4wg3:A (ASP228) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1610 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4wg4:A (ASP228) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1613 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR
3rny:A (GLU584) to (HIS672) CRYSTAL STRUCTURE OF HUMAN RSK1 C-TERMINAL KINASE DOMAIN | PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE
3rny:B (LYS587) to (HIS672) CRYSTAL STRUCTURE OF HUMAN RSK1 C-TERMINAL KINASE DOMAIN | PROTEIN KINASE, AUTOINHIBITION, TRANSFERASE
1ny3:A (CYS244) to (HIS322) CRYSTAL STRUCTURE OF ADP BOUND TO MAP KAP KINASE 2 | MAP KAP KINASE 2, MK2, ADP, KINASE, SER/THR KINASE, TRANSFERASE
2bdw:A (PRO193) to (VAL268) CRYSTAL STRUCTURE OF THE AUTO-INHIBITED KINASE DOMAIN OF CALCIUM/CALMODULIN ACTIVATED KINASE II | KINASE; CALMODULIN ACTIVATED, TRANSFERASE
2bdw:B (PRO193) to (VAL268) CRYSTAL STRUCTURE OF THE AUTO-INHIBITED KINASE DOMAIN OF CALCIUM/CALMODULIN ACTIVATED KINASE II | KINASE; CALMODULIN ACTIVATED, TRANSFERASE
3f3z:A (GLY202) to (HIS279) CRYSTAL STRUCTURE OF CRYPTOSPORIDIUM PARVUM CALCIUM DEPENDENT PROTEIN KINASE CGD7_1840 IN PRESENCE OF INDIRUBIN E804 | CALCIUM DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, SGC
3faa:A (GLU394) to (GLN498) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A 2- AMINOIMIDAZOLE INHIBITOR | KINASE, TGFBETA, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3faa:B (GLU394) to (GLY500) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A 2- AMINOIMIDAZOLE INHIBITOR | KINASE, TGFBETA, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3faa:C (GLU394) to (SER496) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A 2- AMINOIMIDAZOLE INHIBITOR | KINASE, TGFBETA, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3faa:D (GLU394) to (GLN498) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A 2- AMINOIMIDAZOLE INHIBITOR | KINASE, TGFBETA, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
2pmo:X (ASN224) to (ALA322) CRYSTAL STRUCTURE OF PFPK7 IN COMPLEX WITH HYMENIALDISINE | SER/THR PROTEIN KINASE; PLASMODIUM FALCIPARUM; TRANSFERASE; PHOSPHORYLATION, TRANSFERASE
3fpm:A (TYR240) to (HIS322) CRYSTAL STRUCTURE OF A SQUARATE INHIBITOR BOUND TO MAPKAP KINASE-2 | 3D-STRUCTURE, ATP-BINDING, ALTERNATIVE SPLICING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3soa:A (PRO193) to (VAL277) FULL-LENGTH HUMAN CAMKII | KINASE, PROTEIN KINASE, PHOSPHORYLATION, CALCIUM/CALMODULIN, CYTOSOLIC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3soc:B (GLN378) to (LEU485) CRYSTAL STRUCTURE OF ACTIVIN RECEPTOR TYPE-IIA (ACVR2A) KINASE DOMAIN IN COMPLEX WITH A QUINAZOLIN | STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE, PROTEIN KINASE
2pzy:C (TYR240) to (HIS322) STRUCTURE OF MK2 COMPLEXED WITH COMPOUND 76 | MK2, PROTEIN KINASE, TRANSFERASE
2pzy:D (TYR240) to (HIS322) STRUCTURE OF MK2 COMPLEXED WITH COMPOUND 76 | MK2, PROTEIN KINASE, TRANSFERASE
4ifg:A (CYS231) to (HIS305) CRYSTAL STRUCTURE OF TGCDPK1 WITH INHIBITOR BOUND | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3fxz:A (VAL445) to (HIS518) CRYSTAL STRUCTURE OF PAK1 KINASE DOMAIN WITH RUTHENIUM COMPLEX LAMBDA-FL172 | TRANSFERASE, KINASE, ATP-BINDING, PHOSPHORYLATION, ALLOSTERIC ENZYME, ALTERNATIVE SPLICING, APOPTOSIS, CELL JUNCTION, CYTOPLASM, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE
4ih8:A (CYS231) to (HIS305) CRYSTAL STRUCTURE OF TGCDPK1 WITH INHIBITOR BOUND | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ihp:A (ASP228) to (HIS305) CRYSTAL STRUCTURE OF TGCDPK1 WITH INHIBITOR BOUND | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3sx9:A (ASP228) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR, RM-1-132 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
