4wa9:B (GLU255) to (ASN336) THE CRYSTAL STRUCTURE OF HUMAN ABL1 WILD TYPE KINASE DOMAIN IN COMPLEX WITH AXITINIB | KINASE, KINASE INHIBITOR, AXITINIB, ACTIVATION LOOP, DFG-OUT, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gt4:A (GLY485) to (HIS610) STRUCTURE OF UNLIGANDED, INACTIVE ROR2 KINASE DOMAIN | ATP BINDING, PHOSPHORYLATION, MEMBRANE, TRANSFERASE
4gt4:B (LYS489) to (HIS610) STRUCTURE OF UNLIGANDED, INACTIVE ROR2 KINASE DOMAIN | ATP BINDING, PHOSPHORYLATION, MEMBRANE, TRANSFERASE
4gt5:A (ALA527) to (HIS645) CRYSTAL STRUCTURE OF THE INACTIVE TRKA KINASE DOMAIN | TYROSINE KINASE DOMAIN, TRANSFERASE
2of2:A (PHE256) to (LEU336) CRYSTAL STRUCTURE OF FURANOPYRIMIDINE 8 BOUND TO LCK | LCK, KINASE DOMAIN, TRANSFERASE
2of4:A (PHE256) to (LEU336) CRYSTAL STRUCTURE OF FURANOPYRIMIDINE 1 BOUND TO LCK | LCK, KINASE DOMAIN, TRANSFERASE
2ofv:A (MET261) to (LEU336) CRYSTAL STRUCTURE OF AMINOQUINAZOLINE 1 BOUND TO LCK | LCK, KINASE DOMAIN, TRANSFERASE
2ofv:B (GLY257) to (LEU336) CRYSTAL STRUCTURE OF AMINOQUINAZOLINE 1 BOUND TO LCK | LCK, KINASE DOMAIN, TRANSFERASE
2og8:A (GLY257) to (LEU336) CRYSTAL STRUCTURE OF AMINOQUINAZOLINE 36 BOUND TO LCK | LCK, KINASE DOMAIN, TRANSFERASE
2og8:B (MET261) to (LEU336) CRYSTAL STRUCTURE OF AMINOQUINAZOLINE 36 BOUND TO LCK | LCK, KINASE DOMAIN, TRANSFERASE
2ogv:A (ASP608) to (ASN773) CRYSTAL STRUCTURE OF THE AUTOINHIBITED HUMAN C-FMS KINASE DOMAIN | RECEPTOR TYROSINE KINASE, MACROPHAGE COLONY STIMULATING FACTOR RECEPTOR, TRANSFERASE
4whz:A (GLY76) to (GLY184) DESIGN AND SYNTHESIS OF HIGHLY POTENT AND ISOFORM SELECTIVE JNK3 INHIBITORS: SAR STUDIES ON AMINOPYRAZOLE DERIVATIVES | JNK3, JNK2, JNK1, P38, KINASE INHIBITOR, PARKINSON DISEASE, ISOFORM- SELECTIVITY, AMINOPYRAZOLE
2oid:D (GLY198) to (HIS306) CRYSTAL STRUCTURE OF IRAK4 KINASE DOMAIN COMPLEXED WITH AMPPNP | KINASE, TRANSFERASE
3efj:B (GLY1090) to (LYS1199) STRUCTURE OF C-MET WITH PYRIMIDONE INHIBITOR 7 | C-MET, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
2onl:B (SER37) to (ASP145) CRYSTAL STRUCTURE OF THE P38A-MAPKAP KINASE 2 HETERODIMER | HETERODIMER, KINASE, NLS, NES, DOCKING GROOVE, TRANSFERASE
4wnp:A (VAL29) to (PHE118) STRUCTURE OF ULK1 BOUND TO A POTENT INHIBITOR | KINASE, AUTOPHAGY, INHIBITOR
4wo5:A (GLY469) to (SER571) CRYSTAL STRUCTURE OF A BRAF KINASE DOMAIN MONOMER | KINASE, MONOMER, INHIBITOR, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4h58:A (LYS472) to (GLU544) BRAF IN COMPLEX WITH COMPOUND 3 | PROTEIN KINASE, STRUCTURE BASED DRUG DISCOVERY, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3el8:B (GLU280) to (LEU358) CRYSTAL STRUCTURE OF C-SRC IN COMPLEX WITH PYRAZOLOPYRIMIDINE 5 | C-SRC, KINASE, PYRAZOLOPYRIMIDINE 5, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
4wsq:A (ALA58) to (HIS166) CRYSTAL STRUCTURE OF ADAPTOR PROTEIN 2 ASSOCIATED KINASE (AAK1) IN COMPLEX WITH SMALL MOLECULE INHIBITOR | KINASE, SMALL-MOLECULE, CATALYTIC DOMAIN, PROTEIN KINASE, PROTEIN BINDING, PROTEIN KINASE INHIBITORS, TRANSFERASE
4wsq:B (PHE57) to (HIS166) CRYSTAL STRUCTURE OF ADAPTOR PROTEIN 2 ASSOCIATED KINASE (AAK1) IN COMPLEX WITH SMALL MOLECULE INHIBITOR | KINASE, SMALL-MOLECULE, CATALYTIC DOMAIN, PROTEIN KINASE, PROTEIN BINDING, PROTEIN KINASE INHIBITORS, TRANSFERASE
1nw1:A (MET88) to (LEU183) CRYSTAL STRUCTURE OF CHOLINE KINASE | CHOLINE KINASE, PHOSPHOLIPID SYNTHESIS, PROTEIN KINASE FOLD, TRANSFERASE
1nw1:B (LEU89) to (LEU183) CRYSTAL STRUCTURE OF CHOLINE KINASE | CHOLINE KINASE, PHOSPHOLIPID SYNTHESIS, PROTEIN KINASE FOLD, TRANSFERASE
4wun:B (ASN506) to (LYS618) STRUCTURE OF FGFR1 IN COMPLEX WITH AZD4547 (N-{3-[2-(3,5- DIMETHOXYPHENYL)ETHYL]-1H-PYRAZOL-5-YL}-4-[(3R,5S)-3,5- DIMETHYLPIPERAZIN-1-YL]BENZAMIDE) AT 1.65 ANGSTROM | TRANSFERASE; TRANSFERASE INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ww7:A (ILE29) to (ASP156) CRYSTAL STRUCTURE OF BINARY COMPLEX BUD32-CGI121 IN COMPLEX WITH AMP | KEOPS, BINARY COMPLEX, BUD32-CGI121, TRNA T6A, TRANSFERASE
2bdj:A (GLU280) to (LEU358) SRC KINASE IN COMPLEX WITH INHIBITOR AP23464 | SRC KINASE INHIBITOR, TRANSFERASE
2bdw:A (SER25) to (GLY130) CRYSTAL STRUCTURE OF THE AUTO-INHIBITED KINASE DOMAIN OF CALCIUM/CALMODULIN ACTIVATED KINASE II | KINASE; CALMODULIN ACTIVATED, TRANSFERASE
2bdw:B (SER25) to (GLY130) CRYSTAL STRUCTURE OF THE AUTO-INHIBITED KINASE DOMAIN OF CALCIUM/CALMODULIN ACTIVATED KINASE II | KINASE; CALMODULIN ACTIVATED, TRANSFERASE
1b6c:B (GLY217) to (MET318) CRYSTAL STRUCTURE OF THE CYTOPLASMIC DOMAIN OF THE TYPE I TGF-BETA RECEPTOR IN COMPLEX WITH FKBP12 | COMPLEX (ISOMERASE/PROTEIN KINASE), RECEPTOR SERINE/THREONINE KINASE
1b6c:D (GLY217) to (MET318) CRYSTAL STRUCTURE OF THE CYTOPLASMIC DOMAIN OF THE TYPE I TGF-BETA RECEPTOR IN COMPLEX WITH FKBP12 | COMPLEX (ISOMERASE/PROTEIN KINASE), RECEPTOR SERINE/THREONINE KINASE
1b6c:F (GLY217) to (MET318) CRYSTAL STRUCTURE OF THE CYTOPLASMIC DOMAIN OF THE TYPE I TGF-BETA RECEPTOR IN COMPLEX WITH FKBP12 | COMPLEX (ISOMERASE/PROTEIN KINASE), RECEPTOR SERINE/THREONINE KINASE
1b6c:H (GLY217) to (MET318) CRYSTAL STRUCTURE OF THE CYTOPLASMIC DOMAIN OF THE TYPE I TGF-BETA RECEPTOR IN COMPLEX WITH FKBP12 | COMPLEX (ISOMERASE/PROTEIN KINASE), RECEPTOR SERINE/THREONINE KINASE
4hgt:A (ASP22) to (ASN123) CRYSTAL STRUCTURE OF CK1D WITH COMPOUND 13 | CK1D, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4hgt:B (ASP22) to (ASN123) CRYSTAL STRUCTURE OF CK1D WITH COMPOUND 13 | CK1D, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4hjo:A (VAL714) to (ARG808) CRYSTAL STRUCTURE OF THE INACTIVE EGFR TYROSINE KINASE DOMAIN WITH ERLOTINIB | INACTIVE TYROSINE KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ezr:A (GLY16) to (ARG122) CDK-2 WITH INDAZOLE INHIBITOR 17 BOUND AT ITS ACTIVE SITE | KINASE, PKC, PROTEIN KINASE, INHIBITOR, ATP-BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4hnf:A (GLY21) to (ASN123) CRYSTAL STRUCTURE OF CK1D IN COMPLEX WITH PF4800567 | CK1D, KINASE, INHIBITOR, PF4800567, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4hni:A (GLY21) to (ASN123) CRYSTAL STRUCTURE OF CK1E IN COMPLEX WITH PF4800567 | CK1E, KINASE, INHIBITOR, PF4800567, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3f3t:B (GLY279) to (LEU358) KINASE DOMAIN OF CSRC IN COMPLEX WITH INHIBITOR RL38 (TYPE III) | ALLOSTERIC, TYPE III, DFG-OUT, ALTERNATIVE SPLICING, ATP- BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3f3z:A (LYS43) to (ILE128) CRYSTAL STRUCTURE OF CRYPTOSPORIDIUM PARVUM CALCIUM DEPENDENT PROTEIN KINASE CGD7_1840 IN PRESENCE OF INDIRUBIN E804 | CALCIUM DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, SGC
3f5p:E (PRO1026) to (LYS1130) COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR | IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3f5p:F (PRO1026) to (LYS1130) COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR | IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3f5p:G (PRO1026) to (LYS1130) COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR | IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3f5p:H (PRO1026) to (LYS1130) COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR | IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3f5p:I (PRO1026) to (LYS1130) COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR | IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3f5p:L (PRO1026) to (LYS1130) COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR | IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3f5p:R (PRO1026) to (LYS1130) COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR | IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3f6x:A (GLY279) to (LEU358) C-SRC KINASE DOMAIN IN COMPLEX WITH SMALL MOLECULE INHIBITOR | KINASE, ATP-BINDING, ALTERNATIVE SPLICING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE
4hok:A (TYR24) to (ASN123) CRYSTAL STRUCTURE OF APO CK1E | CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE
4hok:C (TYR24) to (ASN123) CRYSTAL STRUCTURE OF APO CK1E | CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE
4hok:E (ILE23) to (SER121) CRYSTAL STRUCTURE OF APO CK1E | CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE
4hok:G (ASP22) to (ASN123) CRYSTAL STRUCTURE OF APO CK1E | CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE
4hok:I (GLY21) to (ASN123) CRYSTAL STRUCTURE OF APO CK1E | CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE
4hok:Q (ASP22) to (ASN123) CRYSTAL STRUCTURE OF APO CK1E | CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE
4hok:S (TYR24) to (LYS122) CRYSTAL STRUCTURE OF APO CK1E | CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE
4hok:U (TYR24) to (ASN123) CRYSTAL STRUCTURE OF APO CK1E | CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE
4x7n:A (GLY605) to (GLY932) CO-CRYSTAL STRUCTURE OF PERK BOUND TO 4-[2-AMINO-4-METHYL-3-(2- METHYLQUINOLIN-6-YL)BENZOYL]-1-METHYL-2,5-DIPHENYL-1,2-DIHYDRO-3H- PYRAZOL-3-ONE INHIBITOR | CATALYTIC DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR, COMPLEX
3faa:A (GLU218) to (HIS317) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A 2- AMINOIMIDAZOLE INHIBITOR | KINASE, TGFBETA, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3faa:B (GLY217) to (HIS317) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A 2- AMINOIMIDAZOLE INHIBITOR | KINASE, TGFBETA, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3faa:C (GLU218) to (MET318) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A 2- AMINOIMIDAZOLE INHIBITOR | KINASE, TGFBETA, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3faa:D (GLY217) to (HIS317) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A 2- AMINOIMIDAZOLE INHIBITOR | KINASE, TGFBETA, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3faa:E (GLU218) to (MET318) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A 2- AMINOIMIDAZOLE INHIBITOR | KINASE, TGFBETA, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
2buj:A (PHE31) to (GLY143) CRYSTAL STRUCTURE OF THE HUMAN SERINE-THREONINE KINASE 16 IN COMPLEX WITH STAUROSPORINE | TRANSFERASE, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, PALMITATE, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE
2buj:B (SER32) to (GLY143) CRYSTAL STRUCTURE OF THE HUMAN SERINE-THREONINE KINASE 16 IN COMPLEX WITH STAUROSPORINE | TRANSFERASE, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, PALMITATE, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE
4hvs:A (ALA606) to (ASN787) CRYSTAL STRUCTURE OF KIT KINASE DOMAIN WITH A SMALL MOLECULE INHIBITOR, PLX647 | TRANSFERASE, TYROSINE-PROTEIN KINASE, ATP-BINDING, KINASE-KINASE INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3fe3:B (ALA68) to (ARG173) CRYSTAL STRUCTURE OF THE KINASE MARK3/PAR-1: T211A-S215A DOUBLE MUTANT | SERINE/THREONINE PROTEIN KINASE; MARK;PAR-1; KIN1; UBA DOMAIN;C- TAK1;P78;MARK3, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4hys:A (GLY38) to (GLY146) CRYSTAL STRUCTURE OF JNK1 IN COMPLEX WITH JIP1 PEPTIDE AND 4-(4- INDAZOL-1-YL-PYRIMIDIN-2-YLAMINO)-CYCLOHEXAN | KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2c0i:A (MET257) to (GLN332) SRC FAMILY KINASE HCK WITH BOUND INHIBITOR A-420983 | TYROSINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHORYLATION, SH2 DOMAIN, SH3 DOMAIN
2c0i:B (MET257) to (GLN332) SRC FAMILY KINASE HCK WITH BOUND INHIBITOR A-420983 | TYROSINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHORYLATION, SH2 DOMAIN, SH3 DOMAIN
2c0o:A (MET257) to (GLN332) SRC FAMILY KINASE HCK WITH BOUND INHIBITOR A-770041 | TYROSINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHORYLATION, SH2 DOMAIN, SH3 DOMAIN
2c0o:B (MET257) to (GLN332) SRC FAMILY KINASE HCK WITH BOUND INHIBITOR A-770041 | TYROSINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHORYLATION, SH2 DOMAIN, SH3 DOMAIN
4xh0:A (TYR24) to (SER123) STRUCTURE OF C. GLABRATA HRR25 BOUND TO ADP (SO4 CONDITION) | CASEIN KINASE, MONOPOLIN, TRANSFERASE
4xhh:A (ASP22) to (GLY121) STRUCTURE OF C. GLABRATA HRR25, APO STATE | CASEIN KINASE, MONOPOLIN, TRANSFERASE
3sg8:A (ILE35) to (ILE133) CRYSTAL STRUCTURE OF AMINOGLYCOSIDE-2''-PHOSPHOTRANSFERASE TYPE IVA TOBRAMYCIN COMPLEX | ANTIBIOTIC RESISTANCE ENZYME, TRANSFERASE, AMINOGLYCOSIDE, PHOSPHORYLATION, TRANSFERASE-ANTIBIOTIC COMPLEX
3sg9:A (ILE35) to (ILE133) CRYSTAL STRUCTURE OF AMINOGLYCOSIDE-2''-PHOSPHOTRANSFERASE TYPE IVA KANAMYCIN A COMPLEX | ANTIBIOTIC RESISTANCE ENZYME, TRANSFERASE, AMINOGLYCOSIDE, PHOSPHOTRANSFERASE, TRANSFERASE-ANTIBIOTIC COMPLEX
4xhl:A (ASP22) to (ARG122) STRUCTURE OF S. CEREVISIAE HRR25 1-394 (K38R MUTANT) | CASEIN KINASE, MONOPOLIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3she:A (LEU59) to (ILE150) NOVEL ATP-COMPETITIVE MK2 INHIBITORS WITH POTENT BIOCHEMICAL AND CELL- BASED ACTIVITY THROUGHOUT THE SERIES | KINASE DOMAIN WITH BOUND INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2pyw:A (ASN48) to (SER155) STRUCTURE OF A. THALIANA 5-METHYLTHIORIBOSE KINASE IN COMPLEX WITH ADP AND MTR | 5-METHYLTHIORIBOSE KINASE, PLANT METHIONINE RECYCLING, REFOLDING, TRANSFERASE
2pyw:B (ASN48) to (SER155) STRUCTURE OF A. THALIANA 5-METHYLTHIORIBOSE KINASE IN COMPLEX WITH ADP AND MTR | 5-METHYLTHIORIBOSE KINASE, PLANT METHIONINE RECYCLING, REFOLDING, TRANSFERASE
1ckj:A (GLY24) to (ASN126) CASEIN KINASE I DELTA TRUNCATION MUTANT CONTAINING RESIDUES 1-317 COMPLEX WITH BOUND TUNGSTATE | PROTEIN KINASE, PHOSPHOTRANSFERASE
4i92:A (ASN71) to (GLY175) STRUCTURE OF THE BSK8 KINASE DOMAIN | PROTEIN KINASE, PSEUDO KINASE, CFG, ALANINE GATEKEEPER, TRANSFERASE BRASSINOSTEROID-SIGNALING, TRANSFERASE
4i93:A (ASN71) to (GLY175) STRUCTURE OF THE BSK8 KINASE DOMAIN (SEMET LABELED) | PROTEIN KINASE, PSEUDO KINASE, CFG, ALANINE GATEKEEPER, TRANSFERASE BRASSINOSTEROID-SIGNALING, SEMET DERIVATIVE, TRANSFERASE
4i93:B (PRO70) to (GLY175) STRUCTURE OF THE BSK8 KINASE DOMAIN (SEMET LABELED) | PROTEIN KINASE, PSEUDO KINASE, CFG, ALANINE GATEKEEPER, TRANSFERASE BRASSINOSTEROID-SIGNALING, SEMET DERIVATIVE, TRANSFERASE
4i94:A (PRO70) to (TRP147) STRUCTURE OF BSK8 IN COMPLEX WITH AMP-PNP | PROTEIN KINASE, PSEUDO KINASE, CFG, ALANINE GATEKEEPER, TRANSFERASE, BRASSINOSTEROID-SIGNALING, AMP-PNP, MG2+
4i94:B (PRO70) to (TRP147) STRUCTURE OF BSK8 IN COMPLEX WITH AMP-PNP | PROTEIN KINASE, PSEUDO KINASE, CFG, ALANINE GATEKEEPER, TRANSFERASE, BRASSINOSTEROID-SIGNALING, AMP-PNP, MG2+
4ieb:A (GLU64) to (LYS169) CRYSTAL STRUCTURE OF A GLY128MET MUTANT OF THE TOXOPLASMA CDPK, TGME49_101440 | CDPKS, TOXOPLASMA, KINASE, PROTIST, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4ifg:A (GLY63) to (LYS169) CRYSTAL STRUCTURE OF TGCDPK1 WITH INHIBITOR BOUND | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1p14:A (GLY1013) to (LYS1127) CRYSTAL STRUCTURE OF A CATALYTIC-LOOP MUTANT OF THE INSULIN RECEPTOR TYROSINE KINASE | RECEPTOR, TYROSINE KINASE, CATALYSIS, MUTANT, TRANSFERASE
3sv0:A (GLY21) to (SER123) CRYSTAL STRUCTURE OF CASEIN KINASE-1 LIKE PROTEIN IN PLANT | KINASE, TYPICAL KINASE DOMAIN FOLD, CYTOSOL, TRANSFERASE
3fzs:A (GLY442) to (ASN544) CRYSTAL STRUCTURE OF PYK2 COMPLEXED WITH BIRB796 | PYK2, KINASE, DFG, ALTERNATIVE SPLICING, ATP-BINDING, CELL MEMBRANE, CYTOPLASM, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TYROSINE-PROTEIN KINASE
4ih8:A (GLY63) to (LYS169) CRYSTAL STRUCTURE OF TGCDPK1 WITH INHIBITOR BOUND | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ihp:A (GLY63) to (LYS169) CRYSTAL STRUCTURE OF TGCDPK1 WITH INHIBITOR BOUND | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3sx9:A (GLY63) to (LYS169) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR, RM-1-132 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3g5d:A (GLU280) to (LEU358) KINASE DOMAIN OF CSRC IN COMPLEX WITH DASATINIB | TYPE II, DFG-OUT, TYROSINE-PROTEIN KINASE, DASATINIB, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
2cjm:A (GLY16) to (GLY98) MECHANISM OF CDK INHIBITION BY ACTIVE SITE PHOSPHORYLATION: CDK2 Y15P T160P IN COMPLEX WITH CYCLIN A STRUCTURE | PHOSPHORYLATION, NUCLEOTIDE-BINDING, MITOSIS, CELL CYCLE, REGULATION, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, TRANSFERASE, CELL DIVISION, CYCLIN-DEPENDENT KINASE, COMPLEX (TRANSFERASE/CELL DIVISION)
1dd5:A (ALA55) to (ILE182) CRYSTAL STRUCTURE OF THERMOTOGA MARITIMA RIBOSOME RECYCLING FACTOR, RRF | THREE-HELIX BUNDLE, BETA-ALPHA-BETA SANDWICH, RIBOSOME
2qg7:A (ASN122) to (ILE212) PLASMODIUM VIVAX ETHANOLAMINE KINASE PV091845 | MALARIA, ETHANOLAMINE KINASE, PV091845, SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSFERASE
2qg7:D (ILE123) to (ASP211) PLASMODIUM VIVAX ETHANOLAMINE KINASE PV091845 | MALARIA, ETHANOLAMINE KINASE, PV091845, SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSFERASE
2cke:B (PHE24) to (LYS134) HUMAN DEATH-ASSOCIATED DRP-1 KINASE IN COMPLEX WITH INHIBITOR | TRANSFERASE-INHIBITOR COMPLEX, TRANSFERASE/INHIBITOR COMPLEX, CALMODULIN-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, APOPTOSIS
