1nl6:A (ARG108) to (MET215) CRYSTAL STRUCTURE OF THE CYSTEINE PROTEASE HUMAN CATHEPSIN K IN COMPLEX WITH A COVALENT AZEPANONE INHIBITOR | HYDROLASE, SULFHYDRYL PROTEINASE
4i04:A (LYS219) to (ILE322) STRUCTURE OF ZYMOGEN OF CATHEPSIN B1 FROM SCHISTOSOMA MANSONI | PEPTIDASE, DIGESTIVE TRACT, HYDROLASE
4i04:B (LYS219) to (ILE322) STRUCTURE OF ZYMOGEN OF CATHEPSIN B1 FROM SCHISTOSOMA MANSONI | PEPTIDASE, DIGESTIVE TRACT, HYDROLASE
4i04:C (SER221) to (ILE322) STRUCTURE OF ZYMOGEN OF CATHEPSIN B1 FROM SCHISTOSOMA MANSONI | PEPTIDASE, DIGESTIVE TRACT, HYDROLASE
4i04:D (LYS219) to (ILE322) STRUCTURE OF ZYMOGEN OF CATHEPSIN B1 FROM SCHISTOSOMA MANSONI | PEPTIDASE, DIGESTIVE TRACT, HYDROLASE
4i05:A (LYS219) to (ILE322) STRUCTURE OF INTERMEDIATE PROCESSING FORM OF CATHEPSIN B1 FROM SCHISTOSOMA MANSONI | PEPTIDASE, DIGESTIVE TRACT, HYDROLASE
1csb:E (TYR148) to (ASP254) CRYSTAL STRUCTURE OF CATHEPSIN B INHIBITED WITH CA030 AT 2.1 ANGSTROMS RESOLUTION: A BASIS FOR THE DESIGN OF SPECIFIC EPOXYSUCCINYL INHIBITORS | PAPAIN-LIKE LYSOSOMAL DICARBOXY-PEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2dc6:A (CYS148) to (MET250) X-RAY CRYSTAL STRUCTURE ANALYSIS OF BOVINE SPLEEN CATHEPSIN B-CA073 COMPLEX | CATHEPSIN B, CYSTEINE PROTEASE, CA073, HYDROLASE, EC 3.4.22.1
2dc7:A (CYS148) to (MET250) X-RAY CRYSTAL STRUCTURE ANALYSIS OF BOVINE SPLEEN CATHEPSIN B-CA042 COMPLEX | CATHEPSIN B, CYSTEINE PROTEASE, CA042, HYDROLASE, EC 3.4.22.1
2dc8:A (CYS148) to (MET250) X-RAY CRYSTAL STRUCTURE ANALYSIS OF BOVINE SPLEEN CATHEPSIN B-CA059 COMPLEX | CATHEPSIN B, CYSTEINE PROTEASE, CA059, HYDROLASE, EC 3.4.22.1
2dc9:A (CYS148) to (MET250) X-RAY CRYSTAL STRUCTURE ANALYSIS OF BOVINE SPLEEN CATHEPSIN B-CA074ME COMPLEX | CATHEPSIN B, CYSTEINE PROTEASE, CA074ME, HYDROLASE, EC 3.4.22.1
2dcb:A (CYS148) to (MET250) X-RAY CRYSTAL STRUCTURE ANALYSIS OF BOVINE SPLEEN CATHEPSIN B-CA076 COMPLEX | CATHEPSIN B, CYSTEINE PROTEASE, CA076, HYDROLASE, EC 3.4.22.1
2dcc:A (CYS148) to (MET250) X-RAY CRYSTAL STRUCTURE ANALYSIS OF BOVINE SPLEEN CATHEPSIN B-CA077 COMPLEX | CATHEPSIN B, CYSTEINE PROTEASE, CA077, HYDROLASE, EC 3.4.22.1
2dcd:A (CYS148) to (MET250) X-RAY CRYSTAL STRUCTURE ANALYSIS OF BOVINE SPLEEN CATHEPSIN B-CA078 COMPLEX | CATHEPSIN B, CYSTEINE PROTEASE, CA078, HYDROLASE, EC 3.4.22.1
1qdq:A (SER150) to (MET250) X-RAY CRYSTAL STRUCTURE OF BOVINE CATHEPSIN B-CA074 COMPLEX | CATHEPSIN B, PAPAIN, CATHEPSIN B-SPECIFIC INHIBITOR COMPLEX, HYDROLASE