2qlu:A (GLN377) to (SER484) CRYSTAL STRUCTURE OF ACTIVIN RECEPTOR TYPE II KINASE DOMAIN FROM HUMAN | TGF-BETA, ACTRIIB, SERINE/THREONINE KINASE RECEPTOR, ALTERNATIVE SPLICING, ATP-BINDING, DISEASE MUTATION, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3t3u:A (ASP228) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR, RM-1-130 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3t3v:A (ASP228) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR, RM-1-87 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4iti:A (GLU207) to (SER291) CRYSTAL STRUCTURE OF RIP1 KINASE IN COMPLEX WITH NECROSTATIN-3 ANALOG | ALPHA/BETA, RIP1 KINASE, NECROPTOSIS, NECROSTATINS, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3tac:A (PRO199) to (HIS273) CRYSTAL STRUCTURE OF THE LIPRIN-ALPHA/CASK COMPLEX | TRANSFERASE-PROTEIN BINDING COMPLEX
3gok:A (TYR240) to (HIS322) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:B (TYR240) to (HIS322) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:C (TYR240) to (HIS322) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:D (TYR240) to (HIS322) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:E (TYR240) to (HIS322) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:F (TYR240) to (HIS322) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:G (TYR240) to (HIS322) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:H (TYR240) to (HIS322) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:I (TYR240) to (HIS322) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:J (TYR240) to (HIS322) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:K (TYR240) to (HIS322) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3gok:L (TYR240) to (HIS322) BINDING SITE MAPPING OF PROTEIN LIGANDS | MK2, MAPKAP KINASE 2, ISOTOPE LABELLING, INSECT CELL EXPRESSION, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4jbv:A (CYS231) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1268 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jdi:A (GLY493) to (HIS569) CRYSTAL STRUCTURE OF SERINE/THREONINE-PROTEIN KINASE PAK 4 IN COMPLEX WITH PAKTIDE S PEPTIDE SUBSTRATE | TRANSFERASE-PEPTIDE COMPLEX, TRANSFERASE/PEPTIDE, SERINE/THREONINE- PROTEIN KINASE PAK4, ATP BINDING, PHOSPHORYLATION
4jg8:A (ALA586) to (HIS676) STRUCTURE OF RSK2 T493M CTD MUTANT BOUND TO 2-CYANO-N-(1-HYDROXY-2- METHYLPROPAN-2-YL)-3-(3-(3,4,5-TRIMETHOXYPHENYL)-1H-INDAZOL-5-YL) ACRYLAMIDE | PROTEIN KINASE, PHOSPHORYLATION, COVALENT INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4jnw:A (THR199) to (HIS275) BACTERIALLY EXPRESSED TITIN KINASE | MUSCLE CYTOSKELETON, TRANSFERASE
4jnw:B (THR199) to (HIS275) BACTERIALLY EXPRESSED TITIN KINASE | MUSCLE CYTOSKELETON, TRANSFERASE
4yjn:A (CYS231) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1639 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3tzm:A (GLU394) to (SER496) TGF-BETA RECEPTOR TYPE 1 IN COMPLEX WITH SB431542 | ALK5, SB431542, KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ysj:A (ASP205) to (HIS282) CALCIUM-DEPENDENT PROTEIN KINASE FROM EIMERIA TENELLA IN COMPLEX WITH ADP | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING
4ysj:B (ASP205) to (HIS282) CALCIUM-DEPENDENT PROTEIN KINASE FROM EIMERIA TENELLA IN COMPLEX WITH ADP | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING
4ysm:A (ASP205) to (HIS282) CALCIUM-DEPENDENT PROTEIN KINASE FROM EIMERIA TENELLA | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING
4ysm:B (ASP205) to (HIS282) CALCIUM-DEPENDENT PROTEIN KINASE FROM EIMERIA TENELLA | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING
2v7o:A (PRO194) to (HIS269) CRYSTAL STRUCTURE OF HUMAN CALCIUM-CALMODULIN-DEPENDENT PROTEIN KINASE II GAMMA | KINASE, S/T KINASE, TRANSFERASE, ATP-BINDING, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, CALMODULIN-BINDING
4yuq:A (CYS208) to (HIS282) CDPK1 FROM EIMERIA TENELLA IN COMPLEX WITH INHIBITOR UW1354 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yuq:B (CYS208) to (HIS282) CDPK1 FROM EIMERIA TENELLA IN COMPLEX WITH INHIBITOR UW1354 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2f57:A (GLY621) to (HIS697) CRYSTAL STRUCTURE OF THE HUMAN P21-ACTIVATED KINASE 5 | PAK5, KINASE DOMAINS, GROUPII PAKS, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
4yzb:A (LYS207) to (HIS282) CDPK1 FROM EIMERIA TENELLA IN COMPLEX WITH INHIBITOR UW1521 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3upz:A (ASP228) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH BUMPLESS BKI ANALOG UW1243 | SERINE/THREONINE PROTEIN KINASE, CALCIUM-BINDING, ATP-BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uto:A (TYR333) to (HIS408) TWITCHIN KINASE REGION FROM C.ELEGANS (FN31-NL-KIN-CRD-IG26) | KINASE, MUSCLE SARCOMERE, TRANSFERASE
3hx4:A (ASP228) to (HIS305) CRYSTAL STRUCTURE OF CDPK1 OF TOXOPLASMA GONDII, TGME49_101440, IN PRESENCE OF CALCIUM | CDPKS, TOXOPLASMA, KINASE, PROTIST, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3v51:A (ASP228) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR RM-1-176 | SERINE/THREONINE PROTEIN KINASE, CALCIUM-BINDING, ATP-BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3v5p:A (ASP228) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1288 | SERINE/THREONINE PROTEIN KINASE, CALCIUM-BINDING, ATP-BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3hzt:A (ASP253) to (HIS330) CRYSTAL STRUCTURE OF TOXOPLASMA GONDII CDPK3, TGME49_105860 | CALCIUM DEPENDENT KINASE, CALMODULIN, TROPONIN PARASITE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2vn9:A (PRO194) to (HIS269) CRYSTAL STRUCTURE OF HUMAN CALCIUM CALMODULIN DEPENDENT PROTEIN KINASE II DELTA ISOFORM 1, CAMKD | SERINE/THREONINE-PROTEIN KINASE, SERINE-THREONINE KINASE, CELLULAR DIFFERENTIATION, VASCULAR SMOOTH MUSCLE, KINASE, TRANSFERASE, ATP-BINDING, PHOSPHOPROTEIN, CALMODULIN-BINDING, NUCLEOTIDE-BINDING
2vn9:B (PRO194) to (HIS269) CRYSTAL STRUCTURE OF HUMAN CALCIUM CALMODULIN DEPENDENT PROTEIN KINASE II DELTA ISOFORM 1, CAMKD | SERINE/THREONINE-PROTEIN KINASE, SERINE-THREONINE KINASE, CELLULAR DIFFERENTIATION, VASCULAR SMOOTH MUSCLE, KINASE, TRANSFERASE, ATP-BINDING, PHOSPHOPROTEIN, CALMODULIN-BINDING, NUCLEOTIDE-BINDING
3i7b:A (CYS231) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR NM-PP1 | PROTEIN KINASE, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, TRANSFERASE
3i7c:A (CYS231) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR NA-PP2 | PROTEIN KINASE, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, TRANSFERASE
2vwi:C (LYS207) to (HIS288) STRUCTURE OF THE OSR1 KINASE, A HYPERTENSION DRUG TARGET | KINASE, STE KINASE, HYPERTENSION, TRANSFERASE
2vwi:D (LYS207) to (HIS288) STRUCTURE OF THE OSR1 KINASE, A HYPERTENSION DRUG TARGET | KINASE, STE KINASE, HYPERTENSION, TRANSFERASE
4zji:A (LYS444) to (HIS518) PAK1 IN COMPLEX WITH 2-CHLORO-5-ETHYL-8-FLUORO-11-(4-METHYLPIPERAZIN- 1-YL)-DIBENZODIAZEPINE | INHIBITOR, KINASE, PAK1, ALLOSTERIC, TRANSFERASE
4zji:B (LYS444) to (HIS518) PAK1 IN COMPLEX WITH 2-CHLORO-5-ETHYL-8-FLUORO-11-(4-METHYLPIPERAZIN- 1-YL)-DIBENZODIAZEPINE | INHIBITOR, KINASE, PAK1, ALLOSTERIC, TRANSFERASE