2cko:A (LEU124) to (GLY237) CRYSTAL STRUCTURE OF HUMAN CHOLINE KINASE ALPHA 2 | KINASE, TRANSFERASE, CHOLINE KINASE, PHOSPHATYDILCHOLINE, ALTERNATIVE SPLICING
2cko:B (MET123) to (GLY237) CRYSTAL STRUCTURE OF HUMAN CHOLINE KINASE ALPHA 2 | KINASE, TRANSFERASE, CHOLINE KINASE, PHOSPHATYDILCHOLINE, ALTERNATIVE SPLICING
4xuf:A (ALA627) to (SER806) CRYSTAL STRUCTURE OF THE FLT3 KINASE DOMAIN BOUND TO THE INHIBITOR QUIZARTINIB (AC220) | FLT3, RECEPTOR TYROSINE KINASE, AC220, QUIZARTINIB, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
2qnj:B (PHE67) to (ARG173) KINASE AND UBIQUITIN-ASSOCIATED DOMAINS OF MARK3/PAR-1 | SERINE/THREONINE PROTEIN KINASE, UBIQUITIN-ASSOCIATED DOMAIN, MARK, PAR-1, TRANSFERASE
3geq:A (GLY279) to (LEU358) STRUCTURAL BASIS FOR THE CHEMICAL RESCUE OF SRC KINASE ACTIVITY | KINASE, CHEMICAL RESCUE, PP2, ALTERNATIVE SPLICING, ATP- BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3geq:B (GLU280) to (LEU358) STRUCTURAL BASIS FOR THE CHEMICAL RESCUE OF SRC KINASE ACTIVITY | KINASE, CHEMICAL RESCUE, PP2, ALTERNATIVE SPLICING, ATP- BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
2qr8:A (SER434) to (GLY534) 2.0A X-RAY STRUCTURE OF C-TERMINAL KINASE DOMAIN OF P90 RIBOSOMAL S6 KINASE 2 (RSK2) | KINASE DOMAIN, RSK2, AUTOINHIBITORY, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2qr7:A (SER434) to (GLY534) 2.0A X-RAY STRUCTURE OF C-TERMINAL KINASE DOMAIN OF P90 RIBOSOMAL S6 KINASE 2: SE-MET DERIVATIVE | KINASE DOMAIN, RSK2, AUTOINHIBITORY, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
1pmn:A (GLY76) to (GLY184) CRYSTAL STRUCTURE OF JNK3 IN COMPLEX WITH AN IMIDAZOLE- PYRIMIDINE INHIBITOR | MAP KINASE, APOPTOSIS, INHIBITION, TRANSFERASE
3ggf:A (GLY36) to (GLY114) CRYSTAL STRUCTURE OF HUMAN SERINE/THREONINE-PROTEIN KINASE MST4 IN COMPLEX WITH AN QUINAZOLIN | SERINE/THREONINE-PROTEIN KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, APOPTOSIS, ATP-BINDING, GOLGI APPARATUS, KINASE, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, TRANSFERASE
4iw0:A (ALA72) to (ALA215) CRYSTAL STRUCTURE AND MECHANISM OF ACTIVATION OF TBK1 | KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4y12:A (GLY163) to (GLY271) CRYSTAL STRUCTURE OF THE S/T PROTEIN KINASE PKNG FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH AGS | S/T PROTEIN KINASE, PKNG, TRANSFERASE
4y46:A (GLY76) to (GLY184) PYRIDOPYRIMIDINONE DERIVATIVES AS POTENT AND SELECTIVE C-JUN N- TERMINAL KINASE (JNK) INHIBITORS | JNK, MAP KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2r2p:A (GLY692) to (GLY795) KINASE DOMAIN OF HUMAN EPHRIN TYPE-A RECEPTOR 5 (EPHA5) | ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, RECEPTOR, SIGNAL, TRANSFERASE, PHOSPHORYLATION, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE, ALTERNATIVE SPLICING, GLYCOPROTEIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
3tcp:A (VAL601) to (ASN718) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE-PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR UNC569 | TYROSINE KINASE, ACUTE LYMPHOBLASTIC LEUKEMIA, RATIONAL STRUCTURE- BASED DRUG DESIGN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2r4b:A (THR743) to (ARG838) ERBB4 KINASE DOMAIN COMPLEXED WITH A THIENOPYRIMIDINE INHIBITOR | ERB, KINASE, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE
2r4b:B (THR743) to (ARG838) ERBB4 KINASE DOMAIN COMPLEXED WITH A THIENOPYRIMIDINE INHIBITOR | ERB, KINASE, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE
4j96:B (ALA498) to (LYS621) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC GAIN-OF-FUNCTION K659M MUTATION IDENTIFIED IN CERVICAL CANCER. | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, RECEPTOR TYROSINE KINASE, ATP BINDING, TRANSFERASE
4y8d:A (PHE51) to (GLY141) CRYSTAL STRUCTURE OF CYCLIN-G ASSOCIATED KINASE (GAK) COMPLEXED WITH SELECTIVE 12I INHIBITOR | TRANSFERASE, KINASE, NANOBODY, INHIBITOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
4y8d:B (PHE51) to (GLY141) CRYSTAL STRUCTURE OF CYCLIN-G ASSOCIATED KINASE (GAK) COMPLEXED WITH SELECTIVE 12I INHIBITOR | TRANSFERASE, KINASE, NANOBODY, INHIBITOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
4jbv:A (GLY63) to (LYS169) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1268 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jg7:A (SER434) to (GLY534) STRUCTURE OF RSK2 CTD BOUND TO 3-(3-(1H-PYRROLO[2,3-B]PYRIDINE-3- CARBONYL)PHENYL)-2-CYANOACRYLAMIDE | PROTEIN KINASE, PHOSPHORYLATION, COVALENT INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4yc8:B (GLU255) to (ASN336) C-HELIX-OUT BINDING OF DASATINIB ANALOG TO C-ABL KINASE | KINASE, C-HELIX-OUT, TRANSFERASE
4jjr:A (GLY21) to (ASN123) A P21 CRYSTAL FORM OF MAMMALIAN CASEIN KINASE 1 DELTA | CK1D, KINASE, CASEIN KINASE, TRANSFERASE
2rei:A (GLU646) to (GLY753) KINASE DOMAIN OF HUMAN EPHRIN TYPE-A RECEPTOR 7 (EPHA7) | ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, RECEPTOR, SIGNAL, TRANSFERASE, PHOSPHORYLATION, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE, ALTERNATIVE SPLICING, GLYCOPROTEIN, STRUCTURAL GENOMICS CONSORTIUM, SGC, POLYMORPHISM
2rfn:A (GLY1102) to (LYS1199) X-RAY STRUCTURE OF C-MET WITH INHIBITOR. | C-MET HGF RECEPTOR TYROSINE KINSE KINASE DOMAIN, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, PROTO- ONCOGENE, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3ttj:A (GLY76) to (GLY184) CRYSTAL STRUCTURE OF JNK3 COMPLEXED WITH CC-359, A JNK INHIBITOR FOR THE PREVENTION OF ISCHEMIA-REPERFUSION INJURY | MITOGEN-ACTIVATED PROTEIN KINASE 10, JNK3, PROTEIN KINASE INHIBITORS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yff:A (GLY480) to (LYS555) TNNI3K COMPLEXED WITH INHIBITOR 2 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yff:B (GLY480) to (LYS555) TNNI3K COMPLEXED WITH INHIBITOR 2 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yff:C (GLY480) to (LYS555) TNNI3K COMPLEXED WITH INHIBITOR 2 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yff:D (GLY480) to (LYS555) TNNI3K COMPLEXED WITH INHIBITOR 2 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yfi:A (GLY480) to (LYS555) TNNI3K COMPLEXED WITH INHIBITOR 1 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yfi:C (GLY480) to (LYS555) TNNI3K COMPLEXED WITH INHIBITOR 1 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yfi:D (GLY475) to (LYS555) TNNI3K COMPLEXED WITH INHIBITOR 1 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2e2b:A (GLU255) to (ASN336) CRYSTAL STRUCTURE OF THE C-ABL KINASE DOMAIN IN COMPLEX WITH INNO-406 | C-ABL, KINASE, INNO-406, TRANSFERASE
2e2b:B (GLU255) to (ASN336) CRYSTAL STRUCTURE OF THE C-ABL KINASE DOMAIN IN COMPLEX WITH INNO-406 | C-ABL, KINASE, INNO-406, TRANSFERASE
3tv4:A (THR470) to (GLU545) HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH AN BROMOPYRIDINE BENZAMIDE INHIBITOR | KINASE, KINASE INHIBITOR, TRANSFERASE, RAS, C-RAF, MEK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3tv4:B (PHE468) to (GLU545) HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH AN BROMOPYRIDINE BENZAMIDE INHIBITOR | KINASE, KINASE INHIBITOR, TRANSFERASE, RAS, C-RAF, MEK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3tv6:A (LYS473) to (GLU545) HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH A METHOXYPYRAZOLOPYRIDINYL BENZAMIDE INHIBITOR | B-RAF, KINASE, KINASE INHIBITOR, TRANSFERASE, C-RAF, RAS, MEK, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1qpc:A (PHE256) to (LEU336) STRUCTURAL ANALYSIS OF THE LYMPHOCYTE-SPECIFIC KINASE LCK IN COMPLEX WITH NON-SELECTIVE AND SRC FAMILY SELECTIVE KINASE INHIBITORS | ALPHA BETA FOLD, TRANSFERASE
1qpj:A (GLU258) to (LEU336) CRYSTAL STRUCTURE OF THE LYMPHOCYTE-SPECIFIC KINASE LCK IN COMPLEX WITH STAUROSPORINE. | ALPHA BETA FOLD, TRANSFERASE
4yht:A (LYS472) to (GLU544) BRAF COMPLEXED WITH AN INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yht:B (LYS472) to (GLU544) BRAF COMPLEXED WITH AN INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2uv2:A (GLY46) to (LYS150) CRYSTAL STRUCTURE OF HUMAN STE20-LIKE KINASE BOUND TO 4-(4-( 5-CYCLOPROPYL-1H-PYRAZOL-3-YLAMINO)-QUINAZOLIN-2-YLAMINO)- PHENYL)-ACETONITRILE | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, MUSCLE DEVELOPMENT, KINASE, APOPTOSIS, GERMINAL CENTRE KINASE, SERINE- THREONINE KINASE 2, NUCLEOTIDE-BINDING, SERINE-THREONINE-PROTEIN KINASE
4yjn:A (GLY63) to (LYS169) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1639 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jt3:A (SER537) to (GLY642) CRYSTAL STRUCTURE OF TTK KINASE DOMAIN WITH AN INHIBITOR: 400740 | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3h9r:A (GLY220) to (ILE321) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF TYPE I ACTIVIN RECEPTOR (ACVR1) IN COMPLEX WITH FKBP12 AND DORSOMORPHIN | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP- BINDING, DISEASE MUTATION, GLYCOPROTEIN, KINASE, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE, ISOMERASE, ROTAMASE, ISOMERASE-PROTEIN KINASE COMPLEX
4jvg:A (LYS473) to (SER544) B-RAF KINASE IN COMPLEX WITH BIRB796 | KINASE, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jvg:D (LYS473) to (SER544) B-RAF KINASE IN COMPLEX WITH BIRB796 | KINASE, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1r0e:A (GLY68) to (GLY176) GLYCOGEN SYNTHASE KINASE-3 BETA IN COMPLEX WITH 3-INDOLYL-4- ARYLMALEIMIDE INHIBITOR | SER/THR PROTEIN KINASE, TRANSFERASE
2uzb:A (GLY16) to (GLN113) CRYSTAL STRUCTURE OF HUMAN CDK2 COMPLEXED WITH A THIAZOLIDINONE INHIBITOR | TRANSFERASE, ATP-BINDING, PHOSPHORYLATION, CDK2, KINASE, CYCLIN, MITOSIS, CELL CYCLE, CELL DIVISION, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, THIAZOLIDINONE LIGAND
4yo6:A (GLY198) to (HIS306) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yo6:B (GLY198) to (HIS306) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4k11:A (GLY279) to (LEU358) THE STRUCTURE OF 1NA IN COMPLEX WITH SRC T338G | 1NA, C-SRC, KINASE, PHOSPHORYLATION, TRANSFERASE
4yom:B (GLY32) to (SER137) STRUCTURE OF SAD KINASE | KINASE DOMAIN, UBA DOMAIN, KA1 DOMAIN, TRANSFERASE
3uc4:A (VAL34) to (MET134) THE CRYSTAL STRUCTURE OF SNF1-RELATED KINASE 2.6 | SNRK2.6, KINASE, ABA SIGNALING, TRANSFERASE
4yps:A (ALA527) to (HIS645) (R)-2-PHENYLPYRROLIDINE SUBSTITUTE IMIDAZOPYRIDAZINES: A NEW CLASS OF POTENT AND SELECTIVE PAN-TRK INHIBITORS | TRKA, KINASE, ONCOLOGY, INHIBITOR COMPLEX., TRANSFEASE-TRANSFERASE INHIBITOR COMPLEX
3ue4:B (GLU255) to (ASN336) STRUCTURAL AND SPECTROSCOPIC ANALYSIS OF THE KINASE INHIBITOR BOSUTINIB BINDING TO THE ABL TYROSINE KINASE DOMAIN | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2exc:X (GLY76) to (GLY184) INHIBITOR COMPLEX OF JNK3 | ENZYME-INHIBITOR COMPLEX, KINASE INHIBITOR, TRANSFERASE
1fpu:B (GLU255) to (SER336) CRYSTAL STRUCTURE OF ABL KINASE DOMAIN IN COMPLEX WITH A SMALL MOLECULE INHIBITOR | KINASE, KINASE INHIBITOR, STI-571, ACTIVATION LOOP, TRANSFERASE
1rjb:A (ALA627) to (SER806) CRYSTAL STRUCTURE OF FLT3 | KINASE, STRUCTURE, AUTOINHIBITION, JUXTAMEMBRANE DOMAIN, TRANSFERASE
2f4j:A (GLU255) to (ASN336) STRUCTURE OF THE KINASE DOMAIN OF AN IMATINIB-RESISTANT ABL MUTANT IN COMPLEX WITH THE AURORA KINASE INHIBITOR VX-680 | KINASE, KINASE INHIBITOR, ABL, TRANSFERASE
4kaw:X (ALA55) to (GLU184) CRYSTAL STRUCTURE OF RIBOSOME RECYCLING FACTOR MUTANT R39G FROM MYCOBACTERIUM TUBERCULOSIS | RIBOSOME RECYCLING, TRANSLATION, EUBACTERIA, DISASSEMBLY, POST- TERMINATION COMPLEX, RIBOSOME, ELONGATION FACTOR G, BACTERIAL CYTOSOL
4kb4:A (ILE57) to (LEU183) CRYSTAL STRUCTURE OF RIBOSOME RECYCLING FACTOR MUTANT R31A FROM MYCOBACTERIUM TUBERCULOSIS | RIBOSOME RECYCLING, POST-TERMINATION COMPLEX, TRANSLATION, ELONGATION FACTOR G, BACTERIAL CYTOSOL
4kb8:B (GLY21) to (ASN123) CK1D IN COMPLEX WITH 1-{4-[3-(4-FLUOROPHENYL)-1-METHYL-1H-PYRAZOL-4- YL]PYRIDIN-2-YL}-N-METHYLMETHANAMINE LIGAND | SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4kb8:D (ASP22) to (ASN123) CK1D IN COMPLEX WITH 1-{4-[3-(4-FLUOROPHENYL)-1-METHYL-1H-PYRAZOL-4- YL]PYRIDIN-2-YL}-N-METHYLMETHANAMINE LIGAND | SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4kba:B (GLY21) to (ASN123) CK1D IN COMPLEX WITH 9-[3-(4-FLUOROPHENYL)-1-METHYL-1H-PYRAZOL-4-YL]- 2,3,4,5-TETRAHYDROPYRIDO[2,3-F][1,4]OXAZEPINE INHIBITOR | SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4kba:D (ASP22) to (ASN123) CK1D IN COMPLEX WITH 9-[3-(4-FLUOROPHENYL)-1-METHYL-1H-PYRAZOL-4-YL]- 2,3,4,5-TETRAHYDROPYRIDO[2,3-F][1,4]OXAZEPINE INHIBITOR | SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4kbk:A (GLY21) to (ASN123) CK1D IN COMPLEX WITH (3S)-3-{4-[3-(4-FLUOROPHENYL)-1-METHYL-1H- PYRAZOL-4-YL]PYRIDIN-2-YL}MORPHOLINE INHIBITOR | SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4kbk:D (ASP22) to (ASN123) CK1D IN COMPLEX WITH (3S)-3-{4-[3-(4-FLUOROPHENYL)-1-METHYL-1H- PYRAZOL-4-YL]PYRIDIN-2-YL}MORPHOLINE INHIBITOR | SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yz9:C (ARG588) to (ASN683) CRYSTAL STRUCTURE OF HUMAN PHOSPHORYLATED IRE1ALPHA IN COMPLEX WITH A TYPE III KINASE INHIBITOR (GSK2850163A) | ACTIVE, INHIBITOR, COMPLEX, IRE1, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2fb8:B (GLY469) to (GLU545) STRUCTURE OF THE B-RAF KINASE DOMAIN BOUND TO SB-590885 | KINASE DOMAIN, TRANSFERASE
3uqc:D (GLN45) to (GLY145) STRUCTURE OF THE INTRACELLULAR KINASE HOMOLOGY DOMAIN OF RV3910 AT 2.2 A RESOLUTION | STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, KINASE FOLD, FHAA, TRANSFERASE
1gag:A (GLY1013) to (LYS1126) CRYSTAL STRUCTURE OF THE INSULIN RECEPTOR KINASE IN COMPLEX WITH A BISUBSTRATE INHIBITOR | PROTEIN KINASE INHIBITOR, TYROSINE KINASE, TRANSFERASE, SIGNALING PROTEIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4z7h:A (ARG588) to (LEU661) CRYSTAL STRUCTURE OF HUMAN IRE1 CYTOPLASMIC KINASE-RNASE REGION - COMPLEX WITH IMIDAZOPYRIDINE COMPOUND 3 | TRANSFERASE, KINASE, RNASE, UNFOLDED PROTEIN RESPONSE
4z7h:B (ARG588) to (LEU661) CRYSTAL STRUCTURE OF HUMAN IRE1 CYTOPLASMIC KINASE-RNASE REGION - COMPLEX WITH IMIDAZOPYRIDINE COMPOUND 3 | TRANSFERASE, KINASE, RNASE, UNFOLDED PROTEIN RESPONSE
4z9l:A (GLY76) to (GLY184) THE STRUCTURE OF JNK3 IN COMPLEX WITH AN IMIDAZOLE-PYRIMIDINE INHIBITOR | MAP KINASE, APOPTOSIS, INHIBITION, TRANSFERASE
3uyt:A (ASP22) to (ASN123) CRYSTAL STRUCTURE OF CK1D WITH PF670462 FROM P1 CRYSTAL FORM | CK1D, KINASE, INHIBITOR, PF670462, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uyt:B (ASP22) to (ASN123) CRYSTAL STRUCTURE OF CK1D WITH PF670462 FROM P1 CRYSTAL FORM | CK1D, KINASE, INHIBITOR, PF670462, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uyt:C (GLY21) to (ASN123) CRYSTAL STRUCTURE OF CK1D WITH PF670462 FROM P1 CRYSTAL FORM | CK1D, KINASE, INHIBITOR, PF670462, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3hx4:A (GLU64) to (ILE154) CRYSTAL STRUCTURE OF CDPK1 OF TOXOPLASMA GONDII, TGME49_101440, IN PRESENCE OF CALCIUM | CDPKS, TOXOPLASMA, KINASE, PROTIST, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3hyh:A (LYS70) to (LYS172) CRYSTAL STRUCTURE OF THE PROTEIN KINASE DOMAIN OF YEAST AMP-ACTIVATED PROTEIN KINASE SNF1 | KINASE DOMAIN, TRANSFERASE, ATP-BINDING, CARBOHYDRATE METABOLISM, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE
2g1t:A (GLY254) to (ASN336) A SRC-LIKE INACTIVE CONFORMATION IN THE ABL TYROSINE KINASE DOMAIN | KINASE, TRANSFERASE
2g1t:B (GLY254) to (ASN336) A SRC-LIKE INACTIVE CONFORMATION IN THE ABL TYROSINE KINASE DOMAIN | KINASE, TRANSFERASE
2g1t:D (GLU255) to (ASN336) A SRC-LIKE INACTIVE CONFORMATION IN THE ABL TYROSINE KINASE DOMAIN | KINASE, TRANSFERASE
2g2h:B (GLU274) to (ASN355) A SRC-LIKE INACTIVE CONFORMATION IN THE ABL TYROSINE KINASE DOMAIN | PROTEIN KINASE, TRANSFERASE
4ksp:A (GLY468) to (GLU544) CRYSTAL STRUCTURE OF HUMAN B-RAF BOUND TO A DFG-OUT INHIBITOR TAK-632 | HUMAN SERINE/THERONINE PROTEIN KINASE, KINASE DRUG COMPLEX,, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ksp:B (LYS472) to (GLU544) CRYSTAL STRUCTURE OF HUMAN B-RAF BOUND TO A DFG-OUT INHIBITOR TAK-632 | HUMAN SERINE/THERONINE PROTEIN KINASE, KINASE DRUG COMPLEX,, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1snu:B (GLY375) to (CYS477) CRYSTAL STRUCTURE OF THE UNPHOSPHORYLATED INTERLEUKIN-2 TYROSINE KINASE CATALYTIC DOMAIN | PROTEIN KINASE, IMMUNOLOGY, TRANSFERASE
3i5n:A (HIS1094) to (LYS1199) CRYSTAL STRUCTURE OF C-MET WITH TRIAZOLOPYRIDAZINE INHIBITOR 13 | PROTO-ONCOGENE, RTK, RECEPTOR TYROSINE KINASE, SCATTER FACTOR RECEPTOR, HGF/SF, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
1gup:A (ALA89) to (ASP208) STRUCTURE OF NUCLEOTIDYLTRANSFERASE COMPLEXED WITH UDP- GALACTOSE | TRANSFERASE, NUCLEOTIDYLTRANSFERASE, GALACTOSE METABOLISM
1guq:D (PRO87) to (ASP208) STRUCTURE OF NUCLEOTIDYLTRANSFERASE COMPLEXED WITH UDP-GLUCOSE | TRANSFERASE, NUCLEOTIDYLTRANSFERASE, GALACTOSE METABOLISM
