1a06:A (ALA186) to (HIS273) CALMODULIN-DEPENDENT PROTEIN KINASE FROM RAT | KINASE, SIGNAL TRANSDUCTION, CALCIUM/CALMODULIN
4gue:A (ALA236) to (HIS324) STRUCTURE OF N-TERMINAL KINASE DOMAIN OF RSK2 WITH FLAVONOID GLYCOSIDE QUERCITRIN | SERINE/THREONINE KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4wnk:A (ALA353) to (HIS445) CRYSTAL STRUCTURE OF BOVINE G PROTEIN COUPLED-RECEPTOR KINASE 5 IN COMPLEX WITH CCG215022 | G PROTEIN-COUPLED RECEPTOR KINASE 5, HYDROLASE, PHOSPHORYLATION, CARDIOVASCULAR DISEASE, LIGASE
4wno:A (ALA189) to (ASP279) STRUCTURE OF ULK1 BOUND TO AN INHIBITOR | KINASE, AUTOPHAGY, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4wnp:A (ALA189) to (ALA280) STRUCTURE OF ULK1 BOUND TO A POTENT INHIBITOR | KINASE, AUTOPHAGY, INHIBITOR
4wnp:B (ALA189) to (ASP279) STRUCTURE OF ULK1 BOUND TO A POTENT INHIBITOR | KINASE, AUTOPHAGY, INHIBITOR
4wnp:C (ALA189) to (ASP279) STRUCTURE OF ULK1 BOUND TO A POTENT INHIBITOR | KINASE, AUTOPHAGY, INHIBITOR
4wo5:B (ALA621) to (LEU721) CRYSTAL STRUCTURE OF A BRAF KINASE DOMAIN MONOMER | KINASE, MONOMER, INHIBITOR, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1atp:E (ALA206) to (ALA298) 2.2 ANGSTROM REFINED CRYSTAL STRUCTURE OF THE CATALYTIC SUBUNIT OF CAMP-DEPENDENT PROTEIN KINASE COMPLEXED WITH MNATP AND A PEPTIDE INHIBITOR | TRANSFERASE(PHOSPHOTRANSFERASE)
2bfx:B (PRO257) to (HIS340) MECHANISM OF AURORA-B ACTIVATION BY INCENP AND INHIBITION BY HESPERADIN. | TRANSFERASE, KINASE, MITOSIS, INHIBITION, TRANSFERASE COMPLEX
1bi7:A (ALA187) to (GLN301) MECHANISM OF G1 CYCLIN DEPENDENT KINASE INHIBITION FROM THE STRUCTURE OF THE CDK6-P16INK4A TUMOR SUPPRESSOR COMPLEX | CYCLIN DEPENDENT KINASE, CYCLIN DEPENDENT KINASE INHIBITORY PROTEIN, CDK, INK4, CELL CYCLE, MULTIPLE TUMOR SUPPRESSOR, MTS1, COMPLEX (KINASE/ANTI-ONCOGENE)
4x3f:A (ALA185) to (ALA276) CRYSTAL STRUCTURE OF THE INTRACELLULAR DOMAIN OF THE M. TUBERCULOSIS SER/THR KINASE PKNA | KINASE, AUTOINHIBITION, PHOSPHORYLATION, TRANSFERASE
4x3f:B (ALA185) to (GLY277) CRYSTAL STRUCTURE OF THE INTRACELLULAR DOMAIN OF THE M. TUBERCULOSIS SER/THR KINASE PKNA | KINASE, AUTOINHIBITION, PHOSPHORYLATION, TRANSFERASE
4x3f:C (ALA185) to (ALA276) CRYSTAL STRUCTURE OF THE INTRACELLULAR DOMAIN OF THE M. TUBERCULOSIS SER/THR KINASE PKNA | KINASE, AUTOINHIBITION, PHOSPHORYLATION, TRANSFERASE
4hni:B (SER181) to (GLY281) CRYSTAL STRUCTURE OF CK1E IN COMPLEX WITH PF4800567 | CK1E, KINASE, INHIBITOR, PF4800567, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1o6y:A (SER184) to (ASN278) CATALYTIC DOMAIN OF PKNB KINASE FROM MYCOBACTERIUM TUBERCULOSIS | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TB, TBSGC
3f66:B (ALA1251) to (ARG1336) HUMAN C-MET KINASE IN COMPLEX WITH QUINOXALINE INHIBITOR | C-MET, PROTEIN KINASE, QUINOXALINE, ALTERNATIVE SPLICING; ATP-BINDING; CHROMOSOMAL REARRANGEMENT; DISEASE MUTATION; GLYCOPROTEIN; KINASE; MEMBRANE; NUCLEOTIDE-BINDING; PHOSPHOPROTEIN; POLYMORPHISM; PROTO-ONCOGENE; RECEPTOR; REPEAT; SIGNAL; TRANSFERASE; TRANSMEMBRANE; TYROSINE- PROTEIN KINASE.
3f69:A (SER184) to (GLY279) CRYSTAL STRUCTURE OF THE MYCOBACTERIUM TUBERCULOSIS PKNB MUTANT KINASE DOMAIN IN COMPLEX WITH KT5720 | PROTEIN KINASE, PKNB, MYCOBACTERIUM TUBERCULOSIS, KT5720, STRUCTURAL GENOMICS, STRUCTUAL GENOMICS, COCRYSTALLIZATION OF PKNB KINASE DOMAIN AND INHIBITORS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, ATP-BINDING, KINASE, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3f69:B (SER184) to (GLY279) CRYSTAL STRUCTURE OF THE MYCOBACTERIUM TUBERCULOSIS PKNB MUTANT KINASE DOMAIN IN COMPLEX WITH KT5720 | PROTEIN KINASE, PKNB, MYCOBACTERIUM TUBERCULOSIS, KT5720, STRUCTURAL GENOMICS, STRUCTUAL GENOMICS, COCRYSTALLIZATION OF PKNB KINASE DOMAIN AND INHIBITORS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, ATP-BINDING, KINASE, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4hok:K (SER181) to (GLY281) CRYSTAL STRUCTURE OF APO CK1E | CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE
4hok:U (SER181) to (GLY281) CRYSTAL STRUCTURE OF APO CK1E | CK1E, KINASE, INHIBITOR, PF 4800567, TRANSFERASE
1ob3:A (ALA168) to (HIS281) STRUCTURE OF P. FALCIPARUM PFPK5 | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, CDK
3fe3:A (ALA215) to (ASP304) CRYSTAL STRUCTURE OF THE KINASE MARK3/PAR-1: T211A-S215A DOUBLE MUTANT | SERINE/THREONINE PROTEIN KINASE; MARK;PAR-1; KIN1; UBA DOMAIN;C- TAK1;P78;MARK3, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3skc:A (ALA621) to (LEU721) HUMAN B-RAF KINASE IN COMPLEX WITH AN AMIDE LINKED PYRAZOLOPYRIDINE INHIBITOR | KINASE, ATP-COMPETITIVE INHIBITOR, TRANSFERASE, RAS, MEK, C-RAF, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3skc:B (ALA621) to (LEU721) HUMAN B-RAF KINASE IN COMPLEX WITH AN AMIDE LINKED PYRAZOLOPYRIDINE INHIBITOR | KINASE, ATP-COMPETITIVE INHIBITOR, TRANSFERASE, RAS, MEK, C-RAF, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4i5p:A (SER248) to (HIS331) SELECTIVE & BRAIN-PERMEABLE POLO-LIKE KINASE-2 (PLK-2) INHIBITORS THAT REDUCE -SYNUCLEIN PHOSPHORYLATION IN RAT BRAIN | POLO-LIKE KINASE-2 (PLK-2), SYNUCLEIN, PARKINSON'S DISEASE, KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3sls:A (SER231) to (HIS320) CRYSTAL STRUCTURE OF HUMAN MEK-1 KINASE IN COMPLEX WITH UCB1353770 AND AMPPNP | SERINE-THREONINE KINASE, SIGNALLING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3sls:B (SER231) to (HIS320) CRYSTAL STRUCTURE OF HUMAN MEK-1 KINASE IN COMPLEX WITH UCB1353770 AND AMPPNP | SERINE-THREONINE KINASE, SIGNALLING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4i6h:A (SER248) to (HIS331) SELECTIVE & BRAIN-PERMEABLE POLO-LIKE KINASE-2 (PLK-2) INHIBITORS THAT REDUCE ALPHA-SYNUCLEIN PHOSPHORYLATION IN RAT BRAIN | PARKINSON S DISEASE, KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2c47:B (SER220) to (GLY320) STRUCTURE OF CASEIN KINASE 1 GAMMA 2 | SERINE/THREONINE KINASE, ACTIN CYTOSKELETON ORGANISATION, ATP-BINDING, TRANSFERASE, WNT SIGNALING PATHWAY
2c5x:C (ALA170) to (GLN287) DIFFERENTIAL BINDING OF INHIBITORS TO ACTIVE AND INACTIVE CDK2 PROVIDES INSIGHTS FOR DRUG DESIGN | TRANSFERASE/INHIBITOR, INHIBITION, ACTIVE, INACTIVE, CDK2, CELL CYCLE, CELL DIVISION, KINASE, MITOSIS, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, COMPLEX (TRANSFERASE/INHIBITOR)
2q0n:A (ALA483) to (ALA575) STRUCTURE OF HUMAN P21 ACTIVATING KINASE 4 (PAK4) IN COMPLEX WITH A CONSENSUS PEPTIDE | PROTEIN KINASE, PHOSPHORYLATION, NUCLEOTIDE-BINDING, PAK4, STE20, KINASE, TRANSFERASE, ATP-BINDING, SERINE/THREONINE-PROTEIN KINASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
1ctp:E (ALA206) to (HIS294) STRUCTURE OF THE MAMMALIAN CATALYTIC SUBUNIT OF CAMP-DEPENDENT PROTEIN KINASE AND AN INHIBITOR PEPTIDE DISPLAYS AN OPEN CONFORMATION | TRANSFERASE(PHOSPHOTRANSFERASE), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3g51:A (ALA236) to (HIS324) STRUCTURAL DIVERSITY OF THE ACTIVE CONFORMATION OF THE N- TERMINAL KINASE DOMAIN OF P90 RIBOSOMAL S6 KINASE 2 | N-TERMINAL KINASE DOMAIN OF P90 RIBOSOMAL S6 KINASE 2, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2qnj:A (SER215) to (ASP304) KINASE AND UBIQUITIN-ASSOCIATED DOMAINS OF MARK3/PAR-1 | SERINE/THREONINE PROTEIN KINASE, UBIQUITIN-ASSOCIATED DOMAIN, MARK, PAR-1, TRANSFERASE
4xv9:A (ALA621) to (SER722) B-RAF KINASE DOMAIN IN COMPLEX WITH PLX5568 | B-RAF, BRAF, PROTO-ONCOGENE, V600E, KINASE, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4xyf:A (ALA1251) to (THR1343) CRYSTAL STRUCTURE OF C-MET IN COMPLEX WITH (S)-5-(8-FLUORO-3-(1-(3-(2- METHOXYETHOXY)QUINOLIN-6-YL)ETHYL)-[1,2,4]TRIAZOLO[4,3-A]PYRIDIN-6- YL)-3-METHYLISOXAZOLE | RECEPTOR TYROSINE KINASE, INHIBITOR, COMPLEX, INTRACELLULAR CATALYTIC DOMAIN
