1a2a:A (LEU2) to (LEU110) AGKISTROTOXIN, A PHOSPHOLIPASE A2-TYPE PRESYNAPTIC NEUROTOXIN FROM AGKISTRODON HALYS PALLAS | PRESYNAPTIC NEUROTOXIN, PHOSPHOLIPASE A2, HYDROLASE, LIPID DEGRADATION
1a2a:C (LEU2) to (ASN109) AGKISTROTOXIN, A PHOSPHOLIPASE A2-TYPE PRESYNAPTIC NEUROTOXIN FROM AGKISTRODON HALYS PALLAS | PRESYNAPTIC NEUROTOXIN, PHOSPHOLIPASE A2, HYDROLASE, LIPID DEGRADATION
1a2a:E (LEU2) to (ASN109) AGKISTROTOXIN, A PHOSPHOLIPASE A2-TYPE PRESYNAPTIC NEUROTOXIN FROM AGKISTRODON HALYS PALLAS | PRESYNAPTIC NEUROTOXIN, PHOSPHOLIPASE A2, HYDROLASE, LIPID DEGRADATION
1a2a:G (LEU2) to (ASN109) AGKISTROTOXIN, A PHOSPHOLIPASE A2-TYPE PRESYNAPTIC NEUROTOXIN FROM AGKISTRODON HALYS PALLAS | PRESYNAPTIC NEUROTOXIN, PHOSPHOLIPASE A2, HYDROLASE, LIPID DEGRADATION
2aoz:A (LEU2) to (ASN99) CRYSTAL STRUCTURE OF THE MYOTOXIN-II FROM ATROPOIDES NUMMIFER VENOM | X-RAY DIFFRATION, MYOTOXICITY, PHOSPHOLIPASE A2, ATROPOIDES NUMMIFER, TOXIN
2arm:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX OF PHOSPHOLIPASE A2 WITH A NATURAL COMPOUND ATROPINE AT 1.2 A RESOLUTION | ENZYME, COMPLEX, HYDROLASE
2ok9:A (PHE3) to (ASN109) PRTX-I-BPB | PRTX-I-BPB COMPLEX, LYS49-PLA2, BOTHROPS PIRAJAI, PIRATOXIN I
2ok9:B (PHE3) to (ASN109) PRTX-I-BPB | PRTX-I-BPB COMPLEX, LYS49-PLA2, BOTHROPS PIRAJAI, PIRATOXIN I
2oli:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN A GROUP II PHOSPHOLIPASE A2 AND AN INDOLE DERIVATIVE AT 2.2 A RESOLUTION | INHIBITOR, BINDING, HYDROLASE
1ae7:A (LEU2) to (ALA109) NOTEXIN, A PRESYNAPTIC NEUROTOXIC PHOSPHOLIPASE A2 | HYDROLASE, PHOSPHOLIPASE A2, LIPID DEGRADATION, PRESYNAPTIC NEUROTOXIN, VENOM
2b01:A (ALA1) to (ALA109) CRYSTAL STRUCTURE OF PORCINE PANCREATIC PHOSPHOLIPASE A2 IN COMPLEX WITH TAUROCHENODEOXYCHOLATE | BILE SALT, TAUROCHENODEOXYCHOLATE, CARBOXYLIC ESTER HYDROLASE, PLA2, PANCREATIC ENZYME, HYDROLASE
2b03:A (ALA1) to (LYS108) CRYSTAL STRUCTURE OF PORCINE PANCREATIC PHOSPHOLIPASE A2 IN COMPLEX WITH TAUROCHENODEOXYCHOLATE | BILE SALT, TAUROCHENODEOXYCHOLATE, CARBOXY ESTER HYDROLASE, PANCREATIC ENZYME, HYDROLASE
2b04:A (ALA1) to (ALA109) CRYSTAL STRUCTURE OF PORCINE PANCREATIC PHOSPHOLIPASE A2 IN COMPLEX WITH GLYCOCHENODEOXYCHOLATE | BILE SALT, GLYCOCHENODEOXYCHOLATE, CARBOXYLIC ESTER HYDROLASE, PANCREATIC ENZYME, HYDROLASE
4h0s:A (SER1) to (ASN109) CRYSTAL STRUCTURE ANALYSIS OF A BASIC PHOSPHOLIPASE A2 FROM TRIMERESURUS STEJNEGERI VENOM | ALPHA-HELIX, GLYCEROPHOSPHOLIPID, VENOM GLAND, HYDROLASE
4h0s:C (SER1) to (ASN109) CRYSTAL STRUCTURE ANALYSIS OF A BASIC PHOSPHOLIPASE A2 FROM TRIMERESURUS STEJNEGERI VENOM | ALPHA-HELIX, GLYCEROPHOSPHOLIPID, VENOM GLAND, HYDROLASE
2b17:A (SER1) to (ASN109) SPECIFIC BINDING OF NON-STEROIDAL ANTI-INFLAMMATORY DRUGS (NSAIDS) TO PHOSPHOLIPASE A2: CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND DICLOFENAC AT 2.7 A RESOLUTION: | DRUGS, BINDING, COMPLEX, INHIBITON, HYDROLASE
2oth:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF A TERNARY COMPLEX OF PHOSPHOLIPASE A2 WITH INDOMETHACIN AND NIMESULIDE AT 2.9 A RESOLUTION | COMPLEX, INHIBITOR, HYDROLASE
3elo:A (VAL2) to (ALA109) CRYSTAL STRUCTURE OF HUMAN PANCREATIC PROPHOSPHOLIPASE A2 | HUMAN PANCREATIC PROPHOSPHOLIPASE A2, TRIMERIC, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, SECRETED
2oyf:A (LEU2) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX OF PHOSPHOLIPASE A2 WITH INDOLE ACETIC ACID AT 1.2 A RESOLUTION | PHOSPHOLIPASE A2, INDOLE ACETIC ACID, CRYTSAL STRUCTURE, DABOIA RUSELLI PULCHELLA, HYDROLASE
1ayp:A (LEU2) to (ASN101) A PROBE MOLECULE COMPOSED OF SEVENTEEN PERCENT OF TOTAL DIFFRACTING MATTER GIVES CORRECT SOLUTIONS IN MOLECULAR REPLACEMENT | HYDROLASE
1ayp:C (VAL3) to (ASN101) A PROBE MOLECULE COMPOSED OF SEVENTEEN PERCENT OF TOTAL DIFFRACTING MATTER GIVES CORRECT SOLUTIONS IN MOLECULAR REPLACEMENT | HYDROLASE
1ayp:D (LEU2) to (ASN101) A PROBE MOLECULE COMPOSED OF SEVENTEEN PERCENT OF TOTAL DIFFRACTING MATTER GIVES CORRECT SOLUTIONS IN MOLECULAR REPLACEMENT | HYDROLASE
1ayp:E (LEU2) to (ASN101) A PROBE MOLECULE COMPOSED OF SEVENTEEN PERCENT OF TOTAL DIFFRACTING MATTER GIVES CORRECT SOLUTIONS IN MOLECULAR REPLACEMENT | HYDROLASE
1ayp:F (LEU2) to (LYS102) A PROBE MOLECULE COMPOSED OF SEVENTEEN PERCENT OF TOTAL DIFFRACTING MATTER GIVES CORRECT SOLUTIONS IN MOLECULAR REPLACEMENT | HYDROLASE
4wtb:A (SER1) to (LEU100) BTHTX-I, A SVPLA2S-LIKE TOXIN, COMPLEXED WITH ZINC IONS | SVPLA2-LIKE INHIBITOR, BTHTX-I, TOXIN
4wtb:B (SER1) to (LEU100) BTHTX-I, A SVPLA2S-LIKE TOXIN, COMPLEXED WITH ZINC IONS | SVPLA2-LIKE INHIBITOR, BTHTX-I, TOXIN
1b4w:A (LEU2) to (ASN109) BASIC PHOSPHOLIPASE A2 FROM AGKISTRODON HALYS PALLAS- IMPLICATIONS FOR ITS ASSOCIATION AND ANTICOAGULANT ACTIVITIES BY X-RAY CRYSTALLOGRAPHY | BASIC PHOSPHOLIPASE A2, AGKISTRODON HALYS PALLAS, DIMER, ANTICOAGULANT ACTIVITY, HYDROLASE
1b4w:B (LEU2) to (ASN109) BASIC PHOSPHOLIPASE A2 FROM AGKISTRODON HALYS PALLAS- IMPLICATIONS FOR ITS ASSOCIATION AND ANTICOAGULANT ACTIVITIES BY X-RAY CRYSTALLOGRAPHY | BASIC PHOSPHOLIPASE A2, AGKISTRODON HALYS PALLAS, DIMER, ANTICOAGULANT ACTIVITY, HYDROLASE
1b4w:C (LEU2) to (ASN109) BASIC PHOSPHOLIPASE A2 FROM AGKISTRODON HALYS PALLAS- IMPLICATIONS FOR ITS ASSOCIATION AND ANTICOAGULANT ACTIVITIES BY X-RAY CRYSTALLOGRAPHY | BASIC PHOSPHOLIPASE A2, AGKISTRODON HALYS PALLAS, DIMER, ANTICOAGULANT ACTIVITY, HYDROLASE
1b4w:D (LEU2) to (ASN109) BASIC PHOSPHOLIPASE A2 FROM AGKISTRODON HALYS PALLAS- IMPLICATIONS FOR ITS ASSOCIATION AND ANTICOAGULANT ACTIVITIES BY X-RAY CRYSTALLOGRAPHY | BASIC PHOSPHOLIPASE A2, AGKISTRODON HALYS PALLAS, DIMER, ANTICOAGULANT ACTIVITY, HYDROLASE
2pb8:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND PEPTIDE ALA-VAL-TYR-SER AT 2.0 A RESOLUTION | INHIBITOR, BINDING, HYDROLASE
4hmb:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX OF GROUP II PHOSPHOLIPASE A2 WITH A 3-{3-[(DIMETHYLAMINO)METHYL]-1H-INDOL-7-YL}PROPAN-1-OL AT 2.21 A RESOLUTION | PLA2, HYDROLASE
1bjj:A (LEU2) to (ASN109) AGKISTRODOTOXIN, A PHOSPHOLIPASE A2-TYPE PRESYNAPTIC NEUROTOXIN FROM AGKISTRODON HALYS PALLAS | PRESYNAPTIC NEUROTOXIN, PHOSPHOLIPASE A2, HYDROLASE
1bjj:C (LEU2) to (ASN109) AGKISTRODOTOXIN, A PHOSPHOLIPASE A2-TYPE PRESYNAPTIC NEUROTOXIN FROM AGKISTRODON HALYS PALLAS | PRESYNAPTIC NEUROTOXIN, PHOSPHOLIPASE A2, HYDROLASE
1bjj:D (LEU2) to (ASN109) AGKISTRODOTOXIN, A PHOSPHOLIPASE A2-TYPE PRESYNAPTIC NEUROTOXIN FROM AGKISTRODON HALYS PALLAS | PRESYNAPTIC NEUROTOXIN, PHOSPHOLIPASE A2, HYDROLASE
2ph4:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF A NOVEL ARG49 PHOSPHOLIPASE A2 HOMOLOGUE FROM ZHAOERMIA MANGSHANENSIS VENOM | SNAKE VENOM, ARG49, PHOSPHOLIPASE A2, MYOTOXIN, TOXIN
2ph4:B (SER1) to (LEU110) CRYSTAL STRUCTURE OF A NOVEL ARG49 PHOSPHOLIPASE A2 HOMOLOGUE FROM ZHAOERMIA MANGSHANENSIS VENOM | SNAKE VENOM, ARG49, PHOSPHOLIPASE A2, MYOTOXIN, TOXIN
2phi:A (LEU2) to (LYS108) A LARGE CONFORMATIONAL CHANGE IS FOUND IN THE CRYSTAL STRUCTURE OF THE PORCINE PANCREATIC PHOSPHOLIPASE A2 POINT MUTANT F63V | HYDROLASE (CARBOXYLIC ESTER)
1c1j:A (LEU2) to (ASN109) STRUCTURE OF CADMIUM-SUBSTITUTED PHOSPHOLIPASE A2 FROM AGKISTRONDON HALYS PALLAS AT 2.8 ANGSTROMS RESOLUTION | VENOM,PHOSPHOLIPASE A2,X-RAY CRYSTALLOGRAPHY,CADMIUM, CATALYTIC MECHANISM, HYDROLASE
1c1j:B (LEU2) to (ASN109) STRUCTURE OF CADMIUM-SUBSTITUTED PHOSPHOLIPASE A2 FROM AGKISTRONDON HALYS PALLAS AT 2.8 ANGSTROMS RESOLUTION | VENOM,PHOSPHOLIPASE A2,X-RAY CRYSTALLOGRAPHY,CADMIUM, CATALYTIC MECHANISM, HYDROLASE
1c1j:C (LEU2) to (ASN109) STRUCTURE OF CADMIUM-SUBSTITUTED PHOSPHOLIPASE A2 FROM AGKISTRONDON HALYS PALLAS AT 2.8 ANGSTROMS RESOLUTION | VENOM,PHOSPHOLIPASE A2,X-RAY CRYSTALLOGRAPHY,CADMIUM, CATALYTIC MECHANISM, HYDROLASE
1c1j:D (LEU2) to (ASN109) STRUCTURE OF CADMIUM-SUBSTITUTED PHOSPHOLIPASE A2 FROM AGKISTRONDON HALYS PALLAS AT 2.8 ANGSTROMS RESOLUTION | VENOM,PHOSPHOLIPASE A2,X-RAY CRYSTALLOGRAPHY,CADMIUM, CATALYTIC MECHANISM, HYDROLASE
2pmj:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND 1, 2 BENZOPYRONE AT 2.4 A RESOLUTION | COMPLEX, BINDING, HYDROLASE
