4wb5:A (GLY66) to (ASP161) CRYSTAL STRUCTURE OF HUMAN CAMP-DEPENDENT PROTEIN KINASE A (CATALYTIC ALPHA SUBUNIT) | CATALYSIS, PROTEIN KINASE, ADENOSINE TRIPHOSPHATE, PHOSPHORYLATION
4wb8:A (GLY66) to (ASP161) CRYSTAL STRUCTURE OF HUMAN CAMP-DEPENDENT PROTEIN KINASE A (CATALYTIC ALPHA SUBUNIT), EXON 1 DELETION | CATALYSIS, PROTEIN KINASE, ADENOSINE TRIPHOSPHATE, PHOSPHORYLATION
3e87:A (ARG176) to (TYR255) CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF AKT2 IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS | AKT2, KINASE, GSK3 BETA, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
3e87:B (ARG176) to (TYR255) CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF AKT2 IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS | AKT2, KINASE, GSK3 BETA, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
3e8c:B (GLY66) to (ASP161) CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS | PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, PROTEIN KINASE INHIBITOR
3e8c:C (GLY66) to (ASP161) CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS | PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, PROTEIN KINASE INHIBITOR
3e8c:E (GLY66) to (ASP161) CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS | PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, PROTEIN KINASE INHIBITOR
3e8e:A (GLY66) to (ASP161) CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS | PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3e8e:B (GLY66) to (ASP161) CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS | PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3e8e:P (GLY66) to (TYR146) CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS | PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4gu6:A (VAL451) to (SER539) FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH N-{3-[(5-CYANO- 2-PHENYL-1H-PYRROLO[2,3-B]PYRIDIN-4-YLAMINO)- METHYL]-PYRIDIN-2-YL}- N-METHYL-METHANESULFONAMIDE | PROTEIN TYROSINE KINASE, ATP BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gv1:A (GLY173) to (ASN269) PKB ALPHA IN COMPLEX WITH AZD5363 | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2oh0:E (GLY66) to (TYR146) CRYSTAL STRUCTURE OF PROTEIN KINASE A IN COMPLEX WITH PYRIDINE-PYRAZOLOPYRIDINE BASED INHIBITORS | PROTEIN KINASE A, AKT, TRANSFERASE
4wih:A (GLY67) to (ASP162) CRYSTAL STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE A FROM CRICETULUS GRISEUS | PKA, KINASE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ATP- BINDING, CAMP, NUCLEOTIDE-BINDING
3rwp:A (ARG106) to (GLY200) DISCOVERY OF A NOVEL, POTENT AND SELECTIVE INHIBITOR OF 3- PHOSPHOINOSITIDE DEPENDENT KINASE (PDK1) | KINASE DOMAIN, TRANSFERASE, PHOSPHOSERINE: SEP, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4wot:A (GLN115) to (GLY209) ROCK2 IN COMPLEX WITH 1426382-07-1 | TRANSFERASE
4wot:B (GLN115) to (GLY209) ROCK2 IN COMPLEX WITH 1426382-07-1 | TRANSFERASE
4wot:C (LYS116) to (GLY209) ROCK2 IN COMPLEX WITH 1426382-07-1 | TRANSFERASE
4wot:D (GLN115) to (GLY209) ROCK2 IN COMPLEX WITH 1426382-07-1 | TRANSFERASE
2bfx:B (LYS116) to (LYS211) MECHANISM OF AURORA-B ACTIVATION BY INCENP AND INHIBITION BY HESPERADIN. | TRANSFERASE, KINASE, MITOSIS, INHIBITION, TRANSFERASE COMPLEX
2biy:A (SER105) to (GLY200) STRUCTURE OF PDK1-S241A MUTANT KINASE DOMAIN | AGC KINASE, AC-HELIX, ATP-BINDING, PHOSPHORYLATION, PHOSPHOINOSITIDE DEPENDENT PROTEIN KINASE, PI3-KINASE SIGNALLING, PIF-POCKET, PKA, PKB, T-LOOP MUTANT, SERINE- THREONINE-PROTEIN KINASE, TRANSFERASE
2pe0:A (SER105) to (GLY200) CRYSTAL STRUCTURE OF HUMAN PHOSPHOINOSITIDE-DEPENDENT PROTEIN KINASE 1 (PDK1) 5-HYDROXY-3-[1-(1H-PYRROL-2-YL)-ETH-(Z)-YLIDENE]-1,3-DIHYDRO- INDOL-2-ONE COMPLEX | PROTEIN INHIBITOR COMPLEX, SERINE KINASE, TRANSFERASE
2pe2:A (ARG106) to (GLY200) CRYSTAL STRUCTURE OF HUMAN PHOSPHOINOSITIDE-DEPENDENT PROTEIN KINASE 1 (PDK1) 3-{5-[2-OXO-5-UREIDO-1,2-DIHYDRO-INDOL-(3Z)-YLIDENEMETHYL]-1H- PYRROL-3-YL}-N-(2-PIPERIDIN-1-YL-ETHYL)-BENZAMIDE COMPLEX | PROTEIN INHIBITOR COMPLEX, SERINE KINASE, TRANSFERASE
4hpt:E (GLY66) to (ASP161) CRYSTAL STRUCTURE OF THE CATALYTIC SUBUNIT OF CAMP-DEPENDENT PROTEIN KINASE DISPLAYING COMPLETE PHOSPHORYL TRANSFER OF AMP-PNP ONTO A SUBSTRATE PEPTIDE | PROTEIN KINASE, PHOSPHOTRANSFERASE, REGULATORY SUBUNITS, PKI, MAGNESIUM, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3sc1:A (SER105) to (GLY200) NOVEL ISOQUINOLONE PDK1 INHIBITORS DISCOVERED THROUGH FRAGMENT-BASED LEAD DISCOVERY | KINASE DOMAIN, PHOSPHOSERINE, SEP, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3fe3:A (ARG80) to (ARG173) CRYSTAL STRUCTURE OF THE KINASE MARK3/PAR-1: T211A-S215A DOUBLE MUTANT | SERINE/THREONINE PROTEIN KINASE; MARK;PAR-1; KIN1; UBA DOMAIN;C- TAK1;P78;MARK3, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3fhi:A (GLY66) to (ASP161) CRYSTAL STRUCTURE OF A COMPLEX BETWEEN THE CATALYTIC AND REGULATORY (RI{ALPHA}) SUBUNITS OF PKA | CAMP, CAMP DEPENDENT PROTEIN KINASE, PROTEIN-PROTEIN COMPLEX, AMP- PNP, PROTEIN KINASE REGULATION, NUCLEOTIDE BINDING, PROTEIN KINASE ACTIVITY, PROTEIN SERINE/THREONINE KINASE ACTIVITY, CAMP-DEPENDENT PROTEIN KINASE ACTIVITY, PROTEIN BINDING, ATP BINDING, KINASE ACTIVITY, TRANSFERASE ACTIVITY, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, CAMP-BINDING
1cdk:B (ASN67) to (ASP161) CAMP-DEPENDENT PROTEIN KINASE CATALYTIC SUBUNIT (E.C.2.7.1.37) (PROTEIN KINASE A) COMPLEXED WITH PROTEIN KINASE INHIBITOR PEPTIDE FRAGMENT 5-24 (PKI(5-24) ISOELECTRIC VARIANT CA) AND MN2+ ADENYLYL IMIDODIPHOSPHATE (MNAMP-PNP) AT PH 5.6 AND 7C AND 4C | COMPLEX (TRANSFERASE-INHIBITOR), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1oky:A (ARG106) to (GLY200) STRUCTURE OF HUMAN PDK1 KINASE DOMAIN IN COMPLEX WITH STAUROSPORINE | PROTEIN KINASE, PKB, PDK1, STAUROSPORINE, TRANSFERASE
1okz:A (SER105) to (GLY200) STRUCTURE OF HUMAN PDK1 KINASE DOMAIN IN COMPLEX WITH UCN-01 | PROTEIN KINASE, PKB, PDK1, UCN-01, 7-HYDROXY STAUROSPORINE, INHIBITOR, TRANSFERASE, ATP-BINDING, PHOSPHORYLATION
1ol7:A (LYS156) to (ARG251) STRUCTURE OF HUMAN AURORA-A 122-403 PHOSPHORYLATED ON THR287, THR288 | KINASE, CELL CYCLE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION
2c47:A (GLU70) to (SER160) STRUCTURE OF CASEIN KINASE 1 GAMMA 2 | SERINE/THREONINE KINASE, ACTIN CYTOSKELETON ORGANISATION, ATP-BINDING, TRANSFERASE, WNT SIGNALING PATHWAY
2c6e:A (ALA159) to (ARG250) AURORA A KINASE ACTIVATED MUTANT (T287D) IN COMPLEX WITH A 5-AMINOPYRIMIDINYL QUINAZOLINE INHIBITOR | TRANSFERASE/INHIBITOR, TRANSFERASE/INHIBITOR COMPLEX, AURORA, KINASE, CANCER, ATP-BINDING, CELL CYCLE, NUCLEOTIDE- BINDING, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4iaf:A (GLY66) to (TYR146) ROOM TEMPERATURE X-RAY STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A IN COMPLEX WITH HIGH MG2+ CONCENTRATION, ADP AND PHOSPHORYLATED PEPTIDE PSP20 | KINASE ENZYME, PHOSPHOTRANSFER, PHOSPHORYLATION, TRANSFERASE-PEPTIDE COMPLEX
4iak:A (GLY66) to (ASP161) LOW TEMPERATURE X-RAY STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A IN COMPLEX WITH HIGH SR2+ CONCENTRATION, ADP AND PHOSPHORYLATED PEPTIDE PSP20 | KINASE ENZYME, PHOSPHOTRANSFER, PHOSPHORYLATION, TRANSFERASE-PEPTIDE COMPLEX
4iay:A (GLY66) to (ASP161) ROOM TEMPERATURE X-RAY STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A IN COMPLEX WITH HIGH SR2+ CONCENTRATION, ADP AND PHOSPHORYLATED PEPTIDE PSP20 | KINASE ENZYME, PHOSPHOTRANSFER, PHOSPHORYLATION, TRANSFERASE-PEPTIDE COMPLEX
4iaz:A (GLY66) to (ASP161) STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A IN COMPLEX WITH HIGH BA2+ CONCENTRATION, ADP AND PHOSPHORYLATED PEPTIDE PSP20 | KINASE ENZYME, PHOSPHOTRANSFER, PHOSPHORYLATED, TRANSFERASE-PEPTIDE COMPLEX
4ib1:A (GLY66) to (ASP161) STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A IN COMPLEX WITH HIGH K+ CONCENTRATION, ADP AND PHOSPHORYLATED PEPTIDE PSP20 | KINASE ENZYME, PHOSPHOTRANSFER, PHOSPHORYLATED, TRANSFERASE-PEPTIDE COMPLEX
