4w9x:A (HIS49) to (LEU129) CRYSTAL STRUCTURE OF BMP-2-INDUCIBLE KINASE IN COMPLEX WITH BARICITINIB | KINASE, SMALL-MOLECULE, CATALYTIC DOMAIN, PROTEIN BINDING, INHIBITOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
4wbo:C (TRP186) to (MET264) BOVINE G PROTEIN COUPLED RECEPTOR KINASE 1 IN COMPLEX WITH AMLEXANOX | G-PROTEIN-COUPLED RECEPTOR KINASE 1, AMLEXANOX, PHOSPHORYLATION, PROTEIN CONFORMATION, PROTEIN KINASE INHIBITORS, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
2obj:A (GLN37) to (GLU121) CRYSTAL STRUCTURE OF HUMAN PIM-1 KINASE IN COMPLEX WITH INHIBITOR | PIM, PIM-1, PIM1, HUMAN PIM-1 KINASE, SERINE/THREONINE KINASE, KINASE INHIBITOR COMPLEX, PYRIDONE, KINASE INHIBITOR, TRANSFERASE
4gw8:A (GLN37) to (ILE119) HUMAN PROTO-ONCOGENE SERINE THREONINE KINASE (PIM1) IN COMPLEX WITH A CONSENSUS PEPTIDE AND LEUCETTINE L41 | ONCOGENE, KINASE, SERINE-THREONINE, PIM1, STRUCTURAL GENOMICS CONSORTIUM, SGC, ALTERNATIVE INITIATION, ATP-BINDING, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, HOST-VIRUS INTERACTION, VIRAL IMMUNOEVASION, VIRION, VIRULENCE, CELL CYCLE, CELL MEMBRANE
4wsy:A (GLN37) to (ILE119) CRYSTAL STRUCTURE OF HUMAN PIM-1 KINASE IN COMPLEX WITH A THIAZOLAMINE-INDAZOLE INHIBITOR. | TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4hyh:A (ASP8) to (PHE83) X-RAY CRYSTAL STRUCTURE OF COMPOUND 39 BOUND TO HUMAN CHK1 KINASE DOMAIN | SERINE/THREONINE-PROTEIN KINASE CHK1 INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4xh6:A (GLN37) to (LEU120) CRYSTAL STRUCTURE OF PROTO-ONCOGENE KINASE PIM1 BOUND TO HISPIDULIN | PIM1, HISPIDULIN, INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2c3i:B (GLN37) to (ILE119) CRYSTAL STRUCTURE OF HUMAN PIM1 IN COMPLEX WITH IMIDAZOPYRIDAZIN I | TRANSFERASE-PEPTIDE COMPLEX, COMPLEX TRANSFERASE/PEPTIDE, PIM1, KINASE, CANCER, LEUKEMIA, ATP-BINDING, NUCLEAR PROTEIN, NUCLEOTIDE-BINDING, PHOSPHORYLATION, PROTO- ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
1csn:A (HIS11) to (ILE85) BINARY COMPLEX OF CASEIN KINASE-1 WITH MGATP | PHOSPHOTRANSFERASE
3fwq:B (ASP38) to (GLU114) INACTIVE CONFORMATION OF HUMAN PROTEIN KINASE CK2 CATALYTIC SUBUNIT | CASEIN KINASE 2, PROTEIN KINASE CK2, EUKARYOTIC PROTEIN KINASES, INACTIVE CONFORMATION, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
3g2f:A (ASN202) to (GLU280) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF BONE MORPHOGENETIC PROTEIN RECEPTOR TYPE II (BMPR2) AT 2.35 A RESOLUTION | KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
2qg5:D (TYR28) to (VAL101) CRYPTOSPORIDIUM PARVUM CALCIUM DEPENDENT PROTEIN KINASE CGD7_1840 | MALARIA, CALCIUM DEPENDENT KINASE, SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSFERASE
2cke:A (PHE12) to (GLU94) HUMAN DEATH-ASSOCIATED DRP-1 KINASE IN COMPLEX WITH INHIBITOR | TRANSFERASE-INHIBITOR COMPLEX, TRANSFERASE/INHIBITOR COMPLEX, CALMODULIN-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, APOPTOSIS
2cke:C (PHE12) to (GLU94) HUMAN DEATH-ASSOCIATED DRP-1 KINASE IN COMPLEX WITH INHIBITOR | TRANSFERASE-INHIBITOR COMPLEX, TRANSFERASE/INHIBITOR COMPLEX, CALMODULIN-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, APOPTOSIS
2cke:D (TYR13) to (GLU94) HUMAN DEATH-ASSOCIATED DRP-1 KINASE IN COMPLEX WITH INHIBITOR | TRANSFERASE-INHIBITOR COMPLEX, TRANSFERASE/INHIBITOR COMPLEX, CALMODULIN-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, APOPTOSIS
2qnj:A (TYR56) to (MET132) KINASE AND UBIQUITIN-ASSOCIATED DOMAINS OF MARK3/PAR-1 | SERINE/THREONINE PROTEIN KINASE, UBIQUITIN-ASSOCIATED DOMAIN, MARK, PAR-1, TRANSFERASE
3h30:A (ASP38) to (GLU114) CRYSTAL STRUCTURE OF THE CATALYTIC SUBUNIT OF HUMAN PROTEIN KINASE CK2 WITH 5,6-DICHLORO-1-BETA-D- RIBOFURANOSYLBENZIMIDAZOLE | PROTEIN KINASE CK2, CASEIN KINASE 2, CASEIN KINASE II, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
4jnw:B (LYS23) to (ILE96) BACTERIALLY EXPRESSED TITIN KINASE | MUSCLE CYTOSKELETON, TRANSFERASE
3u9n:A (ASP8) to (PHE83) X-RAY CRYSTAL STRUCTURE OF COMPOUND 1 BOUND TO HUMAN CHK1 KINASE DOMAIN | PROTEIN KINASE DOMAIN, ATPASE, ATP BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uix:A (GLN37) to (ILE119) CRYSTAL STRUCTURE OF PIM1 KINASE IN COMPLEX WITH SMALL MOLECULE INHIBITOR | PIM-1, LEUKEMIA CELL LETHALITY, SUBSTRATE-PEPTIDE-BINDING RESIDUE, FLUORESCENT CORRELATION SPECTROSCOPY, INHIBITOR COMPLEX, IN SILICO SCREENING, TRANSFERASE-INHIBITOR COMPLEX
