4wb5:A   (ALA218) to   (ALA298)  CRYSTAL STRUCTURE OF HUMAN CAMP-DEPENDENT PROTEIN KINASE A (CATALYTIC ALPHA SUBUNIT)  |   CATALYSIS, PROTEIN KINASE, ADENOSINE TRIPHOSPHATE, PHOSPHORYLATION 
4wb6:A   (ASN216) to   (ALA298)  CRYSTAL STRUCTURE OF A L205R MUTANT OF HUMAN CAMP-DEPENDENT PROTEIN KINASE A (CATALYTIC ALPHA SUBUNIT)  |   CUSHING'S SYNDROME, PROTEIN KINASE, PHOSPHORYLATION, MUTANT, ADENOSINE TRIPHOSPHATE, CATALYSIS 
4wb8:A   (VAL219) to   (ALA298)  CRYSTAL STRUCTURE OF HUMAN CAMP-DEPENDENT PROTEIN KINASE A (CATALYTIC ALPHA SUBUNIT), EXON 1 DELETION  |   CATALYSIS, PROTEIN KINASE, ADENOSINE TRIPHOSPHATE, PHOSPHORYLATION 
3e87:A   (VAL331) to   (LEU410)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF AKT2 IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   AKT2, KINASE, GSK3 BETA, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY 
3e87:B   (VAL331) to   (LEU410)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF AKT2 IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   AKT2, KINASE, GSK3 BETA, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY 
3e88:A   (VAL331) to   (LEU410)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF AKT2 IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   AKT2, KINASE, GSK3 BETA, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY 
3e88:B   (GLY328) to   (LEU410)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF AKT2 IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   AKT2, KINASE, GSK3 BETA, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY 
3e8d:A   (GLY328) to   (LEU410)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF AKT2 IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   AKT2, KINASE, GSK3 BETA, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY 
3e8d:B   (VAL331) to   (LEU410)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF AKT2 IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   AKT2, KINASE, GSK3 BETA, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY 
3e8c:A   (ALA218) to   (ALA298)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, PROTEIN KINASE INHIBITOR 
3e8c:B   (ALA218) to   (ALA298)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, PROTEIN KINASE INHIBITOR 
3e8c:C   (ALA218) to   (ALA298)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, PROTEIN KINASE INHIBITOR 
3e8c:E   (ALA218) to   (ALA298)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, PROTEIN KINASE INHIBITOR 
3e8e:B   (ALA218) to   (ALA298)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3e8e:L   (ALA218) to   (ALA298)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3e8e:P   (ALA218) to   (ALA298)  CRYSTAL STRUCTURES OF THE KINASE DOMAIN OF PKA IN COMPLEX WITH ATP- COMPETITIVE INHIBITORS  |   PKA, AKT2, KINASE, PKI, BOVINE, INHIBITOR, ATP-BINDING, CAMP, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
4gv1:A   (GLY327) to   (ALA409)  PKB ALPHA IN COMPLEX WITH AZD5363  |   PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2oh0:E   (ALA218) to   (ALA298)  CRYSTAL STRUCTURE OF PROTEIN KINASE A IN COMPLEX WITH PYRIDINE-PYRAZOLOPYRIDINE BASED INHIBITORS  |   PROTEIN KINASE A, AKT, TRANSFERASE 
3efw:A   (VAL310) to   (ASN386)  STRUCTURE OF AURORAA WITH PYRIDYL-PYRIMIDINE UREA INHIBITOR  |   AURORAA, STK6_HUMAN, ATP-BINDING, CELL CYCLE, KINASE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE-INHIBITOR COMPLEX 
2ayp:A   (HIS185) to   (LYS267)  CRYSTAL STRUCTURE OF CHK1 WITH AN INDOL INHIBITOR  |   PROTEIN-INHIBITOR COMPLEX, TRANSFERASE 
2b54:A   (ALA183) to   (VAL289)  HUMAN CYCLIN DEPENDENT KINASE 2 (CKD2)COMPLEXED WITH DIN- 232305  |   PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION, TRANSFERASE 
1nvq:A   (PRO188) to   (LYS267)  THE COMPLEX STRUCTURE OF CHECKPOINT KINASE CHK1/UCN-01  |   CHK1-UCN-01 COMPLEX, TRANSFERASE 
1nvr:A   (PRO188) to   (LYS267)  THE COMPLEX STRUCTURE OF CHECKPOINT KINASE CHK1/STAUROSPORINE  |   CHK1-STAUROSPORINE COMPLEX, TRANSFERASE 
1nvs:A   (PRO188) to   (LYS267)  THE COMPLEX STRUCTURE OF CHECKPOINT KINASE CHK1/SB218078  |   CHK1-SB218078 COMPLEX, TRANSFERASE 
4wsy:A   (ARG221) to   (GLN291)  CRYSTAL STRUCTURE OF HUMAN PIM-1 KINASE IN COMPLEX WITH A THIAZOLAMINE-INDAZOLE INHIBITOR.  |   TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2bfy:B   (LYS269) to   (ASN346)  COMPLEX OF AURORA-B WITH INCENP AND HESPERADIN.  |   TRANSFERASE, KINASE, MITOSIS, INHIBITION, TRANSFERASE COMPLEX 
2bmc:A   (HIS306) to   (SER387)  AURORA-2 T287D T288D COMPLEXED WITH PHA-680632  |   CELL CYCLE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION 
2bmc:C   (ASP307) to   (SER387)  AURORA-2 T287D T288D COMPLEXED WITH PHA-680632  |   CELL CYCLE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION 
2bmc:D   (HIS306) to   (SER387)  AURORA-2 T287D T288D COMPLEXED WITH PHA-680632  |   CELL CYCLE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION 
2bmc:E   (HIS306) to   (SER387)  AURORA-2 T287D T288D COMPLEXED WITH PHA-680632  |   CELL CYCLE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION 
2bmc:F   (VAL310) to   (SER387)  AURORA-2 T287D T288D COMPLEXED WITH PHA-680632  |   CELL CYCLE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION 
1o6k:A   (GLY328) to   (LEU410)  STRUCTURE OF ACTIVATED FORM OF PKB KINASE DOMAIN S474D WITH GSK3 PEPTIDE AND AMP-PNP  |   PROTEIN KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE 
2br1:A   (PRO188) to   (LYS267)  STRUCTURE-BASED DESIGN OF NOVEL CHK1 INHIBITORS: INSIGHTS INTO HYDROGEN BONDING AND PROTEIN-LIGAND AFFINITY  |   TRANSFERASE, DRUG DESIGN, FURANOPYRIMIDINE, MOLECULAR RECOGNITION, ONCOLOGY, PYRROLOPYRIMIDINE, X-RAY CRYSTALLOGRAPHY, KINASE 
2brb:A   (PRO188) to   (LYS267)  STRUCTURE-BASED DESIGN OF NOVEL CHK1 INHIBITORS: INSIGHTS INTO HYDROGEN BONDING AND PROTEIN-LIGAND AFFINITY  |   DRUG DESIGN, FURANOPYRIMIDINE, MOLECULAR RECOGNITION, ONCOLOGY, PYRROLOPYRIMIDINE, TRANSFERASE 
2brg:A   (PRO188) to   (LYS267)  STRUCTURE-BASED DESIGN OF NOVEL CHK1 INHIBITORS: INSIGHTS INTO HYDROGEN BONDING AND PROTEIN-LIGAND AFFINITY  |   DRUG DESIGN, FURANOPYRIMIDINE, MOLECULAR RECOGNITION, ONCOLOGY, PYRROLOPYRIMIDINE, ATP-BINDING, CELL CYCLE, DNA DAMAGE, KINASE, NUCLEAR PROTEIN, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
2brm:A   (PRO188) to   (LYS267)  STRUCTURE-BASED DESIGN OF NOVEL CHK1 INHIBITORS: INSIGHTS INTO HYDROGEN BONDING AND PROTEIN-LIGAND AFFINITY  |   DRUG DESIGN, FURANOPYRIMIDINE, MOLECULAR RECOGNITION, ONCOLOGY, PYRROLOPYRIMIDINE, ATP-BINDING, CELL CYCLE, DNA DAMAGE, KINASE, NUCLEAR PROTEIN, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
2brn:A   (PRO188) to   (LYS267)  STRUCTURE-BASED DESIGN OF NOVEL CHK1 INHIBITORS: INSIGHTS INTO HYDROGEN BONDING AND PROTEIN-LIGAND AFFINITY  |   DRUG DESIGN, FURANOPYRIMIDINE, MOLECULAR RECOGNITION, ONCOLOGY, PYRROLOPYRIMIDINE, ATP-BINDING, CELL CYCLE, DNA DAMAGE, KINASE, NUCLEAR PROTEIN, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
4x7q:A   (LEU217) to   (GLN287)  PIM2 KINASE IN COMPLEX WITH COMPOUND 1S  |   TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4hpu:E   (VAL219) to   (ALA298)  CRYSTAL STRUCTURE OF THE CATALYTIC SUBUNIT OF CAMP-DEPENDENT PROTEIN KINASE DISPLAYING PARTIAL PHOSPHORYL TRANSFER OF AMP-PNP ONTO A SUBSTRATE PEPTIDE  |   PROTEIN KINASE FOLD, PHOSPHOTRANSFERASE, REGULATORY SUBUNITS, PKI, MAGNESIUM, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3f9n:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHK1 KINASE IN COMPLEX WITH INHIBITOR 38  |   CHEK1, CHK1, KINASE, CELL CYCLE CHECKPOINT, ATP-BINDING, CYTOPLASM, DNA DAMAGE, DNA REPAIR, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE, UBL CONJUGATION 
2phk:A   (GLY207) to   (GLN288)  THE CRYSTAL STRUCTURE OF A PHOSPHORYLASE KINASE PEPTIDE SUBSTRATE COMPLEX: KINASE SUBSTRATE RECOGNITION  |   CATALYTIC MECHANISM, DIMERIZATION, PHOSPHORYLASE KINASE, REVERSIBLE PHOSPHORYLISATION, SUBSTRATE RECOGNITION, COMPLEX (TRANSFERASE- PEPTIDE), COMPLEX (TRANSFERASE-PEPTIDE) COMPLEX 
3fdn:A   (ASP307) to   (ASN386)  STRUCTURE-BASED DRUG DESIGN OF NOVEL AURORA KINASE A INHIBITORS: STRUCTURE BASIS FOR POTENCY AND SPECIFICITY  |   AURORA KINASE INHIBITORS, VIRTUAL SCREENING, X-RAY CO- CRYSTAL ANALYSIS, STRUCTURE-BASED DRUG DESIGN (SBDD), H- BONDING., ATP-BINDING, CELL CYCLE, KINASE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE 
3fe3:B   (PRO232) to   (ALA309)  CRYSTAL STRUCTURE OF THE KINASE MARK3/PAR-1: T211A-S215A DOUBLE MUTANT  |   SERINE/THREONINE PROTEIN KINASE; MARK;PAR-1; KIN1; UBA DOMAIN;C- TAK1;P78;MARK3, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
4hyh:A   (PRO188) to   (LYS267)  X-RAY CRYSTAL STRUCTURE OF COMPOUND 39 BOUND TO HUMAN CHK1 KINASE DOMAIN  |   SERINE/THREONINE-PROTEIN KINASE CHK1 INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4hyi:A   (PRO188) to   (LYS267)  X-RAY CRYSTAL STRUCTURE OF COMPOUND 40 BOUND TO HUMAN CHK1 KINASE DOMAIN  |   SERINE/THREONINE-PROTEIN KINASE CHK1 INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
2bzj:A   (ARG221) to   (GLN291)  CRYSTAL STRUCTURE OF THE HUMAN PIM1 IN COMPLEX WITH A RUTHENIUM ORGANOMETALLIC LIGAND RU3  |   PIM1, KINASE, CANCER, LEUKEMIA, NUCLEAR PROTEIN, NUCLEOTIDE- BINDING, TRANSFERASE 
4i20:A   (HIS893) to   (LEU979)  CRYSTAL STRUCTURE OF MONOMERIC (V948R) PRIMARY ONCOGENIC MUTANT L858R EGFR KINASE DOMAIN  |   KINASE DOMAIN, PHOSPHOTRANSFER, ATP BINDING, TRANSFERASE 