2qcs:A (GLY66) to (ASP161) A COMPLEX STRUCTURE BETWEEN THE CATALYTIC AND REGULATORY SUBUNIT OF PROTEIN KINASE A THAT REPRESENTS THE INHIBITED STATE | CYCLIC ADENOSINE MONOPHOSPHATE, CAMP-DEPENDENT PROTEIN KINASE, PKA HOLOENZYME, CYCLIC NUCLEOTIDE BINDING DOMAIN, PROTEIN-PROTEIN INTERACTION, CONFORMATIONAL CHANGE, PROTEIN BINDING, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4ij9:A (ASN67) to (ASP161) BOVINE PKA C-ALPHA IN COMPLEX WITH 2-[[5-(4-PYRIDYL)-1H-1,2,4-TRIAZOL- 3-YL]SULFANYL]-1-(2-THIOPHENYL)ETHANONE | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4xx9:A (SER105) to (GLY200) CRYSTAL STRUCTURE OF PDK1 IN COMPLEX WITH ATP AND THE PIF-POCKET LIGAND RF4 | PROTEIN KINASE, ALLOSTERY, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3tac:A (GLY35) to (ASN136) CRYSTAL STRUCTURE OF THE LIPRIN-ALPHA/CASK COMPLEX | TRANSFERASE-PROTEIN BINDING COMPLEX
3gni:B (GLU95) to (GLY190) STRUCTURE OF STRAD AND MO25 | KINASE FOLD, PSEUDOKINASE, ALPHA HELICAL REPEAT PROTEIN, ADAPTOR PROTEIN, ATP-BINDING, CELL CYCLE, KINASE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE, METAL BINDING PROTEIN- TRANSFERASE COMPLEX, SIGNALING PROTEIN-SIGNALING PROTEIN COMPLEX
4j8m:A (ALA160) to (TYR246) AURORA A IN COMPLEX WITH CD532 | AURORA A, TYPE II, KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jaj:A (ALA160) to (ARG251) CRYSTAL STRUCTURE OF AURORA KINASE A IN COMPLEX WITH BENZO[C][1, 8]NAPHTHYRIDIN-6(5H)-ONE | KINASE INHIBITOR COMPLEX, ATP-BINDING, CELL CYCLE,CYTOPLASM, CYTOSKELETON, NUCLEOTIDE-BINDING,PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE, PROTEIN KINASE-LIKE CYTOPLASM, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jbp:A (ALA160) to (ARG251) NOVEL AURORA KINASE INHIBITORS REVEAL MECHANISMS OF HURP IN NUCLEATION OF CENTROSOMAL AND KINETOCHORE MICROTUBULES | AURORA KINASE INHIBITORS, HURP, MITOTIC SPINDLE, TRANSFERASE
4jbo:A (ALA160) to (ARG251) NOVEL AURORA KINASE INHIBITORS REVEAL MECHANISMS OF HURP IN NUCLEATION OF CENTROSOMAL AND KINETOCHORE MICROTUBULES | AURORA KINASE INHIBITORS, HURP, MITOTIC SPINDLE, TRANSFERASE
1q61:A (GLY66) to (TYR146) PKA TRIPLE MUTANT MODEL OF PKB | PKB-MODEL, RESTORATION OF ATP-SITE, POINT MUTATION, TRANSFERASE/TRANSFERASE INHIBITOR COMPLEX
3tku:A (GLU99) to (HIS195) MRCK BETA IN COMPLEX WITH FASUDIL | PROTEIN KINASE, SERINE THREONINE KINASE, MRCK, MRCK BETA, CD BINDING PROTEIN KINASE BETA, FASUDIL, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3tnp:C (GLY66) to (ASP161) STRUCTURE AND ALLOSTERY OF THE PKA RIIB TETRAMERIC HOLOENZYME | PKA RIIB TETRAMERIC HOLOENZYME, TRANSFERASE
3tnp:F (GLY66) to (ASP161) STRUCTURE AND ALLOSTERY OF THE PKA RIIB TETRAMERIC HOLOENZYME | PKA RIIB TETRAMERIC HOLOENZYME, TRANSFERASE
2dwb:A (LEU159) to (ARG251) AURORA-A KINASE COMPLEXED WITH AMPPNP | AURORA, PROTEIN KINASE, ATP-BINDING, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, TRANSFERASE
3h0z:A (ALA160) to (ALA243) AURORA A IN COMPLEX WITH A BISANILINOPYRIMIDINE | PROTEIN:INHIBITOR COMPLEX AURORA-A, CELL CYCLE, SERINE/THREONINE, PROTEIN KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3h10:B (ALA160) to (ARG251) AURORA A INHIBITOR COMPLEX | PROTEIN:INHIBITOR COMPLEX AURORA-A, CELL CYCLE, SERINE/THREONINE, PROTEIN KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3tv7:A (ARG99) to (MET192) HUMAN RHO-ASSOCIATED PROTEIN KINASE 1 (ROCK 1) IN COMPLEX WITH RKI1342 | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3tv7:C (ARG99) to (MET192) HUMAN RHO-ASSOCIATED PROTEIN KINASE 1 (ROCK 1) IN COMPLEX WITH RKI1342 | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3txo:A (GLY378) to (GLY474) PKC ETA KINASE IN COMPLEX WITH A NAPHTHYRIDINE | KINASE, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3h9o:A (SER105) to (GLY200) PHOSPHOINOSITIDE-DEPENDENT PROTEIN KINASE 1 (PDK-1) IN COMPLEX WITH COMPOUND 9 | PDK-1, KINASE, PROTEIN STRUCTURE, X-RAY CRYSATLLOGRAPHY, ALTERNATIVE SPLICING, ATP-BINDING, CYTOPLASM, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
2uw3:A (GLY66) to (TYR146) STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH 5-METHYL-4- PHENYL-1H-PYRAZOLE | TRANSFERASE/INHIBITOR, CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION, TRANSFERASE/INHIBITOR COMPLEX
2uw9:A (GLY175) to (ASP270) STRUCTURE OF PKB-BETA (AKT2) COMPLEXED WITH 4-(4-CHLORO- PHENYL)-4-(4-(1H-PYRAZOL-4-YL)-PHENYL)-PIPERIDINE | TRANSFERASE/INHIBITOR, TRANSFERASE/INHIBITOR COMPLEX, WNT SIGNALING PATHWAY, SERINE/THREONINE-PROTEIN KINASE, KINASE, TRANSFERASE, ATP-BINDING, PHOSPHORYLATION, NUCLEOTIDE-BINDING, ALTERNATIVE SPLICING
2uzu:E (GLY66) to (ASP161) PKA STRUCTURES OF INDAZOLE-PYRIDINE SERIES OF AKT INHIBITORS | CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, PHOSPHORYLATION, PROTEIN KINASE A, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP- BINDING, AKT INHIBITORS, NUCLEAR PROTEIN
2uzv:A (GLY66) to (ASP161) PKA STRUCTURES OF INDAZOLE-PYRIDINE SERIES OF AKT INHIBITORS | CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, PHOSPHORYLATION, PROTEIN KINASE A, NUCLEOTIDE-BINDING, ATP-BINDING, AKT INHIBITORS, NUCLEAR PROTEIN
4ynz:A (GLN44) to (SER137) STRUCTURE OF THE N-TERMINAL DOMAIN OF SAD | KINASE DOMAIN, UBA DOMAIN, TRANSFERASE
2esm:A (ARG99) to (SER191) CRYSTAL STRUCTURE OF ROCK 1 BOUND TO FASUDIL | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE
2esm:B (ARG99) to (SER191) CRYSTAL STRUCTURE OF ROCK 1 BOUND TO FASUDIL | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE
2etk:A (ARG99) to (SER191) CRYSTAL STRUCTURE OF ROCK 1 BOUND TO HYDROXYFASUDIL | DIMER, DIMERIZATION, KINASE, FASUDIL, HYDROXYFASUDIL, TRANSFERASE
2etk:B (ARG99) to (SER191) CRYSTAL STRUCTURE OF ROCK 1 BOUND TO HYDROXYFASUDIL | DIMER, DIMERIZATION, KINASE, FASUDIL, HYDROXYFASUDIL, TRANSFERASE
2etr:A (ARG99) to (MET192) CRYSTAL STRUCTURE OF ROCK I BOUND TO Y-27632 | DIMERIZATION, DIMER, PHOSPHORYLATION, KINASE, YOSHITOMI, TRANSFERASE
2etr:B (ARG99) to (MET192) CRYSTAL STRUCTURE OF ROCK I BOUND TO Y-27632 | DIMERIZATION, DIMER, PHOSPHORYLATION, KINASE, YOSHITOMI, TRANSFERASE
2v55:A (ARG99) to (MET192) MECHANISM OF MULTI-SITE PHOSPHORYLATION FROM A ROCK-I:RHOE COMPLEX STRUCTURE | SERINE/THREONINE-PROTEIN KINASE, RHOE, ZINC, KINASE, ROCK-I, MEMBRANE, APOPTOSIS, CYTOPLASM, G-PROTEINS, METHYLATION, ZINC-FINGER, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, ATP-BINDING, PRENYLATION, TRANSFERASE, LIPOPROTEIN, MULTI-SITE PHOSPHORYLATION, COILED COIL, GTP-BINDING, POLYMORPHISM, STRESS FIBRES, METAL-BINDING, PHOSPHOPROTEIN, GOLGI APPARATUS
2v55:C (ARG99) to (MET192) MECHANISM OF MULTI-SITE PHOSPHORYLATION FROM A ROCK-I:RHOE COMPLEX STRUCTURE | SERINE/THREONINE-PROTEIN KINASE, RHOE, ZINC, KINASE, ROCK-I, MEMBRANE, APOPTOSIS, CYTOPLASM, G-PROTEINS, METHYLATION, ZINC-FINGER, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, ATP-BINDING, PRENYLATION, TRANSFERASE, LIPOPROTEIN, MULTI-SITE PHOSPHORYLATION, COILED COIL, GTP-BINDING, POLYMORPHISM, STRESS FIBRES, METAL-BINDING, PHOSPHOPROTEIN, GOLGI APPARATUS
1rdq:E (GLY66) to (TYR146) HYDROLYSIS OF ATP IN THE CRYSTAL OF Y204A MUTANT OF CAMP-DEPENDENT PROTEIN KINASE | CAMP-DEPENDENT PROTEIN KINASE,CATALYTIC MECHANISM, ATP HYDROLYSIS, TWO NUCLEOTIDE STATES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1re8:A (GLY66) to (ASP161) CRYSTAL STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE COMPLEXED WITH BALANOL ANALOG 2 | PROTEIN KINASE, NATURAL PRODUCT INHIBITOR, LIGAND BINDING, SPECIFICITY DETERMINANTS, CONFORMATIONAL MALLEABILITY, TRANSFERASE
1rej:A (GLY66) to (ASP161) CRYSTAL STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE COMPLEXED WITH BALANOL ANALOG 1 | PROTEIN KINASE, NATURAL PRODUCT INHIBITOR, LIGAND BINDING, SPECIFICITY DETERMINANTS, CONFORMATIONAL MALLEABILITY, TRANSFERASE
4yur:A (GLY35) to (GLY131) CRYSTAL STRUCTURE OF PLK4 KINASE DOMAIN BOUND TO CENTRINONE | TRANSFERASE, PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yve:A (ARG99) to (MET192) ROCK 1 BOUND TO METHOXYPHENYL THIAZOLE INHIBITOR | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yve:B (ARG99) to (GLY193) ROCK 1 BOUND TO METHOXYPHENYL THIAZOLE INHIBITOR | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yvc:A (ARG99) to (GLY193) ROCK 1 BOUND TO THIAZOLE INHIBITOR | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yvc:B (ARG99) to (GLY193) ROCK 1 BOUND TO THIAZOLE INHIBITOR | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2f2u:A (GLN115) to (GLY209) CRYSTAL STRUCTURE OF THE RHO-KINASE KINASE DOMAIN | ENZYME-INHIBITOR COMPLEX, TRANSFERASE