3umw:A (GLN37) to (LEU120) CRYSTAL STRUCTURE OF PIM1 KINASE IN COMPLEX WITH INHIBITOR (Z)-2-[(1H- INDAZOL-3-YL)METHYLENE]-6-METHOXY-7-(PIPERAZIN-1-YLMETHYL)BENZOFURAN- 3(2H)-ONE | PIM1, KINASE INHIBITOR, RATIONAL DRUG DESIGN, LEUKEMIA, TRANSFERASE- INHIBITOR COMPLEX
2fb8:A (GLN456) to (GLN530) STRUCTURE OF THE B-RAF KINASE DOMAIN BOUND TO SB-590885 | KINASE DOMAIN, TRANSFERASE
3vbq:A (GLN37) to (GLU121) EXPLOITATION OF HYDROGEN BONDING CONSTRAINTS AND FLAT HYDROPHOBIC ENERGY LANDSCAPES IN PIM-1 KINASE NEEDLE SCREENING AND INHIBITOR DESIGN | PIM1, ROSSMANN FOLD, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2gdo:A (ASP8) to (PHE83) 4-(AMINOALKYLAMINO)-3-BENZIMIDAZOLE-QUINOLINONES AS POTENT CHK1 INHIBITORS | DRUG DESIGN, ATP-BINDING, CELL CYCLE, DNA DAMAGE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2gqg:A (ASP241) to (GLU316) X-RAY CRYSTAL STRUCTURE OF DASATINIB (BMS-354825) BOUND TO ACTIVATED ABL KINASE DOMAIN | KINASE, TRANSFERASE
4lgd:A (VAL26) to (GLU100) STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5 | HIPPO, MST AUTOACTIVATION, RASSF, SARAH DOMAIN, DIMERIZATION, SIGNALING PROTEIN
1tki:A (LYS23) to (GLU98) AUTOINHIBITED SERINE KINASE DOMAIN OF THE GIANT MUSCLE PROTEIN TITIN | SERINE KINASE, TITIN, MUSCLE, AUTOINHIBITION
1tki:B (LYS23) to (GLU98) AUTOINHIBITED SERINE KINASE DOMAIN OF THE GIANT MUSCLE PROTEIN TITIN | SERINE KINASE, TITIN, MUSCLE, AUTOINHIBITION
2hak:A (ASN52) to (GLY134) CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1 | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE
2hak:F (TYR53) to (MET129) CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1 | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE
2hak:G (ASN52) to (GLY134) CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1 | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE
4ll5:A (TYR38) to (ILE119) CRYSTAL STRUCTURE OF PIM-1 IN COMPLEX WITH THE FLUORESCENT COMPOUND SKF86002 | CO-CRYSTALLIZATION, SKF86002, FLUORESCENCE, INHIBITOR SCREENING, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2wnt:A (GLY417) to (THR489) CRYSTAL STRUCTURE OF THE HUMAN RIBOSOMAL PROTEIN S6 KINASE | ATP-BINDING, POLYMORPHISM, METAL-BINDING, HUMAN, KINASE, RIBOSOMAL, MAGNESIUM, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, PHOSPHOPROTEIN, NUCLEOTIDE-BINDING
2wnt:B (GLY417) to (THR489) CRYSTAL STRUCTURE OF THE HUMAN RIBOSOMAL PROTEIN S6 KINASE | ATP-BINDING, POLYMORPHISM, METAL-BINDING, HUMAN, KINASE, RIBOSOMAL, MAGNESIUM, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, PHOSPHOPROTEIN, NUCLEOTIDE-BINDING
1u59:A (ASN336) to (GLU415) CRYSTAL STRUCTURE OF THE ZAP-70 KINASE DOMAIN IN COMPLEX WITH STAUROSPORINE | TRANSFERASE
1ia8:A (GLU7) to (PHE83) THE 1.7 A CRYSTAL STRUCTURE OF HUMAN CELL CYCLE CHECKPOINT KINASE CHK1 | PROTEIN KINASE, TRANSFERASE
2wtc:A (GLU219) to (VAL300) CRYSTAL STRUCTURE OF CHK2 IN COMPLEX WITH AN INHIBITOR | TRANSFERASE, KINASE, CELL CYCLE, LI-FRAUMENI SYNDROME
4m8t:A (TYR422) to (MET493) RSK2 T493M C-TERMINAL KINASE DOMAIN IN COMPLEX WITH 3-(3-(1H-PYRAZOL- 4-YL)PHENYL)-2-CYANOACRYLAMIDE | PROTEIN KINASE, PHOSPHORYLATION, COVALENT INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4mbl:A (GLN37) to (ILE119) DISCOVERY OF PYRAZOLO[1,5A]PYRIMIDINE-BASED PIM1 INHIBITORS | KINASE, PIM1, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ajq:B (VAL35) to (GLU111) HUMAN LOK (STK10) IN COMPLEX WITH BOSUTINIB | TRANSFERASE
4mne:B (GLN456) to (GLN530) CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4mnf:B (GLN456) to (GLN530) CRYSTAL STRUCTURE OF BRAF-V600E BOUND TO GDC0879 | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, ACTIVE CONFORMATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2xbj:A (GLU219) to (VAL300) CRYSTAL STRUCTURE OF CHK2 IN COMPLEX WITH AN INHIBITOR | TRANSFERASE, DNA REPAIR, PARP
5auu:A (TYR13) to (GLU94) CRYSTAL STRUCTURE OF DAPK1 IN COMPLEX WITH LUTEOLIN. | DEATH-ASSOCIATED PROTEIN KINASE 1, SERINE/THREONINE PROTEIN KINASE, NATURAL FLAVONOID
5av0:A (TYR13) to (GLU94) CRYSTAL STRUCTURE OF DAPK1 IN COMPLEX WITH 7,3',4'- TRIHYDROXYISOFLAVONE. | DEATH-ASSOCIATED PROTEIN KINASE 1, SERINE/THREONINE PROTEIN KINASE, NATURAL FLAVONOID
2xik:A (LEU19) to (ILE94) STRUCTURE OF HUMAN YSK1 (YEAST SPS1-STE20-RELATED KINASE 1) | TRANSFERASE
2xiy:A (GLN37) to (GLU121) PROTEIN KINASE PIM-1 IN COMPLEX WITH FRAGMENT-2 FROM CRYSTALLOGRAPHIC FRAGMENT SCREEN | PHOSPHORYLATION, TRANSFERASE
2xj1:A (GLN37) to (PRO125) PROTEIN KINASE PIM-1 IN COMPLEX WITH SMALL MOLECULE INIBITOR | PHOSPHORYLATION, TRANSFERASE