4ixp:A (ALA176) to (MET264) CRYSTAL STRUCTURE OF MATERNAL EMBRYONIC LEUCINE ZIPPER KINASE (MELK) | PROTEIN KINASE, REGULATED BY PHOSPHORYLATION, TRANSFERASE
2r4b:A (ALA888) to (ARG979) ERBB4 KINASE DOMAIN COMPLEXED WITH A THIENOPYRIMIDINE INHIBITOR | ERB, KINASE, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE
2r4b:B (ALA888) to (ARG979) ERBB4 KINASE DOMAIN COMPLEXED WITH A THIENOPYRIMIDINE INHIBITOR | ERB, KINASE, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE
2r5t:A (ALA265) to (HIS352) CRYSTAL STRUCTURE OF INACTIVE SERUM AND GLUCOCORTICOID- REGULATED KINASE 1 IN COMPLEX WITH AMP-PNP | AGC PROTEIN KINASE, APOPTOSIS, ATP-BINDING, CYTOPLASM, ENDOPLASMIC RETICULUM, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, UBL CONJUGATION
1e9h:C (ALA170) to (GLN287) THR 160 PHOSPHORYLATED CDK2 - HUMAN CYCLIN A3 COMPLEX WITH THE INHIBITOR INDIRUBIN-5-SULPHONATE BOUND | CELL CYCLE, COMPLEX (PROTEIN KINASE/CYCLIN), KINASES, INHIBITOR, CYCLIN, COMPLEX, PHOSPHORYLATION
2r9s:B (ALA231) to (HIS356) C-JUN N-TERMINAL KINASE 3 WITH 3,5-DISUBSTITUTED QUINOLINE INHIBITOR | JNK3, SIGNALING PROTEIN, TRANSFERASE
4jjr:B (SER181) to (GLY281) A P21 CRYSTAL FORM OF MAMMALIAN CASEIN KINASE 1 DELTA | CK1D, KINASE, CASEIN KINASE, TRANSFERASE
2dwb:A (PRO297) to (HIS380) AURORA-A KINASE COMPLEXED WITH AMPPNP | AURORA, PROTEIN KINASE, ATP-BINDING, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, TRANSFERASE
3tt0:B (ALA668) to (LEU760) CO-STRUCTURE OF FIBROBLAST GROWTH FACTOR RECEPTOR 1 KINASE DOMAIN WITH 3-(2,6-DICHLORO-3,5-DIMETHOXY-PHENYL)-1-{6-[4-(4-ETHYL-PIPERAZIN-1- YL)-PHENYLAMINO]-PYRIMIDIN-4-YL}-1-METHYL-UREA (BGJ398) | KINASE DOMAIN, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3tv4:B (ALA621) to (LEU721) HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH AN BROMOPYRIDINE BENZAMIDE INHIBITOR | KINASE, KINASE INHIBITOR, TRANSFERASE, RAS, C-RAF, MEK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4yhj:A (ALA354) to (HIS446) STRUCTURE AND FUNCTION OF THE HYPERTENSION VARIANT A486V OF G PROTEIN- COUPLED RECEPTOR KINASE 4 (GRK4) | TRANSFERASE
4yhj:B (ALA354) to (GLN445) STRUCTURE AND FUNCTION OF THE HYPERTENSION VARIANT A486V OF G PROTEIN- COUPLED RECEPTOR KINASE 4 (GRK4) | TRANSFERASE
4yht:A (ALA620) to (THR715) BRAF COMPLEXED WITH AN INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1f3m:C (ALA432) to (HIS518) CRYSTAL STRUCTURE OF HUMAN SERINE/THREONINE KINASE PAK1 | KINASE DOMAIN, AUTOINHIBITORY FRAGMENT, HOMODIMER, TRANSFERASE
1f3m:D (ALA432) to (HIS518) CRYSTAL STRUCTURE OF HUMAN SERINE/THREONINE KINASE PAK1 | KINASE DOMAIN, AUTOINHIBITORY FRAGMENT, HOMODIMER, TRANSFERASE
3hdm:A (ALA265) to (HIS352) CRYSTAL STRUCTURE OF SERUM AND GLUCOCORTICOID-REGULATED KINASE 1 IN COMPLEX WITH COMPOUND 1 | AGC PROTEIN KINASE, APOPTOSIS, ATP-BINDING, ENDOPLASMIC RETICULUM, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHORYLATION, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE, KINASE, PHOSPHOPROTEIN
3hdn:A (ALA265) to (SER356) CRYSTAL STRUCTURE OF SERUM AND GLUCOCORTICOID-REGULATED KINASE 1 IN COMPLEX WITH COMPOUND 2 | AGC PROTEIN KINASE, APOPTOSIS, ATP-BINDING, ENDOPLASMIC RETICULUM, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHORYLATION, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE, KINASE, PHOSPHOPROTEIN
2uzu:E (ALA206) to (ALA298) PKA STRUCTURES OF INDAZOLE-PYRIDINE SERIES OF AKT INHIBITORS | CAMP, KINASE, MYRISTATE, TRANSFERASE, LIPOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, PHOSPHORYLATION, PROTEIN KINASE A, NUCLEOTIDE-BINDING, PROTEIN KINASE INHIBITOR, ATP- BINDING, AKT INHIBITORS, NUCLEAR PROTEIN
3ubd:A (ALA236) to (HIS324) STRUCTURE OF N-TERMINAL DOMAIN OF RSK2 KINASE IN COMPLEX WITH FLAVONOID GLYCOSIDE SL0101 | KINASE-INHIBITOR COMPLEX, INDUCED FIT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1fin:C (ALA170) to (GLN287) CYCLIN A-CYCLIN-DEPENDENT KINASE 2 COMPLEX | COMPLEX (TRANSFERASE/CYCLIN), CYCLIN, CDK, PHOSPHORYLATION
2vd5:A (GLU241) to (HIS336) STRUCTURE OF HUMAN MYOTONIC DYSTROPHY PROTEIN KINASE IN COMPLEX WITH THE BISINDOYLMALEIDE INHIBITOR BIM VIII | SERINE/THREONINE-PROTEIN KINASE, KINASE, TRANSFERASE, ATP-BINDING, NUCLEOTIDE-BINDING, CARDIAC CONTRACTILITY, MUSCLE DIFFERENTIATION
2vd5:B (PRO240) to (HIS336) STRUCTURE OF HUMAN MYOTONIC DYSTROPHY PROTEIN KINASE IN COMPLEX WITH THE BISINDOYLMALEIDE INHIBITOR BIM VIII | SERINE/THREONINE-PROTEIN KINASE, KINASE, TRANSFERASE, ATP-BINDING, NUCLEOTIDE-BINDING, CARDIAC CONTRACTILITY, MUSCLE DIFFERENTIATION
3hmo:A (PRO692) to (HIS788) CRYSTAL STRUCTURE OF HUMAN MPS1 CATALYTIC DOMAIN IN COMPLEX WITH THE INHIBITOR STAUROSPORINE | MPS1, TTK, STU, STAUROSPORINE, KINASE, ATP-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TYROSINE- PROTEIN KINASE, TRANSFERASE
2fb8:B (ALA621) to (SER720) STRUCTURE OF THE B-RAF KINASE DOMAIN BOUND TO SB-590885 | KINASE DOMAIN, TRANSFERASE
1g3n:A (ALA187) to (GLN301) STRUCTURE OF A P18(INK4C)-CDK6-K-CYCLIN TERNARY COMPLEX | CYCLIN-DEPENDENT KINASE, INK4 INHIBITOR, VIRAL CYCLIN, CELL CYCLE, SIGNALING PROTEIN
1g3n:E (ALA187) to (HIS297) STRUCTURE OF A P18(INK4C)-CDK6-K-CYCLIN TERNARY COMPLEX | CYCLIN-DEPENDENT KINASE, INK4 INHIBITOR, VIRAL CYCLIN, CELL CYCLE, SIGNALING PROTEIN
3uo5:A (PRO297) to (HIS380) AURORA A IN COMPLEX WITH YL1-038-31 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-IN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uoj:A (PRO297) to (HIS380) AURORA A IN COMPLEX WITH RPM1715 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uok:A (PRO297) to (HIS380) AURORA A IN COMPLEX WITH YL5-81-1 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uok:B (PRO297) to (HIS380) AURORA A IN COMPLEX WITH YL5-81-1 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2fh9:A (ALA219) to (ASP303) STRUCTURE AND DIMERIZATION OF THE KINASE DOMAIN FROM YEAST SNF1 | KINASE DOMAIN; DIMER, SIGNALING PROTEIN, TRANSFERASE, SIGNALING PROTEIN,TRANSFERASE
2vgo:B (PRO257) to (HIS340) CRYSTAL STRUCTURE OF AURORA B KINASE IN COMPLEX WITH REVERSINE INHIBITOR | NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, TRANSFERASE, COILED COIL, CELL DIVISION, KINASE, CANCER, INCENP, NUCLEUS, MITOSIS, AURORA B, METAL-BINDING, AMINOTHIAZOLE, PHOSPHORYLATION, MAGNESIUM, CELL CYCLE, CENTROMERE, MICROTUBULE
2fum:A (SER184) to (HIS277) CATALYTIC DOMAIN OF PROTEIN KINASE PKNB FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH MITOXANTRONE | PROTEIN KINASE-INHIBITOR COMPLEX, TRANSFERASE
2fum:B (SER184) to (ASN278) CATALYTIC DOMAIN OF PROTEIN KINASE PKNB FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH MITOXANTRONE | PROTEIN KINASE-INHIBITOR COMPLEX, TRANSFERASE
2fum:C (SER184) to (HIS277) CATALYTIC DOMAIN OF PROTEIN KINASE PKNB FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH MITOXANTRONE | PROTEIN KINASE-INHIBITOR COMPLEX, TRANSFERASE
2fum:D (SER184) to (HIS277) CATALYTIC DOMAIN OF PROTEIN KINASE PKNB FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH MITOXANTRONE | PROTEIN KINASE-INHIBITOR COMPLEX, TRANSFERASE
2g15:A (ALA1251) to (PHE1344) STRUCTURAL CHARACTERIZATION OF AUTOINHIBITED C-MET KINASE | KINASE DOMAIN, TRANSFERASE