3fg5:A (SER1) to (ASN109) CRYSTAL STRUCTURE DETERMINATION OF A TERNARY COMPLEX OF PHOSPHOLIPASE A2 WITH A PENTAPETIDE FLSYK AND AJMALINE AT 2.5 A RESOLUTION | PLA2, PENTAPEPTIDE, FLSYK, AJMALINE, TERNARY COMPLEX, HYDROLASE
1ceh:A (LEU2) to (LYS108) STRUCTURE AND FUNCTION OF THE CATALYTIC SITE MUTANT ASP99ASN OF PHOSPHOLIPASE A2: ABSENCE OF CONSERVED STRUCTURAL WATER | HYDROLASE (CARBOXYLIC ESTER)
2pvt:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF A NEW ISOFORM OF PHOSPHOLIPASE A2 FROM RUSSELLS VIPER AT 2.1 A RESOLUTION | CATALYSIS, ACTIVE SITE, ISOFORM, HYDROLASE
2pyc:A (LEU2) to (ASN109) CRYSTAL STRUCTURE OF A MONOMERIC PHOSPHOLIPASE A2 FROM RUSSELL'S VIPER AT 1.5A RESOLUTION | ACTIVE SITE, TOXIN, HYDROLASE
1oqs:D (ASN1) to (ASN109) CRYSTAL STRUCTURE OF RV4/RV7 COMPLEX | HYDROLASE
1oqs:F (LEU2) to (ASN109) CRYSTAL STRUCTURE OF RV4/RV7 COMPLEX | HYDROLASE
1oqs:H (LEU2) to (ASN109) CRYSTAL STRUCTURE OF RV4/RV7 COMPLEX | HYDROLASE
1cl5:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 FROM DABOIA RUSSELLI PULCHELLA | PHOSPHOLIPASE A2, X-RAY STRUCTURE, NEUROTOXIC, DABOIA RUSSELLI PULCHELLA, HYDROLASE
1clp:A (SER1) to (GLU108) CRYSTAL STRUCTURE OF A CALCIUM-INDEPENDENT PHOSPHOLIPASELIKE MYOTOXIC PROTEIN FROM BOTHROPS ASPER VENOM | HYDROLASE
1clp:B (SER1) to (LEU110) CRYSTAL STRUCTURE OF A CALCIUM-INDEPENDENT PHOSPHOLIPASELIKE MYOTOXIC PROTEIN FROM BOTHROPS ASPER VENOM | HYDROLASE
2q1p:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 COMPLEX WITH PROPANOL AT 1.5 A RESOLUTION | PHOSPHOLIPASE A2, PROPANOL, HYDROLASE
2q2j:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF PRTX-I, A PLA2 HOMOLOG FROM BOTHROPS PIRAJAI | MYOTOXIN, PLA2 LIKE, LYS49-PLA2, PHOSPHOLIPASE A2
2q2j:B (PHE3) to (ASN109) CRYSTAL STRUCTURE OF PRTX-I, A PLA2 HOMOLOG FROM BOTHROPS PIRAJAI | MYOTOXIN, PLA2 LIKE, LYS49-PLA2, PHOSPHOLIPASE A2
1oxl:A (SER1) to (ASN109) INHIBITION OF PHOSPHOLIPASE A2 (PLA2) BY (2-CARBAMOYLMETHYL- 5-PROPYL-OCTAHYDRO-INDOL-7-YL)-ACETIC ACID (INDOLE): CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PLA2 FROM RUSSELL'S VIPER AND INDOLE AT 1.8 RESOLUTION | PHOSPHOLIPASE A2, INDOLE DERIVATIVE, INHIBITION, CRYSTAL STRUCTURE, HYDROLASE
1oxl:B (SER1) to (ASN109) INHIBITION OF PHOSPHOLIPASE A2 (PLA2) BY (2-CARBAMOYLMETHYL- 5-PROPYL-OCTAHYDRO-INDOL-7-YL)-ACETIC ACID (INDOLE): CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PLA2 FROM RUSSELL'S VIPER AND INDOLE AT 1.8 RESOLUTION | PHOSPHOLIPASE A2, INDOLE DERIVATIVE, INHIBITION, CRYSTAL STRUCTURE, HYDROLASE
1oxr:A (LEU2) to (GLY103) ASPIRIN INDUCES ITS ANTI-INFLAMMATORY EFFECTS THROUGH ITS SPECIFIC BINDING TO PHOSPHOLIPASE A2: CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND ASPIRIN AT 1.9A RESOLUTION | O-ACETYL-OXY PHENOL, COMPLEX, PLA2, NAJA NAJA SAGITTIFERA, CRYSTAL STRUCTURE, HYDROLASE
3fvi:A (ALA1) to (ALA109) CRYSTAL STRUCTURE OF COMPLEX OF PHOSPHOLIPASE A2 WITH OCTYL SULFATES | PHOSPHOLIPASE A2, PLA2-1B, OCTYL SULFATE BINDING, PROTEIN DETERGENT AGGREGATES, HYDROLASE, LIPID DEGRADATION, LIPOPROTEIN, METAL- BINDING, PALMITATE, PYRROLIDONE CARBOXYLIC ACID, SECRETED
3fvi:B (LEU2) to (ALA109) CRYSTAL STRUCTURE OF COMPLEX OF PHOSPHOLIPASE A2 WITH OCTYL SULFATES | PHOSPHOLIPASE A2, PLA2-1B, OCTYL SULFATE BINDING, PROTEIN DETERGENT AGGREGATES, HYDROLASE, LIPID DEGRADATION, LIPOPROTEIN, METAL- BINDING, PALMITATE, PYRROLIDONE CARBOXYLIC ACID, SECRETED
3fvi:C (ALA1) to (LYS108) CRYSTAL STRUCTURE OF COMPLEX OF PHOSPHOLIPASE A2 WITH OCTYL SULFATES | PHOSPHOLIPASE A2, PLA2-1B, OCTYL SULFATE BINDING, PROTEIN DETERGENT AGGREGATES, HYDROLASE, LIPID DEGRADATION, LIPOPROTEIN, METAL- BINDING, PALMITATE, PYRROLIDONE CARBOXYLIC ACID, SECRETED
3fvi:D (ALA1) to (ALA109) CRYSTAL STRUCTURE OF COMPLEX OF PHOSPHOLIPASE A2 WITH OCTYL SULFATES | PHOSPHOLIPASE A2, PLA2-1B, OCTYL SULFATE BINDING, PROTEIN DETERGENT AGGREGATES, HYDROLASE, LIPID DEGRADATION, LIPOPROTEIN, METAL- BINDING, PALMITATE, PYRROLIDONE CARBOXYLIC ACID, SECRETED
3fvj:A (ALA1) to (LYS108) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 1B CRYSTALLIZED IN THE PRESENCE OF OCTYL SULFATE | PHOSPHOLIPASE A2, PLA2-1B, OCTYL SULFATE BINDING, HYDROLASE, LIPID DEGRADATION, LIPOPROTEIN, METAL-BINDING, PALMITATE, PYRROLIDONE CARBOXYLIC ACID, SECRETED
1ozy:A (ASN1) to (LYS108) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 (MIPLA3) FROM MICROPECHIS IKAHEKA | PHOSPHOLIPASE A2, MICROPECHIS IKAHEKA, PANCREATIC LOOP, HYDROLASE
1ozy:B (ASN1) to (LYS108) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 (MIPLA3) FROM MICROPECHIS IKAHEKA | PHOSPHOLIPASE A2, MICROPECHIS IKAHEKA, PANCREATIC LOOP, HYDROLASE
1p2p:A (ALA1) to (ALA109) STRUCTURE OF PORCINE PANCREATIC PHOSPHOLIPASE A2 AT 2.6 ANGSTROMS RESOLUTION AND COMPARISON WITH BOVINE PHOSPHOLIPASE A2 | CARBOXYLIC ESTER HYDROLASE
1p7o:A (ASN1) to (ALA109) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 (MIPLA4) FROM MICROPECHIS IKAHEKA | PHOSPHOLIPASE A2, MICROPECHIS IKAHEKA, PANCREATIC LOOP, HYDROLASE
1p7o:C (ASN1) to (ALA109) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 (MIPLA4) FROM MICROPECHIS IKAHEKA | PHOSPHOLIPASE A2, MICROPECHIS IKAHEKA, PANCREATIC LOOP, HYDROLASE
1p7o:D (ASN1) to (ALA109) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 (MIPLA4) FROM MICROPECHIS IKAHEKA | PHOSPHOLIPASE A2, MICROPECHIS IKAHEKA, PANCREATIC LOOP, HYDROLASE
1p7o:E (ASN1) to (LYS108) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 (MIPLA4) FROM MICROPECHIS IKAHEKA | PHOSPHOLIPASE A2, MICROPECHIS IKAHEKA, PANCREATIC LOOP, HYDROLASE
1p7o:F (LEU2) to (ALA109) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 (MIPLA4) FROM MICROPECHIS IKAHEKA | PHOSPHOLIPASE A2, MICROPECHIS IKAHEKA, PANCREATIC LOOP, HYDROLASE
1db4:A (LEU2) to (ASN101) HUMAN S-PLA2 IN COMPLEX WITH INDOLE 8 | S-PLA2, STRUCTURE-BASED DRUG DESIGN, HYDROLASE/HYDROLASE INHIBITOR
1pa0:A (SER1) to (LEU110) CRYSTAL STRUCTURE OF BNSP-7, A LYS49-PHOSPHOLIPASE A2 | LYS49-PHOSPHOLIPASE A2, MYOTOXIN, CRYSTAL STRUCTURE, BOTHROPIC VENOM, HYDROLASE
1pa0:B (SER1) to (ASN109) CRYSTAL STRUCTURE OF BNSP-7, A LYS49-PHOSPHOLIPASE A2 | LYS49-PHOSPHOLIPASE A2, MYOTOXIN, CRYSTAL STRUCTURE, BOTHROPIC VENOM, HYDROLASE
1pc9:B (SER1) to (ASN109) CRYSTAL STRUCTURE OF BNSP-6, A LYS49-PHOSPHOLIPASE A2 | LYS49-PHOSPHOLIPASE A2, MYOTOXIN, CRYSTAL STRUCTURE, BOTHROPS, VENOM., HYDROLASE
2qhd:A (VAL2) to (ASN109) CRYSTAL STRUCTURE OF ECARPHOLIN S (SER49-PLA2) COMPLEXED WITH FATTY ACID | BETA SHEET, THREE HELICES, PROTEIN-LIGAND COMPLEX, HYDROLASE
2qhd:B (SER1) to (ASN109) CRYSTAL STRUCTURE OF ECARPHOLIN S (SER49-PLA2) COMPLEXED WITH FATTY ACID | BETA SHEET, THREE HELICES, PROTEIN-LIGAND COMPLEX, HYDROLASE
2qhw:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF A COMPLEX OF PHOSPHOLIPASE A2 WITH A GRAMINE DERIVATIVE AT 2.2 RESOLUTION | ACTIVE SITE, INHIBITOR, HYDROLASE
3t0r:A (VAL3) to (ASN109) CRYSTAL STRUCTURE OF MJTX-I, A MYOTOXIC LYS49-PHOSPHOLIPASE A2 FROM BOTHROPS MOOJENI | LYS49-PHOSPHOLIPASE A2, MYOTOXIN, VENOM GLANDS, TOXIN
3t0r:B (SER1) to (ASN109) CRYSTAL STRUCTURE OF MJTX-I, A MYOTOXIC LYS49-PHOSPHOLIPASE A2 FROM BOTHROPS MOOJENI | LYS49-PHOSPHOLIPASE A2, MYOTOXIN, VENOM GLANDS, TOXIN
3t0r:C (SER1) to (LYS110) CRYSTAL STRUCTURE OF MJTX-I, A MYOTOXIC LYS49-PHOSPHOLIPASE A2 FROM BOTHROPS MOOJENI | LYS49-PHOSPHOLIPASE A2, MYOTOXIN, VENOM GLANDS, TOXIN
3t0r:D (SER1) to (ASN109) CRYSTAL STRUCTURE OF MJTX-I, A MYOTOXIC LYS49-PHOSPHOLIPASE A2 FROM BOTHROPS MOOJENI | LYS49-PHOSPHOLIPASE A2, MYOTOXIN, VENOM GLANDS, TOXIN
3g8f:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN A GROUP II PHOSPHOLIPASE A2 AND DESIGNED PEPTIDE INHIBITOR CARBOBENZOXY-DEHYDRO- VAL-ALA-ARG-SER AT 1.2 A RESOLUTION | PHOSPHOLIPASE A2, CRYSTAL STRUCTRE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3g8g:A (SER1) to (ASN99) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 AMMODYTOXIN A FROM VIPERA AMMODYTES AMMODYTES | PHOSPHOLIPASE A2, AMMODYTOXIN, PRESYNAPTIC NEUROTOXIN, ANTICOAGULANT, SNAKE VENOM, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, SECRETED, NEUROTOXIN, TOXIN
3g8h:A (SER1) to (ASN99) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 AMMODYTOXIN C FROM VIPERA AMMODYTES AMMODYTES | PHOSPHOLIPASE A2, AMMODYTOXIN, PRESYNAPTIC NEUROTOXIN, ANTICOAGULANT, SNAKE VENOM, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, SECRETED, NEUROTOXIN, TOXIN
3gci:A (ASN1) to (ALA104) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN A NEW ISOFORM OF PHOSPHOLIPASE A2 WITH C-TERMINAL AMYLOID BETA HEPTAPEPTIDE AT 2 A RESOLUTION | PHOSPHOLIPASE A2, HEPTAPEPTIDE, AMYLOID BETA, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, SECRETED
1dpy:A (ASN1) to (SER103) THREE-DIMENSIONAL STRUCTURE OF A NOVEL PHOSPHOLIPASE A2 FROM INDIAN COMMON KRAIT AT 2.45 A RESOLUTION | INDIAN COMMON KRAIT VENOM, PHOSPHOLIPASE A2, CRYSTAL STRUCTURE, REFINEMENT, HYDROLASE
1po8:A (ASN1) to (LYS103) CRYSTAL STRUCTURE OF A COMPLEX FORMED BETWEEN KRAIT VENOM PHOSPHOLIPASE A2 AND HEPTANOIC ACID AT 2.7 A RESOLUTION. | PHOSPHOLIPASE A2, CRYSTAL STRUCTURE,INHIBITOR,COMPLEX, HYDROLASE
1pod:A (LEU2) to (ASN101) STRUCTURES OF FREE AND INHIBITED HUMAN SECRETORY PHOSPHOLIPASE A2 FROM INFLAMMATORY EXUDATE | HYDROLASE
1poe:A (LEU2) to (ASN101) STRUCTURES OF FREE AND INHIBITED HUMAN SECRETORY PHOSPHOLIPASE A2 FROM INFLAMMATORY EXUDATE | HYDROLASE
1poe:B (LEU2) to (ASN101) STRUCTURES OF FREE AND INHIBITED HUMAN SECRETORY PHOSPHOLIPASE A2 FROM INFLAMMATORY EXUDATE | HYDROLASE
1pp2:L (SER1) to (ASN109) THE REFINED CRYSTAL STRUCTURE OF DIMERIC PHOSPHOLIPASE A2 AT 2.5 ANGSTROMS. ACCESS TO A SHIELDED CATALYTIC CENTER | HYDROLASE
1ppa:A (VAL2) to (ASN109) THE CRYSTAL STRUCTURE OF A LYSINE 49 PHOSPHOLIPASE A2 FROM THE VENOM OF THE COTTONMOUTH SNAKE AT 2.0 ANGSTROMS RESOLUTION | HYDROLASE(CARBOXYLIC ESTERASE)
2qu9:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX OF GROUP II PHOSPHOLIPASE A2 WITH EUGENOL | PLA2, EUGENOL, COMPLEX, CALCIUM, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, NEUROTOXIN, PRESYNAPTIC NEUROTOXIN, SECRETED, TOXIN
2que:A (SER1) to (ASN109) SATURATION OF SUBSTRATE-BINDING SITE USING TWO NATURAL LIGANDS: CRYSTAL STRUCTURE OF A TERNARY COMPLEX OF PHOSPHOLIPASE A2 WITH ANISIC ACID AND AJMALINE AT 2.25 A RESOLUTION | ACTIVE SITE, LIPID HYDROLYSIS, BINDING AFFINITY, CALCIUM, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, NEUROTOXIN, PRESYNAPTIC NEUROTOXIN, SECRETED, TOXIN
2qvd:A (SER1) to (ASN109) IDENTIFICATION OF A POTENT ANTI-INFLAMMATORY AGENT FROM THE NATURAL EXTRACT OF PLANT CARDIOSPERMUN HELICACABUM: CRYSTAL STRUCTURE OF THE COMPLEX OF PHOSPHOLIPASE A2 WITH BENZO(G)-1,3-BENZODIOXOLO(5,6-A) QUINOLIZINIUM, 5,6-DIHYDRO-9,10-DIMETHOXY AT 1.93 A RESOLUTION | PHOSPHOLIPIDS, MEMBRANE, HYDROLYSIS, INHIBITOR, PLANT EXTRAXT, LIPID DEGRADATION, METAL-BINDING, NEUROTOXIN, PRESYNAPTIC NEUROTOXIN, SECRETED, TOXIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1pwo:A (ASN1) to (ALA109) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 (MIPLA2) FROM MICROPECHIS IKAHEKA | PHOSPHOLIPASE A2, MICROPECHIS IKAHEKA, PANCREATIC LOOP, HYDROLASE
1pwo:B (ASN1) to (ALA109) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 (MIPLA2) FROM MICROPECHIS IKAHEKA | PHOSPHOLIPASE A2, MICROPECHIS IKAHEKA, PANCREATIC LOOP, HYDROLASE
1pwo:C (ASN1) to (LYS108) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 (MIPLA2) FROM MICROPECHIS IKAHEKA | PHOSPHOLIPASE A2, MICROPECHIS IKAHEKA, PANCREATIC LOOP, HYDROLASE
1pwo:D (ASN1) to (LYS108) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 (MIPLA2) FROM MICROPECHIS IKAHEKA | PHOSPHOLIPASE A2, MICROPECHIS IKAHEKA, PANCREATIC LOOP, HYDROLASE
2do2:A (SER1) to (ASN109) DESIGN OF SPECIFIC INHIBITORS OF PHOSPHOLIPASE A2: CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN A GROUP II CYS 49 PHOSPHOLIPASE A2 AND A DESIGNED PENTAPEPTIDE ALA-LEU-ALA- SER-LYS AT 2.6A RESOLUTION | CYS 49 PHOSPHOLIPASE A2, SYNTHETIC PENTAPEPTIDE, COMPLEX, HYDROLASE
2dpz:A (LEU2) to (ASN109) STRUCTURE OF THE COMPLEX OF PHOSPHOLIPASE A2 WITH N-(4- HYDROXYPHENYL)- ACETAMIDE AT 2.1 A RESOLUTION | NSAIDS, COMPLEX, HYDROLASE
1q7a:A (LEU2) to (ASN99) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN RUSSELL'S VIPER PHOSPHOLIPASE A2 AND AN ANTIINFLAMMATORY AGENT OXYPHENBUTAZONE AT 1.6A RESOLUTION | PHOSPHOLIPASE A2, VENOM, ANTIINFLAMMATORY COMPOUND, HYDROLASE
1qll:A (SER1) to (ASN99) PIRATOXIN-II (PRTX-II) - A K49 PLA2 FROM BOTHROPS PIRAJAI | NEUROTOXIN, K49 PHOSPHOLIPASE A2 (PLA2)
1qll:B (SER1) to (ASN99) PIRATOXIN-II (PRTX-II) - A K49 PLA2 FROM BOTHROPS PIRAJAI | NEUROTOXIN, K49 PHOSPHOLIPASE A2 (PLA2)
3u8b:A (LEU2) to (ASN101) FUNCTIONALLY SELECTIVE INHIBITION OF GROUP IIA PHOSPHOLIPASE A2 REVEALS A ROLE FOR VIMENTIN IN REGULATING ARACHIDONIC ACID METABOLISM | SECRETED PHOSPHOLIPASE A2, PHOSPHOLIPASE A2 ACTIVITY, HYDROLASE
3u8i:A (LEU2) to (ASN101) FUNCTIONALLY SELECTIVE INHIBITION OF GROUP IIA PHOSPHOLIPASE A2 REVEALS A ROLE FOR VIMENTIN IN REGULATING ARACHIDONIC ACID METABOLISM | SECRETED PHOSPHOLIPASE A2, HYDROLASE
3u8i:B (LEU2) to (ASN101) FUNCTIONALLY SELECTIVE INHIBITION OF GROUP IIA PHOSPHOLIPASE A2 REVEALS A ROLE FOR VIMENTIN IN REGULATING ARACHIDONIC ACID METABOLISM | SECRETED PHOSPHOLIPASE A2, HYDROLASE
3u8h:A (ASN1) to (ASN101) FUNCTIONALLY SELECTIVE INHIBITION OF GROUP IIA PHOSPHOLIPASE A2 REVEALS A ROLE FOR VIMENTIN IN REGULATING ARACHIDONIC ACID METABOLISM | SECRETED PHOSPHOLIPASE A2, PHOSPHOLIPASE A2 ACTIVITY, HYDROLASE
3u8h:B (ASN1) to (ASN101) FUNCTIONALLY SELECTIVE INHIBITION OF GROUP IIA PHOSPHOLIPASE A2 REVEALS A ROLE FOR VIMENTIN IN REGULATING ARACHIDONIC ACID METABOLISM | SECRETED PHOSPHOLIPASE A2, PHOSPHOLIPASE A2 ACTIVITY, HYDROLASE
1fe5:A (ASN1) to (SER103) SEQUENCE AND CRYSTAL STRUCTURE OF A BASIC PHOSPHOLIPASE A2 FROM COMMON KRAIT (BUNGARUS CAERULEUS) AT 2.4 RESOLUTION: IDENTIFICATION AND CHARACTERIZATION OF ITS PHARMACOLOGICAL SITES. | BUNGARUS CAERULEUS; PHOSPHOLIPASE A2 (PLA2); PRESYNAPTIC NEUROTOXIN; NEUROTOXIC SITE; X-RAY STRUCTURE; MOLECULAR REPLACEMENT
4k06:A (SER1) to (ASN110) CRYSTAL STRUCTURE OF MTX-II FROM BOTHROPS BRAZILI VENOM COMPLEXED WITH POLYETHYLENE GLYCOL | PHOSPHOLIPASE A2, TOXIN
4k06:B (PHE3) to (ASN109) CRYSTAL STRUCTURE OF MTX-II FROM BOTHROPS BRAZILI VENOM COMPLEXED WITH POLYETHYLENE GLYCOL | PHOSPHOLIPASE A2, TOXIN
4k09:A (SER1) to (LEU110) CRYSTAL STRUCTURE OF BBTX-II FROM BOTHROPS BRAZILI VENOM | PHOSPHOLIPASES A2, TOXIN
4k09:B (SER1) to (LEU110) CRYSTAL STRUCTURE OF BBTX-II FROM BOTHROPS BRAZILI VENOM | PHOSPHOLIPASES A2, TOXIN
3hhm:A (THR876) to (SER965) CRYSTAL STRUCTURE OF P110ALPHA H1047R MUTANT IN COMPLEX WITH NISH2 OF P85ALPHA AND THE DRUG WORTMANNIN | P110, P85, PI3KCA, PI3K, PIK3R1, PHOSPHATIDILYNOSITOL 3,4,5- TRIPHOSPHATE, WORTMANNIN, H1047R, ATP-BINDING, DISEASE MUTATION, KINASE, NUCLEOTIDE-BINDING, ONCOGENE, POLYMORPHISM, TRANSFERASE, TRANSFERASE/ONCOPROTEIN COMPLEX
4yu7:B (SER1) to (ASN99) CRYSTAL STRUCTURE OF PIRATOXIN I (PRTX-I) COMPLEXED TO CAFFEIC ACID | PHOSPHOLIPASE A2 PHOSPHOLIPASE A2-LIKE BOTHROPS SNAKE VENOM INHIBITOR, TOXIN
4yu7:A (SER1) to (ASN99) CRYSTAL STRUCTURE OF PIRATOXIN I (PRTX-I) COMPLEXED TO CAFFEIC ACID | PHOSPHOLIPASE A2 PHOSPHOLIPASE A2-LIKE BOTHROPS SNAKE VENOM INHIBITOR, TOXIN
1rgb:A (ASN1) to (ASN109) PHOSPHOLIPASE A2 FROM VIPERA AMMODYTES MERIDIONALIS | PHOSPHOLIPASE A2, NEUROTOXIN, ELAIDOYLAMIDE, HYDROLASE
1rgb:B (ASN1) to (ASN109) PHOSPHOLIPASE A2 FROM VIPERA AMMODYTES MERIDIONALIS | PHOSPHOLIPASE A2, NEUROTOXIN, ELAIDOYLAMIDE, HYDROLASE
1rgb:L (ASN1) to (LYS110) PHOSPHOLIPASE A2 FROM VIPERA AMMODYTES MERIDIONALIS | PHOSPHOLIPASE A2, NEUROTOXIN, ELAIDOYLAMIDE, HYDROLASE
1fv0:A (SER1) to (ASN109) FIRST STRUCTURAL EVIDENCE OF THE INHIBITION OF PHOSPHOLIPASE A2 BY ARISTOLOCHIC ACID: CRYSTAL STRUCTURE OF A COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND ARISTOLOCHIC ACID | PHOSPHOLIPASE A2, DABOIA RUSSELLI PULCHELLA, NEUROTOXIC, EDEMA, TOXIN
1fv0:B (LEU3) to (ASN109) FIRST STRUCTURAL EVIDENCE OF THE INHIBITION OF PHOSPHOLIPASE A2 BY ARISTOLOCHIC ACID: CRYSTAL STRUCTURE OF A COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND ARISTOLOCHIC ACID | PHOSPHOLIPASE A2, DABOIA RUSSELLI PULCHELLA, NEUROTOXIC, EDEMA, TOXIN
1fx9:A (ALA1) to (LYS108) CARBOXYLIC ESTER HYDROLASE COMPLEX (DIMERIC PLA2 + MJ33 INHIBITOR + SULPHATE IONS) | HYDROLASE, ENZYME, CARBOXYLIC ESTER HYDROLASE, DIMER, SULPHATE BINDING, INHIBITOR BINDING
1fx9:B (ALA1) to (LYS108) CARBOXYLIC ESTER HYDROLASE COMPLEX (DIMERIC PLA2 + MJ33 INHIBITOR + SULPHATE IONS) | HYDROLASE, ENZYME, CARBOXYLIC ESTER HYDROLASE, DIMER, SULPHATE BINDING, INHIBITOR BINDING
1fxf:A (ALA1) to (LYS108) CARBOXYLIC ESTER HYDROLASE COMPLEX (DIMERIC PLA2 + MJ33 INHIBITOR + PHOSPHATE IONS) | HYDROLASE, ENZYME, CARBOXYLIC ESTER HYDROLASE, DIMER, PHOSPHATE BINDING, INHIBITOR BINDING
1fxf:B (ALA1) to (LYS108) CARBOXYLIC ESTER HYDROLASE COMPLEX (DIMERIC PLA2 + MJ33 INHIBITOR + PHOSPHATE IONS) | HYDROLASE, ENZYME, CARBOXYLIC ESTER HYDROLASE, DIMER, PHOSPHATE BINDING, INHIBITOR BINDING
4kf3:B (SER1) to (ASN109) CRYSTAL STRUCTURE OF MYOTOXIN II (MJTX-II), A MYOTOXIC LYS49- PHOSPHOLIPASE A2 FROM BOTHROPS MOOJENI. | PHOSPHOLIPASE A2-LIKE MYOTOXIN, TOXIN, VENOM GLANDS
4kf3:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF MYOTOXIN II (MJTX-II), A MYOTOXIC LYS49- PHOSPHOLIPASE A2 FROM BOTHROPS MOOJENI. | PHOSPHOLIPASE A2-LIKE MYOTOXIN, TOXIN, VENOM GLANDS
1g2x:C (LEU2) to (SER103) SEQUENCE INDUCED TRIMERIZATION OF KRAIT PLA2: CRYSTAL STRUCTURE OF THE TRIMERIC FORM OF KRAIT PLA2 | STRUCTURE, PHOSPHOLIPASE A2, HOMOTRIMER, BUNGARUS CAERULEUS, TOXIN
3ux7:H (VAL2) to (ASN99) CRYSTAL STRUCTURE OF A DIMERIC MYOTOXIC COMPONENT OF THE VIPERA AMMODYTES MERIDIONALIS VENOM REVEALS DETERMINANTS OF MYOTOXICITY AND MEMBRANE DAMAGING ACTIVITY | TOXIN, SNAKE VENOM, SER49 MYOTOXIN
3hsw:A (ALA1) to (LYS108) CRYSTAL STRUCTURE OF PORCINE PANCREATIC PHOSPHOLIPASE A2 IN COMPLEX WITH 2-METHOXYCYCLOHEXA-2-5-DIENE-1,4-DIONE | HYDROLASE, CURCUMIN BINDING, PLA2, PANCREATIC ENZYME, DISULFIDE BOND, LIPID DEGRADATION, LIPOPROTEIN, METAL-BINDING, PALMITATE, PYRROLIDONE CARBOXYLIC ACID, SECRETED
1gh4:A (LEU2) to (LYS108) STRUCTURE OF THE TRIPLE MUTANT (K56M, K120M, K121M) OF PHOSPHOLIPASE A2 | ALPHA HELIX, BETA SHEET, TRIPLE MUTANT, HYDROLASE
1s8g:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF LYS49-PHOSPHOLIPASE A2 FROM AGKISTRODON CONTORTRIX LATICINCTUS, FATTY ACID BOUND FORM | LYS49-PHOSPHOLIPASE A2, SNAKE VENOM, MYOTOXICITY, FATTY ACID BOUND FORM, HYDROLASE, TOXIN
1s8i:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF LYS49-PHOSPHOLIPASE A2 FROM AGKISTRODON CONTORTRIX LATICINCTUS, SECOND FATTY ACID FREE FORM | LYS49-PHOSPHOLIPASE A2, SNAKE VENOM, MYOTOXICITY, FATTY ACID FREE FORM, HYDROLASE, TOXIN
3hzd:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF BOTHROPSTOXIN-I (BTHTX-I), A PLA2 HOMOLOGUE FROM BOTHROPS JARARACUSSU VENOM | BOTHROPS, SNAKE VENOM, PHOSPHOLIPASE A2, LYS49-PLA2S, MYOTOXICITY, ANTIBIOTIC, ANTIMICROBIAL, DISULFIDE BOND, MYOTOXIN, SECRETED, TOXIN
3hzd:B (SER1) to (ASN109) CRYSTAL STRUCTURE OF BOTHROPSTOXIN-I (BTHTX-I), A PLA2 HOMOLOGUE FROM BOTHROPS JARARACUSSU VENOM | BOTHROPS, SNAKE VENOM, PHOSPHOLIPASE A2, LYS49-PLA2S, MYOTOXICITY, ANTIBIOTIC, ANTIMICROBIAL, DISULFIDE BOND, MYOTOXIN, SECRETED, TOXIN
1god:A (SER1) to (ASN109) MONOMERIC LYS-49 PHOSPHOLIPASE A2 HOMOLOGUE ISOLATED FROM THE VENOM OF CERROPHIDION (BOTHROPS) GODMANI | LYS49-PHOSPHOLIPASE A2, SNAKE VENOM, BOTHROPS, HYDROLASE
3i03:A (SER1) to (ASN99) CRYSTAL STRUCTURE OF BOTHROPSTOXIN-I CHEMICALLY MODIFIED BY P- BROMOPHENACYL BROMIDE (BPB) - MONOMERIC FORM AT A HIGH RESOLUTION | LYS49-PLA2S, PHOSPHOLIPASE HOMOLOGUE, BOTHROPSTOXIN-I, P- BROMOPHENACYL BROMIDE, MYOTOXICITY, ANTIBIOTIC, ANTIMICROBIAL, DISULFIDE BOND, MYOTOXIN, SECRETED, TOXIN
1gp7:A (HIS1) to (SER109) ACIDIC PHOSPHOLIPASE A2 FROM VENOM OF OPHIOPHAGUS HANNAH | PHOSPHOLIPASE A2, SNAKE VENOM, KING COBRA, CARDIOTOXIC ACTIVITY, MYOTOXIC ACTIVITY, PANCREATIC LOOP, CRYSTAL STRUCTURE, HYDROLASE, LIPID DEGRADATION, CALCIUM
3v9m:B (LEU2) to (ALA102) PHOSPHOLIPASE ACII4 FROM AUSTRALIAN KING BROWN SNAKE | WING MOTIF, PHOSPHOLIPASE, HYDROLASE
3i3h:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF BOTHROPSTOXIN-I CRYSTALLIZED AT 291K | HOMOLOGUE PHOSPHOLIPASE A2, BOTHROPSTOXIN-I, BTHTX-I_18C, LYS49-PLA2 FROM BOTHROPS JARARACUSSU, SNAKE VENOM, ANTIMICROBIAL, DISULFIDE BOND, MYOTOXIN, SECRETED, TOXIN
3i3h:B (PHE3) to (LEU110) CRYSTAL STRUCTURE OF BOTHROPSTOXIN-I CRYSTALLIZED AT 291K | HOMOLOGUE PHOSPHOLIPASE A2, BOTHROPSTOXIN-I, BTHTX-I_18C, LYS49-PLA2 FROM BOTHROPS JARARACUSSU, SNAKE VENOM, ANTIMICROBIAL, DISULFIDE BOND, MYOTOXIN, SECRETED, TOXIN
2g58:A (LEU2) to (ASN109) CRYSTAL STRUCTURE OF A COMPLEX OF PHOSPHOLIPASE A2 WITH A DESIGNED PEPTIDE INHIBITOR DEHYDRO-ILE-ALA-ARG-SER AT 0.98 A RESOLUTION | PHOSPHOLIPASE A2, DIARS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3vbz:A (LEU2) to (GLN101) CRYSTAL STRUCTURE OF TAIPOXIN BETA SUBUNIT ISOFORM 2 | PHOSPHOLIPASE A2 FOLD, PLA2 FOLD, NEUROTOXIN, PHOSPHOLIPASE, CALCIUM BINDING, TAIPOXIN ALPHA SUBUNIT BINDING, TAIPOXIN GAMMA SUBUNIT BINDING, SECRETED, TOXIN
3vc0:A (ASN1) to (GLN101) CRYSTAL STRUCTURE OF TAIPOXIN BETA SUBUNIT ISOFORM 1 | PHOSPHOLIPASE A2 FOLD, PLA2 FOLD, NEUROTOXIN, PHOSPHOLIPASE, CALCIUM BINDING, TAIPOXIN ALPHA SUBUNIT BINDING, TAIPOXIN GAMMA SUBUNIT BINDING, SECRETED, TOXIN
1sqz:A (LEU2) to (ASN109) DESIGN OF SPECIFIC INHIBITORS OF PHOPHOLIPASE A2: CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN GROUP II PHOPHOLIPASE A2 AND A DESIGNED PEPTIDE DEHYDRO-ILE-ALA-ARG-SER AT 1.2A RESOLUTION | PHOSPHOLIPASE A2, DEHYDRO-IARS, TOXIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1sv3:A (LEU2) to (ASN109) STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND 4-METHOXYBENZOIC ACID AT 1.3A RESOLUTION. | PHOSPHOLIPASE A2, COMPLEX, 4-METHOXYBENZOIC ACID, CRYSTAL STRUCTURE, 1.3A RESOLUTION, HYDROLASE
1sv9:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN GROUPII PHOSPHOLIPASE A2 AND ANTI-INFLAMMATORY AGENT 2-[(2,6- DICHLOROPHENYL)AMINO] BENZENEACETIC ACID AT 2.7A RESOLUTION | PHOSPHOLIPASE A2,COMPLEX,DICLOFENAC,CRYSTAL STRUCTURE,2.7A RESOLUTION, TOXIN
1sxk:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF A COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND A NON-SPECIFIC ANTI-INFLAMMATORY AMINO SALICYLIC ACID AT 1.2 A RESOLUTION | COMPLEX, PHOSPHOLIPASE A2, AMINO SALICYLIC ACID, DABOIA RUSSELI PULCHELLA, TOXIN
1sz8:A (ASN1) to (ALA104) CRYSTAL STRUCTURE OF AN ACIDIC PHOSPHOLIPASE A2 FROM NAJA NAJA SAGITTIFERA AT 1.5 A RESOLUTION | PHOSPHOLIPASE A2, MOLECULAR CONFORMATION, ENZYME ACTIVITY, HYDROLASE
2gns:A (SER1) to (ASN109) DESIGN OF SPECIFIC PEPTIDE INHIBITORS OF PHOSPHOLIPASE A2: CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN A GROUP II PHOSPHOLIPASE A2 AND A DESIGNED PENTAPEPTIDE ALA- LEU- VAL- TYR- LYS AT 2.3 A RESOLUTION | PEPTIDE INHIBITOR, BINDING CONSTANT, HYDROLASE
1tc8:A (ASN1) to (LYS103) CRYSTAL STRUCTURE OF KRAIT-VENOM PHOSPHOLIPASE A2 IN A COMPLEX WITH A NATURAL FATTY ACID TRIDECANOIC ACID | PHOSPHOLIPASEA2, COMPLEX, CRYSTAL, FATTY ACID, TOXIN
1td7:A (ASN1) to (ALA104) INTERACTIONS OF A SPECIFIC NON-STEROIDAL ANTI-INFLAMMATORY DRUG (NSAID) WITH GROUP I PHOSPHOLIPASE A2 (PLA2): CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PLA2 AND NIFLUMIC ACID AT 2.5 A RESOLUTION | PHOSPHOLIPASE A2, ENZYME, INHIBITOR, HYDROLASE
1tdv:A (SER1) to (ASN109) NON-SPECIFIC BINDING TO PHOSPHOLIPASE A2:CRYSTAL STRUCTURE OF THE COMPLEX OF PLA2 WITH A DESIGNED PEPTIDE TYR-TRP-ALA- ALA-ALA-ALA AT 1.7A RESOLUTION | NON-SPECIFIC, YWAAAA COMPLEX, PHOSPHOLIPASE A2, HYDROLASE
1tg4:A (LEU2) to (ASN109) DESIGN OF SPECIFIC INHIBITORS OF GROUPII PHOSPHOLIPASE A2(PLA2): CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN RUSSELLS VIPER PLA2 AND DESIGNED PEPTIDE PHE-LEU-ALA-TYR- LYS AT 1.7A RESOLUTION | PHOSPHOLIPASE A2,FLAYK,COMPLEX,SPECIFIC INHIBITOR,CRYSTAL STRUCTURE, HYDROLASE
1tgm:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF A COMPLEX FORMED BETWEEN GROUP II PHOSPHOLIPASE A2 AND ASPIRIN AT 1.86 A RESOLUTION | PHOSPHOLIPASE A2, ENZYME, COMPLEX, HYDROLASE
1th6:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 IN COMPLEX WITH ATROPINE AT 1.23A RESOLUTION | PHOSPHOLIPIDS, EICOSANOIDS, INHIBITION, HYDROLASE
3iq3:A (SER1) to (ASN99) CRYSTAL STRUCTURE OF BOTHROPSTOXIN-I COMPLEXED WITH POLIETILENE GLICOL 4000 - CRYSTALLIZED AT 283 K | HOMOLOGUE PHOSPHOLIPASE A2, BOTHROPSTOXIN-I, BTHTX-I_10C, LYS49-PLA2 FROM BOTHROPS JARARACUSSU, SNAKE VENOM, ANTIBIOTIC, ANTIMICROBIAL, DISULFIDE BOND, MYOTOXIN, SECRETED, TOXIN
3iq3:B (SER1) to (ASN99) CRYSTAL STRUCTURE OF BOTHROPSTOXIN-I COMPLEXED WITH POLIETILENE GLICOL 4000 - CRYSTALLIZED AT 283 K | HOMOLOGUE PHOSPHOLIPASE A2, BOTHROPSTOXIN-I, BTHTX-I_10C, LYS49-PLA2 FROM BOTHROPS JARARACUSSU, SNAKE VENOM, ANTIBIOTIC, ANTIMICROBIAL, DISULFIDE BOND, MYOTOXIN, SECRETED, TOXIN
1tjk:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN GROUP II PHOSPHOLIPASE A2 WITH A DESIGNED PENTAPEPTIDE, PHE- LEU- SER- THR- LYS AT 1.2 A RESOLUTION | PHOSPHOLIPASE A2, ENZYME, COMPLEX, HYDROLASE
2h4c:C (ASN1) to (ASN109) STRUCTURE OF DABOIATOXIN (HETERODIMERIC PLA2 VENOM) | PHOSPHOLIPASE A2, NON-INHIBITOR ACIDIC PLA2, BASIC PLA2, HETERODIMER, HYDROLASE
2h4c:E (ASN1) to (ASN109) STRUCTURE OF DABOIATOXIN (HETERODIMERIC PLA2 VENOM) | PHOSPHOLIPASE A2, NON-INHIBITOR ACIDIC PLA2, BASIC PLA2, HETERODIMER, HYDROLASE
2h4c:G (ASN1) to (ASN109) STRUCTURE OF DABOIATOXIN (HETERODIMERIC PLA2 VENOM) | PHOSPHOLIPASE A2, NON-INHIBITOR ACIDIC PLA2, BASIC PLA2, HETERODIMER, HYDROLASE
2h4c:H (ASN1) to (ASN109) STRUCTURE OF DABOIATOXIN (HETERODIMERIC PLA2 VENOM) | PHOSPHOLIPASE A2, NON-INHIBITOR ACIDIC PLA2, BASIC PLA2, HETERODIMER, HYDROLASE
1tp2:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX OF GROUP II PHOSPHOLIPASEA2 DIMER WITH A FATTY ACID TRIDECANOIC ACID AT 2.4 A RESOLUTION | CATALYSIS, INHIBITION, FATTY ACID, HYDROLASE
1tp2:B (LEU3) to (LEU110) CRYSTAL STRUCTURE OF THE COMPLEX OF GROUP II PHOSPHOLIPASEA2 DIMER WITH A FATTY ACID TRIDECANOIC ACID AT 2.4 A RESOLUTION | CATALYSIS, INHIBITION, FATTY ACID, HYDROLASE
1hn4:B (SER-3) to (LYS108) PROPHOSPHOLIPASE A2 DIMER COMPLEXED WITH MJ33, SULFATE, AND CALCIUM | HYDROLASE, ENZYME, CARBOXYLIC ESTER HYDROLASE, DIMER, SULFATE BINDING, INHIBITOR BINDING
1u4j:A (LEU2) to (SER103) CRYSTAL STRUCTURE OF A CARBOHYDRATE INDUCED DIMER OF GROUP I PHOSPHOLIPASE A2 FROM BUNGARUS CAERULEUS AT 2.1 A RESOLUTION | PHOSPHOLIPASE A2, HOMODIMER, BUNGARUS CAERULEUS, MANNOSE, HYDROLASE
1u4j:B (LEU2) to (SER103) CRYSTAL STRUCTURE OF A CARBOHYDRATE INDUCED DIMER OF GROUP I PHOSPHOLIPASE A2 FROM BUNGARUS CAERULEUS AT 2.1 A RESOLUTION | PHOSPHOLIPASE A2, HOMODIMER, BUNGARUS CAERULEUS, MANNOSE, HYDROLASE
2i0u:E (LEU2) to (ASN109) CRYSTAL STRUCTURES OF PHOSPHOLIPASES A2 FROM VIPERA NIKOLSKII VENOM REVEALING TRITON X-100 BOUND IN HYDROPHOBIC CHANNEL | ALPHA-BETA-ALPHA, HYDROLASE
2i0u:A (ASN1) to (ASN109) CRYSTAL STRUCTURES OF PHOSPHOLIPASES A2 FROM VIPERA NIKOLSKII VENOM REVEALING TRITON X-100 BOUND IN HYDROPHOBIC CHANNEL | ALPHA-BETA-ALPHA, HYDROLASE
1ijl:B (SER1) to (ASN99) CRYSTAL STRUCTURE OF ACIDIC PHOSPHOLIPASE A2 FROM DEINAGKISTRODON ACUTUS | THREE LONG HELIX, ONE TWO STRAND BETA SHEET, CALCIUM BINDING LOOP, HYDROLASE
1j1a:A (ASN1) to (ASN101) PANCREATIC SECRETORY PHOSPHOLIPASE A2 (IIA) WITH ANTI- INFLAMMATORY ACTIVITY | MEDICINAL CHEMISTRY, ENZYME INHIBITOR, STRUCTURE-ACTIVITY RELATIONSHIPS, INFLAMMATION, HYDROLASE
1j1a:B (ASN1) to (ASN101) PANCREATIC SECRETORY PHOSPHOLIPASE A2 (IIA) WITH ANTI- INFLAMMATORY ACTIVITY | MEDICINAL CHEMISTRY, ENZYME INHIBITOR, STRUCTURE-ACTIVITY RELATIONSHIPS, INFLAMMATION, HYDROLASE
1jia:A (LEU2) to (ASN109) STRUCTURE OF A BASIC PHOSPHOLIPASE A2 FROM AGKISTRODON HALYS PALLAS AT 2.13A RESOLUTION | PHOSPHOLIPASE A2, AGKISTRODON HALYS PALLAS CRYSTAL STRUCTURE
1jia:B (LEU2) to (ASN109) STRUCTURE OF A BASIC PHOSPHOLIPASE A2 FROM AGKISTRODON HALYS PALLAS AT 2.13A RESOLUTION | PHOSPHOLIPASE A2, AGKISTRODON HALYS PALLAS CRYSTAL STRUCTURE
1vip:A (LEU2) to (ASN109) ANTICOAGULANT CLASS II PHOSPHOLIPASE A2 FROM THE VENOM OF VIPERA RUSSELLI RUSSELLI | HYDROLASE, PHOSPHOLIPASE A2, ANTICOAGULANT
1vl9:A (ALA1) to (VAL109) ATOMIC RESOLUTION (0.97A) STRUCTURE OF THE TRIPLE MUTANT (K53,56,121M) OF BOVINE PANCREATIC PHOSPHOLIPASE A2 | ALPHA HELIX, BETA SHEET, TRIPLE MUTANT, CALCIUM ION, HYDROLASE
1jq9:B (LEU3) to (ASN109) CRYSTAL STRUCTURE OF A COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 FROM DABOIA RUSSELLI PULCHELLA AND A DESIGNED PENTAPEPTIDE PHE-LEU-SER- TYR-LYS AT 1.8 RESOLUTION | PHOSPHOLIPASE A2, DABOIA RUSSELLI PULCHELLA, NEUROTOXIC, DESIGNED PEPTIDE, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1kpm:A (SER1) to (ASN109) FIRST STRUCTURAL EVIDENCE OF A SPECIFIC INHIBITION OF PHOSPHOLIPASE A2 BY VITAMIN E AND ITS IMPLICATIONS IN INFLAMMATION: CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND VITAMIN E AT 1.8 A RESOLUTION. | PHOSPHOLIPASE A2, DABOIA RUSSELLI PULCHELLA, NEUROTOXIC, INFLAMMATION, HYDROLASE
1kpm:B (SER1) to (ASN109) FIRST STRUCTURAL EVIDENCE OF A SPECIFIC INHIBITION OF PHOSPHOLIPASE A2 BY VITAMIN E AND ITS IMPLICATIONS IN INFLAMMATION: CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND VITAMIN E AT 1.8 A RESOLUTION. | PHOSPHOLIPASE A2, DABOIA RUSSELLI PULCHELLA, NEUROTOXIC, INFLAMMATION, HYDROLASE
1kqu:A (ASN1) to (ALA99) HUMAN PHOSPHOLIPASE A2 COMPLEXED WITH A SUBSTRATE ANOLOGUE | PHOSPHOLIPASE A2, INHIBITOR, STRUCTURE, HYDROLASE
1kvo:A (LEU2) to (ASN101) HUMAN PHOSPHOLIPASE A2 COMPLEXED WITH A HIGHLY POTENT SUBSTRATE ANOLOGUE | HYDROLASE, LIPID DEGRADATION, MEMBRANE, SIGNAL, CALCIUM
1kvo:B (LEU2) to (ASN101) HUMAN PHOSPHOLIPASE A2 COMPLEXED WITH A HIGHLY POTENT SUBSTRATE ANOLOGUE | HYDROLASE, LIPID DEGRADATION, MEMBRANE, SIGNAL, CALCIUM
1kvo:C (ASN1) to (ASN101) HUMAN PHOSPHOLIPASE A2 COMPLEXED WITH A HIGHLY POTENT SUBSTRATE ANOLOGUE | HYDROLASE, LIPID DEGRADATION, MEMBRANE, SIGNAL, CALCIUM
1kvo:D (LEU2) to (ASN101) HUMAN PHOSPHOLIPASE A2 COMPLEXED WITH A HIGHLY POTENT SUBSTRATE ANOLOGUE | HYDROLASE, LIPID DEGRADATION, MEMBRANE, SIGNAL, CALCIUM
1kvo:E (LEU2) to (ASN101) HUMAN PHOSPHOLIPASE A2 COMPLEXED WITH A HIGHLY POTENT SUBSTRATE ANOLOGUE | HYDROLASE, LIPID DEGRADATION, MEMBRANE, SIGNAL, CALCIUM
1kvo:F (LEU2) to (ASN101) HUMAN PHOSPHOLIPASE A2 COMPLEXED WITH A HIGHLY POTENT SUBSTRATE ANOLOGUE | HYDROLASE, LIPID DEGRADATION, MEMBRANE, SIGNAL, CALCIUM
1kvw:A (LEU2) to (LYS108) CARBOXYLIC ESTER HYDROLASE, SINGLE MUTANT H48Q OF BOVINE PANCREATIC PLA2 ENZYME | HYDROLASE, ENZYME, CARBOXYLIC ESTER HYDROLASE
1kvy:A (ALA1) to (LYS108) CARBOXYLIC ESTER HYDROLASE, SINGLE MUTANT D49E COORDINATED TO CALCIUM | HYDROLASE, ENZYME, CARBOXYLIC ESTER HYDROLASE, MUTANT
4o1y:A (ALA1) to (LYS108) CRYSTAL STRUCTURE OF PORCINE PANCREATIC PHOSPHOLIPASE A2 IN COMPLEX WITH 1-NAPHTHALENEACETIC ACID | HYDROLASE, 1-NAPHTHALENEACETIC ACID BINDING, PLA2, PANCREATIC ENZYME
3jq5:A (ASN1) to (GLY103) PHOSPHOLIPASE A2 PREVENTS THE AGGREGATION OF AMYLOID BETA PEPTIDES: CRYSTAL STRUCTURE OF THE COMPLEX OF PHOSPHOLIPASE A2 WITH OCTAPEPTIDE FRAGMENT OF AMYLOID BETA PEPTIDE, ASP- ALA-GLU-PHE-ARG-HIS-ASP-SER AT 2 A RESOLUTION | PHOSPHOLIPASE A2, CRYSTAL STRUCTURE, OCTAPEPTIDE, AMYLOID BETA, HYDROLASE, CALCIUM, DISULFIDE BOND, LIPID DEGRADATION, METAL-BINDING, SECRETED
3jql:A (LEU2) to (GLY103) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND A HEXAPEPTIDE FRAGMENT OF AMYLOID BETA PEPTIDE, LYS-LEU-VAL-PHE-PHE-ALA AT 1.2 A RESOLUTION | PHOSPHOLIPASE A2, CRYSTAL STRUCTURE, HEXAPEPTIDE, AMYLOID BETA, HYDROLASE, CALCIUM, DISULFIDE BOND, LIPID DEGRADATION, METAL-BINDING, SECRETED
3jti:A (LEU2) to (ALA104) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 WITH BETA-AMYLOID FRAGMENT, LYS-GLY-ALA-ILE-ILE-GLY-LEU-MET AT 1.8 A RESOLUTION | PHOSPHOLIPASE A2, HEPTAPEPTIDE, AMYLOID BETA, HYDROLASE, LIPID DEGRADATION, DISULFIDE BOND, METAL-BINDING, SECRETED, AMYLOID, AMYLOIDOSIS, PROTEASE INHIBITOR, PROTEOGLYCAN, SERINE PROTEASE INHIBITOR
1l8s:A (ALA1) to (LYS108) CARBOXYLIC ESTER HYDROLASE COMPLEX (DIMERIC PLA2 + LPC- ETHER + ACETATE + PHOSPHATE IONS) | HYDROLASE, ENZYME, CARBOXYLIC ESTER HYDROLASE, DIMER, PAF HYDROLYSIS PRODUCTS BINDING, PHOSPHATE BINDING
1l8s:B (TRP3) to (LYS108) CARBOXYLIC ESTER HYDROLASE COMPLEX (DIMERIC PLA2 + LPC- ETHER + ACETATE + PHOSPHATE IONS) | HYDROLASE, ENZYME, CARBOXYLIC ESTER HYDROLASE, DIMER, PAF HYDROLYSIS PRODUCTS BINDING, PHOSPHATE BINDING
1le6:A (GLY1) to (THR101) CARBOXYLIC ESTER HYDROLASE, P 1 21 1 SPACE GROUP | HUMAN PHOSPHATIDYLCHOLINE 2-ACYLHYDROLASE GX, GX SPLA2, SPLA2-X
1le6:B (GLY1) to (THR101) CARBOXYLIC ESTER HYDROLASE, P 1 21 1 SPACE GROUP | HUMAN PHOSPHATIDYLCHOLINE 2-ACYLHYDROLASE GX, GX SPLA2, SPLA2-X
1le6:C (GLY1) to (THR101) CARBOXYLIC ESTER HYDROLASE, P 1 21 1 SPACE GROUP | HUMAN PHOSPHATIDYLCHOLINE 2-ACYLHYDROLASE GX, GX SPLA2, SPLA2-X
1le7:B (GLY1) to (THR101) CARBOXYLIC ESTER HYDROLASE, C 2 2 21 SPACE GROUP | HUMAN PHOSPHATIDYLCHOLINE 2-ACYLHYDROLASE GX, GX SPLA2, SPLA2-X
1ln8:A (ASN1) to (ALA104) CRYSTAL STRUCTURE OF A NEW ISOFORM OF PHOSPHOLIPASE A2 FROM NAJA NAJA SAGITTIFERA AT 1.6 A RESOLUTION | PHOSPHOLIPASE A2, ISOFORM, NAJA NAJA SAGITTIFERA, HYDROLASE
2zbh:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX OF PHOSPHOLIPASE A2 WITH BAVACHALCONE FROM AERVA LANATA AT 2.6 A RESOLUTION | COMPLEX, DAUCOSTEROL, AERVA LANATA, PHOSPHOLIPSE A2, CALCIUM, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, NEUROTOXIN, PRESYNAPTIC NEUROTOXIN, SECRETED, TOXIN
1m8r:A (SER1) to (THR112) CRYSTAL STRUCTURES OF CADMIUM-BINDING ACIDIC PHOSPHOLIPASE A2 FROM THE VENOM OF AGKISTRODON HALYS PALLAS AT 1.9 RESOLUTION (CRYSTAL GROWN AT PH 7.4) | PHOPHOLIPASE A2-METAL CATION COMPLEX, THREE ALPHA, TWO BETA, HYDROLASE
1m8s:A (SER1) to (THR112) CRYSTAL STRUCTURES OF CADMIUM-BINDING ACIDIC PHOSPHOLIPASE A2 FROM THE VENOM OF AGKISTRODON HALYS PALLAS AT 1.9 RESOLUTION (CRYSTAL GROWN AT PH 5.9) | PHOPHOLIPASE A2-METAL CATION COMPLEX, THREE ALPHA, TWO BETA, HYDROLASE
1m8t:A (HIS1) to (ALA109) STRUCTURE OF AN ACIDIC PHOSPHOLIPASE A2 FROM THE VENOM OF OPHIOPHAGUS HANNAH AT 2.1 RESOLUTION FROM A HEMIHEDRALLY TWINNED CRYSTAL FORM | PHOSPHOLIPASE A2 STRUCTURE, TWINNED CRYSTAL, ALPHA, BETA, HYDROLASE
1m8t:B (HIS1) to (ALA109) STRUCTURE OF AN ACIDIC PHOSPHOLIPASE A2 FROM THE VENOM OF OPHIOPHAGUS HANNAH AT 2.1 RESOLUTION FROM A HEMIHEDRALLY TWINNED CRYSTAL FORM | PHOSPHOLIPASE A2 STRUCTURE, TWINNED CRYSTAL, ALPHA, BETA, HYDROLASE
1m8t:C (HIS1) to (ALA109) STRUCTURE OF AN ACIDIC PHOSPHOLIPASE A2 FROM THE VENOM OF OPHIOPHAGUS HANNAH AT 2.1 RESOLUTION FROM A HEMIHEDRALLY TWINNED CRYSTAL FORM | PHOSPHOLIPASE A2 STRUCTURE, TWINNED CRYSTAL, ALPHA, BETA, HYDROLASE
1m8t:D (HIS1) to (ALA109) STRUCTURE OF AN ACIDIC PHOSPHOLIPASE A2 FROM THE VENOM OF OPHIOPHAGUS HANNAH AT 2.1 RESOLUTION FROM A HEMIHEDRALLY TWINNED CRYSTAL FORM | PHOSPHOLIPASE A2 STRUCTURE, TWINNED CRYSTAL, ALPHA, BETA, HYDROLASE
1m8t:E (HIS1) to (ALA109) STRUCTURE OF AN ACIDIC PHOSPHOLIPASE A2 FROM THE VENOM OF OPHIOPHAGUS HANNAH AT 2.1 RESOLUTION FROM A HEMIHEDRALLY TWINNED CRYSTAL FORM | PHOSPHOLIPASE A2 STRUCTURE, TWINNED CRYSTAL, ALPHA, BETA, HYDROLASE
1m8t:F (HIS1) to (GLY108) STRUCTURE OF AN ACIDIC PHOSPHOLIPASE A2 FROM THE VENOM OF OPHIOPHAGUS HANNAH AT 2.1 RESOLUTION FROM A HEMIHEDRALLY TWINNED CRYSTAL FORM | PHOSPHOLIPASE A2 STRUCTURE, TWINNED CRYSTAL, ALPHA, BETA, HYDROLASE
1mc2:A (SER1001) to (ASN1109) MONOMERIC LYS-49 PHOSPHOLIPASE A2 HOMOLOGUE PURIFIED FROM AG | YS49-PHOSPHOLIPASE A2, SNAKE VENOM, AGKISTRODON ACUTUS, TOXIN
1y38:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 DIMER AND GLYCEROPHOSPHATE AT 2.4 A RESOLUTION | CATALYSIS, INHIBITION, COMPLEX, HYDROLASE
1y38:B (LEU3) to (LEU110) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 DIMER AND GLYCEROPHOSPHATE AT 2.4 A RESOLUTION | CATALYSIS, INHIBITION, COMPLEX, HYDROLASE
1y4l:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF BOTHROPS ASPER MYOTOXIN II COMPLEXED WITH THE ANTI-TRYPANOSOMAL DRUG SURAMIN | BOTHROPS ASPER MYOTOXIN II, ANTI-TRYPANOSOMAL DRUG SURAMIN, HYDROLASE
1y4l:B (SER1) to (ASN109) CRYSTAL STRUCTURE OF BOTHROPS ASPER MYOTOXIN II COMPLEXED WITH THE ANTI-TRYPANOSOMAL DRUG SURAMIN | BOTHROPS ASPER MYOTOXIN II, ANTI-TRYPANOSOMAL DRUG SURAMIN, HYDROLASE
4p2p:A (ALA1) to (ALA109) AN INDEPENDENT CRYSTALLOGRAPHIC REFINEMENT OF PORCINE PHOSPHOLIPASE A2 AT 2.4 ANGSTROMS RESOLUTION | CARBOXYLIC ESTER HYDROLASE
1y6o:A (ALA1) to (LYS108) CRYSTAL STRUCTURE OF DISULFIDE ENGINEERED PORCINE PANCREATIC PHOSPHOLIPASE A2 TO GROUP-X ISOZYME IN COMPLEX WITH INHIBITOR MJ33 AND PHOSPHATE IONS | HYDROLASE. DISULFIDE ENGINEERED PLA2. PORCINE PANCRATIC ISOZYME., HYDROLASE
1y6o:B (ALA1) to (LYS108) CRYSTAL STRUCTURE OF DISULFIDE ENGINEERED PORCINE PANCREATIC PHOSPHOLIPASE A2 TO GROUP-X ISOZYME IN COMPLEX WITH INHIBITOR MJ33 AND PHOSPHATE IONS | HYDROLASE. DISULFIDE ENGINEERED PLA2. PORCINE PANCRATIC ISOZYME., HYDROLASE
1y6p:B (ALA1) to (LYS108) CRYSTAL STRUCTURE OF DISULFIDE ENGINEERED PORCINE PANCRATIC PHOSPHOLIPASE A2 TO GROUP-X ISOZYME | HYDROLASE, DISULFIDE ENGINEERED PLA2, PORCINE PANCRATIC ISOZYME
1y75:A (THR2) to (ALA104) A NEW FORM OF CATALYTICALLY INACTIVE PHOSPHOLIPASE A2 WITH AN UNUSUAL DISULPHIDE BRIDGE CYS 32- CYS 49 REVEALS RECOGNITION FOR N- ACETYLGLUCOSMINE | ENZYME, ACTIVITY, MOLECULAR ASSOCIATION, HYDROLASE
1n28:B (LEU2) to (ASN101) CRYSTAL STRUCTURE OF THE H48Q MUTANT OF HUMAN GROUP IIA PHOSPHOLIPASE A2 | HYDROLASE
1n28:A (ALA1) to (ASN101) CRYSTAL STRUCTURE OF THE H48Q MUTANT OF HUMAN GROUP IIA PHOSPHOLIPASE A2 | HYDROLASE
1n29:A (ALA1) to (ASN101) CRYSTAL STRUCTURE OF THE N1A MUTANT OF HUMAN GROUP IIA PHOSPHOLIPASE A2 | HYDROLASE
3l30:A (ALA1) to (LYS108) CRYSTAL STRUCTURE OF PORCINE PANCREATIC PHOSPHOLIPASE A2 COMPLEXED WITH DIHYDROXYBERBERINE | PHOSPHOLIPASE A2, DIHYDROXYBERBERINE, DISULFIDE BOND, HYDROLASE, LIPID DEGRADATION, LIPOPROTEIN, METAL-BINDING, PALMITATE, PYRROLIDONE CARBOXYLIC ACID, SECRETED
1yxh:A (ILE2) to (GLY103) CRYSTAL STRUCTURE OF A NOVEL PHOSPHOLIPASE A2 FROM NAJA NAJA SAGITTIFERA WITH A STRONG ANTICOAGULANT ACTIVITY | PLA2, ANTICOAGULATION, MONOMER, HYDROLASE
1zwp:A (SER1) to (ASN109) THE ATOMIC RESOLUTION CRYSTAL STRUCTURE OF THE PHOSPHOLIPASE A2 (PLA2) COMPLEX WITH NIMESULIDE REVEALS ITS WEAKER BINDING TO PLA2 | PHOSPHOLIPASE A2, NIMESULIDE, COMPLEX, CRYSTAL STRUCTURE, 1.1A RESOLUTION, HYDROLASE
1zyx:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX OF A GROUP IIA PHOSPHOLIPASE A2 WITH A SYNTHETIC ANTI-INFLAMMATORY AGENT LICOFELONE AT 1.9A RESOLUTION | INHIBITOR, COMPLEX, DRUG, HYDROLASE
4qem:A (LEU2) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX OF PHOSPHOLIPASE A2 WITH P-COUMARIC ACID AT 1.2 A RESOLUTION | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4qer:A (LEU2) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX OF PHOSPHOLIPASE A2 WITH RESVERATROL AT 1.20 A RESOLUTION | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4qf7:A (LEU2) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX OF PHOSPHOLIPASE A2 WITH CORTICOSTERONE AT 1.48 A RESOLUTION | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4qf8:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX OF PHOSPHOLIPASE A2 WITH SPERMIDINE AT 1.65 A RESOLUTION | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4qgd:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX OF PHOSPHOLIPASE A2 WITH GRAMINE DERIVATIVE AT 1.80 A RESOLUTION | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4qmc:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND BIOTIN-SULFOXIDE AT 1.09 A RESOLUTION | HYDROLASE
3mlm:A (SER1) to (ASN99) CRYSTAL STRUCTURE OF BN IV IN COMPLEX WITH MYRISTIC ACID: A LYS49 MYOTOXIC PHOSPHOLIPASE A2 FROM BOTHROPS NEUWIEDI VENOM | MYOTOXIN, PHOSPHOLIPASE-LIKE PROTEIN, HYDROLASE
3mlm:B (SER1) to (ASN99) CRYSTAL STRUCTURE OF BN IV IN COMPLEX WITH MYRISTIC ACID: A LYS49 MYOTOXIC PHOSPHOLIPASE A2 FROM BOTHROPS NEUWIEDI VENOM | MYOTOXIN, PHOSPHOLIPASE-LIKE PROTEIN, HYDROLASE
3bjw:B (VAL2) to (ASN109) CRYSTAL STRUCTURE OF ECARPHOLIN S COMPLEXED WITH SURAMIN | SNAKE VENOM, PHOSPHOLIPASE A2, SURAMIN, SER49, COMPLEX, CALCIUM, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, SECRETED, TOXIN
3bjw:E (SER1) to (ASN109) CRYSTAL STRUCTURE OF ECARPHOLIN S COMPLEXED WITH SURAMIN | SNAKE VENOM, PHOSPHOLIPASE A2, SURAMIN, SER49, COMPLEX, CALCIUM, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, SECRETED, TOXIN
3bjw:F (SER1) to (ASN109) CRYSTAL STRUCTURE OF ECARPHOLIN S COMPLEXED WITH SURAMIN | SNAKE VENOM, PHOSPHOLIPASE A2, SURAMIN, SER49, COMPLEX, CALCIUM, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, SECRETED, TOXIN
3bjw:H (VAL3) to (ASN109) CRYSTAL STRUCTURE OF ECARPHOLIN S COMPLEXED WITH SURAMIN | SNAKE VENOM, PHOSPHOLIPASE A2, SURAMIN, SER49, COMPLEX, CALCIUM, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, SECRETED, TOXIN
4bp2:A (ALA1) to (LYS108) CRYSTALLOGRAPHIC REFINEMENT OF BOVINE PRO-PHOSPHOLIPASE A2 AT 1.6 ANGSTROMS RESOLUTION | CARBOXYLIC ESTER HYDROLASE ZYMOGEN
3cbi:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE TERNARY COMPLEX OF PHOSPHOLIPASE A2 WITH AJMALINE AND ANISIC ACID AT 3.1 A RESOLUTION | PLA2, TERNARY COMPLEX, AJMALINE, ANISIC ACID, PHOSPHOLIPASE A2, CALCIUM, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, NEUROTOXIN, PRESYNAPTIC NEUROTOXIN, SECRETED, TOXIN
3cbi:B (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE TERNARY COMPLEX OF PHOSPHOLIPASE A2 WITH AJMALINE AND ANISIC ACID AT 3.1 A RESOLUTION | PLA2, TERNARY COMPLEX, AJMALINE, ANISIC ACID, PHOSPHOLIPASE A2, CALCIUM, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, NEUROTOXIN, PRESYNAPTIC NEUROTOXIN, SECRETED, TOXIN
3cbi:C (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE TERNARY COMPLEX OF PHOSPHOLIPASE A2 WITH AJMALINE AND ANISIC ACID AT 3.1 A RESOLUTION | PLA2, TERNARY COMPLEX, AJMALINE, ANISIC ACID, PHOSPHOLIPASE A2, CALCIUM, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, NEUROTOXIN, PRESYNAPTIC NEUROTOXIN, SECRETED, TOXIN
3cbi:D (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE TERNARY COMPLEX OF PHOSPHOLIPASE A2 WITH AJMALINE AND ANISIC ACID AT 3.1 A RESOLUTION | PLA2, TERNARY COMPLEX, AJMALINE, ANISIC ACID, PHOSPHOLIPASE A2, CALCIUM, HYDROLASE, LIPID DEGRADATION, METAL-BINDING, NEUROTOXIN, PRESYNAPTIC NEUROTOXIN, SECRETED, TOXIN
4rfp:A (ASN1) to (THR102) CRYSTAL STRUCTURE OF A ACIDIC PLA2 FROM TRIMERESURUS STEJNEGERI VENOM | ALPHA-HELIX, HYDROLASE, GLYCEROPHOSPHOLIPID, VENOM GLAND
3nju:A (LEU2) to (ALA104) CRYSTAL STRUCTURE OF THE COMPLEX OF GROUP I PHOSPHOLIPASE A2 WITH 4- METHOXY-BENZOICACID AT 1.4A RESOLUTION | PLA2, COMPLEX, ANISIC ACID, NAJA SAGITTIFERA, HYDROLASE
3cyl:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF PIRATOXIN I (A MYOTOXIC LYS49-PLA2) COMPLEXED WITH ALPHA-TOCOPHEROL | LYS49-PLA2, BOTHROPS PIRAJAI, SANKE VENOM, X-RAY CRYSTALLOGRAPHY, ALPHA-TOCOPHEROL, PRTX-I, MYOTOXIN, SECRETED, TOXIN
3cyl:B (SER1) to (ASN109) CRYSTAL STRUCTURE OF PIRATOXIN I (A MYOTOXIC LYS49-PLA2) COMPLEXED WITH ALPHA-TOCOPHEROL | LYS49-PLA2, BOTHROPS PIRAJAI, SANKE VENOM, X-RAY CRYSTALLOGRAPHY, ALPHA-TOCOPHEROL, PRTX-I, MYOTOXIN, SECRETED, TOXIN
3o4m:A (ALA1) to (LYS108) CRYSTAL STRUCTURE OF PORCINE PANCREATIC PHOSPHOLIPASE A2 IN COMPLEX WITH 1,2-DIHYDROXYBENZENE | CATECHOL BINDING, PLA2, PANCREATIC ENZYME, DISULFIDE BOND, LIPID DEGRADATION, LIPOPROTEIN, METAL-BINDING, PALMITATE, PYRROLIDONE CARBOXYLIC ACID, PANCREAS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5g3m:A (GLY1) to (THR101) DISCOVERY OF A NOVEL SECRETED PHOSPHOLIPASE A2 (SPLA2) INHIBITOR. | HYDROLASE, SPLA2, CARDIOVASCULAR DISEASE, INHIBITOR, FRAGMENT
5g3m:B (GLY1) to (THR101) DISCOVERY OF A NOVEL SECRETED PHOSPHOLIPASE A2 (SPLA2) INHIBITOR. | HYDROLASE, SPLA2, CARDIOVASCULAR DISEASE, INHIBITOR, FRAGMENT
4dbk:A (ALA1) to (LYS108) CRYSTAL STRUCTURE OF PORCINE PANCREATIC PHOSPHOLIPASE A2 COMPLEXED WITH BERBERINE | MONOMERIC PROTEIN, BERBERINE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4dcf:A (SER1) to (ASN99) STRUCTURE OF MTX-II FROM BOTHROPS BRAZILI | LYS49 PHOSPHOLIPASE, PHOSPHOLIPASE, HYDROLASE
4dcf:B (SER1) to (ASN99) STRUCTURE OF MTX-II FROM BOTHROPS BRAZILI | LYS49 PHOSPHOLIPASE, PHOSPHOLIPASE, HYDROLASE
4dcf:C (SER1) to (ASN99) STRUCTURE OF MTX-II FROM BOTHROPS BRAZILI | LYS49 PHOSPHOLIPASE, PHOSPHOLIPASE, HYDROLASE
4dcf:D (SER1) to (ASN99) STRUCTURE OF MTX-II FROM BOTHROPS BRAZILI | LYS49 PHOSPHOLIPASE, PHOSPHOLIPASE, HYDROLASE
3p2p:A (ALA1) to (ALA109) ENHANCED ACTIVITY AND ALTERED SPECIFICITY OF PHOSPHOLIPASE A2 BY DELETION OF A SURFACE LOOP | HYDROLASE(CARBOXYL ESTER)
3p2p:B (ALA1) to (LYS108) ENHANCED ACTIVITY AND ALTERED SPECIFICITY OF PHOSPHOLIPASE A2 BY DELETION OF A SURFACE LOOP | HYDROLASE(CARBOXYL ESTER)
4e4c:A (ASN1) to (LYS102) CRYSTAL STRUCTURE OF NOTEXIN AT 1.8 A RESOLUTION | HYDROLASE
4eix:A (SER1) to (ASN109) STRUCTURAL STUDIES OF THE TERNARY COMPLEX OF PHASPHOLIPASE A2 WITH NIMESULIDE AND INDOMETHACIN | HYDROLASE
3qlm:A (ALA1) to (ALA109) CRYSTAL STRUCTURE OF PORCINE PANCREATIC PHOSPHOLIPASE A2 IN COMPLEX WITH N-HEXADECANOIC ACID | HYDROLASE, PLA2, PANCREATIC ENZYME, PALMITIC ACID BINDING
3qnl:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF PRTX-I COMPLEXED TO ROSMARINIC ACID | HYDROLASE
3qnl:B (SER1) to (ASN109) CRYSTAL STRUCTURE OF PRTX-I COMPLEXED TO ROSMARINIC ACID | HYDROLASE
4g5i:A (ALA1) to (LYS108) CRYSTAL STRUCTURE OF PORCINE PANCREATIC PLA2 IN COMPLEX WITH DBP | PHOSPHOLIPASE A2, DISULFIDE BOND, HYDROLASE, 2 LIPID DEGRADATION, LIPOPROTEIN, METAL-BINDING, PALMITATE
4gfy:A (SER1) to (ASN109) DESIGN OF PEPTIDE INHIBITORS OF PHOSPHOLIPASE A2: CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 COMPLEXED WITH A DESIGNED TETRAPEPTIDE VAL - ILU- ALA - LYS AT 2.7 A RESOLUTION | PLA2, ANTI-INFLAMMATORY, ANTI-COAGULANT, PEPTIDE-INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4gld:A (LEU2) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX OF TYPE II PHOSPHOLIPASE A2 WITH A DESIGNED PEPTIDE INHIBITOR PHE - LEU - ALA - TYR - LYS AT 1.69 A RESOLUTION | PLA2, ANTI-INFLAMMATORY, ANTI-COAGULANT, PEPTIDE-INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5p2p:A (ALA1) to (LYS108) X-RAY STRUCTURE OF PHOSPHOLIPASE A2 COMPLEXED WITH A SUBSTRATE-DERIVED INHIBITOR | HYDROLASE(CARBOXYLIC ESTER)
5p2p:B (ALA1) to (ALA109) X-RAY STRUCTURE OF PHOSPHOLIPASE A2 COMPLEXED WITH A SUBSTRATE-DERIVED INHIBITOR | HYDROLASE(CARBOXYLIC ESTER)
1aok:B (LEU2) to (ASN109) VIPOXIN COMPLEX | PHOSPHOLIPASE, HYDROLASE, VIPOXIN, PLA2-ACTIVITY, SNAKE- VENOM
2osh:A (ASN1) to (GLY102) CRYSTAL STRUCTURE OF NATRATOXIN, A SNAKE SPLA2 THAT BLOCKS A-TYPE K+ CHANNEL | NAJA ATRA VENOM, STRUCTURE, PHOSPHOLIPASE A2, A-TYPE K+ CHANNEL INHIBITOR, HYDROLASE
2otf:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND ATENOLOL AT 1.95 A RESOLUTION | INHIBITION, COMPLEX, HYDROLASE
2oub:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND ATENOLOL AT 2.75 A RESOLUTION | INHIBITION, COMPLEX, HYDROLASE
2bd1:A (ALA1) to (VAL109) A POSSIBLE ROLE OF THE SECOND CALCIUM ION IN INTERFACIAL BINDING: ATOMIC AND MEDIUM RESOLUTION CRYSTAL STRUCTURES OF THE QUADRUPLE MUTANT OF PHOSPHOLIPASE A2 | ALPHA HELIX, BETA SHEET, HYDROLASE
2bd1:B (ALA1) to (LYS108) A POSSIBLE ROLE OF THE SECOND CALCIUM ION IN INTERFACIAL BINDING: ATOMIC AND MEDIUM RESOLUTION CRYSTAL STRUCTURES OF THE QUADRUPLE MUTANT OF PHOSPHOLIPASE A2 | ALPHA HELIX, BETA SHEET, HYDROLASE
1bbc:A (ASN1) to (ASN109) STRUCTURE OF RECOMBINANT HUMAN RHEUMATOID ARTHRITIC SYNOVIAL FLUID PHOSPHOLIPASE A2 AT 2.2 ANGSTROMS RESOLUTION | CARBOXYLIC ESTER HYDROLASE, HYDROLASE
3fo7:A (LEU2) to (ASN109) SIMULTANEOUS INHIBITION OF ANTI-COAGULATION AND INFLAMMATION: CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 COMPLEXED WITH INDOMETHACIN AT 1.4 A RESOLUTION REVEALS THE PRESENCE OF THE NEW COMMON LIGAND BINDING SITE | PLA2, ANTI-INFLAMMATORY, ANTI-COAGULANT, INDOMETHACIN, CRYSTAL STRUCTURE, HYDROLASE
2pws:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND 2-(4-ISOBUTYL-PHENYL)-PROPIONIC ACID AT 2.2 A RESOLUTION | NSAIDS, ACTIVE SITE, INHIBITOR, HYDROLASE
1oyf:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF RUSSELLES VIPER (DABOIA RUSSELLII PULCHELLA) PHOSPHOLIPASE A2 IN A COMPLEX WITH VENOM 6- METHYL HEPTANOL | PHOSPHOLIPASE A2, COMPLEX, CATALYSIS, INHIBITION, HYDROLASE
1oyf:B (SER1) to (LEU110) CRYSTAL STRUCTURE OF RUSSELLES VIPER (DABOIA RUSSELLII PULCHELLA) PHOSPHOLIPASE A2 IN A COMPLEX WITH VENOM 6- METHYL HEPTANOL | PHOSPHOLIPASE A2, COMPLEX, CATALYSIS, INHIBITION, HYDROLASE
1oz6:A (LEU2) to (ASN109) X-RAY STRUCTURE OF ACIDIC PHOSPHOLIPASE A2 FROM INDIAN SAW- SCALED VIPER (ECHIS CARINATUS) WITH A POTENT PLATELET AGGREGATION INHIBITORY ACTIVITY | ENZYME, PLA2, HYDROLASE
3h1x:A (LEU2) to (ASN109) SIMULTANEOUS INHIBITION OF ANTI-COAGULATION AND INFLAMMATION: CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 COMPLEXED WITH INDOMETHACIN AT 1.4 A RESOLUTION REVEALS THE PRESENCE OF THE NEW COMMON LIGAND BINDING SITE | PLA2, ANTI-INFLAMMATORY, ANTI-COAGULANT, INDOMETHACIN, CRYSTAL STRUCTURE, HYDROLASE
1fb2:A (LEU3) to (ASN109) STRUCTURE OF PHOSPHOLIPASE A2 FROM DABOIA RUSSELLI PULCHELLA AT 1.95 | STRUCTURE, PHOSPHOLIPASE A2, DABOIA RUSSELLI PULCHELLA, NEUROTOXIC, TOXIN
4yv5:B (SER1) to (ASN109) CRYSTAL STRUCTURE OF MYOTOXIN II FROM BOTHROPS MOOJENI COMPLEXED TO SURAMIN | BOTHROPS MOOJENI, MYOTOXIN II, LYS49-PLA2, SURAMIN, TOXIN
4yv5:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF MYOTOXIN II FROM BOTHROPS MOOJENI COMPLEXED TO SURAMIN | BOTHROPS MOOJENI, MYOTOXIN II, LYS49-PLA2, SURAMIN, TOXIN
4yz7:A (SER1) to (ASN99) CRYSTAL STRUCTURE OF PIRATOXIN I (PRTX-I) COMPLEXED TO ARISTOLOCHIC ACID | TOXIN, PHOSPHOLIPASE A2, PHOSPHOLIPASE A2-LIKE, INHIBITOR
4yz7:B (SER1) to (ASN99) CRYSTAL STRUCTURE OF PIRATOXIN I (PRTX-I) COMPLEXED TO ARISTOLOCHIC ACID | TOXIN, PHOSPHOLIPASE A2, PHOSPHOLIPASE A2-LIKE, INHIBITOR
1g0z:A (LEU2) to (SER103) SPECIFIC MUTATIONS IN KRAIT PLA2 LEAD TO DIMERIZATION OF PROTEIN MOLECULES: CRYSTAL STRUCTURE OF KRAIT PLA2 AT 2.1 RESOLUTION | STRUCTURE,PHOSPHOLIPASE A2,HOMODIMER,BUNGARUS CAERULEUS, TOXIN
1g0z:B (LEU2) to (SER103) SPECIFIC MUTATIONS IN KRAIT PLA2 LEAD TO DIMERIZATION OF PROTEIN MOLECULES: CRYSTAL STRUCTURE OF KRAIT PLA2 AT 2.1 RESOLUTION | STRUCTURE,PHOSPHOLIPASE A2,HOMODIMER,BUNGARUS CAERULEUS, TOXIN
1s8h:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF LYS49-PHOSPHOLIPASE A2 FROM AGKISTRODON CONTORTRIX LATICINCTUS, FIRST FATTY ACID FREE FORM | LYS49-PHOSPHOLIPASE A2, SNAKE VENOM, MYOTOXICITY, FATTY ACID FREE FORM, HYDROLASE, TOXIN
3hzw:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF BOTHROPSTOXIN-I CHEMICALLY MODIFIED BY P- BROMOPHENACYL BROMIDE (BPB) | LYS49-PLA2, PHOSPHOLIPASE HOMOLOGUE, MYOTOXICITY, P-BROMOPHENACYL BROMIDE, BOTHROPSTOXIN-I, ANTIBIOTIC, ANTIMICROBIAL, DISULFIDE BOND, MYOTOXIN, SECRETED, TOXIN
3hzw:B (SER1) to (ASN109) CRYSTAL STRUCTURE OF BOTHROPSTOXIN-I CHEMICALLY MODIFIED BY P- BROMOPHENACYL BROMIDE (BPB) | LYS49-PLA2, PHOSPHOLIPASE HOMOLOGUE, MYOTOXICITY, P-BROMOPHENACYL BROMIDE, BOTHROPSTOXIN-I, ANTIBIOTIC, ANTIMICROBIAL, DISULFIDE BOND, MYOTOXIN, SECRETED, TOXIN
1skg:A (SER2001) to (ASN2109) STRUCTURE-BASED RATIONAL DRUG DESIGN: CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND A PENTAPEPTIDE VAL-ALA-PHE-ARG-SER | RATIONAL DRUG DESIGN, VAFRS COMPLEX, PHOSPHOLIPASE A2, CRYSTAL STRUCTURE, HYDROLASE
3i3i:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF BOTHROPSTOXIN-I CRYSTALLIZED AT 283 K | HOMOLOGUE PHOSPHOLIPASE A2, BOTHROPSTOXIN-I, BTHTX-I_10C, LYS49-PLA2 FROM BOTHROPS JARARACUSSU, SNAKE VENOM, ANTIBIOTIC, ANTIMICROBIAL, DISULFIDE BOND, MYOTOXIN, SECRETED, TOXIN
1tg1:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN RUSSELLS VIPER PHOSPHOLIPASE A2 AND A DESIGNED PEPTIDE INHIBITOR PHQ-LEU-VAL-ARG-TYR AT 1.2A RESOLUTION | PHOSPHOLIPASE A2, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1tj9:A (SER1) to (ASN109) STRUCTURE OF THE COMPLEXED FORMED BETWEEN GROUP II PHOSPHOLIPASE A2 AND A RATIONALLY DESIGNED TETRA PEPTIDE, VAL-ALA-ARG-SER AT 1.1A RESOLUTION | PHOSPHOLIPASE,COMPLEX,VARS,CRYSTAL STRUCTURE,1.1 RESOLUTION, HYDROLASE
1tk4:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF RUSSELLS VIPER PHOSPHOLIPASE A2 IN COMPLEX WITH A SPECIFICALLY DESIGNED TETRAPEPTIDE ALA-ILE- ARG-SER AT 1.1 A RESOLUTION | CRYSTAL STRUCTURE, TETRAPEPTIDE, PHOSPHOLIPASE A2, HYDROLASE
2h8i:A (SER1) to (ASN99) CRYSTAL STRUCTURE OF THE BOTHROPSTOXIN-I COMPLEXED WITH POLYETHYLENE GLYCOL | LYS49-PLA2S, MYOTOXICITY, TOXIN
2h8i:B (SER1) to (LEU100) CRYSTAL STRUCTURE OF THE BOTHROPSTOXIN-I COMPLEXED WITH POLYETHYLENE GLYCOL | LYS49-PLA2S, MYOTOXICITY, TOXIN
1jq8:A (SER1) to (ASN109) DESIGN OF SPECIFIC INHIBITORS OF PHOSPHOLIPASE A2: CRYSTAL STRUCTURE OF A COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 FROM DABOIA RUSSELLI PULCHELLA AND A DESIGNED PENTAPEPTIDE LEU-ALA-ILE-TYR-SER AT 2.0 RESOLUTION | NEUROTOXIC, DESIGNED PEPTIDE, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1jq8:B (SER1) to (ASN109) DESIGN OF SPECIFIC INHIBITORS OF PHOSPHOLIPASE A2: CRYSTAL STRUCTURE OF A COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 FROM DABOIA RUSSELLI PULCHELLA AND A DESIGNED PENTAPEPTIDE LEU-ALA-ILE-TYR-SER AT 2.0 RESOLUTION | NEUROTOXIC, DESIGNED PEPTIDE, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2o1n:A (SER1) to (ASN109) CRYSTAL STRUCTURE OF A COMPLEX OF PHOSPHOLIPASE A2 WITH A PEPTIDE ALA-ILE-ALA-SER AT 2.8 A RESOLUTION | PEPTIDE INHIBITOR, HYDROLASE
1xxs:A (SER1) to (ASN109) STRUCTURAL INSIGHTS FOR FATTY ACID BINDING IN A LYS49 PHOSPHOLIPASE A2: CRYSTAL STRUCTURE OF MYOTOXIN II FROM BOTHROPS MOOJENI COMPLEXED WITH STEARIC ACID | PHOSPHOLIPASE A2, STEARIC ACID, CRYSTAL STRUCTURE, DIMER INTERFACE, FATTY ACID BINDING, HYDROLASE
1xxs:B (PHE3) to (ASN109) STRUCTURAL INSIGHTS FOR FATTY ACID BINDING IN A LYS49 PHOSPHOLIPASE A2: CRYSTAL STRUCTURE OF MYOTOXIN II FROM BOTHROPS MOOJENI COMPLEXED WITH STEARIC ACID | PHOSPHOLIPASE A2, STEARIC ACID, CRYSTAL STRUCTURE, DIMER INTERFACE, FATTY ACID BINDING, HYDROLASE
1mf4:A (ASN1) to (ALA104) STRUCTURE-BASED DESIGN OF POTENT AND SELECTIVE INHIBITORS OF PHOSPHOLIPASE A2: CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN PHOSHOLIPASE A2 FROM NAJA NAJA SAGITTIFERA AND A DESIGNED PEPTIDE INHIBITOR AT 1.9 A RESOLUTION | NAJA NAJA SAGITTIFERA, PHOSPHOLIPASE A2, DESIGNED INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1mg6:A (SER1) to (ASN109) THE CRYSTAL STRUCTURE OF A K49 PLA2 FROM THE SNAKE VENOM OF AGKISTRODON ACUTUS | PLA2, HYDROLASE
1mks:A (LEU2) to (LYS108) CARBOXYLIC ESTER HYDROLASE, TRIGONAL FORM OF THE TRIPLE MUTANT | HYDROLASE, ENZYME, CARBOXYLIC ESTER HYDROLASE, TRIGONAL FORM
1yxl:A (ASN1) to (ALA104) CRYSTAL STRUCTURE OF A NOVEL PHOSPHOLIPASE A2 FROM NAJA NAJA SAGITTIFERA AT 1.5 A RESOLUTION | PHOSPHOLIPASE A2, MONOMER, COBRA, NAJA NAJA SAGITTIFERA, HYDROLASE
3cxi:A (SER1) to (ASN109) STRUCTURE OF BTHTX-I COMPLEXED WITH ALPHA-TOCOPHEROL | MYOTOXIN, BOTHROPS JARACUSSU, LYS49-PLA2, SNAKE VENOM, PHOSPHOLIPASE A2, X-RAY CRYSTALLOGRAPHY, SECRETED
3cxi:B (SER1) to (ASN109) STRUCTURE OF BTHTX-I COMPLEXED WITH ALPHA-TOCOPHEROL | MYOTOXIN, BOTHROPS JARACUSSU, LYS49-PLA2, SNAKE VENOM, PHOSPHOLIPASE A2, X-RAY CRYSTALLOGRAPHY, SECRETED
4uy1:A (GLY1) to (THR101) NOVEL PYRAZOLE SERIES OF GROUP X SECRETORY PHOSPHOLIPASE A2 (SPLA2-X) INHIBITORS | HYDROLASE, FRAGMENT BASED LEAD GENERATION, VIRTUAL SCREENING, DRUG DISCOVERY
4uy1:B (GLY1) to (THR101) NOVEL PYRAZOLE SERIES OF GROUP X SECRETORY PHOSPHOLIPASE A2 (SPLA2-X) INHIBITORS | HYDROLASE, FRAGMENT BASED LEAD GENERATION, VIRTUAL SCREENING, DRUG DISCOVERY