2xk9:A (TYR220) to (VAL300) STRUCTURAL ANALYSIS OF CHECKPOINT KINASE 2 (CHK2) IN COMPLEX WITH INHIBITOR PV1533 | STRUCTURE-BASED DRUG DESIGN, TRANSFERASE
4n6z:A (GLN37) to (ILE119) PIM1 COMPLEXED WITH A PYRIDYLCARBOXAMIDE | KINASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3zh8:A (PHE245) to (GLU324) A NOVEL SMALL MOLECULE APKC INHIBITOR | TRANSFERASE, AGC KINASES, CELL POLARITY, CELL MIGRATION
3zh8:C (ASP244) to (GLU324) A NOVEL SMALL MOLECULE APKC INHIBITOR | TRANSFERASE, AGC KINASES, CELL POLARITY, CELL MIGRATION
2xzs:A (TYR13) to (GLU94) DEATH ASSOCIATED PROTEIN KINASE 1 RESIDUES 1-312 | TRANSFERASE, CALMODULIN, ESPRIT
2xzs:B (TYR13) to (GLU94) DEATH ASSOCIATED PROTEIN KINASE 1 RESIDUES 1-312 | TRANSFERASE, CALMODULIN, ESPRIT
2y0a:A (TYR13) to (GLU94) STRUCTURE OF DAPK1 CONSTRUCT RESIDUES 1-304 | TRANSFERASE, CALMODULIN, ESPRIT
1wmk:A (PHE12) to (GLU94) HUMAN DEATH-ASSOCIATED KINASE DRP-1, MUTANT S308D D40 | PROTEIN KINASE, AUTOINHIBITORY HELIX, TRANSFERASE
1wmk:E (PHE12) to (GLU94) HUMAN DEATH-ASSOCIATED KINASE DRP-1, MUTANT S308D D40 | PROTEIN KINASE, AUTOINHIBITORY HELIX, TRANSFERASE
1wmk:C (PHE12) to (GLU94) HUMAN DEATH-ASSOCIATED KINASE DRP-1, MUTANT S308D D40 | PROTEIN KINASE, AUTOINHIBITORY HELIX, TRANSFERASE
1wmk:B (PHE12) to (GLU94) HUMAN DEATH-ASSOCIATED KINASE DRP-1, MUTANT S308D D40 | PROTEIN KINASE, AUTOINHIBITORY HELIX, TRANSFERASE
1wmk:F (PHE12) to (GLU94) HUMAN DEATH-ASSOCIATED KINASE DRP-1, MUTANT S308D D40 | PROTEIN KINASE, AUTOINHIBITORY HELIX, TRANSFERASE
1wmk:D (PHE12) to (GLU94) HUMAN DEATH-ASSOCIATED KINASE DRP-1, MUTANT S308D D40 | PROTEIN KINASE, AUTOINHIBITORY HELIX, TRANSFERASE
1wmk:H (PHE12) to (GLU94) HUMAN DEATH-ASSOCIATED KINASE DRP-1, MUTANT S308D D40 | PROTEIN KINASE, AUTOINHIBITORY HELIX, TRANSFERASE
1wmk:G (PHE12) to (GLU94) HUMAN DEATH-ASSOCIATED KINASE DRP-1, MUTANT S308D D40 | PROTEIN KINASE, AUTOINHIBITORY HELIX, TRANSFERASE
4nif:A (GLY417) to (THR489) HETERODIMERIC STRUCTURE OF ERK2 AND RSK1 | KINASE DOMAIN, SIGNALING, SUBSTRATE KINASE BINDING, TRANSFERASE
4nif:D (GLY417) to (THR489) HETERODIMERIC STRUCTURE OF ERK2 AND RSK1 | KINASE DOMAIN, SIGNALING, SUBSTRATE KINASE BINDING, TRANSFERASE
1wvy:A (TYR12) to (GLU94) CRYSTAL STRUCTURES OF KINASE DOMAIN OF DAP KINASE IN COMPLEX WITH SMALL MOLECULAR INHIBITORS | PROTEIN KINASE, APOPTOSIS, STAUROSPORINE, TRANSFERASE
2yaa:B (TYR13) to (GLU94) CRYSTAL STRUCTURE OF THE AUTOINHIBITED FORM OF MOUSE DAPK2 IN COMPLEX WITH ATP | TRANSFERASE, APOPTOSIS
2ya9:A (TYR13) to (GLU94) CRYSTAL STRUCTURE OF THE AUTOINHIBITED FORM OF MOUSE DAPK2 | TRANSFERASE, APOPTOSIS
2ycf:A (TYR220) to (VAL300) CRYSTAL STRUCTURE OF CHECKPOINT KINASE 2 IN COMPLEX WITH INHIBITOR PV1531 | TRANSFERASE, ANTICANCER, ANTICANCER DRUG DESIGN
2ycq:A (TYR220) to (VAL300) CRYSTAL STRUCTURE OF CHECKPOINT KINASE 2 IN COMPLEX WITH INHIBITOR PV1115 | TRANSFERASE, ANTICANCER DRUG DESIGN
4o0s:A (ASP132) to (ILE209) CRYSTAL STRUCTURES OF HUMAN KINASE AURORA A | PROTEIN KINASE, TRANSFERASE
2yit:A (TYR220) to (VAL300) STRUCTURAL ANALYSIS OF CHECKPOINT KINASE 2 IN COMPLEX WITH PV1162, A NOVEL INHIBITOR | TRANSFERASE, STRUCTURE-BASED DRUG DESIGN, CELL CYCLE
3juh:A (ASP38) to (GLU114) CRYSTAL STRUCTURE OF A MUTANT OF HUMAN PROTEIN KINASE CK2ALPHA WITH ALTERED COSUBSTRATE SPECIFICITY | EUKARYOTIC PROTEIN KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
3jxw:A (GLN37) to (LEU120) DISCOVERY OF 3H-BENZO[4,5]THIENO[3,2-D]PYRIMIDIN-4-ONES AS POTENT, HIGHLY SELECTIVE AND ORALLY BIOAVAILABLE PIM KINASES INHIBITORS | PIM-1, ALTERNATIVE INITIATION, ATP-BINDING, CELL MEMBRANE, CYTOPLASM, KINASE, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3jya:A (GLN37) to (ILE119) DISCOVERY OF 3H-BENZO[4,5]THIENO[3,2-D]PYRIMIDIN-4-ONES AS POTENT, HIGHLY SELECTIVE AND ORALLY BIOAVAILABLE PIM KINASES INHIBITORS | PIM-1, ALTERNATIVE INITIATION, ATP-BINDING, CELL MEMBRANE, CYTOPLASM, KINASE, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
5cqu:A (ASP38) to (GLU114) MONOCLINIC COMPLEX STRUCTURE OF PROTEIN KINASE CK2 CATALYTIC SUBUNIT WITH A BENZOTRIAZOLE-BASED INHIBITOR GENERATED BY CLICK-CHEMISTRY | TRANSFERASE, ATP-COMPETITIVE INHIBITOR, PROTEIN KINASE CK2, CASEIN KINASE 2
5cs6:A (ASP38) to (GLU114) CRYSTAL STRUCTURE OF CK2ALPHA WITH COMPOUND 3 BOUND | TRANSFERASE, CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION
5cs6:B (ASP38) to (GLU114) CRYSTAL STRUCTURE OF CK2ALPHA WITH COMPOUND 3 BOUND | TRANSFERASE, CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION
5csh:B (ASP38) to (GLU114) CRYSTAL STRUCTURE OF CK2ALPHA WITH COMPOUND 4 BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
2o64:A (TYR38) to (ILE119) CRYSTAL STRUCTURE OF PIM1 WITH QUERCETAGETIN | PIM1, QUERCETAGETIN, TRANSFERASE
5csv:A (ASP38) to (GLU114) CRYSTAL STRUCTURE OF CK2ALPHA WITH COMPOUND 6 BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
1xqz:A (TYR38) to (GLU121) CRYSTAL STRUCTURE OF HPIM-1 KINASE AT 2.1 A RESOLUTION | PROTEIN KINASE FOLD, TRANSFERASE
5cx9:A (TYR39) to (GLU114) CRYSTAL STRUCTURE OF CK2ALPHA WITH (METHYL 4-((3-(3-CHLORO-4-(PHENYL) BENZYLAMINO)PROPYL)AMINO)-4-OXOBUTANOATE BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
1m7n:A (LYS995) to (GLU1077) CRYSTAL STRUCTURE OF UNACTIVATED APO INSULIN-LIKE GROWTH FACTOR-1 RECEPTOR KINASE DOMAIN | TRANSFERASE
3kn5:A (TYR423) to (GLU499) CRYSTAL STRUCTURE OF THE C-TERMINAL KINASE DOMAIN OF MSK1 IN COMPLEX WITH AMP-PNP | KINASE, AMP-PNP, MSK1, MSK, ATP-BINDING, METAL-BINDING, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kn5:B (TYR423) to (GLU499) CRYSTAL STRUCTURE OF THE C-TERMINAL KINASE DOMAIN OF MSK1 IN COMPLEX WITH AMP-PNP | KINASE, AMP-PNP, MSK1, MSK, ATP-BINDING, METAL-BINDING, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kn6:A (TYR423) to (GLU499) CRYSTAL STRUCTURE OF THE C-TERMINAL KINASE DOMAIN OF MSK1 | KINASE, AMP-PNP, MSK1, MSK, ATP-BINDING, METAL-BINDING, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kn6:B (TYR423) to (GLU499) CRYSTAL STRUCTURE OF THE C-TERMINAL KINASE DOMAIN OF MSK1 | KINASE, AMP-PNP, MSK1, MSK, ATP-BINDING, METAL-BINDING, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
1y8g:B (ASN52) to (MSE129) CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK2/PAR-1: INACTIVE DOUBLE MUTANT WITH SELENOMETHIONINE | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE
1yi3:A (GLN37) to (GLU121) CRYSTAL STRUCTURE OF PIM-1 BOUND TO LY294002 | PROTEIN KINASE, PI3K, TRANSFERASE
5dgz:A (GLN37) to (LEU120) DISCOVERY OF 3,5-SUBSTITUTED 6-AZAINDAZOLES AS POTENT PAN-PIM INHIBITORS | PIM-1, KINASE, ATP-COMPETITIVE, STRUCTURE-BASED DRUG DESIGN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1yxs:A (GLN37) to (LEU120) CRYSTAL STRUCTURE OF KINASE PIM1 WITH P123M MUTATION | SER/THR PROTEIN KINASE, TRANSFERASE
1yxx:A (GLN37) to (ILE119) CRYSTAL STRUCTURE OF KINASE PIM1 IN COMPLEX WITH (3E)-3-[(4- HYDROXYPHENYL)IMINO]-1H-INDOL-2(3H)-ONE | SER/THR PROTEIN KINASE, TRANSFERASE
4alw:A (GLN37) to (LEU120) BENZOFUROPYRIMIDINONE INHIBITORS OF PIM-1 | TRANSFERASE, PROTO-ONCOGENE SERINE/THREONINE-PROTEIN KINASE PIM-1
3llt:A (ALA551) to (GLU631) CRYSTAL STRUCTURE OF PF14_0431, KINASE DOMAIN. | LAMMER KINASE, MALARIA, PLASMODIUM FALCIPARUM, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE
3lm5:A (PHE31) to (GLU111) CRYSTAL STRUCTURE OF HUMAN SERINE/THREONINE KINASE 17B (STK17B) IN COMPLEX WITH QUERCETIN | STK17B, SERINE/THREONINE KINASE 17B, DRAK2, DAP KINASE RELATED APOPTOSIS-INDUCING PROTEIN KINASE 2, DEATH-ASSOCIATED PROTEIN KINASE-RELATED 2, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, APOPTOSIS, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
1zmw:B (ASN52) to (MET129) CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK2/PAR-1: T208A/S212A INACTIVE DOUBLE MUTANT | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE
1zys:A (ASP8) to (PHE83) CO-CRYSTAL STRUCTURE OF CHECKPOINT KINASE CHK1 WITH A PYRROLO-PYRIDINE INHIBITOR | CHK1; CRYSTAL STRUCTURE, SIGNALING PROTEIN, TRANSFERASE
3lzb:A (PHE688) to (GLN767) EGFR KINASE DOMAIN COMPLEXED WITH AN IMIDAZO[2,1-B]THIAZOLE INHIBITOR | EPIDERMAL GROWTH FACTOR KINASE DOMAIN, MULTITARGETED SMALL MOLECULE KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2a27:A (PHE12) to (GLU94) HUMAN DRP-1 KINASE, W305S S308A D40 MUTANT, CRYSTAL FORM WITH 8 MONOMERS IN THE ASYMMETRIC UNIT | PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE
2a27:C (PHE12) to (GLU94) HUMAN DRP-1 KINASE, W305S S308A D40 MUTANT, CRYSTAL FORM WITH 8 MONOMERS IN THE ASYMMETRIC UNIT | PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE
2a27:D (TYR13) to (GLU94) HUMAN DRP-1 KINASE, W305S S308A D40 MUTANT, CRYSTAL FORM WITH 8 MONOMERS IN THE ASYMMETRIC UNIT | PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE
2a27:E (PHE12) to (GLU94) HUMAN DRP-1 KINASE, W305S S308A D40 MUTANT, CRYSTAL FORM WITH 8 MONOMERS IN THE ASYMMETRIC UNIT | PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE
2a27:F (PHE12) to (GLU94) HUMAN DRP-1 KINASE, W305S S308A D40 MUTANT, CRYSTAL FORM WITH 8 MONOMERS IN THE ASYMMETRIC UNIT | PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE
2a27:G (TYR13) to (GLU94) HUMAN DRP-1 KINASE, W305S S308A D40 MUTANT, CRYSTAL FORM WITH 8 MONOMERS IN THE ASYMMETRIC UNIT | PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE
2a27:H (PHE12) to (GLU94) HUMAN DRP-1 KINASE, W305S S308A D40 MUTANT, CRYSTAL FORM WITH 8 MONOMERS IN THE ASYMMETRIC UNIT | PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE
2a2a:A (PHE12) to (GLU94) HIGH-RESOLUTION CRYSTALLOGRAPHIC ANALYSIS OF THE AUTOINHIBITED CONFORMATION OF A HUMAN DEATH-ASSOCIATED PROTEIN KINASE | PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE
2a2a:B (TYR13) to (GLU94) HIGH-RESOLUTION CRYSTALLOGRAPHIC ANALYSIS OF THE AUTOINHIBITED CONFORMATION OF A HUMAN DEATH-ASSOCIATED PROTEIN KINASE | PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE
2a2a:D (TYR13) to (GLU94) HIGH-RESOLUTION CRYSTALLOGRAPHIC ANALYSIS OF THE AUTOINHIBITED CONFORMATION OF A HUMAN DEATH-ASSOCIATED PROTEIN KINASE | PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE
4qmn:A (LEU23) to (GLU100) MST3 IN COMPLEX WITH BOSUTINIB | PROTEIN KINASE, MST3, STK24, STERILE 20-LIKE KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4bdc:A (GLU219) to (VAL300) FRAGMENT-BASED SCREENING IDENTIFIES A NEW AREA FOR INHIBITOR BINDING TO CHECKPOINT KINASE 2 (CHK2) | TRANSFERASE
5eol:A (GLN37) to (GLU121) CRYSTAL STRUCTURE OF HUMAN PIM-1 KINASE IN COMPLEX WITH A MACROCYCLIC QUINOXALINE-PYRROLODIHYDROPIPERIDINONE INHIBITOR | TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3bgq:A (GLN37) to (ILE119) HUMAN PIM-1 KINASE IN COMPLEX WITH AN TRIAZOLO PYRIDAZINE INHIBITOR VX2 | KINASE INHIBITOR PHOSPHORYLATION, ALTERNATIVE INITIATION, ATP-BINDING, CYTOPLASM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4bn1:A (ASP132) to (ILE209) CRYSTAL STRUCTURE OF V174M MUTANT OF AURORA-A KINASE | TRANSFERASE, PROTEIN KINASE, MITOSIS
3bqc:A (ASP38) to (GLU114) HIGH PH-VALUE CRYSTAL STRUCTURE OF EMODIN IN COMPLEX WITH THE CATALYTIC SUBUNIT OF PROTEIN KINASE CK2 | PROTEIN KINASE CK2, CASEIN KINASE 2, EUKARYOTIC PROTEIN KINASES, EMODIN, ATP-COMPETITIVE INHIBITOR, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
3bqr:A (HIS12) to (GLU94) CRYSTAL STRUCTURE OF HUMAN DEATH ASSOCIATED PROTEIN KINASE 3 (DAPK3) IN COMPLEX WITH AN IMIDAZO-PYRIDAZINE LIGAND | DEATH ASSOCIATED KINASE, DAPK3, ZIP KINASE, ZIPK, DAP KINASE 3, DAP LIKE KINASE, DLK, STRUCTURAL GENOMICS CONSORTIUM, SGC, APOPTOSIS, ATP-BINDING, CHROMATIN REGULATOR, NUCLEOTIDE-BINDING, NUCLEUS, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4btj:A (ARG57) to (GLN132) TTBK1 IN COMPLEX WITH ATP | TRANSFERASE, LIGAND COMPLEX, STRUCTURE-KINETICS RELATIONSHIP
3c4e:A (TYR38) to (ILE119) PIM-1 KINASE DOMAIN IN COMPLEX WITH 3-AMINOPHENYL-7- AZAINDOLE | PIM-1, PROTO-ONCOGENE, SERINE/THREONINE KINASE, ALTERNATIVE INITIATION, ATP-BINDING, CYTOPLASM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3c4e:B (GLN37) to (ILE119) PIM-1 KINASE DOMAIN IN COMPLEX WITH 3-AMINOPHENYL-7- AZAINDOLE | PIM-1, PROTO-ONCOGENE, SERINE/THREONINE KINASE, ALTERNATIVE INITIATION, ATP-BINDING, CYTOPLASM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4r5y:A (GLN456) to (GLN530) THE COMPLEX STRUCTURE OF BRAF V600E KINASE DOMAIN WITH A NOVEL BRAF INHIBITOR | KINASE, SIGNAL TRANSDUCTION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4bzn:A (GLN37) to (GLU121) CRYSTAL STRUCTURE OF PIM1 IN COMPLEX WITH A PYRROLO(1,2-A) PYRAZINONE INHIBITOR | PIM1, ATP BINDING, KINASE INHIBITOR, TRANSFERASE
3nr9:C (ARG162) to (GLU244) STRUCTURE OF HUMAN CDC2-LIKE KINASE 2 (CLK2) | STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, DUAL SPECIFICITY PROTEIN KINASE, TRANSFERASE
4rll:A (ASP38) to (GLU114) CRYSTAL STRUCTURE OF HUMAN CK2ALPHA IN COMPLEX WITH THE ATP- COMPETITIVE INHIBITOR 4-[(E)-(FLUOREN-9-YLIDENEHYDRAZINYLIDENE)- METHYL] BENZOATE | TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4rpv:A (GLN37) to (ILE119) CO-CRYSTAL STRUCTURE OF PIM1 WITH COMPOUND 3 | PIM1, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4rvk:A (ASP8) to (PHE83) CHK1 KINASE DOMAIN WITH DIAZACARBAZOLE COMPOUND 8: N-[3-(6-CYANO-9H- PYRROLO[2,3-B:5,4-C']DIPYRIDIN-3-YL)PHENYL]ACETAMIDE | PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3cxw:A (GLN37) to (GLU121) CRYSTAL STRUCTURE OF HUMAN PROTO-ONCOGENE SERINE THREONINE KINASE (PIM1) IN COMPLEX WITH A CONSENSUS PEPTIDE AND A BETA CARBOLINE LIGAND I | ONCOGENE, KINASE, SERINE-THREONINE, PIM1, STRUCTURAL GENOMICS CONSORTIUM, SGC, ALTERNATIVE INITIATION, ATP-BINDING, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, HOST-VIRUS INTERACTION, VIRAL IMMUNOEVASION, VIRION, VIRULENCE