3i7c:A (GLY63) to (LYS169) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR NA-PP2 | PROTEIN KINASE, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, TRANSFERASE
3i81:A (PRO996) to (LYS1100) CRYSTAL STRUCTURE OF INSULIN-LIKE GROWTH FACTOR 1 RECEPTOR (IGF-1R-WT) COMPLEX WITH BMS-754807 [1-(4-((5-CYCLOPROPYL- 1H-PYRAZOL-3-YL)AMINO)PYRROLO[2,1-F][1,2,4]TRIAZIN-2-YL)-N- (6-FLUORO-3-PYRIDINYL)-2-METHYL-L-PROLINAMIDE] | HORMONE/GROWTH FACTOR, IGF-1R, KINASE DOMAIN, ATP-BINDING, DISEASE MUTATION, DISULFIDE BOND, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
4l01:A (SER599) to (ASP709) CRYSTAL STRUCTURE OF THE V658F APO JAK1 PSEUDOKINASE DOMAIN | KINASE DOMAIN FOLD, REGULATORY, TRANSFERASE
4zly:A (GLY414) to (GLN516) CRYSTAL STRUCTURE OF BRUTON'S TYROSINE KINASE BOUND TO A CINNOLINE FRAGMENT | CYTOPLASMIC TYROSINE KINASE, TRANSCRIPTIONAL REGULATION, NUCLEAR FACTOR-KAPPAB, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3idp:A (LYS473) to (GLU545) B-RAF V600E KINASE DOMAIN IN COMPLEX WITH AN AMINOISOQUINOLINE INHIBITOR | ONCOGENE, ATP-BINDING, DFG-OUT, TRANSFERASE, CARDIOMYOPATHY, DISEASE MUTATION, KINASE, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, ZINC-FINGER
3idp:B (LYS473) to (GLU545) B-RAF V600E KINASE DOMAIN IN COMPLEX WITH AN AMINOISOQUINOLINE INHIBITOR | ONCOGENE, ATP-BINDING, DFG-OUT, TRANSFERASE, CARDIOMYOPATHY, DISEASE MUTATION, KINASE, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, ZINC-FINGER
4l68:B (GLY319) to (HIS418) STRUCTURE OF THE PSEDUDOKINASE DOMAIN OF BIR2, AN IMMUNE REGULATOR OF THE RLK/PELLE FAMILY | PSEUDOKINASE, NEGATIVE IMMUNE REGULATOR, SIGNALING PROTEIN
3iec:A (ALA65) to (PHE170) HELICOBACTER PYLORI CAGA INHIBITS PAR1/MARK FAMILY KINASES BY MIMICKING HOST SUBSTRATES | PROTEIN-PROTEIN COMPLEX, KINASE, VIRULENCE FACTOR, ALTERNATIVE PROMOTER USAGE, ATP-BINDING, CELL MEMBRANE, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, MAGNESIUM, MEMBRANE, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, SIGNALING PROTEIN-TOXIN COMPLEX
3iec:B (ALA65) to (PHE170) HELICOBACTER PYLORI CAGA INHIBITS PAR1/MARK FAMILY KINASES BY MIMICKING HOST SUBSTRATES | PROTEIN-PROTEIN COMPLEX, KINASE, VIRULENCE FACTOR, ALTERNATIVE PROMOTER USAGE, ATP-BINDING, CELL MEMBRANE, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, MAGNESIUM, MEMBRANE, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, SIGNALING PROTEIN-TOXIN COMPLEX
3iec:C (ALA65) to (PHE170) HELICOBACTER PYLORI CAGA INHIBITS PAR1/MARK FAMILY KINASES BY MIMICKING HOST SUBSTRATES | PROTEIN-PROTEIN COMPLEX, KINASE, VIRULENCE FACTOR, ALTERNATIVE PROMOTER USAGE, ATP-BINDING, CELL MEMBRANE, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, MAGNESIUM, MEMBRANE, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, SIGNALING PROTEIN-TOXIN COMPLEX
3iec:D (LYS66) to (LYS155) HELICOBACTER PYLORI CAGA INHIBITS PAR1/MARK FAMILY KINASES BY MIMICKING HOST SUBSTRATES | PROTEIN-PROTEIN COMPLEX, KINASE, VIRULENCE FACTOR, ALTERNATIVE PROMOTER USAGE, ATP-BINDING, CELL MEMBRANE, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, MAGNESIUM, MEMBRANE, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, SIGNALING PROTEIN-TOXIN COMPLEX
4l7f:A (GLY38) to (SER144) CO-CRYSTAL STRUCTURE OF JNK1 AND AX13587 | PROTEIN KINASE FOLD, PROTEIN KINASE, JUN-C, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3igo:A (LEU91) to (ILE178) CRYSTAL STRUCTURE OF CRYPTOSPORIDIUM PARVUM CDPK1, CGD3_920 | PARASITE, KINASE, CDPK, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
4zog:B (GLU255) to (ASN336) VX-680/MK-0457 BINDS TO HUMAN ABL1 ALSO IN INACTIVE DFG CONFORMATIONS. | KINASE, TRANSFERASE, ABL1, DFG CONFORMATIONS
4zp5:A (TYR40) to (HIS148) MAP4K4 IN COMPLEX WITH INHIBITOR | KINASE, INHIBITOR, TRANSFERASE-INHIBITOR COMPLEX
2gs7:B (LYS713) to (ARG808) CRYSTAL STRUCTURE OF THE INACTIVE EGFR KINASE DOMAIN IN COMPLEX WITH AMP-PNP | EGFR, KINASE, INACTIVE, AMP-PNP, TRANSFERASE
3ii5:A (GLY468) to (GLU544) THE COMPLEX OF WILD-TYPE B-RAF WITH PYRAZOLO PYRIMIDINE INHIBITOR | B-RAF, KINASE, PROTEIN-INHIBITOR COMPLEX, ACETYLATION, ATP- BINDING, CARDIOMYOPATHY, CYTOPLASM, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ZINC, ZINC- FINGER
3ii5:B (LYS472) to (GLU544) THE COMPLEX OF WILD-TYPE B-RAF WITH PYRAZOLO PYRIMIDINE INHIBITOR | B-RAF, KINASE, PROTEIN-INHIBITOR COMPLEX, ACETYLATION, ATP- BINDING, CARDIOMYOPATHY, CYTOPLASM, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ZINC, ZINC- FINGER
3ik3:A (GLU255) to (SER336) AP24534, A PAN-BCR-ABL INHIBITOR FOR CHRONIC MYELOID LEUKEMIA, POTENTLY INHIBITS THE T315I MUTANT AND OVERCOMES MUTATION-BASED RESISTANCE | BCR-ABL, CML, T315I, INHIBITOR, MUTATION, DRUG RESISTANCE, ALTERNATIVE SPLICING, ATP-BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3ik3:B (GLU255) to (SER336) AP24534, A PAN-BCR-ABL INHIBITOR FOR CHRONIC MYELOID LEUKEMIA, POTENTLY INHIBITS THE T315I MUTANT AND OVERCOMES MUTATION-BASED RESISTANCE | BCR-ABL, CML, T315I, INHIBITOR, MUTATION, DRUG RESISTANCE, ALTERNATIVE SPLICING, ATP-BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
4ztl:A (PHE197) to (HIS306) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ztl:B (GLY198) to (HIS306) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ztl:C (GLY198) to (HIS306) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ztl:D (GLY198) to (HIS306) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ztm:B (GLY198) to (HIS306) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ztn:A (GLY198) to (HIS306) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ztn:B (GLY198) to (HIS306) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4lgd:B (GLY39) to (ARG141) STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5 | HIPPO, MST AUTOACTIVATION, RASSF, SARAH DOMAIN, DIMERIZATION, SIGNALING PROTEIN
3is5:D (LEU151) to (HIS255) CRYSTAL STRUCTURE OF CDPK KINASE DOMAIN FROM TOXOPLASMA GONDII, TGME49_018720 | TOXOPLASMA GONDII, CDPK, STRUCTURAL GENOMICS, PARASITOLOGY, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3is5:E (LEU151) to (HIS255) CRYSTAL STRUCTURE OF CDPK KINASE DOMAIN FROM TOXOPLASMA GONDII, TGME49_018720 | TOXOPLASMA GONDII, CDPK, STRUCTURAL GENOMICS, PARASITOLOGY, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2hak:C (ALA65) to (LYS169) CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1 | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE
2hak:H (PHE64) to (LYS169) CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1 | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE
2hiw:A (GLU276) to (ASN354) CRYSTAL STRUCTURE OF INACTIVE CONFORMATION ABL KINASE CATALYTIC DOMAIN COMPLEXED WITH TYPE II INHIBITOR | KINASE DOMAIN, TRANSFERASE
3vrz:B (MET283) to (GLN358) CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRROLO-PYRIMIDINE INHIBITOR 1-[4-(4-AMINO-7-CYCLOPENTYL-7H-PYRROLO[2,3-D]PYRIMIDIN-5-YL)PHENYL]- 3-BENZYLUREA | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3vs1:A (MET283) to (GLN358) CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRROLO-PYRIMIDINE INHIBITOR 1-[4-(4-AMINO-7-CYCLOPENTYL-7H-PYRROLO[2,3-D]PYRIMIDIN-5-YL)PHENYL]- 3-PHENYLUREA | TYROSINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3vs3:A (MET283) to (GLN358) CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRROLO-PYRIMIDINE INHIBITOR 7-[TRANS-4-(4-METHYLPIPERAZIN-1-YL)CYCLOHEXYL]-5-(4-PHENOXYPHENYL)- 7H-PYRROLO[2,3-D]PYRIMIDIN-4-AMINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2hk5:A (MET261) to (GLN336) HCK KINASE IN COMPLEX WITH LCK TARGETTED INHIBITOR PG-1009247 | HCK, SRC-FAMILY, KINASE DOMAIN, TRANSFERASE
3vs4:A (MET283) to (GLN358) CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRROLO-PYRIMIDINE INHIBITOR 5-(4-PHENOXYPHENYL)-7-(TETRAHYDRO-2H-PYRAN-4-YL)-7H-PYRROLO[2,3- D]PYRIMIDIN-4-AMINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3vs7:B (MET283) to (GLN358) CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRAZOLO-PYRIMIDINE INHIBITOR 1-CYCLOPENTYL-3-(1H-PYRROLO[2,3-B]PYRIDIN-5-YL)-1H- PYRAZOLO[3,4-D]PYRIMIDIN-4-AMINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1hxp:A (PRO87) to (ASP208) NUCLEOTIDE TRANSFERASE | METALLOENZYME, GALACTOSEMIA, NUCLEOTIDYL TRANSFERASE, COMPLEX (SERINE PROTEASE/INHIBITOR)
3vum:A (GLY38) to (GLY146) CRYSTAL STRUCTURE OF A CYSTEINE-DEFICIENT MUTANT M7 IN MAP KINASE JNK1 | TRANSCRIPTION, PHOSPHORYLATION, ATP BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3vwa:B (ASP34) to (GLY125) CRYSTAL STRUCTURE OF CEX1P | TRNA, NUCLEAR EXPORT, HEAT REPEAT, KINASE LIKE DOMAIN, HYDROLASE
4lrm:D (GLY729) to (ASN811) EGFR D770_N771INSNPG IN COMPLEX WITH PD168393 | EGFR, KINASE, PD168393, 34-JAB, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1u5r:B (GLY40) to (ASN146) CRYSTAL STRUCTURE OF THE TAO2 KINASE DOMAIN: ACTIVATION AND SPECIFITY OF A STE20P MAP3K | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE
3w2c:G (LEU149) to (CYS247) STRUCTURE OF AURORA KINASE A COMPLEXED TO BENZOIMIDAZOLE-INDAZOLE INHIBITOR XV | KINASE, ATP COMPETITOR, TRANSFERASE
2hw6:A (ALA61) to (GLY165) CRYSTAL STRUCTURE OF MNK1 CATALYTIC DOMAIN | PROTEIN KINASE, DRUG DESIGN, MNK1, PHOSPHORYLATION, TRANSFERASE
2hw6:B (GLY65) to (GLY165) CRYSTAL STRUCTURE OF MNK1 CATALYTIC DOMAIN | PROTEIN KINASE, DRUG DESIGN, MNK1, PHOSPHORYLATION, TRANSFERASE
5a4e:A (GLY171) to (ALA277) DYRK1A IN COMPLEX WITH METHOXY BENZOTHIAZOLE FRAGMENT | TRANSFERASE
5a4q:A (GLY171) to (ALA277) DYRK1A IN COMPLEX WITH CHLORO BENZOTHIAZOLE FRAGMENT | TRANSFERASE
2hyy:A (GLU255) to (ASN336) HUMAN ABL KINASE DOMAIN IN COMPLEX WITH IMATINIB (STI571, GLIVEC) | TYROSINE KINASE, TRANSFERASE
2hyy:B (GLU255) to (ASN336) HUMAN ABL KINASE DOMAIN IN COMPLEX WITH IMATINIB (STI571, GLIVEC) | TYROSINE KINASE, TRANSFERASE
2hyy:D (GLU255) to (ASN336) HUMAN ABL KINASE DOMAIN IN COMPLEX WITH IMATINIB (STI571, GLIVEC) | TYROSINE KINASE, TRANSFERASE
1ias:A (GLY217) to (MET318) CYTOPLASMIC DOMAIN OF UNPHOSPHORYLATED TYPE I TGF-BETA RECEPTOR CRYSTALLIZED WITHOUT FKBP12 | KINASE, TGF-BETA RECEPTOR, GS REGION, TRANSFERASE
1ias:B (GLY217) to (HIS317) CYTOPLASMIC DOMAIN OF UNPHOSPHORYLATED TYPE I TGF-BETA RECEPTOR CRYSTALLIZED WITHOUT FKBP12 | KINASE, TGF-BETA RECEPTOR, GS REGION, TRANSFERASE
1ias:C (GLY217) to (HIS317) CYTOPLASMIC DOMAIN OF UNPHOSPHORYLATED TYPE I TGF-BETA RECEPTOR CRYSTALLIZED WITHOUT FKBP12 | KINASE, TGF-BETA RECEPTOR, GS REGION, TRANSFERASE
1ias:D (GLY217) to (HIS317) CYTOPLASMIC DOMAIN OF UNPHOSPHORYLATED TYPE I TGF-BETA RECEPTOR CRYSTALLIZED WITHOUT FKBP12 | KINASE, TGF-BETA RECEPTOR, GS REGION, TRANSFERASE
1ias:E (GLY217) to (HIS317) CYTOPLASMIC DOMAIN OF UNPHOSPHORYLATED TYPE I TGF-BETA RECEPTOR CRYSTALLIZED WITHOUT FKBP12 | KINASE, TGF-BETA RECEPTOR, GS REGION, TRANSFERASE
2i0y:A (ALA599) to (ASN773) CFMS TYROSINE KINASE (FGF KID) IN COMPLEX WITH AN ARYLAMIDE INHIBITOR | TYROSINE KINASE, KINASE INHIBITOR COMPLEX, TRANSFERASE
2i1m:A (ALA599) to (ASN773) CFMS TYROSINE KINASE (TIE2 KID) IN COMPLEX WITH AN ARYLAMIDE INHIBITOR | KINASE DOMAIN, KINASE INHIBITOR COMPLEX, TRANSFERASE
2wu6:A (LYS169) to (GLN278) CRYSTAL STRUCTURE OF THE HUMAN CLK3 IN COMPLEX WITH DKI | TRANSFERASE, KINASE, TYROSINE-PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING
2wu7:A (LYS169) to (GLN278) CRYSTAL STRUCTURE OF THE HUMAN CLK3 IN COMPLEX WITH V25 | TRANSFERASE, KINASE, TYROSINE-PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING
1iep:A (GLU255) to (SER336) CRYSTAL STRUCTURE OF THE C-ABL KINASE DOMAIN IN COMPLEX WITH STI-571. | KINASE, KINASE INHIBITOR, STI-571, ACTIVATION LOOP, TRANSFERASE
1iep:B (GLU255) to (SER336) CRYSTAL STRUCTURE OF THE C-ABL KINASE DOMAIN IN COMPLEX WITH STI-571. | KINASE, KINASE INHIBITOR, STI-571, ACTIVATION LOOP, TRANSFERASE
1ukh:A (GLY38) to (GLY146) STRUCTURAL BASIS FOR THE SELECTIVE INHIBITION OF JNK1 BY THE SCAFFOLDING PROTEIN JIP1 AND SP600125 | TRANSFERASE, PHOSPHORYLATION
2i7q:A (LEU124) to (GLY237) CRYSTAL STRUCTURE OF HUMAN CHOLINE KINASE A | NON-PROTEIN KINASE, CHOLINE KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
4m69:A (GLY78) to (GLY222) CRYSTAL STRUCTURE OF THE MOUSE RIP3-MLKL COMPLEX | KINASE, PHOSPHORYLATION, TRANSFERASE-SIGNALING PROTEIN COMPLEX
1is1:A (ALA55) to (MET183) CRYSTAL STRUCTURE OF RIBOSOME RECYCLING FACTOR FROM VIBRIO PARAHAEMOLYTICUS | TRANSLATION
5aab:A (GLY1128) to (HIS1244) STRUCTURE OF C1156Y,L1198F MUTANT HUMAN ANAPLASTIC LYMPHOMA KINASE IN COMPLEX WITH CRIZOTINIB | TRANSFERASE, RECEPTOR TYROSINE KINASE, ANAPLASTIC LYMPHOMA KINASE, INHIBITOR, MUTANT
2wzj:F (ALA65) to (PHE170) CATALYTIC AND UBA DOMAIN OF KINASE MARK2/(PAR-1) K82R, T208E DOUBLE MUTANT | UBA DOMAIN, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, SIGNALING PROTEIN, S/T PROTEIN KINASE, DIFFERENTIATION, DEVELOPMENTAL PROTEIN
4mao:A (SER434) to (GLY534) RSK2 T493M C-TERMINAL KINASE DOMAIN IN COMPLEX WITH RMM58 | PROTEIN KINASE, PHOSPHORYLATION, COVALENT INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4mbj:A (THR470) to (GLU545) HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH AN IMIDAZOPYRIDINE-BASED INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1uwh:A (LYS472) to (GLU544) THE COMPLEX OF WILD TYPE B-RAF AND BAY439006 | TRANSFERASE
1uwh:B (LYS472) to (GLU544) THE COMPLEX OF WILD TYPE B-RAF AND BAY439006 | TRANSFERASE
1uwj:A (LYS472) to (GLU544) THE COMPLEX OF MUTANT V599E B-RAF AND BAY439006 | TRANSFERASE, THREONINE-PROTEIN KINASE, SIGNAL TRANSDUCTION
1uwj:B (LYS472) to (GLU544) THE COMPLEX OF MUTANT V599E B-RAF AND BAY439006 | TRANSFERASE, THREONINE-PROTEIN KINASE, SIGNAL TRANSDUCTION
3wf9:A (GLN107) to (GLY213) CRYSTAL STRUCTURE OF S6K1 KINASE DOMAIN IN COMPLEX WITH A QUINOLINE DERIVATIVE 1-OXO-1-[(4-SULFAMOYLPHENYL)AMINO]PROPAN-2-YL-2-METHYL-1, 2,3,4-TETRAHYDROACRIDINE-9-CARBOXYLATE | SERINE/THREONINE PROTEIN KINASE DOMAIN, TRANSFERASE, PHOSPHORYLATION, ATP-BINDING, ZINC-BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2in6:A (PHE310) to (SER421) WEE1 KINASE COMPLEX WITH INHIBITOR PD311839 | PROTEIN-INHIBITOR COMPLEX, TRANSFERASE
5afv:A (LEU124) to (MET238) PHARMACOPHORE-BASED VIRTUAL SCREENING TO DISCOVER NEW ACTIVE COMPOUNDS FOR HUMAN CHOLINE KINASE ALPHA1. | TRANSFERASE, VIRTUAL SCREENING, PHARMACOPHORE
5afv:B (LEU124) to (MET238) PHARMACOPHORE-BASED VIRTUAL SCREENING TO DISCOVER NEW ACTIVE COMPOUNDS FOR HUMAN CHOLINE KINASE ALPHA1. | TRANSFERASE, VIRTUAL SCREENING, PHARMACOPHORE
4mh7:A (SER600) to (ASN718) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE-PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR UNC1896 | TYROSINE KINASE, ACUTE LYMPHOBLASTIC LEUKEMIA, RATIONAL STRUCTURE BASED DRUG DESIGN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4mh7:B (GLY604) to (ASN718) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE-PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR UNC1896 | TYROSINE KINASE, ACUTE LYMPHOBLASTIC LEUKEMIA, RATIONAL STRUCTURE BASED DRUG DESIGN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4mha:A (GLY604) to (ASN718) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE-PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR UNC1817 | TYROSINE KINASE, ACUTE LYMPHOBLASTIC LEUKEMIA, RATIONAL STRUCTURE- BASED DRUG DESIGN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2x6f:B (LEU677) to (HIS769) THE CRYSTAL STRUCTURE OF THE DROSOPHILA CLASS III PI3-KINASE VPS34 IN COMPLEX WITH 3-METHYLADENINE | TRANSFERASE
2x6k:B (LEU677) to (HIS769) THE CRYSTAL STRUCTURE OF THE DROSOPHILA CLASS III PI3-KINASE VPS34 IN COMPLEX WITH PI-103 | PI103, PI-103, AUTOPHAGY, TRANSFERASE, PI3K CLASS III, PHOSPHOINOSITIDE 3-KINASE CLASS III
2x7f:A (GLY37) to (LYS148) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN TRAF2- AND NCK-INTERACTING KINASE WITH WEE1CHK1 INHIBITOR | SERINE/THREONINE-PROTEIN KINASE, PHOSPHOPROTEIN, KINASE, TRANSFERASE
2x7f:B (GLY37) to (LYS148) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN TRAF2- AND NCK-INTERACTING KINASE WITH WEE1CHK1 INHIBITOR | SERINE/THREONINE-PROTEIN KINASE, PHOSPHOPROTEIN, KINASE, TRANSFERASE
1j7i:A (LYS30) to (ILE125) CRYSTAL STRUCTURE OF 3',5"-AMINOGLYCOSIDE PHOSPHOTRANSFERASE TYPE IIIA APOENZYME | ANTIBIOTIC RESISTANCE, KINASE, ATP-BINDING, TRANSFERASE
1j7l:B (VAL31) to (ILE125) CRYSTAL STRUCTURE OF 3',5"-AMINOGLYCOSIDE PHOSPHOTRANSFERASE TYPE IIIA ADP COMPLEX | ANTIBIOTIC RESISTANCE, KINASE, ATP-BINDING, TRANSFERASE
1j7u:A (PRO28) to (ILE125) CRYSTAL STRUCTURE OF 3',5"-AMINOGLYCOSIDE PHOSPHOTRANSFERASE TYPE IIIA AMPPNP COMPLEX | ANTIBIOTIC RESISTANCE, KINASE, ATP-BINDING, TRANSFERASE
2x9e:A (SER537) to (GLY642) HUMAN MPS1 IN COMPLEX WITH NMS-P715 | KINASE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE, MITOTIC CHECKPOINT
5am6:A (ASN506) to (LYS618) NATIVE FGFR1 WITH AN INHIBITOR | TRANSFERASE, FGFR, GROWTH FACTOR, CANCER, DOVITINIB, TKI258, KINASE
