2oag:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) WITH PYRROLIDINE-CONSTRAINED PHENETHYLAMINE 29G | SERINE-PEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2oag:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) WITH PYRROLIDINE-CONSTRAINED PHENETHYLAMINE 29G | SERINE-PEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2aj8:A (SER511) to (VAL653) PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH 7-BENZYL-1,3- DIMETHYL-8-PIPERAZIN-1-YL-3,7-DIHYDRO-PURINE-2,6-DIONE (BDPX) | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE
2aj8:B (SER511) to (VAL653) PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH 7-BENZYL-1,3- DIMETHYL-8-PIPERAZIN-1-YL-3,7-DIHYDRO-PURINE-2,6-DIONE (BDPX) | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE
2aj8:C (SER511) to (VAL653) PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH 7-BENZYL-1,3- DIMETHYL-8-PIPERAZIN-1-YL-3,7-DIHYDRO-PURINE-2,6-DIONE (BDPX) | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE
2aj8:D (SER511) to (VAL653) PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH 7-BENZYL-1,3- DIMETHYL-8-PIPERAZIN-1-YL-3,7-DIHYDRO-PURINE-2,6-DIONE (BDPX) | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE
2ajc:C (SER511) to (VAL653) PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH 4-(2- AMINOETHYL)-BENZENE SULPHONYL FLUORIDE (AEBSF) | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2ajc:D (SER511) to (VAL653) PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH 4-(2- AMINOETHYL)-BENZENE SULPHONYL FLUORIDE (AEBSF) | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2ajl:J (SER511) to (VAL653) X-RAY STRUCTURE OF NOVEL BIARYL-BASED DIPEPTIDYL PEPTIDASE IV INHIBITOR | AMINOPEPTIDASE, HYDROLASE, PROTEASE, SERINE PROTEASE
2og1:A (GLY19) to (MET135) CRYSTAL STRUCTURE OF BPHD, A C-C HYDROLASE FROM BURKHOLDERIA XENOVORANS LB400 | BPHD, ALPHA/BETA HYDROLASE, PCB DEGRADATION, META CLEAVAGE PRODUCT HYDROLASE, MCP HYDROLASE, 2-HYDROXY-6-OXO-6-PHENYLHEXA-2, 4-DIENOATE HYDROLASE, HYDROLASE
2og1:B (GLY19) to (MET135) CRYSTAL STRUCTURE OF BPHD, A C-C HYDROLASE FROM BURKHOLDERIA XENOVORANS LB400 | BPHD, ALPHA/BETA HYDROLASE, PCB DEGRADATION, META CLEAVAGE PRODUCT HYDROLASE, MCP HYDROLASE, 2-HYDROXY-6-OXO-6-PHENYLHEXA-2, 4-DIENOATE HYDROLASE, HYDROLASE
2ogz:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF DPP-IV COMPLEXED WITH LILLY ARYL KETONE INHIBITOR | DIPEPTIDYL PEPTIDASE IV, CD26, DPIV, DPP-IV, DPP4, SERINE PROTEASE, INHIBITOR, HYDROLASE
2ogz:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF DPP-IV COMPLEXED WITH LILLY ARYL KETONE INHIBITOR | DIPEPTIDYL PEPTIDASE IV, CD26, DPIV, DPP-IV, DPP4, SERINE PROTEASE, INHIBITOR, HYDROLASE
3ebl:C (VAL63) to (LEU224) CRYSTAL STRUCTURE OF RICE GID1 COMPLEXED WITH GA4 | ALPHA/BETA HYDROLASE, LIPASE, GIBBERELLIN SIGNALING PATHWAY, HYDROLASE, NUCLEUS, RECEPTOR, HYDROLASE RECEPTOR
3ebl:F (VAL63) to (LEU224) CRYSTAL STRUCTURE OF RICE GID1 COMPLEXED WITH GA4 | ALPHA/BETA HYDROLASE, LIPASE, GIBBERELLIN SIGNALING PATHWAY, HYDROLASE, NUCLEUS, RECEPTOR, HYDROLASE RECEPTOR
1ni4:D (VAL178) to (THR296) HUMAN PYRUVATE DEHYDROGENASE | THIAMIN PYROPHOSPHATE, PYRUVATE, ALPHA-KETO ACID DEHYDROGENASE, PYRUVATE DEHYDROGENASE, OXIDOREDUCTASE
4wjl:A (LYS532) to (VAL674) STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE 10 (DPPY): A MODULATOR OF NEURONAL KV4 CHANNELS | INACTIVE DIPEPTIDYL PEPTIDASE 10, DPP4 STRUCTURE HOMOLOGUE, ALPHA/BETA HYDROLASE, BETA-PROPELLER, MEMBRANE PROTEIN
4wjl:B (LYS532) to (VAL674) STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE 10 (DPPY): A MODULATOR OF NEURONAL KV4 CHANNELS | INACTIVE DIPEPTIDYL PEPTIDASE 10, DPP4 STRUCTURE HOMOLOGUE, ALPHA/BETA HYDROLASE, BETA-PROPELLER, MEMBRANE PROTEIN
2onc:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-4 | DPP4 PROTEIN-INHIBITOR COMPLEX, HYDROLASE
2onc:B (PRO510) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-4 | DPP4 PROTEIN-INHIBITOR COMPLEX, HYDROLASE
2onc:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-4 | DPP4 PROTEIN-INHIBITOR COMPLEX, HYDROLASE
2onc:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-4 | DPP4 PROTEIN-INHIBITOR COMPLEX, HYDROLASE
4h0c:A (MSE1) to (THR129) CRYSTAL STRUCTURE OF PHOSPHOLIPASE/CARBOXYLESTERASE FROM DYADOBACTER FERMENTANS DSM 18053 | PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, PHOSPHOLIPASE/CARBOXYLESTERASE, HYDROLASE
2oqv:A (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV (DPP4) WITH PIPERIDINE- CONSTRAINED PHENETHYLAMINE | SERINE-PEPTIDASE, INHIBITOR, HYDROLASE
2oqv:B (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV (DPP4) WITH PIPERIDINE- CONSTRAINED PHENETHYLAMINE | SERINE-PEPTIDASE, INHIBITOR, HYDROLASE
3eio:A (SER511) to (VAL653) CRYSTAL STRUCTURE ANALYSIS OF DPPIV INHIBITOR | PROTEIN-INHIBITOR COMPLEX, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
3eio:B (SER511) to (VAL653) CRYSTAL STRUCTURE ANALYSIS OF DPPIV INHIBITOR | PROTEIN-INHIBITOR COMPLEX, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
2oxe:A (GLY26) to (LEU194) STRUCTURE OF THE HUMAN PANCREATIC LIPASE-RELATED PROTEIN 2 | GLYCOPROTEIN, HYDROLASE, LIPID DEGRADATION, PANCREATIC LIPASE, STRUCTURAL GENOMICS CONSORTIUM, SGC
1nu8:A (SER511) to (ALA654) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPP-IV) IN COMPLEX WITH DIPROTIN A (IPI) | B-BARREL, ALPHA/BETA HYDROLASE FOLD, EXOPEPTIDASE, DIPROTIN A, HYDROLASE
1nu8:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPP-IV) IN COMPLEX WITH DIPROTIN A (IPI) | B-BARREL, ALPHA/BETA HYDROLASE FOLD, EXOPEPTIDASE, DIPROTIN A, HYDROLASE
2ozl:D (GLY177) to (THR296) HUMAN PYRUVATE DEHYDROGENASE S264E VARIANT | PYRUVATE_DEHYDROGENASE_COMPLEX; HUMAN; E1; MULTIENZYME_COMPLEX_COMPONENT; THIAMINE_PYROPHOSPHATE; THIAMIN_DIPHOSPHATE; HETEROTETRAMERIC; LIPOYL_SUBSTRATE; PYRUVATE; DIHYDROLIPOAMIDE_ACETYLTRANSFERASE; DIHYDROLIPOAMIDE_DEHYDROGENASE;, OXIDOREDUCTASE
2bgn:D (SER511) to (VAL653) HIV-1 TAT PROTEIN DERIVED N-TERMINAL NONAPEPTIDE TRP2-TAT (1-9) BOUND TO THE ACTIVE SITE OF DIPEPTIDYL PEPTIDASE IV (CD26) | HYDROLASE, HYDROLASE/COMPLEX, DIPETIDYL PEPTIDASE IV, DPPIV, CD26, ALPHA/BETA-HYDROLASE FOLD, BETA-PROPELLER FOLD, PROTEIN-PROTEIN COMPLEX, ADENOSINE DEAMINASE, ADA, SERINE PROTEASE, AMINOPEPTIDASE, HIV-1 TAT PROTEIN
2bgr:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HIV-1 TAT DERIVED NONAPEPTIDES TAT(1-9) BOUND TO THE ACTIVE SITE OF DIPEPTIDYL PEPTIDASE IV (CD26) | HYDROLASE, HYDROLASE/COMPLEX, DPPIV, ALPHA/BETA-HYDROLASE FOLD, BETA-PROPELLER FOLD
2bgr:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HIV-1 TAT DERIVED NONAPEPTIDES TAT(1-9) BOUND TO THE ACTIVE SITE OF DIPEPTIDYL PEPTIDASE IV (CD26) | HYDROLASE, HYDROLASE/COMPLEX, DPPIV, ALPHA/BETA-HYDROLASE FOLD, BETA-PROPELLER FOLD
3exg:F (GLY177) to (THR296) CRYSTAL STRUCTURE OF THE PYRUVATE DEHYDROGENASE (E1P) COMPONENT OF HUMAN PYRUVATE DEHYDROGENASE COMPLEX | HETEROTETRAMER; THIAMINE DIPHOSPHATE-DEPENDENT ENZYME; DISEASE MUTATION; GLYCOLYSIS; LEIGH SYNDROME; MITOCHONDRION; OXIDOREDUCTASE; PHOSPHOPROTEIN; ALTERNATIVE SPLICING; POLYMORPHISM; PYRUVATE; THIAMINE PYROPHOSPHATE; TRANSIT PEPTIDE, OXIDOREDUCTASE
3exg:L (GLY177) to (THR296) CRYSTAL STRUCTURE OF THE PYRUVATE DEHYDROGENASE (E1P) COMPONENT OF HUMAN PYRUVATE DEHYDROGENASE COMPLEX | HETEROTETRAMER; THIAMINE DIPHOSPHATE-DEPENDENT ENZYME; DISEASE MUTATION; GLYCOLYSIS; LEIGH SYNDROME; MITOCHONDRION; OXIDOREDUCTASE; PHOSPHOPROTEIN; ALTERNATIVE SPLICING; POLYMORPHISM; PYRUVATE; THIAMINE PYROPHOSPHATE; TRANSIT PEPTIDE, OXIDOREDUCTASE
3exg:2 (VAL178) to (THR296) CRYSTAL STRUCTURE OF THE PYRUVATE DEHYDROGENASE (E1P) COMPONENT OF HUMAN PYRUVATE DEHYDROGENASE COMPLEX | HETEROTETRAMER; THIAMINE DIPHOSPHATE-DEPENDENT ENZYME; DISEASE MUTATION; GLYCOLYSIS; LEIGH SYNDROME; MITOCHONDRION; OXIDOREDUCTASE; PHOSPHOPROTEIN; ALTERNATIVE SPLICING; POLYMORPHISM; PYRUVATE; THIAMINE PYROPHOSPHATE; TRANSIT PEPTIDE, OXIDOREDUCTASE
3s2z:A (GLY0) to (ALA130) CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536 S106A MUTANT IN COMPLEX WITH CAFFEIC ACID | ALPHA/BETA HYDROLASE FOLD, ESTERASE, HYDROLASE, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES
3s2z:B (GLY0) to (ALA130) CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536 S106A MUTANT IN COMPLEX WITH CAFFEIC ACID | ALPHA/BETA HYDROLASE FOLD, ESTERASE, HYDROLASE, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES
3fak:A (ASP43) to (ILE171) STRUCTURAL AND FUNCTIONAL ANALYSIS OF A HORMONE-SENSITIVE LIPASE LIKE ESTE5 FROM A METAGENOME LIBRARY | HSL, ESTE5, ESTERASE, LIPASE, HYDROLASE
2bua:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A LOW MOLECULAR WEIGHT INHIBITOR. | HYDROLASE/INHIBITOR, DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX (HYDROLASE/INHIBITOR)
2bua:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A LOW MOLECULAR WEIGHT INHIBITOR. | HYDROLASE/INHIBITOR, DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX (HYDROLASE/INHIBITOR)
2bua:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A LOW MOLECULAR WEIGHT INHIBITOR. | HYDROLASE/INHIBITOR, DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX (HYDROLASE/INHIBITOR)
2bua:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A LOW MOLECULAR WEIGHT INHIBITOR. | HYDROLASE/INHIBITOR, DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX (HYDROLASE/INHIBITOR)
2bub:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A REVERSED AMIDE INHIBITOR | HYDROLASE/INHIBITOR, COMPLEX (HYDROLASE/INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX
4hxe:B (GLU350) to (ASN489) PYROCOCCUS HORIKOSHII ACYLAMINOACYL PEPTIDASE (UNCOMPLEXED) | SELF-COMPARTMENTALIZATION, BETA-PROPELLER, ALPHA/BETA HYRDOLASE FOLD, HYDROLASE