4zjj:A (LYS444) to (HIS518) PAK1 IN COMPLEX WITH (S)-N-(TERT-BUTYL)-3-((2-CHLORO-5-ETHYL-8-FLUORO- DIBENZODIAZEPIN-11-YL)AMINO)PYRROLIDINE-1-CARBOXAMIDE | PAK1, INHIBITOR, KINASE, ALLOSTERIC, TRANSFERASE
4zlo:B (GLY442) to (HIS518) SERINE/THREONINE-PROTEIN KINASE PAK1 COMPLEXED WITH A DIBENZODIAZEPINE: IDENTIFICATION OF AN ALLOSTERIC SITE ON PAK1 | DIBENZODAZEPINE, PAK1, KINASE, ALLOSTERIC INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4lgd:A (ASP203) to (HIS275) STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5 | HIPPO, MST AUTOACTIVATION, RASSF, SARAH DOMAIN, DIMERIZATION, SIGNALING PROTEIN
4lgd:B (VAL201) to (HIS275) STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5 | HIPPO, MST AUTOACTIVATION, RASSF, SARAH DOMAIN, DIMERIZATION, SIGNALING PROTEIN
4lgd:C (VAL201) to (HIS275) STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5 | HIPPO, MST AUTOACTIVATION, RASSF, SARAH DOMAIN, DIMERIZATION, SIGNALING PROTEIN
4lgd:D (ASP203) to (HIS275) STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5 | HIPPO, MST AUTOACTIVATION, RASSF, SARAH DOMAIN, DIMERIZATION, SIGNALING PROTEIN
1tki:A (ASP202) to (HIS275) AUTOINHIBITED SERINE KINASE DOMAIN OF THE GIANT MUSCLE PROTEIN TITIN | SERINE KINASE, TITIN, MUSCLE, AUTOINHIBITION
1tki:B (ASP202) to (HIS275) AUTOINHIBITED SERINE KINASE DOMAIN OF THE GIANT MUSCLE PROTEIN TITIN | SERINE KINASE, TITIN, MUSCLE, AUTOINHIBITION
4zy4:B (LYS444) to (HIS518) CRYSTAL STRUCTURE OF P21 ACTIVATED KINASE 1 IN COMPLEX WITH AN INHIBITOR COMPOUND 4 | KINASE, INHIBITOR, COMPLEX
4zy5:A (GLY442) to (HIS518) CRYSTAL STRUCTURE OF P21-ACTIVATED KINASE 1 IN COMPLEX WITH AN INHIBITOR COMPOUND 17 | KINASE, INHIBITOR, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4zy5:B (GLY442) to (HIS518) CRYSTAL STRUCTURE OF P21-ACTIVATED KINASE 1 IN COMPLEX WITH AN INHIBITOR COMPOUND 17 | KINASE, INHIBITOR, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2wei:A (CYS255) to (HIS329) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF CRYPTOSPORIDIUM PARVUM CALCIUM DEPENDENT PROTEIN KINASE IN COMPLEX WITH 3- MB-PP1 | NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, KINASE, TRANSFERASE, ATP-BINDING
2wel:A (PRO194) to (HIS269) CRYSTAL STRUCTURE OF SU6656-BOUND CALCIUM/CALMODULIN- DEPENDENT PROTEIN KINASE II DELTA IN COMPLEX WITH CALMODULIN | CELLULAR DIFFERENTIATION, SERINE/THREONINE-PROTEIN KINASE, PHOSPHOPROTEIN, CALMODULIN-BINDING, CALMODULIN BINDING, KINASE, TRANSFERASE, ATP-BINDING, NUCLEOTIDE-BINDING, VASCULAR SMOOTH MUSCLE, SERINE-THREONINE KINASE
2wtc:A (TYR404) to (HIS483) CRYSTAL STRUCTURE OF CHK2 IN COMPLEX WITH AN INHIBITOR | TRANSFERASE, KINASE, CELL CYCLE, LI-FRAUMENI SYNDROME
4m84:A (CYS231) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1455 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3wi6:A (CYS244) to (HIS322) CRYSTAL STRUCTURE OF MAPKAP KINASE-2 (MK2) IN COMPLEX WITH NON- SELECTIVE INHIBITOR | GLY-RICH LOOP FORMED, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3wi6:B (CYS244) to (HIS322) CRYSTAL STRUCTURE OF MAPKAP KINASE-2 (MK2) IN COMPLEX WITH NON- SELECTIVE INHIBITOR | GLY-RICH LOOP FORMED, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3wi6:C (CYS244) to (HIS322) CRYSTAL STRUCTURE OF MAPKAP KINASE-2 (MK2) IN COMPLEX WITH NON- SELECTIVE INHIBITOR | GLY-RICH LOOP FORMED, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3wi6:D (CYS244) to (HIS322) CRYSTAL STRUCTURE OF MAPKAP KINASE-2 (MK2) IN COMPLEX WITH NON- SELECTIVE INHIBITOR | GLY-RICH LOOP FORMED, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3wi6:E (CYS244) to (HIS322) CRYSTAL STRUCTURE OF MAPKAP KINASE-2 (MK2) IN COMPLEX WITH NON- SELECTIVE INHIBITOR | GLY-RICH LOOP FORMED, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3wi6:F (CYS244) to (HIS322) CRYSTAL STRUCTURE OF MAPKAP KINASE-2 (MK2) IN COMPLEX WITH NON- SELECTIVE INHIBITOR | GLY-RICH LOOP FORMED, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