4mne:C (THR470) to (GLU545) CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4mne:F (THR470) to (GLU545) CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4mne:G (THR470) to (GLU545) CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4mnf:A (LYS473) to (GLU545) CRYSTAL STRUCTURE OF BRAF-V600E BOUND TO GDC0879 | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, ACTIVE CONFORMATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ap5:A (GLN541) to (GLY642) NATURALLY OCCURRING MUTATIONS IN THE MPS1 GENE PREDISPOSE CELLS TO KINASE INHIBITOR DRUG RESISTANCE. | TRANSFERASE, MPS1, PROTEIN KINASE, MITOSIS, DRUG RESISTANCE
4mq1:C (GLY171) to (THR278) THE CRYSTAL STRUCTURE OF DYRK1A WITH A BOUND PYRIDO[2,3-D]PYRIMIDINE INHIBITOR | DYRK1A, DYRK1B, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1jkk:A (ALA25) to (PHE119) 2.4A X-RAY STRUCTURE OF TERNARY COMPLEX OF A CATALYTIC DOMAIN OF DEATH-ASSOCIATED PROTEIN KINASE WITH ATP ANALOGUE AND MG. | TRANSFERASE
4mwi:A (SER215) to (HIS321) CRYSTAL STRUCTURE OF THE HUMAN MLKL PSEUDOKINASE DOMAIN | PSEUDOKINASE, NECROPTOSIS, TRANSFERASE
2j90:A (ALA25) to (ARG134) CRYSTAL STRUCTURE OF HUMAN ZIP KINASE IN COMPLEX WITH A TETRACYCLIC PYRIDONE INHIBITOR (PYRIDONE 6) | NUCLEAR PROTEIN, NUCLEOTIDE-BINDING, SERINE/THREONINE- PROTEIN KINASE, CHROMATIN REGULATOR, MYOSIN PHOSPHORYLATION, KINASE, MUSCLE, APOPTOSIS, TRANSFERASE, ATP-BINDING
5awm:A (ILE37) to (GLY144) THE CRYSTAL STRUCTURE OF JNK FROM DROSOPHILA MELANOGASTER REVEALS AN EVOLUTIONARILY CONSERVED TOPOLOGY WITH THAT OF MAMMALIAN JNK PROTEINS. | C-JUN N-TERMINAL KINASE, MAP KINASE, DROSOPHILA JNK PATHWAY, TRANSFERASE
2xne:A (GLY145) to (ARG251) STRUCTURE OF AURORA-A BOUND TO AN IMIDAZOPYRAZINE INHIBITOR | SER-THR PROTEIN KINASE COMPLEX, PROTO-ONCOGENE, KINASE, MITOSIS, CELL CYCLE, MICROTUBULE, TRANSFERASE, CYTOSKELETON, CELL DIVISION
3wzj:A (SER537) to (GLY642) CRYSTAL STRUCTURE OF HUMAN MPS1 CATALYTIC DOMAIN IN COMPLEX WITH 4-(6- (CYCLOHEXYLAMINO)-8-(((TETRAHYDRO-2H-PYRAN-4-YL)METHYL)AMINO) IMIDAZO[1,2-B]PYRIDAZIN-3-YL)-N-CYCLOPROPYLBENZAMIDE | TRANSFERASE, ATP BINDING, PHOSPHORYLATION
2jbp:H (LEU79) to (ASN181) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:I (GLY76) to (ASN181) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:J (LEU79) to (ASN181) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
3zc6:A (GLY834) to (ARG944) CRYSTAL STRUCTURE OF JAK3 KINASE DOMAIN IN COMPLEX WITH AN INDAZOLE SUBSTITUTED PYRROLOPYRAZINE INHIBITOR | TRANSFERASE, SCID, SEVERE COMBINED IMMUNODEFICIENCY, STAT5, STAT6, INTERLEUKIN-2, COMMON-GAMMA CHAIN, ATP SITE KINASE INHIBITOR, CANCER
2xrw:A (ILE39) to (GLY146) LINEAR BINDING MOTIFS FOR JNK AND FOR CALCINEURIN ANTAGONISTICALLY CONTROL THE NUCLEAR SHUTTLING OF NFAT4 | TRANSCRIPTION, MAPK SIGNALING PATHWAYS, LINEAR BINDING MOTIF
5bmm:B (GLY279) to (ASN381) SRC IN COMPLEX WITH DNA-TEMPLATED MACROCYCLIC INHIBITOR MC25B | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5bpy:A (GLY414) to (GLN516) CRYSTAL STRUCTURE OF BRUTON AGAMMAGLOBULINEMIA TYROSINE KINASE COMPLEXED WITH BMS-824171 AKA 6-[(3R)-3-(4-TERT-BU TYLBENZAMIDO) PIPERIDIN-1-YL]-2-{[4-(MORPHOLINE-4-CARBONYL) PHENYL]AMINO}PYRIDINE- 3-CARBOXAMIDE | KINASE, INHIBITOR, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5bq0:A (GLY414) to (GLN516) CRYSTAL STRUCTURE OF BRUTON AGAMMAGLOBULINEMIA TYROSINE KINASE COMPLEXED WITH BMS-824171 AKA 6-[(3R)-3-(4-TERT-BU TYLBENZAMIDO) PIPERIDIN-1-YL]-2-{[4-(MORPHOLINE-4-CARBONYL) PHENYL]AMINO}PYRIDINE- 3-CARBOXAMIDE | KINASE, INHIBITOR, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2jit:B (LYS737) to (ARG832) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN T790M MUTATION | EGFR, T790M, KINASE, RECEPTOR, CELL CYCLE, PHOSPHORYLATION, DISEASE MUTATION, NUCLEOTIDE-BINDING, TYROSINE-PROTEIN KINASE, ANTI-ONCOGENE, EPIDERMAL GROWTH FACTOR, ATP-BINDING, TRANSFERASE
1k2p:A (GLY414) to (PHE493) CRYSTAL STRUCTURE OF BRUTON'S TYROSINE KINASE DOMAIN | BRUTON TRYOSINE KINASE, KINASE DOMAIN, TRANSFERASE
1wbt:A (ASP88) to (LEU217) IDENTIFICATION OF NOVEL P38 ALPHA MAP KINASE INHIBITORS USING FRAGMENT-BASED LEAD GENERATION. | TRANSFERASE, ATP-BINDING, DIRECT PROTEIN SEQUENCING, NUCLEAR PROTEIN, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, P38 MAP KINASE, INHIBITOR STRUCTURE
1k9a:A (GLY207) to (ASN309) CRYSTAL STRUCTURE ANALYSIS OF FULL-LENGTH CARBOXYL-TERMINAL SRC KINASE AT 2.5 A RESOLUTION | CARBOXYL-TERMINAL SRC KINASE, COOH-TERMINAL SRC KINASE, CSK, SRC, SFK, SIGNAL TRANSDUCTION, SH2, SH3, SRC HOMOLOGY, TYROSINE KINASE, CYTOPLASMIC TYROSINE KINASE, CBP, ONCOGENE, CANCER, TRANSFERASE
1k9a:B (LEU211) to (ASN309) CRYSTAL STRUCTURE ANALYSIS OF FULL-LENGTH CARBOXYL-TERMINAL SRC KINASE AT 2.5 A RESOLUTION | CARBOXYL-TERMINAL SRC KINASE, COOH-TERMINAL SRC KINASE, CSK, SRC, SFK, SIGNAL TRANSDUCTION, SH2, SH3, SRC HOMOLOGY, TYROSINE KINASE, CYTOPLASMIC TYROSINE KINASE, CBP, ONCOGENE, CANCER, TRANSFERASE
1k9a:E (GLY207) to (GLY287) CRYSTAL STRUCTURE ANALYSIS OF FULL-LENGTH CARBOXYL-TERMINAL SRC KINASE AT 2.5 A RESOLUTION | CARBOXYL-TERMINAL SRC KINASE, COOH-TERMINAL SRC KINASE, CSK, SRC, SFK, SIGNAL TRANSDUCTION, SH2, SH3, SRC HOMOLOGY, TYROSINE KINASE, CYTOPLASMIC TYROSINE KINASE, CBP, ONCOGENE, CANCER, TRANSFERASE
1k9a:F (GLY207) to (ASN309) CRYSTAL STRUCTURE ANALYSIS OF FULL-LENGTH CARBOXYL-TERMINAL SRC KINASE AT 2.5 A RESOLUTION | CARBOXYL-TERMINAL SRC KINASE, COOH-TERMINAL SRC KINASE, CSK, SRC, SFK, SIGNAL TRANSDUCTION, SH2, SH3, SRC HOMOLOGY, TYROSINE KINASE, CYTOPLASMIC TYROSINE KINASE, CBP, ONCOGENE, CANCER, TRANSFERASE
2y4p:A (PHE24) to (GLN134) DIMERIC STRUCTURE OF DAPK-1 CATALYTIC DOMAIN | CALMODULIN-BINDING, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, APOPTOSIS, TRANSFERASE, ATP-BINDING
3zmm:A (GLY861) to (ASP949) INHIBITORS OF JAK2 KINASE DOMAIN | TRANSFERASE
1wqf:A (SER56) to (LEU183) CRYSTAL STRUCTURE OF RIBOSOME RECYCLING FACTOR FROM MYCOBACTERIUM TUBERCULOSIS | TRANSLATION FACTOR, TRIPLE-HELIX BUNDLE, PROTEIN SYNTHESIS, TRANSLATION
1wqg:A (SER56) to (LEU183) CRYSTAL STRUCTURE OF RIBOSOME RECYCLING FACTOR FROM MYCOBACTERIUM TUBERCULOSIS | TRANSLATION FACTOR, TRIPLE-HELIX BUNDLE, PROTEIN SYNTHESIS, TRANSLATION
1wvw:A (ALA25) to (GLN134) CRYSTAL STRUCTURES OF KINASE DOMAIN OF DAP KINASE IN COMPLEX WITH SMALL MOLECULAR INHIBITORS | PROTEIN KINASE, APOPTOSIS, TRANSFERASE
1wvx:A (ALA25) to (GLU118) CRYSTAL STRUCTURES OF KINASE DOMAIN OF DAP KINASE IN COMPLEX WITH SMALL MOLECULAR INHIBITORS | PROTEIN KINASE, APOPTOSIS, STAUROSPORINE, TRANSFERASE
2yab:A (LYS29) to (LYS134) CRYSTAL STRUCTURE OF THE AUTOINHIBITED FORM OF MOUSE DAPK2 IN COMPLEX WITH AMP | APOPTOSIS, TRANSFERASE
1kob:A (GLY65) to (SER169) TWITCHIN KINASE FRAGMENT (APLYSIA), AUTOREGULATED PROTEIN KINASE DOMAIN | KINASE, TWITCHIN, INTRASTERIC REGULATION
1kob:B (GLY65) to (SER169) TWITCHIN KINASE FRAGMENT (APLYSIA), AUTOREGULATED PROTEIN KINASE DOMAIN | KINASE, TWITCHIN, INTRASTERIC REGULATION
4nus:A (LEU84) to (GLY188) RSK2 N-TERMINAL KINASE IN COMPLEX WITH LJH685 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3zxt:D (ALA25) to (GLU118) DIMERIC STRUCTURE OF DAPK-1 CATALYTIC DOMAIN IN COMPLEX WITH AMPPCP-MG | APOPTOSIS, TRANSFERASE, ATP BINDING
4o38:A (ALA52) to (GLN165) CRYSTAL STRUCTURE OF THE HUMAN CYCLIN G ASSOCIATED KINASE (GAK) | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE, PROTEIN KINASE, SERINE/THREONINE KINASE, CYCLIN G, P53, CLATHRINE, MEMBRANE TRAFFICKING, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ATP- BINDING, CELL CYCLE, CELL JUNCTION, GOLGI APPARATUS, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN
4o38:B (PHE51) to (GLN165) CRYSTAL STRUCTURE OF THE HUMAN CYCLIN G ASSOCIATED KINASE (GAK) | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE, PROTEIN KINASE, SERINE/THREONINE KINASE, CYCLIN G, P53, CLATHRINE, MEMBRANE TRAFFICKING, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ATP- BINDING, CELL CYCLE, CELL JUNCTION, GOLGI APPARATUS, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN
2nru:A (GLY198) to (HIS306) CRYSTAL STRUCTURE OF IRAK-4 | KINASE, INHIBITOR, IRAK, TRANSFERASE
2nru:C (VAL199) to (HIS306) CRYSTAL STRUCTURE OF IRAK-4 | KINASE, INHIBITOR, IRAK, TRANSFERASE
2nry:A (GLY198) to (HIS306) CRYSTAL STRUCTURE OF IRAK-4 | KINASE, INHIBITOR, STAUROSPORINE, TRANSFERASE
2nry:D (GLY198) to (HIS306) CRYSTAL STRUCTURE OF IRAK-4 | KINASE, INHIBITOR, STAUROSPORINE, TRANSFERASE
4obo:B (TYR40) to (HIS148) MAP4K4 IN COMPLEX WITH INHIBITOR (COMPOUND 22), 6-(3-CHLOROPHENYL) QUINAZOLIN-4-AMINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2z2w:A (GLY311) to (SER421) HUMAND WEE1 KINASE COMPLEXED WITH INHIBITOR PF0335770 | WEE1 KINASE, INHIBITOR COMPLEX, TRANSFERASE
2o0u:A (GLY76) to (GLY184) CRYSTAL STRUCTURE OF HUMAN JNK3 COMPLEXED WITH N-{3-CYANO-6-[3-(1- PIPERIDINYL)PROPANOYL]-4,5,6,7-TETRAHYDROTHIENO[2,3-C]PYRIDIN-2-YL}- 1-NAPHTHALENECARBOXAMIDE | KINASE FOLD, TRANSFERASE
2z60:A (GLU255) to (SER336) CRYSTAL STRUCTURE OF THE T315I MUTANT OF ABL KINASE BOUND WITH PPY-A | ABL, KINASE, MUTANT, T315I, ALTERNATIVE SPLICING, ATP- BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHORYLATION, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
4oli:A (GLY909) to (GLN1017) THE PSEUDOKINASE/KINASE PROTEIN FROM JAK-FAMILY MEMBER TYK2 | PROTEIN KINASE, PHOSPHO-TRANSFER, TRANSFERASE
5csx:A (GLY469) to (GLU545) CRYSTAL STRUCTURE OF B-RAF IN COMPLEX WITH BI 882370 | KINASE, TRANSFERASE
5ct7:A (GLY469) to (GLU545) BRAF IN COMPLEX WITH RAF265 | KINASE, TRANSFERASE
5ct7:B (LYS473) to (GLU545) BRAF IN COMPLEX WITH RAF265 | KINASE, TRANSFERASE
3kcf:A (GLY217) to (MET318) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A PYRAZOLONE INHIBITOR | KINASE, TGFBETARI, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, AORTIC ANEURYSM, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3kcf:C (GLY217) to (HIS317) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A PYRAZOLONE INHIBITOR | KINASE, TGFBETARI, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, AORTIC ANEURYSM, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3kcf:D (GLY217) to (HIS317) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A PYRAZOLONE INHIBITOR | KINASE, TGFBETARI, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, AORTIC ANEURYSM, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3kcf:E (GLY217) to (MET318) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A PYRAZOLONE INHIBITOR | KINASE, TGFBETARI, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, AORTIC ANEURYSM, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
4aaa:A (MET17) to (GLY113) CRYSTAL STRUCTURE OF THE HUMAN CDKL2 KINASE DOMAIN | TRANSFERASE, PHOSPHO-MIMETIC
3kf4:A (GLU258) to (SER336) STRUCTURAL ANALYSIS OF DFG-IN AND DFG-OUT DUAL SRC-ABL INHIBITORS SHARING A COMMON VINYL PURINE TEMPLATE | ABL, CML, DRUG RESISTANCE, INHIBITOR, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, ONCOGENE, TYROSINE-PROTEIN KINASE, TRANSFERASE
3kf4:B (GLU255) to (SER336) STRUCTURAL ANALYSIS OF DFG-IN AND DFG-OUT DUAL SRC-ABL INHIBITORS SHARING A COMMON VINYL PURINE TEMPLATE | ABL, CML, DRUG RESISTANCE, INHIBITOR, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, ONCOGENE, TYROSINE-PROTEIN KINASE, TRANSFERASE
2zm1:A (PHE256) to (LEU336) CRYSTAL STRUCTURE OF IMIDAZO PYRAZIN 1 BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE- BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
2zm3:A (PRO1026) to (LYS1130) COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND ISOQUINOLINEDIONE INHIBITOR | IGFR, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP- BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
1m7n:B (GLY1013) to (LYS1127) CRYSTAL STRUCTURE OF UNACTIVATED APO INSULIN-LIKE GROWTH FACTOR-1 RECEPTOR KINASE DOMAIN | TRANSFERASE
5cyz:A (GLY21) to (SER123) STRUCTURE OF S. CEREVISIAE HRR25:MAM1 COMPLEX, FORM 1 | CASEIN KINASE, MONOPOLIN, TRANSFERASE
5czo:A (GLY21) to (SER123) STRUCTURE OF S. CEREVISIAE HRR25:MAM1 COMPLEX, FORM 2 | CASEIN KINASE, MONOPOLIN, TRANSFERASE
5czo:B (GLY21) to (SER123) STRUCTURE OF S. CEREVISIAE HRR25:MAM1 COMPLEX, FORM 2 | CASEIN KINASE, MONOPOLIN, TRANSFERASE
3kk8:A (SER25) to (GLY130) CAMKII SUBSTRATE COMPLEX A | PROTEIN KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2zv7:A (MET263) to (VAL339) LYN TYROSINE KINASE DOMAIN, APO FORM | LYN KINASE, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
2zv8:A (GLY259) to (VAL339) LYN TYROSINE KINASE DOMAIN-AMP-PNP COMPLEX | LYN KINASE AMPPNP, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
2zv9:A (GLY259) to (VAL339) LYN TYROSINE KINASE DOMAIN-PP2 COMPLEX | LYN KINASE PP2, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
2zva:A (GLY259) to (VAL339) LYN TYROSINE KINASE DOMAIN-DASATINIB COMPLEX | LYN KINASE DASATINIB, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
4agd:A (ALA851) to (SER1021) CRYSTAL STRUCTURE OF VEGFR2 (JUXTAMEMBRANE AND KINASE DOMAINS) IN COMPLEX WITH SUNITINIB (SU11248) (N-2- DIETHYLAMINOETHYL)-5-((Z)-(5-FLUORO-2-OXO-1H-INDOL-3- YLIDENE)METHYL)-2,4-DIMETHYL-1H-PYRROLE-3-CARBOXAMIDE) | TRANSFERASE, ANGIOGENESIS, NUCLEOTIDE-BINDING, INHIBITOR, PHOSPHORYLATION, TRANSMEMBRANE
4agw:A (GLY279) to (LEU358) DISCOVERY OF A SMALL MOLECULE TYPE II INHIBITOR OF WILD- TYPE AND GATEKEEPER MUTANTS OF BCR-ABL, PDGFRALPHA, KIT, AND SRC KINASES | ATP-BINDING, LIPOPROTEIN, MYRISTATE, PHOSPHOPROTEIN, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3kmm:A (GLY257) to (LEU336) STRUCTURE OF HUMAN LCK KINASE WITH A SMALL MOLECULE INHIBITOR | TYROSINE KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
2zyb:A (PHE256) to (LEU336) CRYSTAL STRUCTURE OF PHENYLIMIDAZO PYRAZIN 2 BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, KINASE, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, CELL MEMBRANE, POLYMORPHISM
3a4o:X (GLU29) to (VAL108) LYN KINASE DOMAIN | SRC FAMILY, KINASE DOMAIN, ALTERNATIVE SPLICING, ATP- BINDING, HOST-VIRUS INTERACTION, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, TRANSFERASE, TYROSINE-PROTEIN KINASE
3a60:A (GLN107) to (GLY213) CRYSTAL STRUCTURE OF UNPHOSPHORYLATED P70S6K1 (FORM I) | KINASE, KINASE DOMAIN, INACTIVE, ACTIVE, RIBOSOMAL S6 KINASE, ACTIVATION, ALTERNATIVE INITIATION, ATP-BINDING, CELL JUNCTION, CYTOPLASM, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, SYNAPSE, SYNAPTOSOME, TRANSFERASE
3a61:A (LYS104) to (GLY213) CRYSTAL STRUCTURE OF UNPHOSPHORYLATED P70S6K1 (FORM II) | KINASE, KINASE DOMAIN, INACTIVE, ACTIVE, RIBOSOMAL S6 KINASE, ACTIVATION, ALTERNATIVE INITIATION, ATP-BINDING, CELL JUNCTION, CYTOPLASM, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, SYNAPSE, SYNAPTOSOME, TRANSFERASE
3a62:A (GLN107) to (GLY213) CRYSTAL STRUCTURE OF PHOSPHORYLATED P70S6K1 | KINASE, KINASE DOMAIN, INACTIVE, ACTIVE, RIBOSOMAL S6 KINASE, ACTIVATION, ALTERNATIVE INITIATION, ATP-BINDING, CELL JUNCTION, CYTOPLASM, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, SYNAPSE, SYNAPTOSOME, TRANSFERASE
5d9l:A (GLY80) to (GLY188) RSK2 N-TERMINAL KINASE IN COMPLEX WITH BIS-PHENOL PYRAZOLE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1yi6:A (GLY279) to (LEU358) C-TERM TAIL SEGMENT OF HUMAN TYROSINE KINASE (258-533) | SRC, TYROSINE KINASE, PHOSPHORYLATION, REGULATION, SH2, SH3, TRANSFERASE
3kxz:A (MET261) to (LEU336) THE COMPLEX CRYSTAL STRUCTURE OF LCK WITH A PROBE MOLECULE W259 | LCK, ACETYLATION, ATP-BINDING, CELL MEMBRANE, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, KINASE, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, TRANSFERASE, TYROSINE-PROTEIN KINASE, STRUCTURAL GENOMICS, PROTEIN STRUCTURE FACTORY, PSF
1yom:A (GLY286) to (TYR359) CRYSTAL STRUCTURE OF SRC KINASE DOMAIN IN COMPLEX WITH PURVALANOL A | PROTEIN TYROSINE KINASE, TRANSFERASE
1yom:B (GLY281) to (LEU360) CRYSTAL STRUCTURE OF SRC KINASE DOMAIN IN COMPLEX WITH PURVALANOL A | PROTEIN TYROSINE KINASE, TRANSFERASE
3ac1:A (PHE256) to (LEU336) CRYSTAL STRUCTURE OF PYRAZIN DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3ac4:A (PHE256) to (LEU336) CRYSTAL STRUCTURE OF TRIAZOLO PYRIMIDINE DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3acj:A (PHE256) to (LEU336) CRYSTAL STRUCTURE OF IMIDAZO PYRIMIDINE DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3ack:A (PHE256) to (LEU336) CRYSTAL STRUCTURE OF PYRROLO PYRAZINE DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3ad5:A (PHE256) to (LEU336) CRYSTAL STRUCTURE OF TRIAZOLONE DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
5di1:B (GLN38) to (HIS148) MAP4K4 IN COMPLEX WITH AN INHIBITOR | KINASE, INHIBITOR, COMPLEX, MEDICINAL CHEMISTRY, TRANSFERASE- INHIBITOR COMPLEX
4pmm:A (ALA527) to (HIS645) THE STRUCTURE OF TRKA KINASE BOUND TO THE INHIBITOR N-(3-CYCLOPROPYL- 1-PHENYL-1H-PYRAZOL-5-YL)-2-{4-[3-METHOXY-4-(4-METHYL-1H-IMIDAZOL-1- YL)PHENYL]-1H-1,2,3-TRIAZOL-1-YL}ACETAMIDE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4pmp:A (ALA527) to (HIS645) THE STRUCTURE OF TRKA KINASE BOUND TO THE INHIBITOR 1-CYCLOPROPYL-1- [3-(1,3-THIAZOL-2-YL)BENZYL]-3-[4-(TRIFLUOROMETHOXY)PHENYL]UREA | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4pms:A (ALA527) to (HIS645) THE STRUCTURE OF TRKA KINASE BOUND TO THE INHIBITOR 4-NAPHTHALEN-1-YL- 1-[(5-PHENYL-1,2,4-OXADIAZOL-3-YL)METHYL]-1H-PYRROLO[3,2-C]PYRIDINE- 2-CARBOXYLIC ACID | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5dmz:A (ALA799) to (GLU912) STRUCTURE OF HUMAN BUB1 KINASE DOMAIN PHOSPHORYLATED AT SER969 | KINASE, PHOSPHORYLATION, TRANSFERASE
5dmz:B (ALA799) to (GLU912) STRUCTURE OF HUMAN BUB1 KINASE DOMAIN PHOSPHORYLATED AT SER969 | KINASE, PHOSPHORYLATION, TRANSFERASE
4pp7:A (LYS473) to (GLU545) HIGHLY POTENT AND SELECTIVE 3-N-METHYLQUINAZOLINE-4(3H)-ONE BASED INHIBITORS OF B-RAFV600E KINASE | SERINE/THREONINE-PROTEIN KINASE B-RAF, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4pp7:B (LYS473) to (GLU545) HIGHLY POTENT AND SELECTIVE 3-N-METHYLQUINAZOLINE-4(3H)-ONE BASED INHIBITORS OF B-RAFV600E KINASE | SERINE/THREONINE-PROTEIN KINASE B-RAF, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3lck:A (PHE256) to (LEU336) THE KINASE DOMAIN OF HUMAN LYMPHOCYTE KINASE (LCK), ACTIVATED FORM (AUTO-PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION
4ptc:A (GLY68) to (GLY176) STRUCTURE OF A CARBOXAMIDE COMPOUND (3) (2-{2-[(CYCLOPROPYLCARBONYL) AMINO]PYRIDIN-4-YL}-4-OXO-4H-1LAMBDA~4~,3-THIAZOLE-5-CARBOXAMIDE) TO GSK3B | SERINE/THREONINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ptc:B (GLY68) to (GLY176) STRUCTURE OF A CARBOXAMIDE COMPOUND (3) (2-{2-[(CYCLOPROPYLCARBONYL) AMINO]PYRIDIN-4-YL}-4-OXO-4H-1LAMBDA~4~,3-THIAZOLE-5-CARBOXAMIDE) TO GSK3B | SERINE/THREONINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ptg:B (GLY68) to (GLY176) STRUCTURE OF A CARBOXAMINE COMPOUND (26) (2-{2-[(CYCLOPROPYLCARBONYL) AMINO]PYRIDIN-4-YL}-4-METHOXYPYRIMIDINE-5-CARBOXAMIDE) TO GSK3B | SERINE/THREONINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ano:A (ASP13) to (VAL95) CRYSTAL STRUCTURE GEOBACILLUS THERMODENITRIFICANS ESSB CYTOPLASMIC FRAGMENT | MEMBRANE PROTEIN, MEMBRANE SECRETION, ESS TYPE V SECRETION SYSTEM
4aot:A (GLY48) to (ARG152) CRYSTAL STRUCTURE OF HUMAN SERINE THREONINE KINASE-10 (LOK) BOUND TO GW830263A | TRANSFERASE, STK10, LOK
3lij:A (GLY74) to (ASN179) CRYSTAL STRUCTURE OF FULL LENGTH CPCDPK3 (CGD5_820) IN COMPLEX WITH CA2+ AND AMPPNP | TRANSFERASE, CALCIUM DEPENDENT PROTEIN KINASE, EF HAND, ATP- BINDING, CALCIUM, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
3lj0:A (GLN691) to (LYS792) IRE1 COMPLEXED WITH ADP AND QUERCETIN | KINASE, FLAVONOL, ACTIVATOR, DIMER, ATP-BINDING, ENDOPLASMIC RETICULUM, GLYCOPROTEIN, HYDROLASE, MAGNESIUM, MEMBRANE, METAL- BINDING, MULTIFUNCTIONAL ENZYME, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, TRANSMEMBRANE, UNFOLDED PROTEIN RESPONSE
3lj0:B (GLN691) to (LYS792) IRE1 COMPLEXED WITH ADP AND QUERCETIN | KINASE, FLAVONOL, ACTIVATOR, DIMER, ATP-BINDING, ENDOPLASMIC RETICULUM, GLYCOPROTEIN, HYDROLASE, MAGNESIUM, MEMBRANE, METAL- BINDING, MULTIFUNCTIONAL ENZYME, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, TRANSMEMBRANE, UNFOLDED PROTEIN RESPONSE
4apc:A (LYS17) to (LYS123) CRYSTAL STRUCTURE OF HUMAN NIMA-RELATED KINASE 1 (NEK1) | TRANSFERASE
4apc:B (LYS17) to (LYS123) CRYSTAL STRUCTURE OF HUMAN NIMA-RELATED KINASE 1 (NEK1) | TRANSFERASE
3anq:D (GLY171) to (THR278) HUMAN DYRK1A/INHIBITOR COMPLEX | PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5dvr:A (GLU64) to (LYS169) CRYSTAL STRUCTURE OF TGCDPK1 FROM TOXOPLASMA GONDII COMPLEXED WITH GW780159X | STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPKS, SERINE/THREONINE PROTEIN KINASE, NUCLEOTIDE-BINDING, GW780159X, TRANSFERASE
3lmg:A (SER715) to (GLY810) CRYSTAL STRUCTURE OF THE ERBB3 KINASE DOMAIN IN COMPLEX WITH AMP-PNP | ERBB3, HER3, TYROSINE KINASE DOMAIN, AMP-PNP, NUCLEOTIDE BINDING, TRANSFERASE
4asx:A (GLY204) to (HIS304) CRYSTAL STRUCTURE OF ACTIVIN RECEPTOR TYPE-IIA (ACVR2A) KINASE DOMAIN IN COMPLEX WITH DIHYDRO-BAUERINE C | TRANSFERASE, PROTEIN KINASE
1zmw:A (ALA65) to (PHE170) CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK2/PAR-1: T208A/S212A INACTIVE DOUBLE MUTANT | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE
1zmu:A (LYS66) to (PHE170) CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK2/PAR-1: WILD TYPE | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE
1zmu:B (LYS66) to (PHE170) CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK2/PAR-1: WILD TYPE | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE
1zmv:A (ALA65) to (GLN168) CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK2/PAR-1: K82R MUTANT | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE
3aox:A (GLU1129) to (HIS1244) X-RAY CRYSTAL STRUCTURE OF HUMAN ANAPLASTIC LYMPHOMA KINASE IN COMPLEX WITH CH5424802 | ALK KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4awi:A (GLY38) to (SER144) HUMAN JNK1ALPHA KINASE WITH 4-PHENYL-7-AZAINDOLE IKK2 INHIBITOR. | TRANSFERASE
4ax8:A (SER240) to (GLY346) MEDIUM RESOLUTION STRUCTURE OF THE BIFUNCTIONAL KINASE- METHYLTRANSFERASE WBDD | TRANSFERASE, KINASE, METHYLTRANSFERASE
1zy5:B (GLY611) to (GLY830) CRYSTAL STRUCTURE OF EIF2ALPHA PROTEIN KINASE GCN2: R794G HYPERACTIVATING MUTANT COMPLEXED WITH AMPPNP. | TRANSLATION REGULATOR, PROTEIN KINASE, SIGNAL TRANSDUCTION, AMINO-ACID STARVATION, STARVATION STRESS RESPONSE, EIF2ALPHA KINASE, TRANSFERASE
3ats:A (ARG70) to (SER178) CRYSTAL STRUCTURE OF RV3168 | HYPOTHETICAL PROTEIN, PUTATIVE AMINOGLYCOSIDE PHOSPHORTRANSFERASE, TRANSFERASE
1zz2:A (GLY36) to (ASP145) TWO CLASSES OF P38ALPHA MAP KINASE INHIBITORS HAVING A COMMON DIPHENYLETHER CORE BUT EXHIBITING DIVERGENT BINDING MODES | PROTEIN-INHIBITOR COMPLEX, TRANSFERASE
1zzl:A (ASP88) to (LEU217) CRYSTAL STRUCTURE OF P38 WITH TRIAZOLOPYRIDINE | PHOSPHORYLATION,SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4azt:A (SER240) to (GLY346) CO-CRYSTAL STRUCTURE OF WBDD AND KINASE INHIBITOR LY294002. | TRANSFERASE
2a27:B (ALA25) to (LYS134) HUMAN DRP-1 KINASE, W305S S308A D40 MUTANT, CRYSTAL FORM WITH 8 MONOMERS IN THE ASYMMETRIC UNIT | PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE
5e8y:A (ALA256) to (SER363) TGF-BETA RECEPTOR TYPE 2 KINASE DOMAIN (E431A,R433A,E485A,K488A,R493A, R495A) IN COMPLEX WITH STAUROSPORINE | KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2a2a:C (PHE24) to (LYS134) HIGH-RESOLUTION CRYSTALLOGRAPHIC ANALYSIS OF THE AUTOINHIBITED CONFORMATION OF A HUMAN DEATH-ASSOCIATED PROTEIN KINASE | PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE
5eak:B (ALA65) to (PHE170) OPTIMIZATION OF MICROTUBULE AFFINITY REGULATING KINASE (MARK) INHIBITORS WITH IMPROVED PHYSICAL PROPERTIES | CATALYTIC DOMAIN, PROTEIN-SERINE-THREONINE KINASES, KINASE INHIBITOR, SERINE-THREONINE KINASES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3m42:A (LEU79) to (ASN181) CRYSTAL STRUCTURE OF MAPKAP KINASE 2 (MK2) COMPLEXED WITH A TETRACYCLIC ATP SITE INHIBITOR | SMALL MOLECULE INHIBITOR, ATP-SITE KINASE INHIBITOR, NOVARTIS-PRODUCT NVP-BMA086, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4b9d:A (LYS17) to (LYS123) CRYSTAL STRUCTURE OF HUMAN NIMA-RELATED KINASE 1 (NEK1) WITH INHIBITOR. | TRANSFERASE, INHIBITOR
4b9d:B (LYS17) to (LYS123) CRYSTAL STRUCTURE OF HUMAN NIMA-RELATED KINASE 1 (NEK1) WITH INHIBITOR. | TRANSFERASE, INHIBITOR
5ei6:A (SER537) to (GLY642) RAPID DISCOVERY OF PYRIDO[3,4-D]PYRIMIDINE INHIBITORS OF MONOPOLAR SPINDLE KINASE 1 (MPS1) USING A STRUCTURE-BASED HYDRIDIZATION APPROACH | SPINDLE ASSEMBLY CHECKPOINT (SAC), ONCOLOGY TARGET PYRIDO[3, 4- D]PYRIMIDINE BASED INHIBITORS SELECTIVE AGAINST MPS1, TRANSFERASE
4bbe:A (PHE860) to (ARG971) AMINOALKYLPYRIMIDINE INHIBITOR COMPLEXES WITH JAK2 | TRANSFERASE, INHIBITOR
4bbe:B (GLY861) to (ARG971) AMINOALKYLPYRIMIDINE INHIBITOR COMPLEXES WITH JAK2 | TRANSFERASE, INHIBITOR
4bbe:C (GLY861) to (ARG971) AMINOALKYLPYRIMIDINE INHIBITOR COMPLEXES WITH JAK2 | TRANSFERASE, INHIBITOR
4bbe:D (GLY861) to (ARG971) AMINOALKYLPYRIMIDINE INHIBITOR COMPLEXES WITH JAK2 | TRANSFERASE, INHIBITOR
3mdy:C (GLY216) to (THR317) CRYSTAL STRUCTURE OF THE CYTOPLASMIC DOMAIN OF THE BONE MORPHOGENETIC PROTEIN RECEPTOR TYPE-1B (BMPR1B) IN COMPLEX WITH FKBP12 AND LDN- 193189 | COMPLEX (ISOMERASE-PROTEIN KINASE), RECEPTOR SERINE/THREONINE KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, DISEASE MUTATION, KINASE, TRANSFERASE, ROTAMASE, TRANSFERASE-ISOMERASE COMPLEX
3mes:B (GLN85) to (ILE181) CRYSTAL STRUCTURE OF CHOLINE KINASE FROM CRYPTOSPORIDIUM PARVUM IOWA II, CGD3_2030 | CHOLINE KINASE, MALARIA, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE
4bcj:A (GLU32) to (LYS144) STRUCTURE OF CDK9 IN COMPLEX WITH CYCLIN T AND A 2-AMINO-4- HETEROARYL-PYRIMIDINE INHIBITOR | TRANSFERASE-CELL CYCLE COMPLEX, CDK-CYCLIN COMPLEX, TRANSCRIPTION-PROTEIN BINDING, STRUCTURE-BASED DRUG DESIGN
4qpm:A (ALA799) to (GLU912) STRUCTURE OF BUB1 KINASE DOMAIN | TRANSFERASE
4qpm:B (ALA799) to (GLU912) STRUCTURE OF BUB1 KINASE DOMAIN | TRANSFERASE
3bea:A (ALA599) to (ASN773) CFMS TYROSINE KINASE (TIE2 KID) IN COMPLEX WITH A PYRIMIDINOPYRIDONE INHIBITOR | KINASE DOMAIN, INHIBITOR, TRANSFERASE, JUXTAMEMBRANE DOMAIN, ATP-BINDING, GLYCOPROTEIN, IMMUNOGLOBULIN DOMAIN, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO- ONCOGENE, RECEPTOR, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
5eqy:A (SER121) to (GLY237) CRYSTAL STRUCTURE OF CHOLINE KINASE ALPHA-1 BOUND BY 5-[(4-METHYL-1,4- DIAZEPAN-1-YL)METHYL]-2-[4-[(4-METHYL-1,4-DIAZEPAN-1-YL) METHYL]PHENYL]BENZENECARBONITRILE (COMPOUND 65) | KINASE, INHIBITOR, DRUG TARGET, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4bhz:A (SER537) to (GLY642) SCAFFOLD FOCUSED VIRTUAL SCREENING: PROSPECTIVE APPLICATION TO THE DISCOVERY OF TTK INHIBITOR | TRANSFERASE, MITOSIS
4bi1:A (GLN541) to (GLY642) SCAFFOLD FOCUSED VIRTUAL SCREENING: PROSPECTIVE APPLICATION TO THE DISCOVERY OF TTK INHIBITOR | TRANSFERASE, PROTEIN KINASE, MITOSIS
3mpm:A (MET261) to (LEU336) LCK COMPLEXED WITH A PYRAZOLOPYRIMIDINE | KINASE DOMAIN, TRANSFERASE
4bky:A (ALA23) to (VAL112) CRYSTAL STRUCTURE OF UNPHOSPHORYLATED MATERNAL EMBRYONIC LEUCINE ZIPPER KINASE (MELK) IN COMPLEX WITH PYRROLOPYRAZOLE INHIBITOR | TRANSFERASE
4bkz:A (LYS24) to (VAL112) CRYSTAL STRUCTURE OF UNPHOSPHORYLATED MATERNAL EMBRYONIC LEUCINE ZIPPER KINASE (MELK) IN COMPLEX WITH A BENZODIPYRAZOLE INHIBITOR | TRANSFERASE
4bl1:A (ALA23) to (VAL112) CRYSTAL STRUCTURE OF UNPHOSPHORYLATED MATERNAL EMBRYONIC LEUCINE ZIPPER KINASE (MELK) IN COMPLEX WITH AMP-PNP | TRANSFERASE
3mtf:B (GLY220) to (HIS320) CRYSTAL STRUCTURE OF THE ACVR1 KINASE IN COMPLEX WITH A 2- AMINOPYRIDINE INHIBITOR | PROTEIN KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3bpr:A (GLY604) to (ASN718) CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE- PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR C52 | ATP-BINDING, DISEASE MUTATION, GLYCOPROTEIN, KINASE, NUCLEOTIDE- BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, RECEPTOR, RETINITIS PIGMENTOSA, SENSORY TRANSDUCTION, TRANSFERASE, TYROSINE-PROTEIN KINASE, VISION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, IMMUNOGLOBULIN DOMAIN, MEMBRANE, PHOSPHOPROTEIN, POLYMORPHISM, TRANSMEMBRANE
3bpr:B (GLY604) to (ASN718) CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE- PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR C52 | ATP-BINDING, DISEASE MUTATION, GLYCOPROTEIN, KINASE, NUCLEOTIDE- BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, RECEPTOR, RETINITIS PIGMENTOSA, SENSORY TRANSDUCTION, TRANSFERASE, TYROSINE-PROTEIN KINASE, VISION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, IMMUNOGLOBULIN DOMAIN, MEMBRANE, PHOSPHOPROTEIN, POLYMORPHISM, TRANSMEMBRANE
3bpr:C (GLY604) to (ASN718) CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE- PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR C52 | ATP-BINDING, DISEASE MUTATION, GLYCOPROTEIN, KINASE, NUCLEOTIDE- BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, RECEPTOR, RETINITIS PIGMENTOSA, SENSORY TRANSDUCTION, TRANSFERASE, TYROSINE-PROTEIN KINASE, VISION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, IMMUNOGLOBULIN DOMAIN, MEMBRANE, PHOSPHOPROTEIN, POLYMORPHISM, TRANSMEMBRANE
3brb:A (GLY604) to (ASN718) CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE- PROTEIN KINASE MER IN COMPLEX WITH ADP | ATP-BINDING, DISEASE MUTATION, GLYCOPROTEIN, KINASE, NUCLEOTIDE- BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, RECEPTOR, RETINITIS PIGMENTOSA, SENSORY TRANSDUCTION, TRANSFERASE, TYROSINE-PROTEIN KINASE, VISION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, IMMUNOGLOBULIN DOMAIN, MEMBRANE, PHOSPHOPROTEIN, TRANSMEMBRANE
3brb:B (GLY604) to (ASN718) CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE- PROTEIN KINASE MER IN COMPLEX WITH ADP | ATP-BINDING, DISEASE MUTATION, GLYCOPROTEIN, KINASE, NUCLEOTIDE- BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, RECEPTOR, RETINITIS PIGMENTOSA, SENSORY TRANSDUCTION, TRANSFERASE, TYROSINE-PROTEIN KINASE, VISION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, IMMUNOGLOBULIN DOMAIN, MEMBRANE, PHOSPHOPROTEIN, TRANSMEMBRANE
3mwu:A (GLY88) to (ILE178) ACTIVATED CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM CRYPTOSPORIDIUM PARVUM (CPCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR RM-1-95 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, BUMPED KINASE INHIBITOR, BKI, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3my0:A (GLY214) to (HIS314) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:B (GLY214) to (HIS314) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:D (GLY214) to (HIS314) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:E (GLY214) to (HIS314) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:F (GLY214) to (HIS314) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:G (GLY214) to (HIS314) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:H (GLY214) to (HIS314) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:M (GLY214) to (HIS314) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:Q (GLY214) to (HIS314) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:R (GLY214) to (HIS314) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:T (GLY214) to (HIS314) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:V (GLY214) to (HIS314) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:W (GLY214) to (HIS314) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:X (GLY214) to (HIS314) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3bv3:A (GLY36) to (ASP145) MORPHOLINO PYRROLOTRIAZINE P38 ALPHA MAP KINASE INHIBITOR COMPOUND 2 | SERINE/THREONINE-PROTEIN KINASE, KINASE, TRANSFERASE, P38 MAP KINASE, ALTERNATIVE SPLICING, ATP-BINDING, CYTOPLASM, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN
4br3:B (LEU124) to (GLY237) DETERMINATION OF POTENTIAL SCAFFOLDS FOR HUMAN CHOLINE KINASE ALPHA 1 BY CHEMICAL DECONVOLUTION STUDIES | TRANSFERASE
5f94:B (GLY68) to (GLY176) CRYSTAL STRUCTURE OF GSK3B IN COMPLEX WITH COMPOUND 15: 2- [(CYCLOPROPYLCARBONYL)AMINO]-N-(4-METHOXYPYRIDIN-3-YL)PYRIDINE-4- CARBOXAMIDE | GSK3B, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3bym:A (PHE256) to (LEU336) X-RAY CO-CRYSTAL STRUCTURE AMINOBENZIMIDAZOLE TRIAZINE 1 BOUND TO LCK | LCK, KINASE DOMAIN, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE
3byo:A (PHE256) to (LEU336) X-RAY CO-CRYSTAL STRUCTURE OF 2-AMINO-6-PHENYLPYRIMIDO[5', 4':5,6]PYRIMIDO[1,2-A]BENZIMIDAZOL-5(6H)-ONE 25 BOUND TO LCK | LCK, KINASE DOMAIN, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE
3bys:A (PHE256) to (LEU336) CO-CRYSTAL STRUCTURE OF LCK AND AMINOPYRIMIDINE AMIDE 10B | LCK, KINASE DOMAIN, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE
3byu:A (PHE256) to (LEU336) CO-CRYSTAL STRUCTURE OF LCK AND AMINOPYRIMIDINE REVERSE AMIDE 23 | LCK, KINASE DOMAIN, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE
3n4t:A (ILE35) to (ILE133) APO APH(2")-IVA FORM I | AMINOGLYCOSIDE, PHOSPHOTRANSFERASE, RESISTANCE, UNKNOWN FUNCTION
5fd2:B (THR470) to (GLU545) B-RAF WILD-TYPE KINASE DOMAIN IN COMPLEX WITH A PURINYLPYRIDINYLAMINO- BASED INHIBITOR | PHOSPHOTRANSFERASE, INHIBITOR, MELANOMA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3c4c:A (GLY469) to (GLU545) B-RAF KINASE IN COMPLEX WITH PLX4720 | B-RAF, BRAF, RAF, PROTO-ONCOGENE, SERINE/THREONINE KINASE, ATP-BINDING, CARDIOMYOPATHY, CYTOPLASM, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ZINC, ZINC-FINGER
4r7h:A (ALA599) to (LEU687) CRYSTAL STRUCTURE OF FMS KINASE DOMAIN WITH A SMALL MOLECULAR INHIBITOR, PLX3397 | CSF-1-R, FMS PROTO-ONCOGENE, C-FMS, CD115 ANTIGEN, KINASE, ATP- BINDING, PLX3397, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4r8q:A (ALA799) to (GLU912) STRUCTURE AND SUBSTRATE RECRUITMENT OF THE HUMAN SPINDLE CHECKPOINT KINASE BUB1 | SPINDLE ASSEMBLY CHECKPOINT, MITOSIS, KINASE, ACTIVATION, KEN BOX, CDC20, ATP-BINDING, CELL CYCLE, CELL DIVISION, DISEASE MUTATION, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
3ce3:A (GLY1095) to (LYS1199) CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF THE HEPATOCYTE GROWTH FACTOR RECEPTOR C-MET IN COMPLEX WITH A PYRROLOPYRIDINEPYRIDONE BASED INHIBITOR | RECEPTOR TYROSINE KINASE, SIGNAL TRANSDUCTION, GRB2, SHC, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3ncg:A (GLY88) to (ILE178) ACTIVATED CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM CRYPTOSPORIDIUM PARVUM (CPCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR NM-PP1 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, BUMPED KINASE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP
4c3f:A (MET261) to (LEU336) STRUCTURE OF LCK IN COMPLEX WITH A COMPOUND DISCOVERED BY VIRTUAL FRAGMENT LINKING | TRANSFERASE
4rfm:A (LEU376) to (SER477) ITK KINASE DOMAIN IN COMPLEX WITH COMPOUND 1 N-{1-[(1,1-DIOXO-1-THIAN- 2-YL)(PHENYL)METHYL]-1H- PYRAZOL-4-YL}-5,5-DIFLUORO-5A-METHYL-1H,4H, 4AH,5H,5AH,6H-CYCLOPROPA[F]INDAZOLE-3-CARBOXAMIDE | KINASE, TRANSFERASE-INHIBITOR COMPLEX
4c4g:A (SER537) to (GLY642) STRUCTURE-BASED DESIGN OF ORALLY BIOAVAILABLE PYRROLOPYRIDINE INHIBITORS OF THE MITOTIC KINASE MPS1 | TRANSFERASE, PROTEIN KINASE, MITOSIS, STRUCTURE-BASED DESIGN
4c58:A (ALA52) to (GLN165) STRUCTURE OF GAK KINASE IN COMPLEX WITH NANOBODY (NBGAK_4) | TRANSFERASE, KINASE, CONFORMATIONAL PLASTICITY, ACTIVATION
4c59:A (ALA52) to (ARG164) STRUCTURE OF GAK KINASE IN COMPLEX WITH NANOBODY (NBGAK_4) | TRANSFERASE, KINASE, CONFORMATIONAL PLASTICITY, ACTIVATION
4rix:D (GLY705) to (ASN784) CRYSTAL STRUCTURE OF AN EGFR/HER3 KINASE DOMAIN HETERODIMER CONTAINING THE CANCER-ASSOCIATED HER3-Q790R MUTATION | RECEPTOR TYROSINE KINASE, PSEUDOKINASE, KINASE, ATP BINDING, MEMBRANE, TRANSFERASE
4rmz:B (GLY198) to (HIS306) CRYSTAL STRUCTURE OF IRAK-4 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3cr0:A (SER312) to (SER421) WEE1 KINASE COMPLEX WITH INHIBITOR PD259_809 | KINASE DOMAIN, INHIBITOR COMPLEX, TRANSFERASE
4cg9:A (LEU124) to (GLY237) HUMAN CHOLINE KINASE A1 IN COMPLEX WITH COMPOUND 12 | TRANSFERASE, CANCER, DRUG TARGET, BISCATIONIC COMPOUNDS
3cs9:C (GLU255) to (ASN336) HUMAN ABL KINASE IN COMPLEX WITH NILOTINIB | NILOTINIB, AMN107, KINASE, ABL, ALTERNATIVE SPLICING, ATP- BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, ABL KINASE WT IN COMPLEX WITH NVP-AMN107
3nw5:A (PRO996) to (LYS1100) CRYSTAL STRUCTURE OF INSULIN-LIKE GROWTH FACTOR 1 RECEPTOR (IGF-1R-WT) COMPLEX WITH A CARBON-LINKED PROLINE ISOSTERE INHIBITOR (11B) | HORMONE/GROWTH FACTOR, IGF-1R, KINASE DOMAIN, TRANSFERASE
3nw6:A (PRO996) to (LYS1100) CRYSTAL STRUCTURE OF INSULIN-LIKE GROWTH FACTOR 1 RECEPTOR (IGF-1R-WT) COMPLEX WITH A CARBON-LINKED PROLINE ISOSTERE INHIBITOR (11A) | HORMONE/GROWTH FACTOR, IGF-1R, KINASE DOMAIN, TRANSFERASE
3nw7:A (PRO996) to (LYS1100) CRYSTAL STRUCTURE OF INSULIN-LIKE GROWTH FACTOR 1 RECEPTOR (IGF-1R-WT) COMPLEX WITH A CARBON-LINKED PROLINE ISOSTERE INHIBITOR (34) | HORMONE/GROWTH FACTOR, IGF-1R, KINASE DOMAIN, TRANSFERASE
3nyv:A (GLY63) to (LYS169) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH NON-SPECIFIC INHIBITOR WHI-P180 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3o2m:A (GLY38) to (GLY146) CRYSTAL STRUCTURE OF JNK1-ALPHA1 ISOFORM COMPLEX WITH A BIARYL TETRAZOL (A-82118) | SERINE THREONINE PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, KINASE-INHIBITOR COMPLEX, TRANSFERASE-INHIBITOR COMPLEX
4cqg:A (ALA23) to (VAL112) THE CRYSTAL STRUCTURE OF MPK38 IN COMPLEX WITH OTSSP167, AN ORALLY-ADMINISTRATIVE MELK SELECTIVE INHIBITOR | TRANSFERASE
3d7t:A (GLY207) to (ASN309) STRUCTURAL BASIS FOR THE RECOGNITION OF C-SRC BY ITS INACTIVATOR CSK | CSK SRC TYROSINE KINASE, ATP-BINDING, CYTOPLASM, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, ALTERNATIVE SPLICING, LIPOPROTEIN, MYRISTATE, PROTO- ONCOGENE
3d7t:B (GLU280) to (LEU358) STRUCTURAL BASIS FOR THE RECOGNITION OF C-SRC BY ITS INACTIVATOR CSK | CSK SRC TYROSINE KINASE, ATP-BINDING, CYTOPLASM, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, ALTERNATIVE SPLICING, LIPOPROTEIN, MYRISTATE, PROTO- ONCOGENE
3d7u:A (GLY207) to (ASN309) STRUCTURAL BASIS FOR THE RECOGNITION OF C-SRC BY ITS INACTIVATOR CSK | CSK C-SRC TYROSINE KINASE, ATP-BINDING, KINASE, MEMBRANE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, LIPOPROTEIN, MYRISTATE, PROTO-ONCOGENE
3d7u:B (GLY284) to (TYR357) STRUCTURAL BASIS FOR THE RECOGNITION OF C-SRC BY ITS INACTIVATOR CSK | CSK C-SRC TYROSINE KINASE, ATP-BINDING, KINASE, MEMBRANE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, LIPOPROTEIN, MYRISTATE, PROTO-ONCOGENE
3d7u:C (GLY207) to (ASN309) STRUCTURAL BASIS FOR THE RECOGNITION OF C-SRC BY ITS INACTIVATOR CSK | CSK C-SRC TYROSINE KINASE, ATP-BINDING, KINASE, MEMBRANE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, LIPOPROTEIN, MYRISTATE, PROTO-ONCOGENE
3d7u:D (GLY284) to (TYR357) STRUCTURAL BASIS FOR THE RECOGNITION OF C-SRC BY ITS INACTIVATOR CSK | CSK C-SRC TYROSINE KINASE, ATP-BINDING, KINASE, MEMBRANE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, LIPOPROTEIN, MYRISTATE, PROTO-ONCOGENE
4cva:A (SER536) to (ALA634) MPS1 KINASE WITH 3-AMINOPYRIDIN-2-ONE INHIBITORS | TRANSFERASE, FRAGMENT, INHIBITOR
4tn6:B (GLY21) to (ASN123) CK1D IN COMPLEX WITH INHIBITOR | SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3dak:A (ALA29) to (GLY116) CRYSTAL STRUCTURE OF DOMAIN-SWAPPED OSR1 KINASE DOMAIN | SERINE/THREONINE PROTEIN KINASE, STE20, DOMAIN-SWAPPING, ATP-BINDING, KINASE, MAGNESIUM, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
3dak:D (THR28) to (GLY116) CRYSTAL STRUCTURE OF DOMAIN-SWAPPED OSR1 KINASE DOMAIN | SERINE/THREONINE PROTEIN KINASE, STE20, DOMAIN-SWAPPING, ATP-BINDING, KINASE, MAGNESIUM, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
3od6:X (SER37) to (ASP145) CRYSTAL STRUCTURE OF P38ALPHA Y323T ACTIVE MUTANT | MAP KINASE, P38, TCR INDUCED ACTIVATION, TYR-323 PHOSPHORYLATION, KINASE FOLD, KINASE, PHOSPHORYLAITON, TRANSFERASE
3dbq:A (SER536) to (ALA634) CRYSTAL STRUCTURE OF TTK KINASE DOMAIN | MPS1 STRUCTURE, KINASE ACTIVATION, PHOSPHORYLATION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE
3oez:A (GLY279) to (LEU358) CRYSTAL STRUCTURE OF THE L317I MUTANT OF THE CHICKEN C-SRC TYROSINE KINASE DOMAIN COMPLEXED WITH IMATINIB | C-SRC L317I MUTANT, TYROSINE KINASE, IMATINIB, TRANSFERASE
4d28:C (PHE22) to (GLY129) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF SNRK3.11 AT5G35410 | TRANSFERASE, SALT STRESS, SODIUM TRANSPORT, ION HOMEOSTASIS
3dk3:A (GLY254) to (SER336) CRYSTAL STRUCTURE OF MUTANT ABL KINASE DOMAIN IN COMPLEX WITH SMALL MOLECULE FRAGMENT | DRUG DISCOVERY, ABL KINASE, FRAGMENT BASED, ALTERNATIVE SPLICING, ATP-BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3dk3:B (GLU258) to (SER336) CRYSTAL STRUCTURE OF MUTANT ABL KINASE DOMAIN IN COMPLEX WITH SMALL MOLECULE FRAGMENT | DRUG DISCOVERY, ABL KINASE, FRAGMENT BASED, ALTERNATIVE SPLICING, ATP-BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3dk6:A (GLY254) to (SER336) CRYSTAL STRUCTURE OF MUTANT ABL KINASE DOMAIN IN COMPLEX WITH SMALL MOLECULE FRAGMENT | DRUG DISCOVERY, ABL KINASE, FRAGMENT BASED, ALTERNATIVE SPLICING, ATP-BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3dk6:B (GLU255) to (SER336) CRYSTAL STRUCTURE OF MUTANT ABL KINASE DOMAIN IN COMPLEX WITH SMALL MOLECULE FRAGMENT | DRUG DISCOVERY, ABL KINASE, FRAGMENT BASED, ALTERNATIVE SPLICING, ATP-BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
4d2r:A (PRO1026) to (LYS1130) HUMAN IGF IN COMPLEX WITH A DYRK1B INHIBITOR | TRANSFERASE, KINASE, INHIBITOR, ONCOLOGY
4d2s:A (SER537) to (GLY642) HUMAN TTK IN COMPLEX WITH A DYRK1B INHIBITOR | TRANSFERASE, ONCOLOGY
4d2v:B (PHE22) to (VAL112) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN
4tw9:A (GLY21) to (ASN123) DIFLUORO-DIOXOLO-BENZOIMIDAZOL-BENZAMIDES AS POTENT INHIBITORS OF CK1DELTA AND EPSILON WITH NANOMOLAR INHIBITORY ACTIVITY ON CANCER CELL PROLIFERATION | TRANSFERASE, CK1DELTA, CK1EPSILON, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR
3oom:A (GLY220) to (ILE321) CRYSTAL STRUCTURE OF THE ACVR1 KINASE DOMAIN IN COMPLEX WITH THE IMIDAZO[1,2-B]PYRIDAZINE INHIBITOR K00507 | PROTEIN KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4d9t:A (SER434) to (GLY534) RSK2 C-TERMINAL KINASE DOMAIN WITH INHIBITOR (E)-METHYL 3-(4-AMINO-7- (3-HYDROXYPROPYL)-5-P-TOLYL-7H-PYRROLO[2,3-D]PYRIMIDIN-6-YL)-2- CYANOACRYLATE | KINASE, INHIBITOR, REVERSIBLE, THIOL, PHOSPHORYLATION, MIGRATION,, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4dbn:A (GLY468) to (GLU544) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN B-RAF WITH A [1, 3]THIAZOLO[5,4-B]PYRIDINE DERIVATIVE | KINASE DRUG COMPLEX, SER/THR KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4dbn:B (LYS472) to (GLU544) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN B-RAF WITH A [1, 3]THIAZOLO[5,4-B]PYRIDINE DERIVATIVE | KINASE DRUG COMPLEX, SER/THR KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3otv:D (GLN45) to (GLY145) CRYSTAL STRUCTURE OF THE INTRACELLULAR DOMAIN OF RV3910 FROM MYCOBACTERIUM TUBERCULOSIS | PEPTIDOGLYCAN, SER/THR KINASE, PSEUDOKINASE, REGULATION, MEMBRANE, TRANSFERASE
3oun:B (GLN45) to (GLY145) CRYSTAL STRUCTURE OF THE FHAA FHA DOMAIN COMPLEXED WITH THE INTRACELLULAR DOMAIN OF RV3910 | PEPTIDOGLYCAN, SER/THR KINASE, PSEUDOKINASE, FHA DOMAIN, REGULATION, PHOSPHORYLATION, MEMBRANE ASSOCIATED INTRACELLULAR, PROTEIN BINDING- TRANSFERASE COMPLEX
4u40:A (GLN38) to (HIS148) MITOGEN-ACTIVATED PROTEIN KINASE KINASE KINASE KINASE 4 (MAP4K4) BOUND TO AMPPNP | KINASE, TRANSFERASE
4u43:A (GLY37) to (HIS148) MAP4K4 IN COMPLEX WITH INHIBITOR (COMPOUND 6) | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4u45:A (GLY37) to (HIS148) MAP4K4 IN COMPLEX WITH INHIBITOR (COMPOUND 25) | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4deg:A (GLY1090) to (LYS1199) CRYSTAL STRUCTURE OF C-MET IN COMPLEX WITH TRIAZOLOPYRIDAZINE INHIBITOR 2 | PROTO-ONCOGENE, RECEPTOR TYROSINE KINASE, RTK, ATP-BINDING, HEPATOCYTE GROWTH FACTOR/SCATTER FACTOR, HGF/SF, PHOSPHOPROTEIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3oxi:A (GLY76) to (GLY184) DESIGN AND SYNTHESIS OF DISUBSTITUTED THIOPHENE AND THIAZOLE BASED INHIBITORS OF JNK FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES | JNK INHIBITORS, NEURODEGENERATIVE DISEASES, KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3oy3:A (GLU255) to (SER336) CRYSTAL STRUCTURE OF ABL T315I MUTANT KINASE DOMAIN BOUND WITH A DFG- OUT INHIBITOR AP24589 | PROTEIN-INHIBITOR COMPLEX, PROTEIN KINASE TWO-DOMAIN FOLD, PHOSPHOTRANSFERASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3oy3:B (GLU255) to (SER336) CRYSTAL STRUCTURE OF ABL T315I MUTANT KINASE DOMAIN BOUND WITH A DFG- OUT INHIBITOR AP24589 | PROTEIN-INHIBITOR COMPLEX, PROTEIN KINASE TWO-DOMAIN FOLD, PHOSPHOTRANSFERASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5hie:A (THR470) to (GLU545) BRAF KINASE DOMAIN B3AC LOOP DELETION MUTANT IN COMPLEX WITH DABRAFENIB | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hie:C (THR470) to (GLU545) BRAF KINASE DOMAIN B3AC LOOP DELETION MUTANT IN COMPLEX WITH DABRAFENIB | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hie:D (THR470) to (GLU545) BRAF KINASE DOMAIN B3AC LOOP DELETION MUTANT IN COMPLEX WITH DABRAFENIB | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3p7a:A (GLY36) to (ASP145) P38 INHIBITOR-BOUND | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hu9:A (GLU258) to (ASN336) CRYSTAL STRUCTURE OF ABL1 IN COMPLEX WITH CHMFL-074 | ABL, BCR-ABL, CHMFL-074, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4dt8:B (ILE35) to (ILE133) CRYSTAL STRUCTURE OF AMINOGLYCOSIDE-2''-PHOSPHOTRANSFERASE TYPE IVA IN COMPLEX WITH ADENOSINE | AMINOGLYCOSIDE KINASE, TRANSFERASE
4dt9:A (ILE35) to (ILE133) CRYSTAL STRUCTURE OF AMINOGLYCOSIDE-2''-PHOSPHOTRANSFERASE TYPE IVA IN COMPLEX WITH GUANOSINE | AMINOGLYCOSIDE KINASE, TRANSFERASE
5hzn:A (PRO1023) to (LYS1127) STRUCTURE OF NVP-AEW541 IN COMPLEX WITH IGF-1R KINASE | INHIBITOR, KINASE, TRANSFERASE
5hzn:D (PRO1023) to (LYS1127) STRUCTURE OF NVP-AEW541 IN COMPLEX WITH IGF-1R KINASE | INHIBITOR, KINASE, TRANSFERASE
5hzn:H (PRO1023) to (LYS1127) STRUCTURE OF NVP-AEW541 IN COMPLEX WITH IGF-1R KINASE | INHIBITOR, KINASE, TRANSFERASE
5i3o:A (SER63) to (CYS172) CRYSTAL STRUCTURE OF BMP-2-INDUCIBLE KINASE IN COMPLEX WITH AN INDAZOLE INHIBITOR | TRANSFERASE, PROTEIN KINASE DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5i3o:B (SER63) to (CYS172) CRYSTAL STRUCTURE OF BMP-2-INDUCIBLE KINASE IN COMPLEX WITH AN INDAZOLE INHIBITOR | TRANSFERASE, PROTEIN KINASE DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5i3r:A (SER63) to (CYS172) CRYSTAL STRUCTURE OF BMP-2-INDUCIBLE KINASE IN COMPLEX WITH AN INDAZOLE INHIBITOR | TRANSFERASE, PROTEIN KINASE DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5i3r:B (SER63) to (CYS172) CRYSTAL STRUCTURE OF BMP-2-INDUCIBLE KINASE IN COMPLEX WITH AN INDAZOLE INHIBITOR | TRANSFERASE, PROTEIN KINASE DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5i4n:A (GLY562) to (THR668) CRYSTAL STRUCTURE OF THE E596A V617F MUTANT JAK2 PSEUDOKINASE DOMAIN BOUND TO MG-ATP | TRANSFERASE, PSEUDOKINASE, ATP BINDING
4ump:B (ALA23) to (VAL112) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE
4umt:A (PHE22) to (VAL112) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN
3piz:A (GLY414) to (ARG492) CRYSTAL STRUCTURE OF BTK KINASE DOMAIN COMPLEXED WITH (5-AMINO-1-O- TOLYL-1H-PYRAZOL-4-YL)-[3-(1-METHANESULFONYL-PIPERIDIN-4-YL)-PHENYL]- METHANONE | HELIX C-IN, DFG-IN, TRANSFERASE, TRANSFERASE-INHIBITOR COMPLEX
5i5z:A (LYS37) to (TRP146) CDK8-CYCC IN COMPLEX WITH 8-(1-METHYL-2,2-DIOXO-2,3-DIHYDRO-1H-2L6- BENZO[C]ISOTHIAZOL-5-YL)-[1,6]NAPHTHYRIDINE-2-CARBOXYLIC ACID METHYLAMIDE | CDK8 KINASE / CYCLIN C, TRANSFERASE
4dym:A (GLY220) to (HIS320) CRYSTAL STRUCTURE OF THE ACVR1 KINASE DOMAIN IN COMPLEX WITH THE IMIDAZO[1,2-B]PYRIDAZINE INHIBITOR K00135 | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e26:A (LYS473) to (SER571) BRAF IN COMPLEX WITH AN ORGANIC INHIBITOR 7898734 | KINASE, INHIBITOR, ONCOPROTEIN, MELANOMA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e26:B (GLY469) to (GLU545) BRAF IN COMPLEX WITH AN ORGANIC INHIBITOR 7898734 | KINASE, INHIBITOR, ONCOPROTEIN, MELANOMA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ppk:B (LYS473) to (GLU545) HUMAN B-RAF KINASE IN COMPLEX WITH A NON-OXIME FUROPYRIDINE INHIBITOR | PROTEIN KINASE, B-RAF ATP-COMPETITIVE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3ppz:A (GLY563) to (ASP647) CRYSTAL STRUCTURE OF CTR1 KINASE DOMAIN IN COMPLEX WITH STAUROSPORINE | KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
3ppz:B (THR564) to (ASN667) CRYSTAL STRUCTURE OF CTR1 KINASE DOMAIN IN COMPLEX WITH STAUROSPORINE | KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
4e4m:A (GLY861) to (ARG971) JAK2 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 30 | O-PHOSPHOTYROSINE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e4m:D (SER862) to (THR969) JAK2 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 30 | O-PHOSPHOTYROSINE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e4x:A (THR470) to (GLU545) CRYSTAL STRUCTURE OF B-RAF KINASE DOMAIN IN COMPLEX WITH A DIHYDROPYRIDO[2,3-D]PYRIMIDINONE-BASED INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4e4x:B (LYS473) to (GLU545) CRYSTAL STRUCTURE OF B-RAF KINASE DOMAIN IN COMPLEX WITH A DIHYDROPYRIDO[2,3-D]PYRIMIDINONE-BASED INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3prf:A (LYS473) to (GLU545) CRYSTAL STRUCTURE OF HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH A NON- OXIME FUROPYRIDINE INHIBITOR | PROTEIN KINASE, ATP-COMPETITIVE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3prf:B (LYS473) to (GLU545) CRYSTAL STRUCTURE OF HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH A NON- OXIME FUROPYRIDINE INHIBITOR | PROTEIN KINASE, ATP-COMPETITIVE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ih5:A (ASP22) to (ASN123) HUMAN CASEIN KINASE 1 ISOFORM DELTA (KINASE DOMAIN) IN COMPLEX WITH EPIBLASTIN A | KINASE DOMAIN, STEM CELL REPROGRAMMING, KINASE INHIBITOR COMPLEX, TRANSFERASE
5ih6:A (ASP22) to (SER121) HUMAN CASEIN KINASE 1 ISOFORM DELTA (KINASE DOMAIN) IN COMPLEX WITH EPIBLASTIN A DERIVATIVE | KINASE DOMAIN, STEM CELL REPROGRAMMING, KINASE INHIBITOR COMPLEX, TRANSFERASE
5iha:A (ALA23) to (VAL112) MELK IN COMPLEX WITH NVS-MELK8F | KINASE UBA DOMAIN INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ihc:A (ALA23) to (VAL112) MELK IN COMPLEX WITH NVS-MELK12B | KINASE UBA DOMAIN INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3psd:A (THR470) to (GLU545) NON-OXIME PYRAZOLE BASED INHIBITORS OF B-RAF KINASE | KINASE, ATP-BINDING, CARDIOMYOPATHY, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, ZINC-FINGER, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3psd:B (GLY469) to (GLU545) NON-OXIME PYRAZOLE BASED INHIBITORS OF B-RAF KINASE | KINASE, ATP-BINDING, CARDIOMYOPATHY, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, ZINC-FINGER, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5ikw:A (SER63) to (CYS172) CRYSTAL STRUCTURE OF BMP-2-INDUCIBLE KINASE IN COMPLEX WITH AN INDAZOLE INHIBITOR | TRANSFERASE, PROTEIN KINASE DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ehe:A (LYS473) to (GLU545) B-RAF KINASE DOMAIN IN COMPLEX WITH AN AMINOTHIENOPYRIMIDINE-BASED INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ehe:B (LYS473) to (GLU545) B-RAF KINASE DOMAIN IN COMPLEX WITH AN AMINOTHIENOPYRIMIDINE-BASED INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ehg:B (LYS473) to (GLU545) B-RAF KINASE DOMAIN IN COMPLEX WITH AN AMINOPYRIDIMINE-BASED INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ej7:B (THR39) to (SER133) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, ATP-BOUND | CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR
4ej7:C (THR39) to (SER133) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, ATP-BOUND | CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR
3pyy:B (GLU274) to (ASN355) DISCOVERY AND CHARACTERIZATION OF A CELL-PERMEABLE, SMALL-MOLECULE C- ABL KINASE ACTIVATOR THAT BINDS TO THE MYRISTOYL BINDING SITE | TYROSINE KINASE, TRANSFERASE
3q2j:A (LYS30) to (ILE125) CRYSTAL STRUCTURE OF 3',5"-AMINOGLYCOSIDE PHOSPHOTRANSFERASE TYPE IIIA PROTEIN KINASE INHIBITOR CKI-7 COMPLEX | SER/THR/TYR PROTEIN KINASE, KINASE, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3q2j:B (LYS30) to (ILE125) CRYSTAL STRUCTURE OF 3',5"-AMINOGLYCOSIDE PHOSPHOTRANSFERASE TYPE IIIA PROTEIN KINASE INHIBITOR CKI-7 COMPLEX | SER/THR/TYR PROTEIN KINASE, KINASE, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3q4c:B (THR469) to (GLU544) CRYSTAL STRUCTURE OF WILD TYPE BRAF KINASE DOMAIN IN COMPLEX WITH ORGANOMETALLIC INHIBITOR CNS292 | KINASE, INHIBITOR, ONCOPROTEIN, MELANOMA, KINASE-KINASE INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3q4t:A (GLY204) to (GLU305) CRYSTAL STRUCTURE OF ACTIVIN RECEPTOR TYPE-IIA (ACVR2A) KINASE DOMAIN IN COMPLEX WITH DORSOMORPHIN | STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, TRANSFERASE
3q4u:A (GLY220) to (ILE321) CRYSTAL STRUCTURE OF THE ACVR1 KINASE DOMAIN IN COMPLEX WITH LDN- 193189 | STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, TRANSFERASE
3q4u:B (GLY220) to (HIS320) CRYSTAL STRUCTURE OF THE ACVR1 KINASE DOMAIN IN COMPLEX WITH LDN- 193189 | STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, TRANSFERASE
3q6w:A (GLY1095) to (LYS1199) STRUCTURE OF DUALLY-PHOSPHORYLATED MET RECEPTOR KINASE IN COMPLEX WITH AN MK-2461 ANALOG WITH SPECIFICITY FOR THE ACTIVATED RECEPTOR | TYROSINE KINASE, TWO PHOSPHOTYROSINE RESIUDES, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3q96:A (GLY469) to (GLU545) B-RAF KINASE DOMAIN IN COMPLEX WITH A TETRAHYDRONAPHTHALENE INHIBITOR | DESIGN, OPTIMIZATION, POTENT, ORALLY BIOAVAILABLE, TETRAHYDRONAPHTHALENE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4f0i:B (ALA526) to (HIS644) CRYSTAL STRUCTURE OF APO TRKA | TYROSINE KINASE, ROSSMANN FOLD, TRANSFERASE
3qgw:B (GLY375) to (PHE454) CRYSTAL STRUCTURE OF ITK KINASE BOUND TO AN INHIBITOR | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5j5t:A (GLY28) to (GLY131) GLK CO-CRYSTAL STRUCTURE WITH AMINOPYRROLOPYRIMIDINE INHIBITOR | PROTEIN KINSAE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4f7l:A (GLY33) to (TRP146) CRYSTAL STRUCTURE OF HUMAN CDK8/CYCC IN COMPLEX WITH COMPOUND 2 (TERT- BUTYL [3-({[3-TERT-BUTYL-1-(4-METHYLPHENYL)-1H-PYRAZOL-5- YL]CARBAMOYL}AMINO)PROPYL]CARBAMATE) | PROTEIN KINASE COMPLEX, PROTEROS, TRANSFERASE-TRANSCRIPTION-INHIBITOR COMPLEX
4uwg:A (LEU616) to (TYR707) DISCOVERY OF (2S)-8-((3R)-3-METHYLMORPHOLIN-4-YL)-1-(3- METHYL-2-OXO-BUTYL)-2-(TRIFLUOROMETHYL)-3,4-DIHYDRO-2H- PYRIMIDO(1,2-A)PYRIMIDIN-6-ONE: A NOVEL POTENT AND SELECTIVE INHIBITOR OF VPS34 FOR THE TREATMENT OF SOLID TUMORS | TRANSFERASE
3qqu:A (PRO1023) to (LYS1127) COCRYSTAL STRUCTURE OF UNPHOSPHORYLATED IGF WITH PYRIMIDINE 8 | IGF, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qqu:B (PRO1023) to (LYS1127) COCRYSTAL STRUCTURE OF UNPHOSPHORYLATED IGF WITH PYRIMIDINE 8 | IGF, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qri:B (GLU255) to (ASN336) THE CRYSTAL STRUCTURE OF HUMAN ABL1 KINASE DOMAIN IN COMPLEX WITH DCC- 2036 | ABL1, KINASE, KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4feu:C (THR39) to (SER133) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR ANTHRAPYRAZOLONE SP600125 | ANTHRAPYRAZOLONE, SP600125, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4few:A (THR39) to (SER133) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR PYRAZOLOPYRIMIDINE PP2 | PYRAZOLOPYRIMIDINE, PP2, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4few:B (THR39) to (PRO135) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR PYRAZOLOPYRIMIDINE PP2 | PYRAZOLOPYRIMIDINE, PP2, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4few:E (THR39) to (PRO135) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR PYRAZOLOPYRIMIDINE PP2 | PYRAZOLOPYRIMIDINE, PP2, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fex:E (THR39) to (SER133) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR TYRPHOSTIN AG1478 | TYRPHOSTIN, 4-ANILINOQUINAZOLINE, TYRPHOSTIN AG1478, AG1478, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qup:A (GLY520) to (ASN640) INHIBITOR BOUND STRUCTURE OF THE KINASE DOMAIN OF THE MURINE RECEPTOR TYROSINE KINASE TYRO3 (SKY) | PROTEIN KINASE INHIBITOR, RECEPTOR TYROSINE KINASE, SPIROCYCLE, KINASE DOMAIN, PHOSPHOTRANSFER, GAS6 LIGAND, CYTOPLASMIC SURFACE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fg7:A (SER32) to (GLY136) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE I 1-293 IN COMPLEX WITH ATP | CAMK, CALMODULIN, AUTOINHIBITION, REGULATION MECHANISM, KINASE, TRANSFERASE
4w7p:D (LEU92) to (SER191) CRYSTAL STRUCTURE OF ROCK 1 BOUND TO YB-15-QD37 | INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fku:A (GLY16) to (ARG122) CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH OXINDOLE INHIBITOR | ALPHA AND BETA PROTEIN (A+B), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5jeb:A (VAL714) to (ASP806) CRYSTAL STRUCTURE OF EGFR TYROSINE KINASE DOMAIN WITH NOVEL INHIBITOR OF ACTIVE STATE OF HER2 | INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5jms:A (GLY63) to (LYS169) CRYSTAL STRUCTURE OF TGCDPK1 BOUND TO CGP060476 | KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, HYDROLASE
5jn2:A (GLY63) to (LYS169) CRYSTAL STRUCTURE OF TGCDPK1 BOUND TO NVPACU106 | KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, HYDROLASE
3rin:A (ASP88) to (GLY219) P38 KINASE CRYSTAL STRUCTURE IN COMPLEX WITH SMALL MOLECULE INHIBITOR | P38 MAP KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5jt2:B (LYS473) to (GLU545) BRAFV600E KINASE DOMAIN IN COMPLEX WITH CHEMICALLY LINKED VEMURAFENIB INHIBITOR VEM-BISAMIDE | KINASE, DIMER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5jt2:C (GLY469) to (GLU545) BRAFV600E KINASE DOMAIN IN COMPLEX WITH CHEMICALLY LINKED VEMURAFENIB INHIBITOR VEM-BISAMIDE | KINASE, DIMER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fza:B (GLY36) to (LYS139) CRYSTAL STRUCTURE OF MST4-MO25 COMPLEX | SCAFFOLD PROTEIN, PROTEIN SER/THR KINASE, ATP BINDING, SIGNALING PROTEIN-TRANSFERASE COMPLEX
4fzf:B (GLY36) to (LYS139) CRYSTAL STRUCTURE OF MST4-MO25 COMPLEX WITH DKI | SCAFFOLD PROTEIN, PROTEIN SER/THR KINASE, ATP BINDING, SIGNALING PROTEIN-TRANSFERASE-INHIBITOR COMPLEX
4g31:A (GLY604) to (GLY931) CRYSTAL STRUCTURE OF GSK6414 BOUND TO PERK (R587-R1092, DELETE A660- T867) AT 2.28 A RESOLUTION | DELETION MUTANT, CATALYTIC DOMAIN, SYNTHETIC INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4g34:A (GLY604) to (GLY931) CRYSTAL STRUCTURE OF GSK6924 BOUND TO PERK (R587-R1092, DELETE A660- T867) AT 2.70 A RESOLUTION | DELETION MUTANT, CATALYTIC DOMAIN, SYNTHETIC INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5jzj:A (SER424) to (ASN506) CRYSTAL STRUCTURE OF DCLK1-KD IN COMPLEX WITH AMPPN | KINASE, DOUBLECORTIN, TRANSFERASE
5k5x:A (GLY610) to (ASN813) CRYSTAL STRUCTURE OF HUMAN PDGFRA | TYROSINE KINASE, AUTOINHIBITION, TRANSFERASE
4g9c:A (THR470) to (GLU545) HUMAN B-RAF KINASE DOMAIN BOUND TO A TYPE II PYRAZOLOPYRIDINE INHIBITOR | DFG-OUT, INHIBITOR, TYPE II, TRANSFERASE, KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4g9c:B (LYS473) to (GLU545) HUMAN B-RAF KINASE DOMAIN BOUND TO A TYPE II PYRAZOLOPYRIDINE INHIBITOR | DFG-OUT, INHIBITOR, TYPE II, TRANSFERASE, KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4g9r:A (GLY469) to (SER571) B-RAF V600E KINASE DOMAIN BOUND TO A TYPE II DIHYDROQUINAZOLINE INHIBITOR | INHIBITOR, TYPE II, TRANSFERASE, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gg5:A (GLY1090) to (LYS1199) CRYSTAL STRUCTURE OF CMET IN COMPLEX WITH NOVEL INHIBITOR | CMET INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gkh:C (THR39) to (SER133) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR 1-NA-PP1 | PYRAZOLOPYRIMIDINE, 1-NA-PP1, BUMPED KINASE INHIBITOR, BKI, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR
4gkh:I (THR39) to (SER133) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR 1-NA-PP1 | PYRAZOLOPYRIMIDINE, 1-NA-PP1, BUMPED KINASE INHIBITOR, BKI, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR
4gkh:L (THR39) to (PRO135) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR 1-NA-PP1 | PYRAZOLOPYRIMIDINE, 1-NA-PP1, BUMPED KINASE INHIBITOR, BKI, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR
4gl9:B (GLY861) to (ARG971) CRYSTAL STRUCTURE OF INHIBITORY PROTEIN SOCS3 IN COMPLEX WITH JAK2 KINASE DOMAIN AND FRAGMENT OF GP130 INTRACELLULAR DOMAIN | KINASE INHIBITOR RECEPTOR CYTOKINE SIGNALLING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gmy:A (PHE860) to (ARG971) JAK2 KINASE (JH1 DOMAIN) IN COMPLEX WITH 2,6-DICHLORO-N-{2- [(CYCLOPROPYLCARBONYL)AMINO]PYRIDIN-4-YL}BENZAMIDE | JAK2, JH1 KINASE DOMAIN, TYROSINE KINASE, PHOSPHOTRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5kx8:B (GLY198) to (HIS306) IRAK4-INHIBITOR CO-STRUCTURE | KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5l2i:A (GLY25) to (ARG140) THE X-RAY CO-CRYSTAL STRUCTURE OF HUMAN CDK6 AND PALBOCICLIB. | CYCLIN-DEPENDENT KINASE, KINASE INHIBITOR, KINASE SELECTIVITY, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5l4q:A (ALA58) to (HIS166) CRYSTAL STRUCTURE OF ADAPTOR PROTEIN 2 ASSOCIATED KINASE 1 (AAK1) IN COMPLEX WITH LKB1 (AAK1 DUAL INHIBITOR) | KINASE KINASE DOMAIN, TRANSFERASE
5l4q:B (ALA58) to (HIS166) CRYSTAL STRUCTURE OF ADAPTOR PROTEIN 2 ASSOCIATED KINASE 1 (AAK1) IN COMPLEX WITH LKB1 (AAK1 DUAL INHIBITOR) | KINASE KINASE DOMAIN, TRANSFERASE
5m55:A (ARG21) to (SER131) NEK2 BOUND TO ARYLAMINOPURINE 71 | PROTEIN KINASE, INHIBITOR, CENTROSOME SEPARATION, TRANSFERASE
5t6a:A (GLY63) to (LYS169) CRYSTAL STRUCTURE OF TGCDPK1 FROM TOXOPLASMA GONDII COMPLEXED WITH 5GA | STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPKS, SERINE/THREONINE PROTEIN KINASE, NUCLEOTIDE-BINDING, TRANSFERASE
5t6k:A (GLY63) to (LYS169) CRYSTAL STRUCTURE OF TGCDPK1 FROM TOXOPLASMA GONDII COMPLEXED WITH GW780159X | STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPKS, SERINE/THREONINE PROTEIN KINASE, NUCLEOTIDE-BINDING, TRANSFERASE
3ekk:A (GLY1013) to (LYS1127) INSULIN RECEPTOR KINASE COMPLEXED WITH AN INHIBITOR | INSULIN, TYROSINE KINASE, ATP-BINDING, CARBOHYDRATE METABOLISM, CLEAVAGE ON PAIR OF BASIC RESIDUES, DIABETES MELLITUS, DISEASE MUTATION, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE
2bdf:B (GLU280) to (LEU358) SRC KINASE IN COMPLEX WITH INHIBITOR AP23451 | SRC KINASE INHIBITOR, TRANSFERASE
2c0t:A (MET257) to (GLN332) SRC FAMILY KINASE HCK WITH BOUND INHIBITOR A-641359 | TRANSFERASE, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, SH2 DOMAIN, SH3 DOMAIN
4xhg:A (GLY21) to (SER123) STRUCTURE OF C. GLABRATA HRR25 BOUND TO ADP (FORMATE CONDITION) | CASEIN KINASE, MONOPOLIN, TRANSFERASE
2psq:A (ALA498) to (LYS621) CRYSTAL STRUCTURE OF UNPHOSPHORYLATED UNACTIVATED WILD TYPE FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, TRANSFERASE
2pui:B (LEU43) to (SER152) STRUCTURES OF 5-METHYLTHIORIBOSE KINASE REVEAL SUBSTRATE SPECIFICITY AND UNUSUAL MODE OF NUCLEOTIDE BINDING | 5-METHYLTHIORIBOSE KINASE, METHIONINE RECYCLING PATHWAY, TRANSFERASE
1cki:A (GLY24) to (ASN126) RECOMBINANT CASEIN KINASE I DELTA TRUNCATION MUTANT CONTAINING RESIDUES 1-317 | PROTEIN KINASE, PHOSPHOTRANSFERASE
1cki:B (GLY24) to (ASN126) RECOMBINANT CASEIN KINASE I DELTA TRUNCATION MUTANT CONTAINING RESIDUES 1-317 | PROTEIN KINASE, PHOSPHOTRANSFERASE
2qi8:A (GLY284) to (LEU358) CRYSTAL STRUCTURE OF DRUG RESISTANT SRC KINASE DOMAIN | SRC KINASE DOMAIN; DRUG RESISTANCE, SIGNALING PROTEIN, TRANSFERASE
3g6h:A (GLY279) to (LEU358) SRC THR338ILE INHIBITED IN THE DFG-ASP-OUT CONFORMATION | CANCER, IMATINIB RESISTANCE, DSA COMPOUNDS, KINASE, DFG-ASP- OUT, ALTERNATIVE SPLICING, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE
3g6h:B (GLY279) to (LEU358) SRC THR338ILE INHIBITED IN THE DFG-ASP-OUT CONFORMATION | CANCER, IMATINIB RESISTANCE, DSA COMPOUNDS, KINASE, DFG-ASP- OUT, ALTERNATIVE SPLICING, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE
4y0x:A (GLY163) to (GLY271) CRYSTAL STRUCTURE OF THE S/T PROTEIN KINASE PKNG FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH ADP | S/T PROTEIN KINASE, PKNG, TRANSFERASE
3gp0:A (SER37) to (GLY145) CRYSTAL STRUCTURE OF HUMAN MITOGEN ACTIVATED PROTEIN KINASE 11 (P38 BETA) IN COMPLEX WITH NILOTINIB | MITOGEN-ACTIVATED PROTEIN KINASE 11, P38B, P38BETA, PRKM11, SAPK2, SAPK2B, STRESS-ACTIVATED PROTEIN KINASE-2, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4y5q:A (LEU91) to (ILE178) ACTIVATED CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM CRYPTOSPORIDIUM PARVUM (CPCDPK1) IN COMPLEX WITH AMP | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, BUMPED KINASE INHIBITOR, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP
3tdw:A (TYR34) to (PHE130) THE GDP COMPLEX OF THE AMINOGLYCOSIDE 2'-PHOSPHOTRANSFERE-IIIA F108L MUTANT | KINASE, PHOSPHORYL TRANSFER, ANTIBIOTIC RESISTANCE, TRANSFERASE
3gu8:A (ALA25) to (GLN134) CRYSTAL STRUCTURE OF DAPKL93G WITH N6-CYCLOPENTYLADENOSINE | GATEKEEPER MUTANT, ALTERNATIVE SPLICING, ANK REPEAT, APOPTOSIS, ATP-BINDING, CALMODULIN-BINDING, CYTOPLASM, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4jg6:A (SER434) to (GLY534) RSK2 CTD BOUND TO 2-CYANO-3-(1H-INDAZOL-5-YL)ACRYLAMIDE | PROTEIN KINASE, PHOSPHORYLATION, COVALENT INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
1eh4:A (GLY24) to (GLU124) BINARY COMPLEX OF CASEIN KINASE-1 FROM S. POMBE WITH AN ATP COMPETITIVE INHIBITOR, IC261 | PROTEIN KINASE, CASEIN KINASE-1, PROTEIN-INHIBITOR BINARY COMPLEX, TRANSFERASE
1eh4:B (VAL25) to (GLU124) BINARY COMPLEX OF CASEIN KINASE-1 FROM S. POMBE WITH AN ATP COMPETITIVE INHIBITOR, IC261 | PROTEIN KINASE, CASEIN KINASE-1, PROTEIN-INHIBITOR BINARY COMPLEX, TRANSFERASE
1qcf:A (GLY279) to (GLN358) CRYSTAL STRUCTURE OF HCK IN COMPLEX WITH A SRC FAMILY- SELECTIVE TYROSINE KINASE INHIBITOR | TYROSINE KINASE-INHIBITOR COMPLEX, DOWN-REGULATED KINASE, ORDERED ACTIVATION LOOP
1qpd:A (GLY257) to (LEU336) STRUCTURAL ANALYSIS OF THE LYMPHOCYTE-SPECIFIC KINASE LCK IN COMPLEX WITH NON-SELECTIVE AND SRC FAMILY SELECTIVE KINASE INHIBITORS | ALPHA BETA FOLD, TRANSFERASE
4yne:A (ASP537) to (HIS645) (R)-2-PHENYLPYRROLIDINE SUBSTITUTE IMIDAZOPYRIDAZINES: A NEW CLASS OF POTENT AND SELECTIVE PAN-TRK INHIBITORS | KINASE, TRK, INHIBITOR, ONCOLOGY, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3udb:A (VAL34) to (MET134) CRYSTAL STRUCTURE OF SNRK2.6 | SNRK2.6, KINASE, ABA SIGNALING PATHWAY, ABI1, TRANSFERASE
3udb:C (VAL34) to (GLN135) CRYSTAL STRUCTURE OF SNRK2.6 | SNRK2.6, KINASE, ABA SIGNALING PATHWAY, ABI1, TRANSFERASE
3udb:E (VAL34) to (GLN135) CRYSTAL STRUCTURE OF SNRK2.6 | SNRK2.6, KINASE, ABA SIGNALING PATHWAY, ABI1, TRANSFERASE
2v7a:B (GLY254) to (ASN336) CRYSTAL STRUCTURE OF THE T315I ABL MUTANT IN COMPLEX WITH THE INHIBITOR PHA-739358 | KINASE, NUCLEUS, MYRISTATE, CYTOPLASM, MANGANESE, CELL ADHESION, METAL-BINDING, PROTO-ONCOGENE, TYROSINE-PROTEIN KINASE, CHROMOSOMAL REARRANGEMENT, TRANSFERASE, LIPOPROTEIN, POLYMORPHISM, CYTOSKELETON, MAGNESIUM, SH2 DOMAIN, SH3 DOMAIN, ATP-BINDING, NUCLEOTIDE-BINDING, ALTERNATIVE SPLICING, PHOSPHORYLATION, KINASE INHIBITOR, T315I ABL MUTANT
3hmi:A (GLU301) to (THR382) THE CRYSTAL STRUCTURE OF HUMAN ABL2 IN COMPLEX WITH 5-AMINO-3-{[4- (AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4- TRIAZOLE-1-CARBOTHIOAMIDE | TYROSINE KINASE, ABL, ABL2, ABELSON MURINE LEUKEMIA VIRAL ONCOGENE, ATP-BINDING, CELL ADHESION, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
4kbc:B (GLY21) to (ASN123) CK1D IN COMPLEX WITH {4-[3-(4-FLUOROPHENYL)-1H-PYRAZOL-4-YL]PYRIDIN-2- YL}METHANOL INHIBITOR | SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uzp:A (GLY21) to (ASN123) CRYSTAL STRUCTURE OF CK1D WITH PF670462 FROM P21 CRYSTAL FORM | CK1D, KINASE, INHIBITOR, PF670462, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uzp:B (GLY21) to (ASN123) CRYSTAL STRUCTURE OF CK1D WITH PF670462 FROM P21 CRYSTAL FORM | CK1D, KINASE, INHIBITOR, PF670462, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2g2f:B (GLU255) to (ASN336) A SRC-LIKE INACTIVE CONFORMATION IN THE ABL TYROSINE KINASE DOMAIN | PROTEIN KINASE, TRANSFERASE
1sm2:B (GLY375) to (PHE454) CRYSTAL STRUCTURE OF THE PHOSPHORYLATED INTERLEUKIN-2 TYROSINE KINASE CATALYTIC DOMAIN | PROTEIN KINASE, IMMUNOLOGY, TRANSFERASE
3i79:A (GLY63) to (LYS169) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) | PROTEIN KINASE, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, TRANSFERASE
2vz6:B (SER25) to (GLY130) STRUCTURE OF HUMAN CALCIUM CALMODULIN DEPENDENT PROTEIN KINASE TYPE II ALPHA (CAMK2A) IN COMPLEX WITH INDIRUBIN E804 | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, CELL JUNCTION, CELL MEMBRANE, LONG TERM POTENTIATION, BRAIN, KINASE, SYNAPSE, MEMBRANE, NMDA RECEPTOR SIGNALLING, PHOSPHOPROTEIN, CALMODULIN-BINDING, NUCLEOTIDE-BINDING
4zs0:A (LEU149) to (ARG251) HUMAN AURORA A CATALYTIC DOMAIN BOUND TO SB-6-OH | AURORA, KINASE, INHIBITOR, TRANSFERASE
4lg4:D (SER40) to (ARG141) STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5 | HIPPO, MST AUTOACTIVATION, DIMERIZATION, SIGNALING PROTEIN
3vs0:A (MET283) to (GLN358) CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRROLO-PYRIMIDINE INHIBITOR N-[4-(4-AMINO-7-CYCLOPENTYL-7H-PYRROLO[2,3-D]PYRIMIDIN-5-YL) PHENYL]BENZAMIDE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3vs6:A (MET283) to (GLN358) CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRAZOLO-PYRIMIDINE INHIBITOR TERT-BUTYL {4-[4-AMINO-1-(PROPAN-2-YL)-1H-PYRAZOLO[3,4- D]PYRIMIDIN-3-YL]-2-METHOXYPHENYL}CARBAMATE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5a4l:A (GLY171) to (ALA277) DYRK1A IN COMPLEX WITH FLUORO BENZOTHIAZOLE FRAGMENT | TRANSFERASE
2i0v:A (ALA599) to (ASN773) C-FMS TYROSINE KINASE IN COMPLEX WITH A QUINOLONE INHIBITOR | RECEPTOR TYROSINE KINASE, KINASE-INHIBITOR COMPLEX, TRANSFERASE
5aep:A (GLY861) to (ASP949) NOVEL PYRROLE CARBOXAMIDE INHIBITORS OF JAK2 AS POTENTIAL TREATMENT OF MYELOPROLIFERATIVE DISORDERS | TRANSFERASE, PROTEIN KINASE, JAK2, MYELOPROLIFERATIVE DISORDERS, TUMOUR CELL PROLIFERATION INHIBITION, ANTI-CANCER AGENTS
5ax9:A (GLY37) to (LYS148) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN TRAF2 AND NCK- INTERACTING PROTEIN KINASE IN COMPLEX WITH COMPUND 9 | INHIBITOR, KINASE, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4mxo:A (GLY279) to (LEU358) HUMAN SRC KINASE BOUND TO KINASE INHIBITOR BOSUTINIB | KINASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3zep:C (SER835) to (ARG944) CRYSTAL STRUCTURE OF JAK3 KINASE DOMAIN IN COMPLEX WITH A PYRROLOPYRAZINE-2-PHENYL ETHER INHIBITOR | TRANSFERASE, STAT5, STAT6, INTERLEUKIN-2, COMMON-GAMMA CHAIN, ATP SITE KINASE INHIBITOR, CANCER, SCID, SEVERE COMBINED IMMUNODEFICIENCY
5c9c:A (GLY468) to (GLU544) CRYSTAL STRUCTURE OF BRAF(V600E) IN COMPLEX WITH LY3009120 COMPND | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4o1p:A (GLY380) to (GLY477) CRYSTAL STRUCTURE OF RNASE L IN COMPLEX WITH 2-5A AND AMP-PNP | ANKYRIN REPEAT-KINASE-RNASE, RNA CLEAVAGE, 2-5A, TRANSFERASE, HYDROLASE
4o1p:C (GLY380) to (GLY477) CRYSTAL STRUCTURE OF RNASE L IN COMPLEX WITH 2-5A AND AMP-PNP | ANKYRIN REPEAT-KINASE-RNASE, RNA CLEAVAGE, 2-5A, TRANSFERASE, HYDROLASE
4o1p:D (GLY380) to (GLY477) CRYSTAL STRUCTURE OF RNASE L IN COMPLEX WITH 2-5A AND AMP-PNP | ANKYRIN REPEAT-KINASE-RNASE, RNA CLEAVAGE, 2-5A, TRANSFERASE, HYDROLASE
3k5v:A (GLU274) to (SER355) STRUCTURE OF ABL KINASE IN COMPLEX WITH IMATINIB AND GNF-2 | KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3kc3:A (LYS77) to (ASN181) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:G (LEU79) to (ILE170) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:I (LEU79) to (GLY171) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
5cwz:C (GLY37) to (LYS148) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN TRAF2 AND NCK- INTERACTING PROTEIN KINASE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2zm4:A (PHE256) to (LEU336) CRYSTAL STRUCTURE OF IMIDAZO QUINOXALINE 1 BOUND TO THE KINASE DOMAIN OF HUMAN LCK, ACTIVATED FORM (AUTO- PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE- BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3a2c:G (LEU79) to (ASN181) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3ad6:A (PHE256) to (LEU336) CRYSTAL STRUCTURE OF PYRAZOLO PYRIMIDINE DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
1yrp:A (PHE24) to (PHE119) CATALYTIC DOMAIN OF HUMAN ZIP KINASE PHOSPHORYLATED AT THR265 | KINASE FOLD, PHOSPHOTHREONINE, TRANSFERASE
1yrp:B (PHE24) to (PHE119) CATALYTIC DOMAIN OF HUMAN ZIP KINASE PHOSPHORYLATED AT THR265 | KINASE FOLD, PHOSPHOTHREONINE, TRANSFERASE
4ark:A (LYS84) to (LYS185) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN MAP KINASE KINASE 1 (MEK1) IN COMPLEX WITH A SMALL MOLECULE INHIBITOR AND ADP | TRANSFERASE, KINASE, INHIBITOR
4at3:A (GLY566) to (LEU654) CRYSTAL STRUCTURE OF TRKB KINASE DOMAIN IN COMPLEX WITH CPD5N | TRANSFERASE
4at5:A (ALA571) to (ALA656) CRYSTAL STRUCTURE OF TRKB KINASE DOMAIN IN COMPLEX WITH GW2580 | TRANSFERASE
1zws:A (ALA25) to (LYS134) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE | PROTEIN KINASE, TWINNING, TRANSFERASE
1zws:B (ALA25) to (LYS134) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE | PROTEIN KINASE, TWINNING, TRANSFERASE
1zws:C (ALA25) to (LYS134) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE | PROTEIN KINASE, TWINNING, TRANSFERASE
1zws:D (ALA25) to (LYS134) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE | PROTEIN KINASE, TWINNING, TRANSFERASE
1zws:E (ALA25) to (LYS134) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE | PROTEIN KINASE, TWINNING, TRANSFERASE
1zws:F (ALA25) to (LYS134) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE | PROTEIN KINASE, TWINNING, TRANSFERASE
1zws:G (ALA25) to (LYS134) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE | PROTEIN KINASE, TWINNING, TRANSFERASE
1zws:H (ALA25) to (LYS134) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE | PROTEIN KINASE, TWINNING, TRANSFERASE
3lvp:C (PRO1026) to (LYS1130) CRYSTAL STRUCTURE OF BISPHOSPHORYLATED IGF1-R KINASE DOMAIN (2P) IN COMPLEX WITH A BIS-AZAINDOLE INHIBITOR | PROTEIN KINASE, TYROSINE KINASE, TYROSINE PHOSPHORYLATION, PROTEIN- SUBSTRATE COMPLEX, TRANSFERASE
3att:A (GLU57) to (SER178) CRYSTAL STRUCTURE OF RV3168 WITH ATP | HYPOTHETICAL PROTEIN, PUTATIVE AMINOGLYCOSIDE PHOSPHORTRANSFERASE, TRANSFERASE
5ehl:A (SER537) to (GLY642) RAPID DISCOVERY OF PYRIDO[3,4-D]PYRIMIDINE INHIBITORS OF MONOPOLAR SPINDLE KINASE 1 (MPS1) USING A STRUCTURE-BASED HYDRIDIZATION APPROACH | SPINDLE ASSEMBLY CHECKPOINT (SAC), ONCOLOGY TARGET PYRIDO[3, 4- D]PYRIMIDINE BASED INHIBITORS SELECTIVE AGAINST MPS1, TRANSFERASE
5ei8:A (SER537) to (GLN640) RAPID DISCOVERY OF PYRIDO[3,4-D]PYRIMIDINE INHIBITORS OF MONOPOLAR SPINDLE KINASE 1 (MPS1) USING A STRUCTURE-BASED HYDRIDIZATION APPROACH | SPINDLE ASSEMBLY CHECKPOINT (SAC), ONCOLOGY TARGET PYRIDO[3, 4- D]PYRIMIDINE BASED INHIBITORS SELECTIVE AGAINST MPS1, TRANSFERASE
4bch:A (GLY31) to (LYS144) STRUCTURE OF CDK9 IN COMPLEX WITH CYCLIN T AND A 2-AMINO-4- HETEROARYL-PYRIMIDINE INHIBITOR | TRANSFERASE-CELL CYCLE COMPLEX, CDK-CYCLIN COMPLEX, TRANSCRIPTION-PROTEIN BINDING, STRUCTURE-BASED DRUG DESIGN
4qox:A (GLU83) to (ASN188) CRYSTAL STRUCTURE OF CDPK4 FROM PLASMODIUM FALCIPARUM, PF3D7_0717500 | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPK, PLASMODIUM, MALARIA, TRANSFERASE
3miy:A (LEU379) to (SER477) X-RAY CRYSTAL STRUCTURE OF ITK COMPLEXED WITH SUNITINIB | HELIX C-IN, TRANSFERASE
5eqe:B (LEU124) to (MET238) CRYSTAL STRUCTURE OF CHOLINE KINASE ALPHA-1 BOUND BY [4-[(4-METHYL-1, 4-DIAZEPAN-1-YL)METHYL]PHENYL]METHANAMINE (COMPOUND 11) | KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qrc:A (ALA484) to (LYS607) CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF FGF RECEPTOR 4 IN COMPLEX WITH PONATINIB | KINASE DOMAIN FOLD, CELL SIGNALING, PHOSPHOTRANSFERASE, PLASMAMEMBRANE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4bgg:A (GLY220) to (HIS320) CRYSTAL STRUCTURE OF THE ACVR1 KINASE IN COMPLEX WITH LDN-213844 | TRANSFERASE, INHIBITOR, BMP SIGNALLING
4bgg:B (GLY220) to (HIS320) CRYSTAL STRUCTURE OF THE ACVR1 KINASE IN COMPLEX WITH LDN-213844 | TRANSFERASE, INHIBITOR, BMP SIGNALLING
4bgg:C (GLY220) to (HIS320) CRYSTAL STRUCTURE OF THE ACVR1 KINASE IN COMPLEX WITH LDN-213844 | TRANSFERASE, INHIBITOR, BMP SIGNALLING
4bgg:D (GLY220) to (HIS320) CRYSTAL STRUCTURE OF THE ACVR1 KINASE IN COMPLEX WITH LDN-213844 | TRANSFERASE, INHIBITOR, BMP SIGNALLING
3bhh:A (SER26) to (GLY131) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE IIB ISOFORM 1 (CAMK2B) | CAMK2B, CAM2, CAMK2, CAM KINASE II BETA CHAIN, CAMK II BETA SUBUNIT, CALCIUM/CALMODULION DEPENDENT PROTEIN KINASE II BETA, EC:2.7.1.123, MGC29528, PROLINE RICH CALMODULIN DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, CALMODULIN- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
3bhh:B (SER26) to (GLY131) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE IIB ISOFORM 1 (CAMK2B) | CAMK2B, CAM2, CAMK2, CAM KINASE II BETA CHAIN, CAMK II BETA SUBUNIT, CALCIUM/CALMODULION DEPENDENT PROTEIN KINASE II BETA, EC:2.7.1.123, MGC29528, PROLINE RICH CALMODULIN DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, CALMODULIN- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
3bhh:C (VAL27) to (GLY131) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE IIB ISOFORM 1 (CAMK2B) | CAMK2B, CAM2, CAMK2, CAM KINASE II BETA CHAIN, CAMK II BETA SUBUNIT, CALCIUM/CALMODULION DEPENDENT PROTEIN KINASE II BETA, EC:2.7.1.123, MGC29528, PROLINE RICH CALMODULIN DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, CALMODULIN- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
3bhh:D (VAL27) to (GLY131) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE IIB ISOFORM 1 (CAMK2B) | CAMK2B, CAM2, CAMK2, CAM KINASE II BETA CHAIN, CAMK II BETA SUBUNIT, CALCIUM/CALMODULION DEPENDENT PROTEIN KINASE II BETA, EC:2.7.1.123, MGC29528, PROLINE RICH CALMODULIN DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, CALMODULIN- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
3biz:A (SER312) to (SER421) WEE1 KINASE COMPLEX WITH INHIBITOR PD331618 | KINASE DOMAIN, INHIBITOR COMPLEX, ATP-BINDING, CELL CYCLE, CELL DIVISION, MAGNESIUM, METAL-BINDING, MITOSIS, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3n4v:A (ILE35) to (ILE133) APO APH(2")-IVA FORM III | AMINOGLYCOSIDE, PHOSPHOTRANSFERASE, RESISTANCE, UNKNOWN FUNCTION
4c02:A (GLY220) to (HIS320) CRYSTAL STRUCTURE OF HUMAN ACVR1 (ALK2) IN COMPLEX WITH FKBP12.6 AND DORSOMORPHIN | TRANSFERASE-ISOMERASE COMPLEX, TRANSFERASE, DORSOMORPHIN,
4rfy:A (GLY414) to (GLN516) CRYSTAL STRUCTURE OF BTK KINASE DOMAIN COMPLEXED WITH 6- (DIMETHYLAMINO)-2-[2-(HYDROXYMETHYL)-3-[1-METHYL-5-[[5-(MORPHOLINE-4- CARBONYL)-2-PYRIDYL]AMINO]-6-OXO-3-PYRIDYL]PHENYL]-3,4- DIHYDROISOQUINOLIN-1-ONE | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5fxq:A (PRO1026) to (LYS1130) IGFR-1R COMPLEX WITH A PYRIMIDINE INHIBITOR. | TRANSFERASE
4d2t:A (LYS24) to (VAL112) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN, KINASE
4d2t:C (LYS24) to (VAL112) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN, KINASE
4d2t:D (PHE22) to (VAL112) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN, KINASE
4twc:A (ASP22) to (ASN123) 2-BENZAMIDO-N-(1H-BENZO[D]IMIDAZOL-2-YL)THIAZOLE-4- CARBOXAMIDE DERIVATIVES AS POTENT INHIBITORS OF CK1D/E | CK1D, CK1E, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, TRANSFERASE
3dpk:A (ALA599) to (ASN773) CFMS TYROSINE KINASE IN COMPLEX WITH A PYRIDOPYRIMIDINONE INHIBITOR | RECEPTOR TYROSINE KINASE, KINASE-INHIBITOR COMPLEX, ATP- BINDING, GLYCOPROTEIN, IMMUNOGLOBULIN DOMAIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, ALTERNATIVE SPLICING, CHROMOSOMAL REARRANGEMENT, CRANIOSYNOSTOSIS, DISEASE MUTATION, DWARFISM, HEPARIN-BINDING, KALLMANN SYNDROME
5hbj:A (GLY33) to (TRP146) CDK8-CYCC IN COMPLEX WITH 8-[2-AMINO-3-CHLORO-5-(1-METHYL-1H-INDAZOL- 5-YL)-PYRIDIN-4-YL]-2,8-DIAZA-SPIRO[4.5]DECAN-1-ONE | CDK8 KINASE / CYCLIN C, TRANSFERASE
4u42:A (GLN38) to (HIS148) MAP4K4 T181E MUTANT BOUND TO INHIBITOR COMPOUND 1 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3owe:B (LYS124) to (ASN211) CRYSTAL STRUCTURE OF STAPHYLOCOCCAL ENTEROTOXIN G (SEG) IN COMPLEX WITH A HIGH AFFINITY MUTANT MOUSE T-CELL RECEPTOR CHAIN | T-CELL RECEPTOR V BETA DOMAIN, COMPLEX STRUCTURE, IGG DOMAINS, B GRASP, VIRULENCE FACTORS, IMMUNE SYSTEM
3owe:H (LYS124) to (ASN211) CRYSTAL STRUCTURE OF STAPHYLOCOCCAL ENTEROTOXIN G (SEG) IN COMPLEX WITH A HIGH AFFINITY MUTANT MOUSE T-CELL RECEPTOR CHAIN | T-CELL RECEPTOR V BETA DOMAIN, COMPLEX STRUCTURE, IGG DOMAINS, B GRASP, VIRULENCE FACTORS, IMMUNE SYSTEM
3owe:J (LYS124) to (LEU210) CRYSTAL STRUCTURE OF STAPHYLOCOCCAL ENTEROTOXIN G (SEG) IN COMPLEX WITH A HIGH AFFINITY MUTANT MOUSE T-CELL RECEPTOR CHAIN | T-CELL RECEPTOR V BETA DOMAIN, COMPLEX STRUCTURE, IGG DOMAINS, B GRASP, VIRULENCE FACTORS, IMMUNE SYSTEM
5hx6:B (VAL31) to (GLY133) CRYSTAL STRUCTURE OF RIP1 KINASE WITH A BENZO[B][1,4]OXAZEPIN-4-ONE | KINASE, INHIBITOR COMPLEX, NON-HINGE BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3piy:A (GLY414) to (GLN516) CRYSTAL STRUCTURE OF BTK KINASE DOMAIN COMPLEXED WITH R406 | HELIX C-OUT, DFG-IN, TRANSFERASE, TRANSFERASE-INHIBITOR COMPLEX
4usf:B (LYS47) to (LYS150) HUMAN SLK WITH SB-440719 | TRANSFERASE
5ig1:A (SER30) to (ASN135) CRYSTAL STRUCTURE OF S. ROSETTA CAMKII KINASE DOMAIN | CA2+/CAM-DEPENDENT KINASE, CHOANOFLAGELLATE, TRANSFERASE
5ig1:B (PHE29) to (ASN135) CRYSTAL STRUCTURE OF S. ROSETTA CAMKII KINASE DOMAIN | CA2+/CAM-DEPENDENT KINASE, CHOANOFLAGELLATE, TRANSFERASE
5ih4:A (ASP22) to (LYS122) HUMAN CASEIN KINASE 1 ISOFORM DELTA APO (KINASE DOMAIN) | KINASE DOMAIN, STEM CELL REPROGRAMMING, TRANSFERASE
4w4w:A (ILE77) to (GLY184) JNK2/3 IN COMPLEX WITH N-(2-METHYLPYRIDIN-4-YL)-3-{4- [(PHENYLCARBAMOYL)AMINO]-1H-PYRAZOL-1-YL}BENZAMIDE | JNK, MAP KINASE, ISOFORM SELECTIVE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fig:A (GLY333) to (GLY435) CATALYTIC DOMAIN OF HUMAN PAK4 | SERINE/THREONINE-PROTEIN KINASE PAK4, KINASE DOMAIN, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
4fig:B (GLY333) to (GLY435) CATALYTIC DOMAIN OF HUMAN PAK4 | SERINE/THREONINE-PROTEIN KINASE PAK4, KINASE DOMAIN, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
3r2b:C (LEU79) to (ASN181) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:E (LEU79) to (ILE170) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:G (LEU79) to (ASN181) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r7o:A (CYS1091) to (LYS1199) STRUCTURE OF DUALLY PHOSPHORYLATED C-MET RECEPTOR KINASE IN COMPLEX WITH AN MK-2461 ANALOG | TYROSINE KINASE, PHOSPHOTYROSINE, 1234, 1235, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3raw:A (GLY168) to (GLN278) CRYSTAL STRUCTURE OF HUMAN CDC-LIKE KINASE 3 ISOFORM IN COMPLEX WITH LEUCETTINE L41 | TRANSFERASE, KINASE, TYROSINE-PROTEIN KINASE, SERINE/THREONINE- PROTEIN KINASE, NUCLEOTIDE-BINDING, STRUCTURAL GENOMICS CONSORTIUM, SGC
5jrq:A (LYS473) to (GLU545) BRAFV600E KINASE DOMAIN IN COMPLEX WITH CHEMICALLY LINKED VEMURAFENIB INHIBITOR VEM-6-VEM | KINASE, DIMER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5jrq:B (THR470) to (GLU545) BRAFV600E KINASE DOMAIN IN COMPLEX WITH CHEMICALLY LINKED VEMURAFENIB INHIBITOR VEM-6-VEM | KINASE, DIMER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gfq:A (ASN56) to (VAL185) 2.65 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF RIBOSOME RECYCLING FACTOR (FRR) FROM BACILLUS ANTHRACIS | STRUCTURAL GENOMICS, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, TRANSLATION
5knj:B (SER215) to (HIS321) PSEUDOKINASE DOMAIN OF MLKL BOUND TO COMPOUND 1. | PSEUDOKINASE DOMAIN MLKL COMPOUND 1 GFE OUT TYPE 2 INHIBITOR, MEMBRANE PROTEINS-INHIBITOR COMPLEX
5lih:A (ALA266) to (GLY373) STRUCTURE OF A PEPTIDE-SUBSTRATE BOUND TO PKCIOTA CORE KINASE DOMAIN | APKC, POLARITY, COMPLEX, TRANSFERASE