4hxf:B (GLU350) to (ASN489) ACYLAMINOACYL PEPTIDASE IN COMPLEX WITH Z-GLY-GLY-PHE-CHLOROMETHYL KETONE | SELF-COMPARTMENTALIZATION, BETA-PROPELLER, ALPHA/BETA HYRDOLASE FOLD, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4hxg:A (GLU350) to (ASN489) PYROCOCCUS HORIKOSHII ACYLAMINOACYL PEPTIDASE (ORTHORHOMBIC CRYSTAL FORM) | SELF-COMPARTMENTALIZATION, BETA-PROPELLER, ALPHA/BETA HYRDOLASE FOLD, HYDROLASE
4hxg:B (GLU350) to (ASN489) PYROCOCCUS HORIKOSHII ACYLAMINOACYL PEPTIDASE (ORTHORHOMBIC CRYSTAL FORM) | SELF-COMPARTMENTALIZATION, BETA-PROPELLER, ALPHA/BETA HYRDOLASE FOLD, HYDROLASE
4hxg:G (GLU350) to (ASN489) PYROCOCCUS HORIKOSHII ACYLAMINOACYL PEPTIDASE (ORTHORHOMBIC CRYSTAL FORM) | SELF-COMPARTMENTALIZATION, BETA-PROPELLER, ALPHA/BETA HYRDOLASE FOLD, HYDROLASE
4hxg:H (PHE354) to (ASN489) PYROCOCCUS HORIKOSHII ACYLAMINOACYL PEPTIDASE (ORTHORHOMBIC CRYSTAL FORM) | SELF-COMPARTMENTALIZATION, BETA-PROPELLER, ALPHA/BETA HYRDOLASE FOLD, HYDROLASE
4hxg:J (GLU350) to (ASN489) PYROCOCCUS HORIKOSHII ACYLAMINOACYL PEPTIDASE (ORTHORHOMBIC CRYSTAL FORM) | SELF-COMPARTMENTALIZATION, BETA-PROPELLER, ALPHA/BETA HYRDOLASE FOLD, HYDROLASE
4i19:A (TYR65) to (ASN197) THE CRYSTAL STRUCTURE OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS. | STRUCTURAL GENOMICS, PSI-BIOLOGY, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESI, NATPRO, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, HYDROLASE
2pu5:A (SER10) to (MET135) CRYSTAL STRUCTURE OF A C-C BOND HYDROLASE, BPHD, FROM BURKHOLDERIA XENOVORANS LB400 | C-C BOND HYDROLASE, HYDROLASE
2pu5:B (GLY19) to (GLY136) CRYSTAL STRUCTURE OF A C-C BOND HYDROLASE, BPHD, FROM BURKHOLDERIA XENOVORANS LB400 | C-C BOND HYDROLASE, HYDROLASE
2puh:A (GLY19) to (MET135) CRYSTAL STRUCTURE OF THE S112A MUTANT OF A C-C HYDROLASE, BPHD FROM BURKHOLDERIA XENOVORANS LB400, IN COMPLEX WITH ITS SUBSTRATE HOPDA | C-C BOND HYDROLASE, HYDROLASE
1orv:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) | SERINE PROTEASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, HYDROLASE
1orv:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) | SERINE PROTEASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, HYDROLASE
2q0x:A (HIS16) to (GLY142) ALPHA/BETA HYDROLASE FOLD PROTEIN OF UNKNOWN FUNCTION | ALPHA/BETA HYDROLASE FOLD, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA CONSORTIUM, SGPP, PSI, PROTEIN STRUCTURE INITIATIVE, UNKNOWN FUNCTION
2q0x:B (HIS16) to (GLY142) ALPHA/BETA HYDROLASE FOLD PROTEIN OF UNKNOWN FUNCTION | ALPHA/BETA HYDROLASE FOLD, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA CONSORTIUM, SGPP, PSI, PROTEIN STRUCTURE INITIATIVE, UNKNOWN FUNCTION
3fvr:A (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvr:B (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvr:C (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvr:D (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvr:E (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvr:F (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvr:G (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvr:H (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvr:I (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvr:L (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvr:M (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvr:N (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM I | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3sww:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH SA-(+)-3- (AMINOMETHYL)-4-(2,4-DICHLOROPHENYL)-6-(2-METHOXYPHENYL)- 2-METHYL- 5H-PYRROLO[3,4-B]PYRIDIN-7(6H)-ONE | EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3sww:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH SA-(+)-3- (AMINOMETHYL)-4-(2,4-DICHLOROPHENYL)-6-(2-METHOXYPHENYL)- 2-METHYL- 5H-PYRROLO[3,4-B]PYRIDIN-7(6H)-ONE | EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0b:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH TAK-322 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0b:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH TAK-322 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0b:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH TAK-322 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0b:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH TAK-322 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3sx4:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH SA-(+)-3- (AMINOMETHYL)-4-(2,4-DICHLOROPHENYL)-6-(2-METHOXYPHENYL)- 2-METHYL- 5H-PYRROLO[3,4-B]PYRIDIN-7(6H)-ONE | EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3sx4:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH SA-(+)-3- (AMINOMETHYL)-4-(2,4-DICHLOROPHENYL)-6-(2-METHOXYPHENYL)- 2-METHYL- 5H-PYRROLO[3,4-B]PYRIDIN-7(6H)-ONE | EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0d:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 2 | DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0d:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 2 | DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0d:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 2 | DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0d:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 2 | DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0g:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINONE INHIBITOR 3 | DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0g:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINONE INHIBITOR 3 | DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0g:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINONE INHIBITOR 3 | DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0g:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINONE INHIBITOR 3 | DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2qky:A (SER511) to (VAL653) COMPLEX STRUCTURE OF DIPEPTIDYL PEPTIDASE IV AND A OXADIAZOLYL KETONE | BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
2qky:C (SER511) to (VAL653) COMPLEX STRUCTURE OF DIPEPTIDYL PEPTIDASE IV AND A OXADIAZOLYL KETONE | BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
2qky:D (SER511) to (VAL653) COMPLEX STRUCTURE OF DIPEPTIDYL PEPTIDASE IV AND A OXADIAZOLYL KETONE | BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
3g9u:A (ASP43) to (ILE171) CRYSTAL STRUCTURE OF ESTE5, WAS SOAKED BY P-NITROPHENYL BUTYRATE FOR 5MIN | HSL, ESTE5, ESTERASE, LIPASE, HYDROLASE
2qoe:A (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A TRIAZOLOPIPERAZINE- BASED BETA AMINO ACID INHIBITOR | ALPHA/BETA INHIBITORS, BETA-PROPELLER,DIMER, DIABETES, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
2qoe:B (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A TRIAZOLOPIPERAZINE- BASED BETA AMINO ACID INHIBITOR | ALPHA/BETA INHIBITORS, BETA-PROPELLER,DIMER, DIABETES, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
2qr5:A (GLY332) to (ALA469) AEROPYRUM PERNIX ACYLAMINOACYL PEPTIDASE, H367A MUTANT | ACYLAMINOACYL PEPTIDASE, THERMOPHILIC ENZYME, OXYANION BINDING SITE, CATALYTIC ACTIVITY, HYDROLASE
2qr5:B (GLY332) to (ALA469) AEROPYRUM PERNIX ACYLAMINOACYL PEPTIDASE, H367A MUTANT | ACYLAMINOACYL PEPTIDASE, THERMOPHILIC ENZYME, OXYANION BINDING SITE, CATALYTIC ACTIVITY, HYDROLASE
2qru:A (ASN5) to (PHE128) CRYSTAL STRUCTURE OF AN ALPHA/BETA HYDROLASE SUPERFAMILY PROTEIN FROM ENTEROCOCCUS FAECALIS | ENTEROCOCCUS FAECALIS, ALPHA/BETA-HYDROLASE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, UNKNOWN FUNCTION
2qt9:A (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A 4-ARYL CYCLOHEXYLALANINE INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE
2qt9:B (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A 4-ARYL CYCLOHEXYLALANINE INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE
2qtb:A (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A 4-ARYL CYCLOHEXYLALANINE INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE
2qtb:B (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A 4-ARYL CYCLOHEXYLALANINE INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE
2qzp:A (VAL336) to (ALA469) CRYSTAL STRUCTURE OF MUTATION OF AN ACYLPTIDE HYDROLASE/ESTERASE FROM AEROPYRUM PERNIX K1 | CRYSTAL STRUCTURE, TRUNCATED, ACYLPEPTIDE HYDROLASE, AEROPYRUM PERNIX K1, CYTOPLASM
2qzp:B (GLY332) to (ALA469) CRYSTAL STRUCTURE OF MUTATION OF AN ACYLPTIDE HYDROLASE/ESTERASE FROM AEROPYRUM PERNIX K1 | CRYSTAL STRUCTURE, TRUNCATED, ACYLPEPTIDE HYDROLASE, AEROPYRUM PERNIX K1, CYTOPLASM
2d5l:A (GLU480) to (GLY627) CRYSTAL STRUCTURE OF PROLYL TRIPEPTIDYL AMINOPEPTIDASE FROM PORPHYROMONAS GINGIVALIS | PEPTIDASE FAMILY S9, SERINE PEPTIDASE, PROLYL OLIGOPEPTIDASE FAMILY, HYDROLASE
4j3j:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF DPP-IV WITH COMPOUND C3 | INHIBITOR COMPLEX, SERINE EXOPEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2dcm:A (GLU480) to (GLY627) THE CRYSTAL STRUCTURE OF S603A MUTATED PROLYL TRIPEPTIDYL AMINOPEPTIDASE COMPLEXED WITH SUBSTRATE | PEPTIDASE FAMILY S9, SERINE PEPTIDASE, PROLYL OLIGOPEPTIDASE FAMILY, SITE-DIRECTED MUTANGENESIS, HYDROLASE
4y9s:A (LYS3) to (LEU128) STRUCTURE OF AN H300N MUTANT OF POTATO EPOXIDE HYDROLASE, STEH1 | MUTATION OF CATALYTIC RESIDUE, HYDROLASE
2dst:A (ARG3) to (GLU108) CRYSTAL STRUCTURE ANALYSIS OF TT1977 | CONSERVED HYPOTHETICAL PROTEIN, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, UNKNOWN FUNCTION
4jh0:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL-PEPTIDASE 4 (CD26, ADENOSINE DEAMINASE COMPLEXING PROTEIN 2) (DPP-IV-WT) COMPLEX WITH BMS-767778 AKA 2-(3- (AMINOMETHYL)-4-(2,4- DICHLOROPHENYL)-2-METHYL-5-OXO-5,7-DIHYDRO-6H- PYRROLO[3,4- B]PYRIDIN-6-YL)-N,N-DIMETHYLACETAMIDE | EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP-IV, DIMER, HYDROLASE
4jh0:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL-PEPTIDASE 4 (CD26, ADENOSINE DEAMINASE COMPLEXING PROTEIN 2) (DPP-IV-WT) COMPLEX WITH BMS-767778 AKA 2-(3- (AMINOMETHYL)-4-(2,4- DICHLOROPHENYL)-2-METHYL-5-OXO-5,7-DIHYDRO-6H- PYRROLO[3,4- B]PYRIDIN-6-YL)-N,N-DIMETHYLACETAMIDE | EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP-IV, DIMER, HYDROLASE