2f2u:B (LYS116) to (GLY209) CRYSTAL STRUCTURE OF THE RHO-KINASE KINASE DOMAIN | ENZYME-INHIBITOR COMPLEX, TRANSFERASE
4yxr:A (GLY66) to (TYR146) CRYSTAL STRUCTURE OF PKA IN COMPLEX WITH INHIBITOR. | COMPLEX (PHOSPHOTRANSFERASE-INHIBITOR) COMPLEX, TRANSFERASE
4yxs:A (GLY66) to (TYR146) CAMP-DEPENDENT PROTEIN KINASE PKA CATALYTIC SUBUNIT WITH PKI-5-24 | ATP-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, CAMP, PROTEIN KINASE INHIBITOR, TRANSFERASE-IN COMPLEX, TRANSFERASE-INHIBITOR COMPLEX
2f7e:E (GLY66) to (ASP161) PKA COMPLEXED WITH (S)-2-(1H-INDOL-3-YL)-1-(5-ISOQUINOLIN-6- YL-PYRIDIN-3-YLOXYMETHYL-ETYLAMINE | PROTEIN KINASE A, AKT INHIBITORS, TRANSFERASE
2vd5:A (GLY94) to (GLY190) STRUCTURE OF HUMAN MYOTONIC DYSTROPHY PROTEIN KINASE IN COMPLEX WITH THE BISINDOYLMALEIDE INHIBITOR BIM VIII | SERINE/THREONINE-PROTEIN KINASE, KINASE, TRANSFERASE, ATP-BINDING, NUCLEOTIDE-BINDING, CARDIAC CONTRACTILITY, MUSCLE DIFFERENTIATION
2vd5:B (GLY94) to (GLY190) STRUCTURE OF HUMAN MYOTONIC DYSTROPHY PROTEIN KINASE IN COMPLEX WITH THE BISINDOYLMALEIDE INHIBITOR BIM VIII | SERINE/THREONINE-PROTEIN KINASE, KINASE, TRANSFERASE, ATP-BINDING, NUCLEOTIDE-BINDING, CARDIAC CONTRACTILITY, MUSCLE DIFFERENTIATION
2f7x:E (GLY66) to (TYR146) PROTEIN KINASE A BOUND TO (S)-2-(1H-INDOL-3-YL)-1-[5-((E)-2- PYRIDIN-4-YL-VINYL)-PYRIDIN-3-YLOXYMETHYL]-ETHYLAMINE | PROTEIN KINASE A, AKT INHIBITORS, TRANSFERASE
3unz:A (LEU159) to (ARG251) AURORA A IN COMPLEX WITH RPM1679 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3unz:B (LEU159) to (ARG251) AURORA A IN COMPLEX WITH RPM1679 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uoh:A (LEU159) to (ARG251) AURORA A IN COMPLEX WITH RPM1722 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uoh:B (LEU159) to (ARG251) AURORA A IN COMPLEX WITH RPM1722 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uoj:A (ALA160) to (ARG251) AURORA A IN COMPLEX WITH RPM1715 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uoj:B (ALA160) to (ARG251) AURORA A IN COMPLEX WITH RPM1715 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3up2:A (ALA160) to (ARG251) AURORA A IN COMPLEX WITH RPM1686 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-IN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2vnw:A (GLY66) to (TYR146) STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH (1-(9H-PURIN-6- YL)PIPERIDIN-4-YL)METHANAMINE | TRANSFERASE, LIPOPROTEIN, ATP-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, CAMP, KINASE, NUCLEUS, MYRISTATE, CYTOPLASM
2vo0:A (GLY66) to (ASP161) STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH C-(4-(4- CHLOROPHENYL)-1-(7H-PYRROLO(2,3-D)PYRIMIDIN-4-YL)PIPERIDIN- 4-YL)METHYLAMINE | TRANSFERASE, LIPOPROTEIN, ATP-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, CAMP, KINASE, NUCLEUS, MYRISTATE, CYTOPLASM
2vo3:A (GLY66) to (TYR146) STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH C-(4-(4- CHLOROPHENYL)-1-(7H-PYRROLO(2,3-D)PYRIMIDIN-4-YL)PIPERIDIN- 4-YL)METHYLAMINE | TRANSFERASE, LIPOPROTEIN, ATP-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, CAMP, KINASE, NUCLEUS, MYRISTATE, CYTOPLASM
2vo7:A (GLY66) to (TYR146) STRUCTURE OF PKA COMPLEXED WITH 4-(4-CHLOROBENZYL)-1-(7H- PYRROLO(2,3-D)PYRIMIDIN-4-YL)PIPERIDIN-4-YLAMINE | TRANSFERASE, LIPOPROTEIN, ATP-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, CAMP, KINASE, NUCLEUS, MYRISTATE, CYTOPLASM
3vap:A (ALA160) to (ARG251) SYNTHESIS AND SAR STUDIES OF IMIDAZO-[1,2-A]-PYRAZINE AURORA KINASE INHIBITORS WITH IMPROVED OFF TARGET KINASE SELECTIVITY | KINASE, CELL CYCLE, INHIBITOR, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4zhx:A (GLY39) to (MET134) NOVEL BINDING SITE FOR ALLOSTERIC ACTIVATION OF AMPK | TRANSFERASE, SERINE/THREONINE KINASE, ALLOSTERIC ACTIVATION, NUCLEOTIDE-BINDING
1sve:A (ASN67) to (ASP161) CRYSTAL STRUCTURE OF PROTEIN KINASE A IN COMPLEX WITH AZEPANE DERIVATIVE 1 | KINASE-INHIBITOR-COMPLEX, SERINE/THREONINE-PROTEIN KINASE, BALANOL DERIVATIVE, TRANSFERASE
2gfc:A (GLY66) to (TYR146) CAMP-DEPENDENT PROTEIN KINASE PKA CATALYTIC SUBUNIT WITH PKI-5-24 | BINARY COMPLEX, PEPTIDE INHIBITOR, TRANSFERASE
4l00:B (VAL619) to (ASP709) CRYSTAL STRUCTURE OF THE APO JAK1 PSEUDOKINASE DOMAIN | KINASE DOMAIN FOLD, REGULATORY, TRANSFERASE
1h1w:A (SER105) to (GLY200) HIGH RESOLUTION CRYSTAL STRUCTURE OF THE HUMAN PDK1 CATALYTIC DOMAIN | TRANSFERASE, PHOSPHOINOSITIDE DEPENDENT PROTEIN KINASE, PKA, AGC KINASE ACTIVATION, PIF-POCKET, PI3-KINASE SIGNALLING, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING
4l3j:A (GLY94) to (GLY190) CRYSTAL STRUCTURES OF HUMAN P70S6K1 KINASE DOMAIN | PROTEIN KINASE, TRANSFERASE
4l3l:A (GLY94) to (GLY190) CRYSTAL STRUCTURES OF HUMAN P70S6K1 KINASE DOMAIN (ZINC ANOMALOUS) | PROTEIN KINASE, TRANSFERASE
4l42:A (LYS95) to (GLY190) CRYSTAL STRUCTURES OF HUMAN P70S6K1-PIF | PROTEIN KINASE, TRANSFERASE
4l43:A (LYS95) to (GLY190) CRYSTAL STRUCTURES OF HUMAN P70S6K1-T389A (FORM I) | PROTEIN KINASE, TRANSFERASE
4l44:A (GLY94) to (GLY190) CRYSTAL STRUCTURES OF HUMAN P70S6K1-T389A (FORM II) | PROTEIN KINASE, TRANSFERASE
4l45:A (GLY94) to (GLY190) CRYSTAL STRUCTURES OF HUMAN P70S6K1-T389E | PROTEIN KINASE, TRANSFERASE
4l46:A (LYS95) to (GLY190) CRYSTAL STRUCTURES OF HUMAN P70S6K1-WT | PROTEIN KINASE, TRANSFERASE
2gng:A (GLY66) to (ASP161) PROTEIN KINASE A FIVEFOLD MUTANT MODEL OF RHO-KINASE | PKA, MUTANT, RHO-KINASE, SURROGATE, INHIBITOR, TRANSFERASE/TRANSFERASE INHIBITOR COMPLEX
4l6q:A (GLN115) to (GLY209) ROCK2 IN COMPLEX WITH BENZOXABOROLE | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2w1d:A (ALA160) to (ARG251) STRUCTURE DETERMINATION OF AURORA KINASE IN COMPLEX WITH INHIBITOR | NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, POLYMORPHISM, PHOSPHOPROTEIN, KINASE, CANCER, AURORA, INHIBITOR, CELL CYCLE
2w1e:A (LYS156) to (ARG251) STRUCTURE DETERMINATION OF AURORA KINASE IN COMPLEX WITH INHIBITOR | NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, POLYMORPHISM, PHOSPHOPROTEIN, KINASE, CANCER, AURORA, INHIBITOR, CELL CYCLE
2h9v:A (GLN115) to (GLY209) STRUCTURAL BASIS FOR INDUCED-FIT BINDING OF RHO-KINASE TO THE INHIBITOR Y27632 | PROTEIN KINASE-INHIBITOR COMPLEX, TRANSFERASE
3vqh:A (GLY66) to (TYR146) BROMINE SAD PARTIALLY RESOLVES MULTIPLE BINDING MODES FOR PKA INHIBITOR H-89 | PROTEIN-INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3w10:A (LYS156) to (ARG251) AURORA KINASE A COMPLEXED TO PYRAZOLE AMINOQUINOLINE I | KINASE, PYRAZOLE AMINOQUINOLINE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2wtk:E (VAL97) to (GLY190) STRUCTURE OF THE HETEROTRIMERIC LKB1-STRADALPHA-MO25ALPHA COMPLEX | TRANSFERASE-METAL-BINDING PROTEIN COMPLEX, TRANSFERASE METAL-BINDING PROTEIN COMPLEX, KINASE, NUCLEUS, SERINE/THREONINE-PROTEIN KINASE, PSEUDOKINASE, PHOSPHOPROTEIN, SIGNAL TRANSDUCTION, TRANSFERASE, NUCLEOTIDE-BINDING
2i0e:A (ASP365) to (GLY461) STRUCTURE OF CATALYTIC DOMAIN OF HUMAN PROTEIN KINASE C BETA II COMPLEXED WITH A BISINDOLYLMALEIMIDE INHIBITOR | PROTEIN KINASE C BETA II, PROTEIN KINASE C, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE
2i0e:B (ASP365) to (GLY461) STRUCTURE OF CATALYTIC DOMAIN OF HUMAN PROTEIN KINASE C BETA II COMPLEXED WITH A BISINDOLYLMALEIMIDE INHIBITOR | PROTEIN KINASE C BETA II, PROTEIN KINASE C, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE
2wtv:A (ALA160) to (ARG251) AURORA-A INHIBITOR STRUCTURE | KINASE, CELL CYCLE, TRANSFERASE, PHOSPHOPROTEIN
2wtw:A (ALA160) to (ARG251) AURORA-A INHIBITOR STRUCTURE (2ND CRYSTAL FORM) | KINASE, CELL CYCLE, TRANSFERASE, PHOSPHOPROTEIN, PROTEIN KINASE
5aad:A (LYS156) to (ARG251) AURORA A KINASE BOUND TO AN IMIDAZOPYRIDINE INHIBITOR (7A) | TRANSFERASE, AURORA-A, IMIDAZOPYRIDINE, AURORA KINASE, INHIBITOR
2wzj:B (LYS77) to (LYS155) CATALYTIC AND UBA DOMAIN OF KINASE MARK2/(PAR-1) K82R, T208E DOUBLE MUTANT | UBA DOMAIN, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, SIGNALING PROTEIN, S/T PROTEIN KINASE, DIFFERENTIATION, DEVELOPMENTAL PROTEIN