3h6s:A (THR110) to (VAL221) STRUCURE OF CLITOCYPIN - CATHEPSIN V COMPLEX | CATHEPSIN, CLITOCYPIN, KUNITZ INHIBITOR, CYSTEINE PROTEASE, DISULFIDE BOND, GLYCOPROTEIN, HYDROLASE, LYSOSOME, PROTEASE, THIOL PROTEASE, ZYMOGEN, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
3h7d:A (GLY109) to (MET215) THE CRYSTAL STRUCTURE OF THE CATHEPSIN K VARIANT M5 IN COMPLEX WITH CHONDROITIN-4-SULFATE | GLYCOSAMINOGLYCAN, SULFHYDRYL PEPTIDASE, CATHEPSIN K MUTANT, TERNARY COMPLEX, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, HYDROLASE, LYSOSOME, PROTEASE, THIOL PROTEASE, ZYMOGEN
3hhi:A (TRP232) to (LEU335) CRYSTAL STRUCTURE OF CATHEPSIN B FROM T. BRUCEI IN COMPLEX WITH CA074 | CYSTEINE PROTEASE, OCCLUDING LOOP, HYDROLASE, PROTEASE, THIOL PROTEASE
2f1g:A (LYS112) to (ILE217) CATHEPSIN S IN COMPLEX WITH NON-COVALENT 2-(BENZOXAZOL-2-YLAMINO)- ACETAMIDE | CATHEPSIN S, NONCOVALENT, INHIBITION, 2-(BENZOOXAZOL-2-YLAMINO) ACETAMIDES, HYDROLASE
4yyq:A (SER110) to (PRO214) FICIN A | CYSTEIN PROTEASE, HYDROLASE
2fq9:A (ALA107) to (ILE218) CATHEPSIN S WITH NITRILE INHIBITOR | PAPAIN, CYSTEINE PROTEASE, ANTIGEN PRESENTATION, DRUG DESIGN, HYDROLASE
2fud:A (ALA107) to (ILE218) HUMAN CATHEPSIN S WITH INHIBITOR CRA-27566 | CYSTEINE PROTEASE, PROTEINASE, PAPAIN, 27566, HYDROLASE
1glo:A (LYS112) to (ILE217) CRYSTAL STRUCTURE OF CYS25SER MUTANT OF HUMAN CATHEPSIN S | CATHEPSIN S, PROTEINASE, INHIBITOR, HYDROLASE, THIOL PROTEAS
1gmy:A (TYR148) to (ILE250) CATHEPSIN B COMPLEXED WITH DIPEPTIDYL NITRILE INHIBITOR | HYDROLASE/INHIBITOR, COMPLEX (HYDROLASE/INHIBITOR), COVALENT COMPLEX, PROTEASE, CATHEPSIN B, HYDROLASE, THIOL PROTEASE
1gmy:B (TYR148) to (ILE250) CATHEPSIN B COMPLEXED WITH DIPEPTIDYL NITRILE INHIBITOR | HYDROLASE/INHIBITOR, COMPLEX (HYDROLASE/INHIBITOR), COVALENT COMPLEX, PROTEASE, CATHEPSIN B, HYDROLASE, THIOL PROTEASE
1gmy:C (TYR148) to (ILE250) CATHEPSIN B COMPLEXED WITH DIPEPTIDYL NITRILE INHIBITOR | HYDROLASE/INHIBITOR, COMPLEX (HYDROLASE/INHIBITOR), COVALENT COMPLEX, PROTEASE, CATHEPSIN B, HYDROLASE, THIOL PROTEASE
1sp4:B (CYS148) to (MET250) CRYSTAL STRUCTURE OF NS-134 IN COMPLEX WITH BOVINE CATHEPSIN B: A TWO HEADED EPOXYSUCCINYL INHIBITOR EXTENDS ALONG THE WHOLE ACTIVE SITE CLEFT | CATHEPSIN B, EPOXYSUCCINYL-BASED INHIBITORS, INHIBITOR DESIGN, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3iej:A (ALA107) to (GLN219) PYRAZOLE-BASED CATHEPSIN S INHIBITORS WITH ARYLALKYNES AS P1 BINDING ELEMENTS | CATHEPSIN S, DISULFIDE BOND, GLYCOPROTEIN, HYDROLASE, LYSOSOME, POLYMORPHISM, PROTEASE, THIOL PROTEASE, ZYMOGEN
1the:B (TYR148) to (ILE250) CRYSTAL STRUCTURES OF RECOMBINANT RAT CATHEPSIN B AND A CATHEPSIN B- INHIBITOR COMPLEX: IMPLICATIONS FOR STRUCTURE-BASED INHIBITOR DESIGN | THIOL PROTEASE, GLYCOPROTEIN, PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2h7j:A (LYS112) to (ILE217) CRYSTAL STRUCTURE OF CATHEPSIN S IN COMPLEX WITH A NONPEPTIDIC INHIBITOR. | CATHEPSIN S, NONPEPTIDIC, CHLOROMETHYLKETONE, SUBSTRATE ACTIVITY SCREENING, HYDROLASE
2hhn:A (LYS112) to (ILE217) CATHEPSIN S IN COMPLEX WITH NON COVALENT ARYLAMINOETHYL AMIDE. | CATHEPSIN S, NONCOVALENT, INHIBITION, ARYLAMINOETHYL AMIDE, PROTEASE, HYDROLASE
1huc:B (TYR148) to (ILE250) THE REFINED 2.15 ANGSTROMS X-RAY CRYSTAL STRUCTURE OF HUMAN LIVER CATHEPSIN B: THE STRUCTURAL BASIS FOR ITS SPECIFICITY | THIOL PROTEASE
1ito:A (SER150) to (MET250) CRYSTAL STRUCTURE ANALYSIS OF BOVINE SPLEEN CATHEPSIN B- E64C COMPLEX | CATHEPSIN B, CYSTEINE PROTEASE, E64C, HYDROLASE
2ipp:B (TYR148) to (ILE250) CRYSTAL STRUCTURE OF THE TETRAGONAL FORM OF HUMAN LIVER CATHEPSIN B | CATHEPSIN, CYSTEINE PROTEINASE, HYDROLASE
4n8w:A (GLY109) to (MET215) CATHEPSIN K - CHONDROITIN SULFATE COMPLEX | COLLAGINASE, GLYCOSAMINOGLYCAN, HYDROLASE
3k9m:A (LYS144) to (ILE250) CATHEPSIN B IN COMPLEX WITH STEFIN A | DISULFIDE BOND, GLYCOPROTEIN, LYSOSOME, PROTEASE, THIOL PROTEASE, ZYMOGEN, THIOL PROTEASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1mir:A (TYR148) to (ILE250) RAT PROCATHEPSIN B | HYDROLASE, THIOL PROTEASE, CYSTEINE PROTEASE
1mir:B (TYR148) to (ILE250) RAT PROCATHEPSIN B | HYDROLASE, THIOL PROTEASE, CYSTEINE PROTEASE
4p6e:A (LYS112) to (ILE217) CRYSTAL STRUCTURE OF HUMAN CATHEPSIN S BOUND TO A NON-COVALENT INHIBITOR | CYSTEINE PROTEASE, CATHEPSIN S, INHIBITOR, NON-COVALENT
4p6e:B (ALA107) to (ILE217) CRYSTAL STRUCTURE OF HUMAN CATHEPSIN S BOUND TO A NON-COVALENT INHIBITOR | CYSTEINE PROTEASE, CATHEPSIN S, INHIBITOR, NON-COVALENT
3kwb:X (GLY1109) to (MET1215) STRUCTURE OF CATK COVALENTLY BOUND TO A DIOXO-TRIAZINE INHIBITOR | COVALENT BOND, CYS 25, THIOIMIDATE, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, HYDROLASE, LYSOSOME, PROTEASE, THIOL PROTEASE, ZYMOGEN
3lfy:C (GLY109) to (ASN212) CTD OF TAROCYSTATIN IN COMPLEX WITH PAPAIN | CYSTATIN, TAROCYSTATIN, CECPI, PAPAIN, PHYTOCYSTATIN, HYDROLASE
4qrg:B (ALA211) to (PRO316) CRYSTAL STRUCTURE OF I86L MUTANT OF PAPAIN | PROTEASE, ZYMOGEN, HYDROLASE
3mor:A (TRP232) to (ALA336) CRYSTAL STRUCTURE OF CATHEPSIN B FROM TRYPANOSOMA BRUCEI | THIOL PROTEASE, HYDROLASE
4bpv:B (SER234) to (ILE340) MOUSE CATHEPSIN S WITH COVALENT LIGAND | HYDROLASE, CYSTEINE PROTEASE, COVALENT LIGAND
4bpv:D (ALA230) to (ILE340) MOUSE CATHEPSIN S WITH COVALENT LIGAND | HYDROLASE, CYSTEINE PROTEASE, COVALENT LIGAND
4bqv:E (ARG235) to (ILE340) MOUSE CATHEPSIN S WITH COVALENT LIGAND | HYDROLASE, CYSTEINE PROTEASE
4bqv:G (ARG235) to (ILE340) MOUSE CATHEPSIN S WITH COVALENT LIGAND | HYDROLASE, CYSTEINE PROTEASE
3n4c:B (SER111) to (PRO215) 6-PHENYL-1H-IMIDAZO[4,5-C]PYRIDINE-4-CARBONITRILE AS CATHEPSIN S INHIBITORS | CATHEPSIN S, COVALENT INHIBITOR, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3cbj:A (LYS144) to (ILE250) CHAGASIN-CATHEPSIN B COMPLEX | CHAGASIN, CATHEPSIN B, OCCLUDING LOOP, CHAGAS DISEASE, GLYCOPROTEIN, HYDROLASE, LYSOSOME, PROTEASE, THIOL PROTEASE, ZYMOGEN, CYTOPLASMIC VESICLE, PROTEASE INHIBITOR, THIOL PROTEASE INHIBITOR, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3cbk:A (TYR148) to (GLN255) CHAGASIN-CATHEPSIN B | CHAGASIN, CATHEPSIN B, OCCLUDING LOOP, CHAGAS DISEASE, GLYCOPROTEIN, HYDROLASE, LYSOSOME, PROTEASE, THIOL PROTEASE, ZYMOGEN, CYTOPLASMIC VESICLE, PROTEASE INHIBITOR, THIOL PROTEASE INHIBITOR, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3ch2:X (TYR703) to (PHE820) CRYSTAL STRUCTURE ANALYSIS OF SERA5E FROM PLASMODIUM FALCIPARUM | CYSTEINE PROTEASE, PAPAIN FAMILY, GLYCOPROTEIN, HYDROLASE, MALARIA, THIOL PROTEASE, VACUOLE
3ch3:X (TYR703) to (PHE820) CRYSTAL STRUCTURE ANALYSIS OF SERA5E FROM PLASMODIUM FALCIPARUM | CYSTEINE PROTEASE, PAPAIN FAMILY, GLYCOPROTEIN, HYDROLASE, MALARIA, THIOL PROTEASE, VACUOLE
5fpw:A (ALA209) to (PRO311) PROCATHEPSIN B S9 FROM TRYPANOSOMA CONGOLENSE | HYDROLASE, PRO CATHEPSIN B, TRYPANOSOMA CONGOLENSE, TRYPANOSOME
5fpw:B (ALA1209) to (SER1314) PROCATHEPSIN B S9 FROM TRYPANOSOMA CONGOLENSE | HYDROLASE, PRO CATHEPSIN B, TRYPANOSOMA CONGOLENSE, TRYPANOSOME
5fpw:C (ALA2209) to (PRO2311) PROCATHEPSIN B S9 FROM TRYPANOSOMA CONGOLENSE | HYDROLASE, PRO CATHEPSIN B, TRYPANOSOMA CONGOLENSE, TRYPANOSOME
3pbh:A (TYR148) to (ILE250) REFINED CRYSTAL STRUCTURE OF HUMAN PROCATHEPSIN B AT 2.5 ANGSTROM RESOLUTION | THIOL PROTEASE, CATHEPSIN B, CYSTEINE PROTEASE, PROENZYME, CRYSTAL STRUCTURE, PAPAIN
1atk:A (ALA104) to (MET215) CRYSTAL STRUCTURE OF THE CYSTEINE PROTEASE HUMAN CATHEPSIN K IN COMPLEX WITH THE COVALENT INHIBITOR E-64 | HYDROLASE, SULFHYDRYL PROTEINASE
4hwy:A (TRP232) to (ASN338) TRYPANOSOMA BRUCEI PROCATHEPSIN B SOLVED FROM 40 FS FREE-ELECTRON LASER PULSE DATA BY SERIAL FEMTOSECOND X-RAY CRYSTALLOGRAPHY | PAPAIN FOLD, LYSOSOMAL CYSTEINE PROTEASE, HYDROLASE
1cpj:A (TYR148) to (ILE250) CRYSTAL STRUCTURES OF RECOMBINANT RAT CATHEPSIN B AND A CATHEPSIN B-INHIBITOR COMPLEX: IMPLICATIONS FOR STRUCTURE- BASED INHIBITOR DESIGN | THIOL PROTEASE, HYDROLASE
1cpj:B (TYR148) to (ILE250) CRYSTAL STRUCTURES OF RECOMBINANT RAT CATHEPSIN B AND A CATHEPSIN B-INHIBITOR COMPLEX: IMPLICATIONS FOR STRUCTURE- BASED INHIBITOR DESIGN | THIOL PROTEASE, HYDROLASE
1dki:D (HIS158) to (VAL249) CRYSTAL STRUCTURE OF THE ZYMOGEN FORM OF STREPTOCOCCAL PYROGENIC EXOTOXIN B ACTIVE SITE (C47S) MUTANT | ZYMOGEN, CYSTEINE PROTEASE, PAPAIN-LIKE, TOXIN
2dca:A (SER150) to (MET250) X-RAY CRYSTAL STRUCTURE ANALYSIS OF BOVINE SPLEEN CATHEPSIN B-CA075 COMPLEX | CATHEPSIN B, CYSTEINE PROTEASE, CA075, HYDROLASE, EC 3.4.22.1
3h8b:E (GLY111) to (VAL220) A COMBINED CRYSTALLOGRAPHIC AND MOLECULAR DYNAMICS STUDY OF CATHEPSIN- L RETRO-BINDING INHIBITORS(COMPOUND 9) | CYSTEINE PROTEASES, CATHEPSIN L, DISULFIDE BOND, GLYCOPROTEIN, HYDROLASE, LYSOSOME, PROTEASE, THIOL PROTEASE, ZYMOGEN
3h8b:F (GLY111) to (VAL220) A COMBINED CRYSTALLOGRAPHIC AND MOLECULAR DYNAMICS STUDY OF CATHEPSIN- L RETRO-BINDING INHIBITORS(COMPOUND 9) | CYSTEINE PROTEASES, CATHEPSIN L, DISULFIDE BOND, GLYCOPROTEIN, HYDROLASE, LYSOSOME, PROTEASE, THIOL PROTEASE, ZYMOGEN
2ftd:B (GLY109) to (MET215) CRYSTAL STRUCTURE OF CATHEPSIN K COMPLEXED WITH 7-METHYL- SUBSTITUTED AZEPAN-3-ONE COMPOUND | HYDROLASE, SULFHYDRYL PROTEINASE
1u9v:A (GLY109) to (MET215) CRYSTAL STRUCTURE OF THE CYSTEINE PROTEASE HUMAN CATHEPSIN K IN COMPLEX WITH THE COVALENT INHIBITOR NVP-ABE854 | HYDROLASE, SULFHYDRYL PROTEINASE
3kfq:B (THR110) to (VAL221) UNREDUCED CATHEPSIN V IN COMPLEX WITH STEFIN A | PAPAIN-LIKE CYSTEINE PROTEASE, CATHEPSIN, PROTEASE-INHIBITOR COMPLEX, HYDROLASE, LYSOSOME, PROTEASE, THIOL PROTEASE, ZYMOGEN, PROTEASE INHIBITOR, THIOL PROTEASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3bpf:D (LYS122) to (PRO238) CRYSTAL STRUCTURE OF FALCIPAIN-2 WITH ITS INHIBITOR, E64 | FALCIPAIN, MALARIA, CYSTEINE PROTEASE, HYDROLASE, THIOL PROTEASE
3ovx:B (LYS112) to (ILE217) CATHEPSIN S IN COMPLEX WITH A COVALENT INHIBITOR WITH AN ALDEHYDE WARHEAD | CATHEPSIN S, HYDROLASE, COVALENT INHIBITOR, ALDEHYDE WARHEAD, LIGAND IS COVALENTLY BOUND TO CYS25, LYSOSOMEAL PROTEIN, HYDROLASE- HYDROLASE INHIBITOR COMPLEX