3h04:A (ILE4) to (TYR126) THE CRYSTAL STRUCTURE OF THE PROTEIN WITH UNKNOWN FUNCTION FROM STAPHYLOCOCCUS AUREUS SUBSP. AUREUS MU50 | PROTEIN WITH UNKNOWN FUNCTION, STRUCTURAL GENOMICS, MCSG, PSI, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, UNKNOWN FUNCTION
3h0c:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A REVERSED AMIDE INHIBITOR | COMPLEX (HYDROLASE-INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, CELL MEMBRANE, DISULFIDE BOND, MEMBRANE, SECRETED
3h0c:B (SER511) to (ALA654) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A REVERSED AMIDE INHIBITOR | COMPLEX (HYDROLASE-INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, CELL MEMBRANE, DISULFIDE BOND, MEMBRANE, SECRETED
2rgu:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF COMPLEX OF HUMAN DPP4 AND INHIBITOR | PEPTIDASE, INHIBITOR, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
2rgu:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF COMPLEX OF HUMAN DPP4 AND INHIBITOR | PEPTIDASE, INHIBITOR, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
2rip:A (SER511) to (VAL653) STRUCTURE OF DPPIV IN COMPLEX WITH AN INHIBITOR | DPPIV, DIABETES, DRUG DESIGN, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE
3h19:A (ASP43) to (ILE171) CRYSTAL STRUCTURE OF ESTE5, WAS SOAKED BY METHYL ALCOHOL | HSL, ESTE5, ESTERASE, LIPASE, HYDROLASE
1evq:A (ALA46) to (TYR183) THE CRYSTAL STRUCTURE OF THE THERMOPHILIC CARBOXYLESTERASE EST2 FROM ALICYCLOBACILLUS ACIDOCALDARIUS | ALPHA/BETA HYDROLASE FOLD
1qtr:A (TYR14) to (GLY137) CRYSTAL STRUCTURE ANALYSIS OF THE PROLYL AMINOPEPTIDASE FROM SERRATIA MARCESCENS | ALPHA BETA HYDROLASE FOLD, PROLINE, PROLYL AMINOPEPTIDASE, SERRATIA, IMINOPEPTIDASE
1qz3:A (ALA46) to (TYR183) CRYSTAL STRUCTURE OF MUTANT M211S/R215L OF CARBOXYLESTERASE EST2 COMPLEXED WITH HEXADECANESULFONATE | ALPHA/BETA HYDROLASE FOLD, HYDROLASE
2ecf:A (PRO486) to (ALA634) CRYSTAL STRUCTURE OF DIPEPTIDYL AMINOPEPTIDASE IV FROM STENOTROPHOMONAS MALTOPHILIA | PROLYL OLIGOPEPTIDASE FAMILY, PEPTIDASE FAMILY S9, DIPEPTIDYL PEPTIDASE IV, HYDROLASE
2eep:A (GLU480) to (GLY626) PROLYL TRIPEPTIDYL AMINOPEPTIDASE COMPLEXED WITH AN INHIBITOR | PEPTIDASE FAMILY S9, PROLYL OLIGOPEPTIDASE FAMILY, SERINE PEPTIDASE, INHIBITOR COMPLEX, HYDROLASE
3hea:B (SER1) to (GLY119) THE L29P/L124I MUTATION OF PSEUDOMONAS FLUORESCENS ESTERASE | ALPHA/BETA HYDROLASE, ESTERASE, COVALENT ADDUCT, TETRAHEDRAL INTERMEDIATE, HYDROLASE, OXIDOREDUCTASE, PEROXIDASE
3hea:C (SER1) to (GLY119) THE L29P/L124I MUTATION OF PSEUDOMONAS FLUORESCENS ESTERASE | ALPHA/BETA HYDROLASE, ESTERASE, COVALENT ADDUCT, TETRAHEDRAL INTERMEDIATE, HYDROLASE, OXIDOREDUCTASE, PEROXIDASE
1r9m:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV AT 2.1 ANG. RESOLUTION. | AMINOPEPTIDASE, SERINE PROTEASE, GLYCOPROTEIN, HYDROLASE
1r9m:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV AT 2.1 ANG. RESOLUTION. | AMINOPEPTIDASE, SERINE PROTEASE, GLYCOPROTEIN, HYDROLASE
1r9m:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV AT 2.1 ANG. RESOLUTION. | AMINOPEPTIDASE, SERINE PROTEASE, GLYCOPROTEIN, HYDROLASE
1r9m:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV AT 2.1 ANG. RESOLUTION. | AMINOPEPTIDASE, SERINE PROTEASE, GLYCOPROTEIN, HYDROLASE
2fjp:A (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH AN INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, HYDROLASE
2fjp:B (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH AN INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, HYDROLASE
4z8z:A (LYS63) to (ASN210) CRYSTAL STRUCTURE OF THE HYPOTHETICAL PROTEIN FROM RUMINICLOSTRIDIUM THERMOCELLUM ATCC 27405 | STRUCTURAL GENOMICS, HUMAN MICROBIOME, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, PSI-BIOLOGY
3v1k:A (GLY19) to (MET135) CRYSTAL STRUCTURE OF THE H265Q MUTANT OF A C-C HYDROLASE, BPHD FROM BURKHOLDERIA XENOVORANS LB400. | C-C BOND HYDROLASE, ALPHA/BETA HYDROLASE FOLD, BPHD, ALPHA/BETA HYDROLASE, PCB DEGRADATION, META CLEAVAGE PRODUCT HYDROLASE, MCP HYDROLASE, 2-HYDROXY-6-OXO-6-PHENYL-HEXA-2,4-DIENOATE HYDROLASE, HYDROLASE
3v1k:B (GLY19) to (MET135) CRYSTAL STRUCTURE OF THE H265Q MUTANT OF A C-C HYDROLASE, BPHD FROM BURKHOLDERIA XENOVORANS LB400. | C-C BOND HYDROLASE, ALPHA/BETA HYDROLASE FOLD, BPHD, ALPHA/BETA HYDROLASE, PCB DEGRADATION, META CLEAVAGE PRODUCT HYDROLASE, MCP HYDROLASE, 2-HYDROXY-6-OXO-6-PHENYL-HEXA-2,4-DIENOATE HYDROLASE, HYDROLASE
2fx5:A (THR24) to (ILE147) PSEUDOMONAS MENDOCINA LIPASE | ALPHA-BETA HYDROLASE
4kr0:A (SER511) to (VAL653) COMPLEX STRUCTURE OF MERS-COV SPIKE RBD BOUND TO CD26 | 8-BLADED BETA-PROPELLER DOMAIN, ALPHA/BETA HYDROLASE DOMAIN, BLADES IV AND V, CD26 BETA-PROPELLER, HYDROLASE-VIRAL PROTEIN COMPLEX
4kry:A (ALA59) to (TYR195) STRUCTURE OF AES FROM E. COLI IN COVALENT COMPLEX WITH PMS | ALPHA/BETA-HYDROLASE, HORMONE-SENSITIVE-LIPASE FAMILY, INHIBITION OF MALT, ACYL ESTERASE, PHENYLMETHYLSULFONYL-SERINE, HYDROLASE
3v9a:A (ASP43) to (ILE171) CRYSTAL STRUCTURE OF ESTERASE/LIPASE FROM UNCULTURED BACTERIUM | ESTERASE, LIPASE, HYDROLASE ACTIVATOR
2g5p:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) COMPLEXED WITH CYANOPYRROLIDINE (C5-PRO-PRO) INHIBITOR 21AC | SERINE PEPTIDASE, BETA-PROPELLER, HYDROLASE
2g5p:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) COMPLEXED WITH CYANOPYRROLIDINE (C5-PRO-PRO) INHIBITOR 21AC | SERINE PEPTIDASE, BETA-PROPELLER, HYDROLASE
2g5t:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) COMPLEXED WITH CYANOPYRROLIDINE (C5-PRO-PRO) INHIBITOR 21AG | SERINE PEPTIDASE, BETA-PROPELLER, HYDROLASE
2g63:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) COMPLEXED WITH CYANOPYRROLIDINE (C5-PRO-PRO) INHIBITOR 24B | SERINE PEPTIDASE, BETA-PROPELLER, HYDROLASE
2g63:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) COMPLEXED WITH CYANOPYRROLIDINE (C5-PRO-PRO) INHIBITOR 24B | SERINE PEPTIDASE, BETA-PROPELLER, HYDROLASE
2gbf:A (SER512) to (VAL654) RAT DPP-IV WITH ALKYNYL CYANOPYRROLIDINE #1 | SERINE PEPTIDASE BETA PROPELLER, HYDROLASE
2gbf:B (SER512) to (VAL654) RAT DPP-IV WITH ALKYNYL CYANOPYRROLIDINE #1 | SERINE PEPTIDASE BETA PROPELLER, HYDROLASE
2gbg:A (VAL508) to (VAL654) RAT DPP-IV WITH ALKYNYL CYANOPYRROLIDINE #2 | SERINE PEPTIDASE BETA PROPELLER, HYDROLASE
2gbg:B (VAL508) to (VAL654) RAT DPP-IV WITH ALKYNYL CYANOPYRROLIDINE #2 | SERINE PEPTIDASE BETA PROPELLER, HYDROLASE
2gbi:A (SER512) to (VAL654) RAT DPP-IV WITH XANTHINE INHIBITOR 4 | SERINE PEPTIDASE BETA PROPELLER, HYDROLASE
2gbi:B (SER512) to (VAL654) RAT DPP-IV WITH XANTHINE INHIBITOR 4 | SERINE PEPTIDASE BETA PROPELLER, HYDROLASE
3ia2:B (SER1) to (GLY119) PSEUDOMONAS FLUORESCENS ESTERASE COMPLEXED TO THE R-ENANTIOMER OF A SULFONATE TRANSITION STATE ANALOG | ALPHA-BETA HYDROLASE FOLD, TRANSITION STATE ANALOG, HYDROLASE, OXIDOREDUCTASE, PEROXIDASE
3ia2:D (SER1) to (GLY119) PSEUDOMONAS FLUORESCENS ESTERASE COMPLEXED TO THE R-ENANTIOMER OF A SULFONATE TRANSITION STATE ANALOG | ALPHA-BETA HYDROLASE FOLD, TRANSITION STATE ANALOG, HYDROLASE, OXIDOREDUCTASE, PEROXIDASE
3ia2:E (SER1) to (GLY119) PSEUDOMONAS FLUORESCENS ESTERASE COMPLEXED TO THE R-ENANTIOMER OF A SULFONATE TRANSITION STATE ANALOG | ALPHA-BETA HYDROLASE FOLD, TRANSITION STATE ANALOG, HYDROLASE, OXIDOREDUCTASE, PEROXIDASE
3ib3:B (GLY44) to (TRP192) CRYSTAL STRUCTURE OF SACOL2612 - COCE/NOND FAMILY HYDROLASE FROM STAPHYLOCOCCUS AUREUS | STRUCTURAL GENOMICS, HYDROLASE, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID
3vjk:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DEPIPTIDYL PEPTIDASE IV (DPP-4) IN COMPLEX WITH MP-513 | ALPHA/BETA, BETA-PROPELLER, AMINOPEPTIDASE, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, DIABETES, GLYCOPROTEIN, CELL MEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3vjl:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DEPIPTIDYL PEPTIDASE IV (DPP-4) IN COMPLEX WITH A PROLYLTHIAZOLIDINE INHIBITOR #2 | ALPHA/BETA, BETA-PROPELLER, AMINOPEPTIDASE, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, DIABETES, GLYCOPROTEIN, CELL MEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3vjm:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DEPIPTIDYL PEPTIDASE IV (DPP-4) IN COMPLEX WITH A PROLYLTHIAZOLIDINE INHIBITOR #1 | ALPHA/BETA, BETA-PROPELLER, AMINOPEPTIDASE, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, DIABETES, GLYCOPROTEIN, CELL MEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3vjm:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DEPIPTIDYL PEPTIDASE IV (DPP-4) IN COMPLEX WITH A PROLYLTHIAZOLIDINE INHIBITOR #1 | ALPHA/BETA, BETA-PROPELLER, AMINOPEPTIDASE, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, DIABETES, GLYCOPROTEIN, CELL MEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4l72:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF MERS-COV COMPLEXED WITH HUMAN DPP4 | ALPHA/BETA HYDROLASE BETA-PROPELLER, GLYCOLATION, VIRUS RECEPTOR- BINDING DOMAIN, HYDROLASE-VIRAL PROTEIN COMPLEX
4l9a:A (ALA3) to (LEU124) CRYSTAL STRUCTURE OF SMU.1393C FROM CARIOGENIC PATHOGEN STREPTOCOCCUS MUTANS | ALPHA/BETA HYDROLASE, CARBOXYLESTERASE, HYDROLASE
4l9a:B (ALA3) to (LEU124) CRYSTAL STRUCTURE OF SMU.1393C FROM CARIOGENIC PATHOGEN STREPTOCOCCUS MUTANS | ALPHA/BETA HYDROLASE, CARBOXYLESTERASE, HYDROLASE
1hde:A (PRO22) to (MET147) HALOALKANE DEHALOGENASE MUTANT WITH PHE 172 REPLACED WITH TRP | DEHALOGENASE, HYDROLASE, DETOXIFICATION
1hde:B (PRO22) to (MET147) HALOALKANE DEHALOGENASE MUTANT WITH PHE 172 REPLACED WITH TRP | DEHALOGENASE, HYDROLASE, DETOXIFICATION
4zwn:A (LEU15) to (SER148) CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF THE MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE | MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, SERINE HYDROLASE, ALPHA/BETA HYDROLASE, HYDROLASE
4zwn:B (GLU14) to (SER148) CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF THE MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE | MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, SERINE HYDROLASE, ALPHA/BETA HYDROLASE, HYDROLASE
4zwn:C (GLU14) to (SER148) CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF THE MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE | MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, SERINE HYDROLASE, ALPHA/BETA HYDROLASE, HYDROLASE
4zwn:D (GLN16) to (SER148) CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF THE MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE | MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, SERINE HYDROLASE, ALPHA/BETA HYDROLASE, HYDROLASE
4lko:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH BMS-744891 | EXOPEPTIDASE, BETA BARREL, ALPHA/BETA HYDROLASE FOLD, HYDROLASE
2hm7:A (ALA46) to (ILE182) CRYSTAL STRUCTURE ANALYSIS OF THE G84S EST2 MUTANT | ALPHA/BETA HYDROLASE FOLD, HYDROLASE
2wj6:A (LEU6) to (MET125) CRYSTAL STRUCTURE OF THE COFACTOR-DEVOID 1-H-3-HYDROXY-4- OXOQUINALDINE 2,4-DIOXYGENASE (HOD) FROM ARTHROBACTER NITROGUAJACOLICUS RU61A COMPLEXED WITH ITS NATURAL PRODUCT N-ACETYLANTHRANILATE | OXIDOREDUCTASE, ALPHA/BETA HYDROLASE
1u2e:A (SER8) to (GLY134) CRYSTAL STRUCTURE OF THE C-C BOND HYDROLASE MHPC | ALPHA/BETA HYDROLASE FOLD
1u2e:B (SER1008) to (GLY1134) CRYSTAL STRUCTURE OF THE C-C BOND HYDROLASE MHPC | ALPHA/BETA HYDROLASE FOLD
1u4n:A (ALA46) to (ILE182) CRYSTAL STRUCTURE ANALYSIS OF THE M211S/R215L EST2 MUTANT | ALPHA/BETA HYDROLASE FOLD, HYDROLASE
2hu5:A (VAL336) to (ALA469) BINDING OF INHIBITORS BY ACYLAMINOACYL-PEPTIDASE | ALPHA/BETA HYDROLASE, BETA-PROPELLER, ENZYME-INHIBITOR COMPLEX, HYDROLASE
2hu5:B (GLY332) to (ALA469) BINDING OF INHIBITORS BY ACYLAMINOACYL-PEPTIDASE | ALPHA/BETA HYDROLASE, BETA-PROPELLER, ENZYME-INHIBITOR COMPLEX, HYDROLASE
2hu7:A (VAL336) to (ALA469) BINDING OF INHIBITORS BY ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE, BETA-PROPELLER, ENZYME-INHIBITOR COMPLEX, HYDROLASE
2hu8:A (VAL336) to (ALA469) BINDING OF INHIBITORS BY ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE, BETA-PROPELLER, ENZYME-INHIBITOR COMPLEX, HYDROLASE
2hu8:B (VAL336) to (ALA469) BINDING OF INHIBITORS BY ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE, BETA-PROPELLER, ENZYME-INHIBITOR COMPLEX, HYDROLASE
3w2t:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DEPIPTIDYL PEPTIDASE IV (DPP-4) IN COMPLEX WITH VILDAGLIPTIN | ALPHA/BETA, BETA-PROPELLER, HYDROLASE, AMINOPEPTIDASE, SERINE PROTEASE, SECRETED, SIGNAL-ANCHOR, TRANSMEMBRANE, DIABETES, GLYCOPROTEIN, CELL MEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3w2t:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DEPIPTIDYL PEPTIDASE IV (DPP-4) IN COMPLEX WITH VILDAGLIPTIN | ALPHA/BETA, BETA-PROPELLER, HYDROLASE, AMINOPEPTIDASE, SERINE PROTEASE, SECRETED, SIGNAL-ANCHOR, TRANSMEMBRANE, DIABETES, GLYCOPROTEIN, CELL MEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1u8e:A (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 MUTANT Y547F | ALPHA/BETA HYDROLASE, BETA-PROPELLER, HOMODIMER, HYDROLASE
1u8e:B (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 MUTANT Y547F | ALPHA/BETA HYDROLASE, BETA-PROPELLER, HOMODIMER, HYDROLASE
2wtm:B (GLY-1) to (SER129) EST1E FROM BUTYRIVIBRIO PROTEOCLASTICUS | ESTERASE, HYDROLASE, FERULIC ACID ESTERASE
2wtm:D (GLY-1) to (SER129) EST1E FROM BUTYRIVIBRIO PROTEOCLASTICUS | ESTERASE, HYDROLASE, FERULIC ACID ESTERASE
1ufo:B (ARG2) to (ILE136) CRYSTAL STRUCTURE OF TT1662 FROM THERMUS THERMOPHILUS | ALPHA-BETA FOLD, HYDROLASE, STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
1ufo:C (MSE1) to (ILE136) CRYSTAL STRUCTURE OF TT1662 FROM THERMUS THERMOPHILUS | ALPHA-BETA FOLD, HYDROLASE, STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
1ufo:E (MSE1) to (ILE136) CRYSTAL STRUCTURE OF TT1662 FROM THERMUS THERMOPHILUS | ALPHA-BETA FOLD, HYDROLASE, STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
2i3d:A (PRO2) to (ILE130) CRYSTAL STRUCTURE OF PROTEIN OF UNKNOWN FUNCTION ATU1826, A PUTATIVE ALPHA/BETA HYDROLASE FROM AGROBACTERIUM TUMEFACIENS | STRUCTURAL GENOMICS, APC5865, HYDROLASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, UNKNOWN FUNCTION
2i3d:B (GLU3) to (ILE130) CRYSTAL STRUCTURE OF PROTEIN OF UNKNOWN FUNCTION ATU1826, A PUTATIVE ALPHA/BETA HYDROLASE FROM AGROBACTERIUM TUMEFACIENS | STRUCTURAL GENOMICS, APC5865, HYDROLASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, UNKNOWN FUNCTION
2i3z:A (SER512) to (VAL654) RAT DPP-IV WITH XANTHINE MIMETIC INHIBITOR #7 | ENZYME, PEPTIDASE, INHIBITOR, HYDROLASE
2i3z:B (SER512) to (VAL654) RAT DPP-IV WITH XANTHINE MIMETIC INHIBITOR #7 | ENZYME, PEPTIDASE, INHIBITOR, HYDROLASE
1ik6:A (GLU186) to (ALA294) 3D STRUCTURE OF THE E1BETA SUBUNIT OF PYRUVATE DEHYDROGENASE FROM THE ARCHEON PYROBACULUM AEROPHILUM | E1BETA, PYRUVATE DEHYDROGENASE, TETRAMER, GXXXG, OXIDOREDUCTASE
2i78:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPP IV) COMPLEXED WITH ABT-341, A CYCLOHEXENE-CONSTRAINED PHENETHYLAMINE INHIBITOR | SERINE PEPTIDASE,, HYDROLASE
2i78:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPP IV) COMPLEXED WITH ABT-341, A CYCLOHEXENE-CONSTRAINED PHENETHYLAMINE INHIBITOR | SERINE PEPTIDASE,, HYDROLASE
2i78:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPP IV) COMPLEXED WITH ABT-341, A CYCLOHEXENE-CONSTRAINED PHENETHYLAMINE INHIBITOR | SERINE PEPTIDASE,, HYDROLASE
1j2e:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE IV, CD26, PROLYL OLIGOPEPTIDASE, BETA-PROPELLER STRUCTURE, HYDROLASE
1j2e:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE IV, CD26, PROLYL OLIGOPEPTIDASE, BETA-PROPELLER STRUCTURE, HYDROLASE
2iu4:A (GLN24) to (ASP132) DIHYDROXYACETONE KINASE OPERON CO-ACTIVATOR DHA-DHAQ | TRANSFERASE, LACTOCOCCUS LACTIS, DIHYDROXYACETONE, CO-ACTIVATOR, KINASE
2iu4:B (GLN24) to (ASP133) DIHYDROXYACETONE KINASE OPERON CO-ACTIVATOR DHA-DHAQ | TRANSFERASE, LACTOCOCCUS LACTIS, DIHYDROXYACETONE, CO-ACTIVATOR, KINASE
2iu6:A (GLN24) to (ASP133) REGULATION OF THE DHA OPERON OF LACTOCOCCUS LACTIS | KINASE, DIHYDROXYACETONE KINASE TRANSFERASE, TRANSFERASE
2iu6:B (GLN24) to (ASP133) REGULATION OF THE DHA OPERON OF LACTOCOCCUS LACTIS | KINASE, DIHYDROXYACETONE KINASE TRANSFERASE, TRANSFERASE
1va4:A (SER1) to (GLY119) PSEUDOMONAS FLUORESCENS ARYL ESTERASE | ALPHA/BETA HYDROLASE, ESTERASE, NON-COFACTOR DEPENDENT HALOPEROXIDASE, HYDROLASE
1va4:C (SER1) to (GLY119) PSEUDOMONAS FLUORESCENS ARYL ESTERASE | ALPHA/BETA HYDROLASE, ESTERASE, NON-COFACTOR DEPENDENT HALOPEROXIDASE, HYDROLASE
1va4:E (SER1) to (GLY119) PSEUDOMONAS FLUORESCENS ARYL ESTERASE | ALPHA/BETA HYDROLASE, ESTERASE, NON-COFACTOR DEPENDENT HALOPEROXIDASE, HYDROLASE
1jfr:A (SER26) to (THR154) CRYSTAL STRUCTURE OF THE STREPTOMYCES EXFOLIATUS LIPASE AT 1.9A RESOLUTION: A MODEL FOR A FAMILY OF PLATELET- ACTIVATING FACTOR ACETYLHYDROLASES | SERINE HYDROLASE, LIPASE
1jfr:B (SER26) to (THR154) CRYSTAL STRUCTURE OF THE STREPTOMYCES EXFOLIATUS LIPASE AT 1.9A RESOLUTION: A MODEL FOR A FAMILY OF PLATELET- ACTIVATING FACTOR ACETYLHYDROLASES | SERINE HYDROLASE, LIPASE
1ve6:A (VAL336) to (ALA469) CRYSTAL STRUCTURE OF AN ACYLPEPTIDE HYDROLASE/ESTERASE FROM AEROPYRUM PERNIX K1 | BETA PROPELLER DOMAIN, ALPHA/BETA HYDROLASE DOMAIN, HYDROLASE
1ve6:B (GLY332) to (ALA469) CRYSTAL STRUCTURE OF AN ACYLPEPTIDE HYDROLASE/ESTERASE FROM AEROPYRUM PERNIX K1 | BETA PROPELLER DOMAIN, ALPHA/BETA HYDROLASE DOMAIN, HYDROLASE
1ve7:A (VAL336) to (ALA469) CRYSTAL STRUCTURE OF AN ACYLPEPTIDE HYDROLASE/ESTERASE FROM AEROPYRUM PERNIX K1 IN COMPLEX WITH P-NITROPHENYL PHOSPHATE | BETA PROPELLER DOMAIN, ALPHA/BETA HYDROLASE DOMAIN, HYDROLASE
1ve7:B (ARG334) to (ALA469) CRYSTAL STRUCTURE OF AN ACYLPEPTIDE HYDROLASE/ESTERASE FROM AEROPYRUM PERNIX K1 IN COMPLEX WITH P-NITROPHENYL PHOSPHATE | BETA PROPELLER DOMAIN, ALPHA/BETA HYDROLASE DOMAIN, HYDROLASE
3wqh:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH ANAGLIPTIN | DIABETES, BETA-PROPELLER, AMINOPEPTIDASE, MEMBRANE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3wqh:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH ANAGLIPTIN | DIABETES, BETA-PROPELLER, AMINOPEPTIDASE, MEMBRANE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1w1i:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV (DPPIV OR CD26) IN COMPLEX WITH ADENOSINE DEAMINASE | HYDROLASE, HYDROLASE/COMPLEX, DIPETIDYL PEPTIDASE IV, DPPIV, CD26, ALPHA/BETA-HYDROLASE FOLD, BETA-PROPELLER FOLD, PROTEIN-PROTEIN COMPLEX, ADENOSINE DEAMINASE, ADA, SERINE PROTEASE, AMINOPEPTIDASE
2jgd:B (ASN796) to (TYR901) E. COLI 2-OXOGLUTARATE DEHYDROGENASE (E1O) | 2-OXOGLUTARATE DEHYDROGENASE, FLAVOPROTEIN, OXIDOREDUCTASE, THIAMINE DIPHOSPHATE, THIAMINE PYROPHOSPHATE, ADENOSINE MONOPHOSPHATE, E1O, KGDH, OGDH, GLYCOLYSIS, OXALOACETATE
4n8d:A (SER511) to (VAL653) DPP4 COMPLEXED WITH SYN-7AA | HYDROLASE
4n8d:B (SER511) to (VAL653) DPP4 COMPLEXED WITH SYN-7AA | HYDROLASE
4n8e:A (SER511) to (VAL653) DPP4 COMPLEXED WITH COMPOUND 12A | HYDROLASE
4n8e:B (SER511) to (VAL653) DPP4 COMPLEXED WITH COMPOUND 12A | HYDROLASE
2jid:A (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH 1-(3,4- DIMETHOXY-PHENYL)-3-M-TOLYL-PIPERIDINE-4-YLAMINE | HYDROLASE, DIABETES TYPE II, DIPEPTIDYL PEPTIDASE, PROTEASE, MEMBRANE, B-PROPELLER, STRUCTURE BASED DESIGN, GLYCOPROTEIN, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE FOLD, AMINOPEPTIDASE, SERINE PROTEASE
3jw8:A (PRO30) to (ILE155) CRYSTAL STRUCTURE OF HUMAN MONO-GLYCERIDE LIPASE | ALPHA-BETA HYDROLASE, HYDROLASE
3jw8:B (PRO30) to (ILE155) CRYSTAL STRUCTURE OF HUMAN MONO-GLYCERIDE LIPASE | ALPHA-BETA HYDROLASE, HYDROLASE
3jwe:B (PRO30) to (ILE155) CRYSTAL STRUCTURE OF HUMAN MONO-GLYCERIDE LIPASE IN COMPLEX WITH SAR629 | ALPHA-BETA HYDROLASE, HYDROLASE
2z3z:A (GLU480) to (GLY627) PROLYL TRIPEPTIDYL AMINOPEPTIDASE MUTANT E636A COMPLEXD WITH AN INHIBITOR | PEPTIDASE FAMILY S9, PROLYL OLIGOPEPTIDASE FAMILY, SERINE PROTEASE, PROLINE-SPECIFIC PEPTIDASE, HYDROLASE
2z3w:A (GLU480) to (GLY627) PROLYL TRIPEPTIDYL AMINOPEPTIDASE MUTANT E636A | PROLYL OLIGOPEPTIDASE FAMILY, PEPTIDASE FAMILY S9, SERINE PROTEASE, PROLINE-SPECIFIC PEPTIDASE, HYDROLASE
3kwj:A (SER511) to (VAL653) STRUCUTRE OF HUMAN DPP-IV WITH (2S,3S,11BS)-3-(3-FLUOROMETHYL-PHENYL)- 9,10-DIMETHOXY-1,3,4,6,7,11B-HEXAHYDRO-2H-PYRIDO[2,1-A]ISOQUINOLIN-2- YLAMINE | DIABETES TYPE II, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
3l1h:A (ASP43) to (ILE171) CRYSTAL STRUCTURE OF ESTE5, WAS SOAKED BY FECL3 | HSL, ESTE5, ESTERASE, LIPASE, HYDROLASE
3l1i:A (ASP43) to (ILE171) CRYSTAL STRUCTURE OF ESTE5, WAS SOAKED BY CUSO4 | HSL, ESTE5, ESTERASE, LIPASE, HYDROLASE
4pnz:A (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH THE LONG-ACTING INHIBITOR OMARIGLIPTIN (MK-3102) | ALPHA/BETA, BETA-PROPELLER, DIMER, DIABETES, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4pnz:B (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH THE LONG-ACTING INHIBITOR OMARIGLIPTIN (MK-3102) | ALPHA/BETA, BETA-PROPELLER, DIMER, DIABETES, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4pv7:A (SER511) to (VAL653) COCRYSTAL STRUCTURE OF DIPEPTIDYL-PEPTIDASE 4 WITH AN INDOLE SCAFFOLD INHIBITOR | BETA-PROPELLER, HYDROLASE, EXTROCELLULAR SIDE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4pw0:A (THR13) to (GLY131) ALPHA/BETA HYDROLASE FOLD PROTEIN FROM CHITINOPHAGA PINENSIS | STRUCTURAL GENOMICS, APC103277, ALPHA/BETA HYDROLASE FOLD PROTEIN, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, HYDROLASE
4q3k:A (MET1) to (GLY136) CRYSTAL STRUCTURE OF MGS-M1, AN ALPHA/BETA HYDROLASE ENZYME FROM A MEDEE BASIN DEEP-SEA METAGENOME LIBRARY | METAGENOME, METAGENOMIC LIBRARY, ALPHA AND BETA PROTEINS, ALPHA/BETA HYDROLASE SUPERFAMILY, ESTERASE/LIPASE FOLD, HYDROLASE
4q3l:A (SER2) to (ASN121) CRYSTAL STRUCTURE OF MGS-M2, AN ALPHA/BETA HYDROLASE ENZYME FROM A MEDEE BASIN DEEP-SEA METAGENOME LIBRARY | METAGENOME, METAGENOMIC LIBRARY, ALPHA AND BETA PROTEINS, ALPHA/BETA HYDROLASE SUPERFAMILY, ESTERASE/LIPASE FOLD, HYDROLASE
4q3l:C (SER2) to (ASN121) CRYSTAL STRUCTURE OF MGS-M2, AN ALPHA/BETA HYDROLASE ENZYME FROM A MEDEE BASIN DEEP-SEA METAGENOME LIBRARY | METAGENOME, METAGENOMIC LIBRARY, ALPHA AND BETA PROTEINS, ALPHA/BETA HYDROLASE SUPERFAMILY, ESTERASE/LIPASE FOLD, HYDROLASE
4q3l:D (SER2) to (ASN121) CRYSTAL STRUCTURE OF MGS-M2, AN ALPHA/BETA HYDROLASE ENZYME FROM A MEDEE BASIN DEEP-SEA METAGENOME LIBRARY | METAGENOME, METAGENOMIC LIBRARY, ALPHA AND BETA PROTEINS, ALPHA/BETA HYDROLASE SUPERFAMILY, ESTERASE/LIPASE FOLD, HYDROLASE
4q3l:H (SER2) to (ASN121) CRYSTAL STRUCTURE OF MGS-M2, AN ALPHA/BETA HYDROLASE ENZYME FROM A MEDEE BASIN DEEP-SEA METAGENOME LIBRARY | METAGENOME, METAGENOMIC LIBRARY, ALPHA AND BETA PROTEINS, ALPHA/BETA HYDROLASE SUPERFAMILY, ESTERASE/LIPASE FOLD, HYDROLASE
4q3o:F (VAL92) to (GLY221) CRYSTAL STRUCTURE OF MGS-MT1, AN ALPHA/BETA HYDROLASE ENZYME FROM A LAKE MATAPAN DEEP-SEA METAGENOME LIBRARY | METAGENOME, METAGENOMIC LIBRARY, ALPHA AND BETA PROTEINS, ALPHA/BETA HYDROLASE SUPERFAMILY, ESTERASE/LIPASE FOLD, HYDROLASE
4qa9:A (TYR65) to (ASN197) ENSEMBLE REFINEMENT OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS. | STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, EPOXIDE HYDROLASE, PSI-BIOLOGY, HYDROLASE
3b5e:B (PRO10) to (LEU141) CRYSTAL STRUCTURE OF CARBOXYLESTERASE (NP_108484.1) FROM MESORHIZOBIUM LOTI AT 1.75 A RESOLUTION | NP_108484.1, CARBOXYLESTERASE, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, HYDROLASE
5f4z:A (PRO67) to (ASN198) THE CRYSTAL STRUCTURE OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS | EPOXIDE HYDROLASE, STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, HYDROLASE
5f4z:B (PRO67) to (ASN198) THE CRYSTAL STRUCTURE OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS | EPOXIDE HYDROLASE, STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, HYDROLASE
5f4z:C (PRO67) to (ASN198) THE CRYSTAL STRUCTURE OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS | EPOXIDE HYDROLASE, STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, HYDROLASE
5f4z:D (VAL66) to (ASN198) THE CRYSTAL STRUCTURE OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS | EPOXIDE HYDROLASE, STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, HYDROLASE
5f4z:E (PRO67) to (ASN198) THE CRYSTAL STRUCTURE OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS | EPOXIDE HYDROLASE, STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, HYDROLASE
4qzv:A (SER511) to (VAL653) BAT-DERIVED CORONAVIRUS HKU4 USES MERS-COV RECEPTOR HUMAN CD26 FOR CELL ENTRY | 8-BLADED BETA-PROPELLER DOMAIN, ALPHA/BETA HYDROLASE DOMAIN, BLADES IV AND V, CD26 BETA-PROPELLER, HYDROLASE-VIRAL PROTEIN COMPLEX
4qzv:C (VAL507) to (VAL653) BAT-DERIVED CORONAVIRUS HKU4 USES MERS-COV RECEPTOR HUMAN CD26 FOR CELL ENTRY | 8-BLADED BETA-PROPELLER DOMAIN, ALPHA/BETA HYDROLASE DOMAIN, BLADES IV AND V, CD26 BETA-PROPELLER, HYDROLASE-VIRAL PROTEIN COMPLEX
3c43:A (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A FLOUROOLEFIN INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE
3c43:B (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A FLOUROOLEFIN INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE
3c45:A (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A FLUOROOLEFIN INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE
3c45:B (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A FLUOROOLEFIN INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE
3ccb:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A BENZIMIDAZOLE DERIVATIVE | STRUCTURE-BASED DESIGN, DENZIMIDAZOLE DERIVATIVES, PEPTIDASE, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
3ccb:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A BENZIMIDAZOLE DERIVATIVE | STRUCTURE-BASED DESIGN, DENZIMIDAZOLE DERIVATIVES, PEPTIDASE, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
3ccb:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A BENZIMIDAZOLE DERIVATIVE | STRUCTURE-BASED DESIGN, DENZIMIDAZOLE DERIVATIVES, PEPTIDASE, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
3ccc:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A BENZIMIDAZOLE DERIVATIVE | STRUCTURE-BASED DESIGN, DENZIMIDAZOLE DERIVATIVES, PEPTIDASE, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
3ccc:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A BENZIMIDAZOLE DERIVATIVE | STRUCTURE-BASED DESIGN, DENZIMIDAZOLE DERIVATIVES, PEPTIDASE, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
3ccc:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A BENZIMIDAZOLE DERIVATIVE | STRUCTURE-BASED DESIGN, DENZIMIDAZOLE DERIVATIVES, PEPTIDASE, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
3ccc:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A BENZIMIDAZOLE DERIVATIVE | STRUCTURE-BASED DESIGN, DENZIMIDAZOLE DERIVATIVES, PEPTIDASE, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
4re5:A (VAL336) to (ALA469) ACYLAMINOACYL PEPTIDASE COMPLEXED WITH A CHLOROMETHYLKETONE INHIBITOR | BETA-PROPELLER, ALPHA-BETA-HYDROLASE FOLD, CHLOROMETHYL-KETONE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4re5:B (VAL336) to (ALA469) ACYLAMINOACYL PEPTIDASE COMPLEXED WITH A CHLOROMETHYLKETONE INHIBITOR | BETA-PROPELLER, ALPHA-BETA-HYDROLASE FOLD, CHLOROMETHYL-KETONE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4re6:A (GLY332) to (ALA469) ACYLAMINOACYL PEPTIDASE COMPLEXED WITH A CHLOROMETHYLKETONE INHIBITOR | BETA-PROPELLER, ALPHA-BETA-HYDROLASE FOLD, CHLOROMETHYL-KETONE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4re6:B (GLY332) to (ALA469) ACYLAMINOACYL PEPTIDASE COMPLEXED WITH A CHLOROMETHYLKETONE INHIBITOR | BETA-PROPELLER, ALPHA-BETA-HYDROLASE FOLD, CHLOROMETHYL-KETONE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4re6:C (GLY332) to (ALA469) ACYLAMINOACYL PEPTIDASE COMPLEXED WITH A CHLOROMETHYLKETONE INHIBITOR | BETA-PROPELLER, ALPHA-BETA-HYDROLASE FOLD, CHLOROMETHYL-KETONE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4re6:D (GLY332) to (ALA469) ACYLAMINOACYL PEPTIDASE COMPLEXED WITH A CHLOROMETHYLKETONE INHIBITOR | BETA-PROPELLER, ALPHA-BETA-HYDROLASE FOLD, CHLOROMETHYL-KETONE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4c88:B (ARG76) to (LEU201) ESTERASE LPEST1 FROM LACTOBACILLUS PLANTARUM: NATIVE STRUCTURE | HYDROLASE
4c88:C (ARG76) to (LEU201) ESTERASE LPEST1 FROM LACTOBACILLUS PLANTARUM: NATIVE STRUCTURE | HYDROLASE
4c89:B (ARG76) to (LEU201) CRYSTAL STRUCTURE OF CARBOXYLESTERASE LPEST1 FROM LACTOBACILLUS PLANTARUM: HIGH RESOLUTION MODEL | HYDROLASE
4c89:C (ARG76) to (LEU201) CRYSTAL STRUCTURE OF CARBOXYLESTERASE LPEST1 FROM LACTOBACILLUS PLANTARUM: HIGH RESOLUTION MODEL | HYDROLASE
3nox:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH SA-(+)-(6- (AMINOMETHYL)-5-(2,4-DICHLOROPHENYL)-7-METHYLIMIDAZO[1,2-A]PYRIMIDIN- 2-YL)(MORPHOLINO)METHANONE | EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE
3nox:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH SA-(+)-(6- (AMINOMETHYL)-5-(2,4-DICHLOROPHENYL)-7-METHYLIMIDAZO[1,2-A]PYRIMIDIN- 2-YL)(MORPHOLINO)METHANONE | EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE
3cxu:A (LYS3) to (LEU128) STRUCTURE OF A Y149F MUTANT OF EPOXIDE HYDROLASE FROM SOLANUM TUBEROSUM | EPOXIDE HYDROLASE, ALPHA/BETA HYDROLASE FOLD, Y149F, PROTON WIRE
3o4h:A (VAL336) to (ALA469) STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY
3o4h:B (VAL336) to (ALA469) STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY
3o4h:C (VAL336) to (ALA469) STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY
3o4h:D (VAL336) to (ALA469) STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY
3o4j:A (GLY332) to (ALA469) STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY
3o4j:B (GLY332) to (ALA469) STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY
3o4j:C (GLY332) to (ALA469) STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY
3o4j:D (GLY332) to (ALA469) STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY
3o95:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-100 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX
3o95:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-100 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX
3o95:C (SER511) to (ALA654) CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-100 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX
3o95:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-100 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX
3d4l:A (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A NOVEL INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE
3d4l:B (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A NOVEL INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE
3o9v:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-986 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX
3o9v:B (SER511) to (ALA654) CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-986 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX
3o9v:C (SER511) to (ALA654) CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-986 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX
3o9v:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-986 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN, HYDROLASE,SIGNALING PROTEIN-INHIBITOR COMPLEX
3doi:A (PHE162) to (CYS310) CRYSTAL STRUCTURE OF A THERMOSTABLE ESTERASE COMPLEX WITH PARAOXON | ALPHA-BETA HYDROLASE, BETA SHEET
3opm:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-294 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE-HYDROLASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3opm:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-294 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE-HYDROLASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3opm:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-294 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE-HYDROLASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3opm:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 BOUND TO TAK-294 | PROTEASE AND 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, SIGNALING PROTEIN, HYDROLASE-HYDROLASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3e3a:A (LEU-11) to (ALA111) THE STRUCTURE OF RV0554 FROM MYCOBACTERIUM TUBERCULOSIS | ALPHA/BETA HYDROLASE, OXIDOREDUCTASE, PEROXIDASE
3e3a:B (GLU-13) to (ALA111) THE STRUCTURE OF RV0554 FROM MYCOBACTERIUM TUBERCULOSIS | ALPHA/BETA HYDROLASE, OXIDOREDUCTASE, PEROXIDASE
4dsz:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF DPP-IV WITH COMPOUND C2 | INHIBITOR COMPLEX, SERINE EXOPEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4dsz:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF DPP-IV WITH COMPOUND C2 | INHIBITOR COMPLEX, SERINE EXOPEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4dtc:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF DPP-IV WITH COMPOUND C5 | INHIBITOR COMPLEX, SERINE EXOPEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4dtc:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF DPP-IV WITH COMPOUND C5 | INHIBITOR COMPLEX, SERINE EXOPEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3pf8:A (GLY0) to (ALA130) CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536 | ALPHA/BETA HYDROLASE FOLD, ESTERASE, HYDROLASE, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES, EXTRACELLULAR
3pf8:B (ALA2) to (ALA130) CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536 | ALPHA/BETA HYDROLASE FOLD, ESTERASE, HYDROLASE, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES, EXTRACELLULAR
3pf9:A (GLY0) to (ALA130) CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536 S106A MUTANT | ALPHA/BETA HYDROLASE FOLD, ESTERASE, HYDROLASE, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES, EXTRACELLULAR
3pfb:A (GLY0) to (LEU129) CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536 S106A MUTANT IN COMPLEX WITH ETHYLFERULATE | ALPHA/BETA HYDROLASE FOLD, ESTERASE, HYDROLASE, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES, EXTRACELLULAR
3pfc:A (GLY0) to (ALA130) CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536 S106A MUTANT IN COMPLEX WITH FERULIC ACID | ALPHA/BETA HYDROLASE FOLD, ESTERASE, HYDROLASE, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES, EXTRACELLULAR
4ufn:B (LYS3) to (LEU128) LABORATORY EVOLVED VARIANT R-C1B1 OF POTATO EPOXIDE HYDROLASE STEH1 | HYDROLASE, EPOXIDE HYDROLYSIS, ALPHA/BETA-HYDROLASE, DIRECTED EVOLUTION, ASYMMETRIC SYNTHESES
4ufo:B (LYS3) to (LEU128) LABORATORY EVOLVED VARIANT R-C1B1D33E6 OF POTATO EPOXIDE HYDROLASE STEH1 | HYDROLASE, EPOXIDE HYDROLYSIS, ALPHA/BETA-HYDROLASE, DIRECTED EVOLUTION, ASYMMETRIC SYNTHESES
4ufp:A (LYS3) to (LEU128) LABORATORY EVOLVED VARIANT R-C1B1D33 OF POTATO EPOXIDE HYDROLASE STEH1 | HYDROLASE, EPOXIDE HYDROLYSIS, ALPHA/BETA-HYDROLASE, DIRECTED EVOLUTION, ASYMMETRIC SYNTHESES
4ufp:B (LYS3) to (LEU128) LABORATORY EVOLVED VARIANT R-C1B1D33 OF POTATO EPOXIDE HYDROLASE STEH1 | HYDROLASE, EPOXIDE HYDROLYSIS, ALPHA/BETA-HYDROLASE, DIRECTED EVOLUTION, ASYMMETRIC SYNTHESES
3q0t:A (SER511) to (ALA654) CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITHSA-(+)- METHYL2-(3- (AMINOMETHYL)-4-(2,4-DICHLOROPHENYL)-2-METHYL- 7-OXO-5H-PYRROLO[3,4- B]PYRIDIN-6(7H)-YL)ACETATE | EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3q0t:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITHSA-(+)- METHYL2-(3- (AMINOMETHYL)-4-(2,4-DICHLOROPHENYL)-2-METHYL- 7-OXO-5H-PYRROLO[3,4- B]PYRIDIN-6(7H)-YL)ACETATE | EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5ivi:A (CYS89) to (SER244) THE ALPHA-ESTERASE-7 CARBOXYLESTERASE, E3, FROM THE BLOWFLY LUCILIA CUPRINA: PHOSPHORYLATED ENZYME QFIT MULTI-CONFORMER MODEL | CARBOXYLESTERASE, ORGANOPHOSPHATE, PROTEIN DYNAMICS, ACETYLCHOLINESTERASE, HYDROLASE
3qm1:A (GLY0) to (ALA130) CRYSTAL STRUCTURE OF THE LACTOBACILLUS JOHNSONII CINNAMOYL ESTERASE LJ0536 S106A MUTANT IN COMPLEX WITH ETHYLFERULATE, FORM II | ALPHA/BETA HYDROLASE FOLD, CINNAMOYL/FERULOYL ESTERASE, HYDROXYCINAMMATES, HYDROLASE
4w1p:A (CYS89) to (SER244) KINETIC CRYSTALLOGRAPHY OF ALPHA_E7-CARBOXYLESTERSE FROM LUCILLA CUPRINA - ABSORBED X-RAY DOSE 5.54 MGY TEMP 150K | ALPHA/BETA HYDROLASE FOLD, CARBOXYLESTERASE, HYDROLASE
4w1r:A (CYS89) to (SER244) KINETIC CRYSTALLOGRAPHY OF ALPHA_E7-CARBOXYLESTERSE FROM LUCILLA CUPRINA - ABSORBED X-RAY DOSE 9.24 MGY TEMP 150K | ALPHA/BETA HYDROLASE FOLD, CARBOXYLESTERASE, HYDROLASE
3r3u:A (GLY10) to (LEU133) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - WT/APO | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r3u:B (GLY10) to (LEU133) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - WT/APO | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r3v:B (GLY10) to (LEU133) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - ASP110ASN/FLUOROACETATE | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r3w:A (GLY10) to (LEU133) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - ASP110ASN/CHLOROACETATE | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r3w:B (GLY10) to (LEU133) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - ASP110ASN/CHLOROACETATE | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r3x:A (GLY12) to (LEU133) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - ASP110ASN/BROMOACETATE | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r3x:B (GLY10) to (LEU133) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - ASP110ASN/BROMOACETATE | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r3y:A (GLY12) to (ASP134) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - HIS280ASN/FLUOROACETATE | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r3y:B (GLY10) to (ASP134) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - HIS280ASN/FLUOROACETATE | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r3z:A (GLY10) to (LEU133) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - WT/GLYCOLATE | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r3z:B (GLY10) to (LEU133) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - WT/GLYCOLATE | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r3z:C (GLY10) to (ASP134) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - WT/GLYCOLATE | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r3z:D (GLY10) to (LEU133) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - WT/GLYCOLATE | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r40:A (GLY10) to (LEU133) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - ASP110ASN/APO | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r40:B (GLY10) to (LEU133) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - ASP110ASN/APO | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r41:A (GLY10) to (ASP134) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - HIS280ASN/APO | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
3r41:B (GLY10) to (ASP134) CRYSTAL STRUCTURE OF THE FLUOROACETATE DEHALOGENASE RPA1163 - HIS280ASN/APO | FACD, DEFLUORINASE, ALPHA/BETA HYDROLASE, HYDROLASE
4g1f:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIDOPYRIMIDINEDIONE ANALOGUE | PROTEASE, 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, SECRETED, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4g1f:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIDOPYRIMIDINEDIONE ANALOGUE | PROTEASE, 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, SECRETED, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4g1f:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIDOPYRIMIDINEDIONE ANALOGUE | PROTEASE, 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, SECRETED, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4g1f:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIDOPYRIMIDINEDIONE ANALOGUE | PROTEASE, 8-BLADED BETA-PROPELLER DOMAIN, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, SECRETED, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5l8s:A (MET341) to (PHE482) THE CRYSTAL STRUCTURE OF A COLD-ADAPTED ACYLAMINOACYL PEPTIDASE REVEALS A NOVEL QUATERNARY ARCHITECTURE BASED ON THE ARM-EXCHANGE MECHANISM | ACYL AMINOACYL PEPTIDASE, ALPHA/BETA HYDROLASE DOMAIN, ARM EXCHANGE, BETA-PROPELLER DOMAIN, COLD ADAPTATION, DIMERIZATION, PROLINE HINGE, SPOROSARCINA PSYCHROPHILA, HYDROLASE
5l8s:B (MET341) to (PHE482) THE CRYSTAL STRUCTURE OF A COLD-ADAPTED ACYLAMINOACYL PEPTIDASE REVEALS A NOVEL QUATERNARY ARCHITECTURE BASED ON THE ARM-EXCHANGE MECHANISM | ACYL AMINOACYL PEPTIDASE, ALPHA/BETA HYDROLASE DOMAIN, ARM EXCHANGE, BETA-PROPELLER DOMAIN, COLD ADAPTATION, DIMERIZATION, PROLINE HINGE, SPOROSARCINA PSYCHROPHILA, HYDROLASE
5t4b:A (SER511) to (VAL653) HUMAN DPP4 IN COMPLEX WITH A LIGAND 34A | STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5t4b:B (SER511) to (VAL653) HUMAN DPP4 IN COMPLEX WITH A LIGAND 34A | STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5t4e:A (SER511) to (VAL653) HUMAN DPP4 IN COMPLEX WITH LIGAND 19A | STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5t4e:B (SER511) to (VAL653) HUMAN DPP4 IN COMPLEX WITH LIGAND 19A | STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5t4f:A (SER511) to (VAL653) HUMAN DPP4 IN COMPLEX WITH LIGAND 34P | STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5t4f:B (SER511) to (VAL653) HUMAN DPP4 IN COMPLEX WITH LIGAND 34P | STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5t4h:A (SER511) to (VAL653) HUMAN DPP4 IN COMPLEX WITH LIGAND 34N | STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5t4h:B (SER511) to (VAL653) HUMAN DPP4 IN COMPLEX WITH LIGAND 34N | STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2ajb:B (SER511) to (ALA654) PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH THE TRIPEPTIDE TERT-BUTYL-GLY-L-PRO-L-ILE (TBU-GPI) | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2ajb:C (SER511) to (VAL653) PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH THE TRIPEPTIDE TERT-BUTYL-GLY-L-PRO-L-ILE (TBU-GPI) | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2ajb:D (SER511) to (VAL653) PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH THE TRIPEPTIDE TERT-BUTYL-GLY-L-PRO-L-ILE (TBU-GPI) | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2ajd:B (SER511) to (VAL653) PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH L-PRO-BORO-L- PRO (BOROPRO) | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE
2ajd:C (SER511) to (ALA654) PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH L-PRO-BORO-L- PRO (BOROPRO) | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE
2ajd:D (SER511) to (VAL653) PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH L-PRO-BORO-L- PRO (BOROPRO) | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE, ALPHA/BETA-HYDROLASE, BETA- PROPELLER, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, FLEXIBILITY, HYDROLASE
3ed1:C (VAL63) to (LEU224) CRYSTAL STRUCTURE OF RICE GID1 COMPLEXED WITH GA3 | ALPHA/BETA HYDROLASE, LIPASE, GIBBERELLIN SIGNALING PATHWAY, HYDROLASE, NUCLEUS, RECEPTOR, HYDROLASE RECEPTOR
3ed1:E (VAL63) to (LEU224) CRYSTAL STRUCTURE OF RICE GID1 COMPLEXED WITH GA3 | ALPHA/BETA HYDROLASE, LIPASE, GIBBERELLIN SIGNALING PATHWAY, HYDROLASE, NUCLEUS, RECEPTOR, HYDROLASE RECEPTOR
3ed1:F (VAL63) to (LEU224) CRYSTAL STRUCTURE OF RICE GID1 COMPLEXED WITH GA3 | ALPHA/BETA HYDROLASE, LIPASE, GIBBERELLIN SIGNALING PATHWAY, HYDROLASE, NUCLEUS, RECEPTOR, HYDROLASE RECEPTOR
2oph:A (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH AN ALPHA AMINO ACID INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, TYPE 2 DIABETES, SELECTIVE INHIBITOR, HYDROLASE
2oph:B (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH AN ALPHA AMINO ACID INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, TYPE 2 DIABETES, SELECTIVE INHIBITOR, HYDROLASE
2p8s:A (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A CYCLOHEXALAMINE INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, STRUCTURE-BASED DESIGN, HYDROLASE
2p8s:B (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 IN COMPLEX WITH A CYCLOHEXALAMINE INHIBITOR | ALPHA/BETA, BETA-PROPELLER, DIMER, STRUCTURE-BASED DESIGN, HYDROLASE
1bn6:A (ASP22) to (MET140) HALOALKANE DEHALOGENASE FROM A RHODOCOCCUS SPECIES | DEHALOGENASE, ALPHA/BETA-HYDROLASE, DHLA, CRYSTAL STRUCTURE
2buc:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A TETRAHYDROISOQUINOLINE INHIBITOR | HYDROLASE/INHIBITOR, COMPLEX (HYDROLASE/INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX
2buc:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A TETRAHYDROISOQUINOLINE INHIBITOR | HYDROLASE/INHIBITOR, COMPLEX (HYDROLASE/INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX
2buc:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A TETRAHYDROISOQUINOLINE INHIBITOR | HYDROLASE/INHIBITOR, COMPLEX (HYDROLASE/INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX
2buc:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A TETRAHYDROISOQUINOLINE INHIBITOR | HYDROLASE/INHIBITOR, COMPLEX (HYDROLASE/INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, COMPLEX
1orw:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A PEPTIDOMIMETIC INHIBITOR | SERINE PROTEASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, HYDROLASE
1orw:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF PORCINE DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A PEPTIDOMIMETIC INHIBITOR | SERINE PROTEASE, OXYANION HOLE, SUBSTRATE CHANNELING, DRUG DESIGN, DIABETES MELLITUS, HYDROLASE
2q2e:A (GLY178) to (GLY289) CRYSTAL STRUCTURE OF THE TOPOISOMERASE VI HOLOENZYME FROM METHANOSARCINA MAZEI | TOPOISOMERASE, DNA-BINDING, SPO11, ATPASE, ISOMERASE
3fvt:B (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM II | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvt:F (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM II | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvt:I (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM II | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvt:L (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM II | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3fvt:M (GLY53) to (ASP203) CRYSTAL STRUCTURE OF ACETYL XYLAN ESTERASE FROM BACILLUS PUMILUS, MONOCLINIC CRYSTAL FORM II | ALPHA/BETA HYDROLASE, CARBOHYDRATE ESTERASE, CE7, BACILLUS PUMILUS, HYDROLASE
3g0c:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 1 | DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0c:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 1 | DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0c:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 1 | DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g0c:D (VAL507) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH A PYRIMIDINEDIONE INHIBITOR 1 | DPP4, PYRIMIDINONE, PYRIMIDINDIONE, AMINOPEPTIDASE, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2qjr:A (SER511) to (VAL653) DIPEPDYL PEPTIDASE IV IN COMPLEX WITH INHIBITOR PZF | PROTEIN-INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
2qjr:B (SER511) to (VAL653) DIPEPDYL PEPTIDASE IV IN COMPLEX WITH INHIBITOR PZF | PROTEIN-INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
3t4u:A (SER1) to (GLY119) L29I MUTATION IN AN ARYL ESTERASE FROM PSEUDOMONAS FLUORESCENS LEADS TO UNIQUE PEPTIDE FLIP AND INCREASED ACTIVITY | OXIDOREDUCTASE, HYDRLOASE
3t4u:B (SER1) to (GLY119) L29I MUTATION IN AN ARYL ESTERASE FROM PSEUDOMONAS FLUORESCENS LEADS TO UNIQUE PEPTIDE FLIP AND INCREASED ACTIVITY | OXIDOREDUCTASE, HYDRLOASE
3t4u:C (SER1) to (GLY119) L29I MUTATION IN AN ARYL ESTERASE FROM PSEUDOMONAS FLUORESCENS LEADS TO UNIQUE PEPTIDE FLIP AND INCREASED ACTIVITY | OXIDOREDUCTASE, HYDRLOASE
3t4u:D (SER1) to (GLY119) L29I MUTATION IN AN ARYL ESTERASE FROM PSEUDOMONAS FLUORESCENS LEADS TO UNIQUE PEPTIDE FLIP AND INCREASED ACTIVITY | OXIDOREDUCTASE, HYDRLOASE
3t4u:E (SER1) to (GLY119) L29I MUTATION IN AN ARYL ESTERASE FROM PSEUDOMONAS FLUORESCENS LEADS TO UNIQUE PEPTIDE FLIP AND INCREASED ACTIVITY | OXIDOREDUCTASE, HYDRLOASE
3t4u:F (SER1) to (GLY119) L29I MUTATION IN AN ARYL ESTERASE FROM PSEUDOMONAS FLUORESCENS LEADS TO UNIQUE PEPTIDE FLIP AND INCREASED ACTIVITY | OXIDOREDUCTASE, HYDRLOASE
3h17:A (ASP43) to (ILE171) CRYSTAL STRUCTURE OF ESTE5-PMSF (I) | HSL, ESTE5, ESTERASE, LIPASE, HYDROLASE, PMSF, PHENYLMETHYLSULFONYL FLUORIDE
3hab:A (SER511) to (VAL653) THE STRUCTURE OF DPP4 IN COMPLEX WITH PIPERIDINE FUSED BENZIMIDAZOLE 25 | ALPHA/BETA, BETA-PROPELLER, DIMER, HYDROLASE, DIABETES, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3hab:B (SER511) to (VAL653) THE STRUCTURE OF DPP4 IN COMPLEX WITH PIPERIDINE FUSED BENZIMIDAZOLE 25 | ALPHA/BETA, BETA-PROPELLER, DIMER, HYDROLASE, DIABETES, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3hac:A (SER511) to (VAL653) THE STRUCTURE OF DPP-4 IN COMPLEX WITH PIPERIDINE FUSED IMIDAZOPYRIDINE 34 | ALPHA/BETA, BETA-PROPELLER, DIMER, HYDROLASE, DIABETES, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3hac:B (SER511) to (VAL653) THE STRUCTURE OF DPP-4 IN COMPLEX WITH PIPERIDINE FUSED IMIDAZOPYRIDINE 34 | ALPHA/BETA, BETA-PROPELLER, DIMER, HYDROLASE, DIABETES, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3hju:A (PRO20) to (ILE145) CRYSTAL STRUCTURE OF HUMAN MONOGLYCERIDE LIPASE | ALPHA/BETA HYDROLASE, HYDROLASE, SERINE ESTERASE
2fuk:A (LEU13) to (ALA141) CRYSTAL STRUCTURE OF XC6422 FROM XANTHOMONAS CAMPESTRIS: A MEMBER OF A/B SERINE HYDROLASE WITHOUT LID AT 1.6 RESOLUTION | A/B HYDROLASE, XANTHOMONAS CAMPESTRIS, STRUCTURAL GENOMICS, X-RAY DIFFRACTION
1sfr:A (PRO7) to (MET149) CRYSTAL STRUCTURE OF THE MYCOBACTERIUM TUBERCULOSIS ANTIGEN 85A PROTEIN | ALPHA/BETA HYDROLASE, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, TRANSFERASE
2gbc:A (SER512) to (VAL654) NATIVE DPP-IV (CD26) FROM RAT | BETA PROPELLER, HYDROLASE
2gbc:B (SER512) to (VAL654) NATIVE DPP-IV (CD26) FROM RAT | BETA PROPELLER, HYDROLASE
1tht:A (LYS6) to (ALA135) STRUCTURE OF A MYRISTOYL-ACP-SPECIFIC THIOESTERASE FROM VIBRIO HARVEYI | THIOESTERASE
1tht:B (LYS6) to (VAL136) STRUCTURE OF A MYRISTOYL-ACP-SPECIFIC THIOESTERASE FROM VIBRIO HARVEYI | THIOESTERASE
1tk3:A (SER511) to (ALA654) CRYSTAL STRUCTURE OF HUMAN APO DIPEPTIDYL PEPTIDASE IV/CD26 | ALPHA/BETA HYDROLASE, BETA-PROPELLER, HOMODIMER, HYDROLASE
1tk3:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN APO DIPEPTIDYL PEPTIDASE IV/CD26 | ALPHA/BETA HYDROLASE, BETA-PROPELLER, HOMODIMER, HYDROLASE
1tkr:B (SER511) to (ALA654) HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 INHIBITED WITH DIISOPROPYL FLUOROPHOSPHATE | ALPHA/BETA HYDROLASE, BETA-PROPELLER, HOMODIMER, HYDROLASE
4zxf:A (GLU14) to (SER148) CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE IN COMPLEX WITH A SUBSTRATE ANALOG | HYDROLASE, MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, COMPLEX, SUBSTRATE ANALOG
4zxf:B (GLU14) to (GLY149) CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE IN COMPLEX WITH A SUBSTRATE ANALOG | HYDROLASE, MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, COMPLEX, SUBSTRATE ANALOG
4zxf:C (GLU14) to (SER148) CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE IN COMPLEX WITH A SUBSTRATE ANALOG | HYDROLASE, MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, COMPLEX, SUBSTRATE ANALOG
4zxf:D (PRO13) to (GLY149) CRYSTAL STRUCTURE OF A SOLUBLE VARIANT OF MONOGLYCERIDE LIPASE FROM SACCHAROMYCES CEREVISIAE IN COMPLEX WITH A SUBSTRATE ANALOG | HYDROLASE, MONOGLYCERIDE LIPASE, MONOACYLGLYCEROL LIPASE, COMPLEX, SUBSTRATE ANALOG
2hha:A (SER511) to (VAL653) THE STRUCTURE OF DPP4 IN COMPLEX WITH AN OXADIAZOLE INHIBITOR | HYDROLASE, ALPHA/BETA, BETA-PROPELLER, DIMER
2hha:B (SER511) to (VAL653) THE STRUCTURE OF DPP4 IN COMPLEX WITH AN OXADIAZOLE INHIBITOR | HYDROLASE, ALPHA/BETA, BETA-PROPELLER, DIMER
2i03:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE 4 (DPP IV) WITH POTENT ALKYNYL CYANOPYRROLIDINE (ABT-279) | ENZYME, SERINE PEPTIDASE, HYDROLASE
2iit:A (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE 4 IN COMPLEX WITH A DIAZEPAN-2-ONE INHIBITOR | HYDROLASE; ALPHA/BETA; BETA-PROPELLER; DIMER, HYDROLASE
2iit:B (SER511) to (VAL653) HUMAN DIPEPTIDYL PEPTIDASE 4 IN COMPLEX WITH A DIAZEPAN-2-ONE INHIBITOR | HYDROLASE; ALPHA/BETA; BETA-PROPELLER; DIMER, HYDROLASE
1wcy:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (DPPIV) COMPLEX WITH DIPROTIN A | SERINE PROTEASE, DIPEPTIDYL PEPTIDASE IV, CD26, PROLYL OLIGOPEPTIDASE, BETA-PROPELLER STRUCTURE, DIPROTIN A, HYDROLASE
4a5s:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A NOVAL HETEROCYCLIC DPP4 INHIBITOR | HYDROLASE, TYPE 2 DIABETES, NOVARTIS COMPOUND NVP-BIV988
4a5s:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP4 IN COMPLEX WITH A NOVAL HETEROCYCLIC DPP4 INHIBITOR | HYDROLASE, TYPE 2 DIABETES, NOVARTIS COMPOUND NVP-BIV988
3kwf:B (SER511) to (VAL653) HUMAN DPP-IV WITH CARMEGLIPTIN (S)-1-((2S,3S,11BS)-2-AMINO- 9,10-DIMETHOXY-1,3,4,6,7,11B-HEXAHYDRO-2H-PYRIDO[2,1- A]ISOQUINOLIN-3-YL)-4-FLUOROMETHYL-PYRROLIDIN-2-ONE | DIABETES TYPE II, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
1z68:A (ASN500) to (VAL647) CRYSTAL STRUCTURE OF HUMAN FIBROBLAST ACTIVATION PROTEIN ALPHA | SEPRASE, FIBROBLAST ACTIVATION PROTEIN ALPHA,FAPALPHA, DIPEPTIDYLPEPTIDASE,S9B, INTEGRAL MEMBRANE SERINE PROTEASE, LYASE
1z68:B (PRO504) to (VAL647) CRYSTAL STRUCTURE OF HUMAN FIBROBLAST ACTIVATION PROTEIN ALPHA | SEPRASE, FIBROBLAST ACTIVATION PROTEIN ALPHA,FAPALPHA, DIPEPTIDYLPEPTIDASE,S9B, INTEGRAL MEMBRANE SERINE PROTEASE, LYASE
4q1v:A (TYR476) to (GLY626) CRYSTAL STRUCTURE OF A PUTATIVE DIPEPTIDYL AMINOPEPTIDASE IV (BACOVA_01349) FROM BACTEROIDES OVATUS ATCC 8483 AT 2.48 A RESOLUTION | TWO DOMAIN PROTEIN, DIPEPTIDYL-PEPTIDASE IV FAMILY (PF00930), PROLYL OLIGOPEPTIDASE FAMILY (PF00326), STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI- BIOLOGY, HYDROLASE
4q1v:B (TYR476) to (GLY627) CRYSTAL STRUCTURE OF A PUTATIVE DIPEPTIDYL AMINOPEPTIDASE IV (BACOVA_01349) FROM BACTEROIDES OVATUS ATCC 8483 AT 2.48 A RESOLUTION | TWO DOMAIN PROTEIN, DIPEPTIDYL-PEPTIDASE IV FAMILY (PF00930), PROLYL OLIGOPEPTIDASE FAMILY (PF00326), STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI- BIOLOGY, HYDROLASE
3bjm:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH (1S,3S, 5S)-2-[(2S)- 2-AMINO-2-(3-HYDROXYTRICYCLO[3.3.1.13,7]DEC-1- YL)ACETYL]-2- AZABICYCLO[3.1.0]HEXANE-3-CARBONITRILE (CAS), (1S,3S,5S)-2-((2S)-2- AMINO-2-(3-HYDROXYADAMANTAN-1- YL)ACETYL)-2-AZABICYCLO[3.1.0]HEXANE- 3-CARBONITRILE (IUPAC), OR BMS-477118 | EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE
3bjm:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF HUMAN DPP-IV IN COMPLEX WITH (1S,3S, 5S)-2-[(2S)- 2-AMINO-2-(3-HYDROXYTRICYCLO[3.3.1.13,7]DEC-1- YL)ACETYL]-2- AZABICYCLO[3.1.0]HEXANE-3-CARBONITRILE (CAS), (1S,3S,5S)-2-((2S)-2- AMINO-2-(3-HYDROXYADAMANTAN-1- YL)ACETYL)-2-AZABICYCLO[3.1.0]HEXANE- 3-CARBONITRILE (IUPAC), OR BMS-477118 | EXOPEPTIDASE, ALPHA/BETA HYDROLASE FOLD, BETA BARREL, BETA PROPELLER, DPP4, DIMER, PROTEIN:INHIBITOR COMPLEX, AMINOPEPTIDASE, GLYCOPROTEIN, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE, HYDROLASE
4c87:C (ARG76) to (LEU201) ESTERASE LPEST1 FROM LACTOBACILLUS PLANTARUM WCFS1 | HYDROLASE
3o4g:A (GLY332) to (ALA469) STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY
3o4g:B (VAL336) to (ALA469) STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY
3o4g:C (GLY332) to (ALA469) STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY
3o4g:D (VAL336) to (ALA469) STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY
3o4i:A (VAL336) to (ALA469) STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY
3o4i:B (VAL336) to (ALA469) STRUCTURE AND CATALYSIS OF ACYLAMINOACYL PEPTIDASE | ALPHA/BETA HYDROLASE FOLD, BETA PROPELLER, HYDROLASE, OLIGOPEPTIDASE, SIZE SELECTIVITY
3our:C (TYR166) to (GLY296) CRYSTAL STRUCTURE OF COMPLEX BETWEEN EIIA AND A NOVEL PYRUVATE DECARBOXYLASE | EXHIBIT NO HYDROLASE ACTIVITY1, LYASE-TRANSFERASE COMPLEX
5i7u:A (SER511) to (VAL653) HUMAN DPP4 IN COMPLEX WITH A NOVEL TRICYCLIC HETERO-CYCLE INHIBITOR | STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5i7u:B (SER511) to (VAL653) HUMAN DPP4 IN COMPLEX WITH A NOVEL TRICYCLIC HETERO-CYCLE INHIBITOR | STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4uuq:A (PRO30) to (ILE155) CRYSTAL STRUCTURE OF HUMAN MONO-GLYCERIDE LIPASE IN COMPLEX WITH SAR127303 | HYDROLASE
5ism:A (SER511) to (VAL653) HUMAN DPP4 IN COMPLEX WITH A NOVEL 5,5,6-TRICYCLIC PYRROLIDINE INHIBITOR | STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5ism:B (SER511) to (VAL653) HUMAN DPP4 IN COMPLEX WITH A NOVEL 5,5,6-TRICYCLIC PYRROLIDINE INHIBITOR | STRUCTURE-BASED DRUG DESIGN, DIABETES, DPP4 INHIBITORS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3qbj:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH INHIBITOR | DIABETES MELLITUS, DIPEPTIDYL-PEPTIDASE IV INHIBITOR, HYPOGLYCEMIC AGENT, PYRROLIDINES, SPRAGUE-DAWLEY, STRUCTURE-ACTIVITY RELATIONSHIP, HYDROLASE, GLYCOSYLATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3qbj:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH INHIBITOR | DIABETES MELLITUS, DIPEPTIDYL-PEPTIDASE IV INHIBITOR, HYPOGLYCEMIC AGENT, PYRROLIDINES, SPRAGUE-DAWLEY, STRUCTURE-ACTIVITY RELATIONSHIP, HYDROLASE, GLYCOSYLATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5kby:A (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH SYR-472 | PEPTIDASE, GLP-1, METABOLIC DISEASE, CO-COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5kby:B (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH SYR-472 | PEPTIDASE, GLP-1, METABOLIC DISEASE, CO-COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5kby:C (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH SYR-472 | PEPTIDASE, GLP-1, METABOLIC DISEASE, CO-COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5kby:D (SER511) to (VAL653) CRYSTAL STRUCTURE OF DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH SYR-472 | PEPTIDASE, GLP-1, METABOLIC DISEASE, CO-COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5lls:A (SER511) to (VAL653) PORCINE DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH 8-(3-AMINOPIPERIDIN-1- YL)-7-[(2-BROMOPHENYL)METHYL]-1,3-DIMETHYL-2,3,6,7-TETRAHYDRO-1H- PURINE-2,6-DIONE | PEPTIDASE, INHIBITOR, COMPLEX, HYDROLASE
5lls:B (SER511) to (VAL653) PORCINE DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH 8-(3-AMINOPIPERIDIN-1- YL)-7-[(2-BROMOPHENYL)METHYL]-1,3-DIMETHYL-2,3,6,7-TETRAHYDRO-1H- PURINE-2,6-DIONE | PEPTIDASE, INHIBITOR, COMPLEX, HYDROLASE
5lls:C (SER511) to (VAL653) PORCINE DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH 8-(3-AMINOPIPERIDIN-1- YL)-7-[(2-BROMOPHENYL)METHYL]-1,3-DIMETHYL-2,3,6,7-TETRAHYDRO-1H- PURINE-2,6-DIONE | PEPTIDASE, INHIBITOR, COMPLEX, HYDROLASE
5lls:D (SER511) to (VAL653) PORCINE DIPEPTIDYL PEPTIDASE IV IN COMPLEX WITH 8-(3-AMINOPIPERIDIN-1- YL)-7-[(2-BROMOPHENYL)METHYL]-1,3-DIMETHYL-2,3,6,7-TETRAHYDRO-1H- PURINE-2,6-DIONE | PEPTIDASE, INHIBITOR, COMPLEX, HYDROLASE