2x4f:A (SER281) to (HIS358) THE CRYSTAL STRUCTURE OF THE HUMAN MYOSIN LIGHT CHAIN KINASE LOC340156. | LUNG, KINASE, MYOSIN, BREAST CANCER, TRANSFERASE
2x4f:B (PRO283) to (HIS358) THE CRYSTAL STRUCTURE OF THE HUMAN MYOSIN LIGHT CHAIN KINASE LOC340156. | LUNG, KINASE, MYOSIN, BREAST CANCER, TRANSFERASE
2x4z:A (GLY493) to (HIS569) CRYSTAL STRUCTURE OF THE HUMAN P21-ACTIVATED KINASE 4 IN COMPLEX WITH PF-03758309 | TRANSFERASE, NUCLEOTIDE-BINDING ATP-BINDING, PHOSPHOPROTEIN
2xbj:A (ALA402) to (HIS483) CRYSTAL STRUCTURE OF CHK2 IN COMPLEX WITH AN INHIBITOR | TRANSFERASE, DNA REPAIR, PARP
1vjy:A (GLU394) to (GLU499) CRYSTAL STRUCTURE OF A NAPHTHYRIDINE INHIBITOR OF HUMAN TGF- BETA TYPE I RECEPTOR | TRANSFERASE, PROTEIN KINASE, INHIBITOR COMPLEX
4mx9:A (ASP227) to (HIS304) CDPK1 FROM NEOSPORA CANINUM IN COMPLEX WITH INHIBITOR UW1294 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4mxa:A (CYS230) to (HIS304) CDPK1 FROM NEOSPORA CANINUM IN COMPLEX WITH INHIBITOR RM-1-132 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2xm8:A (ALA402) to (HIS483) CO-CRYSTAL STRUCTURE OF A SMALL MOLECULE INHIBITOR BOUND TO THE KINASE DOMAIN OF CHK2 | TRANSFERASE, CANCER
2jam:A (SER198) to (HIS275) CRYSTAL STRUCTURE OF HUMAN CALMODULIN-DEPENDENT PROTEIN KINASE I G | TRANSFERASE, KINASE, MEMBRANE, ATP-BINDING, PRENYLATION, SERINE/THREONINE-PROTEIN KINASE, ALTERNATIVE SPLICING, PROTEIN SERINE/THREONINE KINASE, CALMODULIN BINDING, CALMODULIN-BINDING, NUCLEOTIDE BINDING, NUCLEOTIDE-BINDING, LIPOPROTEIN, POLYMORPHISM, GOLGI APPARATUS, PHOSPHORYLATION, ALLOSTERIC ENZYME
2jam:B (SER198) to (HIS275) CRYSTAL STRUCTURE OF HUMAN CALMODULIN-DEPENDENT PROTEIN KINASE I G | TRANSFERASE, KINASE, MEMBRANE, ATP-BINDING, PRENYLATION, SERINE/THREONINE-PROTEIN KINASE, ALTERNATIVE SPLICING, PROTEIN SERINE/THREONINE KINASE, CALMODULIN BINDING, CALMODULIN-BINDING, NUCLEOTIDE BINDING, NUCLEOTIDE-BINDING, LIPOPROTEIN, POLYMORPHISM, GOLGI APPARATUS, PHOSPHORYLATION, ALLOSTERIC ENZYME
2jbo:A (TYR240) to (HIS322) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-1, SOAKING) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, MK2, KINASE, ATP SITE, TRANSFERASE, ATP-BINDING, SERINE/THREONINE-PROTEIN KINASE, SMALL MOLECULE INHIBITOR, NUCLEOTIDE-BINDING
2jbp:A (TYR240) to (HIS322) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:B (TYR240) to (HIS322) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:E (TYR240) to (HIS322) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:F (TYR240) to (HIS322) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:G (TYR240) to (HIS322) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:H (TYR240) to (HIS322) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:I (TYR240) to (HIS322) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:K (SER243) to (HIS322) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jbp:L (SER243) to (HIS322) PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-2, CO-CRYSTALLIZATION) | SER-THR KINASE, MAPKAP KINASE 2, PHOSPHORYLATION, SMALL MOLECULE INHIBITOR, MK2, KINASE, ATP SITE, TRANSFERASE, ATP- BINDING, SERINE/THREONINE-PROTEIN KINASE, CO- CRYSTALLIZATION, NUCLEOTIDE-BINDING
2jc6:A (SER199) to (HIS276) CRYSTAL STRUCTURE OF HUMAN CALMODULIN-DEPENDENT PROTEIN KINASE 1D | TRANSFERASE, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION
2jc6:C (SER199) to (HIS276) CRYSTAL STRUCTURE OF HUMAN CALMODULIN-DEPENDENT PROTEIN KINASE 1D | TRANSFERASE, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION
1kob:A (TYR230) to (HIS305) TWITCHIN KINASE FRAGMENT (APLYSIA), AUTOREGULATED PROTEIN KINASE DOMAIN | KINASE, TWITCHIN, INTRASTERIC REGULATION
1kob:B (PHE229) to (HIS305) TWITCHIN KINASE FRAGMENT (APLYSIA), AUTOREGULATED PROTEIN KINASE DOMAIN | KINASE, TWITCHIN, INTRASTERIC REGULATION
4o0r:B (GLY442) to (HIS518) BACK POCKET FLEXIBILITY PROVIDES GROUP-II PAK SELECTIVITY FOR TYPE 1 KINASE INHIBITORS | PAK1, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4o0t:B (LYS444) to (HIS518) BACK POCKET FLEXIBILITY PROVIDES GROUP-II PAK SELECTIVITY FOR TYPE 1 KINASE INHIBITORS | PAK1, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ona:A (CYS231) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1517 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3kcf:A (GLU394) to (GLN498) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A PYRAZOLONE INHIBITOR | KINASE, TGFBETARI, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, AORTIC ANEURYSM, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3kcf:B (GLU394) to (GLY500) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A PYRAZOLONE INHIBITOR | KINASE, TGFBETARI, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, AORTIC ANEURYSM, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3kcf:C (GLU394) to (GLY500) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A PYRAZOLONE INHIBITOR | KINASE, TGFBETARI, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, AORTIC ANEURYSM, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3kcf:D (GLU394) to (GLY500) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH A PYRAZOLONE INHIBITOR | KINASE, TGFBETARI, STRUCTURE-BASED DRUG DESIGN, PROTEIN- INHIBITOR COMPLEX, AORTIC ANEURYSM, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
4a9u:A (ALA402) to (HIS483) CRYSTAL STRUCTURE OF HUMAN CHK2 IN COMPLEX WITH BENZIMIDAZOLE CARBOXAMIDE INHIBITOR | TRANSFERASE
3kk8:A (SER190) to (VAL267) CAMKII SUBSTRATE COMPLEX A | PROTEIN KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kk9:A (PRO192) to (VAL267) CAMKII SUBSTRATE COMPLEX B | CAMKII, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
3kl8:A (SER190) to (VAL267) CAMKIINTIDE INHIBITOR COMPLEX | CAMKII, CAMKIINTIDE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL JUNCTION, CELL MEMBRANE, MEMBRANE, POSTSYNAPTIC CELL MEMBRANE, PROTEIN KINASE INHIBITOR, SYNAPSE, SYNAPTOSOME, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3kl8:C (SER190) to (VAL267) CAMKIINTIDE INHIBITOR COMPLEX | CAMKII, CAMKIINTIDE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL JUNCTION, CELL MEMBRANE, MEMBRANE, POSTSYNAPTIC CELL MEMBRANE, PROTEIN KINASE INHIBITOR, SYNAPSE, SYNAPTOSOME, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3kl8:E (PRO192) to (VAL267) CAMKIINTIDE INHIBITOR COMPLEX | CAMKII, CAMKIINTIDE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL JUNCTION, CELL MEMBRANE, MEMBRANE, POSTSYNAPTIC CELL MEMBRANE, PROTEIN KINASE INHIBITOR, SYNAPSE, SYNAPTOSOME, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3kl8:G (SER190) to (VAL267) CAMKIINTIDE INHIBITOR COMPLEX | CAMKII, CAMKIINTIDE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL JUNCTION, CELL MEMBRANE, MEMBRANE, POSTSYNAPTIC CELL MEMBRANE, PROTEIN KINASE INHIBITOR, SYNAPSE, SYNAPTOSOME, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3kl8:I (PRO192) to (VAL267) CAMKIINTIDE INHIBITOR COMPLEX | CAMKII, CAMKIINTIDE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, CELL JUNCTION, CELL MEMBRANE, MEMBRANE, POSTSYNAPTIC CELL MEMBRANE, PROTEIN