3cy2:A (GLN37) to (GLU121) CRYSTAL STRUCTURE OF HUMAN PROTO-ONCOGENE SERINE THREONINE KINASE (PIM1) IN COMPLEX WITH A CONSENSUS PEPTIDE AND A BETA CARBOLINE LIGAND II | ONCOGENE, KINASE, SERINE-THREONINE, PIM1, STRUCTURAL GENOMICS CONSORTIUM, SGC, ALTERNATIVE INITIATION, ATP-BINDING, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, HOST-VIRUS INTERACTION, VIRAL IMMUNOEVASION, VIRION, VIRULENCE
4tl0:A (TYR13) to (GLU94) CRYSTAL STRUCTURE OF DEATH-ASSOCIATED PROTEIN KINASE 1 WITH A CRUCIAL PHOSPHOMIMICKING MUTATION | KINASE, DEATH-ASSOCIATED, CALMODULIN BINDING, ACTIVATION MUTANT, PHOSPHOMIMICKING MUTANT, TRANSFERASE
3dae:B (ASN54) to (ASN137) CRYSTAL STRUCTURE OF PHOSPHORYLATED SNF1 KINASE DOMAIN | KINASE, AMPK, SNF1, ATP-BINDING, CARBOHYDRATE METABOLISM, MEMBRANE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3dcv:A (TYR38) to (ILE119) CRYSTAL STRUCTURE OF HUMAN PIM1 KINASE COMPLEXED WITH 4-(4- HYDROXY-3-METHYL-PHENYL)-6-PHENYLPYRIMIDIN-2(1H)-ONE | SER/THR PROTEIN KINASE, NUCLEOTIDE-BINDING, PHSPHORYLATION, ATP-BINDING, CANCER, ONCOGENE, ALTERNATIVE INITIATION, CYTOPLASM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3ofm:A (TYR40) to (GLU115) STRUCTURE OF A HUMAN CK2ALPHA PRIME, THE PARALOG ISOFORM OF THE CATALYTIC SUBUNIT OF PROTEIN KINASE CK2 FROM HOMO SAPIENS | EUKARYPTIC PROTEIN KINASE FOLD, PHOSPHO TRANSFERASE, ATP BINDING, PHOSPHORYLATION, CYTOPLASM AND NUCLEUS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4czt:B (TYR31) to (GLU109) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF SNRK3.23 AT1G30270 | TRANSFERASE, POTASSIUM TRANSPORT, SNRK3
4czu:A (TYR31) to (THR112) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF SNRK3.23 AT1G30270 T190D MUTANT | TRANSFERASE, POTASSIUM TRANSPORT, SNRK3
4d2p:A (TYR10) to (GLU87) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT STERBASED DRUG DESIGN, KINASE
4d2p:C (TYR10) to (GLU87) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT STERBASED DRUG DESIGN, KINASE
4d2p:D (TYR10) to (GLU87) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT STERBASED DRUG DESIGN, KINASE
4d2v:C (TYR10) to (GLU87) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN
4d2w:A (GLU12) to (GLU87) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN
4d2w:B (TYR10) to (GLU87) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN
4d2w:C (GLU12) to (GLU87) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN
4txc:A (TYR13) to (GLU94) CRYSTAL STRUCTURE OF DAPK1 KINASE DOMAIN IN COMPLEX WITH A SMALL MOLECULE INHIBITOR | PROTEIN-LIGAND COMPLEX, KINASE, SMALL-MOLECULE, CATALYTIC DOMAIN, PROTEIN KINASE, PROTEIN BINDING, PROTEIN KINASE INHIBITORS, TRANSFERASE
4d9u:A (GLY421) to (GLU494) RSK2 C-TERMINAL KINASE DOMAIN, (E)-TERT-BUTYL 3-(4-AMINO-7-(3- HYDROXYPROPYL)-5-P-TOLYL-7H-PYRROLO[2,3-D]PYRIMIDIN-6-YL)-2- CYANOACRYLATE | KINASE, REVERSIBLE INHIBITOR, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4dgl:C (ASP38) to (GLU114) CRYSTAL STRUCTURE OF THE CK2 TETRAMERIC HOLOENZYME | PROTEIN KINASE, TRANSFERASE
5hie:B (GLN456) to (GLN530) BRAF KINASE DOMAIN B3AC LOOP DELETION MUTANT IN COMPLEX WITH DABRAFENIB | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4umr:A (TYR10) to (VAL85) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN
3pri:A (GLN456) to (GLN530) CRYSTAL STRUCTURE OF HUMAN B-RAF KINASE IN COMPLEX WITH A NON-OXIME FUROPYRIDINE INHIBITOR | PROTEIN KINASE, ATP-COMPETITIVE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3pri:B (GLN456) to (GLN530) CRYSTAL STRUCTURE OF HUMAN B-RAF KINASE IN COMPLEX WITH A NON-OXIME FUROPYRIDINE INHIBITOR | PROTEIN KINASE, ATP-COMPETITIVE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5iis:A (GLN37) to (ILE119) DESIGN, SYNTHESIS AND STRUCTURE ACTIVITY RELATIONSHIP OF POTENT PAN- PIM KINASE INHIBITORS DERIVED FROM THE PYRIDYL-AMIDE SCAFFOLD | PIM1, MOLONEY MURINE LEUKEMIA, PIM447, KINASE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4uv0:A (TYR13) to (GLU94) STRUCTURE OF A SEMISYNTHETIC PHOSPHORYLATED DAPK | TRANSFERASE, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NATIVE CHEMICAL LIGATION, CALMODULIN-BINDING, NUCLEOTIDE-BINDING, APOPTOSIS