2wzj:D (LYS77) to (PHE170) CATALYTIC AND UBA DOMAIN OF KINASE MARK2/(PAR-1) K82R, T208E DOUBLE MUTANT | UBA DOMAIN, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, SIGNALING PROTEIN, S/T PROTEIN KINASE, DIFFERENTIATION, DEVELOPMENTAL PROTEIN
1uu7:A (SER105) to (GLY200) STRUCTURE OF HUMAN PDK1 KINASE DOMAIN IN COMPLEX WITH BIM-2 | PROTEIN KINASE, PKB, PDK1, INHIBITOR, LY333531, BISINDOLYL MALEIMIDE, BIM-1, DIABETES, CANCER, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE
1uu8:A (SER105) to (GLY200) STRUCTURE OF HUMAN PDK1 KINASE DOMAIN IN COMPLEX WITH BIM-1 | PROTEIN KINASE, PKB, PDK1, INHIBITOR, LY333531, BISINDOLYL MALEIMIDE, BIM-1, DIABETES, CANCER, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE
1uu9:A (SER105) to (GLY200) STRUCTURE OF HUMAN PDK1 KINASE DOMAIN IN COMPLEX WITH BIM-3 | PROTEIN KINASE, PKB, PDK1, INHIBITOR, LY333531, BISINDOLYL MALEIMIDE, BIM-1, DIABETES, CANCER, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE
1uvr:A (ARG106) to (GLY200) STRUCTURE OF HUMAN PDK1 KINASE DOMAIN IN COMPLEX WITH BIM-8 | PROTEIN KINASE, PKB, PDK1, INHIBITOR, LY333531, BISINDOLYL MALEIMIDE, BIM-8, DIABETES, CANCER, TRANSFERASE
3wf8:A (LYS118) to (GLY213) CRYSTAL STRUCTURE OF S6K1 KINASE DOMAIN IN COMPLEX WITH A QUINOLINE DERIVATIVE 2-OXO-2-[(4-SULFAMOYLPHENYL)AMINO]ETHYL 7,8,9,10- TETRAHYDRO-6H-CYCLOHEPTA[B]QUINOLINE-11-CARBOXYLATE | SERINE/THREONINE PROTEIN KINASE DOMAIN, TRANSFERASE, PHOSPHORYLATION, ATP-BINDING, ZINC-BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2x39:A (GLY175) to (ASP270) STRUCTURE OF 4-AMINO-N-(4-CHLOROBENZYL)-1-(7H-PYRROLO(2,3-D) PYRIMIDIN-4-YL)PIPERIDINE-4-CARBOXAMIDE BOUND TO PKB | SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, WNT SIGNALING PATHWAY, KINASE, TRANSFERASE, PHOSPHOPROTEIN
1jbp:E (GLY66) to (ASP161) CRYSTAL STRUCTURE OF THE CATALYTIC SUBUNIT OF CAMP- DEPENDENT PROTEIN KINASE COMPLEXED WITH A SUBSTRATE PEPTIDE, ADP AND DETERGENT | PROTEIN-SUBSTRATE COMPLEX, TRANSFERASE
2xch:A (SER105) to (GLY200) CRYSTAL STRUCTURE OF PDK1 IN COMPLEX WITH A PYRAZOLOQUINAZOLINE INHIBITOR | PI3-KINASE SIGNALLING, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING
1veb:A (GLY66) to (ASP161) CRYSTAL STRUCTURE OF PROTEIN KINASE A IN COMPLEX WITH AZEPANE DERIVATIVE 5 | KINASE-INHIBITOR-COMPLEX, SERINE/THREONINE-PROTEIN KINASE, BALANOL DERIVATIVE, TRANSFERASE
1jlu:E (GLY66) to (ASP161) CRYSTAL STRUCTURE OF THE CATALYTIC SUBUNIT OF CAMP-DEPENDENT PROTEIN KINASE COMPLEXED WITH A PHOSPHORYLATED SUBSTRATE PEPTIDE AND DETERGENT | PROTEIN KINASE-PHOSPHORYLATED SUBSTRATE COMPLEX, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
2j4z:A (ALA160) to (ARG251) STRUCTURE OF AURORA-2 IN COMPLEX WITH PHA-680626 | TRANSFERASE, PHOSPHORYLATION, NUCLEOTIDE-BINDING, KINASE, CELL CYCLE, ATP-BINDING, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, SERINE-THREONINE-PROTEIN KINASE
2xh5:A (GLY175) to (ASP270) STRUCTURE OF 4-(4-TERT-BUTYLBENZYL)-1-(7H-PYRROLO(2,3-D) PYRIMIDIN-4-YL)PIPERIDIN-4-AMINE BOUND TO PKB | SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, WNT SIGNALING PATHWAY, KINASE, TRANSFERASE, PHOSPHOPROTEIN
3x2v:A (ASN67) to (ASP161) MICHAELIS-LIKE COMPLEX OF CAMP-DEPENDENT PROTEIN KINASE CATALYTIC SUBUNIT | MICHAELIS-LIKE COMPLEX, PROTEIN-SUBSTRATE, PKAC-ATPMG2 TERNARY, SER/THR KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-PEPTIDE COMPLEX
3x2w:A (ASN67) to (ASP161) MICHAELIS COMPLEX OF CAMP-DEPENDENT PROTEIN KINASE CATALYTIC SUBUNIT | MICHAELIS COMPLEX, PROTEIN-SUBSTRATE, PKAC-ATPMG2 TERNARY, SER/THR KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-PEPTIDE COMPLEX
2xru:A (LYS156) to (ARG251) AURORA-A T288E COMPLEXED WITH PHA-828300 | NUCLEOTIDE-BINDING, KINASE, CELL CYCLE, TRANSFERASE
2jdo:A (GLY175) to (ASP270) STRUCTURE OF PKB-BETA (AKT2) COMPLEXED WITH ISOQUINOLINE-5- SULFONIC ACID (2-(2-(4-CHLOROBENZYLOXY) ETHYLAMINO)ETHYL) AMIDE | WNT SIGNALING PATHWAY, SERINE/THREONINE-PROTEIN KINASE, KINASE, TRANSFERASE, ATP-BINDING, PHOSPHORYLATION, NUCLEOTIDE-BINDING, ALTERNATIVE SPLICING
2jdr:A (GLY175) to (ASP270) STRUCTURE OF PKB-BETA (AKT2) COMPLEXED WITH THE INHIBITOR A- 443654 | WNT SIGNALING PATHWAY, SERINE/THREONINE-PROTEIN KINASE, KINASE, TRANSFERASE, ATP-BINDING, PHOSPHORYLATION, NUCLEOTIDE-BINDING, ALTERNATIVE SPLICING
2jds:A (GLY66) to (TYR146) STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE COMPLEXED WITH A- 443654 | CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION
2jdt:A (GLY66) to (TYR146) STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH ISOQUINOLINE-5- SULFONIC ACID (2-(2-(4-CHLOROBENZYLOXY) ETHYLAMINO)ETHYL) AMIDE | CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION
2jdv:A (GLY66) to (TYR146) STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH A-443654 | CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION
2jed:A (ASN403) to (GLY491) THE CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF THE PROTEIN KINASE C THETA IN COMPLEX WITH NVP-XAA228 AT 2.32A RESOLUTION. | PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, POLYMORPHISM, METAL-BINDING, ZINC, KINASE, PKC THETA, MAGNESIUM, ZINC-FINGER, ALTERNATIVE SPLICING, PHORBOL-ESTER BINDING
2jed:B (GLN404) to (GLY499) THE CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF THE PROTEIN KINASE C THETA IN COMPLEX WITH NVP-XAA228 AT 2.32A RESOLUTION. | PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, POLYMORPHISM, METAL-BINDING, ZINC, KINASE, PKC THETA, MAGNESIUM, ZINC-FINGER, ALTERNATIVE SPLICING, PHORBOL-ESTER BINDING
3zh8:B (ASP268) to (GLY364) A NOVEL SMALL MOLECULE APKC INHIBITOR | TRANSFERASE, AGC KINASES, CELL POLARITY, CELL MIGRATION
5bx6:A (GLY66) to (TYR146) PKA IN COMPLEX WITH A HALOGENATED PHTHALAZINONE FRAGMENT COMPOUND. | INHIBITOR, PROTEIN KINASE, STRUCTURE-GUIDED, FRAGMENT-BASED, TRANSFERASE
5bx7:A (GLY66) to (TYR146) PKA IN COMPLEX WITH A BENZOTHIOPHENE FRAGMENT COMPOUND. | INHIBITOR, PROTEIN KINASE, STRUCTURE-GUIDED, FRAGMENT-BASED, TRANSFERASE
5byy:A (VAL81) to (GLN177) ERK5 IN COMPLEX WITH SMALL MOLECULE | ERK5 KINASE, KINASE INHIBITOR, PROTEROS BIOSTRUCTURES GMBH, TRANSFERASE
3zo1:A (GLY66) to (ASP161) THE SYNTHESIS AND EVALUATION OF DIAZASPIROCYCLIC PROTEIN KINASE INHIBITORS | TRANSFERASE-INHIBITOR COMPLEX
3zo2:A (GLY66) to (ASP161) THE SYNTHESIS AND EVALUATION OF DIAZASPIROCYCLIC PROTEIN KINASE INHIBITORS | TRANSFERASE-INHIBITOR COMPLEX
3zo3:A (GLY66) to (ASP161) THE SYNTHESIS AND EVALUATION OF DIAZASPIROCYCLIC PROTEIN KINASE INHIBITORS | TRANSFERASE-INHIBITOR COMPLEX
3ztx:A (ALA120) to (LYS211) AURORA KINASE SELECTIVE INHIBITORS IDENTIFIED USING A TAXOL- INDUCED CHECKPOINT SENSITIVITY SCREEN. | TRANSFERASE-CELL CYCLE COMPLEX, TRANSFERASE, TAXOL-INDUCED CHECKPOINT INHIBITOR
4nts:A (GLY66) to (TYR146) APO STRUCTURE OF THE CATALYTIC SUBUNIT OF CAMP-DEPENDENT PROTEIN KINASE | PROTEIN KINASE FOLD, PHOSPHORYL TRANSFERASE, KINASE, REGULATORY SUBUNIT OF PKA, PKI, PHOSPHORYLATION, TRANSFERASE
4nw5:A (ARG94) to (GLY188) RSK2 N-TERMINAL KINASE IN COMPLEX WITH 2-AMINO-7-SUBSTITUTED BENZOXAZOLE COMPOUND 8 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4nw6:A (ARG94) to (GLY188) RSK2 N-TERMINAL KINASE IN COMPLEX WITH 2-AMINO-7-SUBSTITUTED BENZOXAZOLE COMPOUND 27 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4o0w:A (ALA160) to (ARG251) CRYSTAL STRUCTURES OF HUMAN KINASE AURORA A | PROTEIN KINASE, TRANSFERASE
2np8:A (ALA160) to (ARG251) STRUCTURAL BASIS FOR THE INHIBITION OF AURORA A KINASE BY A NOVEL CLASS OF HIGH AFFINITY DISUBSTITUTED PYRIMIDINE INHIBITORS | AURORA A KINASE, AIK, AURORA 2 KINASE, KINASE, KINASE INHIBITOR, TRANSFERASE
4o21:A (GLY66) to (TYR146) PRODUCT COMPLEX OF METAL-FREE PKAC, ATP-GAMMA-S AND SP20. | SER/THR KINASE, PHOSPHORYL TRANSFER, NUCLEOTIDE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4o22:A (GLY66) to (ASP161) BINARY COMPLEX OF METAL-FREE PKAC WITH SP20. | SER/THR KINASE, PHOSPHORYL TRANSFER, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2yza:A (HIS40) to (ARG132) CRYSTAL STRUCTURE OF KINASE DOMAIN OF HUMAN 5'-AMP-ACTIVATED PROTEIN KINASE ALPHA-2 SUBUNIT MUTANT (T172D) | SIGNALING PROTEIN, SERINE/THREONINE PROTEIN KINASE, PHOSPHORYLATION, ATP-BINDING, NUCLEOTIDE-BINDING, CHOLESTEROL BIOSYNTHESIS, FATTY ACID BIOSYNTHESIS, LIPID SYNTHESIS, GLUCOSE METABOLISM, MAGNESIUM, METAL-BINDING, SERINE/THREONINE-PROTEIN KINASE, STEROID BIOSYNTHESIS, TRANSFERASE, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