3fhi:A   (VAL219) to   (ALA298)  CRYSTAL STRUCTURE OF A COMPLEX BETWEEN THE CATALYTIC AND REGULATORY (RI{ALPHA}) SUBUNITS OF PKA  |   CAMP, CAMP DEPENDENT PROTEIN KINASE, PROTEIN-PROTEIN COMPLEX, AMP- PNP, PROTEIN KINASE REGULATION, NUCLEOTIDE BINDING, PROTEIN KINASE ACTIVITY, PROTEIN SERINE/THREONINE KINASE ACTIVITY, CAMP-DEPENDENT PROTEIN KINASE ACTIVITY, PROTEIN BINDING, ATP BINDING, KINASE ACTIVITY, TRANSFERASE ACTIVITY, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, CAMP-BINDING 
2c3j:A   (PRO188) to   (LYS267)  IDENTIFICATION OF A BURIED POCKET FOR POTENT AND SELECTIVE INHIBITION OF CHK1: PREDICTION AND VERIFICATION  |   DRUG DESIGN, MOLECULAR MODELING, MOLECULAR RECOGNITION, ONCOLOGY, TRANSFERASE, CELL CYCLE, DNA DAMAGE, DNA REPAIR, ATP-BINDING, KINASE, NUCLEAR PROTEIN, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, UBL CONJUGATION 
2c3k:A   (PRO188) to   (LYS267)  IDENTIFICATION OF A BURIED POCKET FOR POTENT AND SELECTIVE INHIBITION OF CHK1: PREDICTION AND VERIFICATION  |   DRUG DESIGN, MOLECULAR MODELING, MOLECULAR RECOGNITION, ONCOLOGY, ATP-BINDING, CELL CYCLE, DNA DAMAGE, DNA REPAIR, KINASE, NUCLEAR PROTEIN, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, UBL CONJUGATION 
4i41:A   (ARG221) to   (GLN291)  CRYSTAL STRUCTURE OF HUMAN SER/THR KINASE PIM1 IN COMPLEX WITH MITOXANTRONE  |   SER/THR KINASE, MITOXANTRONE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1ol2:C   (ALA183) to   (ASP288)  CYCLIN A BINDING GROOVE INHIBITOR H-ARG-ARG-LEU-ASN-(P-F-PHE)-NH2  |   CELL CYCLE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, CYCLIN A, LIGAND EXCHANGE, PEPTIDOMIMETICS, KINASE 
4iai:A   (VAL219) to   (ALA298)  X-RAY STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A IN COMPLEX WITH HIGH CA2+ CONCENTRATION, ADP AND PHOSPHORYLATED PEPTIDE PSP20  |   KINASE ENZYME, PHOSPHOTRANSFER, PHOSPHORYLATION, TRANSFERASE-PEPTIDE COMPLEX 
4iak:A   (VAL219) to   (ALA298)  LOW TEMPERATURE X-RAY STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A IN COMPLEX WITH HIGH SR2+ CONCENTRATION, ADP AND PHOSPHORYLATED PEPTIDE PSP20  |   KINASE ENZYME, PHOSPHOTRANSFER, PHOSPHORYLATION, TRANSFERASE-PEPTIDE COMPLEX 
4iaz:A   (VAL219) to   (ALA298)  STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A IN COMPLEX WITH HIGH BA2+ CONCENTRATION, ADP AND PHOSPHORYLATED PEPTIDE PSP20  |   KINASE ENZYME, PHOSPHOTRANSFER, PHOSPHORYLATED, TRANSFERASE-PEPTIDE COMPLEX 
4ib0:A   (VAL219) to   (ALA298)  X-RAY STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A IN COMPLEX WITH HIGH NA+ CONCENTRATION, ADP AND PHOSPHORYLATED PEPTIDE PSP20  |   KINASE ENZYME, PHOSPHOTRANSFER, PHOSPHORYLATED, TRANSFERASE-PEPTIDE COMPLEX 
4ib1:A   (VAL219) to   (ALA298)  STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A IN COMPLEX WITH HIGH K+ CONCENTRATION, ADP AND PHOSPHORYLATED PEPTIDE PSP20  |   KINASE ENZYME, PHOSPHOTRANSFER, PHOSPHORYLATED, TRANSFERASE-PEPTIDE COMPLEX 
2cgu:A   (PRO188) to   (LYS267)  IDENTIFICATION OF CHEMICALLY DIVERSE CHK1 INHIBITORS BY RECEPTOR-BASED VIRTUAL SCREENING  |   TRANSFERASE, DOCKING, DRUG DESIGN, ONCOLOGY, VIRTUAL SCREENING, ATP- BINDING, CELL CYCLE, DNA DAMAGE, DNA REPAIR, KINASE, NUCLEAR PROTEIN, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, UBL CONJUGATION 
2cgv:A   (PRO188) to   (LYS267)  IDENTIFICATION OF CHEMICALLY DIVERSE CHK1 INHIBITORS BY RECEPTOR-BASED VIRTUAL SCREENING  |   TRANSFERASE, DOCKING, DRUG DESIGN, ONCOLOGY, VIRTUAL SCREENING, ATP- BINDING, CELL CYCLE, DNA DAMAGE, DNA REPAIR, KINASE, NUCLEAR PROTEIN, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, UBL CONJUGATION 
2cgw:A   (PRO188) to   (LYS267)  IDENTIFICATION OF CHEMICALLY DIVERSE CHK1 INHIBITORS BY RECEPTOR-BASED VIRTUAL SCREENING  |   TRANSFERASE, DOCKING, DRUG DESIGN, ONCOLOGY, VIRTUAL SCREENING, ATP- BINDING, CELL CYCLE, DNA DAMAGE, DNA REPAIR, KINASE, NUCLEAR PROTEIN, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, UBL CONJUGATION 
2cgx:A   (PRO188) to   (LYS267)  IDENTIFICATION OF CHEMICALLY DIVERSE CHK1 INHIBITORS BY RECEPTOR-BASED VIRTUAL SCREENING  |   TRANSFERASE, DOCKING, DRUG DESIGN, ONCOLOGY, VIRTUAL SCREENING, ATP- BINDING, CELL CYCLE, DNA DAMAGE, DNA REPAIR, KINASE, NUCLEAR PROTEIN, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, UBL CONJUGATION 
4ij9:A   (VAL219) to   (ALA298)  BOVINE PKA C-ALPHA IN COMPLEX WITH 2-[[5-(4-PYRIDYL)-1H-1,2,4-TRIAZOL- 3-YL]SULFANYL]-1-(2-THIOPHENYL)ETHANONE  |   PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2qg5:D   (GLY202) to   (LEU286)  CRYPTOSPORIDIUM PARVUM CALCIUM DEPENDENT PROTEIN KINASE CGD7_1840  |   MALARIA, CALCIUM DEPENDENT KINASE, SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSFERASE 
2qhm:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHEK1 IN COMPLEX WITH INHIBITOR 2A  |   CHEK1, KINASE, CELL CYCLE CHECKPOINT, TRANSFERASE 
2qhn:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHEK1 IN COMPLEX WITH INHIBITOR 1A  |   CHEK1, KINASE, CELL CYCLE CHECKPOINT, TRANSFERASE 
3gc0:A   (SER197) to   (HIS303)  STRUCTURE OF THE CMGC CDK KINASE FROM GIARDIA LAMBLIA IN COMPLEX WITH AMP  |   SSGCID, KINASE, CMGC CDK, AMP, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE 
2qnj:B   (PRO232) to   (ALA309)  KINASE AND UBIQUITIN-ASSOCIATED DOMAINS OF MARK3/PAR-1  |   SERINE/THREONINE PROTEIN KINASE, UBIQUITIN-ASSOCIATED DOMAIN, MARK, PAR-1, TRANSFERASE 
4xw5:A   (VAL219) to   (ALA298)  X-RAY STRUCTURE OF PKAC WITH ATP, CP20, CALCIUM IONS  |   PROTEIN KINASE A, PHOSPHORYLATION, CATALYTIC SUBUNIT, REACTANT COMPLEX, TRANSFERASE 
4xw6:A   (ALA218) to   (ALA298)  X-RAY STRUCTURE OF PKAC WITH ADP, FREE PHOSPHATE ION, CP20, MAGNESIUM IONS  |   PROTEIN KINASE A, ATP HYDROLYSIS, CATALYTIC SUBUNIT, ATPASE, TRANSFERASE 
4iti:B   (GLU207) to   (GLN292)  CRYSTAL STRUCTURE OF RIP1 KINASE IN COMPLEX WITH NECROSTATIN-3 ANALOG  |   ALPHA/BETA, RIP1 KINASE, NECROPTOSIS, NECROSTATINS, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2qr8:A   (PRO587) to   (HIS681)  2.0A X-RAY STRUCTURE OF C-TERMINAL KINASE DOMAIN OF P90 RIBOSOMAL S6 KINASE 2 (RSK2)  |   KINASE DOMAIN, RSK2, AUTOINHIBITORY, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
2qr7:A   (PRO587) to   (HIS681)  2.0A X-RAY STRUCTURE OF C-TERMINAL KINASE DOMAIN OF P90 RIBOSOMAL S6 KINASE 2: SE-MET DERIVATIVE  |   KINASE DOMAIN, RSK2, AUTOINHIBITORY, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
2qvs:E   (VAL219) to   (ALA298)  CRYSTAL STRUCTURE OF TYPE IIA HOLOENZYME OF CAMP-DEPENDENT PROTEIN KINASE  |   CRYSTAL STRUCTURE, CAMP-DEPENDENT PROTEIN KINASE, TYPE IIA HOLOENZYME, ISOFORM DIVERSITY, ALTERNATIVE SPLICING, ATP- BINDING, CYTOPLASM, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ACETYLATION, CAMP-BINDING, TRANSFERASE/TRANSFERASE REGULATOR COMPLEX 
2r0u:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHEK1 IN COMPLEX WITH INHIBITOR 54  |   CHEK1, KINASE, CELL CYCLE CHECK POINT, ATP-BINDING, CYTOPLASM, DNA DAMAGE, DNA REPAIR, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE, UBL CONJUGATION 
4j8m:A   (ASP307) to   (ASN386)  AURORA A IN COMPLEX WITH CD532  |   AURORA A, TYPE II, KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4j8n:A   (LYS309) to   (ASN386)  AURORA A KINASE APO  |   AURORA A, KINASE DOMAIN, TRANSFERASE 
4j8n:B   (LYS309) to   (SER387)  AURORA A KINASE APO  |   AURORA A, KINASE DOMAIN, TRANSFERASE 
4j8n:C   (LYS309) to   (ASN386)  AURORA A KINASE APO  |   AURORA A, KINASE DOMAIN, TRANSFERASE 
4j8n:D   (LYS309) to   (ASN386)  AURORA A KINASE APO  |   AURORA A, KINASE DOMAIN, TRANSFERASE 
4jbp:A   (ASP307) to   (ASN386)  NOVEL AURORA KINASE INHIBITORS REVEAL MECHANISMS OF HURP IN NUCLEATION OF CENTROSOMAL AND KINETOCHORE MICROTUBULES  |   AURORA KINASE INHIBITORS, HURP, MITOTIC SPINDLE, TRANSFERASE 
3tki:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHK1 IN COMPLEX WITH INHIBITOR S25  |   CHK1, KINASE, CELL CHECKPOINT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1q8u:A   (ALA218) to   (ALA298)  THE CATALYTIC SUBUNIT OF CAMP-DEPENDENT PROTEIN KINASE IN COMPLEX WITH RHO-KINASE INHIBITOR H-1152P  |   KINASE-INHIBITOR-COMPLEX, PHOSPHOTRANSFERASE/INHIBITOR, CAMP, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, ATP- BINDING, PKA, RHO-KINASE, TRANSFERASE/TRANSFERASE INHIBITOR COMPLEX 
4jik:A   (PRO188) to   (LYS267)  X-RAY CRYSTAL STRUCTURE OF COMPOUND 22A (R)-2-(4-CHLOROPHENYL)-8- (PIPERIDIN-3-YLAMINO)IMIDAZO[1,2-C]PYRIMIDINE-5-CARBOXAMIDE BOUND TO HUMAN CHK1 KINASE DOMAIN  |   KINASE PHOSPHATASE TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3h0z:B   (VAL310) to   (ASN386)  AURORA A IN COMPLEX WITH A BISANILINOPYRIMIDINE  |   PROTEIN:INHIBITOR COMPLEX AURORA-A, CELL CYCLE, SERINE/THREONINE, PROTEIN KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
1ql6:A   (GLY207) to   (GLN288)  THE CATALYTIC MECHANISM OF PHOSPHORYLASE KINASE PROBED BY MUTATIONAL STUDIES  |   KINASE (GLYCOGEN METABOLISM), GLYCOGEN METABOLISM, TRANSFERASE, SERINE/THREONINE-PROTEIN, KINASE, ATP-BINDING, CALMODULIN-BINDING 
2uw3:A   (VAL219) to   (ALA298)  STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH 5-METHYL-4- PHENYL-1H-PYRAZOLE  |   TRANSFERASE/INHIBITOR, CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION, TRANSFERASE/INHIBITOR COMPLEX 
4jx3:A   (ARG221) to   (GLN291)  CRYSTAL STRUCTURE OF PIM1 KINASE  |   HUMAN PROTEIN KINASES, SERINE/THREONINE-PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE 
4jx7:A   (ARG221) to   (GLN291)  CRYSTAL STRUCTURE OF PIM1 KINASE IN COMPLEX WITH INHIBITOR 2-[(TRANS- 4-AMINOCYCLOHEXYL)AMINO]-4-{[3-(TRIFLUOROMETHYL) PHENYL]AMINO}PYRIDO[4,3-D]PYRIMIDIN-5(6H)-ONE  |   SERINE/THREONINE-PROTEIN KINASES, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3u9n:A   (PRO188) to   (LYS267)  X-RAY CRYSTAL STRUCTURE OF COMPOUND 1 BOUND TO HUMAN CHK1 KINASE DOMAIN  |   PROTEIN KINASE DOMAIN, ATPASE, ATP BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2uzw:E   (VAL219) to   (ALA298)  PKA STRUCTURES OF INDAZOLE-PYRIDINE SERIES OF AKT INHIBITORS  |   CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, PHOSPHORYLATION, PROTEIN KINASE A, NUCLEOTIDE-BINDING, ATP-BINDING, AKT INHIBITORS, NUCLEAR PROTEIN 
4ynz:B   (GLY195) to   (LYS275)  STRUCTURE OF THE N-TERMINAL DOMAIN OF SAD  |   KINASE DOMAIN, UBA DOMAIN, TRANSFERASE 
4yom:B   (GLY195) to   (GLY273)  STRUCTURE OF SAD KINASE  |   KINASE DOMAIN, UBA DOMAIN, KA1 DOMAIN, TRANSFERASE 
3uc4:A   (ASP194) to   (LYS279)  THE CRYSTAL STRUCTURE OF SNF1-RELATED KINASE 2.6  |   SNRK2.6, KINASE, ABA SIGNALING, TRANSFERASE 
2etr:A   (GLU258) to   (LYS339)  CRYSTAL STRUCTURE OF ROCK I BOUND TO Y-27632  |   DIMERIZATION, DIMER, PHOSPHORYLATION, KINASE, YOSHITOMI, TRANSFERASE 
2etr:B   (GLU258) to   (LYS339)  CRYSTAL STRUCTURE OF ROCK I BOUND TO Y-27632  |   DIMERIZATION, DIMER, PHOSPHORYLATION, KINASE, YOSHITOMI, TRANSFERASE 
2euf:B   (PRO199) to   (LEU303)  X-RAY STRUCTURE OF HUMAN CDK6-VCYCLIN IN COMPLEX WITH THE INHIBITOR PD0332991  |   INHIBITOR COMPLEX OF HUMAN CYCLIN-DEPENDENT KINASE 6, CELL CYCLE- TRANSFERASE COMPLEX 
1rdq:E   (VAL219) to   (ALA298)  HYDROLYSIS OF ATP IN THE CRYSTAL OF Y204A MUTANT OF CAMP-DEPENDENT PROTEIN KINASE  |   CAMP-DEPENDENT PROTEIN KINASE,CATALYTIC MECHANISM, ATP HYDROLYSIS, TWO NUCLEOTIDE STATES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1re8:A   (ALA218) to   (ALA298)  CRYSTAL STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE COMPLEXED WITH BALANOL ANALOG 2  |   PROTEIN KINASE, NATURAL PRODUCT INHIBITOR, LIGAND BINDING, SPECIFICITY DETERMINANTS, CONFORMATIONAL MALLEABILITY, TRANSFERASE 
3ujg:A   (ASP194) to   (LYS279)  CRYSTAL STRUCTURE OF SNRK2.6 IN COMPLEX WITH HAB1  |   SNRK2.6, KINASE, PROTEIN PHOSPHATASE 2C, ABA SIGNALING, SIGNALING PROTEIN 
4yxs:A   (ALA218) to   (ALA298)  CAMP-DEPENDENT PROTEIN KINASE PKA CATALYTIC SUBUNIT WITH PKI-5-24  |   ATP-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, CAMP, PROTEIN KINASE INHIBITOR, TRANSFERASE-IN COMPLEX, TRANSFERASE-INHIBITOR COMPLEX 
2f7e:E   (VAL219) to   (ALA298)  PKA COMPLEXED WITH (S)-2-(1H-INDOL-3-YL)-1-(5-ISOQUINOLIN-6- YL-PYRIDIN-3-YLOXYMETHYL-ETYLAMINE  |   PROTEIN KINASE A, AKT INHIBITORS, TRANSFERASE 
3unz:A   (ASP307) to   (ALA385)  AURORA A IN COMPLEX WITH RPM1679  |   PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3unz:B   (ASP307) to   (ALA385)  AURORA A IN COMPLEX WITH RPM1679  |   PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3uod:A   (LYS309) to   (ASN386)  AURORA A IN COMPLEX WITH RPM1693  |   PROTEIN KINASE, AURORA A, INHIBITOR, DFG-IN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3up2:A   (LYS309) to   (ASN386)  AURORA A IN COMPLEX WITH RPM1686  |   PROTEIN KINASE, AURORA A, INHIBITOR, DFG-IN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3hyh:A   (GLU232) to   (VAL308)  CRYSTAL STRUCTURE OF THE PROTEIN KINASE DOMAIN OF YEAST AMP-ACTIVATED PROTEIN KINASE SNF1  |   KINASE DOMAIN, TRANSFERASE, ATP-BINDING, CARBOHYDRATE METABOLISM, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE 
3hyh:B   (GLU232) to   (VAL308)  CRYSTAL STRUCTURE OF THE PROTEIN KINASE DOMAIN OF YEAST AMP-ACTIVATED PROTEIN KINASE SNF1  |   KINASE DOMAIN, TRANSFERASE, ATP-BINDING, CARBOHYDRATE METABOLISM, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE 
3v5t:A   (CYS231) to   (THR312)  CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1299  |   SERINE/THREONINE PROTEIN KINASE, CALCIUM-BINDING, ATP-BINDING, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2vnw:A   (ALA218) to   (ALA298)  STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH (1-(9H-PURIN-6- YL)PIPERIDIN-4-YL)METHANAMINE  |   TRANSFERASE, LIPOPROTEIN, ATP-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, CAMP, KINASE, NUCLEUS, MYRISTATE, CYTOPLASM 
2vo0:A   (ALA218) to   (ALA298)  STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH  C-(4-(4- CHLOROPHENYL)-1-(7H-PYRROLO(2,3-D)PYRIMIDIN-4-YL)PIPERIDIN- 4-YL)METHYLAMINE  |   TRANSFERASE, LIPOPROTEIN, ATP-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, CAMP, KINASE, NUCLEUS, MYRISTATE, CYTOPLASM 
2vo3:A   (VAL219) to   (ALA298)  STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH  C-(4-(4- CHLOROPHENYL)-1-(7H-PYRROLO(2,3-D)PYRIMIDIN-4-YL)PIPERIDIN- 4-YL)METHYLAMINE  |   TRANSFERASE, LIPOPROTEIN, ATP-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, CAMP, KINASE, NUCLEUS, MYRISTATE, CYTOPLASM 
2vo7:A   (VAL219) to   (ALA298)  STRUCTURE OF PKA COMPLEXED WITH 4-(4-CHLOROBENZYL)-1-(7H- PYRROLO(2,3-D)PYRIMIDIN-4-YL)PIPERIDIN-4-YLAMINE  |   TRANSFERASE, LIPOPROTEIN, ATP-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, CAMP, KINASE, NUCLEUS, MYRISTATE, CYTOPLASM 
3vap:A   (LYS309) to   (ASN386)  SYNTHESIS AND SAR STUDIES OF IMIDAZO-[1,2-A]-PYRAZINE AURORA KINASE INHIBITORS WITH IMPROVED OFF TARGET KINASE SELECTIVITY  |   KINASE, CELL CYCLE, INHIBITOR, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3i6u:A   (ALA402) to   (GLN487)  STRUCTURE AND ACTIVATION MECHANISM OF THE CHK2 DNA-DAMAGE CHECKPOINT KINASE  |   SER/THR PROTEIN KINASE, FHA DOMAIN, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, KINASE, LI-FRAUMENI SYNDROME, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3i6u:B   (ALA407) to   (GLN487)  STRUCTURE AND ACTIVATION MECHANISM OF THE CHK2 DNA-DAMAGE CHECKPOINT KINASE  |   SER/THR PROTEIN KINASE, FHA DOMAIN, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, KINASE, LI-FRAUMENI SYNDROME, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3i6w:A   (ASN405) to   (GLN487)  STRUCTURE AND ACTIVATION MECHANISM OF THE CHK2 DNA-DAMAGE CHECKPOINT KINASE  |   SER/THR PROTEIN KINASE, FHA DOMAIN, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, KINASE, LI-FRAUMENI SYNDROME, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3i6w:B   (ASN405) to   (GLN487)  STRUCTURE AND ACTIVATION MECHANISM OF THE CHK2 DNA-DAMAGE CHECKPOINT KINASE  |   SER/THR PROTEIN KINASE, FHA DOMAIN, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, KINASE, LI-FRAUMENI SYNDROME, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3i6w:C   (ASN405) to   (GLN487)  STRUCTURE AND ACTIVATION MECHANISM OF THE CHK2 DNA-DAMAGE CHECKPOINT KINASE  |   SER/THR PROTEIN KINASE, FHA DOMAIN, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, KINASE, LI-FRAUMENI SYNDROME, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3i6w:D   (ASN405) to   (GLN487)  STRUCTURE AND ACTIVATION MECHANISM OF THE CHK2 DNA-DAMAGE CHECKPOINT KINASE  |   SER/THR PROTEIN KINASE, FHA DOMAIN, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, KINASE, LI-FRAUMENI SYNDROME, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3i6w:E   (ASN405) to   (GLN487)  STRUCTURE AND ACTIVATION MECHANISM OF THE CHK2 DNA-DAMAGE CHECKPOINT KINASE  |   SER/THR PROTEIN KINASE, FHA DOMAIN, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, KINASE, LI-FRAUMENI SYNDROME, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3i6w:F   (ASN405) to   (GLN487)  STRUCTURE AND ACTIVATION MECHANISM OF THE CHK2 DNA-DAMAGE CHECKPOINT KINASE  |   SER/THR PROTEIN KINASE, FHA DOMAIN, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, KINASE, LI-FRAUMENI SYNDROME, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3i6w:G   (ASN405) to   (GLN487)  STRUCTURE AND ACTIVATION MECHANISM OF THE CHK2 DNA-DAMAGE CHECKPOINT KINASE  |   SER/THR PROTEIN KINASE, FHA DOMAIN, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, KINASE, LI-FRAUMENI SYNDROME, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3i6w:H   (ASN405) to   (GLN487)  STRUCTURE AND ACTIVATION MECHANISM OF THE CHK2 DNA-DAMAGE CHECKPOINT KINASE  |   SER/THR PROTEIN KINASE, FHA DOMAIN, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, KINASE, LI-FRAUMENI SYNDROME, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
2gdo:A   (HIS185) to   (LYS267)  4-(AMINOALKYLAMINO)-3-BENZIMIDAZOLE-QUINOLINONES AS POTENT CHK1 INHIBITORS  |   DRUG DESIGN, ATP-BINDING, CELL CYCLE, DNA DAMAGE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
2gfc:A   (ALA218) to   (ALA298)  CAMP-DEPENDENT PROTEIN KINASE PKA CATALYTIC SUBUNIT WITH PKI-5-24  |   BINARY COMPLEX, PEPTIDE INHIBITOR, TRANSFERASE 
1syk:A   (VAL219) to   (ALA298)  CRYSTAL STRUCTURE OF E230Q MUTANT OF CAMP-DEPENDENT PROTEIN KINASE REVEALS UNEXPECTED APOENZYME CONFORMATION  |   E230Q MUTANT; CATALYTIC SUBUNIT; CAMP-DEPENDENT PROTEIN KINASE; APOENZYME CONFORMATION; N-TERMINAL A-HELIX, TRANSFERASE 
1syk:B   (VAL219) to   (ALA298)  CRYSTAL STRUCTURE OF E230Q MUTANT OF CAMP-DEPENDENT PROTEIN KINASE REVEALS UNEXPECTED APOENZYME CONFORMATION  |   E230Q MUTANT; CATALYTIC SUBUNIT; CAMP-DEPENDENT PROTEIN KINASE; APOENZYME CONFORMATION; N-TERMINAL A-HELIX, TRANSFERASE 
1szm:B   (VAL219) to   (ALA298)  DUAL BINDING MODE OF BISINDOLYLMALEIMIDE 2 TO PROTEIN KINASE A (PKA)  |   PKA, PKC, BISINDOLYL MALEIMIDE 2, LY333531, SELECTIVITY, SURROGATE KINASE, AMINO ACID RESIDUE EXCHANGE, X-RAY STRUCTURE, TRANSFERASE 
2gng:A   (ALA218) to   (ALA298)  PROTEIN KINASE A FIVEFOLD MUTANT MODEL OF RHO-KINASE  |   PKA, MUTANT, RHO-KINASE, SURROGATE, INHIBITOR, TRANSFERASE/TRANSFERASE INHIBITOR COMPLEX 
2w1d:A   (VAL310) to   (ASN386)  STRUCTURE DETERMINATION OF AURORA KINASE IN COMPLEX WITH INHIBITOR  |   NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, POLYMORPHISM, PHOSPHOPROTEIN, KINASE, CANCER, AURORA, INHIBITOR, CELL CYCLE 
2w1e:A   (GLU308) to   (ASN386)  STRUCTURE DETERMINATION OF AURORA KINASE IN COMPLEX WITH INHIBITOR  |   NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, POLYMORPHISM, PHOSPHOPROTEIN, KINASE, CANCER, AURORA, INHIBITOR, CELL CYCLE 
2w96:B   (ALA192) to   (LEU295)  CRYSTAL STRUCTURE OF CDK4 IN COMPLEX WITH A D-TYPE CYCLIN  |   SERINE/THREONINE-PROTEIN KINASE, CHROMOSOMAL REARRANGEMENT, ATP-BINDING, TRANSFERASE, POLYMORPHISM, CELL DIVISION, PROTO-ONCOGENE, PHOSPHOPROTEIN, DISEASE MUTATION, NUCLEOTIDE-BINDING, CYCLIN DEPENDENT KINASE, KINASE, CYCLIN, ONCOLOGY, CELL CYCLE, DRUG DESGN 
3is5:A   (ASP318) to   (GLN395)  CRYSTAL STRUCTURE OF CDPK KINASE DOMAIN FROM TOXOPLASMA GONDII, TGME49_018720  |   TOXOPLASMA GONDII, CDPK, STRUCTURAL GENOMICS, PARASITOLOGY, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
2h6d:A   (GLY192) to   (GLN270)  PROTEIN KINASE DOMAIN OF THE HUMAN 5'-AMP-ACTIVATED PROTEIN KINASE CATALYTIC SUBUNIT ALPHA-2 (AMPK ALPHA-2 CHAIN)  |   ATP-BINDING; CHOLESTEROL BIOSYNTHESIS; FATTY ACID BIOSYNTHESIS;KINASE; LIPID SYNTHESIS; NUCLEOTIDE-BINDING; PHOSPHORYLATION; SERINE/THREONINE-PROTEIN KINASE; STEROID BIOSYNTHESIS; STEROL BIOSYNTHESIS; TRANSFERASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, SIGNALING PROTEIN, TRANSFERASE, SIGNALING PROTEIN,TRANSFERASE 
2hak:A   (GLY228) to   (VAL306)  CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1  |   SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
2hak:C   (PRO229) to   (ASN305)  CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1  |   SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
2hak:D   (PRO229) to   (ASN305)  CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1  |   SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
2hak:E   (PRO229) to   (VAL306)  CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1  |   SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
2hak:F   (PRO229) to   (VAL306)  CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1  |   SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
2hak:G   (ASP232) to   (VAL306)  CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1  |   SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
3vqh:A   (VAL219) to   (ALA298)  BROMINE SAD PARTIALLY RESOLVES MULTIPLE BINDING MODES FOR PKA INHIBITOR H-89  |   PROTEIN-INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2wmq:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   SERINE/THREONINE-PROTEIN KINASE, POLYMORPHISM, PHOSPHOPROTEIN, UBL CONJUGATION, ISOPEPTIDE BOND, CHECKPOINT KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE KINASE, DNA DAMAGE, DNA REPAIR, ATP-BINDING, TRANSFERASE, CHK1, KINASE, NUCLEUS, CYTOPLASM, CELL CYCLE 
2wmr:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   SERINE/THREONINE-PROTEIN KINASE, POLYMORPHISM, PHOSPHOPROTEIN, UBL CONJUGATION, ISOPEPTIDE BOND, CHECKPOINT KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE KINASE, DNA DAMAGE, DNA REPAIR, ATP-BINDING, TRANSFERASE, CHK1, KINASE, NUCLEUS, CYTOPLASM, CELL CYCLE 
2wms:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   SERINE/THREONINE-PROTEIN KINASE, POLYMORPHISM, PHOSPHOPROTEIN, UBL CONJUGATION, ISOPEPTIDE BOND, CHECKPOINT KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE KINASE, DNA DAMAGE, DNA REPAIR, ATP-BINDING, TRANSFERASE, CHK1, KINASE, NUCLEUS, CYTOPLASM, CELL CYCLE 
2wmt:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   SERINE/THREONINE-PROTEIN KINASE, POLYMORPHISM, PHOSPHOPROTEIN, UBL CONJUGATION, ISOPEPTIDE BOND, CHECKPOINT KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE KINASE, DNA DAMAGE, DNA REPAIR, ATP-BINDING, TRANSFERASE, CHK1, KINASE, NUCLEUS, CYTOPLASM, CELL CYCLE 
2wmu:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   SERINE/THREONINE-PROTEIN KINASE, POLYMORPHISM, PHOSPHOPROTEIN, UBL CONJUGATION, ISOPEPTIDE BOND, CHECKPOINT KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE KINASE, DNA DAMAGE, DNA REPAIR, ATP-BINDING, TRANSFERASE, CHK1, KINASE, NUCLEUS, CYTOPLASM, CELL CYCLE 
2wmw:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   SERINE/THREONINE-PROTEIN KINASE, POLYMORPHISM, PHOSPHOPROTEIN, UBL CONJUGATION, ISOPEPTIDE BOND, CHECKPOINT KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE KINASE, DNA DAMAGE, DNA REPAIR, ATP-BINDING, TRANSFERASE, CHK1, KINASE, NUCLEUS, CYTOPLASM, CELL CYCLE 
2wtk:E   (ASP261) to   (ILE382)  STRUCTURE OF THE HETEROTRIMERIC LKB1-STRADALPHA-MO25ALPHA COMPLEX  |   TRANSFERASE-METAL-BINDING PROTEIN COMPLEX, TRANSFERASE METAL-BINDING PROTEIN COMPLEX, KINASE, NUCLEUS, SERINE/THREONINE-PROTEIN KINASE, PSEUDOKINASE, PHOSPHOPROTEIN, SIGNAL TRANSDUCTION, TRANSFERASE, NUCLEOTIDE-BINDING 
2wtk:F   (PHE234) to   (LYS311)  STRUCTURE OF THE HETEROTRIMERIC LKB1-STRADALPHA-MO25ALPHA COMPLEX  |   TRANSFERASE-METAL-BINDING PROTEIN COMPLEX, TRANSFERASE METAL-BINDING PROTEIN COMPLEX, KINASE, NUCLEUS, SERINE/THREONINE-PROTEIN KINASE, PSEUDOKINASE, PHOSPHOPROTEIN, SIGNAL TRANSDUCTION, TRANSFERASE, NUCLEOTIDE-BINDING 
2i0e:B   (VAL522) to   (ARG601)  STRUCTURE OF CATALYTIC DOMAIN OF HUMAN PROTEIN KINASE C BETA II COMPLEXED WITH A BISINDOLYLMALEIMIDE INHIBITOR  |   PROTEIN KINASE C BETA II, PROTEIN KINASE C, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE 
2wtv:B   (ASP307) to   (ASN386)  AURORA-A INHIBITOR STRUCTURE  |   KINASE, CELL CYCLE, TRANSFERASE, PHOSPHOPROTEIN 
2wtv:D   (ASP307) to   (ASN386)  AURORA-A INHIBITOR STRUCTURE  |   KINASE, CELL CYCLE, TRANSFERASE, PHOSPHOPROTEIN 
1ung:A   (SER180) to   (PHE289)  STRUCTURAL MECHANISM FOR THE INHIBITION OF CDK5-P25 BY ROSCOVITINE, ALOISINE AND INDIRUBIN.  |   CELL CYCLE, COMPLEX(KINASE/ACTIVATOR), INHIBITORS, NEURODEGENERATIVE DISEASES 
1unh:A   (SER180) to   (SER287)  STRUCTURAL MECHANISM FOR THE INHIBITION OF CDK5-P25 BY ROSCOVITINE, ALOISINE AND INDIRUBIN.  |   CELL CYCLE, NEURODEGENERATIVE DISEASES, INDIRUBIN 
5aae:A   (LYS309) to   (ASN386)  AURORA A KINASE BOUND TO AN IMIDAZOPYRIDINE INHIBITOR (14D)  |   TRANSFERASE, AURORA-A, IMIDAZOPYRIDINE, AURORA KINASE, INHIBITOR 
4med:A   (GLY220) to   (GLN291)  CRYSTAL STRUCTURE OF SER/THR KINASE PIM1 IN COMPLEX WITH THIORIDAZINE DERIVATIVES  |   PROTEIN-LIGAND COMPLEX, KINASE, ONCOGENE, ATP BINDING, PHOSPHORYLATION, NUCLEUS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1v0p:A   (SER179) to   (GLU286)  STRUCTURE OF P. FALCIPARUM PFPK5-PURVALANOL B LIGAND COMPLEX  |   TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, CDK 
2x8d:A   (PRO188) to   (LYS267)  DISCOVERY OF A NOVEL CLASS OF TRIAZOLONES AS CHECKPOINT KINASE INHIBITORS - HIT TO LEAD EXPLORATION  |   NUCLEOTIDE-BINDING, CYTOSKELETON, PHOSPHOPROTEIN, ISOPEPTIDE BOND, CELL CYCLE, TRANSFERASE, DNA DAMAGE, DNA REPAIR 
2x8e:A   (PRO188) to   (LYS267)  DISCOVERY OF A NOVEL CLASS OF TRIAZOLONES AS CHECKPOINT KINASE INHIBITORS - HIT TO LEAD EXPLORATION  |   NUCLEOTIDE-BINDING, CYTOSKELETON, PHOSPHOPROTEIN, ISOPEPTIDE BOND, CELL CYCLE, TRANSFERASE, DNA DAMAGE, DNA REPAIR 
2x8i:A   (PRO188) to   (LYS267)  DISCOVERY OF A NOVEL CLASS OF TRIAZOLONES AS CHECKPOINT KINASE INHIBITORS - HIT TO LEAD EXPLORATION  |   NUCLEOTIDE-BINDING, CYTOSKELETON, PHOSPHOPROTEIN, ISOPEPTIDE BOND, CELL CYCLE, TRANSFERASE, DNA DAMAGE, DNA REPAIR 
2iwi:A   (LEU217) to   (GLN287)  CRYSTAL STRUCTURE OF THE HUMAN PIM2 IN COMPLEX WITH A RUTHENIUM ORGANOMETALLIC LIGAND RU1  |   NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, PIM2, KINASE, CANCER, LEUKEMIA, TRANSFERASE, ATP-BINDING, PROTO- ONCOGENE, PHOSPHORYLATION 
2iwi:B   (LEU217) to   (GLN287)  CRYSTAL STRUCTURE OF THE HUMAN PIM2 IN COMPLEX WITH A RUTHENIUM ORGANOMETALLIC LIGAND RU1  |   NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, PIM2, KINASE, CANCER, LEUKEMIA, TRANSFERASE, ATP-BINDING, PROTO- ONCOGENE, PHOSPHORYLATION 
3j4q:D   (VAL219) to   (ALA298)  PSEUDO-ATOMIC MODEL OF THE AKAP18-PKA COMPLEX IN A BENT CONFORMATION DERIVED FROM ELECTRON MICROSCOPY  |   A-KINASE ANCHORING PROTEIN, CAMP-DEPENDENT KINASE, RII, PKA REGULATORY SUBUNIT II, PHOSPHORYLATION, ANCHORING, INTRINSIC DISORDER, TRANSFERASE 
3j4q:E   (VAL219) to   (ALA298)  PSEUDO-ATOMIC MODEL OF THE AKAP18-PKA COMPLEX IN A BENT CONFORMATION DERIVED FROM ELECTRON MICROSCOPY  |   A-KINASE ANCHORING PROTEIN, CAMP-DEPENDENT KINASE, RII, PKA REGULATORY SUBUNIT II, PHOSPHORYLATION, ANCHORING, INTRINSIC DISORDER, TRANSFERASE 
3j4r:D   (VAL219) to   (ALA298)  PSEUDO-ATOMIC MODEL OF THE AKAP18-PKA COMPLEX IN A LINEAR CONFORMATION DERIVED FROM ELECTRON MICROSCOPY  |   A-KINASE ANCHORING PROTEIN, CAMP-DEPENDENT KINASE, RII, PKA REGULATORY SUBUNIT II, PHOSPHORYLATION, ANCHORING, INTRINSIC DISORDER, TRANSFERASE 
3j4r:E   (VAL219) to   (ALA298)  PSEUDO-ATOMIC MODEL OF THE AKAP18-PKA COMPLEX IN A LINEAR CONFORMATION DERIVED FROM ELECTRON MICROSCOPY  |   A-KINASE ANCHORING PROTEIN, CAMP-DEPENDENT KINASE, RII, PKA REGULATORY SUBUNIT II, PHOSPHORYLATION, ANCHORING, INTRINSIC DISORDER, TRANSFERASE 
5ap7:A   (LYS714) to   (GLN792)  NATURALLY OCCURRING MUTATIONS IN THE MPS1 GENE PREDISPOSE CELLS TO KINASE INHIBITOR DRUG RESISTANCE.  |   TRANSFERASE, MPS1, MITOSIS 
1jkt:A   (LEU196) to   (LYS276)  TETRAGONAL CRYSTAL FORM OF A CATALYTIC DOMAIN OF DEATH-ASSOCIATED PROTEIN KINASE  |   TRANSFERASE 
1jkt:B   (GLY195) to   (PRO277)  TETRAGONAL CRYSTAL FORM OF A CATALYTIC DOMAIN OF DEATH-ASSOCIATED PROTEIN KINASE  |   TRANSFERASE 
2xey:A   (GLU187) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   TRANSFERASE,  DNA REPAIR, CELL CYCLE 
2xez:A   (GLU187) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   TRANSFERASE, DNA REPAIR, CELL CYCLE 
1jlu:E   (ASN216) to   (ALA298)  CRYSTAL STRUCTURE OF THE CATALYTIC SUBUNIT OF CAMP-DEPENDENT PROTEIN KINASE COMPLEXED WITH A PHOSPHORYLATED SUBSTRATE PEPTIDE AND DETERGENT  |   PROTEIN KINASE-PHOSPHORYLATED SUBSTRATE COMPLEX, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
2xj1:A   (ARG221) to   (GLN291)  PROTEIN KINASE PIM-1 IN COMPLEX WITH SMALL MOLECULE INIBITOR  |   PHOSPHORYLATION, TRANSFERASE 
2j90:A   (GLU197) to   (ILE278)  CRYSTAL STRUCTURE OF HUMAN ZIP KINASE IN COMPLEX WITH A TETRACYCLIC PYRIDONE INHIBITOR (PYRIDONE 6)  |   NUCLEAR PROTEIN, NUCLEOTIDE-BINDING, SERINE/THREONINE- PROTEIN KINASE, CHROMATIN REGULATOR, MYOSIN PHOSPHORYLATION, KINASE, MUSCLE, APOPTOSIS, TRANSFERASE, ATP-BINDING 
2j90:B   (GLU197) to   (ALA277)  CRYSTAL STRUCTURE OF HUMAN ZIP KINASE IN COMPLEX WITH A TETRACYCLIC PYRIDONE INHIBITOR (PYRIDONE 6)  |   NUCLEAR PROTEIN, NUCLEOTIDE-BINDING, SERINE/THREONINE- PROTEIN KINASE, CHROMATIN REGULATOR, MYOSIN PHOSPHORYLATION, KINASE, MUSCLE, APOPTOSIS, TRANSFERASE, ATP-BINDING 
1vzo:A   (ALA235) to   (GLN319)  THE STRUCTURE OF THE N-TERMINAL KINASE DOMAIN OF MSK1 REVEALS A NOVEL AUTOINHIBITORY CONFORMATION FOR A DUAL KINASE PROTEIN  |   PROTEIN KINASE, TRANSFERASE, PHOSPHORYLATION, SERINE/THREONINE PROTEIN KINASE 
3wzu:A   (ASP316) to   (THR401)  THE STRUCTURE OF MAP2K7 IN COMPLEX WITH 5Z-7-OXOZEAENOL  |   PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3x2v:A   (VAL219) to   (ALA298)  MICHAELIS-LIKE COMPLEX OF CAMP-DEPENDENT PROTEIN KINASE CATALYTIC SUBUNIT  |   MICHAELIS-LIKE COMPLEX, PROTEIN-SUBSTRATE, PKAC-ATPMG2 TERNARY, SER/THR KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-PEPTIDE COMPLEX 
3x2w:A   (VAL219) to   (ALA298)  MICHAELIS COMPLEX OF CAMP-DEPENDENT PROTEIN KINASE CATALYTIC SUBUNIT  |   MICHAELIS COMPLEX, PROTEIN-SUBSTRATE, PKAC-ATPMG2 TERNARY, SER/THR KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-PEPTIDE COMPLEX 
2jdt:A   (VAL219) to   (ALA298)  STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH ISOQUINOLINE-5- SULFONIC ACID (2-(2-(4-CHLOROBENZYLOXY) ETHYLAMINO)ETHYL) AMIDE  |   CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION 
3zh8:A   (VAL425) to   (ARG514)  A NOVEL SMALL MOLECULE APKC INHIBITOR  |   TRANSFERASE, AGC KINASES, CELL POLARITY, CELL MIGRATION 
3zh8:B   (SER424) to   (ARG514)  A NOVEL SMALL MOLECULE APKC INHIBITOR  |   TRANSFERASE, AGC KINASES, CELL POLARITY, CELL MIGRATION 
4neu:A   (GLU207) to   (LEU293)  X-RAY STRUCTURE OF RECEPTOR INTERACTING PROTEIN 1 (RIP1)KINASE DOMAIN WITH A 1-AMINOISOQUINOLINE INHIBITOR  |   KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE 
5bx6:A   (ALA218) to   (ALA298)  PKA IN COMPLEX WITH A HALOGENATED PHTHALAZINONE FRAGMENT COMPOUND.  |   INHIBITOR, PROTEIN KINASE, STRUCTURE-GUIDED, FRAGMENT-BASED, TRANSFERASE 
4nif:A   (PRO583) to   (GLN677)  HETERODIMERIC STRUCTURE OF ERK2 AND RSK1  |   KINASE DOMAIN, SIGNALING, SUBSTRATE KINASE BINDING, TRANSFERASE 
4nif:D   (PRO583) to   (GLN677)  HETERODIMERIC STRUCTURE OF ERK2 AND RSK1  |   KINASE DOMAIN, SIGNALING, SUBSTRATE KINASE BINDING, TRANSFERASE 
1wvw:A   (GLY195) to   (LYS276)  CRYSTAL STRUCTURES OF KINASE DOMAIN OF DAP KINASE IN COMPLEX WITH SMALL MOLECULAR INHIBITORS  |   PROTEIN KINASE, APOPTOSIS, TRANSFERASE 
1wvx:A   (GLU197) to   (LYS276)  CRYSTAL STRUCTURES OF KINASE DOMAIN OF DAP KINASE IN COMPLEX WITH SMALL MOLECULAR INHIBITORS  |   PROTEIN KINASE, APOPTOSIS, STAUROSPORINE, TRANSFERASE 
2ydi:A   (PRO188) to   (LYS267)  DISCOVERY OF CHECKPOINT KINASE INHIBITOR AZD7762 BY STRUCTURE BASED DESIGN AND OPTIMIZATION OF THIOPHENE CARBOXAMIDE UREAS  |   TRANSFERASE, CHK 
2ydj:A   (PRO188) to   (LYS267)  DISCOVERY OF CHECKPOINT KINASE INHIBITOR AZD7762 BY STRUCTURE BASED DESIGN AND OPTIMIZATION OF THIOPHENE CARBOXAMIDE UREAS  |   TRANSFERASE 
2ydj:B   (PRO188) to   (LYS267)  DISCOVERY OF CHECKPOINT KINASE INHIBITOR AZD7762 BY STRUCTURE BASED DESIGN AND OPTIMIZATION OF THIOPHENE CARBOXAMIDE UREAS  |   TRANSFERASE 
2ydk:A   (PRO188) to   (LYS267)  DISCOVERY OF CHECKPOINT KINASE INHIBITOR AZD7762 BY STRUCTURE BASED DESIGN AND OPTIMIZATION OF THIOPHENE CARBOXAMIDE UREAS  |   TRANSFERASE 
4nts:B   (ALA218) to   (ALA298)  APO STRUCTURE OF THE CATALYTIC SUBUNIT OF CAMP-DEPENDENT PROTEIN KINASE  |   PROTEIN KINASE FOLD, PHOSPHORYL TRANSFERASE, KINASE, REGULATORY SUBUNIT OF PKA, PKI, PHOSPHORYLATION, TRANSFERASE 
3zxt:A   (GLU197) to   (LYS276)  DIMERIC STRUCTURE OF DAPK-1 CATALYTIC DOMAIN IN COMPLEX WITH AMPPCP-MG  |   APOPTOSIS, TRANSFERASE, ATP BINDING 
3zxt:C   (GLU197) to   (LYS276)  DIMERIC STRUCTURE OF DAPK-1 CATALYTIC DOMAIN IN COMPLEX WITH AMPPCP-MG  |   APOPTOSIS, TRANSFERASE, ATP BINDING 
3zxt:D   (GLU197) to   (LYS276)  DIMERIC STRUCTURE OF DAPK-1 CATALYTIC DOMAIN IN COMPLEX WITH AMPPCP-MG  |   APOPTOSIS, TRANSFERASE, ATP BINDING 
2ym5:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   TRANSFERASE, DNA REPAIR 
2ym7:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   TRANSFERASE, DNA REPAIR, CELL CYCLE 
2ym8:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   TRANSFERASE, DNA REPAIR, SERINE/THREONINE KINASE 
3jvs:A   (PRO188) to   (LYS267)  CHARACTERIZATION OF THE CHK1 ALLOSTERIC INHIBITOR BINDING SITE  |   PROTEIN KINASE, ATP-BINDING, CELL CYCLE, CYTOPLASM, DNA DAMAGE, DNA REPAIR, ISOPEPTIDE BOND, KINASE, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, UBL CONJUGATION 
5cek:A   (GLY262) to   (LEU342)  PSEUDOKINASE DOMAIN OF HUMAN TRIBBLES HOMOLOG 1  |   KINASE, TRANSFERASE 
2z1q:B   (LEU445) to   (LEU532)  CRYSTAL STRUCTURE OF ACYL COA DEHYDROGENASE  |   ACYL-COA DEHYDROGENASE, FAD, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, OXIDOREDUCTASE 
3ka0:A   (LYS239) to   (GLN327)  MK2 COMPLEX WITH INHIBITOR 6-(5-(2-AMINOPYRIMIDIN-4-YLAMINO)-2- HYDROXYPHENYL)-N-METHYLBENZO[B]THIOPHENE-2-CARBOXAMIDE  |   MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
2zv2:A   (ALA371) to   (ARG449)  CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE KINASE 2, BETA, CAMKK2 KINASE DOMAIN IN COMPLEX WITH STO-609  |   CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE KINASE 2, BETA, STO-609, CAMKK2, E.C.2.7.11.17, PHOSPHORYLATION, AMPKK, METABOLISM, ATP- BINDING, KINASE, CALMODULIN-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ae9:B   (VAL219) to   (ALA298)  STRUCTURE AND FUNCTION OF THE HUMAN SPERM-SPECIFIC ISOFORM OF PROTEIN KINASE A (PKA) CATALYTIC SUBUNIT C ALPHA 2  |   TRANSFERASE 
1ydt:E   (VAL219) to   (ALA298)  STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE, ALPHA-CATALYTIC SUBUNIT IN COMPLEX WITH H89 PROTEIN KINASE INHIBITOR N-[2- (4-BROMOCINNAMYLAMINO)ETHYL]-5-ISOQUINOLINE  |   COMPLEX (PHOSPHOTRANSFERASE/INHIBITOR), TRANSFERASE, CAMP, PHOSPHORYLATION, ISOQUINOLINE SULFONAMIDE, SERINE/THREONINE- PROTEIN KINASE, ATP-BINDING 
3ku2:A   (ASP228) to   (LYS313)  CRYSTAL STRUCTURE OF INACTIVATED FORM OF CDPK1 FROM TOXOPLASMA GONDII, TGME49.101440  |   CDPKS, TOXOPLASMA, PROTIST, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE 
3a8w:B   (VAL425) to   (ARG514)  CRYSTAL STRUCTURE OF PKCIOTA KINASE DOMAIN  |   PROTEIN KINASE C IOTA, KINASE DOMAIN, ATP COMPLEX, TRANSFERASE 
5dhj:A   (ARG221) to   (GLN291)  PIM1 IN COMPLEX WITH CPD4 (3-METHYL-5-(PYRIDIN-3-YL)-1H-PYRAZOLO[3,4- C]PYRIDINE)  |   PIM-1, KINASE, ATP-COMPETITIVE, STRUCTURE-BASED DRUG DESIGN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3agl:A   (ALA218) to   (ALA298)  COMPLEX OF PKA WITH THE BISUBSTRATE PROTEIN KINASE INHIBITOR ARC-1039  |   PKA, PROTEIN KINASE A, BISUBSTRATE INHIBITOR, ARC-1039, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4pl5:C   (THR754) to   (PHE832)  CRYSTAL STRUCTURE OF MURINE IRE1 IN COMPLEX WITH OICR573 INHIBITOR  |   SCHIFF BASE, HYDROXY ARYL ALDEHYDES (HAA), INHIBITOR COMPLEX, UNFOLDED PROTEIN RESPONSE, ENDORIBONUCLEASE 
5dls:A   (GLU187) to   (LYS267)  IDENTIFICATION OF NOVEL, IN VIVO ACTIVE CHK1 INHIBITORS UTILIZING STRUCTURE GUIDED DRUG DESIGN  |   CHK1, V158411, FRAGMENT, KINASE, TRANSFERASE 
3lau:A   (ASP307) to   (ASN386)  CRYSTAL STRUCTURE OF AURORA2 KINASE IN COMPLEX WITH A GSK3BETA INHIBITOR  |   KINASE INHIBITOR COMPLEX, ATP-BINDING, CELL CYCLE, CYTOPLASM, CYTOSKELETON, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, UBL CONJUGATION 
5dr2:A   (LYS309) to   (ASN386)  AURORA A KINASE IN COMPLEX WITH AA30 AND ATP IN SPACE GROUP P6122  |   AURORA A KINASE, MITOTIC KINASE, PPI, TRANSFERASE 
3ama:A   (ALA218) to   (ALA298)  PROTEIN KINASE A SIXFOLD MUTANT MODEL OF AURORA B WITH INHIBITOR JNJ- 7706621  |   PKA, PROTEIN KINASE A, SURROGATE, JNJ-7706621, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3lij:A   (ASP238) to   (SER327)  CRYSTAL STRUCTURE OF FULL LENGTH CPCDPK3 (CGD5_820) IN COMPLEX WITH CA2+ AND AMPPNP  |   TRANSFERASE, CALCIUM DEPENDENT PROTEIN KINASE, EF HAND, ATP- BINDING, CALCIUM, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC 
4apc:B   (ASN181) to   (LEU266)  CRYSTAL STRUCTURE OF HUMAN NIMA-RELATED KINASE 1 (NEK1)  |   TRANSFERASE 
5dt0:A   (LYS309) to   (ASN386)  AURORA A KINASE IN COMPLEX WITH JNJ-7706621 IN SPACE GROUP P6122  |   AURORA A KINASE, MITOTIC KINASE, PPI, TRANSFERASE 
1zlt:A   (GLU187) to   (LYS267)  CRYSTAL STRUCTURE OF CHK1 COMPLEXED WITH A HYMENALDISINE ANALOG  |   KINASE, TRANSFERASE 
1zmu:A   (GLU230) to   (VAL306)  CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK2/PAR-1: WILD TYPE  |   SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
1zmv:A   (GLU230) to   (VAL306)  CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK2/PAR-1: K82R MUTANT  |   SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE 
4au8:A   (SER182) to   (PHE289)  CRYSTAL STRUCTURE OF COMPOUND 4A IN COMPLEX WITH CDK5, SHOWING AN UNUSUAL BINDING MODE TO THE HINGE REGION VIA A WATER MOLECULE  |   TRANSFERASE, CDK2, ALZHEIMER DISEASE 
4au8:B   (SER180) to   (PHE289)  CRYSTAL STRUCTURE OF COMPOUND 4A IN COMPLEX WITH CDK5, SHOWING AN UNUSUAL BINDING MODE TO THE HINGE REGION VIA A WATER MOLECULE  |   TRANSFERASE, CDK2, ALZHEIMER DISEASE 
1zrz:A   (PHE423) to   (ARG514)  CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF ATYPICAL PROTEIN KINASE C-IOTA  |   PROTEIN-INHIBITOR COMPLEX, STRUCTURAL GENOMICS, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, TRANSFERASE 
3aqv:A   (GLY192) to   (GLN270)  HUMAN AMP-ACTIVATED PROTEIN KINASE ALPHA 2 SUBUNIT KINASE DOMAIN (T172D) COMPLEXED WITH COMPOUND C  |   STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, TRANSFERASE, SIGNALING PROTEIN, SERINE/THREONINE PROTEIN KINASE, PHOSPHORYLATION, ATP-BINDING, NUCLEOTIDE-BINDING, CHOLESTEROL BIOSYNTHESIS, FATTY ACID BIOSYNTHESIS, LIPID SYNTHESIS, GLUCOSE METABOLISM, MAGNESIUM, METAL-BINDING, SERINE/THREONINE- PROTEIN KINASE, STEROID BIOSYNTHESIS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
1zys:A   (PRO188) to   (LYS267)  CO-CRYSTAL STRUCTURE OF CHECKPOINT KINASE CHK1 WITH A PYRROLO-PYRIDINE INHIBITOR  |   CHK1; CRYSTAL STRUCTURE, SIGNALING PROTEIN, TRANSFERASE 
4b0g:A   (ASP311) to   (ASN386)  COMPLEX OF AURORA-A BOUND TO AN IMIDAZOPYRIDINE-BASED INHIBITOR  |   TRANSFERASE, MITOSIS 
4b9d:B   (LYS183) to   (LEU266)  CRYSTAL STRUCTURE OF HUMAN NIMA-RELATED KINASE 1 (NEK1) WITH INHIBITOR.  |   TRANSFERASE, INHIBITOR 
3ma6:A   (ASP211) to   (THR295)  CRYSTAL STRUCTURE OF KINASE DOMAIN OF TGCDPK1 IN PRESENCE OF 3BRB-PP1  |   CDPK, PARASITOLOGY, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC 
3ma6:B   (ASP215) to   (THR295)  CRYSTAL STRUCTURE OF KINASE DOMAIN OF TGCDPK1 IN PRESENCE OF 3BRB-PP1  |   CDPK, PARASITOLOGY, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC 
2ac3:A   (SER266) to   (GLN369)  STRUCTURE OF HUMAN MNK2 KINASE DOMAIN  |   DFD MOTIF, TRANSFERASE 
2ac5:A   (SER266) to   (GLY370)  STRUCTURE OF HUMAN MNK2 KINASE DOMAIN MUTANT D228G  |   DFG MOTIF, TRANSFERASE 
5eol:A   (ARG221) to   (GLN291)  CRYSTAL STRUCTURE OF HUMAN PIM-1 KINASE IN COMPLEX WITH A MACROCYCLIC QUINOXALINE-PYRROLODIHYDROPIPERIDINONE INHIBITOR  |   TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5ew9:A   (ASP307) to   (ASN386)  CRYSTAL STRUCTURE OF AURORA A KINASE DOMAIN BOUND TO MK-5108  |   TRANSFERASE, PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3bqr:A   (GLU197) to   (ALA277)  CRYSTAL STRUCTURE OF HUMAN DEATH ASSOCIATED PROTEIN KINASE 3 (DAPK3) IN COMPLEX WITH AN IMIDAZO-PYRIDAZINE LIGAND  |   DEATH ASSOCIATED KINASE, DAPK3, ZIP KINASE, ZIPK, DAP KINASE 3, DAP LIKE KINASE, DLK, STRUCTURAL GENOMICS CONSORTIUM, SGC, APOPTOSIS, ATP-BINDING, CHROMATIN REGULATOR, NUCLEOTIDE-BINDING, NUCLEUS, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
4qye:A   (PRO188) to   (LYS267)  CHK1 KINASE DOMAIN IN COMPLEX WITH DIARYLPYRAZINE COMPOUND 1  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4qyf:A   (PRO188) to   (LYS267)  CHK1 KINASE DOMAIN IN COMPLEX WITH AMINOPYRAZINE COMPOUND 13  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5f4n:A   (GLU187) to   (LYS267)  MULTI-PARAMETER LEAD OPTIMIZATION TO GIVE AN ORAL CHK1 INHIBITOR CLINICAL CANDIDATE: (R)-5-((4-((MORPHOLIN-2-YLMETHYL)AMINO)-5- (TRIFLUOROMETHYL)PYRIDIN-2-YL)AMINO)PYRAZINE-2-CARBONITRILE (CCT245737)  |   INHIBITOR DNA-DAMAGE CHK1-POTENCY HERG-ACTIVITY, TRANSFERASE 
4qyg:A   (PRO188) to   (LYS267)  CHK1 KINASE DOMAIN IN COMPLEX WITH DIAZACARBAZOLE COMPOUND 14  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4qyg:B   (PRO188) to   (LYS267)  CHK1 KINASE DOMAIN IN COMPLEX WITH DIAZACARBAZOLE COMPOUND 14  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4qyh:A   (PRO188) to   (LYS267)  CHK1 KINASE DOMAIN IN COMPLEX WITH DIAZACARBAZOLE GNE-783  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4qyh:B   (PRO188) to   (LYS267)  CHK1 KINASE DOMAIN IN COMPLEX WITH DIAZACARBAZOLE GNE-783  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3mwu:A   (LYS254) to   (SER336)  ACTIVATED CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM CRYPTOSPORIDIUM PARVUM (CPCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR RM-1-95  |   SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, BUMPED KINASE INHIBITOR, BKI, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ncz:D   (GLU258) to   (LYS339)  X-RAY CO-STRUCTURE OF RHO-ASSOCIATED PROTEIN KINASE (ROCK1) WITH A POTENT 2H-ISOQUINOLIN-1-ONE INHIBITOR  |   RHO KINASE, DIMER, PHOSPHORYLATION, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4c34:A   (ALA218) to   (ALA298)  PKA-S6K1 CHIMERA WITH STAUROSPORINE BOUND  |   TRANSFERASE-INHIBITOR COMPLEX 
4c35:A   (ALA218) to   (ALA298)  PKA-S6K1 CHIMERA WITH COMPOUND 1 (NU1085) BOUND  |   TRANSFERASE-INHIBITOR COMPLEX, CHIMERA, S6K1 
4c36:A   (ALA218) to   (ALA298)  PKA-S6K1 CHIMERA WITH COMPOUND 15E (CCT147581) BOUND  |   TRANSFERASE-INHIBITOR COMPLEX, CHIMERA, S6K1 
4red:A   (GLY194) to   (GLN272)  CRYSTAL STRUCTURE OF HUMAN AMPK ALPHA1 KD-AID WITH K43A MUTATION  |   KINASE DOMAIN FOLD, PHOSPHORYLATE NUMEROUS CELLULAR TARGETS, UPREGULATE ATP-GENERATING PATHWAYS UPON ACTIVATION, AMPK BETA AND GAMMA SUBUNITS, TRANSFERASE 
4red:B   (GLY194) to   (GLN272)  CRYSTAL STRUCTURE OF HUMAN AMPK ALPHA1 KD-AID WITH K43A MUTATION  |   KINASE DOMAIN FOLD, PHOSPHORYLATE NUMEROUS CELLULAR TARGETS, UPREGULATE ATP-GENERATING PATHWAYS UPON ACTIVATION, AMPK BETA AND GAMMA SUBUNITS, TRANSFERASE 
4rer:A   (GLU196) to   (GLN272)  CRYSTAL STRUCTURE OF THE PHOSPHORYLATED HUMAN ALPHA1 BETA2 GAMMA1 HOLO-AMPK COMPLEX BOUND TO AMP AND CYCLODEXTRIN  |   HUMAN ALPHA1 BETA2 GAMMA1 HOLO-AMPK COMPLEX, SERINE/THREONINE PROTEIN KINASE, AXIN, CAMKKBETA, LKB1, GLYCOGEN, PHOSPHORYLATION, TRANSFERASE 
4c4e:A   (LYS714) to   (GLN792)  STRUCTURE-BASED DESIGN OF ORALLY BIOAVAILABLE PYRROLOPYRIDINE INHIBITORS OF THE MITOTIC KINASE MPS1  |   TRANSFERASE, MPS1, TTK, PROTEIN KINASE, MITOSIS, STRUCTURE-BASED DESIGN 
3nrm:A   (LYS309) to   (ASN386)  IMIDAZO[1,2-A]PYRAZINE-BASED AURORA KINASE INHIBITORS  |   KINASE, CELL CYCLE, INHIBITOR, TRANSFERASE 
4ceg:A   (LYS309) to   (ASN386)  CRYSTAL STRUCTURE OF AURORA A 122-403 C290A, C393A BOUND TO ADP  |   TRANSFERASE, PROTEIN KINASE, MITOSIS 
3nup:A   (PRO199) to   (PHE300)  CDK6 (MONOMERIC) IN COMPLEX WITH INHIBITOR  |   KINASE, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
3cqu:A   (VAL330) to   (ALA409)  CRYSTAL STRUCTURE OF AKT-1 COMPLEXED WITH SUBSTRATE PEPTIDE AND INHIBITOR  |   KINASE, APOPTOSIS, ATP-BINDING, CARBOHYDRATE METABOLISM, CYTOPLASM, GLUCOSE METABOLISM, GLYCOGEN BIOSYNTHESIS, GLYCOGEN METABOLISM, MEMBRANE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, SUGAR TRANSPORT, TRANSFERASE, TRANSLATION REGULATION, TRANSPORT, ALTERNATIVE SPLICING, WNT SIGNALING PATHWAY 
4rpv:A   (ARG221) to   (GLN291)  CO-CRYSTAL STRUCTURE OF PIM1 WITH COMPOUND 3  |   PIM1, KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3nyn:B   (PRO366) to   (LEU451)  CRYSTAL STRUCTURE OF G PROTEIN-COUPLED RECEPTOR KINASE 6 IN COMPLEX WITH SANGIVAMYCIN  |   KINASE, GRK, RGS HOMOLOGY DOMAIN, G PROTEIN-COUPLED RECEPTOR KINASE, TRANSFERASE 
3nyo:A   (PRO366) to   (LYS449)  CRYSTAL STRUCTURE OF G PROTEIN-COUPLED RECEPTOR KINASE 6 IN COMPLEX WITH AMP  |   KINASE, GRK, RGS HOMOLOGY DOMAIN, G PROTEIN-COUPLED RECEPTOR KINASE, TRANSFERASE 
3o0g:A   (SER180) to   (PHE289)  CRYSTAL STRUCTURE OF CDK5:P25 IN COMPLEX WITH AN ATP ANALOGUE  |   KINASE, KINASE ACTIVATOR COMPLEX, KINASE INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE ACTIVATOR COMPLEX 
4rvk:A   (PRO188) to   (LYS267)  CHK1 KINASE DOMAIN WITH DIAZACARBAZOLE COMPOUND 8: N-[3-(6-CYANO-9H- PYRROLO[2,3-B:5,4-C']DIPYRIDIN-3-YL)PHENYL]ACETAMIDE  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4rvm:A   (PRO188) to   (LYS267)  CHK1 KINASE DOMAIN WITH DIAZACARBAZOLE COMPOUND 19  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3o50:A   (ASP307) to   (ASN386)  CRYSTAL STRUCTURE OF BENZAMIDE 9 BOUND TO AURORAA  |   AURORAA, KINASE DOMAIN, TRANSFERASE 
3o50:B   (ASP307) to   (ALA385)  CRYSTAL STRUCTURE OF BENZAMIDE 9 BOUND TO AURORAA  |   AURORAA, KINASE DOMAIN, TRANSFERASE 
3d0e:A   (VAL331) to   (LEU410)  CRYSTAL STRUCTURE OF HUMAN AKT2 IN COMPLEX WITH GSK690693  |   HUMAN, AKT2, INHIBITOR, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSFERASE INHIBITOR 
3d0e:B   (GLY328) to   (LEU410)  CRYSTAL STRUCTURE OF HUMAN AKT2 IN COMPLEX WITH GSK690693  |   HUMAN, AKT2, INHIBITOR, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSFERASE INHIBITOR 
3d15:A   (LYS322) to   (ASN399)  CRYSTAL STRUCTURE OF MOUSE AURORA A (ASN186->GLY, LYS240->ARG, MET302- >LEU) IN COMPLEX WITH 1-(3-CHLORO-PHENYL)-3-{5-[2-(THIENO[3,2- D]PYRIMIDIN-4-YLAMINO)- ETHYL]-THIAZOL-2-YL}-UREA [SNS-314]  |   AURORA A, SMALL-MOLECULE INHIBITOR, KINASE, TRANSFERASE 
3ocb:B   (VAL330) to   (ALA409)  AKT1 KINASE DOMAIN WITH PYRROLOPYRIMIDINE INHIBITOR  |   SERINE-THREONINE KINASE, TRANSFERASE 
3dae:A   (PRO231) to   (VAL308)  CRYSTAL STRUCTURE OF PHOSPHORYLATED SNF1 KINASE DOMAIN  |   KINASE, AMPK, SNF1, ATP-BINDING, CARBOHYDRATE METABOLISM, MEMBRANE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3daj:A   (ASP307) to   (ASN386)  CRYSTAL STRUCTURE OF AURORA A COMPLEXED WITH AN INHIBITOR DISCOVERED THROUGH SITE-DIRECTED DYNAMIC TETHERING  |   PROTEIN-SMALL MOLECULE INHIBITOR COMPLEX, KINASE, TRANSFERASE 
3dak:D   (ASP205) to   (ALA294)  CRYSTAL STRUCTURE OF DOMAIN-SWAPPED OSR1 KINASE DOMAIN  |   SERINE/THREONINE PROTEIN KINASE, STE20, DOMAIN-SWAPPING, ATP-BINDING, KINASE, MAGNESIUM, METAL-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE 
4czt:D   (ASP209) to   (LYS288)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF SNRK3.23 AT1G30270  |   TRANSFERASE, POTASSIUM TRANSPORT, SNRK3 
4czu:C   (GLY210) to   (LYS288)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF SNRK3.23 AT1G30270 T190D MUTANT  |   TRANSFERASE, POTASSIUM TRANSPORT, SNRK3 
4czu:D   (ASP209) to   (LYS288)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF SNRK3.23 AT1G30270 T190D MUTANT  |   TRANSFERASE, POTASSIUM TRANSPORT, SNRK3 
4d28:A   (SER189) to   (LYS266)  CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF SNRK3.11 AT5G35410  |   TRANSFERASE, SALT STRESS, SODIUM TRANSPORT, ION HOMEOSTASIS 
3os3:A   (SER241) to   (GLU367)  MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1 (MEK1) IN COMPLEX WITH CH4858061 AND MGATP  |   KINASE, KINASE INHIBITOR, ALLOSTERIC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ot3:A   (PRO188) to   (LYS267)  X-RAY CRYSTAL STRUCTURE OF COMPOUND 22K BOUND TO HUMAN CHK1 KINASE DOMAIN  |   KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ot8:A   (PRO188) to   (LYS267)  X-RAY CRYSTAL STRUCTURE OF COMPOUND 17R BOUND TO HUMAN CHK1 KINASE DOMAIN  |   KINASE, PHOSPHATASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ow3:A   (ALA218) to   (ALA298)  DISCOVERY OF DIHYDROTHIENO- AND DIHYDROFUROPYRIMIDINES AS POTENT PAN AKT INHIBITORS  |   CYCLIC-AMP DEPENDENT PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ow4:A   (GLY327) to   (ALA409)  DISCOVERY OF DIHYDROTHIENO- AND DIHYDROFUROPYRIMIDINES AS POTENT PAN AKT INHIBITORS  |   SERINE-THREONINE KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4dee:A   (LYS309) to   (ASN386)  AURORA A IN COMPLEX WITH ADP  |   PROTEIN KINASE, AURORA A, DFG-IN, TRANSFERASE 
4dfx:E   (ALA218) to   (ALA298)  CRYSTAL STRUCTURE OF MYRISTOYLATED K7C CATALYTIC SUBUNIT OF CAMP- DEPENDENT PROTEIN KINASE IN COMPLEX WITH SP20 AND AMP-PNP  |   PROTEIN KINASE, MYRISTOYLATED, PHOSPHOTRANSFERASE ONTO SER/THR, MG, PKI, PKA REGULATORY SUBUNITS, PHOSPHORYLATED ON S139, T197, S338, MYRISTOYLATED ON G1, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4dg0:E   (VAL219) to   (ALA298)  CRYSTAL STRUCTURE OF MYRISTOYLATED WT CATALYTIC SUBUNIT OF CAMP- DEPENDENT PROTEIN KINASE IN COMPLEX WITH SP20 AND AMP-PNP  |   PROTEIN KINASE, MYRISTOYLATED, PHOSPHOTRANSFERASE OF SER/THR, MG, PKI, PKA REGULATORY SUBUNITS, PHOSPHORYLATED ON S139, T197, S338, MYRISTOYLATED ON G1, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4dg3:E   (VAL219) to   (ALA298)  CRYSTAL STRUCTURE OF R336A MUTANT OF CAMP-DEPENDENT PROTEIN KINASE WITH UNPHOSPHORYLATED TURN MOTIF.  |   PROTEIN KINASE, PHOSPHOTRANSFERASE, SERINE/THREONINE PROTEIN KINASE, REGULATORY SUBUNIT, PKI, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4dh1:A   (VAL219) to   (ALA298)  LOW TEMPERATURE X-RAY STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A CATALYTIC SUBUNIT WITH LOW MG2+, ATP AND IP20  |   PROTEIN KINASE, PHOSPHORYLATION, PEPTIDIC INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4dh7:A   (VAL219) to   (ALA298)  LOW TEMPERATURE X-RAY STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A CATALYTIC SUBUNIT WITH HIGH MG2+, AMP-PNP AND IP20'  |   PROTEIN KINASE, PHOSPHOTRANFER, PEPTIDIC INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4dh8:A   (VAL219) to   (ALA298)  ROOM TEMPERATURE X-RAY STRUCTURE OF CAMP DEPENDENT PROTEIN KINASE A CATALYTIC SUBUNIT WITH HIGH MG2+, AMP-PNP AND IP20  |   PROTEIN KINASE, PHOSPHOTRANSFER, PEPTIDIC INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
5hlw:A  (THR1261) to  (PHE1344)  CRYSTAL STRUCTURE OF C-MET MUTANT Y1230H IN COMPLEX WITH COMPOUND 14  |   TRANSFERASE, TRANSFERASE INHIBITOR 
5hoa:A  (THR1262) to  (PHE1344)  CRYSTAL STRUCTURE OF C-MET L1195V IN COMPLEX WITH SAR125844  |   TRANSFERASE, INHIBITOR 
4ual:A   (GLY259) to   (GLU343)  MRCK BETA IN COMPLEX WITH BDP00005290  |   MYOTONIC DYSTROPHY KINASE-RELATED CDC42-BINDING KINASE, METASTASIS, CELL INVASION, TRANSFERASE 
3pa3:A   (PRO188) to   (LYS267)  X-RAY CRYSTAL STRUCTURE OF COMPOUND 70 BOUND TO HUMAN CHK1 KINASE DOMAIN  |   KINASE, PHOSPHATASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3pa4:A   (PRO188) to   (LYS267)  X-RAY CRYSTAL STRUCTURE OF COMPOUND 2A BOUND TO HUMAN CHK1 KINASE DOMAIN  |   KINASE, PHOSPHATASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3pa5:A   (PRO188) to   (LYS267)  X-RAY CRYSTAL STRUCTURE OF COMPOUND 1 BOUND TO HUMAN CHK1 KINASE DOMAIN  |   KINASE, PHOSPHATASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3pfq:A   (ASP523) to   (ARG601)  CRYSTAL STRUCTURE AND ALLOSTERIC ACTIVATION OF PROTEIN KINASE C BETA II  |   KINASE, PHOSPHORYLATION, TRANSFERASE 
3pvb:A   (VAL219) to   (ASP301)  CRYSTAL STRUCTURE OF (73-244)RIA:C HOLOENZYME OF CAMP-DEPENDENT PROTEIN KINASE  |   KINASE, RIA HOLOENZYME, TETRAMERIC PROTEIN KINASE A, TRANSFERASE 
4ejn:A   (ALA329) to   (ALA409)  CRYSTAL STRUCTURE OF AUTOINHIBITED FORM OF AKT1 IN COMPLEX WITH N-(4- (5-(3-ACETAMIDOPHENYL)-2-(2-AMINOPYRIDIN-3-YL)-3H-IMIDAZO[4,5- B]PYRIDIN-3-YL)BENZYL)-3-FLUOROBENZAMIDE  |   AKT1, AUTOINHIBITION, ALLOSTERIC INHIBITOR, KINASE INHIBITOR, HYDROPHOBIC COLLAPASE, KINASE, ATPASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ekk:A   (VAL330) to   (ALA409)  AKT1 WITH AMP-PNP  |   PHOSPHOTRANSFERASE, TRANSFERASE 
4ekk:B   (VAL330) to   (ALA409)  AKT1 WITH AMP-PNP  |   PHOSPHOTRANSFERASE, TRANSFERASE 
4ekl:A   (ARG328) to   (ALA409)  AKT1 WITH GDC0068  |   PHOSPHOTRANSFERASE, TRANSFERASE 
4enx:A   (ARG221) to   (GLN291)  CRYSTAL STRUCTURE OF PIM-1 KINASE IN COMPLEX WITH INHIBITOR (2E,5Z)-2- (2-CHLOROPHENYLIMINO)-5-(4-HYDROXY-3-NITROBENZYLIDENE)THIAZOLIDIN-4- ONE  |   PIM-1 KINASE, TRANSFERASE-INHIBITOR COMPLEX 
5iu2:A   (SER305) to   (ASN389)  DISCOVERY OF IMIDAZOQUINOLINES AS A NOVEL CLASS OF POTENT, SELECTIVE AND IN VIVO EFFICACIOUS COT KINASE INHIBITORS  |   COT, TPL-2, MAP3K8, KINASE, INHIBITOR, COMPLEX, TRANSFERASE 
3qal:E   (VAL219) to   (ALA298)  CRYSTAL STRUCTURE OF ARG280ALA MUTANT OF CATALYTIC SUBUNIT OF CAMP- DEPENDENT PROTEIN KINASE  |   PROTEIN KINASE, GLU208/ARG280 PAIR, PKA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qbn:A   (GLU308) to   (ALA385)  STRUCTURE OF HUMAN AURORA A IN COMPLEX WITH A DIAMINOPYRIMIDINE  |   KINASE DOMAIN, DIAMINOPYRIMIDINE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5j5x:A   (VAL219) to   (ALA298)  COMPLEX OF PKA WITH THE BISUBSTRATE PROTEIN KINASE INHIBITOR ARC-1416  |   PROTEIN KINASE, INHIBITOR, BISUBSTRATE, OLIGOARGININE, PKA, TRANSFERASE 
3qkk:A   (GLY327) to   (ALA409)  SPIROCHROMANE AKT INHIBITORS  |   KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qkl:A   (GLY327) to   (ALA409)  SPIROCHROMANE AKT INHIBITORS  |   KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3qkm:A   (VAL330) to   (ALA409)  SPIROCYCLIC SULFONAMIDES AS AKT INHIBITORS  |   KINASE DOMAIN, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5jn2:A   (ASP228) to   (THR312)  CRYSTAL STRUCTURE OF TGCDPK1 BOUND TO NVPACU106  |   KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, HYDROLASE 
4fsm:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fsq:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fsr:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fst:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fsw:A   (GLU187) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fsy:A   (GLU187) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fsz:A   (GLU187) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ft0:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ft3:A   (GLU187) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ft5:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ft7:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fta:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ftc:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ftj:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ftl:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ftm:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ftn:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fto:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ftq:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ftr:A   (GLU187) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ftt:A   (GLU187) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ftu:A   (GLU187) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
5kbq:B   (GLY442) to   (ALA524)  PAK1 IN COMPLEX WITH BIS-ANILINO PYRIMIDINE INHIBITOR  |   SERINE/THREONINE-PROTEIN KINASE PAK1, KINASE, TRANSFERASE 
5kcv:A   (ALA329) to   (ALA409)  CRYSTAL STRUCTURE OF ALLOSTERIC INHIBITOR, ARQ 092, IN COMPLEX WITH AUTOINHIBITED FORM OF AKT1  |   AKT, ALLOSTERIC INHIBITOR, KINASE INHIBITOR, TRANSFERASE-INHIBITOR COMPLEX 
4gh2:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
2bro:A   (GLU187) to   (LYS267)  STRUCTURE-BASED DESIGN OF NOVEL CHK1 INHIBITORS: INSIGHTS INTO HYDROGEN BONDING AND PROTEIN-LIGAND AFFINITY  |   DRUG DESIGN, FURANOPYRIMIDINE, MOLECULAR RECOGNITION, ONCOLOGY, PYRROLOPYRIMIDINE, ATP-BINDING, CELL CYCLE, DNA DAMAGE, KINASE, NUCLEAR PROTEIN, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
2c1b:A   (ALA218) to   (ALA298)  STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE COMPLEXED WITH ( 4R,2S)-5'-(4-(4-CHLOROBENZYLOXY)PYRROLIDIN-2- YLMETHANESULFONYL)ISOQUINOLINE  |   TRANSFERASE/INHIBITOR, COMPLEX (TRANSFERASE/INHIBITOR), ATP-BINDING, CAMP, PHOSPHORYLATION, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, PROTEIN KINASE INHIBITOR 
2c3l:A   (PRO188) to   (LYS267)  IDENTIFICATION OF A BURIED POCKET FOR POTENT AND SELECTIVE INHIBITION OF CHK1: PREDICTION AND VERIFICATION  |   DRUG DESIGN, MOLECULAR MODELING, MOLECULAR RECOGNITION, ONCOLOGY, ATP-BINDING, CELL CYCLE, DNA DAMAGE, DNA REPAIR, KINASE, NUCLEAR PROTEIN, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, UBL CONJUGATION 
3g33:A   (ALA197) to   (LEU300)  CRYSTAL STRUCTURE OF CDK4/CYCLIN D3  |   SER/THR PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, ATP-BINDING, CELL DIVISION, DISEASE MUTATION, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, CYCLIN 
3g33:C   (ALA197) to   (LEU300)  CRYSTAL STRUCTURE OF CDK4/CYCLIN D3  |   SER/THR PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, ATP-BINDING, CELL DIVISION, DISEASE MUTATION, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, CYCLIN 
1phk:A   (GLY207) to   (GLN288)  TWO STRUCTURES OF THE CATALYTIC DOMAIN OF PHOSPHORYLASE, KINASE: AN ACTIVE PROTEIN KINASE COMPLEXED WITH NUCLEOTIDE, SUBSTRATE-ANALOGUE AND PRODUCT  |   GLYCOGEN METABOLISM, TRANSFERASE, SERINE/THREONINE-PROTEIN, KINASE, ATP-BINDING, CALMODULIN-BINDING 
3gbz:A   (SER197) to   (HIS303)  STRUCTURE OF THE CMGC CDK KINASE FROM GIARDIA LAMBLIA  |   SSGCID, KINASE, CMGC CDK, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE 
3t9i:A   (ARG221) to   (GLN291)  PIM1 COMPLEXED WITH A NOVEL 3,6-DISUBSTITUTED INDOLE AT 2.6 ANG RESOLUTION  |   KINASE, PHOSPHOTRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4y5q:A   (LYS254) to   (SER336)  ACTIVATED CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM CRYPTOSPORIDIUM PARVUM (CPCDPK1) IN COMPLEX WITH AMP  |   SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, BUMPED KINASE INHIBITOR, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP 
3tkh:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHK1 IN COMPLEX WITH INHIBITOR S01  |   CHK1, KINASE, CELL CHECKPOINT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4jdh:A   (GLY493) to   (ALA575)  CRYSTAL STRUCTURE OF SERINE/THREONINE-PROTEIN KINASE PAK 4 IN COMPLEX WITH PAKTIDE T PEPTIDE SUBSTRATE  |   TRANSFERASE-PEPTIDE COMPLEX, TRANSFERASE/PEPTIDE, SERINE/THREONINE- PROTEIN KINASE PAK4, ATP BINDING, PHOSPHORYLATION 
4yga:G   (CYS231) to   (THR312)  CDPK1, FROM TOXOPLASMA GONDII, BOUND TO INHIBITORY VHH-1B7  |   SERINE/THREONINE PROTEIN KINASE, VHH DOMAIN, INHIBITOR, METAL BINDING PROTEIN 
2e9v:B   (PRO188) to   (LYS267)  STRUCTURE OF H-CHK1 COMPLEXED WITH A859017  |   PROTEIN-INHIBITOR COMPLEX, TRANSFERASE 
2uw7:A   (ALA218) to   (ALA298)  STRUCTURE OF PKA-PKB CHIMERA COMPLEXED WITH  4-(4-CHLORO- PHENYL)-4-(4-(1H-PYRAZOL-4-YL)-PHENYL)-PIPERIDINE  |   TRANSFERASE/INHIBITOR, CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION, TRANSFERASE/INHIBITOR COMPLEX 
3udb:C   (GLY195) to   (LYS279)  CRYSTAL STRUCTURE OF SNRK2.6  |   SNRK2.6, KINASE, ABA SIGNALING PATHWAY, ABI1, TRANSFERASE 
2v5q:A   (GLU231) to   (SER307)  CRYSTAL STRUCTURE OF WILD-TYPE PLK-1 KINASE DOMAIN IN COMPLEX WITH A SELECTIVE DARPIN  |   DESIGN ANKYRIN REPEAT PROTEIN, TRANSFERASE COMPLEX, PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, KINASE, NUCLEUS, TRANSFERASE, ATP-BINDING, SERINE/THREONINE PROTEIN KINASE 
3uol:A   (ASP307) to   (ALA385)  AURORA A IN COMPLEX WITH SO2-162  |   PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3uol:B   (ASP307) to   (ALA385)  AURORA A IN COMPLEX WITH SO2-162  |   PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4loq:C   (ASN201) to   (ALA309)  STRUCTURAL BASIS OF AUTOACTIVATION OF P38 ALPHA INDUCED BY TAB1 (TETRAGONAL CRYSTAL FORM WITH BOUND SULPHATE)  |   STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, KINASE-REGULATORY PROTEIN COMPLEX, MAPK, AUTOACTIVATION, AUTOPHOSPHORYLATION, TRANSFERASE 
2wmv:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   SERINE/THREONINE-PROTEIN KINASE, POLYMORPHISM, PHOSPHOPROTEIN, UBL CONJUGATION, ISOPEPTIDE BOND, CHECKPOINT KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE KINASE, DNA DAMAGE, DNA REPAIR, ATP-BINDING, TRANSFERASE, CHK1, KINASE, NUCLEUS, CYTOPLASM, CELL CYCLE 
2wmx:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   SERINE/THREONINE-PROTEIN KINASE, POLYMORPHISM, PHOSPHOPROTEIN, UBL CONJUGATION, ISOPEPTIDE BOND, CHECKPOINT KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE KINASE, DNA DAMAGE, DNA REPAIR, ATP-BINDING, TRANSFERASE, CHK1, KINASE, NUCLEUS, CYTOPLASM, CELL CYCLE 
5a6n:A   (GLY195) to   (ILE278)  CRYSTAL STRUCTURE OF HUMAN DEATH ASSOCIATED PROTEIN KINASE 3 (DAPK3) IN COMPLEX WITH COMPOUND 2  |   TRANSFERASE, DAPK3, HUMAN DEATH ASSOCIATED PROTEIN KINASE 3, DAP-LIKE KINASE, DLK, ZIPPER-INTERACTING PROTEIN KINASE, ZIP-KINASE, 
5a6o:A   (GLY195) to   (ILE278)  CRYSTAL STRUCTURE OF THE APO FORM OF THE UNPHOSPHORYLATED HUMAN DEATH ASSOCIATED PROTEIN KINASE 3 (DAPK3)  |   TRANSFERASE, DAPK3, APO, DEATH-ASSOCIATED PROTEIN KINASE 3, ZIPPER- INTERACTING PROTEIN KINASE 
2xf0:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   TRANSFERASE,  DNA REPAIR, CELL CYCLE 
2xj2:A   (ARG221) to   (GLN291)  PROTEIN KINASE PIM-1 IN COMPLEX WITH SMALL MOLECULE INHIBITOR  |   TRANSFERASE, PHOSPHORYLATION, PROTEIN KINASE FOLD 
2y7j:B   (GLY211) to   (GLU292)  STRUCTURE OF HUMAN PHOSPHORYLASE KINASE, GAMMA 2  |   TRANSFERASE 
2y7j:C   (GLY211) to   (ARG293)  STRUCTURE OF HUMAN PHOSPHORYLASE KINASE, GAMMA 2  |   TRANSFERASE 
2yer:A   (PRO188) to   (LYS267)  SYNTHESIS AND EVALUATION OF TRIAZOLONES AS CHECKPOINT KINASE 1 INHIBITORS  |   TRANSFERASE 
2yex:A   (PRO188) to   (LYS267)  SYNTHESIS AND EVALUATION OF TRIAZOLONES AS CHECKPOINT KINASE 1 INHIBITORS  |   TRANSFERASE, CELL CYCLE, CHK 
2ym3:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   TRANSFERASE, DNA REPAIR 
2ym4:A   (GLU187) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   TRANSFERASE, DNA REPAIR, SERINE/THREONINE KINASE 
2ym6:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS  |   TRANSFERASE, DNA REPAIR, CELL CYCLE 
3jvr:A   (PRO188) to   (LYS267)  CHARACTERIZATION OF THE CHK1 ALLOSTERIC INHIBITOR BINDING SITE  |   PROTEIN KINASE, ATP-BINDING, CELL CYCLE, CYTOPLASM, DNA DAMAGE, DNA REPAIR, ISOPEPTIDE BOND, KINASE, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, UBL CONJUGATION 
3kc3:K   (TYR240) to   (GLN327)  MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE  |   MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE 
3a8x:A   (VAL425) to   (ARG514)  CRYSTAL STRUCTURE OF PKCIOTA KINASE DOMAIN  |   PROTEIN KINASE C IOTA, TRANSFERASE 
3ag9:A   (ALA218) to   (ALA298)  COMPLEX OF PKA WITH THE BISUBSTRATE PROTEIN KINASE INHIBITOR ARC-1012  |   PKA, PROTEIN KINASE A, BISUBSTRATE INHIBITOR, ARC-1012, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4q4a:B   (ILE186) to   (ASP335)  IMPROVED MODEL OF AMP-PNP BOUND TM287/288  |   ABC EXPORTER, MULTIDRUG TRANSPORT, ABC TRANSPORTER, MEMBRANE TRANSPORTER, HYDROLASE-TRANSPORT PROTEIN COMPLEX 
5es1:A   (PRO232) to   (ILE309)  CRYSTAL STRUCTURE OF MICROTUBULE AFFINITY-REGULATING KINASE 4 CATALYTIC DOMAIN IN COMPLEX WITH A PYRAZOLOPYRIMIDINE INHIBITOR  |   MARK4 PAR-1 SERINE/THREONINE PROTEIN KINASE11, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX 
4c37:A   (ALA218) to   (ALA298)  PKA-S6K1 CHIMERA WITH COMPOUND 21A (CCT196539) BOUND  |   TRANSFERASE-INHIBITOR COMPLEX, CHIMERA, S6K1 
3nlb:A   (PRO188) to   (LYS267)  NOVEL KINASE PROFILE HIGHLIGHTS THE TEMPORAL BASIS OF CONTEXT DEPENDENT CHECKPOINT PATHWAYS TO CELL DEATH  |   KINASE DOMAIN, CHECKPOINT KINASE, ATP BINDING, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4rvl:A   (PRO188) to   (LYS267)  CHK1 KINASE DOMAIN WITH DIAZACARBAZOLE COMPOUND 7: 3-(2- HYDROXYPHENYL)-9H-PYRROLO[2,3-B:5,4-C']DIPYRIDINE-6-CARBONITRILE  |   PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
3ody:X   (ASN201) to   (ALA309)  CRYSTAL STRUCTURE OF P38ALPHA Y323Q ACTIVE MUTANT  |   KINASE FOLD, KINASE, PHOSPJORYLATION, TRANSFERASE 
3dkc:A  (THR1261) to  (PHE1344)  STRUCTURE OF MET RECEPTOR TYROSINE KINASE IN COMPLEX WITH ATP  |   DRUG DISCOVERY, C-MET KINASE, FRAGMENT BASED, MEMBRANE, RECEPTOR, TRANSMEMBRANE, ONCOPROTEIN 
4uj2:A   (ALA218) to   (ALA298)  PROTEIN KINASE A IN COMPLEX WITH AN INHIBITOR  |   TRANSFERASE-INHIBITOR COMPLEX, PROTEIN KINASE A, 
3qf4:B   (ILE186) to   (LEU336)  CRYSTAL STRUCTURE OF A HETERODIMERIC ABC TRANSPORTER IN ITS INWARD- FACING CONFORMATION  |   MULTIDRUG TRANSPORTER, TRANSPORT PROTEIN 
4uyn:A   (ASP307) to   (ASN386)  SAR156497 AN EXQUISITELY SELECTIVE INHIBITOR OF AURORA KINASES  |   TRANSFERASE 
4fsn:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fsu:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ft9:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4fti:A   (PRO188) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX 
4ftk:A   (GLU187) to   (LYS267)  CRYSTAL STRUCTURE OF THE CHK1  |   TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX