2aqb:B (VAL99) to (CYS194) STRUCTURE-ACTIVITY RELATIONSHIPS AT THE 5-POSITION OF THIOLACTOMYCIN: AN INTACT 5(R)-ISOPRENE UNIT IS REQUIRED FOR ACTIVITY AGAINST THE CONDENSING ENZYMES FROM MYCOBACTERIUM TUBERCULOSIS AND ESCHERCHIA COLI | FABB-LIGAND ACTIVE-SITE COMPLEX, TRANSFERASE
2aqb:C (VAL99) to (CYS194) STRUCTURE-ACTIVITY RELATIONSHIPS AT THE 5-POSITION OF THIOLACTOMYCIN: AN INTACT 5(R)-ISOPRENE UNIT IS REQUIRED FOR ACTIVITY AGAINST THE CONDENSING ENZYMES FROM MYCOBACTERIUM TUBERCULOSIS AND ESCHERCHIA COLI | FABB-LIGAND ACTIVE-SITE COMPLEX, TRANSFERASE
2pff:A (GLY1244) to (GLN1336) STRUCTURAL INSIGHTS OF YEAST FATTY ACID SYNTHASE | FATTY ACID SYNTHASE, ACYL-CARRIER-PROTEIN, BETA-KETOACYL REDUCTASE, BETA-KETOACYL SYNTHASE, DEHYDRATASE, ENOYL-[ACYL-CARRIER-PROTEIN] REDUCTASE, ACETYLTRANSFERASE, MALONYLTRANSFERASE, TRANSFERASE
2pff:D (GLY1244) to (GLN1336) STRUCTURAL INSIGHTS OF YEAST FATTY ACID SYNTHASE | FATTY ACID SYNTHASE, ACYL-CARRIER-PROTEIN, BETA-KETOACYL REDUCTASE, BETA-KETOACYL SYNTHASE, DEHYDRATASE, ENOYL-[ACYL-CARRIER-PROTEIN] REDUCTASE, ACETYLTRANSFERASE, MALONYLTRANSFERASE, TRANSFERASE
2pff:G (GLY1244) to (GLN1336) STRUCTURAL INSIGHTS OF YEAST FATTY ACID SYNTHASE | FATTY ACID SYNTHASE, ACYL-CARRIER-PROTEIN, BETA-KETOACYL REDUCTASE, BETA-KETOACYL SYNTHASE, DEHYDRATASE, ENOYL-[ACYL-CARRIER-PROTEIN] REDUCTASE, ACETYLTRANSFERASE, MALONYLTRANSFERASE, TRANSFERASE
4jga:A (THR114) to (THR209) X-RAY CRYSTAL STRUCTURE OF 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE 2 FROM RICKETTSIA RICKETTSII | STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE (SSGCID), SYNTHASE, TRANSFERASE
4jga:B (THR114) to (THR209) X-RAY CRYSTAL STRUCTURE OF 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE 2 FROM RICKETTSIA RICKETTSII | STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE (SSGCID), SYNTHASE, TRANSFERASE
2vb9:C (VAL99) to (CYS194) BETA-KETOACYL-ACP SYNTHASE I (KAS) FROM E. COLI, APO STRUCTURE | FATTY ACID BIOSYNTHESIS, CYTOPLASM, ANTIBIOTIC, TRANSFERASE, ACYLTRANSFERASE, LIPID SYNTHESIS, FATTY ACID SYNTHESIS
2vba:A (VAL99) to (CYS194) BETA-KETOACYL-ACP SYNTHASE I (KAS) FROM E. COLI WITH BOUND AMINO-THIAZOLE INHIBITOR | CYTOPLASM, ANTIBIOTIC, TRANSFERASE, AMINO-THIAZOLE, ACYLTRANSFERASE, LIPID SYNTHESIS, FATTY ACID SYNTHESIS, FATTY ACID BIOSYNTHESIS
2hg4:B (THR143) to (MSE229) STRUCTURE OF THE KETOSYNTHASE-ACYLTRANSFERASE DIDOMAIN OF MODULE 5 FROM DEBS. | KETOSYNTHASE, ACYLTRANSFERASE, MODULE 5, DEBS, TRANSFERASE
4ls5:A (VAL100) to (VAL186) CRYSTAL STRUCTURE OF BETA-KETOACYL-ACP SYNTHASE II (FABF) FROM BACILLUS SUBTILIS | KASII, KETOACYL SYNTHASE, CONDENSING ENZYME, FATTY ACID ELONGATION, TRANSFERASE
4ls5:B (VAL100) to (VAL186) CRYSTAL STRUCTURE OF BETA-KETOACYL-ACP SYNTHASE II (FABF) FROM BACILLUS SUBTILIS | KASII, KETOACYL SYNTHASE, CONDENSING ENZYME, FATTY ACID ELONGATION, TRANSFERASE
4ls6:A (VAL100) to (VAL186) CRYSTAL STRUCTURE OF BETA-KETOACYL-ACP SYNTHASE II (FABF) I108F MUTANT FROM BACILLUS SUBTILIS | KASII, KETOACYL SYNTHASE, FATTY ACID ELONGATION, CERULENIN RESISTANT, TRANSFERASE
4ls6:B (VAL100) to (VAL186) CRYSTAL STRUCTURE OF BETA-KETOACYL-ACP SYNTHASE II (FABF) I108F MUTANT FROM BACILLUS SUBTILIS | KASII, KETOACYL SYNTHASE, FATTY ACID ELONGATION, CERULENIN RESISTANT, TRANSFERASE
4ls7:A (VAL100) to (VAL186) CRYSTAL STRUCTURE OF BACILLUS SUBTILIS BETA-KETOACYL-ACP SYNTHASE II (FABF) IN A NON-COVALENT COMPLEX WITH CERULENIN | KASII, CONDENSING ENZYME, FATTY ACID ELONGATION, DRUG TARGET, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ls7:B (VAL100) to (VAL186) CRYSTAL STRUCTURE OF BACILLUS SUBTILIS BETA-KETOACYL-ACP SYNTHASE II (FABF) IN A NON-COVALENT COMPLEX WITH CERULENIN | KASII, CONDENSING ENZYME, FATTY ACID ELONGATION, DRUG TARGET, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ls8:A (VAL101) to (VAL187) CRYSTAL STRUCTURE OF BACILLUS SUBTILIS BETA-KETOACYL-ACP SYNTHASE II (FABF) IN A COVALENT COMPLEX WITH CERULENIN | KASII, KETOACYL SYNTHASE, CONDENSING ENZYME, FATTY ACID ELONGATION, CERULENIN, DRUG TARGET, TRANSFERASE
4ls8:B (VAL101) to (VAL187) CRYSTAL STRUCTURE OF BACILLUS SUBTILIS BETA-KETOACYL-ACP SYNTHASE II (FABF) IN A COVALENT COMPLEX WITH CERULENIN | KASII, KETOACYL SYNTHASE, CONDENSING ENZYME, FATTY ACID ELONGATION, CERULENIN, DRUG TARGET, TRANSFERASE
2ix4:A (THR146) to (VAL232) ARABIDOPSIS THALIANA MITOCHONDRIAL BETA-KETOACYL ACP SYNTHASE HEXANOIC ACID COMPLEX | BETA-KETOACYL-(ACYL CARRIER PROTEIN) SYNTHASE, LIPID METABOLISM, CONDENSING ENZYME, FATTY ACID ELONGATION, FATTY ACID BIOSYNTHESIS, LIPID SYNTHESIS, TRANSIT PEPTIDE, ACYLTRANSFERASE, SYNTHASE, TRANSFERASE, ACYL COMPLEX, MITOCHONDRION
4mz0:B (THR154) to (LEU239) STRUCTURE OF A KETOSYNTHASE-ACYLTRANSFERASE DI-DOMAIN FROM MODULE CURL OF THE CURACIN A POLYKETIDE SYNTHASE | KETOSYNTHASE, THIOLASE FOLD, ACYLTRANSFERASE, ALPHA/BETA HYDROLASE FOLD, EXTENSION OF POLYKETIDE INTERMEDIATE, TRANSFERASE
1w0i:A (THR146) to (SER238) ARABIDOPSIS THALIANA MITOCHONDRIAL KAS | BETA-KETOACYL-(ACYL CARRIER PROTEIN) SYNTHASE, CONDENSING ENZYME, FATTY ACID ELONGATION, LIPID METABOLISM, SYNTHASE
1w0i:B (THR146) to (ASP241) ARABIDOPSIS THALIANA MITOCHONDRIAL KAS | BETA-KETOACYL-(ACYL CARRIER PROTEIN) SYNTHASE, CONDENSING ENZYME, FATTY ACID ELONGATION, LIPID METABOLISM, SYNTHASE
1l8x:A (SER37) to (SER161) CRYSTAL STRUCTURE OF FERROCHELATASE FROM THE YEAST, SACCHAROMYCES CEREVISIAE, WITH COBALT(II) AS THE SUBSTRATE ION | FERROCHELATASE, HEME BIOSYNTHESIS, PROTOHEME, FERRO-LYASE, PORPHYRIN METALLATION, COBALT, MITOCHONDRIAL INNER MEMBRANE PROTEIN
4ope:A (ARG4337) to (SER4423) STREPTOMCYES ALBUS JA3453 OXAZOLOMYCIN KETOSYNTHASE DOMAIN OZMH KS7 | STRUCTURAL GENOMICS, PKS, OZMH, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, LIGASE, TRANSFERASE
4ope:C (ARG4337) to (SER4423) STREPTOMCYES ALBUS JA3453 OXAZOLOMYCIN KETOSYNTHASE DOMAIN OZMH KS7 | STRUCTURAL GENOMICS, PKS, OZMH, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, LIGASE, TRANSFERASE
4ope:D (ARG4337) to (SER4423) STREPTOMCYES ALBUS JA3453 OXAZOLOMYCIN KETOSYNTHASE DOMAIN OZMH KS7 | STRUCTURAL GENOMICS, PKS, OZMH, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, LIGASE, TRANSFERASE
3kzu:A (THR107) to (SER199) CRYSTAL STRUCTURE OF 3-OXOACYL-(ACYL CARRIER PROTEIN) SYNTHASE II FROM BRUCELLA MELITENSIS | ACYL CARRIER PROTEIN, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, SSGCID, ACYLTRANSFERASE, TRANSFERASE
3kzu:B (THR107) to (SER199) CRYSTAL STRUCTURE OF 3-OXOACYL-(ACYL CARRIER PROTEIN) SYNTHASE II FROM BRUCELLA MELITENSIS | ACYL CARRIER PROTEIN, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, SSGCID, ACYLTRANSFERASE, TRANSFERASE
3kzu:C (THR107) to (SER199) CRYSTAL STRUCTURE OF 3-OXOACYL-(ACYL CARRIER PROTEIN) SYNTHASE II FROM BRUCELLA MELITENSIS | ACYL CARRIER PROTEIN, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, SSGCID, ACYLTRANSFERASE, TRANSFERASE
4c6v:A (PHE108) to (GLY200) CRYSTAL STRUCTURE OF M. TUBERCULOSIS KASA IN COMPLEX WITH TLM5 (SOAK FOR 5 MIN) | TRANSFERASE, KAS ENZYME, TYPE 2 FATTY ACID BIOSYNTHESIS, MYCOLIC ACID SYNTHESIS, THIOLACTOMYCIN
3o04:A (VAL101) to (ILE195) CRYSTAL STRUCTURE OF THE BETA-KETO-ACYL CARRIER PROTEIN SYNTHASE II (LMO2201) FROM LISTERIA MONOCYTOGENES | CSGID, STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, 3-LAYER(ABA) SANDWICH, ACYLTRANSFERASE, TRANSFERASE
4ddo:A (THR109) to (ASP204) CRYSTAL STRUCTURE OF 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE II FROM BURKHOLDERIA VIETNAMIENSIS | SSGCID, 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE II, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, TRANSFERASE
3qea:Z (LYS72) to (GLU170) CRYSTAL STRUCTURE OF HUMAN EXONUCLEASE 1 EXO1 (WT) IN COMPLEX WITH DNA (COMPLEX II) | EXONUCLEASE, HYDROLASE-DNA COMPLEX
4f32:A (THR109) to (ASP204) CRYSTAL STRUCTURE OF 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE II FROM BURKHOLDERIA VIETNAMIENSIS IN COMPLEX WITH PLATENCIN | SSGCID, 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE II, PLATENCIN, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, TRANSFERASE-ANTIBIOTIC COMPLEX
4f32:B (THR109) to (ASP204) CRYSTAL STRUCTURE OF 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE II FROM BURKHOLDERIA VIETNAMIENSIS IN COMPLEX WITH PLATENCIN | SSGCID, 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE II, PLATENCIN, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, TRANSFERASE-ANTIBIOTIC COMPLEX
5ld8:B (PHE108) to (GLY200) GSK3011724A COCRYSTALLISED WITH MYCOBACTERIUM TUBERCULOSIS H37RV KASA | INHIBITOR, COMPLEX, KASA, MYCOBACTERIUM TUBERCULOSIS, TRANSFERASE
5sxo:A (VAL101) to (ILE195) 1.35 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF BETA-KETOACYL-ACP SYNTHASE II (FABF) FROM LISTERIA MONOCYTOGENES | KASII, FABF, CONDENSING ENZYME, TRANSFERASE
3e60:A (THR107) to (LEU193) CRYSTAL STRUCTURE OF 3-OXOACYL-(ACYL CARRIER PROTEIN) SYNTHASE II FROM BARTONELLA HENSELAE | SSGCID, DECODE, TRANSFERASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE
3e60:B (THR107) to (LEU193) CRYSTAL STRUCTURE OF 3-OXOACYL-(ACYL CARRIER PROTEIN) SYNTHASE II FROM BARTONELLA HENSELAE | SSGCID, DECODE, TRANSFERASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE
2c9h:A (THR131) to (CYS224) STRUCTURE OF MITOCHONDRIAL BETA-KETOACYL SYNTHASE | TRANSFERASE, FATTY ACID SYNTHESIS, MITOCHONDRIA, KETOACYL SYNTHASE
2vb8:A (VAL99) to (CYS194) BETA-KETOACYL-ACP SYNTHASE I (KAS) FROM E. COLI WITH BOUND INHIBITOR THIOLACTOMYCIN | CYTOPLASM, ANTIBIOTIC, TRANSFERASE, THIOLACTOMYCIN, ACYLTRANSFERASE, LIPID SYNTHESIS, FATTY ACID SYNTHESIS, FATTY ACID BIOSYNTHESIS
2vb7:A (VAL99) to (CYS194) BETA-KETOACYL-ACP SYNTHASE I (KAS) FROM E. COLI, APO STRUCTURE AFTER SOAK IN PEG SOLUTION | FATTY ACID BIOSYNTHESIS, CYTOPLASM, ANTIBIOTIC, TRANSFERASE, ACYLTRANSFERASE, LIPID SYNTHESIS, FATTY ACID SYNTHESIS
2vb7:C (VAL99) to (CYS194) BETA-KETOACYL-ACP SYNTHASE I (KAS) FROM E. COLI, APO STRUCTURE AFTER SOAK IN PEG SOLUTION | FATTY ACID BIOSYNTHESIS, CYTOPLASM, ANTIBIOTIC, TRANSFERASE, ACYLTRANSFERASE, LIPID SYNTHESIS, FATTY ACID SYNTHESIS
1tqy:B (MET98) to (ALA190) THE ACTINORHODIN KETOSYNTHASE/CHAIN LENGTH FACTOR | ALPHA-BETA-ALPHA-BETA-ALPHA, HETERODIMER, TRANSFERASE
1tqy:F (MET98) to (ALA190) THE ACTINORHODIN KETOSYNTHASE/CHAIN LENGTH FACTOR | ALPHA-BETA-ALPHA-BETA-ALPHA, HETERODIMER, TRANSFERASE
1tqy:H (MET98) to (ALA190) THE ACTINORHODIN KETOSYNTHASE/CHAIN LENGTH FACTOR | ALPHA-BETA-ALPHA-BETA-ALPHA, HETERODIMER, TRANSFERASE
2wgf:F (PHE108) to (GLY200) CRYSTAL STRUCTURE OF MYCOBACTERIUM TUBERCULOSIS C171Q KASA VARIANT | BETA KETOACYL SYNTHASE I, CYTOPLASM, TRANSFERASE, ACYLTRANSFERASE, LIPID SYNTHESIS, FATTY ACID BIOSYNTHESIS
2iwy:A (THR146) to (SER241) HUMAN MITOCHONDRIAL BETA-KETOACYL ACP SYNTHASE | MITOCHONDRIA, MITOCHONDRION, LIPID SYNTHESIS, FATTY ACID SYNTHESIS, FATTY ACID BIOSYNTHESIS, BETA-KETOACYL ACP SYNTHASE, TRANSIT PEPTIDE, ACYLTRANSFERASE, CLAISEN CONDENSATION, KAS, CERULENIN, TRANSFERASE, HOMO SAPIENS
2iwy:B (THR146) to (SER241) HUMAN MITOCHONDRIAL BETA-KETOACYL ACP SYNTHASE | MITOCHONDRIA, MITOCHONDRION, LIPID SYNTHESIS, FATTY ACID SYNTHESIS, FATTY ACID BIOSYNTHESIS, BETA-KETOACYL ACP SYNTHASE, TRANSIT PEPTIDE, ACYLTRANSFERASE, CLAISEN CONDENSATION, KAS, CERULENIN, TRANSFERASE, HOMO SAPIENS
2iwz:A (THR146) to (CYS239) HUMAN MITOCHONDRIAL BETA-KETOACYL ACP SYNTHASE COMPLEXED WITH HEXANOIC ACID | MITOCHONDRIA, MITOCHONDRION, LIPID SYNTHESIS, FATTY ACID SYNTHESIS, FATTY ACID BIOSYNTHESIS, BETA-KETOACYL ACP SYNTHASE, TRANSIT PEPTIDE, ACYLTRANSFERASE, CLAISEN CONDENSATION, KAS, CERULENIN, TRANSFERASE, HOMO SAPIENS
2iwz:B (THR146) to (CYS239) HUMAN MITOCHONDRIAL BETA-KETOACYL ACP SYNTHASE COMPLEXED WITH HEXANOIC ACID | MITOCHONDRIA, MITOCHONDRION, LIPID SYNTHESIS, FATTY ACID SYNTHESIS, FATTY ACID BIOSYNTHESIS, BETA-KETOACYL ACP SYNTHASE, TRANSIT PEPTIDE, ACYLTRANSFERASE, CLAISEN CONDENSATION, KAS, CERULENIN, TRANSFERASE, HOMO SAPIENS
4qyr:A (ASN2654) to (LEU2741) CRYSTAL STRUCTURE OF MGSE (2542-3153) OF AT-LESS POLYKETIDE SYNTHASE FROM STREPTOMYCES PLATENSIS | STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, ALPHA-BETA STRUCTURE, TRANSFERASE