3k5u:A (ALA160) to (ARG251) IDENTIFICATION, SAR STUDIES AND X-RAY COCRYSTAL ANALYSIS OF A NOVEL FURANO-PYRIMIDINE AURORA KINASE A INHIBITOR | AURORA KINASE INHIBITORS, VIRTUAL SCREENING, X-RAY CO-CRYSTAL ANALYSIS, STRUCTURE-BASED DRUG DESIGN (SBDD), H-BONDING, ATP-BINDING SITE, CELL CYCLE, CYTOSKELETON, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4otd:A (GLU645) to (LYS741) CRYSTAL STRUCTURE OF PRK1 CATALYTIC DOMAIN | PRK1, PKN1, PROTEIN KINASE C RELATED KINASE 1, KINASE, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
4ae6:B (GLY66) to (ASP161) STRUCTURE AND FUNCTION OF THE HUMAN SPERM-SPECIFIC ISOFORM OF PROTEIN KINASE A (PKA) CATALYTIC SUBUNIT CALPHA 2 | TRANSFERASE
5d9k:A (ARG94) to (GLY188) RSK2 N-TERMINAL KINASE IN COMPLEX WITH BI-D1870 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3agl:A (GLY66) to (TYR146) COMPLEX OF PKA WITH THE BISUBSTRATE PROTEIN KINASE INHIBITOR ARC-1039 | PKA, PROTEIN KINASE A, BISUBSTRATE INHIBITOR, ARC-1039, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3agl:B (ASN67) to (TYR146) COMPLEX OF PKA WITH THE BISUBSTRATE PROTEIN KINASE INHIBITOR ARC-1039 | PKA, PROTEIN KINASE A, BISUBSTRATE INHIBITOR, ARC-1039, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4pnk:A (GLY214) to (PHE312) G PROTEIN-COUPLED RECEPTOR KINASE 2 IN COMPLEX WITH GSK180736A | PROTEIN KINASE, HYDROLASE, ATP BINDING, PHOSPHORYLATION, PERIPHERAL MEMBRANE PROTEIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5dnr:A (LEU159) to (ARG251) AURORA A KINASE IN COMPLEX WITH ATP IN SPACE GROUP P41212 | AURORA A KINASE, MITOTIC KINASE, PPI, TRANSFERASE
3lau:A (ALA160) to (ARG251) CRYSTAL STRUCTURE OF AURORA2 KINASE IN COMPLEX WITH A GSK3BETA INHIBITOR | KINASE INHIBITOR COMPLEX, ATP-BINDING, CELL CYCLE, CYTOPLASM, CYTOSKELETON, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, UBL CONJUGATION
5dos:A (LYS156) to (ARG251) AURORA A KINASE IN COMPLEX WITH AA35 AND ATP IN SPACE GROUP P6122 | AURORA A KINASE, MITOTIC KINASE, PPI, TRANSFERASE
1z5m:A (SER105) to (GLY200) CRYSTAL STRUCTURE OF N1-[3-[[5-BROMO-2-[[3-[(1-PYRROLIDINYLCARBONYL) AMINO]PHENYL]AMINO]-4-PYRIMIDINYL]AMINO]PROPYL]-2,2- DIMETHYLPROPANEDIAMIDE COMPLEXED WITH HUMAN PDK1 | PROTEIN INHIBITOR COMPLEX, SERINE KINASE, TRANSFERASE
4prj:A (ALA160) to (LYS251) AURORA A KINASE DOMAIN WITH COMPOUND 2 (N-[1-(3-CYANOBENZYL)-1H- PYRAZOL-4-YL]-6-(1H-PYRAZOL-4-YL)-1H-INDAZOLE-3-CARBOXAMIDE) | PROTEIN KINASE, PHOSPHO-TRANSFER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5dr2:A (LYS156) to (ARG251) AURORA A KINASE IN COMPLEX WITH AA30 AND ATP IN SPACE GROUP P6122 | AURORA A KINASE, MITOTIC KINASE, PPI, TRANSFERASE
5dr9:A (ALA160) to (ARG251) AURORA A KINASE IN COMPLEX WITH AA29 AND JNJ-7706621 IN SPACE GROUP P6122 | AURORA A KINASE, MITOTIC KINASE, PPI, TRANSFERASE
5drd:A (ALA160) to (ARG251) AURORA A KINASE IN COMPLEX WITH ATP IN SPACE GROUP P6122 | AURORA A KINASE, MITOTIC KINASE, PPI, TRANSFERASE
5dt0:A (ALA160) to (ARG251) AURORA A KINASE IN COMPLEX WITH JNJ-7706621 IN SPACE GROUP P6122 | AURORA A KINASE, MITOTIC KINASE, PPI, TRANSFERASE
5dt3:A (LEU159) to (ARG251) AURORA A KINASE IN COMPLEX WITH ATP IN SPACE GROUP P6122 | AURORA A KINASE, MITOTIC KINASE, PPI, TRANSFERASE
5dt4:A (LYS156) to (ARG251) AURORA A KINASE IN COMPLEX WITH AA35 AND ATP IN SPACE GROUP P6122 | AURORA A KINASE, MITOTIC KINASE, PPI, TRANSFERASE
3aqv:A (HIS40) to (ARG132) HUMAN AMP-ACTIVATED PROTEIN KINASE ALPHA 2 SUBUNIT KINASE DOMAIN (T172D) COMPLEXED WITH COMPOUND C | STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, TRANSFERASE, SIGNALING PROTEIN, SERINE/THREONINE PROTEIN KINASE, PHOSPHORYLATION, ATP-BINDING, NUCLEOTIDE-BINDING, CHOLESTEROL BIOSYNTHESIS, FATTY ACID BIOSYNTHESIS, LIPID SYNTHESIS, GLUCOSE METABOLISM, MAGNESIUM, METAL-BINDING, SERINE/THREONINE- PROTEIN KINASE, STEROID BIOSYNTHESIS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4aw1:A (SER105) to (GLY200) HUMAN PDK1 KINASE DOMAIN IN COMPLEX WITH ALLOSTERIC COMPOUND PS210 BOUND TO THE PIF-POCKET | TRANSFERASE, ALLOSTERIC REGULATION, ALLOSTERIC SITE, PHOSPHORYLATION, AGC PROTEIN KINASE
4aw2:A (ASP100) to (LEU195) CRYSTAL STRUCTURE OF CDC42 BINDING PROTEIN KINASE ALPHA (MRCK ALPHA) | TRANSFERASE, CDC42BPA
4qfg:A (GLY39) to (MET134) STRUCTURE OF AMPK IN COMPLEX WITH STAUROSPORINE INHIBITOR AND IN THE ABSENCE OF A SYNTHETIC ACTIVATOR | CBM, KINASE, AMPK, SIGNALING PROTEIN-INHIBITOR COMPLEX
3mfr:A (GLY35) to (ASN136) CASK-4M CAM KINASE DOMAIN, NATIVE | CATALYTIC MECHANISM, KINASE CATALYSIS, MG2+-MEDIATED PHOSPHATE TRANSFER, PROTEIN KINASE, TRANSFERASE
4bfm:A (GLY34) to (VAL112) THE CRYSTAL STRUCTURE OF MOUSE PK38 | TRANSFERASE
5eyk:A (LYS116) to (LYS211) CRYSTAL STRUCTURE OF AURORA B IN COMPLEX WITH BI 847325 | KINASE, INHIBITOR, TRANSFERASE
3mv5:A (GLY173) to (ASN269) CRYSTAL STRUCTURE OF AKT-1-INHIBITOR COMPLEXES | KINASE INHIBITOR, TRANSFERASE
3mvj:A (ASN67) to (ASP161) HUMAN CYCLIC AMP-DEPENDENT PROTEIN KINASE PKA INHIBITOR COMPLEX | KINASE INHIBITOR, TRANSFERASE
3mvj:B (GLY66) to (ASP161) HUMAN CYCLIC AMP-DEPENDENT PROTEIN KINASE PKA INHIBITOR COMPLEX | KINASE INHIBITOR, TRANSFERASE
3mvh:A (GLY173) to (ASN269) CRYSTAL STRUCTURE OF AKT-1-INHIBITOR COMPLEXES | KINASE INHIBITOR, TRANSFERASE
3myg:A (LYS156) to (ARG251) AURORA A KINASE COMPLEXED WITH SCH 1473759 | KINASE, CELL CYCLE, INHIBITOR, TRANSFERASE
5f9e:A (ASN403) to (GLY499) STRUCTURE OF PROTEIN KINASE C THETA WITH COMPOUND 10: 2,2-DIMETHYL-7- (2-OXIDANYLIDENE-3~{H}-IMIDAZO[4,5-B]PYRIDIN-1-YL)-1-(PHENYLMETHYL)- 3~{H}-QUINAZOLIN-4-ONE | KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5f9e:B (ASN403) to (GLY499) STRUCTURE OF PROTEIN KINASE C THETA WITH COMPOUND 10: 2,2-DIMETHYL-7- (2-OXIDANYLIDENE-3~{H}-IMIDAZO[4,5-B]PYRIDIN-1-YL)-1-(PHENYLMETHYL)- 3~{H}-QUINAZOLIN-4-ONE | KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3c0g:A (GLY35) to (ASN136) CASK CAM-KINASE DOMAIN- 3'-AMP COMPLEX, P1 FORM | CASK, NEUREXIN, CA2+/CALMODULIN DEPENDENT PROTEIN KINASE, MG2+, SYNAPTIC PLASTICITY, PSEUDOKINASE, MAGUK, MEMBRANE-ASSOCIATED GUANYLATE KINASE, ATP-BINDING, CALMODULIN-BINDING, MAGNESIUM, METAL- BINDING, NUCLEOTIDE-BINDING, NUCLEUS, SERINE/THREONINE-PROTEIN KINASE, SH3 DOMAIN, TRANSFERASE
4byi:A (ALA160) to (ARG251) AURORA A KINASE BOUND TO A HIGHLY SELECTIVE IMIDAZOPYRIDINE INHIBITOR | TRANSFERASE, CELL CYCLE, INHIBITOR
4ra4:A (GLU362) to (GLY458) CRYSTAL STRUCTURE OF HUMAN PROTEIN KINASE C ALPHA IN COMPLEX WITH COMPOUND 28 ((R)-6-((3S,4S)-1,3-DIMETHYL-PIPERIDIN-4-YL)-7-(2-FLUORO- PHENYL)-4-METHYL-2,10-DIHYDRO-9-OXA-1,2,4A-TRIAZA-PHENANTHREN-3-ONE) | KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ra5:A (ASN403) to (GLY491) HUMAN PROTEIN KINASE C THETA IN COMPLEX WITH LIGAND COMPOUND 11A (6- [(1,3-DIMETHYL-AZETIDIN-3-YL)-METHYL-AMINO]-4(R)-METHYL-7-PHENYL-2, 10-DIHYDRO-9-OXA-1,2,4A-TRIAZA-PHENANTHREN-3-ONE) | PKC THETA KINASE, KINASE DOMAIN, PROTEROS BIOSTRUCTURES GMBH, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ra5:B (ASN403) to (GLY491) HUMAN PROTEIN KINASE C THETA IN COMPLEX WITH LIGAND COMPOUND 11A (6- [(1,3-DIMETHYL-AZETIDIN-3-YL)-METHYL-AMINO]-4(R)-METHYL-7-PHENYL-2, 10-DIHYDRO-9-OXA-1,2,4A-TRIAZA-PHENANTHREN-3-ONE) | PKC THETA KINASE, KINASE DOMAIN, PROTEROS BIOSTRUCTURES GMBH, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ncz:A (ARG99) to (MET192) X-RAY CO-STRUCTURE OF RHO-ASSOCIATED PROTEIN KINASE (ROCK1) WITH A POTENT 2H-ISOQUINOLIN-1-ONE INHIBITOR | RHO KINASE, DIMER, PHOSPHORYLATION, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3ncz:C (ARG99) to (SER191) X-RAY CO-STRUCTURE OF RHO-ASSOCIATED PROTEIN KINASE (ROCK1) WITH A POTENT 2H-ISOQUINOLIN-1-ONE INHIBITOR | RHO KINASE, DIMER, PHOSPHORYLATION, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3ncz:D (ARG99) to (SER191) X-RAY CO-STRUCTURE OF RHO-ASSOCIATED PROTEIN KINASE (ROCK1) WITH A POTENT 2H-ISOQUINOLIN-1-ONE INHIBITOR | RHO KINASE, DIMER, PHOSPHORYLATION, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4c34:A (GLY66) to (ASP161) PKA-S6K1 CHIMERA WITH STAUROSPORINE BOUND | TRANSFERASE-INHIBITOR COMPLEX