KINASE INHIBITOR, SYNAPSE, SYNAPTOSOME, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3kn5:A (SER602) to (GLN688) CRYSTAL STRUCTURE OF THE C-TERMINAL KINASE DOMAIN OF MSK1 IN COMPLEX WITH AMP-PNP | KINASE, AMP-PNP, MSK1, MSK, ATP-BINDING, METAL-BINDING, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kn5:B (SER602) to (ASN684) CRYSTAL STRUCTURE OF THE C-TERMINAL KINASE DOMAIN OF MSK1 IN COMPLEX WITH AMP-PNP | KINASE, AMP-PNP, MSK1, MSK, ATP-BINDING, METAL-BINDING, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kn6:A (SER602) to (ASN684) CRYSTAL STRUCTURE OF THE C-TERMINAL KINASE DOMAIN OF MSK1 | KINASE, AMP-PNP, MSK1, MSK, ATP-BINDING, METAL-BINDING, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kn6:B (SER602) to (ASN684) CRYSTAL STRUCTURE OF THE C-TERMINAL KINASE DOMAIN OF MSK1 | KINASE, AMP-PNP, MSK1, MSK, ATP-BINDING, METAL-BINDING, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4p90:A (GLY442) to (HIS518) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN PAK1 IN COMPLEX WITH COMPOUND 15 | INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4p90:B (GLY442) to (HIS518) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF HUMAN PAK1 IN COMPLEX WITH COMPOUND 15 | INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1yhw:A (VAL445) to (HIS518) CRYSTAL STRUCTURE OF PAK1 KINASE DOMAIN WITH ONE POINT MUTATIONS (K299R) | KINASE; ACTIVE CONFORMATION; ACTIVATION LOOP; ATP BINDING SITE, SIGNALING PROTEIN, TRANSFERASE
5dew:B (GLY442) to (HIS518) CRYSTAL STRUCTURE OF PAK1 IN COMPLEX WITH AN INHIBITOR COMPOUND 5 | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5dfp:A (VAL445) to (HIS518) CRYSTAL STRUCTURE OF PAK1 IN COMPLEX WITH AN INHIBITOR COMPOUND FRAX1036 | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4pwn:A (SER402) to (HIS476) CRYSTAL STRUCTURE OF ACTIVE WNK1 KINASE | KINASE, WNK1, SER/THR PROTEIN KINASE, SERINE/THREONINE KINASE, ATP- BINDING, PHOSPHORYLATION, TRANSFERASE
5dvr:A (CYS231) to (HIS305) CRYSTAL STRUCTURE OF TGCDPK1 FROM TOXOPLASMA GONDII COMPLEXED WITH GW780159X | STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPKS, SERINE/THREONINE PROTEIN KINASE, NUCLEOTIDE-BINDING, GW780159X, TRANSFERASE
4asx:A (GLN378) to (LEU485) CRYSTAL STRUCTURE OF ACTIVIN RECEPTOR TYPE-IIA (ACVR2A) KINASE DOMAIN IN COMPLEX WITH DIHYDRO-BAUERINE C | TRANSFERASE, PROTEIN KINASE
4asx:B (ARG379) to (LEU485) CRYSTAL STRUCTURE OF ACTIVIN RECEPTOR TYPE-IIA (ACVR2A) KINASE DOMAIN IN COMPLEX WITH DIHYDRO-BAUERINE C | TRANSFERASE, PROTEIN KINASE
5e8v:A (VAL439) to (LEU541) TGF-BETA RECEPTOR TYPE 2 KINASE DOMAIN (E431A,R433A,E485A,K488A,R493A, R495A) | KINASE DOMAIN, TRANSFERASE
5e91:A (GLU440) to (GLU540) TGF-BETA RECEPTOR TYPE 2 KINASE DOMAIN (E431A,R433A,E485A,K488A,R493A, R495A) IN COMPLEX WITH 3-AMINO-6-[4-(2- HYDROXYETHYL)PHENYL]-N-[4- (MORPHOLIN-4-YL)PYRIDIN-3-YL] PYRAZINE-2-CARBOXAMIDE | KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5e92:A (GLU440) to (GLU540) TGF-BETA RECEPTOR TYPE 2 KINASE DOMAIN (E431A,R433A,E485A,K488A,R493A, R495A) IN COMPLEX WITH AMPPNP | KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3mft:A (PRO199) to (HIS273) CASK-4M CAM KINASE DOMAIN, MN2+ | CATALYTIC MECHANISM, KINASE CATALYSIS, MG2+-MEDIATED PHOSPHATE TRANSFER, PROTEIN KINASE, TRANSFERASE
3mfu:A (PRO199) to (HIS273) CASK-4M CAM KINASE DOMAIN, AMPPNP-MN2+ | CATALYTIC MECHANISM, KINASE CATALYSIS, MG2+-MEDIATED PHOSPHATE TRANSFER, PROTEIN KINASE, TRANSFERASE