5ipj:A (GLN37) to (ILE119) CRYSTAL STRUCTURE OF HUMAN PIM-1 KINASE IN COMPLEX WITH A QUINAZOLINONE-PYRROLOPYRROLONE INHIBITOR. | TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4enx:A (GLN37) to (PRO125) CRYSTAL STRUCTURE OF PIM-1 KINASE IN COMPLEX WITH INHIBITOR (2E,5Z)-2- (2-CHLOROPHENYLIMINO)-5-(4-HYDROXY-3-NITROBENZYLIDENE)THIAZOLIDIN-4- ONE | PIM-1 KINASE, TRANSFERASE-INHIBITOR COMPLEX
3q4c:A (GLN455) to (GLN529) CRYSTAL STRUCTURE OF WILD TYPE BRAF KINASE DOMAIN IN COMPLEX WITH ORGANOMETALLIC INHIBITOR CNS292 | KINASE, INHIBITOR, ONCOPROTEIN, MELANOMA, KINASE-KINASE INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3q9w:A (ASP38) to (GLU114) CRYSTAL STRUCTURE OF HUMAN CK2 ALPHA IN COMPLEX WITH EMODIN AT PH 8.5 | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r04:A (GLN37) to (GLU124) THE DISCOVERY OF NOVEL BENZOFURAN-2-CARBOXYLIC ACIDS AS POTENT PIM-1 INHIBITORS | KINAE, PIM1, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r1n:A (TYR43) to (GLU119) MK3 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fnw:A (ILE1116) to (GLU1197) CRYSTAL STRUCTURE OF THE APO F1174L ANAPLASTIC LYMPHOMA KINASE CATALYTIC DOMAIN | RECEPTOR TYROSINE KINASE, INHIBITOR, CRIZOTINIB, NEUROBLASTOMA, CD246, PHOSPHOTRANSFERASE, NPM-ALK, EML4-ALK, TRANSFERASE
4g9r:B (GLN456) to (GLN530) B-RAF V600E KINASE DOMAIN BOUND TO A TYPE II DIHYDROQUINAZOLINE INHIBITOR | INHIBITOR, TYPE II, TRANSFERASE, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2oi4:X (TYR38) to (ILE119) CRYSTAL STRUCTURE OF HUMAN PIM1 IN COMPLEX WITH FLUORINATED RUTHENIUM PYRIDOCARBAZOLE | TRANSFERASE,PIM1,KINASE, ATP-BINDING,PHOSPHORYLATION
2cn5:A (GLU219) to (GLU302) CRYSTAL STRUCTURE OF HUMAN CHK2 IN COMPLEX WITH ADP | TRANSFERASE, KINASE, KINASE DOMAIN, CHECKPOINT, CANCER, TUMOUR SUPPRESSOR, CHEK2, CHK2, CDS1, RAD53, PHOSPHORYLATION, ACTIVATION SEGMENT, LI-FRAUMENI SYNDROME, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, MAGNESIUM, METAL-BINDING, NUCLEAR PROTEIN, NUCLEOTIDE- BINDING, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE
2csn:A (HIS11) to (ASP86) BINARY COMPLEX OF CASEIN KINASE-1 WITH CKI7 | CASEIN KINASE-1, PROTEIN KINASE
2e9v:A (ASP8) to (PHE83) STRUCTURE OF H-CHK1 COMPLEXED WITH A859017 | PROTEIN-INHIBITOR COMPLEX, TRANSFERASE
4yzc:A (LYS568) to (ILE642) CRYSTAL STRUCTURE OF PIRE1ALPHA IN COMPLEX WITH STAUROSPORINE | IRE1, INHIBITOR, STAUROSPORINE, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2w4k:A (TYR13) to (GLU94) X-RAY STRUCTURE OF A DAP-KINASE 2-302 | POLYMORPHISM, PHOSPHOPROTEIN, CALMODULIN-BINDING, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, ALTERNATIVE SPLICING, DAPK, KINASE, COMPLEX, APOPTOSIS, CYTOPLASM, ANK REPEAT, CALMODULIN, TRANSFERASE, ATP-BINDING
4lm5:A (GLN37) to (ILE119) CRYSTAL STRUCTURE OF PIM1 IN COMPLEX WITH 2-{4-[(3-AMINOPROPYL) AMINO]QUINAZOLIN-2-YL}PHENOL (RESULTING FROM DISPLACEMENT OF SKF86002) | CO-CRYSTALLIZATION, SKF86002, FLUORESCENCE, INHIBITOR SCREENING, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5a6n:A (HIS12) to (GLU94) CRYSTAL STRUCTURE OF HUMAN DEATH ASSOCIATED PROTEIN KINASE 3 (DAPK3) IN COMPLEX WITH COMPOUND 2 | TRANSFERASE, DAPK3, HUMAN DEATH ASSOCIATED PROTEIN KINASE 3, DAP-LIKE KINASE, DLK, ZIPPER-INTERACTING PROTEIN KINASE, ZIP-KINASE,
5a6n:B (HIS12) to (GLU94) CRYSTAL STRUCTURE OF HUMAN DEATH ASSOCIATED PROTEIN KINASE 3 (DAPK3) IN COMPLEX WITH COMPOUND 2 | TRANSFERASE, DAPK3, HUMAN DEATH ASSOCIATED PROTEIN KINASE 3, DAP-LIKE KINASE, DLK, ZIPPER-INTERACTING PROTEIN KINASE, ZIP-KINASE,
5a6o:A (TYR13) to (GLU94) CRYSTAL STRUCTURE OF THE APO FORM OF THE UNPHOSPHORYLATED HUMAN DEATH ASSOCIATED PROTEIN KINASE 3 (DAPK3) | TRANSFERASE, DAPK3, APO, DEATH-ASSOCIATED PROTEIN KINASE 3, ZIPPER- INTERACTING PROTEIN KINASE
5a6o:B (HIS12) to (GLU94) CRYSTAL STRUCTURE OF THE APO FORM OF THE UNPHOSPHORYLATED HUMAN DEATH ASSOCIATED PROTEIN KINASE 3 (DAPK3) | TRANSFERASE, DAPK3, APO, DEATH-ASSOCIATED PROTEIN KINASE 3, ZIPPER- INTERACTING PROTEIN KINASE
4md9:G (ASP38) to (GLU114) CRYSTAL STRUCTURE OF SYMMETRIC CK2 HOLOENZYME WITH MUTATED ALPHA SUBUNIT (F121E TRUNCATED AT AA 336) | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
4md9:K (ASP38) to (GLU114) CRYSTAL STRUCTURE OF SYMMETRIC CK2 HOLOENZYME WITH MUTATED ALPHA SUBUNIT (F121E TRUNCATED AT AA 336) | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