4c35:A (GLY66) to (ASP161) PKA-S6K1 CHIMERA WITH COMPOUND 1 (NU1085) BOUND | TRANSFERASE-INHIBITOR COMPLEX, CHIMERA, S6K1
4c38:A (GLY66) to (ASP161) PKA-S6K1 CHIMERA WITH COMPOUND 21E (CCT239066) BOUND | TRANSFERASE-INHIBITOR COMPLEX
3ndm:A (ARG99) to (GLY193) CRYSTAL STRUCTURE OF RHO-ASSOCIATED PROTEIN KINASE (ROCK1) WITH A POTENT ISOQUINOLONE DERIVATIVE | RHO KINASE, PHOSPHORYLATION, DIMERIZATION, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3ndm:B (ARG99) to (GLY193) CRYSTAL STRUCTURE OF RHO-ASSOCIATED PROTEIN KINASE (ROCK1) WITH A POTENT ISOQUINOLONE DERIVATIVE | RHO KINASE, PHOSPHORYLATION, DIMERIZATION, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3ndm:C (ARG99) to (GLY193) CRYSTAL STRUCTURE OF RHO-ASSOCIATED PROTEIN KINASE (ROCK1) WITH A POTENT ISOQUINOLONE DERIVATIVE | RHO KINASE, PHOSPHORYLATION, DIMERIZATION, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4rer:A (GLY41) to (MET136) CRYSTAL STRUCTURE OF THE PHOSPHORYLATED HUMAN ALPHA1 BETA2 GAMMA1 HOLO-AMPK COMPLEX BOUND TO AMP AND CYCLODEXTRIN | HUMAN ALPHA1 BETA2 GAMMA1 HOLO-AMPK COMPLEX, SERINE/THREONINE PROTEIN KINASE, AXIN, CAMKKBETA, LKB1, GLYCOGEN, PHOSPHORYLATION, TRANSFERASE
4c3p:A (ALA160) to (ARG251) STRUCTURE OF DEPHOSPHORYLATED AURORA A (122-403) BOUND TO TPX2 AND AMPPCP | TRANSFERASE, ACTIVATION, ALLOSTERY, CELL CYCLE, CANCER
3cik:A (ALA218) to (PHE312) HUMAN GRK2 IN COMPLEX WITH GBETAGAMMA SUBUNITS | PROTEIN KINASE, COMPLEX, G PROTEIN, RECEPTOR, WD40 REPEAT, ATP- BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSDUCER, WD REPEAT, LIPOPROTEIN, MEMBRANE, PHOSPHOPROTEIN, PRENYLATION, TRANSFERASE-SIGNALING PROTEIN COMPLEX
5fqd:F (GLY40) to (ASN131) STRUCTURAL BASIS OF LENALIDOMIDE INDUCED CK1A DEGRADATION BY THE CRL4CRBN UBIQUITIN LIGASE | LIGASE, DNA BINDING
3nrm:A (LEU159) to (ARG251) IMIDAZO[1,2-A]PYRAZINE-BASED AURORA KINASE INHIBITORS | KINASE, CELL CYCLE, INHIBITOR, TRANSFERASE
3coh:A (ALA160) to (LYS251) CRYSTAL STRUCTURE OF AURORA-A IN COMPLEX WITH A PENTACYCLIC INHIBITOR | AURORA-A, INHIBITOR COMPLEX, ATP-BINDING, CELL CYCLE, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3coh:B (ALA160) to (LYS251) CRYSTAL STRUCTURE OF AURORA-A IN COMPLEX WITH A PENTACYCLIC INHIBITOR | AURORA-A, INHIBITOR COMPLEX, ATP-BINDING, CELL CYCLE, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3cok:A (GLY34) to (GLY130) CRYSTAL STRUCTURE OF PLK4 KINASE | PLK4, POLO-LIKE KINASE 4, SAK, STK18, PSI, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3cok:B (GLY34) to (GLY130) CRYSTAL STRUCTURE OF PLK4 KINASE | PLK4, POLO-LIKE KINASE 4, SAK, STK18, PSI, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4ceg:A (ALA160) to (ARG251) CRYSTAL STRUCTURE OF AURORA A 122-403 C290A, C393A BOUND TO ADP | TRANSFERASE, PROTEIN KINASE, MITOSIS
3nun:A (SER105) to (GLY200) PHOSPHOINOSITIDE-DEPENDENT KINASE-1 (PDK1) WITH LEAD COMPOUND | KINASE DOMAIN, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3cqu:A (GLY173) to (ASN269) CRYSTAL STRUCTURE OF AKT-1 COMPLEXED WITH SUBSTRATE PEPTIDE AND INHIBITOR | KINASE, APOPTOSIS, ATP-BINDING, CARBOHYDRATE METABOLISM, CYTOPLASM, GLUCOSE METABOLISM, GLYCOGEN BIOSYNTHESIS, GLYCOGEN METABOLISM, MEMBRANE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, SUGAR TRANSPORT, TRANSFERASE, TRANSLATION REGULATION, TRANSPORT, ALTERNATIVE SPLICING, WNT SIGNALING PATHWAY
4rqk:A (SER105) to (GLY200) CRYSTAL STRUCTURE OF PDK1 IN COMPLEX WITH ATP AND THE PIF-POCKET LIGAND RS1 | PROTEIN KINASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4rqv:A (SER105) to (GLY200) CRYSTAL STRUCTURE OF PDK1 IN COMPLEX WITH ATP AND THE PIF-POCKET LIGAND RS2 | PROTEIN KINASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3nx8:A (GLY66) to (ASP161) HUMAN CAMP DEPENDENT PROTEIN KINASE IN COMPLEX WITH PHENOL | TRANSFERASE, ATP BINDING, PHOSPHORYLATION
3d0e:A (ARG176) to (ASP270) CRYSTAL STRUCTURE OF HUMAN AKT2 IN COMPLEX WITH GSK690693 | HUMAN, AKT2, INHIBITOR, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSFERASE INHIBITOR
3d0e:B (GLY175) to (ASP270) CRYSTAL STRUCTURE OF HUMAN AKT2 IN COMPLEX WITH GSK690693 | HUMAN, AKT2, INHIBITOR, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSFERASE INHIBITOR
3d15:A (LYS169) to (ARG264) CRYSTAL STRUCTURE OF MOUSE AURORA A (ASN186->GLY, LYS240->ARG, MET302- >LEU) IN COMPLEX WITH 1-(3-CHLORO-PHENYL)-3-{5-[2-(THIENO[3,2- D]PYRIMIDIN-4-YLAMINO)- ETHYL]-THIAZOL-2-YL}-UREA [SNS-314] | AURORA A, SMALL-MOLECULE INHIBITOR, KINASE, TRANSFERASE
3o7l:D (ASN67) to (ASP161) CRYSTAL STRUCTURE OF PHOSPHOLAMBAN (1-19):PKA C-SUBUNIT:AMP-PNP:MG2+ COMPLEX | PROTEIN KINASE A, PHOSPHOLAMBAN, ALLOSTERY, SUBSTRATE RECOGNITION, CONFORMATIONAL SELECTION, INTRINSICALLY DISORDERED PROTEINS, MEMBRANE PROTEINS, TRANSFERASE
3d2k:A (ALA173) to (ARG264) CRYSTAL STRUCTURE OF MOUSE AURORA A (ASN186->GLY, LYS240- >ARG, MET302->LEU) IN COMPLEX WITH [7-(2-{2-[3-(3-CHLORO- PHENYL)-UREIDO]-THIAZOL-5-YL}-ETHYLAMINO)-PYRAZOLO[4,3- D]PYRIMIDIN-1-YL]-ACETIC ACID | AURORA A, SMALL-MOLECULE INHIBITOR, KINASE, TRANSFERASE
4ct1:A (SER105) to (GLY200) HUMAN PDK1-PKCZETA KINASE CHIMERA IN COMPLEX WITH ALLOSTERIC COMPOUND PS315 BOUND TO THE PIF-POCKET | TRANSFERASE, ALLOSTERIC REGULATION, ALLOSTERIC SITE, PHOSPHORYLATION, AGC PROTEIN KINASE, CHIMERIC PROTEIN
3d9v:A (ARG99) to (SER191) CRYSTAL STRUCTURE OF ROCK I BOUND TO H-1152P A DI- METHYLATED VARIANT OF FASUDIL | DIMER, DIMERIZATION, KINASE, PHOSPHORYLATION, FASUDIL, APOPTOSIS, ATP-BINDING, COILED COIL, CYTOPLASM, GOLGI APPARATUS, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ZINC, ZINC- FINGER
3d9v:B (ARG99) to (SER191) CRYSTAL STRUCTURE OF ROCK I BOUND TO H-1152P A DI- METHYLATED VARIANT OF FASUDIL | DIMER, DIMERIZATION, KINASE, PHOSPHORYLATION, FASUDIL, APOPTOSIS, ATP-BINDING, COILED COIL, CYTOPLASM, GOLGI APPARATUS, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ZINC, ZINC- FINGER
3ocb:B (GLY173) to (ASN269) AKT1 KINASE DOMAIN WITH PYRROLOPYRIMIDINE INHIBITOR | SERINE-THREONINE KINASE, TRANSFERASE
3dj5:A (ALA173) to (LYS263) CRYSTAL STRUCTURE OF THE MOUSE AURORA-A CATALYTIC DOMAIN (ASN186->GLY, LYS240->ARG, MET302->LEU) IN COMPLEX WITH COMPOUND 290. | AURORA A, SMALL-MOLECULE INHIBITOR, FRAGMENT-BASED DRUG DISCOVERY, KINASE, TRANSFERASE
4d28:D (GLY34) to (GLY129) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF SNRK3.11 AT5G35410 | TRANSFERASE, SALT STRESS, SODIUM TRANSPORT, ION HOMEOSTASIS
3oog:A (GLY66) to (TYR146) HUMAN CAMP-DEPENDENT PROTEIN KINASE IN COMPLEX WITH A SMALL FRAGMENT | TRANSFERASE, ATP BINDING, PHOSPHORYLATION
3orz:A (SER105) to (GLY200) PDK1 MUTANT BOUND TO ALLOSTERIC DISULFIDE FRAGMENT ACTIVATOR 2A2 | C HELIX, SER/THR-KINASE, AGC KINASE, ALLOSTERY, TRANSFERASE, ALLOSTERIC ACTIVATOR, BISINDOLYLMALEIMIDE, DISULFIDE, KINASE, PDK1, TRANSFERASE-TRANSFERASE ACTIVATOR COMPLEX
3orz:C (SER105) to (GLY200) PDK1 MUTANT BOUND TO ALLOSTERIC DISULFIDE FRAGMENT ACTIVATOR 2A2 | C HELIX, SER/THR-KINASE, AGC KINASE, ALLOSTERY, TRANSFERASE, ALLOSTERIC ACTIVATOR, BISINDOLYLMALEIMIDE, DISULFIDE, KINASE, PDK1, TRANSFERASE-TRANSFERASE ACTIVATOR COMPLEX
3ovv:A (GLY66) to (ASP161) HUMAN CAMP-DEPENDENT PROTEIN KINASE IN COMPLEX WITH AN INHIBITOR | TRANSFERASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ow3:A (GLY66) to (ASP161) DISCOVERY OF DIHYDROTHIENO- AND DIHYDROFUROPYRIMIDINES AS POTENT PAN AKT INHIBITORS | CYCLIC-AMP DEPENDENT PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ow4:A (GLY173) to (ASN269) DISCOVERY OF DIHYDROTHIENO- AND DIHYDROFUROPYRIMIDINES AS POTENT PAN AKT INHIBITORS | SERINE-THREONINE KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ow4:B (ARG174) to (ASN269) DISCOVERY OF DIHYDROTHIENO- AND DIHYDROFUROPYRIMIDINES AS POTENT PAN AKT INHIBITORS | SERINE-THREONINE KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5he1:A (GLY214) to (PHE312) HUMAN GRK2 IN COMPLEX WITH GBETAGAMMA SUBUNITS AND CCG224062 | RGS, KINASE, PH, WD-40, INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5he2:A (GLY214) to (PHE312) BOVINE GRK2 IN COMPLEX WITH GBETAGAMMA SUBUNITS AND CCG224406 | RGS, KINASE, PH, WD-40, INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3owp:A (GLY66) to (ASP161) HUMAN CAMP-DEPENDENT PROTEIN KINASE IN COMPLEX WITH AN INHIBITOR | TRANSFERASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3oxt:A (GLY66) to (ASP161) HUMAN CAMP-DEPENDENT PROTEIN KINASE IN COMPLEX WITH AN INHIBITOR | TRANSFERASE, PHOSPHORYLATION
4dfx:E (GLY66) to (ASP161) CRYSTAL STRUCTURE OF MYRISTOYLATED K7C CATALYTIC SUBUNIT OF CAMP- DEPENDENT PROTEIN KINASE IN COMPLEX WITH SP20 AND AMP-PNP | PROTEIN KINASE, MYRISTOYLATED, PHOSPHOTRANSFERASE ONTO SER/THR, MG, PKI, PKA REGULATORY SUBUNITS, PHOSPHORYLATED ON S139, T197, S338, MYRISTOYLATED ON G1, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4dg0:E (GLY66) to (ASP161) CRYSTAL STRUCTURE OF MYRISTOYLATED WT CATALYTIC SUBUNIT OF CAMP- DEPENDENT PROTEIN KINASE IN COMPLEX WITH SP20 AND AMP-PNP | PROTEIN KINASE, MYRISTOYLATED, PHOSPHOTRANSFERASE OF SER/THR, MG, PKI, PKA REGULATORY SUBUNITS, PHOSPHORYLATED ON S139, T197, S338, MYRISTOYLATED ON G1, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4dh1:A (ASN67) to (ASP161) LOW TEMPERATURE X-RAY STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A CATALYTIC SUBUNIT WITH LOW MG2+, ATP AND IP20 | PROTEIN KINASE, PHOSPHORYLATION, PEPTIDIC INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4dh8:A (GLY66) to (ASP161) ROOM TEMPERATURE X-RAY STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A CATALYTIC SUBUNIT WITH HIGH MG2+, AMP-PNP AND IP20 | PROTEIN KINASE, PHOSPHOTRANSFER, PEPTIDIC INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4dhf:B (LYS156) to (SER249) STRUCTURE OF AURORA A MUTANT BOUND TO BIOGENIDEC CPD 15 | SER/THR KINASE MITOTIC KINASE PYRAZOLOPYRIMIDINE, PHOSPHORYLATION, TPX2, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4din:A (GLY66) to (ASP161) NOVEL LOCALIZATION AND QUATERNARY STRUCTURE OF THE PKA RI BETA HOLOENZYME | ISOFORM DIVERSITY, RIB2:C2 TETRAMERIC COMPLEX, TRANSFERASE-TRANSPORT PROTEIN COMPLEX
3p0m:A (GLY66) to (TYR146) HUMAN CAMP-DEPENDENT PROTEIN KINASE IN COMPLEX WITH AN INHIBITOR | TRANSFERASE, PHOSPHORYLATION
5hkm:A (ARG106) to (GLY200) DISCOVERY OF NOVEL 7-AZAINDOLES AS PDK1 INHIBITORS | PDK1 INHIBITOR, TRANSFERASE
5hng:A (SER105) to (GLY200) DISCOVERY OF NOVEL 7-AZAINDOLES AS PDK1 INHIBITORS | PDK1 INHIBITOR, TRANSFERASE
5ho7:A (SER105) to (GLY200) DISCOVERY OF NOVEL 7-AZAINDOLES AS PDK1 INHIBITORS | PDK1 INHIBITOR, TRANSFERASE
5ho8:A (SER105) to (GLY200) DISCOVERY OF NOVEL 7-AZAINDOLES AS PDK1 INHIBITORS | PDK1 INHIBITOR, TRANSFERASE
4ual:A (GLU99) to (HIS195) MRCK BETA IN COMPLEX WITH BDP00005290 | MYOTONIC DYSTROPHY KINASE-RELATED CDC42-BINDING KINASE, METASTASIS, CELL INVASION, TRANSFERASE
3pfq:A (ASP365) to (GLY461) CRYSTAL STRUCTURE AND ALLOSTERIC ACTIVATION OF PROTEIN KINASE C BETA II | KINASE, PHOSPHORYLATION, TRANSFERASE
4uj1:A (GLY66) to (TYR146) PROTEIN KINASE A IN COMPLEX WITH AN INHIBITOR | TRANSFERASE-INHIBITOR COMPLEX, PROTEIN KINASE A,
4ujb:A (GLY66) to (TYR146) PROTEIN KINASE A IN COMPLEX WITH AN INHIBITOR | TRANSFERASE
3pwy:A (SER105) to (GLY200) CRYSTAL STRUCTURE OF AN EXTENDER (SPD28345)-MODIFIED HUMAN PDK1 COMPLEX 2 | KINASE, FRAGMENT-BASED DRUG DISCOVERY, TETHERING WITH EXTENDERS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ekk:A (GLY173) to (ASN269) AKT1 WITH AMP-PNP | PHOSPHOTRANSFERASE, TRANSFERASE
4ekk:B (ARG174) to (ASN269) AKT1 WITH AMP-PNP | PHOSPHOTRANSFERASE, TRANSFERASE
4ekl:A (GLY173) to (ASN269) AKT1 WITH GDC0068 | PHOSPHOTRANSFERASE, TRANSFERASE
3qal:E (GLY66) to (ASP161) CRYSTAL STRUCTURE OF ARG280ALA MUTANT OF CATALYTIC SUBUNIT OF CAMP- DEPENDENT PROTEIN KINASE | PROTEIN KINASE, GLU208/ARG280 PAIR, PKA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qbn:A (LYS156) to (ARG251) STRUCTURE OF HUMAN AURORA A IN COMPLEX WITH A DIAMINOPYRIMIDINE | KINASE DOMAIN, DIAMINOPYRIMIDINE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qd3:A (ARG106) to (GLY200) PHOSPHOINOSITIDE-DEPENDENT KINASE-1 (PDK1) KINASE DOMAIN WITH 1,1- DIMETHYLETHYL {(3R,6S)-1-[2-AMINO-6-(3-AMINO-1H-INDAZOL-6-YL)-4- PYRIMIDINYL]-6-METHYL-3-PIPERIDINYL}CARBAMATE | KINASE DOMAIN, AGC KINASE, SIGNAL TRANDUCTION, ATP & PHOSPHOINOSITIDE, PHOSPHORYLATION ON S241, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5j5x:A (GLY66) to (ASP161) COMPLEX OF PKA WITH THE BISUBSTRATE PROTEIN KINASE INHIBITOR ARC-1416 | PROTEIN KINASE, INHIBITOR, BISUBSTRATE, OLIGOARGININE, PKA, TRANSFERASE
3qkk:A (GLY173) to (ASN269) SPIROCHROMANE AKT INHIBITORS | KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qkl:A (GLY173) to (ASN269) SPIROCHROMANE AKT INHIBITORS | KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qkm:A (GLY173) to (ASN269) SPIROCYCLIC SULFONAMIDES AS AKT INHIBITORS | KINASE DOMAIN, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4uzh:A (ALA160) to (ARG251) SAR156497 AN EXQUISITELY SELECTIVE INHIBITOR OF AURORA KINASES | TRANSFERASE
4w7p:A (ARG99) to (SER191) CRYSTAL STRUCTURE OF ROCK 1 BOUND TO YB-15-QD37 | INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4w7p:C (ARG99) to (SER191) CRYSTAL STRUCTURE OF ROCK 1 BOUND TO YB-15-QD37 | INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fvp:A (GLN572) to (THR668) CRYSTAL STRUCTURE OF THE JAK2 PSEUDOKINASE DOMAIN (APO FORM) | JANUS PROTEIN KINASE, PSEUDOKINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
4fvq:A (LEU579) to (THR668) CRYSTAL STRUCTURE OF THE JAK2 PSEUDOKINASE DOMAIN (MG-ATP-BOUND FORM) | JANUS PROTEIN KINASE, PSEUDOKINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
5lpw:A (ILE910) to (HIS998) CRYSTAL STRUCTURE OF THE APO-BRI1 KINASE DOMAIN (865-1160) | BRASSINOSTEROID RECEPTOR, KINASE DOMAIN, DUAL-SPECIFICIFY KINASE, MEMBRANE RECEPTOR KINASE, PLASMA MEMBRANE, TRANSFERASE
5lvl:A (SER105) to (GLY200) HUMAN PDK1 KINASE DOMAIN IN COMPLEX WITH COMPOUND PS653 BOUND TO THE ATP-BINDING SITE | PROTEIN KINASE, ALLOSTERIC REGULATION, SMALL COMPOUNDS, PIF-POCKET, TRANSFERASE
5lvn:A (SER105) to (GLY200) HUMAN PDK1 KINASE DOMAIN IN COMPLEX WITH ADENOSINE BOUND TO THE ATP- BINDING SITE | PROTEIN KINASE, ALLOSTERIC REGULATION, SMALL COMPOUNDS, PIF-POCKET, TRANSFERASE
2c1b:A (GLY66) to (TYR146) STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE COMPLEXED WITH ( 4R,2S)-5'-(4-(4-CHLOROBENZYLOXY)PYRROLIDIN-2- YLMETHANESULFONYL)ISOQUINOLINE | TRANSFERASE/INHIBITOR, COMPLEX (TRANSFERASE/INHIBITOR), ATP-BINDING, CAMP, PHOSPHORYLATION, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, PROTEIN KINASE INHIBITOR
2c1a:A (GLY66) to (TYR146) STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE COMPLEXED WITH ISOQUINOLINE-5-SULFONIC ACID (2-(2-(4-CHLOROBENZYLOXY) ETHYLAMINO)ETHYL)AMIDE | TRANSFERASE/INHIBITOR, COMPLEX (TRANSFERASE/INHIBITOR), ATP-BINDING, CAMP, PHOSPHORYLATION, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, PROTEIN KINASE INHIBITOR
3fjq:E (GLY66) to (ASP161) CRYSTAL STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE CATALYTIC SUBUNIT ALPHA IN COMPLEX WITH PEPTIDE INHIBITOR PKI ALPHA (6-25) | NUCLEOTIDE BINDING, PROTEIN KINASE ACTIVITY, PROTEIN SERINE/THREONINE KINASE ACTIVITY, CAMP-DEPENDENT PROTEIN KINASE ACTIVITY, PROTEIN BINDING, ATP BINDING, KINASE ACTIVITY, TRANSFERASE ACTIVITY, ALTERNATIVE SPLICING, ATP- BINDING, CAMP, CYTOPLASM, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, PROTEIN KINASE INHIBITOR
3twj:B (ARG99) to (GLY193) RHO-ASSOCIATED PROTEIN KINASE 1 (ROCK 1) IN COMPLEX WITH RKI1447 | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3twj:C (ARG99) to (GLY193) RHO-ASSOCIATED PROTEIN KINASE 1 (ROCK 1) IN COMPLEX WITH RKI1447 | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2uw0:A (GLY66) to (TYR146) STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH 6-(4-(4-(4- CHLORO-PHENYL)-PIPERIDIN-4-YL)-PHENYL)-9H-PURINE | TRANSFERASE/INHIBITOR, TRANSFERASE/INHIBITOR COMPLEX, CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION
2uw7:A (GLY66) to (TYR146) STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH 4-(4-CHLORO- PHENYL)-4-(4-(1H-PYRAZOL-4-YL)-PHENYL)-PIPERIDINE | TRANSFERASE/INHIBITOR, CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION, TRANSFERASE/INHIBITOR COMPLEX