4ksp:A (ALA620) to (LEU720) CRYSTAL STRUCTURE OF HUMAN B-RAF BOUND TO A DFG-OUT INHIBITOR TAK-632 | HUMAN SERINE/THERONINE PROTEIN KINASE, KINASE DRUG COMPLEX,, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ksq:A (ALA620) to (LEU720) CRYSTAL STRUCTURE OF HUMAN B-RAF BOUND TO A DFG-OUT INHIBITOR 5B | HUMAN SERINE/THERONINE PROTEIN KINASE, KINASE DRUG COMPLEX,, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2vrx:B (PRO257) to (HIS340) STRUCTURE OF AURORA B KINASE IN COMPLEX WITH ZM447439 | SERINE/THREONINE-PROTEIN KINASE, KINASE, NUCLEUS, MITOSIS, MAGNESIUM, CELL CYCLE/TRANSFERASE, CENTROMERE, MICROTUBULE, ATP-BINDING, TRANSFERASE, ANTI-CANCER DRUG TARGET, PHOSPHOPROTEIN, PROTEIN KINASE, NUCLEOTIDE-BINDING, COILED COIL, CELL DIVISION, METAL-BINDING
4zhx:A (ALA181) to (HIS265) NOVEL BINDING SITE FOR ALLOSTERIC ACTIVATION OF AMPK | TRANSFERASE, SERINE/THREONINE KINASE, ALLOSTERIC ACTIVATION, NUCLEOTIDE-BINDING
4zhx:C (ALA181) to (HIS265) NOVEL BINDING SITE FOR ALLOSTERIC ACTIVATION OF AMPK | TRANSFERASE, SERINE/THREONINE KINASE, ALLOSTERIC ACTIVATION, NUCLEOTIDE-BINDING
1h1r:C (ALA170) to (GLN287) STRUCTURE OF HUMAN THR160-PHOSPHO CDK2/CYCLIN A COMPLEXED WITH THE INHIBITOR NU6086 | KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP- BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, PHOSPHORYLATION
1h25:C (ALA170) to (GLN287) CDK2/CYCLIN A IN COMPLEX WITH AN 11-RESIDUE RECRUITMENT PEPTIDE FROM RETINOBLASTOMA-ASSOCIATED PROTEIN | TRANSFERASE, CELL CYCLE, PROTEIN KINASE, CYCLIN, CDK2, RECRUITMENT, PEPTIDE SPECIFICITY
3idp:B (SER614) to (ALA718) B-RAF V600E KINASE DOMAIN IN COMPLEX WITH AN AMINOISOQUINOLINE INHIBITOR | ONCOGENE, ATP-BINDING, DFG-OUT, TRANSFERASE, CARDIOMYOPATHY, DISEASE MUTATION, KINASE, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, ZINC-FINGER
1h4l:B (PRO169) to (HIS283) STRUCTURE AND REGULATION OF THE CDK5-P25(NCK5A) COMPLEX | KINASE/KINASE ACTIVATOR, COMPLEX(CYCLINS/CDK), CYCLINS, CYCLIN-DEPENDENT KINASES, CDK5, P35, P25, TRANSFERASE, ATP-BINDING, CELL CYCLE, CELL DIVISION, PHOSPHORYLATION
4l67:A (ALA483) to (HIS569) CRYSTAL STRUCTURE OF CATALYTIC DOMAIN OF PAK4 | CATALYTIC DOMAIN OF PAK4, TRANSFERASE
2w1f:A (PRO297) to (HIS380) STRUCTURE DETERMINATION OF AURORA KINASE IN COMPLEX WITH INHIBITOR | CANCER, AURORA, KINASE, INHIBITOR, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ATP-BINDING, POLYMORPHISM, PHOSPHOPROTEIN, CELL CYCLE
3igo:A (ALA243) to (HIS329) CRYSTAL STRUCTURE OF CRYPTOSPORIDIUM PARVUM CDPK1, CGD3_920 | PARASITE, KINASE, CDPK, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
4l9i:A (ALA357) to (ILE455) BOVINE G PROTEIN COUPLED RECEPTOR KINASE 1 IN COMPLEX WITH PAROXETINE | AGC FAMILY KINASE, SER/THR KINASE, RGS HOMOLOGY DOMAIN, G PROTEIN COUPLED RECEPTOR KINASE, GRK, GRK1, RHODOPSIN KINASE, SSRI, HYDROLYASE, GPCR, PHOSPHORYLATION, TRANSFERASE, MEMBRANE PROTEIN- INHIBITOR COMPLEX
3ii5:B (ALA620) to (LEU720) THE COMPLEX OF WILD-TYPE B-RAF WITH PYRAZOLO PYRIMIDINE INHIBITOR | B-RAF, KINASE, PROTEIN-INHIBITOR COMPLEX, ACETYLATION, ATP- BINDING, CARDIOMYOPATHY, CYTOPLASM, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ZINC, ZINC- FINGER
2w5a:A (SER184) to (ASN268) HUMAN NEK2 KINASE ADP-BOUND | SER/THR PROTEIN KINASE, KINASE, NUCLEUS, MEIOSIS, MITOSIS, CYTOPLASM, SERINE/THREONINE-PROTEIN KINASE, METAL-BINDING, PHOSPHOPROTEIN, NUCLEOTIDE-BINDING, MAGNESIUM, CELL CYCLE, ATP-BINDING, TRANSFERASE, CENTROSOME SPLITTING, ALTERNATIVE SPLICING, COILED COIL, POLYMORPHISM, CELL DIVISION
2h34:B (ALA183) to (LEU275) APOENZYME CRYSTAL STRUCTURE OF THE TUBERCULOSIS SERINE/THREONINE KINASE, PKNE | APOENZYME, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE
3is5:C (ALA305) to (LYS394) CRYSTAL STRUCTURE OF CDPK KINASE DOMAIN FROM TOXOPLASMA GONDII, TGME49_018720 | TOXOPLASMA GONDII, CDPK, STRUCTURAL GENOMICS, PARASITOLOGY, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3is5:F (ALA305) to (HIS390) CRYSTAL STRUCTURE OF CDPK KINASE DOMAIN FROM TOXOPLASMA GONDII, TGME49_018720 | TOXOPLASMA GONDII, CDPK, STRUCTURAL GENOMICS, PARASITOLOGY, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3vqu:A (PRO692) to (HIS788) CRYSTAL STRUCTURE OF HUMAN MPS1 CATALYTIC DOMAIN IN COMPLEX WITH 4- [(4-AMINO-5-CYANO-6-ETHOXYPYRIDIN-2- YL)AMINO]BENZAMIDE | KINASE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2whb:A (ALA170) to (HIS283) TRUNCATION AND OPTIMISATION OF PEPTIDE INHIBITORS OF CDK2, CYCLIN A THROUGH STRUCTURE GUIDED DESIGN | CDK2, KINASE, CYCLIN, ACTIVE, NUCLEUS, MITOSIS, SERINE/THREONINE-PROTEIN KINASE, CYTOPLASM, INHIBITION, CELL CYCLE, ATP-BINDING, CELL DIVISION, PHOSPHOPROTEIN, NUCLEOTIDE-BINDING, TRANSFERASE, POLYMORPHISM, BETA-PEPTIDE, CYCLIN GROOVE
2wih:C (ALA170) to (GLN287) STRUCTURE OF CDK2-CYCLIN A WITH PHA-848125 | CELL CYCLE, ATP-BINDING, TRANSFERASE, POLYMORPHISM, PHOSPHORYLATION, NUCLEOTIDE-BINDING, CELL DIVISION, SERINE/THREONINE-PROTEIN 2 KINASE, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, MITOSIS
3vs1:B (PRO431) to (PHE519) CRYSTAL STRUCTURE OF HCK COMPLEXED WITH A PYRROLO-PYRIMIDINE INHIBITOR 1-[4-(4-AMINO-7-CYCLOPENTYL-7H-PYRROLO[2,3-D]PYRIMIDIN-5-YL)PHENYL]- 3-PHENYLUREA | TYROSINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4lop:C (ALA190) to (HIS305) STRUCTURAL BASIS OF AUTOACTIVATION OF P38 ALPHA INDUCED BY TAB1 (TETRAGONAL CRYSTAL FORM) | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, KINASE-REGULATORY PROTEIN COMPLEX, MAPK, AUTOACTIVATION, AUTOPHOSPHORYLATION, TRANSFERASE
3vvh:C (SER231) to (HIS358) X-RAY STRUCTURE OF THE HUMAN MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1 (MEK1) IN COMPLEX WITH AN INHIBITOR AND MGATP | KINASE DOMAIN, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4lqs:A (GLN556) to (HIS669) CRYSTAL STRUCTURE OF THE CBK1-MOB2 KINASE-COACTIVATOR COMPLEX | KINASE, TRANSFERASE-TRANSFERASE ACTIVATOR COMPLEX
2wma:A (ALA170) to (GLN287) STRUCTURAL AND THERMODYNAMIC CONSEQUENCES OF CYCLIZATION OF PEPTIDE LIGANDS FOR THE RECRUITMENT SITE OF CYCLIN A | CELL CYCLE, CELL DIVISION, ANTI-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, PHOSPHORYLATION, NUCLEOTIDE-BINDING, TRANSCRIPTION REGULATION, CHROMATIN REGULATOR, RECRUITMENT, TRANSCRIPTION, NUCLEUS, MITOSIS, ATP-BINDING, TRANSFERASE
3vw8:A (ALA1251) to (ARG1336) CRYSTAL STRUCTURE OF HUMAN C-MET KINASE DOMAIN WITH ITS INHIBITOR | TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3w10:A (PRO297) to (HIS380) AURORA KINASE A COMPLEXED TO PYRAZOLE AMINOQUINOLINE I | KINASE, PYRAZOLE AMINOQUINOLINE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2wqm:A (SER204) to (ALA300) STRUCTURE OF APO HUMAN NEK7 | ATP-BINDING, POLYMORPHISM, METAL-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE KINASE, MITOSIS, CYTOPLASM, MAGNESIUM, TRANSFERASE, PHOSPHOPROTEIN, PROTEIN KINASE, NUCLEOTIDE-BINDING
2wqn:A (SER204) to (ALA300) STRUCTURE OF ADP-BOUND HUMAN NEK7 | ATP-BINDING, POLYMORPHISM, METAL-BINDING, SERINE/THREONINE-PROTEIN KINASE, MITOSIS, CYTOPLASM, TRANSFERASE, PHOSPHOPROTEIN, PROTEIN KINASE, NUCLEOTIDE-BINDING
2hwo:A (ALA430) to (TYR519) CRYSTAL STRUCTURE OF SRC KINASE DOMAIN IN COMPLEX WITH COVALENT INHIBITOR | KINASE, COVALENT, QUINAZOLINE, MODIFICATION, TRANSFERASE
1ua2:A (ALA180) to (ASN297) CRYSTAL STRUCTURE OF HUMAN CDK7 | CELL CYCLE; PHOSPHORYLATION; PROTEIN-PROTEIN INTERACTION; PROTEIN KINASE, CELL CYCLE, TRANSFERASE
1ua2:B (ALA180) to (MET292) CRYSTAL STRUCTURE OF HUMAN CDK7 | CELL CYCLE; PHOSPHORYLATION; PROTEIN-PROTEIN INTERACTION; PROTEIN KINASE, CELL CYCLE, TRANSFERASE
1ua2:C (ALA180) to (MET292) CRYSTAL STRUCTURE OF HUMAN CDK7 | CELL CYCLE; PHOSPHORYLATION; PROTEIN-PROTEIN INTERACTION; PROTEIN KINASE, CELL CYCLE, TRANSFERASE
1ua2:D (ALA180) to (MET292) CRYSTAL STRUCTURE OF HUMAN CDK7 | CELL CYCLE; PHOSPHORYLATION; PROTEIN-PROTEIN INTERACTION; PROTEIN KINASE, CELL CYCLE, TRANSFERASE
2wtw:A (PRO297) to (ASN386) AURORA-A INHIBITOR STRUCTURE (2ND CRYSTAL FORM) | KINASE, CELL CYCLE, TRANSFERASE, PHOSPHOPROTEIN, PROTEIN KINASE
1ung:B (PRO169) to (SER287) STRUCTURAL MECHANISM FOR THE INHIBITION OF CDK5-P25 BY ROSCOVITINE, ALOISINE AND INDIRUBIN. | CELL CYCLE, COMPLEX(KINASE/ACTIVATOR), INHIBITORS, NEURODEGENERATIVE DISEASES
1unh:B (PRO169) to (HIS283) STRUCTURAL MECHANISM FOR THE INHIBITION OF CDK5-P25 BY ROSCOVITINE, ALOISINE AND INDIRUBIN. | CELL CYCLE, NEURODEGENERATIVE DISEASES, INDIRUBIN
1unl:A (PRO169) to (SER287) STRUCTURAL MECHANISM FOR THE INHIBITION OF CD5-P25 FROM THE ROSCOVITINE, ALOISINE AND INDIRUBIN. | CYCLIN DEPENDENT KINASE, INHIBITOR, ATP-ANALOGUE, NEURODEGENERATIVE DISEASES
1unl:B (PRO169) to (SER287) STRUCTURAL MECHANISM FOR THE INHIBITION OF CD5-P25 FROM THE ROSCOVITINE, ALOISINE AND INDIRUBIN. | CYCLIN DEPENDENT KINASE, INHIBITOR, ATP-ANALOGUE, NEURODEGENERATIVE DISEASES
4m69:B (SER365) to (GLU457) CRYSTAL STRUCTURE OF THE MOUSE RIP3-MLKL COMPLEX | KINASE, PHOSPHORYLATION, TRANSFERASE-SIGNALING PROTEIN COMPLEX
5aaf:A (PRO297) to (HIS380) AURORA A KINASE BOUND TO AN IMIDAZOPYRIDINE INHIBITOR (14A) | TRANSFERASE, AURORA-A, IMIDAZOPYRIDINE, AURORA KINASE, INHIBITOR
4mbj:A (SER614) to (LEU721) HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH AN IMIDAZOPYRIDINE-BASED INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4mbj:B (SER607) to (LEU721) HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH AN IMIDAZOPYRIDINE-BASED INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1uwj:A (ALA620) to (LEU720) THE COMPLEX OF MUTANT V599E B-RAF AND BAY439006 | TRANSFERASE, THREONINE-PROTEIN KINASE, SIGNAL TRANSDUCTION
1uwj:B (ALA620) to (LEU720) THE COMPLEX OF MUTANT V599E B-RAF AND BAY439006 | TRANSFERASE, THREONINE-PROTEIN KINASE, SIGNAL TRANSDUCTION
1v0b:B (ALA168) to (HIS281) CRYSTAL STRUCTURE OF THE T198A MUTANT OF PFPK5 | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, CDK
1v0p:B (ALA168) to (GLU286) STRUCTURE OF P. FALCIPARUM PFPK5-PURVALANOL B LIGAND COMPLEX | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, CDK
2x6d:A (PRO297) to (HIS380) AURORA-A BOUND TO AN INHIBITOR | TRANSFERASE, MITOSIS
2x81:A (PRO297) to (HIS380) STRUCTURE OF AURORA A IN COMPLEX WITH MLN8054 | TRANSFERASE, DRUG-RESISTANCE, CELL CYCLE, CYTOSKELETON
1jbp:E (ALA206) to (ALA298) CRYSTAL STRUCTURE OF THE CATALYTIC SUBUNIT OF CAMP- DEPENDENT PROTEIN KINASE COMPLEXED WITH A SUBSTRATE PEPTIDE, ADP AND DETERGENT | PROTEIN-SUBSTRATE COMPLEX, TRANSFERASE
4mne:B (ALA621) to (LEU721) CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4mne:C (ALA621) to (SER720) CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4mne:F (ALA621) to (ARG719) CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4mne:G (ALA621) to (ARG719) CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4mne:H (SER231) to (HIS358) CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4mnf:B (ALA621) to (ARG719) CRYSTAL STRUCTURE OF BRAF-V600E BOUND TO GDC0879 | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, ACTIVE CONFORMATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2j0i:A (ALA483) to (HIS569) CRYSTAL STRUCTURE OF THE HUMAN P21-ACTIVATED KINASE 4 | PROTEIN KINASE, PHOSPHORYLATION, NUCLEOTIDE-BINDING, PAK4, STE20, KINASE, TRANSFERASE, ATP-BINDING, ALTERNATIVE SPLICING, SERINE/THREONINE-PROTEIN KINASE
5ap0:A (PRO692) to (HIS788) NATURALLY OCCURRING MUTATIONS IN THE MPS1 GENE PREDISPOSE CELLS TO KINASE INHIBITOR DRUG RESISTANCE. | TRANSFERASE, MPS1, PROTEIN KINASE, MITOSIS, DRUG RESISTANCE
5ar2:A (PRO194) to (ARG295) RIP2 KINASE CATALYTIC DOMAIN (1 - 310) | TRANSFERASE, KINASE DOMAIN, KINASE INHIBITOR, STRUCTURE-BASED DRUG DESIGN, INHIBITOR SELECTIVITY
2xkd:A (SER184) to (GLU267) STRUCTURE OF NEK2 BOUND TO AMINOPYRAZINE COMPOUND 12 | TRANSFERASE, CENTROSOME, MITOSIS
4mxc:A (ALA1251) to (THR1343) CRYSTAL STRUCTURE OF CMET IN COMPLEX WITH NOVEL INHIBITOR | CMET INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2xne:A (PRO297) to (HIS380) STRUCTURE OF AURORA-A BOUND TO AN IMIDAZOPYRAZINE INHIBITOR | SER-THR PROTEIN KINASE COMPLEX, PROTO-ONCOGENE, KINASE, MITOSIS, CELL CYCLE, MICROTUBULE, TRANSFERASE, CYTOSKELETON, CELL DIVISION
2xno:A (SER184) to (GLU267) STRUCTURE OF NEK2 BOUND TO CCT243779 | TRANSFERASE, CENTROSOME, MITOSIS, CELL CYCLE
2jav:A (SER184) to (ASN268) HUMAN KINASE WITH PYRROLE-INDOLINONE LIGAND | TRANSFERASE, PHOSPHORYLATION, NUCLEOTIDE-BINDING, ATP-BINDING, CELL DIVISION, METAL-BINDING, NUCLEAR PROTEIN, SERINE/THREONINE-PROTEIN KINASE, SERINE/THREONINE PROTEIN KINASE, KINASE, MEIOSIS, MITOSIS, MAGNESIUM, CELL CYCLE
4nfn:A (SER207) to (ARG300) HUMAN TAU TUBULIN KINASE 1 (TTBK1) COMPLEXED WITH 3-({5-[(4-AMINO-4- METHYLPIPERIDIN-1-YL)METHYL]PYRROLO[2,1-F][1,2,4]TRIAZIN-4-YL}AMINO)- 5-BROMOPHENOL | PROTEIN KINASE, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1k9a:D (ALA354) to (HIS446) CRYSTAL STRUCTURE ANALYSIS OF FULL-LENGTH CARBOXYL-TERMINAL SRC KINASE AT 2.5 A RESOLUTION | CARBOXYL-TERMINAL SRC KINASE, COOH-TERMINAL SRC KINASE, CSK, SRC, SFK, SIGNAL TRANSDUCTION, SH2, SH3, SRC HOMOLOGY, TYROSINE KINASE, CYTOPLASMIC TYROSINE KINASE, CBP, ONCOGENE, CANCER, TRANSFERASE
4njd:A (ALA483) to (HIS569) STRUCTURE OF P21-ACTIVATED KINASE 4 WITH A NOVEL INHIBITOR KY-04031 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ztx:B (PRO257) to (HIS340) AURORA KINASE SELECTIVE INHIBITORS IDENTIFIED USING A TAXOL- INDUCED CHECKPOINT SENSITIVITY SCREEN. | TRANSFERASE-CELL CYCLE COMPLEX, TRANSFERASE, TAXOL-INDUCED CHECKPOINT INHIBITOR
4nus:A (ALA236) to (HIS324) RSK2 N-TERMINAL KINASE IN COMPLEX WITH LJH685 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4nw5:A (ALA236) to (HIS324) RSK2 N-TERMINAL KINASE IN COMPLEX WITH 2-AMINO-7-SUBSTITUTED BENZOXAZOLE COMPOUND 8 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4nw6:A (ALA236) to (HIS324) RSK2 N-TERMINAL KINASE IN COMPLEX WITH 2-AMINO-7-SUBSTITUTED BENZOXAZOLE COMPOUND 27 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4o0y:A (ALA483) to (HIS569) BACK POCKET FLEXIBILITY PROVIDES GROUP-II PAK SELECTIVITY FOR TYPE 1 KINASE INHIBITORS | PAK4, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4o27:B (ALA187) to (HIS271) CRYSTAL STRUCTURE OF MST3-MO25 COMPLEX WITH WIF MOTIF | SCAFFOLD PROTEIN, PROTEIN SER/THR KINASE, TRANSFERASE ACTIVATOR- TRANSFERASE COMPLEX, SIGNALING PROTEIN
5cen:A (ALA278) to (THR374) CRYSTAL STRUCTURE OF DLK (KINASE DOMAIN) | KINASE, TRANSFERASE
5ceo:A (ALA278) to (THR374) DLK IN COMPLEX WITH INHIBITOR 2-((6-(3,3-DIFLUOROPYRROLIDIN-1-YL)-4- (1-(OXETAN-3-YL)PIPERIDIN-4-YL)PYRIDIN-2-YL)AMINO)ISONICOTINONITRILE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ceq:A (ALA278) to (THR374) DLK IN COMPLEX WITH INHIBITOR 2-((1-CYCLOPENTYL-5-(1-(OXETAN-3-YL) PIPERIDIN-4-YL)-1H-PYRAZOL-3-YL)AMINO)ISONICOTINONITRILE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2yza:A (ALA181) to (HIS265) CRYSTAL STRUCTURE OF KINASE DOMAIN OF HUMAN 5'-AMP-ACTIVATED PROTEIN KINASE ALPHA-2 SUBUNIT MUTANT (T172D) | SIGNALING PROTEIN, SERINE/THREONINE PROTEIN KINASE, PHOSPHORYLATION, ATP-BINDING, NUCLEOTIDE-BINDING, CHOLESTEROL BIOSYNTHESIS, FATTY ACID BIOSYNTHESIS, LIPID SYNTHESIS, GLUCOSE METABOLISM, MAGNESIUM, METAL-BINDING, SERINE/THREONINE-PROTEIN KINASE, STEROID BIOSYNTHESIS, TRANSFERASE, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
2z7q:A (ALA230) to (HIS318) CRYSTAL STRUCTURE OF THE N-TERMINAL KINASE DOMAIN OF HUMAN RSK-1 BOUND TO AMP-PCP | PROTEIN KINASE; CANCER; KINASE INHIBITOR, ATP-BINDING, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2z7r:A (ALA230) to (HIS318) CRYSTAL STRUCTURE OF THE N-TERMINAL KINASE DOMAIN OF HUMAN RSK1 BOUND TO STAUROSPORINE | PROTEIN KINASE, CANCER, KINASE INHIBITOR, ATP-BINDING, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2z7s:A (ALA230) to (HIS318) CRYSTAL STRUCTURE OF THE N-TERMINAL KINASE DOMAIN OF HUMAN RSK1 BOUND TO PURVALNOL A | PROTEIN KINASE, CANCER, KINASE INHIBITOR, TRANSFERASE
1xo2:B (ALA187) to (GLN301) CRYSTAL STRUCTURE OF A HUMAN CYCLIN-DEPENDENT KINASE 6 COMPLEX WITH A FLAVONOL INHIBITOR, FISETIN | CRYSTAL STRUCTURE,HUMAN CYCLIN-DEPENDENT KINASE 6, FISETIN, CELL CYCLE-TRANSFERASE COMPLEX
5csw:A (ALA621) to (LEU721) B-RAF IN COMPLEX WITH DABRAFENIB | KINASE, PROTEROS BIOSTRUCTURES GMBH, TRANSFERASE
5csx:A (ALA621) to (GLU720) CRYSTAL STRUCTURE OF B-RAF IN COMPLEX WITH BI 882370 | KINASE, TRANSFERASE
5ct7:A (ALA621) to (LEU721) BRAF IN COMPLEX WITH RAF265 | KINASE, TRANSFERASE
5ct7:B (ALA621) to (LEU721) BRAF IN COMPLEX WITH RAF265 | KINASE, TRANSFERASE
5czo:A (SER181) to (GLU281) STRUCTURE OF S. CEREVISIAE HRR25:MAM1 COMPLEX, FORM 2 | CASEIN KINASE, MONOPOLIN, TRANSFERASE
3kmu:A (ALA357) to (GLN450) CRYSTAL STRUCTURE OF THE ILK/ALPHA-PARVIN CORE COMPLEX (APO) | CELL ADHESION, ANK REPEAT, ATP-BINDING, CELL JUNCTION, CELL MEMBRANE, INTEGRIN-BINDING PROTEIN, MEMBRANE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, PSEUDOKINASE, ACTIN-BINDING, ALTERNATIVE SPLICING
3kmw:A (ALA357) to (GLN450) CRYSTAL STRUCTURE OF THE ILK/ALPHA-PARVIN CORE COMPLEX (MGATP) | CELL ADHESION, ANK REPEAT, ATP-BINDING, CELL JUNCTION, CELL MEMBRANE, INTEGRIN-BINDING PROTEIN, MEMBRANE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, PSEUDOKINASE, ACTIN-BINDING, ALTERNATIVE SPLICING, CYTOPLASM, CYTOSKELETON
1mru:A (SER184) to (ASN278) INTRACELLULAR SER/THR PROTEIN KINASE DOMAIN OF MYCOBACTERIUM TUBERCULOSIS PKNB. | REGULATORY, ATP-RECOGNITION, MOLECULAR EVOLUTION, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, TRANSFERASE
1mru:B (SER184) to (HIS277) INTRACELLULAR SER/THR PROTEIN KINASE DOMAIN OF MYCOBACTERIUM TUBERCULOSIS PKNB. | REGULATORY, ATP-RECOGNITION, MOLECULAR EVOLUTION, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, TRANSFERASE
3a61:A (ALA261) to (HIS349) CRYSTAL STRUCTURE OF UNPHOSPHORYLATED P70S6K1 (FORM II) | KINASE, KINASE DOMAIN, INACTIVE, ACTIVE, RIBOSOMAL S6 KINASE, ACTIVATION, ALTERNATIVE INITIATION, ATP-BINDING, CELL JUNCTION, CYTOPLASM, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, SYNAPSE, SYNAPTOSOME, TRANSFERASE
5d9k:A (ALA236) to (HIS324) RSK2 N-TERMINAL KINASE IN COMPLEX WITH BI-D1870 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5d9k:B (ALA236) to (HIS324) RSK2 N-TERMINAL KINASE IN COMPLEX WITH BI-D1870 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5d9l:A (ALA236) to (HIS324) RSK2 N-TERMINAL KINASE IN COMPLEX WITH BIS-PHENOL PYRAZOLE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3a7h:A (ALA187) to (HIS271) HUMAN MST3 KINASE IN COMPLEX WITH ATP | TWO-LOBE PROTEIN KINASE FOLD, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, TRANSFERASE
3a7h:B (ALA187) to (HIS271) HUMAN MST3 KINASE IN COMPLEX WITH ATP | TWO-LOBE PROTEIN KINASE FOLD, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, TRANSFERASE
3a7g:A (ALA187) to (HIS271) HUMAN MST3 KINASE | TWO-LOBE PROTEIN KINASE FOLD, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, TRANSFERASE
5de2:A (SER204) to (ALA300) STRUCTURAL MECHANISM OF NEK7 ACTIVATION BY NEK9-INDUCED DIMERISATION | PROTEIN KINASE, MITOSIS, PROTEIN-PROTEIN INTERACTION, TRANSFERASE
4pp7:A (ALA621) to (LEU721) HIGHLY POTENT AND SELECTIVE 3-N-METHYLQUINAZOLINE-4(3H)-ONE BASED INHIBITORS OF B-RAFV600E KINASE | SERINE/THREONINE-PROTEIN KINASE B-RAF, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4pp7:B (ALA621) to (ALA718) HIGHLY POTENT AND SELECTIVE 3-N-METHYLQUINAZOLINE-4(3H)-ONE BASED INHIBITORS OF B-RAFV600E KINASE | SERINE/THREONINE-PROTEIN KINASE B-RAF, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4prj:A (PRO297) to (HIS380) AURORA A KINASE DOMAIN WITH COMPOUND 2 (N-[1-(3-CYANOBENZYL)-1H- PYRAZOL-4-YL]-6-(1H-PYRAZOL-4-YL)-1H-INDAZOLE-3-CARBOXAMIDE) | PROTEIN KINASE, PHOSPHO-TRANSFER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4an2:A (SER231) to (HIS358) CRYSTAL STRUCTURES OF HUMAN MEK1 WITH CARBOXAMIDE-BASED ALLOSTERIC INHIBITOR XL518 (GDC-0973), OR RELATED ANALOGS. | TRANSFERASE, MAP2K1, ATP-BINDING, ALLOSTERIC INHIBITION
4an9:A (SER231) to (HIS358) CRYSTAL STRUCTURES OF HUMAN MEK1 WITH CARBOXAMIDE-BASED ALLOSTERIC INHIBITOR XL518 (GDC-0973), OR RELATED ANALOGS. | TRANSFERASE, MAP2K1, ATP-BINDING, ALLOSTERIC INHIBITION
5drd:A (PRO297) to (HIS380) AURORA A KINASE IN COMPLEX WITH ATP IN SPACE GROUP P6122 | AURORA A KINASE, MITOTIC KINASE, PPI, TRANSFERASE
4apc:A (SER171) to (GLU254) CRYSTAL STRUCTURE OF HUMAN NIMA-RELATED KINASE 1 (NEK1) | TRANSFERASE
4aw2:A (PRO246) to (HIS340) CRYSTAL STRUCTURE OF CDC42 BINDING PROTEIN KINASE ALPHA (MRCK ALPHA) | TRANSFERASE, CDC42BPA
4qfg:A (ALA181) to (HIS265) STRUCTURE OF AMPK IN COMPLEX WITH STAUROSPORINE INHIBITOR AND IN THE ABSENCE OF A SYNTHETIC ACTIVATOR | CBM, KINASE, AMPK, SIGNALING PROTEIN-INHIBITOR COMPLEX
4qfs:A (ALA181) to (HIS265) STRUCTURE OF AMPK IN COMPLEX WITH BR2-A769662CORE ACTIVATOR AND STAUROSPORINE INHIBITOR | CBM, KINASE, AMPK, SIGNALING PROTEIN-INHIBITOR-ACTIVATOR COMPLEX
4b8l:A (PRO257) to (HIS340) AURORA B KINASE P353G MUTANT | CELL CYCLE, CANCER
4b8m:B (PRO257) to (HIS340) AURORA B KINASE IN COMPLEX WITH VX-680 | CELL CYCLE, CANCER
4b9d:A (SER171) to (LYS255) CRYSTAL STRUCTURE OF HUMAN NIMA-RELATED KINASE 1 (NEK1) WITH INHIBITOR. | TRANSFERASE, INHIBITOR
5ehy:A (PRO691) to (HIS788) RAPID DISCOVERY OF PYRIDO[3,4-D]PYRIMIDINE INHIBITORS OF MONOPOLAR SPINDLE KINASE 1 (MPS1) USING A STRUCTURE-BASED HYDRIDIZATION APPROACH | SPINDLE ASSEMBLY CHECKPOINT (SAC), ONCOLOGY TARGET PYRIDO[3, 4- D]PYRIMIDINE BASED INHIBITORS SELECTIVE AGAINST MPS1, TRANSFERASE
4qo9:A (ALA187) to (ASN277) MST3 IN COMPLEX WITH DANUSERTIB | PROTEIN KINASE, MST3, STK24, STERILE 20-LIKE KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3mn3:A (ALA219) to (ASP303) AN INHIBITED CONFORMATION FOR THE PROTEIN KINASE DOMAIN OF THE SACCHAROMYCES CEREVISIAE AMPK HOMOLOG SNF1 | SNF1, KINASE DOMAIN, AUTOINHIBITORY REGION, TRANSFERASE
4bl1:A (ALA176) to (MET264) CRYSTAL STRUCTURE OF UNPHOSPHORYLATED MATERNAL EMBRYONIC LEUCINE ZIPPER KINASE (MELK) IN COMPLEX WITH AMP-PNP | TRANSFERASE
5ezv:A (ALA181) to (HIS265) X-RAY CRYSTAL STRUCTURE OF AMP-ACTIVATED PROTEIN KINASE ALPHA-2/ALPHA- 1 RIM CHIMAERA (ALPHA-2(1-347)/ALPHA-1(349-401)/ALPHA-2(397-END) BETA-1 GAMMA-1) CO-CRYSTALLIZED WITH C2 (5-(5-HYDROXYL-ISOXAZOL-3- YL)-FURAN-2-PHOSPHONIC ACID) | TRANSFERASE, SERINE/THREONINE KINASE, ALLOSTERIC ACTIVATION, NUCLEOTIDE-BINDING
5ezv:C (ALA181) to (HIS265) X-RAY CRYSTAL STRUCTURE OF AMP-ACTIVATED PROTEIN KINASE ALPHA-2/ALPHA- 1 RIM CHIMAERA (ALPHA-2(1-347)/ALPHA-1(349-401)/ALPHA-2(397-END) BETA-1 GAMMA-1) CO-CRYSTALLIZED WITH C2 (5-(5-HYDROXYL-ISOXAZOL-3- YL)-FURAN-2-PHOSPHONIC ACID) | TRANSFERASE, SERINE/THREONINE KINASE, ALLOSTERIC ACTIVATION, NUCLEOTIDE-BINDING
3mv5:A (ALA317) to (HIS405) CRYSTAL STRUCTURE OF AKT-1-INHIBITOR COMPLEXES | KINASE INHIBITOR, TRANSFERASE
3mvh:A (ALA317) to (HIS405) CRYSTAL STRUCTURE OF AKT-1-INHIBITOR COMPLEXES | KINASE INHIBITOR, TRANSFERASE
3my0:J (ALA377) to (ILE492) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:V (ALA377) to (SER493) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3myg:A (PRO297) to (HIS380) AURORA A KINASE COMPLEXED WITH SCH 1473759 | KINASE, CELL CYCLE, INHIBITOR, TRANSFERASE
5fd2:B (ALA621) to (ALA718) B-RAF WILD-TYPE KINASE DOMAIN IN COMPLEX WITH A PURINYLPYRIDINYLAMINO- BASED INHIBITOR | PHOSPHOTRANSFERASE, INHIBITOR, MELANOMA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4r5y:A (ALA621) to (ARG719) THE COMPLEX STRUCTURE OF BRAF V600E KINASE DOMAIN WITH A NOVEL BRAF INHIBITOR | KINASE, SIGNAL TRANSDUCTION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4r5y:B (ALA621) to (GLU720) THE COMPLEX STRUCTURE OF BRAF V600E KINASE DOMAIN WITH A NOVEL BRAF INHIBITOR | KINASE, SIGNAL TRANSDUCTION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3c4y:A (ALA357) to (HIS449) CRYSTAL STRUCTURE OF APO FORM OF G PROTEIN COUPLED RECEPTOR KINASE 1 AT 7.51A | SER/THR KINASE, RGS HOMOLOGY DOMAIN, G PROTEIN COUPLED RECEPTOR KINASE, GRK, GRK1, RHODOPSIN KINASE, P-LOOP, AUTOPHOSPHORYLATION, ATP-BINDING, LIPOPROTEIN, MEMBRANE, METHYLATION, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PRENYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3c4y:B (ALA357) to (HIS449) CRYSTAL STRUCTURE OF APO FORM OF G PROTEIN COUPLED RECEPTOR KINASE 1 AT 7.51A | SER/THR KINASE, RGS HOMOLOGY DOMAIN, G PROTEIN COUPLED RECEPTOR KINASE, GRK, GRK1, RHODOPSIN KINASE, P-LOOP, AUTOPHOSPHORYLATION, ATP-BINDING, LIPOPROTEIN, MEMBRANE, METHYLATION, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PRENYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3c51:A (ALA357) to (ILE455) CRYSTAL STRUCTURE OF G PROTEIN COUPLED RECEPTOR KINASE 1 BOUND TO ADP AND MAGNESIUM CHLORIDE AT 3.55A | SER/THR KINASE, RGS HOMOLOGY DOMAIN, G PROTEIN COUPLED RECEPTOR KINASE, GRK, GRK1, RHODOPSIN KINASE, P-LOOP, AUTOPHOSPHORYLATION, ADP, ATP-BINDING, LIPOPROTEIN, MEMBRANE, METHYLATION, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, PRENYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4byi:A (PRO297) to (HIS380) AURORA A KINASE BOUND TO A HIGHLY SELECTIVE IMIDAZOPYRIDINE INHIBITOR | TRANSFERASE, CELL CYCLE, INHIBITOR
3cd8:A (ALA1251) to (THR1343) X-RAY STRUCTURE OF C-MET WITH TRIAZOLOPYRIDAZINE INHIBITOR. | C-MET, KINASE, TRIAZOLOPYRIDAZINE, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
4c2v:B (PRO257) to (HIS340) AURORA B KINASE IN COMPLEX WITH THE SPECIFIC INHIBITOR BARASERTIB | TRANSFERASE-CELL CYCLE COMPLEX, AZD1152
3ncz:B (PRO243) to (LYS339) X-RAY CO-STRUCTURE OF RHO-ASSOCIATED PROTEIN KINASE (ROCK1) WITH A POTENT 2H-ISOQUINOLIN-1-ONE INHIBITOR | RHO KINASE, DIMER, PHOSPHORYLATION, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4c2w:B (PRO257) to (HIS340) CRYSTAL STRUCTURE OF AURORA B IN COMPLEX WITH AMP-PNP | TRANSFERASE
5flf:E (ALA668) to (THR761) DISEASE LINKED MUTATION IN FGFR | TRANSFERASE, AUTO-ACTIVATING, CANCER, GROWTH FACTOR, RECEPTOR, MUTATION;
3coh:A (PRO297) to (HIS380) CRYSTAL STRUCTURE OF AURORA-A IN COMPLEX WITH A PENTACYCLIC INHIBITOR | AURORA-A, INHIBITOR COMPLEX, ATP-BINDING, CELL CYCLE, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3coh:B (PRO297) to (HIS380) CRYSTAL STRUCTURE OF AURORA-A IN COMPLEX WITH A PENTACYCLIC INHIBITOR | AURORA-A, INHIBITOR COMPLEX, ATP-BINDING, CELL CYCLE, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4cfe:A (ALA181) to (HIS265) STRUCTURE OF FULL LENGTH HUMAN AMPK IN COMPLEX WITH A SMALL MOLECULE ACTIVATOR, A BENZIMIDAZOLE DERIVATIVE (991) | TRANSFERASE, NUCLEOTIDE-BINDING, STAUROSPORINE-BINDING, SERINE/THREONINE-PROTEIN KINASE, ACTIVATOR, CARBOHYDRATE BINDING MODULE (CBM)
4cfe:C (ALA181) to (HIS265) STRUCTURE OF FULL LENGTH HUMAN AMPK IN COMPLEX WITH A SMALL MOLECULE ACTIVATOR, A BENZIMIDAZOLE DERIVATIVE (991) | TRANSFERASE, NUCLEOTIDE-BINDING, STAUROSPORINE-BINDING, SERINE/THREONINE-PROTEIN KINASE, ACTIVATOR, CARBOHYDRATE BINDING MODULE (CBM)
3nyo:B (ALA353) to (HIS445) CRYSTAL STRUCTURE OF G PROTEIN-COUPLED RECEPTOR KINASE 6 IN COMPLEX WITH AMP | KINASE, GRK, RGS HOMOLOGY DOMAIN, G PROTEIN-COUPLED RECEPTOR KINASE, TRANSFERASE
3o0g:B (PRO169) to (SER287) CRYSTAL STRUCTURE OF CDK5:P25 IN COMPLEX WITH AN ATP ANALOGUE | KINASE, KINASE ACTIVATOR COMPLEX, KINASE INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE ACTIVATOR COMPLEX
4rzv:A (SER614) to (LEU721) CRYSTAL STRUCTURE OF THE BRAF (R509H) KINASE DOMAIN MONOMER BOUND TO VEMURAFENIB | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3d14:A (PRO310) to (HIS393) CRYSTAL STRUCTURE OF MOUSE AURORA A (ASN186->GLY, LYS240->ARG, MET302- >LEU) IN COMPLEX WITH 1-{5-[2-(THIENO[3,2-D]PYRIMIDIN-4-YLAMINO)- ETHYL]- THIAZOL-2-YL}-3-(3-TRIFLUOROMETHYL-PHENYL)-UREA | AURORA A, SMALL-MOLECULE INHIBITOR, KINASE, TRANSFERASE
3d2i:A (PRO310) to (HIS393) CRYSTAL STRUCTURE OF MOUSE AURORA A (ASN186->GLY, LYS240- >ARG, MET302->LEU) IN COMPLEX WITH 1-{5-[2-(1-METHYL-1H- PYRAZOLO[4,3-D]PYRIMIDIN-7-YLAMINO)-ETHYL]-THIAZOL-2-YL}-3- (3-TRIFLUOROMETHYL-PHENYL)-UREA | AURORA A, SMALL-MOLECULE INHIBITOR, KINASE, TRANSFERASE
4tnb:A (ALA353) to (HIS445) CRYSTAL STRUCTURE OF G PROTEIN-COUPLED RECEPTOR KINASE 5 IN COMPLEX WITH SANGIVAMYCIN | GRK5-SANGIVAMYCIN COMPLEX, GPCR KINASE, KINASE, INHIBITOR, SIGNALING PROTEIN
3dae:B (ALA219) to (ASP303) CRYSTAL STRUCTURE OF PHOSPHORYLATED SNF1 KINASE DOMAIN | KINASE, AMPK, SNF1, ATP-BINDING, CARBOHYDRATE METABOLISM, MEMBRANE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4czt:A (ALA199) to (ASN283) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF SNRK3.23 AT1G30270 | TRANSFERASE, POTASSIUM TRANSPORT, SNRK3
4czt:B (ALA199) to (ASN283) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF SNRK3.23 AT1G30270 | TRANSFERASE, POTASSIUM TRANSPORT, SNRK3
4czt:C (ALA199) to (ASN283) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF SNRK3.23 AT1G30270 | TRANSFERASE, POTASSIUM TRANSPORT, SNRK3
4d2p:A (ALA176) to (MET264) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT STERBASED DRUG DESIGN, KINASE
4d2p:D (ALA176) to (MET264) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT STERBASED DRUG DESIGN, KINASE
4d2v:D (ALA176) to (MET264) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN
3dls:A (ALA1170) to (THR1252) CRYSTAL STRUCTURE OF HUMAN PAS KINASE BOUND TO ADP | PAS KINASE, PASK, PROTEIN KINASE, DRUG DISCOVERY, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
3dls:B (ALA1170) to (ASP1248) CRYSTAL STRUCTURE OF HUMAN PAS KINASE BOUND TO ADP | PAS KINASE, PASK, PROTEIN KINASE, DRUG DISCOVERY, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
3dls:C (ALA1170) to (THR1252) CRYSTAL STRUCTURE OF HUMAN PAS KINASE BOUND TO ADP | PAS KINASE, PASK, PROTEIN KINASE, DRUG DISCOVERY, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
3dls:D (ALA1170) to (ASP1248) CRYSTAL STRUCTURE OF HUMAN PAS KINASE BOUND TO ADP | PAS KINASE, PASK, PROTEIN KINASE, DRUG DISCOVERY, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
3dls:E (ALA1170) to (ASP1248) CRYSTAL STRUCTURE OF HUMAN PAS KINASE BOUND TO ADP | PAS KINASE, PASK, PROTEIN KINASE, DRUG DISCOVERY, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
3dls:F (ALA1170) to (ASP1248) CRYSTAL STRUCTURE OF HUMAN PAS KINASE BOUND TO ADP | PAS KINASE, PASK, PROTEIN KINASE, DRUG DISCOVERY, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
3orl:A (SER184) to (GLY279) MYCOBACTERIUM TUBERCULOSIS PKNB KINASE DOMAIN L33D MUTANT (CRYSTAL FORM 3) | STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, KINASE DOMAIN, SIGNAL TRANSDUCTION, TRANSFERASE
3orp:A (SER184) to (GLY279) MYCOBACTERIUM TUBERCULOSIS PKNB KINASE DOMAIN L33D MUTANT (CRYSTAL FORM 5) | STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, KINASE DOMAIN, SIGNAL TRANSDUCTION, TRANSFERASE
3ow4:B (ALA317) to (ALA409) DISCOVERY OF DIHYDROTHIENO- AND DIHYDROFUROPYRIMIDINES AS POTENT PAN AKT INHIBITORS | SERINE-THREONINE KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4dea:A (PRO297) to (HIS380) AURORA A IN COMPLEX WITH YL1-038-18 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-IN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4deb:A (PRO297) to (HIS380) AURORA A IN COMPLEX WITH RK2-17-01 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-IN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hes:A (ALA174) to (ASP266) HUMAN LEUCINE ZIPPER- AND STERILE ALPHA MOTIF-CONTAINING KINASE (ZAK, MLT, HCCS-4, MRK, AZK, MLTK) IN COMPLEX WITH VEMURAFENIB | KINASE, COMPLEX, TRANSFERASE
5hie:A (ALA621) to (LEU721) BRAF KINASE DOMAIN B3AC LOOP DELETION MUTANT IN COMPLEX WITH DABRAFENIB | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hie:B (ALA621) to (SER720) BRAF KINASE DOMAIN B3AC LOOP DELETION MUTANT IN COMPLEX WITH DABRAFENIB | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hie:C (ALA621) to (LEU721) BRAF KINASE DOMAIN B3AC LOOP DELETION MUTANT IN COMPLEX WITH DABRAFENIB | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hie:D (ALA621) to (LEU721) BRAF KINASE DOMAIN B3AC LOOP DELETION MUTANT IN COMPLEX WITH DABRAFENIB | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ho6:A (ALA1251) to (ARG1336) CRYSTAL STRUCTURE OF CMET IN COMPLEX WITH CMPD. | TRANSFERASE
3p86:A (ALA719) to (LYS810) CRYSTAL STRUCTURE OF CTR1 KINASE DOMAIN MUTANT D676N IN COMPLEX WITH STAUROSPORINE | KINASE, ETR1, ERS1, ETR2, PHOSPHORYLATION, TRANSFERASE
3p86:B (ALA719) to (LYS810) CRYSTAL STRUCTURE OF CTR1 KINASE DOMAIN MUTANT D676N IN COMPLEX WITH STAUROSPORINE | KINASE, ETR1, ERS1, ETR2, PHOSPHORYLATION, TRANSFERASE
5i4n:A (PRO720) to (LEU808) CRYSTAL STRUCTURE OF THE E596A V617F MUTANT JAK2 PSEUDOKINASE DOMAIN BOUND TO MG-ATP | TRANSFERASE, PSEUDOKINASE, ATP BINDING
4ump:A (ALA176) to (MET264) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE
4umt:A (ALA176) to (MET264) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN
4umu:A (ALA176) to (MET264) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN, KINASE
3pls:A (ALA1255) to (ALA1347) RON IN COMPLEX WITH LIGAND AMP-PNP | PROTEIN KINASE, CIS AUTOPHOSPHORYLATION CONFORMATION, RECEPTOR TYROSINE KINASE, AMP-PNP, UNPHOSPHORYLATED, SINGLE-SPAN TRANSMEMBRANE RECEPTOR, TRANSFERASE
4e26:A (ALA621) to (LEU721) BRAF IN COMPLEX WITH AN ORGANIC INHIBITOR 7898734 | KINASE, INHIBITOR, ONCOPROTEIN, MELANOMA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ppk:B (ALA621) to (LEU721) HUMAN B-RAF KINASE IN COMPLEX WITH A NON-OXIME FUROPYRIDINE INHIBITOR | PROTEIN KINASE, B-RAF ATP-COMPETITIVE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3ppz:A (ALA719) to (ILE809) CRYSTAL STRUCTURE OF CTR1 KINASE DOMAIN IN COMPLEX WITH STAUROSPORINE | KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
3ppz:B (ALA719) to (LYS810) CRYSTAL STRUCTURE OF CTR1 KINASE DOMAIN IN COMPLEX WITH STAUROSPORINE | KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
3prf:A (ALA621) to (LEU721) CRYSTAL STRUCTURE OF HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH A NON- OXIME FUROPYRIDINE INHIBITOR | PROTEIN KINASE, ATP-COMPETITIVE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3prf:B (ALA621) to (SER720) CRYSTAL STRUCTURE OF HUMAN B-RAF KINASE DOMAIN IN COMPLEX WITH A NON- OXIME FUROPYRIDINE INHIBITOR | PROTEIN KINASE, ATP-COMPETITIVE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ehe:A (ALA621) to (LEU721) B-RAF KINASE DOMAIN IN COMPLEX WITH AN AMINOTHIENOPYRIMIDINE-BASED INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4el9:A (ALA236) to (HIS324) STRUCTURE OF N-TERMINAL KINASE DOMAIN OF RSK2 WITH AFZELIN | SERINE/THREONINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3q4z:B (ALA432) to (HIS518) STRUCTURE OF UNPHOSPHORYLATED PAK1 KINASE DOMAIN | KINASE DOMAIN, SIGNALLING PATHWAY, TRANSFERASE
5ita:A (ALA621) to (ALA718) CRYSTAL STRUCTURE OF BRAF KINASE DOMAIN BOUND TO AZ-VEM | TRANSFERASE, KINASE AND INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3q5i:A (ALA235) to (SER321) CRYSTAL STRUCTURE OF PBANKA_031420 | CDPK, PLASMODIUM, MALARIA, CALCIUM DEPENDENT PROTEIN KINASE, PHOSPHOTRANSFERASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
5iu2:B (SER295) to (ASN389) DISCOVERY OF IMIDAZOQUINOLINES AS A NOVEL CLASS OF POTENT, SELECTIVE AND IN VIVO EFFICACIOUS COT KINASE INHIBITORS | COT, TPL-2, MAP3K8, KINASE, INHIBITOR, COMPLEX, TRANSFERASE
4ez5:A (ALA187) to (GLN301) CDK6 (MONOMERIC) IN COMPLEX WITH INHIBITOR | PROTEIN KINASE, ATP BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qgw:A (SER526) to (GLU617) CRYSTAL STRUCTURE OF ITK KINASE BOUND TO AN INHIBITOR | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qjt:A (PRO292) to (ASN446) THE STRUCTURE OF AND PHOTOLYTIC INDUCED CHANGES OF CARBON MONOXIDE BINDING TO THE CYTOCHROME BA3-OXIDASE FROM THERMUS THERMOPHILUS | CYTOCHROME BA3 OXIDASE, CARBON MONOXIDE, CO PHOTODISSOCIATION, OXIDOREDUCTASE
3qjq:A (ASP291) to (ASN446) THE STRUCTURE OF AND PHOTOLYTIC INDUCED CHANGES OF CARBON MONOXIDE BINDING TO THE CYTOCHROME BA3-OXIDASE FROM THERMUS THERMOPHILUS | CYTOCHROME BA3 OXIDASE, CARBON MONOXIDE, CO PHOTODISSOCIATION, OXIDOREDUCTASE
4uzh:A (PRO297) to (HIS380) SAR156497 AN EXQUISITELY SELECTIVE INHIBITOR OF AURORA KINASES | TRANSFERASE
4fc0:A (ALA620) to (LEU720) CRYSTAL STRUCTURE OF HUMAN KINASE DOMAIN OF B-RAF WITH A DFG-OUT INHIBITOR | HUMAN SERINE/THERONINE PROTEIN KINASE, KINASE DRUG COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fie:A (ALA483) to (HIS569) FULL-LENGTH HUMAN PAK4 | SERINE/THREONINE-PROTEIN KINASE PAK4, KINASE DOMAIN, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
4fie:B (ALA483) to (HIS569) FULL-LENGTH HUMAN PAK4 | SERINE/THREONINE-PROTEIN KINASE PAK4, KINASE DOMAIN, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
4fk3:A (ALA621) to (ALA718) B-RAF KINASE V600E ONCOGENIC MUTANT IN COMPLEX WITH PLX3203 | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, ONCOGENIC V600E, KINASE-KINASE INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5jgd:A (ALA197) to (PRO292) CRYSTAL STRUCTURE OF HUMAN TAK1/TAB1 FUSION PROTEIN IN COMPLEX WITH LIGAND 12 | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, TAK1-TAB1 KINASE
3rhk:A (ALA1251) to (PHE1344) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF C-MET KINASE IN COMPLEX WITH ARQ 197 | KINASE, RECEPTOR TYROSINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fvq:A (PRO720) to (LEU808) CRYSTAL STRUCTURE OF THE JAK2 PSEUDOKINASE DOMAIN (MG-ATP-BOUND FORM) | JANUS PROTEIN KINASE, PSEUDOKINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
5jsm:B (ALA621) to (LEU721) BRAFV600E KINASE DOMAIN IN COMPLEX WITH CHEMICALLY LINKED VEMURAFENIB INHIBITOR VEM-3-VEM | KINASE, DIMER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5jsm:C (ALA621) to (SER722) BRAFV600E KINASE DOMAIN IN COMPLEX WITH CHEMICALLY LINKED VEMURAFENIB INHIBITOR VEM-3-VEM | KINASE, DIMER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5jt2:B (ALA621) to (ARG719) BRAFV600E KINASE DOMAIN IN COMPLEX WITH CHEMICALLY LINKED VEMURAFENIB INHIBITOR VEM-BISAMIDE | KINASE, DIMER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fza:B (ALA187) to (HIS271) CRYSTAL STRUCTURE OF MST4-MO25 COMPLEX | SCAFFOLD PROTEIN, PROTEIN SER/THR KINASE, ATP BINDING, SIGNALING PROTEIN-TRANSFERASE COMPLEX
4g3c:B (ALA566) to (GLY661) CRYSTAL STRUCTURE OF APO MURINE NF-KAPPAB INDUCING KINASE (NIK) | NON-RD KINASE, PROTEIN SERINE/THREONINE KINASE, NF-KAPPAB, MAP3K14, TRANSFERASE
4g3e:A (ALA566) to (GLY661) CRYSTAL STRUCTURE OF MURINE NF-KAPPAB INDUCING KINASE (NIK) BOUND TO A 6-ALKYNYLINDOLINE (CMP1) | NON-RD KINASE, PROTEIN SERINE/THREONINE KINASE, NF-KAPPAB,STRUCTURE- BASED DRUG DESIGN, MAP3K14, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5kbr:B (ALA432) to (HIS518) PAK1 IN COMPLEX WITH 7-AZAINDOLE INHIBITOR | SERINE/THREONINE-PROTEIN KINASE PAK1, KINASE, TRANSFERASE
4gg7:A (ALA1251) to (THR1343) CRYSTAL STRUCTURE OF CMET IN COMPLEX WITH NOVEL INHIBITOR | C-MET INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5kq5:A (ALA181) to (HIS265) AMPK BOUND TO ALLOSTERIC ACTIVATOR | KINASE ALLOSTERIC ACTIVATOR, TRANSFERASE
5l2i:A (ALA187) to (GLN301) THE X-RAY CO-CRYSTAL STRUCTURE OF HUMAN CDK6 AND PALBOCICLIB. | CYCLIN-DEPENDENT KINASE, KINASE INHIBITOR, KINASE SELECTIVITY, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5m51:A (SER184) to (GLU267) NEK2 BOUND TO ARYLAMINOPURINE COMPOUND 8 | PROTEIN KINASE, INHIBITOR, CENTROSOME SEPARATION, TRANSFERASE- INHIBITOR COMPLEX
5m53:A (SER184) to (GLU267) NEK2 BOUND TO ARYLAMINOPURINE INHIBITOR 11 | PROTEIN KINASE, INHIBITOR, CENTROSOME SEPARATION, TRANSFERASE- INHIBITOR COMPLEX
1bi8:A (ALA187) to (GLN301) MECHANISM OF G1 CYCLIN DEPENDENT KINASE INHIBITION FROM THE STRUCTURES CDK6-P19INK4D INHIBITOR COMPLEX | CYCLIN DEPENDENT KINASE, CYCLIN DEPENDENT KINASE INHIBITORY PROTEIN, CDK, INK4, CELL CYCLE, COMPLEX (KINASE/INHIBITOR)
1bi8:C (ALA187) to (GLN301) MECHANISM OF G1 CYCLIN DEPENDENT KINASE INHIBITION FROM THE STRUCTURES CDK6-P19INK4D INHIBITOR COMPLEX | CYCLIN DEPENDENT KINASE, CYCLIN DEPENDENT KINASE INHIBITORY PROTEIN, CDK, INK4, CELL CYCLE, COMPLEX (KINASE/INHIBITOR)
3twj:B (SER242) to (HIS335) RHO-ASSOCIATED PROTEIN KINASE 1 (ROCK 1) IN COMPLEX WITH RKI1447 | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3twj:C (SER242) to (GLY328) RHO-ASSOCIATED PROTEIN KINASE 1 (ROCK 1) IN COMPLEX WITH RKI1447 | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uo6:A (PRO297) to (HIS380) AURORA A IN COMPLEX WITH YL5-083 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uo6:B (PRO297) to (HIS380) AURORA A IN COMPLEX WITH YL5-083 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2vgp:B (PRO257) to (HIS340) CRYSTAL STRUCTURE OF AURORA B KINASE IN COMPLEX WITH A AMINOTHIAZOLE INHIBITOR | NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, TRANSFERASE, COILED COIL, CELL DIVISION, KINASE, CANCER, INCENP, NUCLEUS, MITOSIS, AURORA B, METAL-BINDING, AMINOTHIAZOLE, PHOSPHORYLATION, MAGNESIUM, CELL CYCLE, CENTROMERE, MICROTUBULE
3uzp:B (SER181) to (GLY281) CRYSTAL STRUCTURE OF CK1D WITH PF670462 FROM P21 CRYSTAL FORM | CK1D, KINASE, INHIBITOR, PF670462, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3v8s:B (PRO243) to (GLY328) HUMAN RHO-ASSOCIATED PROTEIN KINASE 1 (ROCK 1) IN COMPLEX WITH INDAZOLE DERIVATIVE (COMPOUND 18) | KINASE, DIMERIZATION, MYOSIN, TRANSFERASE, INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3v8s:D (PRO243) to (HIS335) HUMAN RHO-ASSOCIATED PROTEIN KINASE 1 (ROCK 1) IN COMPLEX WITH INDAZOLE DERIVATIVE (COMPOUND 18) | KINASE, DIMERIZATION, MYOSIN, TRANSFERASE, INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
2wqo:A (SER184) to (GLU267) STRUCTURE OF NEK2 BOUND TO THE AMINOPYRIDINE CCT241950 | KINASE, NUCLEUS, MEIOSIS, MITOSIS, CYTOPLASM, ALTERNATIVE SPLICING, SERINE/THREONINE-PROTEIN KINASE, METAL-BINDING, PHOSPHOPROTEIN, NUCLEOTIDE-BINDING, MAGNESIUM, CELL CYCLE, ATP-BINDING, TRANSFERASE, COILED COIL, POLYMORPHISM, CELL DIVISION
2xnm:A (SER184) to (GLU267) STRUCTURE OF NEK2 BOUND TO CCT | TRANSFERASE, CENTROSOME, MITOSIS, CELL CYCLE
4nfm:A (SER207) to (ARG300) HUMAN TAU TUBULIN KINASE 1 (TTBK1) | PROTEIN KINASE, PHOSPHOTRANSFERASE, TRANSFERASE
2y7j:A (PRO196) to (HIS288) STRUCTURE OF HUMAN PHOSPHORYLASE KINASE, GAMMA 2 | TRANSFERASE
2y7j:D (PRO196) to (HIS288) STRUCTURE OF HUMAN PHOSPHORYLASE KINASE, GAMMA 2 | TRANSFERASE
5cep:A (ALA278) to (THR374) DLK IN COMPLEX WITH INHIBITOR N-(1-ISOPROPYL-5-(PIPERIDIN-4-YL)-1H- PYRAZOL-3-YL)-4-(TRIFLUOROMETHYL)PYRIDIN-2-AMINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ow8:A (ALA185) to (GLY277) CRYSTAL STRUCTURE OF KINASE DOMAIN OF PKNA FROM MTB | PKNA, KINASE, DRUG TARGET, MTB
4aua:A (ALA187) to (GLN301) LIGANDED X-RAY CRYSTAL STRUCTURE OF CYCLIN DEPENDENT KINASE 6 (CDK6) | TRANSFERASE
4qfr:A (ALA181) to (HIS265) STRUCTURE OF AMPK IN COMPLEX WITH CL-A769662 ACTIVATOR AND STAUROSPORINE INHIBITOR | CBM, AMPK, KINASE, SIGNALING PROTEIN-INHIBITOR-ACTIVATOR COMPLEX
4rew:A (ALA183) to (HIS267) CRYSTAL STRUCTURE OF THE NON-PHOSPHORYLATED HUMAN ALPHA1 BETA2 GAMMA1 HOLO-AMPK COMPLEX | HUMAN ALPHA1 BETA2 GAMMA1 HOLO-AMPK COMPLEX, SERINE/THREONINE PROTEIN KINASE, AXIN, CAMKKBETA, LKB1, GLYCOGEN, PHOSPHORYLATION, TRANSFERASE
3nux:A (ALA187) to (GLN301) CDK6 (MONOMERIC) IN COMPLEX WITH INHIBITOR | KINASE, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4cff:C (ALA181) to (HIS265) STRUCTURE OF FULL LENGTH HUMAN AMPK IN COMPLEX WITH A SMALL MOLECULE ACTIVATOR, A THIENOPYRIDONE DERIVATIVE (A-769662) | TRANSFERASE, NUCLEOTIDE-BINDING, STAUROSPORINE-BINDING, SERINE/THREONINE-PROTEIN KINASE, ACTIVATOR, CARBOHYDRATE BINDING MODULE (CBM)
4tnd:A (ALA353) to (HIS445) CRYSTAL STRUCTURE OF G PROTEIN-COUPLED RECEPTOR KINASE 5 IN COMPLEX WITH AMP-PNP | GRK5-(5-ADENYLYLIMIDODIPHOSPHATE) COMPLEX, GRK5-(AMP-PNP) COMPLEX, GPCR KINASE, KINASE, GPCR KINASE 5, SIGNALING PROTEIN
4d2t:A (ALA176) to (MET264) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN, KINASE
4d2t:C (ALA176) to (MET264) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN, KINASE
5hi2:A (ALA621) to (ARG719) BRAF KINASE DOMAIN B3AC LOOP DELETION MUTANT IN COMPLEX WITH SORAFENIB | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hid:A (ALA621) to (SER722) BRAF KINASE DOMAIN B3AC LOOP DELETION MUTANT IN COMPLEX WITH AZ628 | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hid:B (ALA621) to (LEU721) BRAF KINASE DOMAIN B3AC LOOP DELETION MUTANT IN COMPLEX WITH AZ628 | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4umq:A (ALA176) to (MET264) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN
3psb:A (ALA621) to (LEU721) FURO[2,3-C]PYRIDINE-BASED INDANONE OXIMES AS POTENT AND SELECTIVE B- RAF INHIBITORS | KINASE, ATP-BINDING, CARDIOMYOPATHY, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, ZINC-FINGER, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3psb:B (ALA621) to (LEU721) FURO[2,3-C]PYRIDINE-BASED INDANONE OXIMES AS POTENT AND SELECTIVE B- RAF INHIBITORS | KINASE, ATP-BINDING, CARDIOMYOPATHY, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, ZINC-FINGER, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4fig:A (ALA483) to (HIS569) CATALYTIC DOMAIN OF HUMAN PAK4 | SERINE/THREONINE-PROTEIN KINASE PAK4, KINASE DOMAIN, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
4fig:B (ALA483) to (HIS569) CATALYTIC DOMAIN OF HUMAN PAK4 | SERINE/THREONINE-PROTEIN KINASE PAK4, KINASE DOMAIN, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
5k3y:B (PRO257) to (HIS340) CRYSTAL STRUCTURE OF AURORAB/INCENP IN COMPLEX WITH BI 811283 | KINASE, INHIBITOR, TRANSFERASE
5knj:A (SER378) to (SER467) PSEUDOKINASE DOMAIN OF MLKL BOUND TO COMPOUND 1. | PSEUDOKINASE DOMAIN MLKL COMPOUND 1 GFE OUT TYPE 2 INHIBITOR, MEMBRANE PROTEINS-INHIBITOR COMPLEX
5knj:B (SER378) to (LEU466) PSEUDOKINASE DOMAIN OF MLKL BOUND TO COMPOUND 1. | PSEUDOKINASE DOMAIN MLKL COMPOUND 1 GFE OUT TYPE 2 INHIBITOR, MEMBRANE PROTEINS-INHIBITOR COMPLEX