYL-2,3,6,7-TETRAHYDRO-1H- PURINE-2,6-DIONE  |   PEPTIDASE, INHIBITOR, COMPLEX, HYDROLASE 
5lls:B   (SER511) to   (VAL653)  PORCINE DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH 8-(3-AMINOPIPERIDIN-1- YL)-7-[(2-BROMOPHENYL)METHYL]-1,3-DIMETHYL-2,3,6,7-TETRAHYDRO-1H- PURINE-2,6-DIONE  |   PEPTIDASE, INHIBITOR, COMPLEX, HYDROLASE 
5lls:C   (SER511) to   (VAL653)  PORCINE DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH 8-(3-AMINOPIPERIDIN-1- YL)-7-[(2-BROMOPHENYL)METHYL]-1,3-DIMETHYL-2,3,6,7-TETRAHYDRO-1H- PURINE-2,6-DIONE  |   PEPTIDASE, INHIBITOR, COMPLEX, HYDROLASE 
5lls:D   (SER511) to   (VAL653)  PORCINE DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH 8-(3-AMINOPIPERIDIN-1- YL)-7-[(2-BROMOPHENYL)METHYL]-1,3-DIMETHYL-2,3,6,7-TETRAHYDRO-1H- PURINE-2,6-DIONE  |   PEPTIDASE, INHIBITOR, COMPLEX, HYDROLASE