2uw8:A (GLY66) to (TYR146) STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH 2-(4-CHLORO- PHENYL)-2-PHENYL-ETHYLAMINE | TRANSFERASE/INHIBITOR, CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION, TRANSFERASE/INHIBITOR COMPLEX
4kbc:A (GLU33) to (ASN123) CK1D IN COMPLEX WITH {4-[3-(4-FLUOROPHENYL)-1H-PYRAZOL-4-YL]PYRIDIN-2- YL}METHANOL INHIBITOR | SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uo6:A (LEU159) to (ARG251) AURORA A IN COMPLEX WITH YL5-083 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uo6:B (LEU159) to (ARG251) AURORA A IN COMPLEX WITH YL5-083 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uol:A (LEU159) to (ARG251) AURORA A IN COMPLEX WITH SO2-162 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uol:B (LEU159) to (ARG251) AURORA A IN COMPLEX WITH SO2-162 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4z84:A (GLY66) to (ASP161) PKAB3 IN COMPLEX WITH PYRROLIDINE INHIBITOR 34A | INHIBITOR, PROTEIN KINASE, STRUCTURE-GUIDED, TRANSFERASE
3uzt:A (LYS215) to (PHE312) STRUCTURE OF THE C13.18 RNA APTAMER IN COMPLEX WITH G PROTEIN-COUPLED RECEPTOR KINASE 2 | PROTEIN-RNA COMPLEX, PROTEIN KINASE FOLD, RGS HOMOLOGY DOMAIN, PLECKSTRIN HOMOLOGY DOMAIN, G PROTEIN-COUPLED RECEPTOR PHOSPHORYLATION, RNA APTAMER, TRANSFERASE-RNA COMPLEX
3v8s:A (ARG99) to (GLY193) HUMAN RHO-ASSOCIATED PROTEIN KINASE 1 (ROCK 1) IN COMPLEX WITH INDAZOLE DERIVATIVE (COMPOUND 18) | KINASE, DIMERIZATION, MYOSIN, TRANSFERASE, INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3v8s:C (ARG99) to (GLY193) HUMAN RHO-ASSOCIATED PROTEIN KINASE 1 (ROCK 1) IN COMPLEX WITH INDAZOLE DERIVATIVE (COMPOUND 18) | KINASE, DIMERIZATION, MYOSIN, TRANSFERASE, INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3v8s:D (ARG99) to (GLY193) HUMAN RHO-ASSOCIATED PROTEIN KINASE 1 (ROCK 1) IN COMPLEX WITH INDAZOLE DERIVATIVE (COMPOUND 18) | KINASE, DIMERIZATION, MYOSIN, TRANSFERASE, INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
2vz6:A (GLY36) to (GLY130) STRUCTURE OF HUMAN CALCIUM CALMODULIN DEPENDENT PROTEIN KINASE TYPE II ALPHA (CAMK2A) IN COMPLEX WITH INDIRUBIN E804 | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, CELL JUNCTION, CELL MEMBRANE, LONG TERM POTENTIATION, BRAIN, KINASE, SYNAPSE, MEMBRANE, NMDA RECEPTOR SIGNALLING, PHOSPHOPROTEIN, CALMODULIN-BINDING, NUCLEOTIDE-BINDING
3iop:A (SER105) to (GLY200) PDK-1 IN COMPLEX WITH THE INHIBITOR COMPOUND-8I | PDK-1, INHIBITOR, ALTERNATIVE SPLICING, ATP-BINDING, CYTOPLASM, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3iw4:A (GLU362) to (GLY458) CRYSTAL STRUCTURE OF PKC ALPHA IN COMPLEX WITH NVP-AEB071 | KINASE, ATP-BINDING, CELL MEMBRANE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ZINC-FINGER
3iw4:C (GLU362) to (GLY458) CRYSTAL STRUCTURE OF PKC ALPHA IN COMPLEX WITH NVP-AEB071 | KINASE, ATP-BINDING, CELL MEMBRANE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ZINC-FINGER
1uu3:A (SER105) to (GLY200) STRUCTURE OF HUMAN PDK1 KINASE DOMAIN IN COMPLEX WITH LY333531 | PROTEIN KINASE, PKB, PDK1, INHIBITOR, LY333531, DIABETES, CANCER, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE
2xck:A (ALA109) to (GLY200) CRYSTAL STRUCTURE OF PDK1 IN COMPLEX WITH A PYRAZOLOQUINAZOLINE INHIBITOR | PI3-KINASE SIGNALLING, TRANSFERASE, ATP-BINDING, SERINE/THREONINE-PROTEIN KINASE
5bml:B (ARG99) to (GLY193) ROCK 1 BOUND TO A PYRIDINE THIAZOLE INHIBITOR | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3zo4:A (GLY66) to (ASP161) THE SYNTHESIS AND EVALUATION OF DIAZASPIROCYCLIC PROTEIN KINASE INHIBITORS | TRANSFERASE-INHIBITOR COMPLEX
4nzw:B (GLU44) to (ARG135) CRYSTAL STRUCTURE OF STK25-MO25 COMPLEX | SCAFOLDING PROTEIN, SER/THR PROTEIN KINASE, TRANSFERASE ACTIVATOR- TRANSFERASE COMPLEX
4o2z:A (VAL73) to (ASN170) CRYSTAL STRUCTURE OF MPK3 FROM LEISHMANIA DONOVANI, LDBPK_100540 IN THE PRESENCE OF NVP-BBT594 | NEGLECTED DISEASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE
1xh4:A (GLY66) to (ASP161) CRYSTAL STRUCTURES OF PROTEIN KINASE B SELECTIVE INHIBITORS IN COMPLEX WITH PROTEIN KINASE A AND MUTANTS | PKA, KINASE-INHIBITOR-COMPLEX, SERINE/THREONINE-PROTEIN KINASE, BALANOL DERIVATIVE, TRANSFERASE/TRANSFERASE INHIBITOR COMPLEX
4ow8:A (VAL39) to (GLY136) CRYSTAL STRUCTURE OF KINASE DOMAIN OF PKNA FROM MTB | PKNA, KINASE, DRUG TARGET, MTB
1yds:E (GLY66) to (ASP161) STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE, ALPHA-CATALYTIC SUBUNIT IN COMPLEX WITH H8 PROTEIN KINASE INHIBITOR [N-(2-METHYLAMINO)ETHYL]-5- ISOQUINOLINESULFONAMIDE | PHOSPHOTRANSFERASE, TRANSFERASE, CAMP, PHOSPHORYLATION, ISOQUINOLINE SULFONAMIDE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ag9:A (GLY66) to (ASP161) COMPLEX OF PKA WITH THE BISUBSTRATE PROTEIN KINASE INHIBITOR ARC-1012 | PKA, PROTEIN KINASE A, BISUBSTRATE INHIBITOR, ARC-1012, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3ag9:B (GLY66) to (ASP161) COMPLEX OF PKA WITH THE BISUBSTRATE PROTEIN KINASE INHIBITOR ARC-1012 | PKA, PROTEIN KINASE A, BISUBSTRATE INHIBITOR, ARC-1012, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3agm:A (GLY66) to (TYR146) COMPLEX OF PKA WITH THE BISUBSTRATE PROTEIN KINASE INHIBITOR ARC-670 | PKA, PROTEIN KINASE A, BISUBSTRATE, BISUBSTRATE INHIBITOR, ARC-670, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3amb:A (GLY66) to (ASP161) PROTEIN KINASE A SIXFOLD MUTANT MODEL OF AURORA B WITH INHIBITOR VX- 680 | PKA, PROTEIN KINASE A, SURROGATE, VX-680, MK-0457, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4aw0:A (SER105) to (GLY200) HUMAN PDK1 KINASE DOMAIN IN COMPLEX WITH ALLOSTERIC COMPOUND PS182 BOUND TO THE PIF-POCKET | TRANSFERASE, ALLOSTERIC REGULATION, ALLOSTERIC SITE, PHOSPHORYLATION, AGC PROTEIN KINASE
4axa:A (GLY66) to (ASP161) STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH (1S)-2-AMINO-1-( 4-CHLOROPHENYL)-1-(4-(1H-PYRAZOL-4-YL)PHENYL)ETHAN-1-OL | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4q9z:A (ASN403) to (GLY491) HUMAN PROTEIN KINASE C THETA IN COMPLEX WITH COMPOUND35 ((1R)-9- (AZETIDIN-3-YLAMINO)-1,8-DIMETHYL-3,5-DIHYDRO[1,2,4]TRIAZINO[3,4- C][1,4]BENZOXAZIN-2(1H)-ONE) | PKC THETA KINASE, KINASE CATALYTIC DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4q9z:B (ASN403) to (GLY491) HUMAN PROTEIN KINASE C THETA IN COMPLEX WITH COMPOUND35 ((1R)-9- (AZETIDIN-3-YLAMINO)-1,8-DIMETHYL-3,5-DIHYDRO[1,2,4]TRIAZINO[3,4- C][1,4]BENZOXAZIN-2(1H)-ONE) | PKC THETA KINASE, KINASE CATALYTIC DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4c0t:A (GLY263) to (GLY359) CANDIDA ALBICANS PKH KINASE DOMAIN | TRANSFERASE, PDK1 ORTHOLOG
4c37:A (GLY66) to (ASP161) PKA-S6K1 CHIMERA WITH COMPOUND 21A (CCT196539) BOUND | TRANSFERASE-INHIBITOR COMPLEX, CHIMERA, S6K1
3nuu:A (SER105) to (GLY200) PHOSPHOINOSITIDE-DEPENDENT KINASE-1 (PDK1) WITH FRAGMENT11 | KINASE DOMAIN, TRANSFERASE
4rrv:A (ARG106) to (GLY200) CRYSTAL STRUCTURE OF PDK1 IN COMPLEX WITH ATP AND PIFTIDE | PROTEIN KINASE, PIFTIDE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4twc:B (GLU33) to (ASN123) 2-BENZAMIDO-N-(1H-BENZO[D]IMIDAZOL-2-YL)THIAZOLE-4- CARBOXAMIDE DERIVATIVES AS POTENT INHIBITORS OF CK1D/E | CK1D, CK1E, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, TRANSFERASE
4dh5:A (GLY66) to (ASP161) ROOM TEMPERATURE X-RAY STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A CATALYTIC SUBUNIT WITH HIGH MG2+, ADP, PHOSPHATE, AND IP20 | PROTEIN KINASE, PHOSPHOTRANSFER, PEPTIDIC INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4uj2:A (GLY66) to (ASP161) PROTEIN KINASE A IN COMPLEX WITH AN INHIBITOR | TRANSFERASE-INHIBITOR COMPLEX, PROTEIN KINASE A,
4uja:A (GLY66) to (TYR146) PROTEIN KINASE A IN COMPLEX WITH AN INHIBITOR | TRANSFERASE
3qcy:A (SER105) to (GLY200) PHOSPHOINOSITIDE-DEPENDENT KINASE-1 (PDK1) KINASE DOMAIN WITH 4-[2- AMINO-6-(3-AMINO-1H-INDAZOL-6-YL)-4-PYRIMIDINYL]-N-PHENYL-2- MORPHOLINECARBOXAMIDE | KINASE DOMAIN, AGC KINASE, SIGNAL TRANSDUCTION, PHOSPHOINOSITIDE, PHOSPHORYLATION ON S241, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5k3y:A (LYS116) to (LYS211) CRYSTAL STRUCTURE OF AURORAB/INCENP IN COMPLEX WITH BI 811283 | KINASE, INHIBITOR, TRANSFERASE
5lvm:A (SER105) to (GLY200) HUMAN PDK1 KINASE DOMAIN IN COMPLEX WITH ADENINE BOUND TO THE ATP- BINDING SITE | PROTEIN KINASE, ALLOSTERIC REGULATION, SMALL COMPOUNDS, PIF-POCKET, TRANSFERASE