3wil:A (GLN40) to (GLU114) CRYSTAL STRUCTURE OF THE CK2ALPHA/COMPOUND3 COMPLEX | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4mta:A (TYR38) to (GLU121) CRYSTAL STRUCTURE OF PIM-1 KINASE DOMAIN IN COMPLEX WITH 2-METHYL-5- PHENYLFURAN-3-CARBOXYLIC ACID | SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, TRANSFERASE
2xj0:A (TYR38) to (GLU121) PROTEIN KINASE PIM-1 IN COMPLEX WITH FRAGMENT-4 FROM CRYSTALLOGRAPHIC FRAGMENT SCREEN | PHOSPHORYLATION, TRANSFERASE
2y7j:A (LYS23) to (VAL106) STRUCTURE OF HUMAN PHOSPHORYLASE KINASE, GAMMA 2 | TRANSFERASE
2y7j:B (LYS23) to (VAL106) STRUCTURE OF HUMAN PHOSPHORYLASE KINASE, GAMMA 2 | TRANSFERASE
2y7j:C (LYS23) to (VAL106) STRUCTURE OF HUMAN PHOSPHORYLASE KINASE, GAMMA 2 | TRANSFERASE
2y7j:D (LYS23) to (VAL106) STRUCTURE OF HUMAN PHOSPHORYLASE KINASE, GAMMA 2 | TRANSFERASE
5c9c:B (GLN455) to (GLN529) CRYSTAL STRUCTURE OF BRAF(V600E) IN COMPLEX WITH LY3009120 COMPND | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2yir:A (GLU219) to (VAL300) STRUCTURAL ANALYSIS OF CHECKPOINT KINASE 2 IN COMPLEX WITH INHIBITOR PV1352 | TRANSFERASE, STRUCTURE-BASED DRUG DESIGN
1lr4:A (ASP38) to (GLU114) ROOM TEMPERATURE CRYSTAL STRUCTURE OF THE APO-FORM OF THE CATALYTIC SUBUNIT OF PROTEIN KINASE CK2 FROM ZEA MAYS | PROTEIN KINASE, CK2, CASEIN KINASE 2, DUAL-COSUBSTRATE SPECIFICITY, TRANSFERASE
1z9x:A (PHE12) to (GLU94) HUMAN DRP-1 KINASE, W305S S308A D40 MUTANT, CRYSTAL FORM WITH 3 MONOMERS IN THE ASYMMETRIC UNIT | PROTEIN KINASE, AUTOINHIBITORY HELIX, DIMERIZATION, TRANSFERASE
1z9x:B (PHE12) to (GLU94) HUMAN DRP-1 KINASE, W305S S308A D40 MUTANT, CRYSTAL FORM WITH 3 MONOMERS IN THE ASYMMETRIC UNIT | PROTEIN KINASE, AUTOINHIBITORY HELIX, DIMERIZATION, TRANSFERASE
1z9x:C (PHE12) to (LEU93) HUMAN DRP-1 KINASE, W305S S308A D40 MUTANT, CRYSTAL FORM WITH 3 MONOMERS IN THE ASYMMETRIC UNIT | PROTEIN KINASE, AUTOINHIBITORY HELIX, DIMERIZATION, TRANSFERASE
3lm0:A (PHE31) to (GLU111) CRYSTAL STRUCTURE OF HUMAN SERINE/THREONINE KINASE 17B (STK17B) | STK17B, SERINE/THREONINE KINASE 17B, DRAK2, DAP KINASE RELATED APOPTOSIS-INDUCING PROTEIN KINASE 2, DEATH-ASSOCIATED PROTEIN KINASE-RELATED 2, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, APOPTOSIS, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
5eym:A (ASP67) to (GLU144) MEK1 IN COMPLEX WITH BI 847325 | KINASE, INHIBITOR, TRANSFERASE
4bzo:A (GLN37) to (GLU121) CRYSTAL STRUCTURE OF PIM1 IN COMPLEX WITH A PYRROLO- PYRAZINONE INHIBITOR | PIM1, ATP BINDING, KINASE INHIBITOR, TRANSFERASE
3ckx:A (LEU8) to (GLU85) CRYSTAL STRUCTURE OF STERILE 20-LIKE KINASE 3 (MST3, STK24) IN COMPLEX WITH STAUROSPORINE | STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, PROTEIN KINASE, MST3, STK24, STERILE 20-LIKE KINASE, STAUROSPORINE, ALTERNATIVE SPLICING, ATP-BINDING, CYTOPLASM, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3nlb:A (ASP8) to (PHE83) NOVEL KINASE PROFILE HIGHLIGHTS THE TEMPORAL BASIS OF CONTEXT DEPENDENT CHECKPOINT PATHWAYS TO CELL DEATH | KINASE DOMAIN, CHECKPOINT KINASE, ATP BINDING, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4rvl:A (GLU7) to (PHE83) CHK1 KINASE DOMAIN WITH DIAZACARBAZOLE COMPOUND 7: 3-(2- HYDROXYPHENYL)-9H-PYRROLO[2,3-B:5,4-C']DIPYRIDINE-6-CARBONITRILE | PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4d0x:A (HIS848) to (GLU930) PYRROLE-3-CARBOXAMIDES AS POTENT AND SELECTIVE JAK2 INHIBITORS | TRANSFERASE, DRUG DISCOVERY, PROTEIN KINASE INHIBITORS, STRUCTURE-ACTIVITY RELATIONSHIP, POLYCYTHEMIA VERA, TUMOUR CELL PROLIFERATION INHIBITION, ANTI-CANCER AGENTS
3psb:A (GLN456) to (GLN530) FURO[2,3-C]PYRIDINE-BASED INDANONE OXIMES AS POTENT AND SELECTIVE B- RAF INHIBITORS | KINASE, ATP-BINDING, CARDIOMYOPATHY, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, ZINC-FINGER, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3q9x:B (ASP38) to (GLU114) CRYSTAL STRUCTURE OF HUMAN CK2 ALPHA IN COMPLEX WITH EMODIN AT PH 6.5 | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fsn:A (GLU7) to (PHE83) CRYSTAL STRUCTURE OF THE CHK1 | TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ft9:A (ASP8) to (PHE83) CRYSTAL STRUCTURE OF THE CHK1 | TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5jzn:A (ARG389) to (VAL464) CRYSTAL STRUCTURE OF DCLK1-KD IN COMPLEX WITH NVP-TAE684 | KINASE, DOUBLECORTIN, TRANSFERASE
5kzi:A (TYR38) to (ILE119) CRYSTAL STRUCTURE OF HUMAN PIM-1 KINASE IN COMPLEX WITH AN IMIDAZOPYRIDAZINE INHIBITOR. | TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX