Usages in wwPDB of concept: c_0435
nUsages: 733; SSE string: EEHEEHH
4wa9:B   (GLU255) to   (ASN336)  THE CRYSTAL STRUCTURE OF HUMAN ABL1 WILD TYPE KINASE DOMAIN IN COMPLEX WITH AXITINIB  |   KINASE, KINASE INHIBITOR, AXITINIB, ACTIVATION LOOP, DFG-OUT, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4gt4:A   (GLY485) to   (HIS610)  STRUCTURE OF UNLIGANDED, INACTIVE ROR2 KINASE DOMAIN  |   ATP BINDING, PHOSPHORYLATION, MEMBRANE, TRANSFERASE 
4gt4:B   (LYS489) to   (HIS610)  STRUCTURE OF UNLIGANDED, INACTIVE ROR2 KINASE DOMAIN  |   ATP BINDING, PHOSPHORYLATION, MEMBRANE, TRANSFERASE 
4gt5:A   (ALA527) to   (HIS645)  CRYSTAL STRUCTURE OF THE INACTIVE TRKA KINASE DOMAIN  |   TYROSINE KINASE DOMAIN, TRANSFERASE 
2of2:A   (PHE256) to   (LEU336)  CRYSTAL STRUCTURE OF FURANOPYRIMIDINE 8 BOUND TO LCK  |   LCK, KINASE DOMAIN, TRANSFERASE 
2of4:A   (PHE256) to   (LEU336)  CRYSTAL STRUCTURE OF FURANOPYRIMIDINE 1 BOUND TO LCK  |   LCK, KINASE DOMAIN, TRANSFERASE 
2ofv:A   (MET261) to   (LEU336)  CRYSTAL STRUCTURE OF AMINOQUINAZOLINE 1 BOUND TO LCK  |   LCK, KINASE DOMAIN, TRANSFERASE 
2ofv:B   (GLY257) to   (LEU336)  CRYSTAL STRUCTURE OF AMINOQUINAZOLINE 1 BOUND TO LCK  |   LCK, KINASE DOMAIN, TRANSFERASE 
2og8:A   (GLY257) to   (LEU336)  CRYSTAL STRUCTURE OF AMINOQUINAZOLINE 36 BOUND TO LCK  |   LCK, KINASE DOMAIN, TRANSFERASE 
2og8:B   (MET261) to   (LEU336)  CRYSTAL STRUCTURE OF AMINOQUINAZOLINE 36 BOUND TO LCK  |   LCK, KINASE DOMAIN, TRANSFERASE 
2ogv:A   (ASP608) to   (ASN773)  CRYSTAL STRUCTURE OF THE AUTOINHIBITED HUMAN C-FMS KINASE DOMAIN  |   RECEPTOR TYROSINE KINASE, MACROPHAGE COLONY STIMULATING FACTOR RECEPTOR, TRANSFERASE 
4whz:A    (GLY76) to   (GLY184)  DESIGN AND SYNTHESIS OF HIGHLY POTENT AND ISOFORM SELECTIVE JNK3 INHIBITORS: SAR STUDIES ON AMINOPYRAZOLE DERIVATIVES  |   JNK3, JNK2, JNK1, P38, KINASE INHIBITOR, PARKINSON DISEASE, ISOFORM- SELECTIVITY, AMINOPYRAZOLE 
2oid:D   (GLY198) to   (HIS306)  CRYSTAL STRUCTURE OF IRAK4 KINASE DOMAIN COMPLEXED WITH AMPPNP  |   KINASE, TRANSFERASE 
3efj:B  (GLY1090) to  (LYS1199)  STRUCTURE OF C-MET WITH PYRIMIDONE INHIBITOR 7  |   C-MET, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
2onl:B    (SER37) to   (ASP145)  CRYSTAL STRUCTURE OF THE P38A-MAPKAP KINASE 2 HETERODIMER  |   HETERODIMER, KINASE, NLS, NES, DOCKING GROOVE, TRANSFERASE 
4wnp:A    (VAL29) to   (PHE118)  STRUCTURE OF ULK1 BOUND TO A POTENT INHIBITOR  |   KINASE, AUTOPHAGY, INHIBITOR 
4wo5:A   (GLY469) to   (SER571)  CRYSTAL STRUCTURE OF A BRAF KINASE DOMAIN MONOMER  |   KINASE, MONOMER, INHIBITOR, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4h58:A   (LYS472) to   (GLU544)  BRAF IN COMPLEX WITH COMPOUND 3  |   PROTEIN KINASE, STRUCTURE BASED DRUG DISCOVERY, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3el8:B   (GLU280) to   (LEU358)  CRYSTAL STRUCTURE OF C-SRC IN COMPLEX WITH PYRAZOLOPYRIMIDINE 5  |   C-SRC, KINASE, PYRAZOLOPYRIMIDINE 5, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
4wsq:A    (ALA58) to   (HIS166)  CRYSTAL STRUCTURE OF ADAPTOR PROTEIN 2 ASSOCIATED KINASE (AAK1) IN COMPLEX WITH SMALL MOLECULE INHIBITOR  |   KINASE, SMALL-MOLECULE, CATALYTIC DOMAIN, PROTEIN KINASE, PROTEIN BINDING, PROTEIN KINASE INHIBITORS, TRANSFERASE 
4wsq:B    (PHE57) to   (HIS166)  CRYSTAL STRUCTURE OF ADAPTOR PROTEIN 2 ASSOCIATED KINASE (AAK1) IN COMPLEX WITH SMALL MOLECULE INHIBITOR  |   KINASE, SMALL-MOLECULE, CATALYTIC DOMAIN, PROTEIN KINASE, PROTEIN BINDING, PROTEIN KINASE INHIBITORS, TRANSFERASE 
1nw1:A    (MET88) to   (LEU183)  CRYSTAL STRUCTURE OF CHOLINE KINASE  |   CHOLINE KINASE, PHOSPHOLIPID SYNTHESIS, PROTEIN KINASE FOLD, TRANSFERASE 
1nw1:B    (LEU89) to   (LEU183)  CRYSTAL STRUCTURE OF CHOLINE KINASE  |   CHOLINE KINASE, PHOSPHOLIPID SYNTHESIS, PROTEIN KINASE FOLD, TRANSFERASE 
4wun:B   (ASN506) to   (LYS618)  STRUCTURE OF FGFR1 IN COMPLEX WITH AZD4547 (N-{3-[2-(3,5- DIMETHOXYPHENYL)ETHYL]-1H-PYRAZOL-5-YL}-4-[(3R,5S)-3,5- DIMETHYLPIPERAZIN-1-YL]BENZAMIDE) AT 1.65 ANGSTROM  |   TRANSFERASE; TRANSFERASE INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ww7:A    (ILE29) to   (ASP156)  CRYSTAL STRUCTURE OF BINARY COMPLEX BUD32-CGI121 IN COMPLEX WITH AMP  |   KEOPS, BINARY COMPLEX, BUD32-CGI121, TRNA T6A, TRANSFERASE 
2bdj:A   (GLU280) to   (LEU358)  SRC KINASE IN COMPLEX WITH INHIBITOR AP23464  |   SRC KINASE INHIBITOR, TRANSFERASE 
2bdw:A    (SER25) to   (GLY130)  CRYSTAL STRUCTURE OF THE AUTO-INHIBITED KINASE DOMAIN OF CALCIUM/CALMODULIN ACTIVATED KINASE II  |   KINASE; CALMODULIN ACTIVATED, TRANSFERASE 
2bdw:B    (SER25) to   (GLY130)  CRYSTAL STRUCTURE OF THE AUTO-INHIBITED KINASE DOMAIN OF CALCIUM/CALMODULIN ACTIVATED KINASE II  |   KINASE; CALMODULIN ACTIVATED, TRANSFERASE 
1b6c:B   (GLY217) to   (MET318)  CRYSTAL STRUCTURE OF THE CYTOPLASMIC DOMAIN OF THE TYPE I TGF-BETA RECEPTOR IN COMPLEX WITH FKBP12  |   COMPLEX (ISOMERASE/PROTEIN KINASE), RECEPTOR SERINE/THREONINE KINASE 
1b6c:D   (GLY217) to   (MET318)  CRYSTAL STRUCTURE OF THE CYTOPLASMIC DOMAIN OF THE TYPE I TGF-BETA RECEPTOR IN COMPLEX WITH FKBP12  |   COMPLEX (ISOMERASE/PROTEIN KINASE), RECEPTOR SERINE/THREONINE KINASE 
1b6c:F   (GLY217) to   (MET318)  CRYSTAL STRUCTURE OF THE CYTOPLASMIC DOMAIN OF THE TYPE I TGF-BETA RECEPTOR IN COMPLEX WITH FKBP12  |   COMPLEX (ISOMERASE/PROTEIN KINASE), RECEPTOR SERINE/THREONINE KINASE 
1b6c:H   (GLY217) to   (MET318)  CRYSTAL STRUCTURE OF THE CYTOPLASMIC DOMAIN OF THE TYPE I TGF-BETA RECEPTOR IN COMPLEX WITH FKBP12  |   COMPLEX (ISOMERASE/PROTEIN KINASE), RECEPTOR SERINE/THREONINE KINASE 
4hgt:A    (ASP22) to   (ASN123)  CRYSTAL STRUCTURE OF CK1D WITH COMPOUND 13  |   CK1D, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4hgt:B    (ASP22) to   (ASN123)  CRYSTAL STRUCTURE OF CK1D WITH COMPOUND 13  |   CK1D, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4hjo:A   (VAL714) to   (ARG808)  CRYSTAL STRUCTURE OF THE INACTIVE EGFR TYROSINE KINASE DOMAIN WITH ERLOTINIB  |   INACTIVE TYROSINE KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ezr:A    (GLY16) to   (ARG122)  CDK-2 WITH INDAZOLE INHIBITOR 17 BOUND AT ITS ACTIVE SITE  |   KINASE, PKC, PROTEIN KINASE, INHIBITOR, ATP-BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
4hnf:A    (GLY21) to   (ASN123)  CRYSTAL STRUCTURE OF CK1D IN COMPLEX WITH PF4800567  |   CK1D, KINASE, INHIBITOR, PF4800567, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4hni:A    (GLY21) to   (ASN123)  CRYSTAL STRUCTURE OF CK1E IN COMPLEX WITH PF4800567  |   CK1E, KINASE, INHIBITOR, PF4800567, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3f3t:B   (GLY279) to   (LEU358)  KINASE DOMAIN OF CSRC IN COMPLEX WITH INHIBITOR RL38 (TYPE III)  |   ALLOSTERIC, TYPE III, DFG-OUT, ALTERNATIVE SPLICING, ATP- BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3f3z:A    (LYS43) to   (ILE128)  CRYSTAL STRUCTURE OF CRYPTOSPORIDIUM PARVUM CALCIUM DEPENDENT PROTEIN KINASE CGD7_1840 IN PRESENCE OF INDIRUBIN E804  |   CALCIUM DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, SGC 
3f5p:E  (PRO1026) to  (LYS1130)  COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR  |   IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3f5p:F  (PRO1026) to  (LYS1130)  COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR  |   IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3f5p:G  (PRO1026) to  (LYS1130)  COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR  |   IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3f5p:H  (PRO1026) to  (LYS1130)  COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR  |   IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3f5p:I  (PRO1026) to  (LYS1130)  COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR  |   IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3f5p:L  (PRO1026) to  (LYS1130)  COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR  |   IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3f5p:R  (PRO1026) to  (LYS1130)  COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND 3- CYANOQUINOLINE INHIBITOR  |   IGF-1R, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3f6x:A   (GLY279) to   (LEU358)  C-SRC KINASE DOMAIN IN COMPLEX WITH SMALL MOLECULE INHIBITOR  |   KINASE, ATP-BINDING, ALTERNATIVE SPLICING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE 
4hok:A    (TYR24) to   (ASN123)  CRYSTAL STRUCTURE OF APO CK1E  |   CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE 
4hok:C    (TYR24) to   (ASN123)  CRYSTAL STRUCTURE OF APO CK1E  |   CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE 
4hok:E    (ILE23) to   (SER121)  CRYSTAL STRUCTURE OF APO CK1E  |   CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE 
4hok:G    (ASP22) to   (ASN123)  CRYSTAL STRUCTURE OF APO CK1E  |   CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE 
4hok:I    (GLY21) to   (ASN123)  CRYSTAL STRUCTURE OF APO CK1E  |   CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE 
4hok:Q    (ASP22) to   (ASN123)  CRYSTAL STRUCTURE OF APO CK1E  |   CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE 
4hok:S    (TYR24) to   (LYS122)  CRYSTAL STRUCTURE OF APO CK1E  |   CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE 
4hok:U    (TYR24) to   (ASN123)  CRYSTAL STRUCTURE OF APO CK1E  |   CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE 
4x7n:A   (GLY605) to   (GLY932)  CO-CRYSTAL STRUCTURE OF PERK BOUND TO 4-[2-AMINO-4-METHYL-3-(2- METHYLQUINOLIN-6-YL)BENZOYL]-1-METHYL-2,5-DIPHENYL-1,2-DIHYDRO-3H- PYRAZOL-3-ONE INHIBITOR  |   CATALYTIC DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR, COMPLEX 
3faa:A   (GLU218) to   (HIS317)  CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A 2- AMINOIMIDAZOLE INHIBITOR  |   KINASE, TGFBETA, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE 
3faa:B   (GLY217) to   (HIS317)  CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A 2- AMINOIMIDAZOLE INHIBITOR  |   KINASE, TGFBETA, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE 
3faa:C   (GLU218) to   (MET318)  CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A 2- AMINOIMIDAZOLE INHIBITOR  |   KINASE, TGFBETA, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE 
3faa:D   (GLY217) to   (HIS317)  CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A 2- AMINOIMIDAZOLE INHIBITOR  |   KINASE, TGFBETA, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE 
3faa:E   (GLU218) to   (MET318)  CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A 2- AMINOIMIDAZOLE INHIBITOR  |   KINASE, TGFBETA, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE 
2buj:A    (PHE31) to   (GLY143)  CRYSTAL STRUCTURE OF THE HUMAN SERINE-THREONINE KINASE 16 IN COMPLEX WITH STAUROSPORINE  |   TRANSFERASE, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, PALMITATE, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE 
2buj:B    (SER32) to   (GLY143)  CRYSTAL STRUCTURE OF THE HUMAN SERINE-THREONINE KINASE 16 IN COMPLEX WITH STAUROSPORINE  |   TRANSFERASE, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, PALMITATE, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE 
4hvs:A   (ALA606) to   (ASN787)  CRYSTAL STRUCTURE OF KIT KINASE DOMAIN WITH A SMALL MOLECULE INHIBITOR, PLX647  |   TRANSFERASE, TYROSINE-PROTEIN KINASE, ATP-BINDING, KINASE-KINASE INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3fe3:B    (ALA68) to   (ARG173)  CRYSTAL STRUCTURE OF THE KINASE MARK3/PAR-1: T211A-S215A DOUBLE MUTANT  |   SERINE/THREONINE PROTEIN KINASE; MARK;PAR-1; KIN1; UBA DOMAIN;C- TAK1;P78;MARK3, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
4hys:A    (GLY38) to   (GLY146)  CRYSTAL STRUCTURE OF JNK1 IN COMPLEX WITH JIP1 PEPTIDE AND 4-(4- INDAZOL-1-YL-PYRIMIDIN-2-YLAMINO)-CYCLOHEXAN  |   KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2c0i:A   (MET257) to   (GLN332)  SRC FAMILY KINASE HCK WITH BOUND INHIBITOR A-420983  |   TYROSINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHORYLATION, SH2 DOMAIN, SH3 DOMAIN 
2c0i:B   (MET257) to   (GLN332)  SRC FAMILY KINASE HCK WITH BOUND INHIBITOR A-420983  |   TYROSINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHORYLATION, SH2 DOMAIN, SH3 DOMAIN 
2c0o:A   (MET257) to   (GLN332)  SRC FAMILY KINASE HCK WITH BOUND INHIBITOR A-770041  |   TYROSINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHORYLATION, SH2 DOMAIN, SH3 DOMAIN 
2c0o:B   (MET257) to   (GLN332)  SRC FAMILY KINASE HCK WITH BOUND INHIBITOR A-770041  |   TYROSINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHORYLATION, SH2 DOMAIN, SH3 DOMAIN 
4xh0:A    (TYR24) to   (SER123)  STRUCTURE OF C. GLABRATA HRR25 BOUND TO ADP (SO4 CONDITION)  |   CASEIN KINASE, MONOPOLIN, TRANSFERASE 
4xhh:A    (ASP22) to   (GLY121)  STRUCTURE OF C. GLABRATA HRR25, APO STATE  |   CASEIN KINASE, MONOPOLIN, TRANSFERASE 
3sg8:A    (ILE35) to   (ILE133)  CRYSTAL STRUCTURE OF AMINOGLYCOSIDE-2''-PHOSPHOTRANSFERASE TYPE IVA TOBRAMYCIN COMPLEX  |   ANTIBIOTIC RESISTANCE ENZYME, TRANSFERASE, AMINOGLYCOSIDE, PHOSPHORYLATION, TRANSFERASE-ANTIBIOTIC COMPLEX 
3sg9:A    (ILE35) to   (ILE133)  CRYSTAL STRUCTURE OF AMINOGLYCOSIDE-2''-PHOSPHOTRANSFERASE TYPE IVA KANAMYCIN A COMPLEX  |   ANTIBIOTIC RESISTANCE ENZYME, TRANSFERASE, AMINOGLYCOSIDE, PHOSPHOTRANSFERASE, TRANSFERASE-ANTIBIOTIC COMPLEX 
4xhl:A    (ASP22) to   (ARG122)  STRUCTURE OF S. CEREVISIAE HRR25 1-394 (K38R MUTANT)  |   CASEIN KINASE, MONOPOLIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3she:A    (LEU59) to   (ILE150)  NOVEL ATP-COMPETITIVE MK2 INHIBITORS WITH POTENT BIOCHEMICAL AND CELL- BASED ACTIVITY THROUGHOUT THE SERIES  |   KINASE DOMAIN WITH BOUND INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2pyw:A    (ASN48) to   (SER155)  STRUCTURE OF A. THALIANA 5-METHYLTHIORIBOSE KINASE IN COMPLEX WITH ADP AND MTR  |   5-METHYLTHIORIBOSE KINASE, PLANT METHIONINE RECYCLING, REFOLDING, TRANSFERASE 
2pyw:B    (ASN48) to   (SER155)  STRUCTURE OF A. THALIANA 5-METHYLTHIORIBOSE KINASE IN COMPLEX WITH ADP AND MTR  |   5-METHYLTHIORIBOSE KINASE, PLANT METHIONINE RECYCLING, REFOLDING, TRANSFERASE 
1ckj:A    (GLY24) to   (ASN126)  CASEIN KINASE I DELTA TRUNCATION MUTANT CONTAINING RESIDUES 1-317 COMPLEX WITH BOUND TUNGSTATE  |   PROTEIN KINASE, PHOSPHOTRANSFERASE 
4i92:A    (ASN71) to   (GLY175)  STRUCTURE OF THE BSK8 KINASE DOMAIN  |   PROTEIN KINASE, PSEUDO KINASE, CFG, ALANINE GATEKEEPER, TRANSFERASE BRASSINOSTEROID-SIGNALING, TRANSFERASE 
4i93:A    (ASN71) to   (GLY175)  STRUCTURE OF THE BSK8 KINASE DOMAIN (SEMET LABELED)  |   PROTEIN KINASE, PSEUDO KINASE, CFG, ALANINE GATEKEEPER, TRANSFERASE BRASSINOSTEROID-SIGNALING, SEMET DERIVATIVE, TRANSFERASE 
4i93:B    (PRO70) to   (GLY175)  STRUCTURE OF THE BSK8 KINASE DOMAIN (SEMET LABELED)  |   PROTEIN KINASE, PSEUDO KINASE, CFG, ALANINE GATEKEEPER, TRANSFERASE BRASSINOSTEROID-SIGNALING, SEMET DERIVATIVE, TRANSFERASE 
4i94:A    (PRO70) to   (TRP147)  STRUCTURE OF BSK8 IN COMPLEX WITH AMP-PNP  |   PROTEIN KINASE, PSEUDO KINASE, CFG, ALANINE GATEKEEPER, TRANSFERASE, BRASSINOSTEROID-SIGNALING, AMP-PNP, MG2+ 
4i94:B    (PRO70) to   (TRP147)  STRUCTURE OF BSK8 IN COMPLEX WITH AMP-PNP  |   PROTEIN KINASE, PSEUDO KINASE, CFG, ALANINE GATEKEEPER, TRANSFERASE, BRASSINOSTEROID-SIGNALING, AMP-PNP, MG2+ 
4ieb:A    (GLU64) to   (LYS169)  CRYSTAL STRUCTURE OF A GLY128MET MUTANT OF THE TOXOPLASMA CDPK, TGME49_101440  |   CDPKS, TOXOPLASMA, KINASE, PROTIST, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
4ifg:A    (GLY63) to   (LYS169)  CRYSTAL STRUCTURE OF TGCDPK1 WITH INHIBITOR BOUND  |   STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1p14:A  (GLY1013) to  (LYS1127)  CRYSTAL STRUCTURE OF A CATALYTIC-LOOP MUTANT OF THE INSULIN RECEPTOR TYROSINE KINASE  |   RECEPTOR, TYROSINE KINASE, CATALYSIS, MUTANT, TRANSFERASE 
3sv0:A    (GLY21) to   (SER123)  CRYSTAL STRUCTURE OF CASEIN KINASE-1 LIKE PROTEIN IN PLANT  |   KINASE, TYPICAL KINASE DOMAIN FOLD, CYTOSOL, TRANSFERASE 
3fzs:A   (GLY442) to   (ASN544)  CRYSTAL STRUCTURE OF PYK2 COMPLEXED WITH BIRB796  |   PYK2, KINASE, DFG, ALTERNATIVE SPLICING, ATP-BINDING, CELL MEMBRANE, CYTOPLASM, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE, TYROSINE-PROTEIN KINASE 
4ih8:A    (GLY63) to   (LYS169)  CRYSTAL STRUCTURE OF TGCDPK1 WITH INHIBITOR BOUND  |   STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ihp:A    (GLY63) to   (LYS169)  CRYSTAL STRUCTURE OF TGCDPK1 WITH INHIBITOR BOUND  |   STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3sx9:A    (GLY63) to   (LYS169)  CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR, RM-1-132  |   SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3g5d:A   (GLU280) to   (LEU358)  KINASE DOMAIN OF CSRC IN COMPLEX WITH DASATINIB  |   TYPE II, DFG-OUT, TYROSINE-PROTEIN KINASE, DASATINIB, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
2cjm:A    (GLY16) to    (GLY98)  MECHANISM OF CDK INHIBITION BY ACTIVE SITE PHOSPHORYLATION: CDK2 Y15P T160P IN COMPLEX WITH CYCLIN A STRUCTURE  |   PHOSPHORYLATION, NUCLEOTIDE-BINDING, MITOSIS, CELL CYCLE, REGULATION, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, TRANSFERASE, CELL DIVISION, CYCLIN-DEPENDENT KINASE, COMPLEX (TRANSFERASE/CELL DIVISION) 
1dd5:A    (ALA55) to   (ILE182)  CRYSTAL STRUCTURE OF THERMOTOGA MARITIMA RIBOSOME RECYCLING FACTOR, RRF  |   THREE-HELIX BUNDLE, BETA-ALPHA-BETA SANDWICH, RIBOSOME 
2qg7:A   (ASN122) to   (ILE212)  PLASMODIUM VIVAX ETHANOLAMINE KINASE PV091845  |   MALARIA, ETHANOLAMINE KINASE, PV091845, SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSFERASE 
2qg7:D   (ILE123) to   (ASP211)  PLASMODIUM VIVAX ETHANOLAMINE KINASE PV091845  |   MALARIA, ETHANOLAMINE KINASE, PV091845, SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSFERASE 
2cke:B    (PHE24) to   (LYS134)  HUMAN DEATH-ASSOCIATED DRP-1 KINASE IN COMPLEX WITH INHIBITOR  |   TRANSFERASE-INHIBITOR COMPLEX, TRANSFERASE/INHIBITOR COMPLEX, CALMODULIN-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, APOPTOSIS 
2cko:A   (LEU124) to   (GLY237)  CRYSTAL STRUCTURE OF HUMAN CHOLINE KINASE ALPHA 2  |   KINASE, TRANSFERASE, CHOLINE KINASE, PHOSPHATYDILCHOLINE, ALTERNATIVE SPLICING 
2cko:B   (MET123) to   (GLY237)  CRYSTAL STRUCTURE OF HUMAN CHOLINE KINASE ALPHA 2  |   KINASE, TRANSFERASE, CHOLINE KINASE, PHOSPHATYDILCHOLINE, ALTERNATIVE SPLICING 
4xuf:A   (ALA627) to   (SER806)  CRYSTAL STRUCTURE OF THE FLT3 KINASE DOMAIN BOUND TO THE INHIBITOR QUIZARTINIB (AC220)  |   FLT3, RECEPTOR TYROSINE KINASE, AC220, QUIZARTINIB, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
2qnj:B    (PHE67) to   (ARG173)  KINASE AND UBIQUITIN-ASSOCIATED DOMAINS OF MARK3/PAR-1  |   SERINE/THREONINE PROTEIN KINASE, UBIQUITIN-ASSOCIATED DOMAIN, MARK, PAR-1, TRANSFERASE 
3geq:A   (GLY279) to   (LEU358)  STRUCTURAL BASIS FOR THE CHEMICAL RESCUE OF SRC KINASE ACTIVITY  |   KINASE, CHEMICAL RESCUE, PP2, ALTERNATIVE SPLICING, ATP- BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3geq:B   (GLU280) to   (LEU358)  STRUCTURAL BASIS FOR THE CHEMICAL RESCUE OF SRC KINASE ACTIVITY  |   KINASE, CHEMICAL RESCUE, PP2, ALTERNATIVE SPLICING, ATP- BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
2qr8:A   (SER434) to   (GLY534)  2.0A X-RAY STRUCTURE OF C-TERMINAL KINASE DOMAIN OF P90 RIBOSOMAL S6 KINASE 2 (RSK2)  |   KINASE DOMAIN, RSK2, AUTOINHIBITORY, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
2qr7:A   (SER434) to   (GLY534)  2.0A X-RAY STRUCTURE OF C-TERMINAL KINASE DOMAIN OF P90 RIBOSOMAL S6 KINASE 2: SE-MET DERIVATIVE  |   KINASE DOMAIN, RSK2, AUTOINHIBITORY, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
1pmn:A    (GLY76) to   (GLY184)  CRYSTAL STRUCTURE OF JNK3 IN COMPLEX WITH AN IMIDAZOLE- PYRIMIDINE INHIBITOR  |   MAP KINASE, APOPTOSIS, INHIBITION, TRANSFERASE 
3ggf:A    (GLY36) to   (GLY114)  CRYSTAL STRUCTURE OF HUMAN SERINE/THREONINE-PROTEIN KINASE MST4 IN COMPLEX WITH AN QUINAZOLIN  |   SERINE/THREONINE-PROTEIN KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, APOPTOSIS, ATP-BINDING, GOLGI APPARATUS, KINASE, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, TRANSFERASE 
4iw0:A    (ALA72) to   (ALA215)  CRYSTAL STRUCTURE AND MECHANISM OF ACTIVATION OF TBK1  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4y12:A   (GLY163) to   (GLY271)  CRYSTAL STRUCTURE OF THE S/T PROTEIN KINASE PKNG FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH AGS  |   S/T PROTEIN KINASE, PKNG, TRANSFERASE 
4y46:A    (GLY76) to   (GLY184)  PYRIDOPYRIMIDINONE DERIVATIVES AS POTENT AND SELECTIVE C-JUN N- TERMINAL KINASE (JNK) INHIBITORS  |   JNK, MAP KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2r2p:A   (GLY692) to   (GLY795)  KINASE DOMAIN OF HUMAN EPHRIN TYPE-A RECEPTOR 5 (EPHA5)  |   ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, RECEPTOR, SIGNAL, TRANSFERASE, PHOSPHORYLATION, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE, ALTERNATIVE SPLICING, GLYCOPROTEIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC 
3tcp:A   (VAL601) to   (ASN718)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE-PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR UNC569  |   TYROSINE KINASE, ACUTE LYMPHOBLASTIC LEUKEMIA, RATIONAL STRUCTURE- BASED DRUG DESIGN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2r4b:A   (THR743) to   (ARG838)  ERBB4 KINASE DOMAIN COMPLEXED WITH A THIENOPYRIMIDINE INHIBITOR  |   ERB, KINASE, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE 
2r4b:B   (THR743) to   (ARG838)  ERBB4 KINASE DOMAIN COMPLEXED WITH A THIENOPYRIMIDINE INHIBITOR  |   ERB, KINASE, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE 
4j96:B   (ALA498) to   (LYS621)  CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC GAIN-OF-FUNCTION K659M MUTATION IDENTIFIED IN CERVICAL CANCER.  |   KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, RECEPTOR TYROSINE KINASE, ATP BINDING, TRANSFERASE 
4y8d:A    (PHE51) to   (GLY141)  CRYSTAL STRUCTURE OF CYCLIN-G ASSOCIATED KINASE (GAK) COMPLEXED WITH SELECTIVE 12I INHIBITOR  |   TRANSFERASE, KINASE, NANOBODY, INHIBITOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC 
4y8d:B    (PHE51) to   (GLY141)  CRYSTAL STRUCTURE OF CYCLIN-G ASSOCIATED KINASE (GAK) COMPLEXED WITH SELECTIVE 12I INHIBITOR  |   TRANSFERASE, KINASE, NANOBODY, INHIBITOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC 
4jbv:A    (GLY63) to   (LYS169)  CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1268  |   SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4jg7:A   (SER434) to   (GLY534)  STRUCTURE OF RSK2 CTD BOUND TO 3-(3-(1H-PYRROLO[2,3-B]PYRIDINE-3- CARBONYL)PHENYL)-2-CYANOACRYLAMIDE  |   PROTEIN KINASE, PHOSPHORYLATION, COVALENT INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4yc8:B   (GLU255) to   (ASN336)  C-HELIX-OUT BINDING OF DASATINIB ANALOG TO C-ABL KINASE  |   KINASE, C-HELIX-OUT, TRANSFERASE 
4jjr:A    (GLY21) to   (ASN123)  A P21 CRYSTAL FORM OF MAMMALIAN CASEIN KINASE 1 DELTA  |   CK1D, KINASE, CASEIN KINASE, TRANSFERASE 
2rei:A   (GLU646) to   (GLY753)  KINASE DOMAIN OF HUMAN EPHRIN TYPE-A RECEPTOR 7 (EPHA7)  |   ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, RECEPTOR, SIGNAL, TRANSFERASE, PHOSPHORYLATION, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE, ALTERNATIVE SPLICING, GLYCOPROTEIN, STRUCTURAL GENOMICS CONSORTIUM, SGC, POLYMORPHISM 
2rfn:A  (GLY1102) to  (LYS1199)  X-RAY STRUCTURE OF C-MET WITH INHIBITOR.  |   C-MET HGF RECEPTOR TYROSINE KINSE KINASE DOMAIN, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, PROTO- ONCOGENE, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3ttj:A    (GLY76) to   (GLY184)  CRYSTAL STRUCTURE OF JNK3 COMPLEXED WITH CC-359, A JNK INHIBITOR FOR THE PREVENTION OF ISCHEMIA-REPERFUSION INJURY  |   MITOGEN-ACTIVATED PROTEIN KINASE 10, JNK3, PROTEIN KINASE INHIBITORS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4yff:A   (GLY480) to   (LYS555)  TNNI3K COMPLEXED WITH INHIBITOR 2  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4yff:B   (GLY480) to   (LYS555)  TNNI3K COMPLEXED WITH INHIBITOR 2  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4yff:C   (GLY480) to   (LYS555)  TNNI3K COMPLEXED WITH INHIBITOR 2  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4yff:D   (GLY480) to   (LYS555)  TNNI3K COMPLEXED WITH INHIBITOR 2  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4yfi:A   (GLY480) to   (LYS555)  TNNI3K COMPLEXED WITH INHIBITOR 1  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4yfi:C   (GLY480) to   (LYS555)  TNNI3K COMPLEXED WITH INHIBITOR 1  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4yfi:D   (GLY475) to   (LYS555)  TNNI3K COMPLEXED WITH INHIBITOR 1  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2e2b:A   (GLU255) to   (ASN336)  CRYSTAL STRUCTURE OF THE C-ABL KINASE DOMAIN IN COMPLEX WITH INNO-406  |   C-ABL, KINASE, INNO-406, TRANSFERASE 
2e2b:B   (GLU255) to   (ASN336)  CRYSTAL STRUCTURE OF THE C-ABL KINASE DOMAIN IN COMPLEX WITH INNO-406  |   C-ABL, KINASE, INNO-406, TRANSFERASE 
3tv4:A   (THR470) to   (GLU545)  HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH AN BROMOPYRIDINE BENZAMIDE INHIBITOR  |   KINASE, KINASE INHIBITOR, TRANSFERASE, RAS, C-RAF, MEK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3tv4:B   (PHE468) to   (GLU545)  HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH AN BROMOPYRIDINE BENZAMIDE INHIBITOR  |   KINASE, KINASE INHIBITOR, TRANSFERASE, RAS, C-RAF, MEK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3tv6:A   (LYS473) to   (GLU545)  HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH A METHOXYPYRAZOLOPYRIDINYL BENZAMIDE INHIBITOR  |   B-RAF, KINASE, KINASE INHIBITOR, TRANSFERASE, C-RAF, RAS, MEK, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1qpc:A   (PHE256) to   (LEU336)  STRUCTURAL ANALYSIS OF THE LYMPHOCYTE-SPECIFIC KINASE LCK IN COMPLEX WITH NON-SELECTIVE AND SRC FAMILY SELECTIVE KINASE INHIBITORS  |   ALPHA BETA FOLD, TRANSFERASE 
1qpj:A   (GLU258) to   (LEU336)  CRYSTAL STRUCTURE OF THE LYMPHOCYTE-SPECIFIC KINASE LCK IN COMPLEX WITH STAUROSPORINE.  |   ALPHA BETA FOLD, TRANSFERASE 
4yht:A   (LYS472) to   (GLU544)  BRAF COMPLEXED WITH AN INHIBITOR  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4yht:B   (LYS472) to   (GLU544)  BRAF COMPLEXED WITH AN INHIBITOR  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2uv2:A    (GLY46) to   (LYS150)  CRYSTAL STRUCTURE OF HUMAN STE20-LIKE KINASE BOUND TO 4-(4-( 5-CYCLOPROPYL-1H-PYRAZOL-3-YLAMINO)-QUINAZOLIN-2-YLAMINO)- PHENYL)-ACETONITRILE  |   TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, MUSCLE DEVELOPMENT, KINASE, APOPTOSIS, GERMINAL CENTRE KINASE, SERINE- THREONINE KINASE 2, NUCLEOTIDE-BINDING, SERINE-THREONINE-PROTEIN KINASE 
4yjn:A    (GLY63) to   (LYS169)  CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1639  |   SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4jt3:A   (SER537) to   (GLY642)  CRYSTAL STRUCTURE OF TTK KINASE DOMAIN WITH AN INHIBITOR: 400740  |   TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3h9r:A   (GLY220) to   (ILE321)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF TYPE I ACTIVIN RECEPTOR (ACVR1) IN COMPLEX WITH FKBP12 AND DORSOMORPHIN  |   STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP- BINDING, DISEASE MUTATION, GLYCOPROTEIN, KINASE, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE, ISOMERASE, ROTAMASE, ISOMERASE-PROTEIN KINASE COMPLEX 
4jvg:A   (LYS473) to   (SER544)  B-RAF KINASE IN COMPLEX WITH BIRB796  |   KINASE, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4jvg:D   (LYS473) to   (SER544)  B-RAF KINASE IN COMPLEX WITH BIRB796  |   KINASE, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1r0e:A    (GLY68) to   (GLY176)  GLYCOGEN SYNTHASE KINASE-3 BETA IN COMPLEX WITH 3-INDOLYL-4- ARYLMALEIMIDE INHIBITOR  |   SER/THR PROTEIN KINASE, TRANSFERASE 
2uzb:A    (GLY16) to   (GLN113)  CRYSTAL STRUCTURE OF HUMAN CDK2 COMPLEXED WITH A THIAZOLIDINONE INHIBITOR  |   TRANSFERASE, ATP-BINDING, PHOSPHORYLATION, CDK2, KINASE, CYCLIN, MITOSIS, CELL CYCLE, CELL DIVISION, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, THIAZOLIDINONE LIGAND 
4yo6:A   (GLY198) to   (HIS306)  IRAK4-INHIBITOR CO-STRUCTURE  |   KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4yo6:B   (GLY198) to   (HIS306)  IRAK4-INHIBITOR CO-STRUCTURE  |   KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4k11:A   (GLY279) to   (LEU358)  THE STRUCTURE OF 1NA IN COMPLEX WITH SRC T338G  |   1NA, C-SRC, KINASE, PHOSPHORYLATION, TRANSFERASE 
4yom:B    (GLY32) to   (SER137)  STRUCTURE OF SAD KINASE  |   KINASE DOMAIN, UBA DOMAIN, KA1 DOMAIN, TRANSFERASE 
3uc4:A    (VAL34) to   (MET134)  THE CRYSTAL STRUCTURE OF SNF1-RELATED KINASE 2.6  |   SNRK2.6, KINASE, ABA SIGNALING, TRANSFERASE 
4yps:A   (ALA527) to   (HIS645)  (R)-2-PHENYLPYRROLIDINE SUBSTITUTE IMIDAZOPYRIDAZINES: A NEW CLASS OF POTENT AND SELECTIVE PAN-TRK INHIBITORS  |   TRKA, KINASE, ONCOLOGY, INHIBITOR COMPLEX., TRANSFEASE-TRANSFERASE INHIBITOR COMPLEX 
3ue4:B   (GLU255) to   (ASN336)  STRUCTURAL AND SPECTROSCOPIC ANALYSIS OF THE KINASE INHIBITOR BOSUTINIB BINDING TO THE ABL TYROSINE KINASE DOMAIN  |   PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2exc:X    (GLY76) to   (GLY184)  INHIBITOR COMPLEX OF JNK3  |   ENZYME-INHIBITOR COMPLEX, KINASE INHIBITOR, TRANSFERASE 
1fpu:B   (GLU255) to   (SER336)  CRYSTAL STRUCTURE OF ABL KINASE DOMAIN IN COMPLEX WITH A SMALL MOLECULE INHIBITOR  |   KINASE, KINASE INHIBITOR, STI-571, ACTIVATION LOOP, TRANSFERASE 
1rjb:A   (ALA627) to   (SER806)  CRYSTAL STRUCTURE OF FLT3  |   KINASE, STRUCTURE, AUTOINHIBITION, JUXTAMEMBRANE DOMAIN, TRANSFERASE 
2f4j:A   (GLU255) to   (ASN336)  STRUCTURE OF THE KINASE DOMAIN OF AN IMATINIB-RESISTANT ABL MUTANT IN COMPLEX WITH THE AURORA KINASE INHIBITOR VX-680  |   KINASE, KINASE INHIBITOR, ABL, TRANSFERASE 
4kaw:X    (ALA55) to   (GLU184)  CRYSTAL STRUCTURE OF RIBOSOME RECYCLING FACTOR MUTANT R39G FROM MYCOBACTERIUM TUBERCULOSIS  |   RIBOSOME RECYCLING, TRANSLATION, EUBACTERIA, DISASSEMBLY, POST- TERMINATION COMPLEX, RIBOSOME, ELONGATION FACTOR G, BACTERIAL CYTOSOL 
4kb4:A    (ILE57) to   (LEU183)  CRYSTAL STRUCTURE OF RIBOSOME RECYCLING FACTOR MUTANT R31A FROM MYCOBACTERIUM TUBERCULOSIS  |   RIBOSOME RECYCLING, POST-TERMINATION COMPLEX, TRANSLATION, ELONGATION FACTOR G, BACTERIAL CYTOSOL 
4kb8:B    (GLY21) to   (ASN123)  CK1D IN COMPLEX WITH 1-{4-[3-(4-FLUOROPHENYL)-1-METHYL-1H-PYRAZOL-4- YL]PYRIDIN-2-YL}-N-METHYLMETHANAMINE LIGAND  |   SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4kb8:D    (ASP22) to   (ASN123)  CK1D IN COMPLEX WITH 1-{4-[3-(4-FLUOROPHENYL)-1-METHYL-1H-PYRAZOL-4- YL]PYRIDIN-2-YL}-N-METHYLMETHANAMINE LIGAND  |   SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4kba:B    (GLY21) to   (ASN123)  CK1D IN COMPLEX WITH 9-[3-(4-FLUOROPHENYL)-1-METHYL-1H-PYRAZOL-4-YL]- 2,3,4,5-TETRAHYDROPYRIDO[2,3-F][1,4]OXAZEPINE INHIBITOR  |   SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4kba:D    (ASP22) to   (ASN123)  CK1D IN COMPLEX WITH 9-[3-(4-FLUOROPHENYL)-1-METHYL-1H-PYRAZOL-4-YL]- 2,3,4,5-TETRAHYDROPYRIDO[2,3-F][1,4]OXAZEPINE INHIBITOR  |   SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4kbk:A    (GLY21) to   (ASN123)  CK1D IN COMPLEX WITH (3S)-3-{4-[3-(4-FLUOROPHENYL)-1-METHYL-1H- PYRAZOL-4-YL]PYRIDIN-2-YL}MORPHOLINE INHIBITOR  |   SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4kbk:D    (ASP22) to   (ASN123)  CK1D IN COMPLEX WITH (3S)-3-{4-[3-(4-FLUOROPHENYL)-1-METHYL-1H- PYRAZOL-4-YL]PYRIDIN-2-YL}MORPHOLINE INHIBITOR  |   SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4yz9:C   (ARG588) to   (ASN683)  CRYSTAL STRUCTURE OF HUMAN PHOSPHORYLATED IRE1ALPHA IN COMPLEX WITH A TYPE III KINASE INHIBITOR (GSK2850163A)  |   ACTIVE, INHIBITOR, COMPLEX, IRE1, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2fb8:B   (GLY469) to   (GLU545)  STRUCTURE OF THE B-RAF KINASE DOMAIN BOUND TO SB-590885  |   KINASE DOMAIN, TRANSFERASE 
3uqc:D    (GLN45) to   (GLY145)  STRUCTURE OF THE INTRACELLULAR KINASE HOMOLOGY DOMAIN OF RV3910 AT 2.2 A RESOLUTION  |   STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, KINASE FOLD, FHAA, TRANSFERASE 
1gag:A  (GLY1013) to  (LYS1126)  CRYSTAL STRUCTURE OF THE INSULIN RECEPTOR KINASE IN COMPLEX WITH A BISUBSTRATE INHIBITOR  |   PROTEIN KINASE INHIBITOR, TYROSINE KINASE, TRANSFERASE, SIGNALING PROTEIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4z7h:A   (ARG588) to   (LEU661)  CRYSTAL STRUCTURE OF HUMAN IRE1 CYTOPLASMIC KINASE-RNASE REGION - COMPLEX WITH IMIDAZOPYRIDINE COMPOUND 3  |   TRANSFERASE, KINASE, RNASE, UNFOLDED PROTEIN RESPONSE 
4z7h:B   (ARG588) to   (LEU661)  CRYSTAL STRUCTURE OF HUMAN IRE1 CYTOPLASMIC KINASE-RNASE REGION - COMPLEX WITH IMIDAZOPYRIDINE COMPOUND 3  |   TRANSFERASE, KINASE, RNASE, UNFOLDED PROTEIN RESPONSE 
4z9l:A    (GLY76) to   (GLY184)  THE STRUCTURE OF JNK3 IN COMPLEX WITH AN IMIDAZOLE-PYRIMIDINE INHIBITOR  |   MAP KINASE, APOPTOSIS, INHIBITION, TRANSFERASE 
3uyt:A    (ASP22) to   (ASN123)  CRYSTAL STRUCTURE OF CK1D WITH PF670462 FROM P1 CRYSTAL FORM  |   CK1D, KINASE, INHIBITOR, PF670462, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3uyt:B    (ASP22) to   (ASN123)  CRYSTAL STRUCTURE OF CK1D WITH PF670462 FROM P1 CRYSTAL FORM  |   CK1D, KINASE, INHIBITOR, PF670462, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3uyt:C    (GLY21) to   (ASN123)  CRYSTAL STRUCTURE OF CK1D WITH PF670462 FROM P1 CRYSTAL FORM  |   CK1D, KINASE, INHIBITOR, PF670462, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3hx4:A    (GLU64) to   (ILE154)  CRYSTAL STRUCTURE OF CDPK1 OF TOXOPLASMA GONDII, TGME49_101440, IN PRESENCE OF CALCIUM  |   CDPKS, TOXOPLASMA, KINASE, PROTIST, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3hyh:A    (LYS70) to   (LYS172)  CRYSTAL STRUCTURE OF THE PROTEIN KINASE DOMAIN OF YEAST AMP-ACTIVATED PROTEIN KINASE SNF1  |   KINASE DOMAIN, TRANSFERASE, ATP-BINDING, CARBOHYDRATE METABOLISM, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE 
2g1t:A   (GLY254) to   (ASN336)  A SRC-LIKE INACTIVE CONFORMATION IN THE ABL TYROSINE KINASE DOMAIN  |   KINASE, TRANSFERASE 
2g1t:B   (GLY254) to   (ASN336)  A SRC-LIKE INACTIVE CONFORMATION IN THE ABL TYROSINE KINASE DOMAIN  |   KINASE, TRANSFERASE 
2g1t:D   (GLU255) to   (ASN336)  A SRC-LIKE INACTIVE CONFORMATION IN THE ABL TYROSINE KINASE DOMAIN  |   KINASE, TRANSFERASE 
2g2h:B   (GLU274) to   (ASN355)  A SRC-LIKE INACTIVE CONFORMATION IN THE ABL TYROSINE KINASE DOMAIN  |   PROTEIN KINASE, TRANSFERASE 
4ksp:A   (GLY468) to   (GLU544)  CRYSTAL STRUCTURE OF HUMAN B-RAF BOUND TO A DFG-OUT INHIBITOR TAK-632  |   HUMAN SERINE/THERONINE PROTEIN KINASE, KINASE DRUG COMPLEX,, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ksp:B   (LYS472) to   (GLU544)  CRYSTAL STRUCTURE OF HUMAN B-RAF BOUND TO A DFG-OUT INHIBITOR TAK-632  |   HUMAN SERINE/THERONINE PROTEIN KINASE, KINASE DRUG COMPLEX,, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1snu:B   (GLY375) to   (CYS477)  CRYSTAL STRUCTURE OF THE UNPHOSPHORYLATED INTERLEUKIN-2 TYROSINE KINASE CATALYTIC DOMAIN  |   PROTEIN KINASE, IMMUNOLOGY, TRANSFERASE 
3i5n:A  (HIS1094) to  (LYS1199)  CRYSTAL STRUCTURE OF C-MET WITH TRIAZOLOPYRIDAZINE INHIBITOR 13  |   PROTO-ONCOGENE, RTK, RECEPTOR TYROSINE KINASE, SCATTER FACTOR RECEPTOR, HGF/SF, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
1gup:A    (ALA89) to   (ASP208)  STRUCTURE OF NUCLEOTIDYLTRANSFERASE COMPLEXED WITH UDP- GALACTOSE  |   TRANSFERASE, NUCLEOTIDYLTRANSFERASE, GALACTOSE METABOLISM 
1guq:D    (PRO87) to   (ASP208)  STRUCTURE OF NUCLEOTIDYLTRANSFERASE COMPLEXED WITH UDP-GLUCOSE  |   TRANSFERASE, NUCLEOTIDYLTRANSFERASE, GALACTOSE METABOLISM 
3i7c:A    (GLY63) to   (LYS169)  CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR NA-PP2  |   PROTEIN KINASE, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, TRANSFERASE 
3i81:A   (PRO996) to  (LYS1100)  CRYSTAL STRUCTURE OF INSULIN-LIKE GROWTH FACTOR 1 RECEPTOR (IGF-1R-WT) COMPLEX WITH BMS-754807 [1-(4-((5-CYCLOPROPYL- 1H-PYRAZOL-3-YL)AMINO)PYRROLO[2,1-F][1,2,4]TRIAZIN-2-YL)-N- (6-FLUORO-3-PYRIDINYL)-2-METHYL-L-PROLINAMIDE]  |   HORMONE/GROWTH FACTOR, IGF-1R, KINASE DOMAIN, ATP-BINDING, DISEASE MUTATION, DISULFIDE BOND, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
4l01:A   (SER599) to   (ASP709)  CRYSTAL STRUCTURE OF THE V658F APO JAK1 PSEUDOKINASE DOMAIN  |   KINASE DOMAIN FOLD, REGULATORY, TRANSFERASE 
4zly:A   (GLY414) to   (GLN516)  CRYSTAL STRUCTURE OF BRUTON'S TYROSINE KINASE BOUND TO A CINNOLINE FRAGMENT  |   CYTOPLASMIC TYROSINE KINASE, TRANSCRIPTIONAL REGULATION, NUCLEAR FACTOR-KAPPAB, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3idp:A   (LYS473) to   (GLU545)  B-RAF V600E KINASE DOMAIN IN COMPLEX WITH AN AMINOISOQUINOLINE INHIBITOR  |   ONCOGENE, ATP-BINDING, DFG-OUT, TRANSFERASE, CARDIOMYOPATHY, DISEASE MUTATION, KINASE, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, ZINC-FINGER 
3idp:B   (LYS473) to   (GLU545)  B-RAF V600E KINASE DOMAIN IN COMPLEX WITH AN AMINOISOQUINOLINE INHIBITOR  |   ONCOGENE, ATP-BINDING, DFG-OUT, TRANSFERASE, CARDIOMYOPATHY, DISEASE MUTATION, KINASE, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, ZINC-FINGER 
4l68:B   (GLY319) to   (HIS418)  STRUCTURE OF THE PSEDUDOKINASE DOMAIN OF BIR2, AN IMMUNE REGULATOR OF THE RLK/PELLE FAMILY  |   PSEUDOKINASE, NEGATIVE IMMUNE REGULATOR, SIGNALING PROTEIN 
3iec:A    (ALA65) to   (PHE170)  HELICOBACTER PYLORI CAGA INHIBITS PAR1/MARK FAMILY KINASES BY MIMICKING HOST SUBSTRATES  |   PROTEIN-PROTEIN COMPLEX, KINASE, VIRULENCE FACTOR, ALTERNATIVE PROMOTER USAGE, ATP-BINDING, CELL MEMBRANE, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, MAGNESIUM, MEMBRANE, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, SIGNALING PROTEIN-TOXIN COMPLEX 
3iec:B    (ALA65) to   (PHE170)  HELICOBACTER PYLORI CAGA INHIBITS PAR1/MARK FAMILY KINASES BY MIMICKING HOST SUBSTRATES  |   PROTEIN-PROTEIN COMPLEX, KINASE, VIRULENCE FACTOR, ALTERNATIVE PROMOTER USAGE, ATP-BINDING, CELL MEMBRANE, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, MAGNESIUM, MEMBRANE, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, SIGNALING PROTEIN-TOXIN COMPLEX 
3iec:C    (ALA65) to   (PHE170)  HELICOBACTER PYLORI CAGA INHIBITS PAR1/MARK FAMILY KINASES BY MIMICKING HOST SUBSTRATES  |   PROTEIN-PROTEIN COMPLEX, KINASE, VIRULENCE FACTOR, ALTERNATIVE PROMOTER USAGE, ATP-BINDING, CELL MEMBRANE, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, MAGNESIUM, MEMBRANE, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, SIGNALING PROTEIN-TOXIN COMPLEX 
3iec:D    (LYS66) to   (LYS155)  HELICOBACTER PYLORI CAGA INHIBITS PAR1/MARK FAMILY KINASES BY MIMICKING HOST SUBSTRATES  |   PROTEIN-PROTEIN COMPLEX, KINASE, VIRULENCE FACTOR, ALTERNATIVE PROMOTER USAGE, ATP-BINDING, CELL MEMBRANE, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, MAGNESIUM, MEMBRANE, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, SIGNALING PROTEIN-TOXIN COMPLEX 
4l7f:A    (GLY38) to   (SER144)  CO-CRYSTAL STRUCTURE OF JNK1 AND AX13587  |   PROTEIN KINASE FOLD, PROTEIN KINASE, JUN-C, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3igo:A    (LEU91) to   (ILE178)  CRYSTAL STRUCTURE OF CRYPTOSPORIDIUM PARVUM CDPK1, CGD3_920  |   PARASITE, KINASE, CDPK, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE 
4zog:B   (GLU255) to   (ASN336)  VX-680/MK-0457 BINDS TO HUMAN ABL1 ALSO IN INACTIVE DFG CONFORMATIONS.  |   KINASE, TRANSFERASE, ABL1, DFG CONFORMATIONS 
4zp5:A    (TYR40) to   (HIS148)  MAP4K4 IN COMPLEX WITH INHIBITOR  |   KINASE, INHIBITOR, TRANSFERASE-INHIBITOR COMPLEX 
2gs7:B   (LYS713) to   (ARG808)  CRYSTAL STRUCTURE OF THE INACTIVE EGFR KINASE DOMAIN IN COMPLEX WITH AMP-PNP  |   EGFR, KINASE, INACTIVE, AMP-PNP, TRANSFERASE 
3ii5:A   (GLY468) to   (GLU544)  THE COMPLEX OF WILD-TYPE B-RAF WITH PYRAZOLO PYRIMIDINE INHIBITOR  |   B-RAF, KINASE, PROTEIN-INHIBITOR COMPLEX, ACETYLATION, ATP- BINDING, CARDIOMYOPATHY, CYTOPLASM, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ZINC, ZINC- FINGER 
3ii5:B   (LYS472) to   (GLU544)  THE COMPLEX OF WILD-TYPE B-RAF WITH PYRAZOLO PYRIMIDINE INHIBITOR  |   B-RAF, KINASE, PROTEIN-INHIBITOR COMPLEX, ACETYLATION, ATP- BINDING, CARDIOMYOPATHY, CYTOPLASM, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ZINC, ZINC- FINGER 
3ik3:A   (GLU255) to   (SER336)  AP24534, A PAN-BCR-ABL INHIBITOR FOR CHRONIC MYELOID LEUKEMIA, POTENTLY INHIBITS THE T315I MUTANT AND OVERCOMES MUTATION-BASED RESISTANCE  |   BCR-ABL, CML, T315I, INHIBITOR, MUTATION, DRUG RESISTANCE, ALTERNATIVE SPLICING, ATP-BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
3ik3:B   (GLU255) to   (SER336)  AP24534, A PAN-BCR-ABL INHIBITOR FOR CHRONIC MYELOID LEUKEMIA, POTENTLY INHIBITS THE T315I MUTANT AND OVERCOMES MUTATION-BASED RESISTANCE  |   BCR-ABL, CML, T315I, INHIBITOR, MUTATION, DRUG RESISTANCE, ALTERNATIVE SPLICING, ATP-BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
4ztl:A   (PHE197) to   (HIS306)  IRAK4-INHIBITOR CO-STRUCTURE  |   KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ztl:B   (GLY198) to   (HIS306)  IRAK4-INHIBITOR CO-STRUCTURE  |   KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ztl:C   (GLY198) to   (HIS306)  IRAK4-INHIBITOR CO-STRUCTURE  |   KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ztl:D   (GLY198) to   (HIS306)  IRAK4-INHIBITOR CO-STRUCTURE  |   KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ztm:B   (GLY198) to   (HIS306)  IRAK4-INHIBITOR CO-STRUCTURE  |   KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ztn:A   (GLY198) to   (HIS306)  IRAK4-INHIBITOR CO-STRUCTURE  |   KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ztn:B   (GLY198) to   (HIS306)  IRAK4-INHIBITOR CO-STRUCTURE  |   KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4lgd:B    (GLY39) to   (ARG141)  STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5  |   HIPPO, MST AUTOACTIVATION, RASSF, SARAH DOMAIN, DIMERIZATION, SIGNALING PROTEIN 
3is5:D   (LEU151) to   (HIS255)  CRYSTAL STRUCTURE OF CDPK KINASE DOMAIN FROM TOXOPLASMA GONDII, TGME49_018720  |   TOXOPLASMA GONDII, CDPK, STRUCTURAL GENOMICS, PARASITOLOGY, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3is5:E   (LEU151) to   (HIS255)  CRYSTAL STRUCTURE OF CDPK KINASE DOMAIN FROM TOXOPLASMA GONDII, TGME49_018720  |   TOXOPLASMA GONDII, CDPK, STRUCTURAL GENOMICS, PARASITOLOGY, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
2hak:C    (ALA65) to   (LYS169)  CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1  |   SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
2hak:H    (PHE64) to   (LYS169)  CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1  |   SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
2hiw:A   (GLU276) to   (ASN354)  CRYSTAL STRUCTURE OF INACTIVE CONFORMATION ABL KINASE CATALYTIC DOMAIN COMPLEXED WITH TYPE II INHIBITOR  |   KINASE DOMAIN, TRANSFERASE 
3vrz:B   (MET283) to   (GLN358)  CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRROLO-PYRIMIDINE INHIBITOR 1-[4-(4-AMINO-7-CYCLOPENTYL-7H-PYRROLO[2,3-D]PYRIMIDIN-5-YL)PHENYL]- 3-BENZYLUREA  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3vs1:A   (MET283) to   (GLN358)  CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRROLO-PYRIMIDINE INHIBITOR 1-[4-(4-AMINO-7-CYCLOPENTYL-7H-PYRROLO[2,3-D]PYRIMIDIN-5-YL)PHENYL]- 3-PHENYLUREA  |   TYROSINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3vs3:A   (MET283) to   (GLN358)  CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRROLO-PYRIMIDINE INHIBITOR 7-[TRANS-4-(4-METHYLPIPERAZIN-1-YL)CYCLOHEXYL]-5-(4-PHENOXYPHENYL)- 7H-PYRROLO[2,3-D]PYRIMIDIN-4-AMINE  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2hk5:A   (MET261) to   (GLN336)  HCK KINASE IN COMPLEX WITH LCK TARGETTED INHIBITOR PG-1009247  |   HCK, SRC-FAMILY, KINASE DOMAIN, TRANSFERASE 
3vs4:A   (MET283) to   (GLN358)  CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRROLO-PYRIMIDINE INHIBITOR 5-(4-PHENOXYPHENYL)-7-(TETRAHYDRO-2H-PYRAN-4-YL)-7H-PYRROLO[2,3- D]PYRIMIDIN-4-AMINE  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3vs7:B   (MET283) to   (GLN358)  CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRAZOLO-PYRIMIDINE INHIBITOR 1-CYCLOPENTYL-3-(1H-PYRROLO[2,3-B]PYRIDIN-5-YL)-1H- PYRAZOLO[3,4-D]PYRIMIDIN-4-AMINE  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1hxp:A    (PRO87) to   (ASP208)  NUCLEOTIDE TRANSFERASE  |   METALLOENZYME, GALACTOSEMIA, NUCLEOTIDYL TRANSFERASE, COMPLEX (SERINE PROTEASE/INHIBITOR) 
3vum:A    (GLY38) to   (GLY146)  CRYSTAL STRUCTURE OF A CYSTEINE-DEFICIENT MUTANT M7 IN MAP KINASE JNK1  |   TRANSCRIPTION, PHOSPHORYLATION, ATP BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3vwa:B    (ASP34) to   (GLY125)  CRYSTAL STRUCTURE OF CEX1P  |   TRNA, NUCLEAR EXPORT, HEAT REPEAT, KINASE LIKE DOMAIN, HYDROLASE 
4lrm:D   (GLY729) to   (ASN811)  EGFR D770_N771INSNPG IN COMPLEX WITH PD168393  |   EGFR, KINASE, PD168393, 34-JAB, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1u5r:B    (GLY40) to   (ASN146)  CRYSTAL STRUCTURE OF THE TAO2 KINASE DOMAIN: ACTIVATION AND SPECIFITY OF A STE20P MAP3K  |   SERINE/THREONINE PROTEIN KINASE, TRANSFERASE 
3w2c:G   (LEU149) to   (CYS247)  STRUCTURE OF AURORA KINASE A COMPLEXED TO BENZOIMIDAZOLE-INDAZOLE INHIBITOR XV  |   KINASE, ATP COMPETITOR, TRANSFERASE 
2hw6:A    (ALA61) to   (GLY165)  CRYSTAL STRUCTURE OF MNK1 CATALYTIC DOMAIN  |   PROTEIN KINASE, DRUG DESIGN, MNK1, PHOSPHORYLATION, TRANSFERASE 
2hw6:B    (GLY65) to   (GLY165)  CRYSTAL STRUCTURE OF MNK1 CATALYTIC DOMAIN  |   PROTEIN KINASE, DRUG DESIGN, MNK1, PHOSPHORYLATION, TRANSFERASE 
5a4e:A   (GLY171) to   (ALA277)  DYRK1A IN COMPLEX WITH METHOXY BENZOTHIAZOLE FRAGMENT  |   TRANSFERASE 
5a4q:A   (GLY171) to   (ALA277)  DYRK1A IN COMPLEX WITH CHLORO BENZOTHIAZOLE FRAGMENT  |   TRANSFERASE 
2hyy:A   (GLU255) to   (ASN336)  HUMAN ABL KINASE DOMAIN IN COMPLEX WITH IMATINIB (STI571, GLIVEC)  |   TYROSINE KINASE, TRANSFERASE 
2hyy:B   (GLU255) to   (ASN336)  HUMAN ABL KINASE DOMAIN IN COMPLEX WITH IMATINIB (STI571, GLIVEC)  |   TYROSINE KINASE, TRANSFERASE 
2hyy:D   (GLU255) to   (ASN336)  HUMAN ABL KINASE DOMAIN IN COMPLEX WITH IMATINIB (STI571, GLIVEC)  |   TYROSINE KINASE, TRANSFERASE 
1ias:A   (GLY217) to   (MET318)  CYTOPLASMIC DOMAIN OF UNPHOSPHORYLATED TYPE I TGF-BETA RECEPTOR CRYSTALLIZED WITHOUT FKBP12  |   KINASE, TGF-BETA RECEPTOR, GS REGION, TRANSFERASE 
1ias:B   (GLY217) to   (HIS317)  CYTOPLASMIC DOMAIN OF UNPHOSPHORYLATED TYPE I TGF-BETA RECEPTOR CRYSTALLIZED WITHOUT FKBP12  |   KINASE, TGF-BETA RECEPTOR, GS REGION, TRANSFERASE 
1ias:C   (GLY217) to   (HIS317)  CYTOPLASMIC DOMAIN OF UNPHOSPHORYLATED TYPE I TGF-BETA RECEPTOR CRYSTALLIZED WITHOUT FKBP12  |   KINASE, TGF-BETA RECEPTOR, GS REGION, TRANSFERASE 
1ias:D   (GLY217) to   (HIS317)  CYTOPLASMIC DOMAIN OF UNPHOSPHORYLATED TYPE I TGF-BETA RECEPTOR CRYSTALLIZED WITHOUT FKBP12  |   KINASE, TGF-BETA RECEPTOR, GS REGION, TRANSFERASE 
1ias:E   (GLY217) to   (HIS317)  CYTOPLASMIC DOMAIN OF UNPHOSPHORYLATED TYPE I TGF-BETA RECEPTOR CRYSTALLIZED WITHOUT FKBP12  |   KINASE, TGF-BETA RECEPTOR, GS REGION, TRANSFERASE 
2i0y:A   (ALA599) to   (ASN773)  CFMS TYROSINE KINASE (FGF KID) IN COMPLEX WITH AN ARYLAMIDE INHIBITOR  |   TYROSINE KINASE, KINASE INHIBITOR COMPLEX, TRANSFERASE 
2i1m:A   (ALA599) to   (ASN773)  CFMS TYROSINE KINASE (TIE2 KID) IN COMPLEX WITH AN ARYLAMIDE INHIBITOR  |   KINASE DOMAIN, KINASE INHIBITOR COMPLEX, TRANSFERASE 
2wu6:A   (LYS169) to   (GLN278)  CRYSTAL STRUCTURE OF THE HUMAN CLK3 IN COMPLEX WITH DKI  |   TRANSFERASE, KINASE, TYROSINE-PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING 
2wu7:A   (LYS169) to   (GLN278)  CRYSTAL STRUCTURE OF THE HUMAN CLK3 IN COMPLEX WITH V25  |   TRANSFERASE, KINASE, TYROSINE-PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING 
1iep:A   (GLU255) to   (SER336)  CRYSTAL STRUCTURE OF THE C-ABL KINASE DOMAIN IN COMPLEX WITH STI-571.  |   KINASE, KINASE INHIBITOR, STI-571, ACTIVATION LOOP, TRANSFERASE 
1iep:B   (GLU255) to   (SER336)  CRYSTAL STRUCTURE OF THE C-ABL KINASE DOMAIN IN COMPLEX WITH STI-571.  |   KINASE, KINASE INHIBITOR, STI-571, ACTIVATION LOOP, TRANSFERASE 
1ukh:A    (GLY38) to   (GLY146)  STRUCTURAL BASIS FOR THE SELECTIVE INHIBITION OF JNK1 BY THE SCAFFOLDING PROTEIN JIP1 AND SP600125  |   TRANSFERASE, PHOSPHORYLATION 
2i7q:A   (LEU124) to   (GLY237)  CRYSTAL STRUCTURE OF HUMAN CHOLINE KINASE A  |   NON-PROTEIN KINASE, CHOLINE KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
4m69:A    (GLY78) to   (GLY222)  CRYSTAL STRUCTURE OF THE MOUSE RIP3-MLKL COMPLEX  |   KINASE, PHOSPHORYLATION, TRANSFERASE-SIGNALING PROTEIN COMPLEX 
1is1:A    (ALA55) to   (MET183)  CRYSTAL STRUCTURE OF RIBOSOME RECYCLING FACTOR FROM VIBRIO PARAHAEMOLYTICUS  |   TRANSLATION 
5aab:A  (GLY1128) to  (HIS1244)  STRUCTURE OF C1156Y,L1198F MUTANT HUMAN ANAPLASTIC LYMPHOMA KINASE IN COMPLEX WITH CRIZOTINIB  |   TRANSFERASE, RECEPTOR TYROSINE KINASE, ANAPLASTIC LYMPHOMA KINASE, INHIBITOR, MUTANT 
2wzj:F    (ALA65) to   (PHE170)  CATALYTIC AND UBA DOMAIN OF KINASE MARK2/(PAR-1) K82R, T208E DOUBLE MUTANT  |   UBA DOMAIN, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, SIGNALING PROTEIN, S/T PROTEIN KINASE, DIFFERENTIATION, DEVELOPMENTAL PROTEIN 
4mao:A   (SER434) to   (GLY534)  RSK2 T493M C-TERMINAL KINASE DOMAIN IN COMPLEX WITH RMM58  |   PROTEIN KINASE, PHOSPHORYLATION, COVALENT INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4mbj:A   (THR470) to   (GLU545)  HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH AN IMIDAZOPYRIDINE-BASED INHIBITOR  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1uwh:A   (LYS472) to   (GLU544)  THE COMPLEX OF WILD TYPE B-RAF AND BAY439006  |   TRANSFERASE 
1uwh:B   (LYS472) to   (GLU544)  THE COMPLEX OF WILD TYPE B-RAF AND BAY439006  |   TRANSFERASE 
1uwj:A   (LYS472) to   (GLU544)  THE COMPLEX OF MUTANT V599E B-RAF AND BAY439006  |   TRANSFERASE, THREONINE-PROTEIN KINASE, SIGNAL TRANSDUCTION 
1uwj:B   (LYS472) to   (GLU544)  THE COMPLEX OF MUTANT V599E B-RAF AND BAY439006  |   TRANSFERASE, THREONINE-PROTEIN KINASE, SIGNAL TRANSDUCTION 
3wf9:A   (GLN107) to   (GLY213)  CRYSTAL STRUCTURE OF S6K1 KINASE DOMAIN IN COMPLEX WITH A QUINOLINE DERIVATIVE 1-OXO-1-[(4-SULFAMOYLPHENYL)AMINO]PROPAN-2-YL-2-METHYL-1, 2,3,4-TETRAHYDROACRIDINE-9-CARBOXYLATE  |   SERINE/THREONINE PROTEIN KINASE DOMAIN, TRANSFERASE, PHOSPHORYLATION, ATP-BINDING, ZINC-BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2in6:A   (PHE310) to   (SER421)  WEE1 KINASE COMPLEX WITH INHIBITOR PD311839  |   PROTEIN-INHIBITOR COMPLEX, TRANSFERASE 
5afv:A   (LEU124) to   (MET238)  PHARMACOPHORE-BASED VIRTUAL SCREENING TO DISCOVER NEW ACTIVE COMPOUNDS FOR HUMAN CHOLINE KINASE ALPHA1.  |   TRANSFERASE, VIRTUAL SCREENING, PHARMACOPHORE 
5afv:B   (LEU124) to   (MET238)  PHARMACOPHORE-BASED VIRTUAL SCREENING TO DISCOVER NEW ACTIVE COMPOUNDS FOR HUMAN CHOLINE KINASE ALPHA1.  |   TRANSFERASE, VIRTUAL SCREENING, PHARMACOPHORE 
4mh7:A   (SER600) to   (ASN718)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE-PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR UNC1896  |   TYROSINE KINASE, ACUTE LYMPHOBLASTIC LEUKEMIA, RATIONAL STRUCTURE BASED DRUG DESIGN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4mh7:B   (GLY604) to   (ASN718)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE-PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR UNC1896  |   TYROSINE KINASE, ACUTE LYMPHOBLASTIC LEUKEMIA, RATIONAL STRUCTURE BASED DRUG DESIGN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4mha:A   (GLY604) to   (ASN718)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE-PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR UNC1817  |   TYROSINE KINASE, ACUTE LYMPHOBLASTIC LEUKEMIA, RATIONAL STRUCTURE- BASED DRUG DESIGN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2x6f:B   (LEU677) to   (HIS769)  THE CRYSTAL STRUCTURE OF THE DROSOPHILA CLASS III PI3-KINASE VPS34 IN COMPLEX WITH 3-METHYLADENINE  |   TRANSFERASE 
2x6k:B   (LEU677) to   (HIS769)  THE CRYSTAL STRUCTURE OF THE DROSOPHILA CLASS III PI3-KINASE VPS34 IN COMPLEX WITH PI-103  |   PI103, PI-103, AUTOPHAGY, TRANSFERASE, PI3K CLASS III, PHOSPHOINOSITIDE 3-KINASE CLASS III 
2x7f:A    (GLY37) to   (LYS148)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN TRAF2- AND NCK-INTERACTING KINASE WITH WEE1CHK1 INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, PHOSPHOPROTEIN, KINASE, TRANSFERASE 
2x7f:B    (GLY37) to   (LYS148)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN TRAF2- AND NCK-INTERACTING KINASE WITH WEE1CHK1 INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE, PHOSPHOPROTEIN, KINASE, TRANSFERASE 
1j7i:A    (LYS30) to   (ILE125)  CRYSTAL STRUCTURE OF 3',5"-AMINOGLYCOSIDE PHOSPHOTRANSFERASE TYPE IIIA APOENZYME  |   ANTIBIOTIC RESISTANCE, KINASE, ATP-BINDING, TRANSFERASE 
1j7l:B    (VAL31) to   (ILE125)  CRYSTAL STRUCTURE OF 3',5"-AMINOGLYCOSIDE PHOSPHOTRANSFERASE TYPE IIIA ADP COMPLEX  |   ANTIBIOTIC RESISTANCE, KINASE, ATP-BINDING, TRANSFERASE 
1j7u:A    (PRO28) to   (ILE125)  CRYSTAL STRUCTURE OF 3',5"-AMINOGLYCOSIDE PHOSPHOTRANSFERASE TYPE IIIA AMPPNP COMPLEX  |   ANTIBIOTIC RESISTANCE, KINASE, ATP-BINDING, TRANSFERASE 
2x9e:A   (SER537) to   (GLY642)  HUMAN MPS1 IN COMPLEX WITH NMS-P715  |   KINASE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE, MITOTIC CHECKPOINT 
5am6:A   (ASN506) to   (LYS618)  NATIVE FGFR1 WITH AN INHIBITOR  |   TRANSFERASE, FGFR, GROWTH FACTOR, CANCER, DOVITINIB, TKI258, KINASE 
4mne:C   (THR470) to   (GLU545)  CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX  |   RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4mne:F   (THR470) to   (GLU545)  CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX  |   RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4mne:G   (THR470) to   (GLU545)  CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX  |   RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4mnf:A   (LYS473) to   (GLU545)  CRYSTAL STRUCTURE OF BRAF-V600E BOUND TO GDC0879  |   RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, ACTIVE CONFORMATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5ap5:A   (GLN541) to   (GLY642)  NATURALLY OCCURRING MUTATIONS IN THE MPS1 GENE PREDISPOSE CELLS TO KINASE INHIBITOR DRUG RESISTANCE.  |   TRANSFERASE, MPS1, PROTEIN KINASE, MITOSIS, DRUG RESISTANCE 
4mq1:C   (GLY171) to   (THR278)  THE CRYSTAL STRUCTURE OF DYRK1A WITH A BOUND PYRIDO[2,3-D]PYRIMIDINE INHIBITOR  |   DYRK1A, DYRK1B, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1jkk:A    (ALA25) to   (PHE119)  2.4A X-RAY STRUCTURE OF TERNARY COMPLEX OF A CATALYTIC DOMAIN OF DEATH-ASSOCIATED PROTEIN KINASE WITH ATP ANALOGUE AND MG.  |   TRANSFERASE 
4mwi:A   (SER215) to   (HIS321)  CRYSTAL STRUCTURE OF THE HUMAN MLKL PSEUDOKINASE DOMAIN  |   PSEUDOKINASE, NECROPTOSIS, TRANSFERASE 
2j90:A    (ALA25) to   (ARG134)  CRYSTAL STRUCTURE OF HUMAN ZIP KINASE IN COMPLEX WITH A TETRACYCLIC PYRIDONE INHIBITOR (PYRIDONE 6)  |   NUCLEAR PROTEIN, NUCLEOTIDE-BINDING, SERINE/THREONINE- PROTEIN KINASE, CHROMATIN REGULATOR, MYOSIN PHOSPHORYLATION, KINASE, MUSCLE, APOPTOSIS, TRANSFERASE, ATP-BINDING 
5awm:A    (ILE37) to   (GLY144)  THE CRYSTAL STRUCTURE OF JNK FROM DROSOPHILA MELANOGASTER REVEALS AN EVOLUTIONARILY CONSERVED TOPOLOGY WITH THAT OF MAMMALIAN JNK PROTEINS.  |   C-JUN N-TERMINAL KINASE, MAP KINASE, DROSOPHILA JNK PATHWAY, TRANSFERASE 
2xne:A   (GLY145) to   (ARG251)  STRUCTURE OF AURORA-A BOUND TO AN IMIDAZOPYRAZINE INHIBITOR  |   SER-THR PROTEIN KINASE COMPLEX, PROTO-ONCOGENE, KINASE, MITOSIS, CELL CYCLE, MICROTUBULE, TRANSFERASE, CYTOSKELETON, CELL DIVISION 
3wzj:A   (SER537) to   (GLY642)  CRYSTAL STRUCTURE OF HUMAN MPS1 CATALYTIC DOMAIN IN COMPLEX WITH 4-(6- (CYCLOHEXYLAMINO)-8-(((TETRAHYDRO-2H-PYRAN-4-YL)METHYL)AMINO) IMIDAZO[1,2-B]PYRIDAZIN-3-YL)-N-CYCLOPROPYLBENZAMIDE  |   TRANSFERASE, ATP BINDING, PHOSPHORYLATION 
2jbp:H    (LEU79) to   (ASN181)  PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION)  |   SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING 
2jbp:I    (GLY76) to   (ASN181)  PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION)  |   SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING 
2jbp:J    (LEU79) to   (ASN181)  PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION)  |   SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING 
3zc6:A   (GLY834) to   (ARG944)  CRYSTAL STRUCTURE OF JAK3 KINASE DOMAIN IN COMPLEX WITH AN INDAZOLE SUBSTITUTED PYRROLOPYRAZINE INHIBITOR  |   TRANSFERASE, SCID, SEVERE COMBINED IMMUNODEFICIENCY, STAT5, STAT6, INTERLEUKIN-2, COMMON-GAMMA CHAIN, ATP SITE KINASE INHIBITOR, CANCER 
2xrw:A    (ILE39) to   (GLY146)  LINEAR BINDING MOTIFS FOR JNK AND FOR CALCINEURIN ANTAGONISTICALLY CONTROL THE NUCLEAR SHUTTLING OF NFAT4  |   TRANSCRIPTION, MAPK SIGNALING PATHWAYS, LINEAR BINDING MOTIF 
5bmm:B   (GLY279) to   (ASN381)  SRC IN COMPLEX WITH DNA-TEMPLATED MACROCYCLIC INHIBITOR MC25B  |   TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5bpy:A   (GLY414) to   (GLN516)  CRYSTAL STRUCTURE OF BRUTON AGAMMAGLOBULINEMIA TYROSINE KINASE COMPLEXED WITH BMS-824171 AKA 6-[(3R)-3-(4-TERT-BU TYLBENZAMIDO) PIPERIDIN-1-YL]-2-{[4-(MORPHOLINE-4-CARBONYL) PHENYL]AMINO}PYRIDINE- 3-CARBOXAMIDE  |   KINASE, INHIBITOR, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5bq0:A   (GLY414) to   (GLN516)  CRYSTAL STRUCTURE OF BRUTON AGAMMAGLOBULINEMIA TYROSINE KINASE COMPLEXED WITH BMS-824171 AKA 6-[(3R)-3-(4-TERT-BU TYLBENZAMIDO) PIPERIDIN-1-YL]-2-{[4-(MORPHOLINE-4-CARBONYL) PHENYL]AMINO}PYRIDINE- 3-CARBOXAMIDE  |   KINASE, INHIBITOR, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2jit:B   (LYS737) to   (ARG832)  CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN T790M MUTATION  |   EGFR, T790M, KINASE, RECEPTOR, CELL CYCLE, PHOSPHORYLATION, DISEASE MUTATION, NUCLEOTIDE-BINDING, TYROSINE-PROTEIN KINASE, ANTI-ONCOGENE, EPIDERMAL GROWTH FACTOR, ATP-BINDING, TRANSFERASE 
1k2p:A   (GLY414) to   (PHE493)  CRYSTAL STRUCTURE OF BRUTON'S TYROSINE KINASE DOMAIN  |   BRUTON TRYOSINE KINASE, KINASE DOMAIN, TRANSFERASE 
1wbt:A    (ASP88) to   (LEU217)  IDENTIFICATION OF NOVEL P38 ALPHA MAP KINASE INHIBITORS USING FRAGMENT-BASED LEAD GENERATION.  |   TRANSFERASE, ATP-BINDING, DIRECT PROTEIN SEQUENCING, NUCLEAR PROTEIN, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, P38 MAP KINASE, INHIBITOR STRUCTURE 
1k9a:A   (GLY207) to   (ASN309)  CRYSTAL STRUCTURE ANALYSIS OF FULL-LENGTH CARBOXYL-TERMINAL SRC KINASE AT 2.5 A RESOLUTION  |   CARBOXYL-TERMINAL SRC KINASE, COOH-TERMINAL SRC KINASE, CSK, SRC, SFK, SIGNAL TRANSDUCTION, SH2, SH3, SRC HOMOLOGY, TYROSINE KINASE, CYTOPLASMIC TYROSINE KINASE, CBP, ONCOGENE, CANCER, TRANSFERASE 
1k9a:B   (LEU211) to   (ASN309)  CRYSTAL STRUCTURE ANALYSIS OF FULL-LENGTH CARBOXYL-TERMINAL SRC KINASE AT 2.5 A RESOLUTION  |   CARBOXYL-TERMINAL SRC KINASE, COOH-TERMINAL SRC KINASE, CSK, SRC, SFK, SIGNAL TRANSDUCTION, SH2, SH3, SRC HOMOLOGY, TYROSINE KINASE, CYTOPLASMIC TYROSINE KINASE, CBP, ONCOGENE, CANCER, TRANSFERASE 
1k9a:E   (GLY207) to   (GLY287)  CRYSTAL STRUCTURE ANALYSIS OF FULL-LENGTH CARBOXYL-TERMINAL SRC KINASE AT 2.5 A RESOLUTION  |   CARBOXYL-TERMINAL SRC KINASE, COOH-TERMINAL SRC KINASE, CSK, SRC, SFK, SIGNAL TRANSDUCTION, SH2, SH3, SRC HOMOLOGY, TYROSINE KINASE, CYTOPLASMIC TYROSINE KINASE, CBP, ONCOGENE, CANCER, TRANSFERASE 
1k9a:F   (GLY207) to   (ASN309)  CRYSTAL STRUCTURE ANALYSIS OF FULL-LENGTH CARBOXYL-TERMINAL SRC KINASE AT 2.5 A RESOLUTION  |   CARBOXYL-TERMINAL SRC KINASE, COOH-TERMINAL SRC KINASE, CSK, SRC, SFK, SIGNAL TRANSDUCTION, SH2, SH3, SRC HOMOLOGY, TYROSINE KINASE, CYTOPLASMIC TYROSINE KINASE, CBP, ONCOGENE, CANCER, TRANSFERASE 
2y4p:A    (PHE24) to   (GLN134)  DIMERIC STRUCTURE OF DAPK-1 CATALYTIC DOMAIN  |   CALMODULIN-BINDING, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, APOPTOSIS, TRANSFERASE, ATP-BINDING 
3zmm:A   (GLY861) to   (ASP949)  INHIBITORS OF JAK2 KINASE DOMAIN  |   TRANSFERASE 
1wqf:A    (SER56) to   (LEU183)  CRYSTAL STRUCTURE OF RIBOSOME RECYCLING FACTOR FROM MYCOBACTERIUM TUBERCULOSIS  |   TRANSLATION FACTOR, TRIPLE-HELIX BUNDLE, PROTEIN SYNTHESIS, TRANSLATION 
1wqg:A    (SER56) to   (LEU183)  CRYSTAL STRUCTURE OF RIBOSOME RECYCLING FACTOR FROM MYCOBACTERIUM TUBERCULOSIS  |   TRANSLATION FACTOR, TRIPLE-HELIX BUNDLE, PROTEIN SYNTHESIS, TRANSLATION 
1wvw:A    (ALA25) to   (GLN134)  CRYSTAL STRUCTURES OF KINASE DOMAIN OF DAP KINASE IN COMPLEX WITH SMALL MOLECULAR INHIBITORS  |   PROTEIN KINASE, APOPTOSIS, TRANSFERASE 
1wvx:A    (ALA25) to   (GLU118)  CRYSTAL STRUCTURES OF KINASE DOMAIN OF DAP KINASE IN COMPLEX WITH SMALL MOLECULAR INHIBITORS  |   PROTEIN KINASE, APOPTOSIS, STAUROSPORINE, TRANSFERASE 
2yab:A    (LYS29) to   (LYS134)  CRYSTAL STRUCTURE OF THE AUTOINHIBITED FORM OF MOUSE DAPK2 IN COMPLEX WITH AMP  |   APOPTOSIS, TRANSFERASE 
1kob:A    (GLY65) to   (SER169)  TWITCHIN KINASE FRAGMENT (APLYSIA), AUTOREGULATED PROTEIN KINASE DOMAIN  |   KINASE, TWITCHIN, INTRASTERIC REGULATION 
1kob:B    (GLY65) to   (SER169)  TWITCHIN KINASE FRAGMENT (APLYSIA), AUTOREGULATED PROTEIN KINASE DOMAIN  |   KINASE, TWITCHIN, INTRASTERIC REGULATION 
4nus:A    (LEU84) to   (GLY188)  RSK2 N-TERMINAL KINASE IN COMPLEX WITH LJH685  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3zxt:D    (ALA25) to   (GLU118)  DIMERIC STRUCTURE OF DAPK-1 CATALYTIC DOMAIN IN COMPLEX WITH AMPPCP-MG  |   APOPTOSIS, TRANSFERASE, ATP BINDING 
4o38:A    (ALA52) to   (GLN165)  CRYSTAL STRUCTURE OF THE HUMAN CYCLIN G ASSOCIATED KINASE (GAK)  |   STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE, PROTEIN KINASE, SERINE/THREONINE KINASE, CYCLIN G, P53, CLATHRINE, MEMBRANE TRAFFICKING, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ATP- BINDING, CELL CYCLE, CELL JUNCTION, GOLGI APPARATUS, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN 
4o38:B    (PHE51) to   (GLN165)  CRYSTAL STRUCTURE OF THE HUMAN CYCLIN G ASSOCIATED KINASE (GAK)  |   STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE, PROTEIN KINASE, SERINE/THREONINE KINASE, CYCLIN G, P53, CLATHRINE, MEMBRANE TRAFFICKING, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ATP- BINDING, CELL CYCLE, CELL JUNCTION, GOLGI APPARATUS, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN 
2nru:A   (GLY198) to   (HIS306)  CRYSTAL STRUCTURE OF IRAK-4  |   KINASE, INHIBITOR, IRAK, TRANSFERASE 
2nru:C   (VAL199) to   (HIS306)  CRYSTAL STRUCTURE OF IRAK-4  |   KINASE, INHIBITOR, IRAK, TRANSFERASE 
2nry:A   (GLY198) to   (HIS306)  CRYSTAL STRUCTURE OF IRAK-4  |   KINASE, INHIBITOR, STAUROSPORINE, TRANSFERASE 
2nry:D   (GLY198) to   (HIS306)  CRYSTAL STRUCTURE OF IRAK-4  |   KINASE, INHIBITOR, STAUROSPORINE, TRANSFERASE 
4obo:B    (TYR40) to   (HIS148)  MAP4K4 IN COMPLEX WITH INHIBITOR (COMPOUND 22), 6-(3-CHLOROPHENYL) QUINAZOLIN-4-AMINE  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2z2w:A   (GLY311) to   (SER421)  HUMAND WEE1 KINASE COMPLEXED WITH INHIBITOR PF0335770  |   WEE1 KINASE, INHIBITOR COMPLEX, TRANSFERASE 
2o0u:A    (GLY76) to   (GLY184)  CRYSTAL STRUCTURE OF HUMAN JNK3 COMPLEXED WITH N-{3-CYANO-6-[3-(1- PIPERIDINYL)PROPANOYL]-4,5,6,7-TETRAHYDROTHIENO[2,3-C]PYRIDIN-2-YL}- 1-NAPHTHALENECARBOXAMIDE  |   KINASE FOLD, TRANSFERASE 
2z60:A   (GLU255) to   (SER336)  CRYSTAL STRUCTURE OF THE T315I MUTANT OF ABL KINASE BOUND WITH PPY-A  |   ABL, KINASE, MUTANT, T315I, ALTERNATIVE SPLICING, ATP- BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHORYLATION, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
4oli:A   (GLY909) to  (GLN1017)  THE PSEUDOKINASE/KINASE PROTEIN FROM JAK-FAMILY MEMBER TYK2  |   PROTEIN KINASE, PHOSPHO-TRANSFER, TRANSFERASE 
5csx:A   (GLY469) to   (GLU545)  CRYSTAL STRUCTURE OF B-RAF IN COMPLEX WITH BI 882370  |   KINASE, TRANSFERASE 
5ct7:A   (GLY469) to   (GLU545)  BRAF IN COMPLEX WITH RAF265  |   KINASE, TRANSFERASE 
5ct7:B   (LYS473) to   (GLU545)  BRAF IN COMPLEX WITH RAF265  |   KINASE, TRANSFERASE 
3kcf:A   (GLY217) to   (MET318)  CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A PYRAZOLONE INHIBITOR  |   KINASE, TGFBETARI, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, AORTIC ANEURYSM, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE 
3kcf:C   (GLY217) to   (HIS317)  CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A PYRAZOLONE INHIBITOR  |   KINASE, TGFBETARI, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, AORTIC ANEURYSM, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE 
3kcf:D   (GLY217) to   (HIS317)  CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A PYRAZOLONE INHIBITOR  |   KINASE, TGFBETARI, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, AORTIC ANEURYSM, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE 
3kcf:E   (GLY217) to   (MET318)  CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A PYRAZOLONE INHIBITOR  |   KINASE, TGFBETARI, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, AORTIC ANEURYSM, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE 
4aaa:A    (MET17) to   (GLY113)  CRYSTAL STRUCTURE OF THE HUMAN CDKL2 KINASE DOMAIN  |   TRANSFERASE, PHOSPHO-MIMETIC 
3kf4:A   (GLU258) to   (SER336)  STRUCTURAL ANALYSIS OF DFG-IN AND DFG-OUT DUAL SRC-ABL INHIBITORS SHARING A COMMON VINYL PURINE TEMPLATE  |   ABL, CML, DRUG RESISTANCE, INHIBITOR, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, ONCOGENE, TYROSINE-PROTEIN KINASE, TRANSFERASE 
3kf4:B   (GLU255) to   (SER336)  STRUCTURAL ANALYSIS OF DFG-IN AND DFG-OUT DUAL SRC-ABL INHIBITORS SHARING A COMMON VINYL PURINE TEMPLATE  |   ABL, CML, DRUG RESISTANCE, INHIBITOR, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, ONCOGENE, TYROSINE-PROTEIN KINASE, TRANSFERASE 
2zm1:A   (PHE256) to   (LEU336)  CRYSTAL STRUCTURE OF IMIDAZO PYRAZIN 1 BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394)  |   TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE- BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
2zm3:A  (PRO1026) to  (LYS1130)  COMPLEX STRUCTURE OF INSULIN-LIKE GROWTH FACTOR RECEPTOR AND ISOQUINOLINEDIONE INHIBITOR  |   IGFR, PROTEIN-INHIBITOR COMPLEX, TYROSINE KINASE, ATP- BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
1m7n:B  (GLY1013) to  (LYS1127)  CRYSTAL STRUCTURE OF UNACTIVATED APO INSULIN-LIKE GROWTH FACTOR-1 RECEPTOR KINASE DOMAIN  |   TRANSFERASE 
5cyz:A    (GLY21) to   (SER123)  STRUCTURE OF S. CEREVISIAE HRR25:MAM1 COMPLEX, FORM 1  |   CASEIN KINASE, MONOPOLIN, TRANSFERASE 
5czo:A    (GLY21) to   (SER123)  STRUCTURE OF S. CEREVISIAE HRR25:MAM1 COMPLEX, FORM 2  |   CASEIN KINASE, MONOPOLIN, TRANSFERASE 
5czo:B    (GLY21) to   (SER123)  STRUCTURE OF S. CEREVISIAE HRR25:MAM1 COMPLEX, FORM 2  |   CASEIN KINASE, MONOPOLIN, TRANSFERASE 
3kk8:A    (SER25) to   (GLY130)  CAMKII SUBSTRATE COMPLEX A  |   PROTEIN KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
2zv7:A   (MET263) to   (VAL339)  LYN TYROSINE KINASE DOMAIN, APO FORM  |   LYN KINASE, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
2zv8:A   (GLY259) to   (VAL339)  LYN TYROSINE KINASE DOMAIN-AMP-PNP COMPLEX  |   LYN KINASE AMPPNP, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
2zv9:A   (GLY259) to   (VAL339)  LYN TYROSINE KINASE DOMAIN-PP2 COMPLEX  |   LYN KINASE PP2, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
2zva:A   (GLY259) to   (VAL339)  LYN TYROSINE KINASE DOMAIN-DASATINIB COMPLEX  |   LYN KINASE DASATINIB, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
4agd:A   (ALA851) to  (SER1021)  CRYSTAL STRUCTURE OF VEGFR2 (JUXTAMEMBRANE AND KINASE DOMAINS) IN COMPLEX WITH SUNITINIB (SU11248) (N-2- DIETHYLAMINOETHYL)-5-((Z)-(5-FLUORO-2-OXO-1H-INDOL-3- YLIDENE)METHYL)-2,4-DIMETHYL-1H-PYRROLE-3-CARBOXAMIDE)  |   TRANSFERASE, ANGIOGENESIS, NUCLEOTIDE-BINDING, INHIBITOR, PHOSPHORYLATION, TRANSMEMBRANE 
4agw:A   (GLY279) to   (LEU358)  DISCOVERY OF A SMALL MOLECULE TYPE II INHIBITOR OF WILD- TYPE AND GATEKEEPER MUTANTS OF BCR-ABL, PDGFRALPHA, KIT, AND SRC KINASES  |   ATP-BINDING, LIPOPROTEIN, MYRISTATE, PHOSPHOPROTEIN, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
3kmm:A   (GLY257) to   (LEU336)  STRUCTURE OF HUMAN LCK KINASE WITH A SMALL MOLECULE INHIBITOR  |   TYROSINE KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
2zyb:A   (PHE256) to   (LEU336)  CRYSTAL STRUCTURE OF PHENYLIMIDAZO PYRAZIN 2 BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394)  |   TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, KINASE, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, CELL MEMBRANE, POLYMORPHISM 
3a4o:X    (GLU29) to   (VAL108)  LYN KINASE DOMAIN  |   SRC FAMILY, KINASE DOMAIN, ALTERNATIVE SPLICING, ATP- BINDING, HOST-VIRUS INTERACTION, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3a60:A   (GLN107) to   (GLY213)  CRYSTAL STRUCTURE OF UNPHOSPHORYLATED P70S6K1 (FORM I)  |   KINASE, KINASE DOMAIN, INACTIVE, ACTIVE, RIBOSOMAL S6 KINASE, ACTIVATION, ALTERNATIVE INITIATION, ATP-BINDING, CELL JUNCTION, CYTOPLASM, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, SYNAPSE, SYNAPTOSOME, TRANSFERASE 
3a61:A   (LYS104) to   (GLY213)  CRYSTAL STRUCTURE OF UNPHOSPHORYLATED P70S6K1 (FORM II)  |   KINASE, KINASE DOMAIN, INACTIVE, ACTIVE, RIBOSOMAL S6 KINASE, ACTIVATION, ALTERNATIVE INITIATION, ATP-BINDING, CELL JUNCTION, CYTOPLASM, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, SYNAPSE, SYNAPTOSOME, TRANSFERASE 
3a62:A   (GLN107) to   (GLY213)  CRYSTAL STRUCTURE OF PHOSPHORYLATED P70S6K1  |   KINASE, KINASE DOMAIN, INACTIVE, ACTIVE, RIBOSOMAL S6 KINASE, ACTIVATION, ALTERNATIVE INITIATION, ATP-BINDING, CELL JUNCTION, CYTOPLASM, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, SYNAPSE, SYNAPTOSOME, TRANSFERASE 
5d9l:A    (GLY80) to   (GLY188)  RSK2 N-TERMINAL KINASE IN COMPLEX WITH BIS-PHENOL PYRAZOLE  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1yi6:A   (GLY279) to   (LEU358)  C-TERM TAIL SEGMENT OF HUMAN TYROSINE KINASE (258-533)  |   SRC, TYROSINE KINASE, PHOSPHORYLATION, REGULATION, SH2, SH3, TRANSFERASE 
3kxz:A   (MET261) to   (LEU336)  THE COMPLEX CRYSTAL STRUCTURE OF LCK WITH A PROBE MOLECULE W259  |   LCK, ACETYLATION, ATP-BINDING, CELL MEMBRANE, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, KINASE, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, TRANSFERASE, TYROSINE-PROTEIN KINASE, STRUCTURAL GENOMICS, PROTEIN STRUCTURE FACTORY, PSF 
1yom:A   (GLY286) to   (TYR359)  CRYSTAL STRUCTURE OF SRC KINASE DOMAIN IN COMPLEX WITH PURVALANOL A  |   PROTEIN TYROSINE KINASE, TRANSFERASE 
1yom:B   (GLY281) to   (LEU360)  CRYSTAL STRUCTURE OF SRC KINASE DOMAIN IN COMPLEX WITH PURVALANOL A  |   PROTEIN TYROSINE KINASE, TRANSFERASE 
3ac1:A   (PHE256) to   (LEU336)  CRYSTAL STRUCTURE OF PYRAZIN DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394)  |   TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
3ac4:A   (PHE256) to   (LEU336)  CRYSTAL STRUCTURE OF TRIAZOLO PYRIMIDINE DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394)  |   TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
3acj:A   (PHE256) to   (LEU336)  CRYSTAL STRUCTURE OF IMIDAZO PYRIMIDINE DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394)  |   TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
3ack:A   (PHE256) to   (LEU336)  CRYSTAL STRUCTURE OF PYRROLO PYRAZINE DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394)  |   TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
3ad5:A   (PHE256) to   (LEU336)  CRYSTAL STRUCTURE OF TRIAZOLONE DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394)  |   TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
5di1:B    (GLN38) to   (HIS148)  MAP4K4 IN COMPLEX WITH AN INHIBITOR  |   KINASE, INHIBITOR, COMPLEX, MEDICINAL CHEMISTRY, TRANSFERASE- INHIBITOR COMPLEX 
4pmm:A   (ALA527) to   (HIS645)  THE STRUCTURE OF TRKA KINASE BOUND TO THE INHIBITOR N-(3-CYCLOPROPYL- 1-PHENYL-1H-PYRAZOL-5-YL)-2-{4-[3-METHOXY-4-(4-METHYL-1H-IMIDAZOL-1- YL)PHENYL]-1H-1,2,3-TRIAZOL-1-YL}ACETAMIDE  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4pmp:A   (ALA527) to   (HIS645)  THE STRUCTURE OF TRKA KINASE BOUND TO THE INHIBITOR 1-CYCLOPROPYL-1- [3-(1,3-THIAZOL-2-YL)BENZYL]-3-[4-(TRIFLUOROMETHOXY)PHENYL]UREA  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4pms:A   (ALA527) to   (HIS645)  THE STRUCTURE OF TRKA KINASE BOUND TO THE INHIBITOR 4-NAPHTHALEN-1-YL- 1-[(5-PHENYL-1,2,4-OXADIAZOL-3-YL)METHYL]-1H-PYRROLO[3,2-C]PYRIDINE- 2-CARBOXYLIC ACID  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5dmz:A   (ALA799) to   (GLU912)  STRUCTURE OF HUMAN BUB1 KINASE DOMAIN PHOSPHORYLATED AT SER969  |   KINASE, PHOSPHORYLATION, TRANSFERASE 
5dmz:B   (ALA799) to   (GLU912)  STRUCTURE OF HUMAN BUB1 KINASE DOMAIN PHOSPHORYLATED AT SER969  |   KINASE, PHOSPHORYLATION, TRANSFERASE 
4pp7:A   (LYS473) to   (GLU545)  HIGHLY POTENT AND SELECTIVE 3-N-METHYLQUINAZOLINE-4(3H)-ONE BASED INHIBITORS OF B-RAFV600E KINASE  |   SERINE/THREONINE-PROTEIN KINASE B-RAF, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4pp7:B   (LYS473) to   (GLU545)  HIGHLY POTENT AND SELECTIVE 3-N-METHYLQUINAZOLINE-4(3H)-ONE BASED INHIBITORS OF B-RAFV600E KINASE  |   SERINE/THREONINE-PROTEIN KINASE B-RAF, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3lck:A   (PHE256) to   (LEU336)  THE KINASE DOMAIN OF HUMAN LYMPHOCYTE KINASE (LCK), ACTIVATED FORM (AUTO-PHOSPHORYLATED ON TYR394)  |   TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION 
4ptc:A    (GLY68) to   (GLY176)  STRUCTURE OF A CARBOXAMIDE COMPOUND (3) (2-{2-[(CYCLOPROPYLCARBONYL) AMINO]PYRIDIN-4-YL}-4-OXO-4H-1LAMBDA~4~,3-THIAZOLE-5-CARBOXAMIDE) TO GSK3B  |   SERINE/THREONINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ptc:B    (GLY68) to   (GLY176)  STRUCTURE OF A CARBOXAMIDE COMPOUND (3) (2-{2-[(CYCLOPROPYLCARBONYL) AMINO]PYRIDIN-4-YL}-4-OXO-4H-1LAMBDA~4~,3-THIAZOLE-5-CARBOXAMIDE) TO GSK3B  |   SERINE/THREONINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ptg:B    (GLY68) to   (GLY176)  STRUCTURE OF A CARBOXAMINE COMPOUND (26) (2-{2-[(CYCLOPROPYLCARBONYL) AMINO]PYRIDIN-4-YL}-4-METHOXYPYRIMIDINE-5-CARBOXAMIDE) TO GSK3B  |   SERINE/THREONINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ano:A    (ASP13) to    (VAL95)  CRYSTAL STRUCTURE GEOBACILLUS THERMODENITRIFICANS ESSB CYTOPLASMIC FRAGMENT  |   MEMBRANE PROTEIN, MEMBRANE SECRETION, ESS TYPE V SECRETION SYSTEM 
4aot:A    (GLY48) to   (ARG152)  CRYSTAL STRUCTURE OF HUMAN SERINE THREONINE KINASE-10 (LOK) BOUND TO GW830263A  |   TRANSFERASE, STK10, LOK 
3lij:A    (GLY74) to   (ASN179)  CRYSTAL STRUCTURE OF FULL LENGTH CPCDPK3 (CGD5_820) IN COMPLEX WITH CA2+ AND AMPPNP  |   TRANSFERASE, CALCIUM DEPENDENT PROTEIN KINASE, EF HAND, ATP- BINDING, CALCIUM, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC 
3lj0:A   (GLN691) to   (LYS792)  IRE1 COMPLEXED WITH ADP AND QUERCETIN  |   KINASE, FLAVONOL, ACTIVATOR, DIMER, ATP-BINDING, ENDOPLASMIC RETICULUM, GLYCOPROTEIN, HYDROLASE, MAGNESIUM, MEMBRANE, METAL- BINDING, MULTIFUNCTIONAL ENZYME, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, TRANSMEMBRANE, UNFOLDED PROTEIN RESPONSE 
3lj0:B   (GLN691) to   (LYS792)  IRE1 COMPLEXED WITH ADP AND QUERCETIN  |   KINASE, FLAVONOL, ACTIVATOR, DIMER, ATP-BINDING, ENDOPLASMIC RETICULUM, GLYCOPROTEIN, HYDROLASE, MAGNESIUM, MEMBRANE, METAL- BINDING, MULTIFUNCTIONAL ENZYME, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, TRANSMEMBRANE, UNFOLDED PROTEIN RESPONSE 
4apc:A    (LYS17) to   (LYS123)  CRYSTAL STRUCTURE OF HUMAN NIMA-RELATED KINASE 1 (NEK1)  |   TRANSFERASE 
4apc:B    (LYS17) to   (LYS123)  CRYSTAL STRUCTURE OF HUMAN NIMA-RELATED KINASE 1 (NEK1)  |   TRANSFERASE 
3anq:D   (GLY171) to   (THR278)  HUMAN DYRK1A/INHIBITOR COMPLEX  |   PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5dvr:A    (GLU64) to   (LYS169)  CRYSTAL STRUCTURE OF TGCDPK1 FROM TOXOPLASMA GONDII COMPLEXED WITH GW780159X  |   STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPKS, SERINE/THREONINE PROTEIN KINASE, NUCLEOTIDE-BINDING, GW780159X, TRANSFERASE 
3lmg:A   (SER715) to   (GLY810)  CRYSTAL STRUCTURE OF THE ERBB3 KINASE DOMAIN IN COMPLEX WITH AMP-PNP  |   ERBB3, HER3, TYROSINE KINASE DOMAIN, AMP-PNP, NUCLEOTIDE BINDING, TRANSFERASE 
4asx:A   (GLY204) to   (HIS304)  CRYSTAL STRUCTURE OF ACTIVIN RECEPTOR TYPE-IIA (ACVR2A) KINASE DOMAIN IN COMPLEX WITH DIHYDRO-BAUERINE C  |   TRANSFERASE, PROTEIN KINASE 
1zmw:A    (ALA65) to   (PHE170)  CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK2/PAR-1: T208A/S212A INACTIVE DOUBLE MUTANT  |   SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
1zmu:A    (LYS66) to   (PHE170)  CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK2/PAR-1: WILD TYPE  |   SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
1zmu:B    (LYS66) to   (PHE170)  CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK2/PAR-1: WILD TYPE  |   SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
1zmv:A    (ALA65) to   (GLN168)  CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK2/PAR-1: K82R MUTANT  |   SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
3aox:A  (GLU1129) to  (HIS1244)  X-RAY CRYSTAL STRUCTURE OF HUMAN ANAPLASTIC LYMPHOMA KINASE IN COMPLEX WITH CH5424802  |   ALK KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4awi:A    (GLY38) to   (SER144)  HUMAN JNK1ALPHA KINASE WITH 4-PHENYL-7-AZAINDOLE IKK2 INHIBITOR.  |   TRANSFERASE 
4ax8:A   (SER240) to   (GLY346)  MEDIUM RESOLUTION STRUCTURE OF THE BIFUNCTIONAL KINASE- METHYLTRANSFERASE WBDD  |   TRANSFERASE, KINASE, METHYLTRANSFERASE 
1zy5:B   (GLY611) to   (GLY830)  CRYSTAL STRUCTURE OF EIF2ALPHA PROTEIN KINASE GCN2: R794G HYPERACTIVATING MUTANT COMPLEXED WITH AMPPNP.  |   TRANSLATION REGULATOR, PROTEIN KINASE, SIGNAL TRANSDUCTION, AMINO-ACID STARVATION, STARVATION STRESS RESPONSE, EIF2ALPHA KINASE, TRANSFERASE 
3ats:A    (ARG70) to   (SER178)  CRYSTAL STRUCTURE OF RV3168  |   HYPOTHETICAL PROTEIN, PUTATIVE AMINOGLYCOSIDE PHOSPHORTRANSFERASE, TRANSFERASE 
1zz2:A    (GLY36) to   (ASP145)  TWO CLASSES OF P38ALPHA MAP KINASE INHIBITORS HAVING A COMMON DIPHENYLETHER CORE BUT EXHIBITING DIVERGENT BINDING MODES  |   PROTEIN-INHIBITOR COMPLEX, TRANSFERASE 
1zzl:A    (ASP88) to   (LEU217)  CRYSTAL STRUCTURE OF P38 WITH TRIAZOLOPYRIDINE  |   PHOSPHORYLATION,SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
4azt:A   (SER240) to   (GLY346)  CO-CRYSTAL STRUCTURE OF WBDD AND KINASE INHIBITOR LY294002.  |   TRANSFERASE 
2a27:B    (ALA25) to   (LYS134)  HUMAN DRP-1 KINASE, W305S S308A D40 MUTANT, CRYSTAL FORM WITH 8 MONOMERS IN THE ASYMMETRIC UNIT  |   PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE 
5e8y:A   (ALA256) to   (SER363)  TGF-BETA RECEPTOR TYPE 2 KINASE DOMAIN (E431A,R433A,E485A,K488A,R493A, R495A) IN COMPLEX WITH STAUROSPORINE  |   KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2a2a:C    (PHE24) to   (LYS134)  HIGH-RESOLUTION CRYSTALLOGRAPHIC ANALYSIS OF THE AUTOINHIBITED CONFORMATION OF A HUMAN DEATH-ASSOCIATED PROTEIN KINASE  |   PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE 
5eak:B    (ALA65) to   (PHE170)  OPTIMIZATION OF MICROTUBULE AFFINITY REGULATING KINASE (MARK) INHIBITORS WITH IMPROVED PHYSICAL PROPERTIES  |   CATALYTIC DOMAIN, PROTEIN-SERINE-THREONINE KINASES, KINASE INHIBITOR, SERINE-THREONINE KINASES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3m42:A    (LEU79) to   (ASN181)  CRYSTAL STRUCTURE OF MAPKAP KINASE 2 (MK2) COMPLEXED WITH A TETRACYCLIC ATP SITE INHIBITOR  |   SMALL MOLECULE INHIBITOR, ATP-SITE KINASE INHIBITOR, NOVARTIS-PRODUCT NVP-BMA086, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
4b9d:A    (LYS17) to   (LYS123)  CRYSTAL STRUCTURE OF HUMAN NIMA-RELATED KINASE 1 (NEK1) WITH INHIBITOR.  |   TRANSFERASE, INHIBITOR 
4b9d:B    (LYS17) to   (LYS123)  CRYSTAL STRUCTURE OF HUMAN NIMA-RELATED KINASE 1 (NEK1) WITH INHIBITOR.  |   TRANSFERASE, INHIBITOR 
5ei6:A   (SER537) to   (GLY642)  RAPID DISCOVERY OF PYRIDO[3,4-D]PYRIMIDINE INHIBITORS OF MONOPOLAR SPINDLE KINASE 1 (MPS1) USING A STRUCTURE-BASED HYDRIDIZATION APPROACH  |   SPINDLE ASSEMBLY CHECKPOINT (SAC), ONCOLOGY TARGET PYRIDO[3, 4- D]PYRIMIDINE BASED INHIBITORS SELECTIVE AGAINST MPS1, TRANSFERASE 
4bbe:A   (PHE860) to   (ARG971)  AMINOALKYLPYRIMIDINE INHIBITOR COMPLEXES WITH JAK2  |   TRANSFERASE, INHIBITOR 
4bbe:B   (GLY861) to   (ARG971)  AMINOALKYLPYRIMIDINE INHIBITOR COMPLEXES WITH JAK2  |   TRANSFERASE, INHIBITOR 
4bbe:C   (GLY861) to   (ARG971)  AMINOALKYLPYRIMIDINE INHIBITOR COMPLEXES WITH JAK2  |   TRANSFERASE, INHIBITOR 
4bbe:D   (GLY861) to   (ARG971)  AMINOALKYLPYRIMIDINE INHIBITOR COMPLEXES WITH JAK2  |   TRANSFERASE, INHIBITOR 
3mdy:C   (GLY216) to   (THR317)  CRYSTAL STRUCTURE OF THE CYTOPLASMIC DOMAIN OF THE BONE MORPHOGENETIC PROTEIN RECEPTOR TYPE-1B (BMPR1B) IN COMPLEX WITH FKBP12 AND LDN- 193189  |   COMPLEX (ISOMERASE-PROTEIN KINASE), RECEPTOR SERINE/THREONINE KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, DISEASE MUTATION, KINASE, TRANSFERASE, ROTAMASE, TRANSFERASE-ISOMERASE COMPLEX 
3mes:B    (GLN85) to   (ILE181)  CRYSTAL STRUCTURE OF CHOLINE KINASE FROM CRYPTOSPORIDIUM PARVUM IOWA II, CGD3_2030  |   CHOLINE KINASE, MALARIA, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE 
4bcj:A    (GLU32) to   (LYS144)  STRUCTURE OF CDK9 IN COMPLEX WITH CYCLIN T AND A 2-AMINO-4- HETEROARYL-PYRIMIDINE INHIBITOR  |   TRANSFERASE-CELL CYCLE COMPLEX, CDK-CYCLIN COMPLEX, TRANSCRIPTION-PROTEIN BINDING, STRUCTURE-BASED DRUG DESIGN 
4qpm:A   (ALA799) to   (GLU912)  STRUCTURE OF BUB1 KINASE DOMAIN  |   TRANSFERASE 
4qpm:B   (ALA799) to   (GLU912)  STRUCTURE OF BUB1 KINASE DOMAIN  |   TRANSFERASE 
3bea:A   (ALA599) to   (ASN773)  CFMS TYROSINE KINASE (TIE2 KID) IN COMPLEX WITH A PYRIMIDINOPYRIDONE INHIBITOR  |   KINASE DOMAIN, INHIBITOR, TRANSFERASE, JUXTAMEMBRANE DOMAIN, ATP-BINDING, GLYCOPROTEIN, IMMUNOGLOBULIN DOMAIN, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO- ONCOGENE, RECEPTOR, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
5eqy:A   (SER121) to   (GLY237)  CRYSTAL STRUCTURE OF CHOLINE KINASE ALPHA-1 BOUND BY 5-[(4-METHYL-1,4- DIAZEPAN-1-YL)METHYL]-2-[4-[(4-METHYL-1,4-DIAZEPAN-1-YL) METHYL]PHENYL]BENZENECARBONITRILE (COMPOUND 65)  |   KINASE, INHIBITOR, DRUG TARGET, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4bhz:A   (SER537) to   (GLY642)  SCAFFOLD FOCUSED VIRTUAL SCREENING: PROSPECTIVE APPLICATION TO THE DISCOVERY OF TTK INHIBITOR  |   TRANSFERASE, MITOSIS 
4bi1:A   (GLN541) to   (GLY642)  SCAFFOLD FOCUSED VIRTUAL SCREENING: PROSPECTIVE APPLICATION TO THE DISCOVERY OF TTK INHIBITOR  |   TRANSFERASE, PROTEIN KINASE, MITOSIS 
3mpm:A   (MET261) to   (LEU336)  LCK COMPLEXED WITH A PYRAZOLOPYRIMIDINE  |   KINASE DOMAIN, TRANSFERASE 
4bky:A    (ALA23) to   (VAL112)  CRYSTAL STRUCTURE OF UNPHOSPHORYLATED MATERNAL EMBRYONIC LEUCINE ZIPPER KINASE (MELK) IN COMPLEX WITH PYRROLOPYRAZOLE INHIBITOR  |   TRANSFERASE 
4bkz:A    (LYS24) to   (VAL112)  CRYSTAL STRUCTURE OF UNPHOSPHORYLATED MATERNAL EMBRYONIC LEUCINE ZIPPER KINASE (MELK) IN COMPLEX WITH A BENZODIPYRAZOLE INHIBITOR  |   TRANSFERASE 
4bl1:A    (ALA23) to   (VAL112)  CRYSTAL STRUCTURE OF UNPHOSPHORYLATED MATERNAL EMBRYONIC LEUCINE ZIPPER KINASE (MELK) IN COMPLEX WITH AMP-PNP  |   TRANSFERASE 
3mtf:B   (GLY220) to   (HIS320)  CRYSTAL STRUCTURE OF THE ACVR1 KINASE IN COMPLEX WITH A 2- AMINOPYRIDINE INHIBITOR  |   PROTEIN KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3bpr:A   (GLY604) to   (ASN718)  CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE- PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR C52  |   ATP-BINDING, DISEASE MUTATION, GLYCOPROTEIN, KINASE, NUCLEOTIDE- BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, RECEPTOR, RETINITIS PIGMENTOSA, SENSORY TRANSDUCTION, TRANSFERASE, TYROSINE-PROTEIN KINASE, VISION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, IMMUNOGLOBULIN DOMAIN, MEMBRANE, PHOSPHOPROTEIN, POLYMORPHISM, TRANSMEMBRANE 
3bpr:B   (GLY604) to   (ASN718)  CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE- PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR C52  |   ATP-BINDING, DISEASE MUTATION, GLYCOPROTEIN, KINASE, NUCLEOTIDE- BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, RECEPTOR, RETINITIS PIGMENTOSA, SENSORY TRANSDUCTION, TRANSFERASE, TYROSINE-PROTEIN KINASE, VISION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, IMMUNOGLOBULIN DOMAIN, MEMBRANE, PHOSPHOPROTEIN, POLYMORPHISM, TRANSMEMBRANE 
3bpr:C   (GLY604) to   (ASN718)  CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE- PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR C52  |   ATP-BINDING, DISEASE MUTATION, GLYCOPROTEIN, KINASE, NUCLEOTIDE- BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, RECEPTOR, RETINITIS PIGMENTOSA, SENSORY TRANSDUCTION, TRANSFERASE, TYROSINE-PROTEIN KINASE, VISION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, IMMUNOGLOBULIN DOMAIN, MEMBRANE, PHOSPHOPROTEIN, POLYMORPHISM, TRANSMEMBRANE 
3brb:A   (GLY604) to   (ASN718)  CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE- PROTEIN KINASE MER IN COMPLEX WITH ADP  |   ATP-BINDING, DISEASE MUTATION, GLYCOPROTEIN, KINASE, NUCLEOTIDE- BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, RECEPTOR, RETINITIS PIGMENTOSA, SENSORY TRANSDUCTION, TRANSFERASE, TYROSINE-PROTEIN KINASE, VISION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, IMMUNOGLOBULIN DOMAIN, MEMBRANE, PHOSPHOPROTEIN, TRANSMEMBRANE 
3brb:B   (GLY604) to   (ASN718)  CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE- PROTEIN KINASE MER IN COMPLEX WITH ADP  |   ATP-BINDING, DISEASE MUTATION, GLYCOPROTEIN, KINASE, NUCLEOTIDE- BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, RECEPTOR, RETINITIS PIGMENTOSA, SENSORY TRANSDUCTION, TRANSFERASE, TYROSINE-PROTEIN KINASE, VISION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, IMMUNOGLOBULIN DOMAIN, MEMBRANE, PHOSPHOPROTEIN, TRANSMEMBRANE 
3mwu:A    (GLY88) to   (ILE178)  ACTIVATED CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM CRYPTOSPORIDIUM PARVUM (CPCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR RM-1-95  |   SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, BUMPED KINASE INHIBITOR, BKI, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3my0:A   (GLY214) to   (HIS314)  CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3my0:B   (GLY214) to   (HIS314)  CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3my0:D   (GLY214) to   (HIS314)  CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3my0:E   (GLY214) to   (HIS314)  CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3my0:F   (GLY214) to   (HIS314)  CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3my0:G   (GLY214) to   (HIS314)  CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3my0:H   (GLY214) to   (HIS314)  CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3my0:M   (GLY214) to   (HIS314)  CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3my0:Q   (GLY214) to   (HIS314)  CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3my0:R   (GLY214) to   (HIS314)  CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3my0:T   (GLY214) to   (HIS314)  CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3my0:V   (GLY214) to   (HIS314)  CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3my0:W   (GLY214) to   (HIS314)  CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3my0:X   (GLY214) to   (HIS314)  CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189  |   PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE 
3bv3:A    (GLY36) to   (ASP145)  MORPHOLINO PYRROLOTRIAZINE P38 ALPHA MAP KINASE INHIBITOR COMPOUND 2  |   SERINE/THREONINE-PROTEIN KINASE, KINASE, TRANSFERASE, P38 MAP KINASE, ALTERNATIVE SPLICING, ATP-BINDING, CYTOPLASM, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN 
4br3:B   (LEU124) to   (GLY237)  DETERMINATION OF POTENTIAL SCAFFOLDS FOR HUMAN CHOLINE KINASE ALPHA 1 BY CHEMICAL DECONVOLUTION STUDIES  |   TRANSFERASE 
5f94:B    (GLY68) to   (GLY176)  CRYSTAL STRUCTURE OF GSK3B IN COMPLEX WITH COMPOUND 15: 2- [(CYCLOPROPYLCARBONYL)AMINO]-N-(4-METHOXYPYRIDIN-3-YL)PYRIDINE-4- CARBOXAMIDE  |   GSK3B, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3bym:A   (PHE256) to   (LEU336)  X-RAY CO-CRYSTAL STRUCTURE AMINOBENZIMIDAZOLE TRIAZINE 1 BOUND TO LCK  |   LCK, KINASE DOMAIN, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE 
3byo:A   (PHE256) to   (LEU336)  X-RAY CO-CRYSTAL STRUCTURE OF 2-AMINO-6-PHENYLPYRIMIDO[5', 4':5,6]PYRIMIDO[1,2-A]BENZIMIDAZOL-5(6H)-ONE 25 BOUND TO LCK  |   LCK, KINASE DOMAIN, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE 
3bys:A   (PHE256) to   (LEU336)  CO-CRYSTAL STRUCTURE OF LCK AND AMINOPYRIMIDINE AMIDE 10B  |   LCK, KINASE DOMAIN, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE 
3byu:A   (PHE256) to   (LEU336)  CO-CRYSTAL STRUCTURE OF LCK AND AMINOPYRIMIDINE REVERSE AMIDE 23  |   LCK, KINASE DOMAIN, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE 
3n4t:A    (ILE35) to   (ILE133)  APO APH(2")-IVA FORM I  |   AMINOGLYCOSIDE, PHOSPHOTRANSFERASE, RESISTANCE, UNKNOWN FUNCTION 
5fd2:B   (THR470) to   (GLU545)  B-RAF WILD-TYPE KINASE DOMAIN IN COMPLEX WITH A PURINYLPYRIDINYLAMINO- BASED INHIBITOR  |   PHOSPHOTRANSFERASE, INHIBITOR, MELANOMA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3c4c:A   (GLY469) to   (GLU545)  B-RAF KINASE IN COMPLEX WITH PLX4720  |   B-RAF, BRAF, RAF, PROTO-ONCOGENE, SERINE/THREONINE KINASE, ATP-BINDING, CARDIOMYOPATHY, CYTOPLASM, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ZINC, ZINC-FINGER 
4r7h:A   (ALA599) to   (LEU687)  CRYSTAL STRUCTURE OF FMS KINASE DOMAIN WITH A SMALL MOLECULAR INHIBITOR, PLX3397  |   CSF-1-R, FMS PROTO-ONCOGENE, C-FMS, CD115 ANTIGEN, KINASE, ATP- BINDING, PLX3397, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4r8q:A   (ALA799) to   (GLU912)  STRUCTURE AND SUBSTRATE RECRUITMENT OF THE HUMAN SPINDLE CHECKPOINT KINASE BUB1  |   SPINDLE ASSEMBLY CHECKPOINT, MITOSIS, KINASE, ACTIVATION, KEN BOX, CDC20, ATP-BINDING, CELL CYCLE, CELL DIVISION, DISEASE MUTATION, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE 
3ce3:A  (GLY1095) to  (LYS1199)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF THE HEPATOCYTE GROWTH FACTOR RECEPTOR C-MET IN COMPLEX WITH A PYRROLOPYRIDINEPYRIDONE BASED INHIBITOR  |   RECEPTOR TYROSINE KINASE, SIGNAL TRANSDUCTION, GRB2, SHC, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE 
3ncg:A    (GLY88) to   (ILE178)  ACTIVATED CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM CRYPTOSPORIDIUM PARVUM (CPCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR NM-PP1  |   SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, BUMPED KINASE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP 
4c3f:A   (MET261) to   (LEU336)  STRUCTURE OF LCK IN COMPLEX WITH A COMPOUND DISCOVERED BY VIRTUAL FRAGMENT LINKING  |   TRANSFERASE 
4rfm:A   (LEU376) to   (SER477)  ITK KINASE DOMAIN IN COMPLEX WITH COMPOUND 1 N-{1-[(1,1-DIOXO-1-THIAN- 2-YL)(PHENYL)METHYL]-1H- PYRAZOL-4-YL}-5,5-DIFLUORO-5A-METHYL-1H,4H, 4AH,5H,5AH,6H-CYCLOPROPA[F]INDAZOLE-3-CARBOXAMIDE  |   KINASE, TRANSFERASE-INHIBITOR COMPLEX 
4c4g:A   (SER537) to   (GLY642)  STRUCTURE-BASED DESIGN OF ORALLY BIOAVAILABLE PYRROLOPYRIDINE INHIBITORS OF THE MITOTIC KINASE MPS1  |   TRANSFERASE, PROTEIN KINASE, MITOSIS, STRUCTURE-BASED DESIGN 
4c58:A    (ALA52) to   (GLN165)  STRUCTURE OF GAK KINASE IN COMPLEX WITH NANOBODY (NBGAK_4)  |   TRANSFERASE, KINASE, CONFORMATIONAL PLASTICITY, ACTIVATION 
4c59:A    (ALA52) to   (ARG164)  STRUCTURE OF GAK KINASE IN COMPLEX WITH NANOBODY (NBGAK_4)  |   TRANSFERASE, KINASE, CONFORMATIONAL PLASTICITY, ACTIVATION 
4rix:D   (GLY705) to   (ASN784)  CRYSTAL STRUCTURE OF AN EGFR/HER3 KINASE DOMAIN HETERODIMER CONTAINING THE CANCER-ASSOCIATED HER3-Q790R MUTATION  |   RECEPTOR TYROSINE KINASE, PSEUDOKINASE, KINASE, ATP BINDING, MEMBRANE, TRANSFERASE 
4rmz:B   (GLY198) to   (HIS306)  CRYSTAL STRUCTURE OF IRAK-4  |   SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3cr0:A   (SER312) to   (SER421)  WEE1 KINASE COMPLEX WITH INHIBITOR PD259_809  |   KINASE DOMAIN, INHIBITOR COMPLEX, TRANSFERASE 
4cg9:A   (LEU124) to   (GLY237)  HUMAN CHOLINE KINASE A1 IN COMPLEX WITH COMPOUND 12  |   TRANSFERASE, CANCER, DRUG TARGET, BISCATIONIC COMPOUNDS 
3cs9:C   (GLU255) to   (ASN336)  HUMAN ABL KINASE IN COMPLEX WITH NILOTINIB  |   NILOTINIB, AMN107, KINASE, ABL, ALTERNATIVE SPLICING, ATP- BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, ABL KINASE WT IN COMPLEX WITH NVP-AMN107 
3nw5:A   (PRO996) to  (LYS1100)  CRYSTAL STRUCTURE OF INSULIN-LIKE GROWTH FACTOR 1 RECEPTOR (IGF-1R-WT) COMPLEX WITH A CARBON-LINKED PROLINE ISOSTERE INHIBITOR (11B)  |   HORMONE/GROWTH FACTOR, IGF-1R, KINASE DOMAIN, TRANSFERASE 
3nw6:A   (PRO996) to  (LYS1100)  CRYSTAL STRUCTURE OF INSULIN-LIKE GROWTH FACTOR 1 RECEPTOR (IGF-1R-WT) COMPLEX WITH A CARBON-LINKED PROLINE ISOSTERE INHIBITOR (11A)  |   HORMONE/GROWTH FACTOR, IGF-1R, KINASE DOMAIN, TRANSFERASE 
3nw7:A   (PRO996) to  (LYS1100)  CRYSTAL STRUCTURE OF INSULIN-LIKE GROWTH FACTOR 1 RECEPTOR (IGF-1R-WT) COMPLEX WITH A CARBON-LINKED PROLINE ISOSTERE INHIBITOR (34)  |   HORMONE/GROWTH FACTOR, IGF-1R, KINASE DOMAIN, TRANSFERASE 
3nyv:A    (GLY63) to   (LYS169)  CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH NON-SPECIFIC INHIBITOR WHI-P180  |   SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3o2m:A    (GLY38) to   (GLY146)  CRYSTAL STRUCTURE OF JNK1-ALPHA1 ISOFORM COMPLEX WITH A BIARYL TETRAZOL (A-82118)  |   SERINE THREONINE PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, KINASE-INHIBITOR COMPLEX, TRANSFERASE-INHIBITOR COMPLEX 
4cqg:A    (ALA23) to   (VAL112)  THE CRYSTAL STRUCTURE OF MPK38 IN COMPLEX WITH OTSSP167, AN ORALLY-ADMINISTRATIVE MELK SELECTIVE INHIBITOR  |   TRANSFERASE 
3d7t:A   (GLY207) to   (ASN309)  STRUCTURAL BASIS FOR THE RECOGNITION OF C-SRC BY ITS INACTIVATOR CSK  |   CSK SRC TYROSINE KINASE, ATP-BINDING, CYTOPLASM, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, ALTERNATIVE SPLICING, LIPOPROTEIN, MYRISTATE, PROTO- ONCOGENE 
3d7t:B   (GLU280) to   (LEU358)  STRUCTURAL BASIS FOR THE RECOGNITION OF C-SRC BY ITS INACTIVATOR CSK  |   CSK SRC TYROSINE KINASE, ATP-BINDING, CYTOPLASM, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, ALTERNATIVE SPLICING, LIPOPROTEIN, MYRISTATE, PROTO- ONCOGENE 
3d7u:A   (GLY207) to   (ASN309)  STRUCTURAL BASIS FOR THE RECOGNITION OF C-SRC BY ITS INACTIVATOR CSK  |   CSK C-SRC TYROSINE KINASE, ATP-BINDING, KINASE, MEMBRANE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, LIPOPROTEIN, MYRISTATE, PROTO-ONCOGENE 
3d7u:B   (GLY284) to   (TYR357)  STRUCTURAL BASIS FOR THE RECOGNITION OF C-SRC BY ITS INACTIVATOR CSK  |   CSK C-SRC TYROSINE KINASE, ATP-BINDING, KINASE, MEMBRANE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, LIPOPROTEIN, MYRISTATE, PROTO-ONCOGENE 
3d7u:C   (GLY207) to   (ASN309)  STRUCTURAL BASIS FOR THE RECOGNITION OF C-SRC BY ITS INACTIVATOR CSK  |   CSK C-SRC TYROSINE KINASE, ATP-BINDING, KINASE, MEMBRANE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, LIPOPROTEIN, MYRISTATE, PROTO-ONCOGENE 
3d7u:D   (GLY284) to   (TYR357)  STRUCTURAL BASIS FOR THE RECOGNITION OF C-SRC BY ITS INACTIVATOR CSK  |   CSK C-SRC TYROSINE KINASE, ATP-BINDING, KINASE, MEMBRANE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, LIPOPROTEIN, MYRISTATE, PROTO-ONCOGENE 
4cva:A   (SER536) to   (ALA634)  MPS1 KINASE WITH 3-AMINOPYRIDIN-2-ONE INHIBITORS  |   TRANSFERASE, FRAGMENT, INHIBITOR 
4tn6:B    (GLY21) to   (ASN123)  CK1D IN COMPLEX WITH INHIBITOR  |   SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3dak:A    (ALA29) to   (GLY116)  CRYSTAL STRUCTURE OF DOMAIN-SWAPPED OSR1 KINASE DOMAIN  |   SERINE/THREONINE PROTEIN KINASE, STE20, DOMAIN-SWAPPING, ATP-BINDING, KINASE, MAGNESIUM, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE 
3dak:D    (THR28) to   (GLY116)  CRYSTAL STRUCTURE OF DOMAIN-SWAPPED OSR1 KINASE DOMAIN  |   SERINE/THREONINE PROTEIN KINASE, STE20, DOMAIN-SWAPPING, ATP-BINDING, KINASE, MAGNESIUM, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE 
3od6:X    (SER37) to   (ASP145)  CRYSTAL STRUCTURE OF P38ALPHA Y323T ACTIVE MUTANT  |   MAP KINASE, P38, TCR INDUCED ACTIVATION, TYR-323 PHOSPHORYLATION, KINASE FOLD, KINASE, PHOSPHORYLAITON, TRANSFERASE 
3dbq:A   (SER536) to   (ALA634)  CRYSTAL STRUCTURE OF TTK KINASE DOMAIN  |   MPS1 STRUCTURE, KINASE ACTIVATION, PHOSPHORYLATION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3oez:A   (GLY279) to   (LEU358)  CRYSTAL STRUCTURE OF THE L317I MUTANT OF THE CHICKEN C-SRC TYROSINE KINASE DOMAIN COMPLEXED WITH IMATINIB  |   C-SRC L317I MUTANT, TYROSINE KINASE, IMATINIB, TRANSFERASE 
4d28:C    (PHE22) to   (GLY129)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF SNRK3.11 AT5G35410  |   TRANSFERASE, SALT STRESS, SODIUM TRANSPORT, ION HOMEOSTASIS 
3dk3:A   (GLY254) to   (SER336)  CRYSTAL STRUCTURE OF MUTANT ABL KINASE DOMAIN IN COMPLEX WITH SMALL MOLECULE FRAGMENT  |   DRUG DISCOVERY, ABL KINASE, FRAGMENT BASED, ALTERNATIVE SPLICING, ATP-BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
3dk3:B   (GLU258) to   (SER336)  CRYSTAL STRUCTURE OF MUTANT ABL KINASE DOMAIN IN COMPLEX WITH SMALL MOLECULE FRAGMENT  |   DRUG DISCOVERY, ABL KINASE, FRAGMENT BASED, ALTERNATIVE SPLICING, ATP-BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
3dk6:A   (GLY254) to   (SER336)  CRYSTAL STRUCTURE OF MUTANT ABL KINASE DOMAIN IN COMPLEX WITH SMALL MOLECULE FRAGMENT  |   DRUG DISCOVERY, ABL KINASE, FRAGMENT BASED, ALTERNATIVE SPLICING, ATP-BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
3dk6:B   (GLU255) to   (SER336)  CRYSTAL STRUCTURE OF MUTANT ABL KINASE DOMAIN IN COMPLEX WITH SMALL MOLECULE FRAGMENT  |   DRUG DISCOVERY, ABL KINASE, FRAGMENT BASED, ALTERNATIVE SPLICING, ATP-BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
4d2r:A  (PRO1026) to  (LYS1130)  HUMAN IGF IN COMPLEX WITH A DYRK1B INHIBITOR  |   TRANSFERASE, KINASE, INHIBITOR, ONCOLOGY 
4d2s:A   (SER537) to   (GLY642)  HUMAN TTK IN COMPLEX WITH A DYRK1B INHIBITOR  |   TRANSFERASE, ONCOLOGY 
4d2v:B    (PHE22) to   (VAL112)  STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS  |   TRANSFERASE, FRAGMENT BASED DRUG DESIGN 
4tw9:A    (GLY21) to   (ASN123)  DIFLUORO-DIOXOLO-BENZOIMIDAZOL-BENZAMIDES AS POTENT INHIBITORS OF CK1DELTA AND EPSILON WITH NANOMOLAR INHIBITORY ACTIVITY ON CANCER CELL PROLIFERATION  |   TRANSFERASE, CK1DELTA, CK1EPSILON, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR 
3oom:A   (GLY220) to   (ILE321)  CRYSTAL STRUCTURE OF THE ACVR1 KINASE DOMAIN IN COMPLEX WITH THE IMIDAZO[1,2-B]PYRIDAZINE INHIBITOR K00507  |   PROTEIN KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4d9t:A   (SER434) to   (GLY534)  RSK2 C-TERMINAL KINASE DOMAIN WITH INHIBITOR (E)-METHYL 3-(4-AMINO-7- (3-HYDROXYPROPYL)-5-P-TOLYL-7H-PYRROLO[2,3-D]PYRIMIDIN-6-YL)-2- CYANOACRYLATE  |   KINASE, INHIBITOR, REVERSIBLE, THIOL, PHOSPHORYLATION, MIGRATION,, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4dbn:A   (GLY468) to   (GLU544)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN B-RAF WITH A [1, 3]THIAZOLO[5,4-B]PYRIDINE DERIVATIVE  |   KINASE DRUG COMPLEX, SER/THR KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4dbn:B   (LYS472) to   (GLU544)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN B-RAF WITH A [1, 3]THIAZOLO[5,4-B]PYRIDINE DERIVATIVE  |   KINASE DRUG COMPLEX, SER/THR KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3otv:D    (GLN45) to   (GLY145)  CRYSTAL STRUCTURE OF THE INTRACELLULAR DOMAIN OF RV3910 FROM MYCOBACTERIUM TUBERCULOSIS  |   PEPTIDOGLYCAN, SER/THR KINASE, PSEUDOKINASE, REGULATION, MEMBRANE, TRANSFERASE 
3oun:B    (GLN45) to   (GLY145)  CRYSTAL STRUCTURE OF THE FHAA FHA DOMAIN COMPLEXED WITH THE INTRACELLULAR DOMAIN OF RV3910  |   PEPTIDOGLYCAN, SER/THR KINASE, PSEUDOKINASE, FHA DOMAIN, REGULATION, PHOSPHORYLATION, MEMBRANE ASSOCIATED INTRACELLULAR, PROTEIN BINDING- TRANSFERASE COMPLEX 
4u40:A    (GLN38) to   (HIS148)  MITOGEN-ACTIVATED PROTEIN KINASE KINASE KINASE KINASE 4 (MAP4K4) BOUND TO AMPPNP  |   KINASE, TRANSFERASE 
4u43:A    (GLY37) to   (HIS148)  MAP4K4 IN COMPLEX WITH INHIBITOR (COMPOUND 6)  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4u45:A    (GLY37) to   (HIS148)  MAP4K4 IN COMPLEX WITH INHIBITOR (COMPOUND 25)  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4deg:A  (GLY1090) to  (LYS1199)  CRYSTAL STRUCTURE OF C-MET IN COMPLEX WITH TRIAZOLOPYRIDAZINE INHIBITOR 2  |   PROTO-ONCOGENE, RECEPTOR TYROSINE KINASE, RTK, ATP-BINDING, HEPATOCYTE GROWTH FACTOR/SCATTER FACTOR, HGF/SF, PHOSPHOPROTEIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3oxi:A    (GLY76) to   (GLY184)  DESIGN AND SYNTHESIS OF DISUBSTITUTED THIOPHENE AND THIAZOLE BASED INHIBITORS OF JNK FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES  |   JNK INHIBITORS, NEURODEGENERATIVE DISEASES, KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3oy3:A   (GLU255) to   (SER336)  CRYSTAL STRUCTURE OF ABL T315I MUTANT KINASE DOMAIN BOUND WITH A DFG- OUT INHIBITOR AP24589  |   PROTEIN-INHIBITOR COMPLEX, PROTEIN KINASE TWO-DOMAIN FOLD, PHOSPHOTRANSFERASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3oy3:B   (GLU255) to   (SER336)  CRYSTAL STRUCTURE OF ABL T315I MUTANT KINASE DOMAIN BOUND WITH A DFG- OUT INHIBITOR AP24589  |   PROTEIN-INHIBITOR COMPLEX, PROTEIN KINASE TWO-DOMAIN FOLD, PHOSPHOTRANSFERASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
5hie:A   (THR470) to   (GLU545)  BRAF KINASE DOMAIN B3AC LOOP DELETION MUTANT IN COMPLEX WITH DABRAFENIB  |   TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5hie:C   (THR470) to   (GLU545)  BRAF KINASE DOMAIN B3AC LOOP DELETION MUTANT IN COMPLEX WITH DABRAFENIB  |   TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5hie:D   (THR470) to   (GLU545)  BRAF KINASE DOMAIN B3AC LOOP DELETION MUTANT IN COMPLEX WITH DABRAFENIB  |   TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3p7a:A    (GLY36) to   (ASP145)  P38 INHIBITOR-BOUND  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5hu9:A   (GLU258) to   (ASN336)  CRYSTAL STRUCTURE OF ABL1 IN COMPLEX WITH CHMFL-074  |   ABL, BCR-ABL, CHMFL-074, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4dt8:B    (ILE35) to   (ILE133)  CRYSTAL STRUCTURE OF AMINOGLYCOSIDE-2''-PHOSPHOTRANSFERASE TYPE IVA IN COMPLEX WITH ADENOSINE  |   AMINOGLYCOSIDE KINASE, TRANSFERASE 
4dt9:A    (ILE35) to   (ILE133)  CRYSTAL STRUCTURE OF AMINOGLYCOSIDE-2''-PHOSPHOTRANSFERASE TYPE IVA IN COMPLEX WITH GUANOSINE  |   AMINOGLYCOSIDE KINASE, TRANSFERASE 
5hzn:A  (PRO1023) to  (LYS1127)  STRUCTURE OF NVP-AEW541 IN COMPLEX WITH IGF-1R KINASE  |   INHIBITOR, KINASE, TRANSFERASE 
5hzn:D  (PRO1023) to  (LYS1127)  STRUCTURE OF NVP-AEW541 IN COMPLEX WITH IGF-1R KINASE  |   INHIBITOR, KINASE, TRANSFERASE 
5hzn:H  (PRO1023) to  (LYS1127)  STRUCTURE OF NVP-AEW541 IN COMPLEX WITH IGF-1R KINASE  |   INHIBITOR, KINASE, TRANSFERASE 
5i3o:A    (SER63) to   (CYS172)  CRYSTAL STRUCTURE OF BMP-2-INDUCIBLE KINASE IN COMPLEX WITH AN INDAZOLE INHIBITOR  |   TRANSFERASE, PROTEIN KINASE DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5i3o:B    (SER63) to   (CYS172)  CRYSTAL STRUCTURE OF BMP-2-INDUCIBLE KINASE IN COMPLEX WITH AN INDAZOLE INHIBITOR  |   TRANSFERASE, PROTEIN KINASE DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5i3r:A    (SER63) to   (CYS172)  CRYSTAL STRUCTURE OF BMP-2-INDUCIBLE KINASE IN COMPLEX WITH AN INDAZOLE INHIBITOR  |   TRANSFERASE, PROTEIN KINASE DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5i3r:B    (SER63) to   (CYS172)  CRYSTAL STRUCTURE OF BMP-2-INDUCIBLE KINASE IN COMPLEX WITH AN INDAZOLE INHIBITOR  |   TRANSFERASE, PROTEIN KINASE DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5i4n:A   (GLY562) to   (THR668)  CRYSTAL STRUCTURE OF THE E596A V617F MUTANT JAK2 PSEUDOKINASE DOMAIN BOUND TO MG-ATP  |   TRANSFERASE, PSEUDOKINASE, ATP BINDING 
4ump:B    (ALA23) to   (VAL112)  STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS  |   TRANSFERASE 
4umt:A    (PHE22) to   (VAL112)  STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS  |   TRANSFERASE, FRAGMENT BASED DRUG DESIGN 
3piz:A   (GLY414) to   (ARG492)  CRYSTAL STRUCTURE OF BTK KINASE DOMAIN COMPLEXED WITH (5-AMINO-1-O- TOLYL-1H-PYRAZOL-4-YL)-[3-(1-METHANESULFONYL-PIPERIDIN-4-YL)-PHENYL]- METHANONE  |   HELIX C-IN, DFG-IN, TRANSFERASE, TRANSFERASE-INHIBITOR COMPLEX 
5i5z:A    (LYS37) to   (TRP146)  CDK8-CYCC IN COMPLEX WITH 8-(1-METHYL-2,2-DIOXO-2,3-DIHYDRO-1H-2L6- BENZO[C]ISOTHIAZOL-5-YL)-[1,6]NAPHTHYRIDINE-2-CARBOXYLIC ACID METHYLAMIDE  |   CDK8 KINASE / CYCLIN C, TRANSFERASE 
4dym:A   (GLY220) to   (HIS320)  CRYSTAL STRUCTURE OF THE ACVR1 KINASE DOMAIN IN COMPLEX WITH THE IMIDAZO[1,2-B]PYRIDAZINE INHIBITOR K00135  |   STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4e26:A   (LYS473) to   (SER571)  BRAF IN COMPLEX WITH AN ORGANIC INHIBITOR 7898734  |   KINASE, INHIBITOR, ONCOPROTEIN, MELANOMA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4e26:B   (GLY469) to   (GLU545)  BRAF IN COMPLEX WITH AN ORGANIC INHIBITOR 7898734  |   KINASE, INHIBITOR, ONCOPROTEIN, MELANOMA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ppk:B   (LYS473) to   (GLU545)  HUMAN B-RAF KINASE IN COMPLEX WITH A NON-OXIME FUROPYRIDINE INHIBITOR  |   PROTEIN KINASE, B-RAF ATP-COMPETITIVE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3ppz:A   (GLY563) to   (ASP647)  CRYSTAL STRUCTURE OF CTR1 KINASE DOMAIN IN COMPLEX WITH STAUROSPORINE  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE 
3ppz:B   (THR564) to   (ASN667)  CRYSTAL STRUCTURE OF CTR1 KINASE DOMAIN IN COMPLEX WITH STAUROSPORINE  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE 
4e4m:A   (GLY861) to   (ARG971)  JAK2 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 30  |   O-PHOSPHOTYROSINE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4e4m:D   (SER862) to   (THR969)  JAK2 KINASE (JH1 DOMAIN) IN COMPLEX WITH COMPOUND 30  |   O-PHOSPHOTYROSINE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4e4x:A   (THR470) to   (GLU545)  CRYSTAL STRUCTURE OF B-RAF KINASE DOMAIN IN COMPLEX WITH A DIHYDROPYRIDO[2,3-D]PYRIMIDINONE-BASED INHIBITOR  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4e4x:B   (LYS473) to   (GLU545)  CRYSTAL STRUCTURE OF B-RAF KINASE DOMAIN IN COMPLEX WITH A DIHYDROPYRIDO[2,3-D]PYRIMIDINONE-BASED INHIBITOR  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3prf:A   (LYS473) to   (GLU545)  CRYSTAL STRUCTURE OF HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH A NON- OXIME FUROPYRIDINE INHIBITOR  |   PROTEIN KINASE, ATP-COMPETITIVE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3prf:B   (LYS473) to   (GLU545)  CRYSTAL STRUCTURE OF HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH A NON- OXIME FUROPYRIDINE INHIBITOR  |   PROTEIN KINASE, ATP-COMPETITIVE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5ih5:A    (ASP22) to   (ASN123)  HUMAN CASEIN KINASE 1 ISOFORM DELTA (KINASE DOMAIN) IN COMPLEX WITH EPIBLASTIN A  |   KINASE DOMAIN, STEM CELL REPROGRAMMING, KINASE INHIBITOR COMPLEX, TRANSFERASE 
5ih6:A    (ASP22) to   (SER121)  HUMAN CASEIN KINASE 1 ISOFORM DELTA (KINASE DOMAIN) IN COMPLEX WITH EPIBLASTIN A DERIVATIVE  |   KINASE DOMAIN, STEM CELL REPROGRAMMING, KINASE INHIBITOR COMPLEX, TRANSFERASE 
5iha:A    (ALA23) to   (VAL112)  MELK IN COMPLEX WITH NVS-MELK8F  |   KINASE UBA DOMAIN INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5ihc:A    (ALA23) to   (VAL112)  MELK IN COMPLEX WITH NVS-MELK12B  |   KINASE UBA DOMAIN INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3psd:A   (THR470) to   (GLU545)  NON-OXIME PYRAZOLE BASED INHIBITORS OF B-RAF KINASE  |   KINASE, ATP-BINDING, CARDIOMYOPATHY, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, ZINC-FINGER, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3psd:B   (GLY469) to   (GLU545)  NON-OXIME PYRAZOLE BASED INHIBITORS OF B-RAF KINASE  |   KINASE, ATP-BINDING, CARDIOMYOPATHY, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, ZINC-FINGER, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
5ikw:A    (SER63) to   (CYS172)  CRYSTAL STRUCTURE OF BMP-2-INDUCIBLE KINASE IN COMPLEX WITH AN INDAZOLE INHIBITOR  |   TRANSFERASE, PROTEIN KINASE DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ehe:A   (LYS473) to   (GLU545)  B-RAF KINASE DOMAIN IN COMPLEX WITH AN AMINOTHIENOPYRIMIDINE-BASED INHIBITOR  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ehe:B   (LYS473) to   (GLU545)  B-RAF KINASE DOMAIN IN COMPLEX WITH AN AMINOTHIENOPYRIMIDINE-BASED INHIBITOR  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ehg:B   (LYS473) to   (GLU545)  B-RAF KINASE DOMAIN IN COMPLEX WITH AN AMINOPYRIDIMINE-BASED INHIBITOR  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ej7:B    (THR39) to   (SER133)  CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, ATP-BOUND  |   CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR 
4ej7:C    (THR39) to   (SER133)  CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, ATP-BOUND  |   CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR 
3pyy:B   (GLU274) to   (ASN355)  DISCOVERY AND CHARACTERIZATION OF A CELL-PERMEABLE, SMALL-MOLECULE C- ABL KINASE ACTIVATOR THAT BINDS TO THE MYRISTOYL BINDING SITE  |   TYROSINE KINASE, TRANSFERASE 
3q2j:A    (LYS30) to   (ILE125)  CRYSTAL STRUCTURE OF 3',5"-AMINOGLYCOSIDE PHOSPHOTRANSFERASE TYPE IIIA PROTEIN KINASE INHIBITOR CKI-7 COMPLEX  |   SER/THR/TYR PROTEIN KINASE, KINASE, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3q2j:B    (LYS30) to   (ILE125)  CRYSTAL STRUCTURE OF 3',5"-AMINOGLYCOSIDE PHOSPHOTRANSFERASE TYPE IIIA PROTEIN KINASE INHIBITOR CKI-7 COMPLEX  |   SER/THR/TYR PROTEIN KINASE, KINASE, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3q4c:B   (THR469) to   (GLU544)  CRYSTAL STRUCTURE OF WILD TYPE BRAF KINASE DOMAIN IN COMPLEX WITH ORGANOMETALLIC INHIBITOR CNS292  |   KINASE, INHIBITOR, ONCOPROTEIN, MELANOMA, KINASE-KINASE INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3q4t:A   (GLY204) to   (GLU305)  CRYSTAL STRUCTURE OF ACTIVIN RECEPTOR TYPE-IIA (ACVR2A) KINASE DOMAIN IN COMPLEX WITH DORSOMORPHIN  |   STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, TRANSFERASE 
3q4u:A   (GLY220) to   (ILE321)  CRYSTAL STRUCTURE OF THE ACVR1 KINASE DOMAIN IN COMPLEX WITH LDN- 193189  |   STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, TRANSFERASE 
3q4u:B   (GLY220) to   (HIS320)  CRYSTAL STRUCTURE OF THE ACVR1 KINASE DOMAIN IN COMPLEX WITH LDN- 193189  |   STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, TRANSFERASE 
3q6w:A  (GLY1095) to  (LYS1199)  STRUCTURE OF DUALLY-PHOSPHORYLATED MET RECEPTOR KINASE IN COMPLEX WITH AN MK-2461 ANALOG WITH SPECIFICITY FOR THE ACTIVATED RECEPTOR  |   TYROSINE KINASE, TWO PHOSPHOTYROSINE RESIUDES, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3q96:A   (GLY469) to   (GLU545)  B-RAF KINASE DOMAIN IN COMPLEX WITH A TETRAHYDRONAPHTHALENE INHIBITOR  |   DESIGN, OPTIMIZATION, POTENT, ORALLY BIOAVAILABLE, TETRAHYDRONAPHTHALENE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4f0i:B   (ALA526) to   (HIS644)  CRYSTAL STRUCTURE OF APO TRKA  |   TYROSINE KINASE, ROSSMANN FOLD, TRANSFERASE 
3qgw:B   (GLY375) to   (PHE454)  CRYSTAL STRUCTURE OF ITK KINASE BOUND TO AN INHIBITOR  |   PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5j5t:A    (GLY28) to   (GLY131)  GLK CO-CRYSTAL STRUCTURE WITH AMINOPYRROLOPYRIMIDINE INHIBITOR  |   PROTEIN KINSAE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4f7l:A    (GLY33) to   (TRP146)  CRYSTAL STRUCTURE OF HUMAN CDK8/CYCC IN COMPLEX WITH COMPOUND 2 (TERT- BUTYL [3-({[3-TERT-BUTYL-1-(4-METHYLPHENYL)-1H-PYRAZOL-5- YL]CARBAMOYL}AMINO)PROPYL]CARBAMATE)  |   PROTEIN KINASE COMPLEX, PROTEROS, TRANSFERASE-TRANSCRIPTION-INHIBITOR COMPLEX 
4uwg:A   (LEU616) to   (TYR707)  DISCOVERY OF (2S)-8-((3R)-3-METHYLMORPHOLIN-4-YL)-1-(3- METHYL-2-OXO-BUTYL)-2-(TRIFLUOROMETHYL)-3,4-DIHYDRO-2H- PYRIMIDO(1,2-A)PYRIMIDIN-6-ONE: A NOVEL POTENT AND SELECTIVE INHIBITOR OF VPS34 FOR THE TREATMENT OF SOLID TUMORS  |   TRANSFERASE 
3qqu:A  (PRO1023) to  (LYS1127)  COCRYSTAL STRUCTURE OF UNPHOSPHORYLATED IGF WITH PYRIMIDINE 8  |   IGF, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qqu:B  (PRO1023) to  (LYS1127)  COCRYSTAL STRUCTURE OF UNPHOSPHORYLATED IGF WITH PYRIMIDINE 8  |   IGF, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qri:B   (GLU255) to   (ASN336)  THE CRYSTAL STRUCTURE OF HUMAN ABL1 KINASE DOMAIN IN COMPLEX WITH DCC- 2036  |   ABL1, KINASE, KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4feu:C    (THR39) to   (SER133)  CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR ANTHRAPYRAZOLONE SP600125  |   ANTHRAPYRAZOLONE, SP600125, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4few:A    (THR39) to   (SER133)  CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR PYRAZOLOPYRIMIDINE PP2  |   PYRAZOLOPYRIMIDINE, PP2, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4few:B    (THR39) to   (PRO135)  CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR PYRAZOLOPYRIMIDINE PP2  |   PYRAZOLOPYRIMIDINE, PP2, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4few:E    (THR39) to   (PRO135)  CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR PYRAZOLOPYRIMIDINE PP2  |   PYRAZOLOPYRIMIDINE, PP2, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fex:E    (THR39) to   (SER133)  CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR TYRPHOSTIN AG1478  |   TYRPHOSTIN, 4-ANILINOQUINAZOLINE, TYRPHOSTIN AG1478, AG1478, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qup:A   (GLY520) to   (ASN640)  INHIBITOR BOUND STRUCTURE OF THE KINASE DOMAIN OF THE MURINE RECEPTOR TYROSINE KINASE TYRO3 (SKY)  |   PROTEIN KINASE INHIBITOR, RECEPTOR TYROSINE KINASE, SPIROCYCLE, KINASE DOMAIN, PHOSPHOTRANSFER, GAS6 LIGAND, CYTOPLASMIC SURFACE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fg7:A    (SER32) to   (GLY136)  CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE I 1-293 IN COMPLEX WITH ATP  |   CAMK, CALMODULIN, AUTOINHIBITION, REGULATION MECHANISM, KINASE, TRANSFERASE 
4w7p:D    (LEU92) to   (SER191)  CRYSTAL STRUCTURE OF ROCK 1 BOUND TO YB-15-QD37  |   INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fku:A    (GLY16) to   (ARG122)  CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH OXINDOLE INHIBITOR  |   ALPHA AND BETA PROTEIN (A+B), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5jeb:A   (VAL714) to   (ASP806)  CRYSTAL STRUCTURE OF EGFR TYROSINE KINASE DOMAIN WITH NOVEL INHIBITOR OF ACTIVE STATE OF HER2  |   INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5jms:A    (GLY63) to   (LYS169)  CRYSTAL STRUCTURE OF TGCDPK1 BOUND TO CGP060476  |   KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, HYDROLASE 
5jn2:A    (GLY63) to   (LYS169)  CRYSTAL STRUCTURE OF TGCDPK1 BOUND TO NVPACU106  |   KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, HYDROLASE 
3rin:A    (ASP88) to   (GLY219)  P38 KINASE CRYSTAL STRUCTURE IN COMPLEX WITH SMALL MOLECULE INHIBITOR  |   P38 MAP KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5jt2:B   (LYS473) to   (GLU545)  BRAFV600E KINASE DOMAIN IN COMPLEX WITH CHEMICALLY LINKED VEMURAFENIB INHIBITOR VEM-BISAMIDE  |   KINASE, DIMER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5jt2:C   (GLY469) to   (GLU545)  BRAFV600E KINASE DOMAIN IN COMPLEX WITH CHEMICALLY LINKED VEMURAFENIB INHIBITOR VEM-BISAMIDE  |   KINASE, DIMER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fza:B    (GLY36) to   (LYS139)  CRYSTAL STRUCTURE OF MST4-MO25 COMPLEX  |   SCAFFOLD PROTEIN, PROTEIN SER/THR KINASE, ATP BINDING, SIGNALING PROTEIN-TRANSFERASE COMPLEX 
4fzf:B    (GLY36) to   (LYS139)  CRYSTAL STRUCTURE OF MST4-MO25 COMPLEX WITH DKI  |   SCAFFOLD PROTEIN, PROTEIN SER/THR KINASE, ATP BINDING, SIGNALING PROTEIN-TRANSFERASE-INHIBITOR COMPLEX 
4g31:A   (GLY604) to   (GLY931)  CRYSTAL STRUCTURE OF GSK6414 BOUND TO PERK (R587-R1092, DELETE A660- T867) AT 2.28 A RESOLUTION  |   DELETION MUTANT, CATALYTIC DOMAIN, SYNTHETIC INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4g34:A   (GLY604) to   (GLY931)  CRYSTAL STRUCTURE OF GSK6924 BOUND TO PERK (R587-R1092, DELETE A660- T867) AT 2.70 A RESOLUTION  |   DELETION MUTANT, CATALYTIC DOMAIN, SYNTHETIC INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
5jzj:A   (SER424) to   (ASN506)  CRYSTAL STRUCTURE OF DCLK1-KD IN COMPLEX WITH AMPPN  |   KINASE, DOUBLECORTIN, TRANSFERASE 
5k5x:A   (GLY610) to   (ASN813)  CRYSTAL STRUCTURE OF HUMAN PDGFRA  |   TYROSINE KINASE, AUTOINHIBITION, TRANSFERASE 
4g9c:A   (THR470) to   (GLU545)  HUMAN B-RAF KINASE DOMAIN BOUND TO A TYPE II PYRAZOLOPYRIDINE INHIBITOR  |   DFG-OUT, INHIBITOR, TYPE II, TRANSFERASE, KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4g9c:B   (LYS473) to   (GLU545)  HUMAN B-RAF KINASE DOMAIN BOUND TO A TYPE II PYRAZOLOPYRIDINE INHIBITOR  |   DFG-OUT, INHIBITOR, TYPE II, TRANSFERASE, KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4g9r:A   (GLY469) to   (SER571)  B-RAF V600E KINASE DOMAIN BOUND TO A TYPE II DIHYDROQUINAZOLINE INHIBITOR  |   INHIBITOR, TYPE II, TRANSFERASE, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4gg5:A  (GLY1090) to  (LYS1199)  CRYSTAL STRUCTURE OF CMET IN COMPLEX WITH NOVEL INHIBITOR  |   CMET INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4gkh:C    (THR39) to   (SER133)  CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR 1-NA-PP1  |   PYRAZOLOPYRIMIDINE, 1-NA-PP1, BUMPED KINASE INHIBITOR, BKI, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR 
4gkh:I    (THR39) to   (SER133)  CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR 1-NA-PP1  |   PYRAZOLOPYRIMIDINE, 1-NA-PP1, BUMPED KINASE INHIBITOR, BKI, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR 
4gkh:L    (THR39) to   (PRO135)  CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR 1-NA-PP1  |   PYRAZOLOPYRIMIDINE, 1-NA-PP1, BUMPED KINASE INHIBITOR, BKI, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR 
4gl9:B   (GLY861) to   (ARG971)  CRYSTAL STRUCTURE OF INHIBITORY PROTEIN SOCS3 IN COMPLEX WITH JAK2 KINASE DOMAIN AND FRAGMENT OF GP130 INTRACELLULAR DOMAIN  |   KINASE INHIBITOR RECEPTOR CYTOKINE SIGNALLING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4gmy:A   (PHE860) to   (ARG971)  JAK2 KINASE (JH1 DOMAIN) IN COMPLEX WITH 2,6-DICHLORO-N-{2- [(CYCLOPROPYLCARBONYL)AMINO]PYRIDIN-4-YL}BENZAMIDE  |   JAK2, JH1 KINASE DOMAIN, TYROSINE KINASE, PHOSPHOTRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5kx8:B   (GLY198) to   (HIS306)  IRAK4-INHIBITOR CO-STRUCTURE  |   KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5l2i:A    (GLY25) to   (ARG140)  THE X-RAY CO-CRYSTAL STRUCTURE OF HUMAN CDK6 AND PALBOCICLIB.  |   CYCLIN-DEPENDENT KINASE, KINASE INHIBITOR, KINASE SELECTIVITY, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5l4q:A    (ALA58) to   (HIS166)  CRYSTAL STRUCTURE OF ADAPTOR PROTEIN 2 ASSOCIATED KINASE 1 (AAK1) IN COMPLEX WITH LKB1 (AAK1 DUAL INHIBITOR)  |   KINASE KINASE DOMAIN, TRANSFERASE 
5l4q:B    (ALA58) to   (HIS166)  CRYSTAL STRUCTURE OF ADAPTOR PROTEIN 2 ASSOCIATED KINASE 1 (AAK1) IN COMPLEX WITH LKB1 (AAK1 DUAL INHIBITOR)  |   KINASE KINASE DOMAIN, TRANSFERASE 
5m55:A    (ARG21) to   (SER131)  NEK2 BOUND TO ARYLAMINOPURINE 71  |   PROTEIN KINASE, INHIBITOR, CENTROSOME SEPARATION, TRANSFERASE 
5t6a:A    (GLY63) to   (LYS169)  CRYSTAL STRUCTURE OF TGCDPK1 FROM TOXOPLASMA GONDII COMPLEXED WITH 5GA  |   STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPKS, SERINE/THREONINE PROTEIN KINASE, NUCLEOTIDE-BINDING, TRANSFERASE 
5t6k:A    (GLY63) to   (LYS169)  CRYSTAL STRUCTURE OF TGCDPK1 FROM TOXOPLASMA GONDII COMPLEXED WITH GW780159X  |   STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPKS, SERINE/THREONINE PROTEIN KINASE, NUCLEOTIDE-BINDING, TRANSFERASE 
3ekk:A  (GLY1013) to  (LYS1127)  INSULIN RECEPTOR KINASE COMPLEXED WITH AN INHIBITOR  |   INSULIN, TYROSINE KINASE, ATP-BINDING, CARBOHYDRATE METABOLISM, CLEAVAGE ON PAIR OF BASIC RESIDUES, DIABETES MELLITUS, DISEASE MUTATION, GLYCOPROTEIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE 
2bdf:B   (GLU280) to   (LEU358)  SRC KINASE IN COMPLEX WITH INHIBITOR AP23451  |   SRC KINASE INHIBITOR, TRANSFERASE 
2c0t:A   (MET257) to   (GLN332)  SRC FAMILY KINASE HCK WITH BOUND INHIBITOR A-641359  |   TRANSFERASE, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, SH2 DOMAIN, SH3 DOMAIN 
4xhg:A    (GLY21) to   (SER123)  STRUCTURE OF C. GLABRATA HRR25 BOUND TO ADP (FORMATE CONDITION)  |   CASEIN KINASE, MONOPOLIN, TRANSFERASE 
2psq:A   (ALA498) to   (LYS621)  CRYSTAL STRUCTURE OF UNPHOSPHORYLATED UNACTIVATED WILD TYPE FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN  |   KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, TRANSFERASE 
2pui:B    (LEU43) to   (SER152)  STRUCTURES OF 5-METHYLTHIORIBOSE KINASE REVEAL SUBSTRATE SPECIFICITY AND UNUSUAL MODE OF NUCLEOTIDE BINDING  |   5-METHYLTHIORIBOSE KINASE, METHIONINE RECYCLING PATHWAY, TRANSFERASE 
1cki:A    (GLY24) to   (ASN126)  RECOMBINANT CASEIN KINASE I DELTA TRUNCATION MUTANT CONTAINING RESIDUES 1-317  |   PROTEIN KINASE, PHOSPHOTRANSFERASE 
1cki:B    (GLY24) to   (ASN126)  RECOMBINANT CASEIN KINASE I DELTA TRUNCATION MUTANT CONTAINING RESIDUES 1-317  |   PROTEIN KINASE, PHOSPHOTRANSFERASE 
2qi8:A   (GLY284) to   (LEU358)  CRYSTAL STRUCTURE OF DRUG RESISTANT SRC KINASE DOMAIN  |   SRC KINASE DOMAIN; DRUG RESISTANCE, SIGNALING PROTEIN, TRANSFERASE 
3g6h:A   (GLY279) to   (LEU358)  SRC THR338ILE INHIBITED IN THE DFG-ASP-OUT CONFORMATION  |   CANCER, IMATINIB RESISTANCE, DSA COMPOUNDS, KINASE, DFG-ASP- OUT, ALTERNATIVE SPLICING, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE 
3g6h:B   (GLY279) to   (LEU358)  SRC THR338ILE INHIBITED IN THE DFG-ASP-OUT CONFORMATION  |   CANCER, IMATINIB RESISTANCE, DSA COMPOUNDS, KINASE, DFG-ASP- OUT, ALTERNATIVE SPLICING, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE 
4y0x:A   (GLY163) to   (GLY271)  CRYSTAL STRUCTURE OF THE S/T PROTEIN KINASE PKNG FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH ADP  |   S/T PROTEIN KINASE, PKNG, TRANSFERASE 
3gp0:A    (SER37) to   (GLY145)  CRYSTAL STRUCTURE OF HUMAN MITOGEN ACTIVATED PROTEIN KINASE 11 (P38 BETA) IN COMPLEX WITH NILOTINIB  |   MITOGEN-ACTIVATED PROTEIN KINASE 11, P38B, P38BETA, PRKM11, SAPK2, SAPK2B, STRESS-ACTIVATED PROTEIN KINASE-2, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4y5q:A    (LEU91) to   (ILE178)  ACTIVATED CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM CRYPTOSPORIDIUM PARVUM (CPCDPK1) IN COMPLEX WITH AMP  |   SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, BUMPED KINASE INHIBITOR, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP 
3tdw:A    (TYR34) to   (PHE130)  THE GDP COMPLEX OF THE AMINOGLYCOSIDE 2'-PHOSPHOTRANSFERE-IIIA F108L MUTANT  |   KINASE, PHOSPHORYL TRANSFER, ANTIBIOTIC RESISTANCE, TRANSFERASE 
3gu8:A    (ALA25) to   (GLN134)  CRYSTAL STRUCTURE OF DAPKL93G WITH N6-CYCLOPENTYLADENOSINE  |   GATEKEEPER MUTANT, ALTERNATIVE SPLICING, ANK REPEAT, APOPTOSIS, ATP-BINDING, CALMODULIN-BINDING, CYTOPLASM, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
4jg6:A   (SER434) to   (GLY534)  RSK2 CTD BOUND TO 2-CYANO-3-(1H-INDAZOL-5-YL)ACRYLAMIDE  |   PROTEIN KINASE, PHOSPHORYLATION, COVALENT INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
1eh4:A    (GLY24) to   (GLU124)  BINARY COMPLEX OF CASEIN KINASE-1 FROM S. POMBE WITH AN ATP COMPETITIVE INHIBITOR, IC261  |   PROTEIN KINASE, CASEIN KINASE-1, PROTEIN-INHIBITOR BINARY COMPLEX, TRANSFERASE 
1eh4:B    (VAL25) to   (GLU124)  BINARY COMPLEX OF CASEIN KINASE-1 FROM S. POMBE WITH AN ATP COMPETITIVE INHIBITOR, IC261  |   PROTEIN KINASE, CASEIN KINASE-1, PROTEIN-INHIBITOR BINARY COMPLEX, TRANSFERASE 
1qcf:A   (GLY279) to   (GLN358)  CRYSTAL STRUCTURE OF HCK IN COMPLEX WITH A SRC FAMILY- SELECTIVE TYROSINE KINASE INHIBITOR  |   TYROSINE KINASE-INHIBITOR COMPLEX, DOWN-REGULATED KINASE, ORDERED ACTIVATION LOOP 
1qpd:A   (GLY257) to   (LEU336)  STRUCTURAL ANALYSIS OF THE LYMPHOCYTE-SPECIFIC KINASE LCK IN COMPLEX WITH NON-SELECTIVE AND SRC FAMILY SELECTIVE KINASE INHIBITORS  |   ALPHA BETA FOLD, TRANSFERASE 
4yne:A   (ASP537) to   (HIS645)  (R)-2-PHENYLPYRROLIDINE SUBSTITUTE IMIDAZOPYRIDAZINES: A NEW CLASS OF POTENT AND SELECTIVE PAN-TRK INHIBITORS  |   KINASE, TRK, INHIBITOR, ONCOLOGY, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3udb:A    (VAL34) to   (MET134)  CRYSTAL STRUCTURE OF SNRK2.6  |   SNRK2.6, KINASE, ABA SIGNALING PATHWAY, ABI1, TRANSFERASE 
3udb:C    (VAL34) to   (GLN135)  CRYSTAL STRUCTURE OF SNRK2.6  |   SNRK2.6, KINASE, ABA SIGNALING PATHWAY, ABI1, TRANSFERASE 
3udb:E    (VAL34) to   (GLN135)  CRYSTAL STRUCTURE OF SNRK2.6  |   SNRK2.6, KINASE, ABA SIGNALING PATHWAY, ABI1, TRANSFERASE 
2v7a:B   (GLY254) to   (ASN336)  CRYSTAL STRUCTURE OF THE T315I ABL MUTANT IN COMPLEX WITH THE INHIBITOR PHA-739358  |   KINASE, NUCLEUS, MYRISTATE, CYTOPLASM, MANGANESE, CELL ADHESION, METAL-BINDING, PROTO-ONCOGENE, TYROSINE-PROTEIN KINASE, CHROMOSOMAL REARRANGEMENT, TRANSFERASE, LIPOPROTEIN, POLYMORPHISM, CYTOSKELETON, MAGNESIUM, SH2 DOMAIN, SH3 DOMAIN, ATP-BINDING, NUCLEOTIDE-BINDING, ALTERNATIVE SPLICING, PHOSPHORYLATION, KINASE INHIBITOR, T315I ABL MUTANT 
3hmi:A   (GLU301) to   (THR382)  THE CRYSTAL STRUCTURE OF HUMAN ABL2 IN COMPLEX WITH 5-AMINO-3-{[4- (AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4- TRIAZOLE-1-CARBOTHIOAMIDE  |   TYROSINE KINASE, ABL, ABL2, ABELSON MURINE LEUKEMIA VIRAL ONCOGENE, ATP-BINDING, CELL ADHESION, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC 
4kbc:B    (GLY21) to   (ASN123)  CK1D IN COMPLEX WITH {4-[3-(4-FLUOROPHENYL)-1H-PYRAZOL-4-YL]PYRIDIN-2- YL}METHANOL INHIBITOR  |   SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3uzp:A    (GLY21) to   (ASN123)  CRYSTAL STRUCTURE OF CK1D WITH PF670462 FROM P21 CRYSTAL FORM  |   CK1D, KINASE, INHIBITOR, PF670462, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3uzp:B    (GLY21) to   (ASN123)  CRYSTAL STRUCTURE OF CK1D WITH PF670462 FROM P21 CRYSTAL FORM  |   CK1D, KINASE, INHIBITOR, PF670462, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2g2f:B   (GLU255) to   (ASN336)  A SRC-LIKE INACTIVE CONFORMATION IN THE ABL TYROSINE KINASE DOMAIN  |   PROTEIN KINASE, TRANSFERASE 
1sm2:B   (GLY375) to   (PHE454)  CRYSTAL STRUCTURE OF THE PHOSPHORYLATED INTERLEUKIN-2 TYROSINE KINASE CATALYTIC DOMAIN  |   PROTEIN KINASE, IMMUNOLOGY, TRANSFERASE 
3i79:A    (GLY63) to   (LYS169)  CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1)  |   PROTEIN KINASE, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, TRANSFERASE 
2vz6:B    (SER25) to   (GLY130)  STRUCTURE OF HUMAN CALCIUM CALMODULIN DEPENDENT PROTEIN KINASE TYPE II ALPHA (CAMK2A) IN COMPLEX WITH INDIRUBIN E804  |   TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, CELL JUNCTION, CELL MEMBRANE, LONG TERM POTENTIATION, BRAIN, KINASE, SYNAPSE, MEMBRANE, NMDA RECEPTOR SIGNALLING, PHOSPHOPROTEIN, CALMODULIN-BINDING, NUCLEOTIDE-BINDING 
4zs0:A   (LEU149) to   (ARG251)  HUMAN AURORA A CATALYTIC DOMAIN BOUND TO SB-6-OH  |   AURORA, KINASE, INHIBITOR, TRANSFERASE 
4lg4:D    (SER40) to   (ARG141)  STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5  |   HIPPO, MST AUTOACTIVATION, DIMERIZATION, SIGNALING PROTEIN 
3vs0:A   (MET283) to   (GLN358)  CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRROLO-PYRIMIDINE INHIBITOR N-[4-(4-AMINO-7-CYCLOPENTYL-7H-PYRROLO[2,3-D]PYRIMIDIN-5-YL) PHENYL]BENZAMIDE  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3vs6:A   (MET283) to   (GLN358)  CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRAZOLO-PYRIMIDINE INHIBITOR TERT-BUTYL {4-[4-AMINO-1-(PROPAN-2-YL)-1H-PYRAZOLO[3,4- D]PYRIMIDIN-3-YL]-2-METHOXYPHENYL}CARBAMATE  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5a4l:A   (GLY171) to   (ALA277)  DYRK1A IN COMPLEX WITH FLUORO BENZOTHIAZOLE FRAGMENT  |   TRANSFERASE 
2i0v:A   (ALA599) to   (ASN773)  C-FMS TYROSINE KINASE IN COMPLEX WITH A QUINOLONE INHIBITOR  |   RECEPTOR TYROSINE KINASE, KINASE-INHIBITOR COMPLEX, TRANSFERASE 
5aep:A   (GLY861) to   (ASP949)  NOVEL PYRROLE CARBOXAMIDE INHIBITORS OF JAK2 AS POTENTIAL TREATMENT OF MYELOPROLIFERATIVE DISORDERS  |   TRANSFERASE, PROTEIN KINASE, JAK2, MYELOPROLIFERATIVE DISORDERS, TUMOUR CELL PROLIFERATION INHIBITION, ANTI-CANCER AGENTS 
5ax9:A    (GLY37) to   (LYS148)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN TRAF2 AND NCK- INTERACTING PROTEIN KINASE IN COMPLEX WITH COMPUND 9  |   INHIBITOR, KINASE, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4mxo:A   (GLY279) to   (LEU358)  HUMAN SRC KINASE BOUND TO KINASE INHIBITOR BOSUTINIB  |   KINASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3zep:C   (SER835) to   (ARG944)  CRYSTAL STRUCTURE OF JAK3 KINASE DOMAIN IN COMPLEX WITH A PYRROLOPYRAZINE-2-PHENYL ETHER INHIBITOR  |   TRANSFERASE, STAT5, STAT6, INTERLEUKIN-2, COMMON-GAMMA CHAIN, ATP SITE KINASE INHIBITOR, CANCER, SCID, SEVERE COMBINED IMMUNODEFICIENCY 
5c9c:A   (GLY468) to   (GLU544)  CRYSTAL STRUCTURE OF BRAF(V600E) IN COMPLEX WITH LY3009120 COMPND  |   TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4o1p:A   (GLY380) to   (GLY477)  CRYSTAL STRUCTURE OF RNASE L IN COMPLEX WITH 2-5A AND AMP-PNP  |   ANKYRIN REPEAT-KINASE-RNASE, RNA CLEAVAGE, 2-5A, TRANSFERASE, HYDROLASE 
4o1p:C   (GLY380) to   (GLY477)  CRYSTAL STRUCTURE OF RNASE L IN COMPLEX WITH 2-5A AND AMP-PNP  |   ANKYRIN REPEAT-KINASE-RNASE, RNA CLEAVAGE, 2-5A, TRANSFERASE, HYDROLASE 
4o1p:D   (GLY380) to   (GLY477)  CRYSTAL STRUCTURE OF RNASE L IN COMPLEX WITH 2-5A AND AMP-PNP  |   ANKYRIN REPEAT-KINASE-RNASE, RNA CLEAVAGE, 2-5A, TRANSFERASE, HYDROLASE 
3k5v:A   (GLU274) to   (SER355)  STRUCTURE OF ABL KINASE IN COMPLEX WITH IMATINIB AND GNF-2  |   KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3kc3:A    (LYS77) to   (ASN181)  MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE  |   MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3kc3:G    (LEU79) to   (ILE170)  MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE  |   MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3kc3:I    (LEU79) to   (GLY171)  MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE  |   MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
5cwz:C    (GLY37) to   (LYS148)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN TRAF2 AND NCK- INTERACTING PROTEIN KINASE  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2zm4:A   (PHE256) to   (LEU336)  CRYSTAL STRUCTURE OF IMIDAZO QUINOXALINE 1 BOUND TO THE KINASE DOMAIN OF HUMAN LCK, ACTIVATED FORM (AUTO- PHOSPHORYLATED ON TYR394)  |   TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE- BINDING, PALMITATE, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
3a2c:G    (LEU79) to   (ASN181)  CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2)  |   GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3ad6:A   (PHE256) to   (LEU336)  CRYSTAL STRUCTURE OF PYRAZOLO PYRIMIDINE DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394)  |   TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE 
1yrp:A    (PHE24) to   (PHE119)  CATALYTIC DOMAIN OF HUMAN ZIP KINASE PHOSPHORYLATED AT THR265  |   KINASE FOLD, PHOSPHOTHREONINE, TRANSFERASE 
1yrp:B    (PHE24) to   (PHE119)  CATALYTIC DOMAIN OF HUMAN ZIP KINASE PHOSPHORYLATED AT THR265  |   KINASE FOLD, PHOSPHOTHREONINE, TRANSFERASE 
4ark:A    (LYS84) to   (LYS185)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN MAP KINASE KINASE 1 (MEK1) IN COMPLEX WITH  A SMALL MOLECULE INHIBITOR AND ADP  |   TRANSFERASE, KINASE, INHIBITOR 
4at3:A   (GLY566) to   (LEU654)  CRYSTAL STRUCTURE OF TRKB KINASE DOMAIN IN COMPLEX WITH CPD5N  |   TRANSFERASE 
4at5:A   (ALA571) to   (ALA656)  CRYSTAL STRUCTURE OF TRKB KINASE DOMAIN IN COMPLEX WITH GW2580  |   TRANSFERASE 
1zws:A    (ALA25) to   (LYS134)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE  |   PROTEIN KINASE, TWINNING, TRANSFERASE 
1zws:B    (ALA25) to   (LYS134)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE  |   PROTEIN KINASE, TWINNING, TRANSFERASE 
1zws:C    (ALA25) to   (LYS134)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE  |   PROTEIN KINASE, TWINNING, TRANSFERASE 
1zws:D    (ALA25) to   (LYS134)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE  |   PROTEIN KINASE, TWINNING, TRANSFERASE 
1zws:E    (ALA25) to   (LYS134)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE  |   PROTEIN KINASE, TWINNING, TRANSFERASE 
1zws:F    (ALA25) to   (LYS134)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE  |   PROTEIN KINASE, TWINNING, TRANSFERASE 
1zws:G    (ALA25) to   (LYS134)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE  |   PROTEIN KINASE, TWINNING, TRANSFERASE 
1zws:H    (ALA25) to   (LYS134)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN DRP-1 KINASE  |   PROTEIN KINASE, TWINNING, TRANSFERASE 
3lvp:C  (PRO1026) to  (LYS1130)  CRYSTAL STRUCTURE OF BISPHOSPHORYLATED IGF1-R KINASE DOMAIN (2P) IN COMPLEX WITH A BIS-AZAINDOLE INHIBITOR  |   PROTEIN KINASE, TYROSINE KINASE, TYROSINE PHOSPHORYLATION, PROTEIN- SUBSTRATE COMPLEX, TRANSFERASE 
3att:A    (GLU57) to   (SER178)  CRYSTAL STRUCTURE OF RV3168 WITH ATP  |   HYPOTHETICAL PROTEIN, PUTATIVE AMINOGLYCOSIDE PHOSPHORTRANSFERASE, TRANSFERASE 
5ehl:A   (SER537) to   (GLY642)  RAPID DISCOVERY OF PYRIDO[3,4-D]PYRIMIDINE INHIBITORS OF MONOPOLAR SPINDLE KINASE 1 (MPS1) USING A STRUCTURE-BASED HYDRIDIZATION APPROACH  |   SPINDLE ASSEMBLY CHECKPOINT (SAC), ONCOLOGY TARGET PYRIDO[3, 4- D]PYRIMIDINE BASED INHIBITORS SELECTIVE AGAINST MPS1, TRANSFERASE 
5ei8:A   (SER537) to   (GLN640)  RAPID DISCOVERY OF PYRIDO[3,4-D]PYRIMIDINE INHIBITORS OF MONOPOLAR SPINDLE KINASE 1 (MPS1) USING A STRUCTURE-BASED HYDRIDIZATION APPROACH  |   SPINDLE ASSEMBLY CHECKPOINT (SAC), ONCOLOGY TARGET PYRIDO[3, 4- D]PYRIMIDINE BASED INHIBITORS SELECTIVE AGAINST MPS1, TRANSFERASE 
4bch:A    (GLY31) to   (LYS144)  STRUCTURE OF CDK9 IN COMPLEX WITH CYCLIN T AND A 2-AMINO-4- HETEROARYL-PYRIMIDINE INHIBITOR  |   TRANSFERASE-CELL CYCLE COMPLEX, CDK-CYCLIN COMPLEX, TRANSCRIPTION-PROTEIN BINDING, STRUCTURE-BASED DRUG DESIGN 
4qox:A    (GLU83) to   (ASN188)  CRYSTAL STRUCTURE OF CDPK4 FROM PLASMODIUM FALCIPARUM, PF3D7_0717500  |   STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPK, PLASMODIUM, MALARIA, TRANSFERASE 
3miy:A   (LEU379) to   (SER477)  X-RAY CRYSTAL STRUCTURE OF ITK COMPLEXED WITH SUNITINIB  |   HELIX C-IN, TRANSFERASE 
5eqe:B   (LEU124) to   (MET238)  CRYSTAL STRUCTURE OF CHOLINE KINASE ALPHA-1 BOUND BY [4-[(4-METHYL-1, 4-DIAZEPAN-1-YL)METHYL]PHENYL]METHANAMINE (COMPOUND 11)  |   KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4qrc:A   (ALA484) to   (LYS607)  CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF FGF RECEPTOR 4 IN COMPLEX WITH PONATINIB  |   KINASE DOMAIN FOLD, CELL SIGNALING, PHOSPHOTRANSFERASE, PLASMAMEMBRANE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4bgg:A   (GLY220) to   (HIS320)  CRYSTAL STRUCTURE OF THE ACVR1 KINASE IN COMPLEX WITH LDN-213844  |   TRANSFERASE, INHIBITOR, BMP SIGNALLING 
4bgg:B   (GLY220) to   (HIS320)  CRYSTAL STRUCTURE OF THE ACVR1 KINASE IN COMPLEX WITH LDN-213844  |   TRANSFERASE, INHIBITOR, BMP SIGNALLING 
4bgg:C   (GLY220) to   (HIS320)  CRYSTAL STRUCTURE OF THE ACVR1 KINASE IN COMPLEX WITH LDN-213844  |   TRANSFERASE, INHIBITOR, BMP SIGNALLING 
4bgg:D   (GLY220) to   (HIS320)  CRYSTAL STRUCTURE OF THE ACVR1 KINASE IN COMPLEX WITH LDN-213844  |   TRANSFERASE, INHIBITOR, BMP SIGNALLING 
3bhh:A    (SER26) to   (GLY131)  CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE IIB ISOFORM 1 (CAMK2B)  |   CAMK2B, CAM2, CAMK2, CAM KINASE II BETA CHAIN, CAMK II BETA SUBUNIT, CALCIUM/CALMODULION DEPENDENT PROTEIN KINASE II BETA, EC:2.7.1.123, MGC29528, PROLINE RICH CALMODULIN DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, CALMODULIN- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE 
3bhh:B    (SER26) to   (GLY131)  CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE IIB ISOFORM 1 (CAMK2B)  |   CAMK2B, CAM2, CAMK2, CAM KINASE II BETA CHAIN, CAMK II BETA SUBUNIT, CALCIUM/CALMODULION DEPENDENT PROTEIN KINASE II BETA, EC:2.7.1.123, MGC29528, PROLINE RICH CALMODULIN DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, CALMODULIN- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE 
3bhh:C    (VAL27) to   (GLY131)  CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE IIB ISOFORM 1 (CAMK2B)  |   CAMK2B, CAM2, CAMK2, CAM KINASE II BETA CHAIN, CAMK II BETA SUBUNIT, CALCIUM/CALMODULION DEPENDENT PROTEIN KINASE II BETA, EC:2.7.1.123, MGC29528, PROLINE RICH CALMODULIN DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, CALMODULIN- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE 
3bhh:D    (VAL27) to   (GLY131)  CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE IIB ISOFORM 1 (CAMK2B)  |   CAMK2B, CAM2, CAMK2, CAM KINASE II BETA CHAIN, CAMK II BETA SUBUNIT, CALCIUM/CALMODULION DEPENDENT PROTEIN KINASE II BETA, EC:2.7.1.123, MGC29528, PROLINE RICH CALMODULIN DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, CALMODULIN- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE 
3biz:A   (SER312) to   (SER421)  WEE1 KINASE COMPLEX WITH INHIBITOR PD331618  |   KINASE DOMAIN, INHIBITOR COMPLEX, ATP-BINDING, CELL CYCLE, CELL DIVISION, MAGNESIUM, METAL-BINDING, MITOSIS, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE, TYROSINE-PROTEIN KINASE 
3n4v:A    (ILE35) to   (ILE133)  APO APH(2")-IVA FORM III  |   AMINOGLYCOSIDE, PHOSPHOTRANSFERASE, RESISTANCE, UNKNOWN FUNCTION 
4c02:A   (GLY220) to   (HIS320)  CRYSTAL STRUCTURE OF HUMAN ACVR1 (ALK2) IN COMPLEX WITH FKBP12.6 AND DORSOMORPHIN  |   TRANSFERASE-ISOMERASE COMPLEX, TRANSFERASE, DORSOMORPHIN, 
4rfy:A   (GLY414) to   (GLN516)  CRYSTAL STRUCTURE OF BTK KINASE DOMAIN COMPLEXED WITH 6- (DIMETHYLAMINO)-2-[2-(HYDROXYMETHYL)-3-[1-METHYL-5-[[5-(MORPHOLINE-4- CARBONYL)-2-PYRIDYL]AMINO]-6-OXO-3-PYRIDYL]PHENYL]-3,4- DIHYDROISOQUINOLIN-1-ONE  |   TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5fxq:A  (PRO1026) to  (LYS1130)  IGFR-1R COMPLEX WITH A PYRIMIDINE INHIBITOR.  |   TRANSFERASE 
4d2t:A    (LYS24) to   (VAL112)  STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS  |   TRANSFERASE, FRAGMENT BASED DRUG DESIGN, KINASE 
4d2t:C    (LYS24) to   (VAL112)  STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS  |   TRANSFERASE, FRAGMENT BASED DRUG DESIGN, KINASE 
4d2t:D    (PHE22) to   (VAL112)  STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS  |   TRANSFERASE, FRAGMENT BASED DRUG DESIGN, KINASE 
4twc:A    (ASP22) to   (ASN123)  2-BENZAMIDO-N-(1H-BENZO[D]IMIDAZOL-2-YL)THIAZOLE-4- CARBOXAMIDE DERIVATIVES AS POTENT INHIBITORS OF CK1D/E  |   CK1D, CK1E, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, TRANSFERASE 
3dpk:A   (ALA599) to   (ASN773)  CFMS TYROSINE KINASE IN COMPLEX WITH A PYRIDOPYRIMIDINONE INHIBITOR  |   RECEPTOR TYROSINE KINASE, KINASE-INHIBITOR COMPLEX, ATP- BINDING, GLYCOPROTEIN, IMMUNOGLOBULIN DOMAIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, ALTERNATIVE SPLICING, CHROMOSOMAL REARRANGEMENT, CRANIOSYNOSTOSIS, DISEASE MUTATION, DWARFISM, HEPARIN-BINDING, KALLMANN SYNDROME 
5hbj:A    (GLY33) to   (TRP146)  CDK8-CYCC IN COMPLEX WITH 8-[2-AMINO-3-CHLORO-5-(1-METHYL-1H-INDAZOL- 5-YL)-PYRIDIN-4-YL]-2,8-DIAZA-SPIRO[4.5]DECAN-1-ONE  |   CDK8 KINASE / CYCLIN C, TRANSFERASE 
4u42:A    (GLN38) to   (HIS148)  MAP4K4 T181E MUTANT BOUND TO INHIBITOR COMPOUND 1  |   KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3owe:B   (LYS124) to   (ASN211)  CRYSTAL STRUCTURE OF STAPHYLOCOCCAL ENTEROTOXIN G (SEG) IN COMPLEX WITH A HIGH AFFINITY MUTANT MOUSE T-CELL RECEPTOR CHAIN  |   T-CELL RECEPTOR V BETA DOMAIN, COMPLEX STRUCTURE, IGG DOMAINS, B GRASP, VIRULENCE FACTORS, IMMUNE SYSTEM 
3owe:H   (LYS124) to   (ASN211)  CRYSTAL STRUCTURE OF STAPHYLOCOCCAL ENTEROTOXIN G (SEG) IN COMPLEX WITH A HIGH AFFINITY MUTANT MOUSE T-CELL RECEPTOR CHAIN  |   T-CELL RECEPTOR V BETA DOMAIN, COMPLEX STRUCTURE, IGG DOMAINS, B GRASP, VIRULENCE FACTORS, IMMUNE SYSTEM 
3owe:J   (LYS124) to   (LEU210)  CRYSTAL STRUCTURE OF STAPHYLOCOCCAL ENTEROTOXIN G (SEG) IN COMPLEX WITH A HIGH AFFINITY MUTANT MOUSE T-CELL RECEPTOR CHAIN  |   T-CELL RECEPTOR V BETA DOMAIN, COMPLEX STRUCTURE, IGG DOMAINS, B GRASP, VIRULENCE FACTORS, IMMUNE SYSTEM 
5hx6:B    (VAL31) to   (GLY133)  CRYSTAL STRUCTURE OF RIP1 KINASE WITH A BENZO[B][1,4]OXAZEPIN-4-ONE  |   KINASE, INHIBITOR COMPLEX, NON-HINGE BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3piy:A   (GLY414) to   (GLN516)  CRYSTAL STRUCTURE OF BTK KINASE DOMAIN COMPLEXED WITH R406  |   HELIX C-OUT, DFG-IN, TRANSFERASE, TRANSFERASE-INHIBITOR COMPLEX 
4usf:B    (LYS47) to   (LYS150)  HUMAN SLK WITH SB-440719  |   TRANSFERASE 
5ig1:A    (SER30) to   (ASN135)  CRYSTAL STRUCTURE OF S. ROSETTA CAMKII KINASE DOMAIN  |   CA2+/CAM-DEPENDENT KINASE, CHOANOFLAGELLATE, TRANSFERASE 
5ig1:B    (PHE29) to   (ASN135)  CRYSTAL STRUCTURE OF S. ROSETTA CAMKII KINASE DOMAIN  |   CA2+/CAM-DEPENDENT KINASE, CHOANOFLAGELLATE, TRANSFERASE 
5ih4:A    (ASP22) to   (LYS122)  HUMAN CASEIN KINASE 1 ISOFORM DELTA APO (KINASE DOMAIN)  |   KINASE DOMAIN, STEM CELL REPROGRAMMING, TRANSFERASE 
4w4w:A    (ILE77) to   (GLY184)  JNK2/3 IN COMPLEX WITH N-(2-METHYLPYRIDIN-4-YL)-3-{4- [(PHENYLCARBAMOYL)AMINO]-1H-PYRAZOL-1-YL}BENZAMIDE  |   JNK, MAP KINASE, ISOFORM SELECTIVE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fig:A   (GLY333) to   (GLY435)  CATALYTIC DOMAIN OF HUMAN PAK4  |   SERINE/THREONINE-PROTEIN KINASE PAK4, KINASE DOMAIN, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE 
4fig:B   (GLY333) to   (GLY435)  CATALYTIC DOMAIN OF HUMAN PAK4  |   SERINE/THREONINE-PROTEIN KINASE PAK4, KINASE DOMAIN, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE 
3r2b:C    (LEU79) to   (ASN181)  MK2 KINASE BOUND TO COMPOUND 5B  |   KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3r2b:E    (LEU79) to   (ILE170)  MK2 KINASE BOUND TO COMPOUND 5B  |   KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3r2b:G    (LEU79) to   (ASN181)  MK2 KINASE BOUND TO COMPOUND 5B  |   KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3r7o:A  (CYS1091) to  (LYS1199)  STRUCTURE OF DUALLY PHOSPHORYLATED C-MET RECEPTOR KINASE IN COMPLEX WITH AN MK-2461 ANALOG  |   TYROSINE KINASE, PHOSPHOTYROSINE, 1234, 1235, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3raw:A   (GLY168) to   (GLN278)  CRYSTAL STRUCTURE OF HUMAN CDC-LIKE KINASE 3 ISOFORM IN COMPLEX WITH LEUCETTINE L41  |   TRANSFERASE, KINASE, TYROSINE-PROTEIN KINASE, SERINE/THREONINE- PROTEIN KINASE, NUCLEOTIDE-BINDING, STRUCTURAL GENOMICS CONSORTIUM, SGC 
5jrq:A   (LYS473) to   (GLU545)  BRAFV600E KINASE DOMAIN IN COMPLEX WITH CHEMICALLY LINKED VEMURAFENIB INHIBITOR VEM-6-VEM  |   KINASE, DIMER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5jrq:B   (THR470) to   (GLU545)  BRAFV600E KINASE DOMAIN IN COMPLEX WITH CHEMICALLY LINKED VEMURAFENIB INHIBITOR VEM-6-VEM  |   KINASE, DIMER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4gfq:A    (ASN56) to   (VAL185)  2.65 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF RIBOSOME RECYCLING FACTOR (FRR) FROM BACILLUS ANTHRACIS  |   STRUCTURAL GENOMICS, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, TRANSLATION 
5knj:B   (SER215) to   (HIS321)  PSEUDOKINASE DOMAIN OF MLKL BOUND TO COMPOUND 1.  |   PSEUDOKINASE DOMAIN MLKL COMPOUND 1 GFE OUT TYPE 2 INHIBITOR, MEMBRANE PROTEINS-INHIBITOR COMPLEX 
5lih:A   (ALA266) to   (GLY373)  STRUCTURE OF A PEPTIDE-SUBSTRATE BOUND TO PKCIOTA CORE KINASE DOMAIN  |   APKC, POLARITY, COMPLEX, TRANSFERASE