3my0:D (GLU391) to (LYS491) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:F (GLU391) to (SER493) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:U (GLU391) to (SER493) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3c0i:A (PRO199) to (HIS273) CASK CAM-KINASE DOMAIN- 3'-AMP COMPLEX, P212121 FORM | CASK, NEUREXIN, CA2+/CALMODULIN DEPENDENT PROTEIN KINASE, MG2+, SYNAPTIC PLASTICITY, PSEUDOKINASE, MAGUK, MEMBRANE-ASSOCIATED GUANYLATE KINASE, ATP-BINDING, CALMODULIN-BINDING, MAGNESIUM, METAL- BINDING, NUCLEOTIDE-BINDING, NUCLEUS, SERINE/THREONINE-PROTEIN KINASE, SH3 DOMAIN, TRANSFERASE
3n51:A (ASP228) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR RM-1-95 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, BUMPED KINASE INHIBITOR, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ncg:A (LYS254) to (HIS329) ACTIVATED CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM CRYPTOSPORIDIUM PARVUM (CPCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR NM-PP1 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, BUMPED KINASE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP
4rgj:A (ASP248) to (HIS325) APO CRYSTAL STRUCTURE OF CDPK4 FROM PLASMODIUM FALCIPARUM, PF3D7_0717500 | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPK, MALARIA, TRANSFERASE
3com:B (CYS203) to (HIS278) CRYSTAL STRUCTURE OF MST1 KINASE | KINASE, MST1, SERINE/THREONINE-PROTEIN KINASE 4, STE20-LIKE KINASE, PSI, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ALTERNATIVE SPLICING, APOPTOSIS, ATP- BINDING, COILED COIL, CYTOPLASM, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, TRANSFERASE
3nyv:A (ASP228) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH NON-SPECIFIC INHIBITOR WHI-P180 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3dfa:A (CYS186) to (HIS260) CRYSTAL STRUCTURE OF KINASE DOMAIN OF CALCIUM-DEPENDENT PROTEIN KINASE CGD3_920 FROM CRYPTOSPORIDIUM PARVUM | CALMODULIN, KINASE, MALARIA, TRANSFERASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
4tzr:A (ASP228) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1561 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE
4d9t:A (ALA586) to (HIS676) RSK2 C-TERMINAL KINASE DOMAIN WITH INHIBITOR (E)-METHYL 3-(4-AMINO-7- (3-HYDROXYPROPYL)-5-P-TOLYL-7H-PYRROLO[2,3-D]PYRIMIDIN-6-YL)-2- CYANOACRYLATE | KINASE, INHIBITOR, REVERSIBLE, THIOL, PHOSPHORYLATION, MIGRATION,, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3dxn:A (CYS203) to (HIS277) CRYSTAL STRUCTURE OF THE CALCIUM-DEPENDENT KINASE FROM TOXOPLASMA GONDII, 541.M00134, KINASE DOMAIN. | CDPK, CALCIUM DEPENDENT KINASE, CALMODULIN, PARASITE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, TRANSFERASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
5ime:A (VAL445) to (HIS518) CRYSTAL STRUCTURE OF P21-ACTIVATED KINASE 1 (PAK1) IN COMPLEX WITH COMPOUND 9 | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ime:B (GLY442) to (HIS518) CRYSTAL STRUCTURE OF P21-ACTIVATED KINASE 1 (PAK1) IN COMPLEX WITH COMPOUND 9 | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4eqc:A (VAL445) to (HIS518) CRYSTAL STRUCTURE OF PAK1 KINASE DOMAIN IN COMPLEX WITH FRAX597 INHIBITOR | SERINE/THREONINE KINASE, PHOSPHORYLATION, ATP-BINDING, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3q4t:B (GLN378) to (LEU485) CRYSTAL STRUCTURE OF ACTIVIN RECEPTOR TYPE-IIA (ACVR2A) KINASE DOMAIN IN COMPLEX WITH DORSOMORPHIN | STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, TRANSFERASE
3q4u:A (ASP397) to (ASP499) CRYSTAL STRUCTURE OF THE ACVR1 KINASE DOMAIN IN COMPLEX WITH LDN- 193189 | STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, TRANSFERASE
3q4z:A (GLY442) to (HIS518) STRUCTURE OF UNPHOSPHORYLATED PAK1 KINASE DOMAIN | KINASE DOMAIN, SIGNALLING PATHWAY, TRANSFERASE
3q52:A (VAL445) to (HIS518) STRUCTURE OF PHOSPHORYLATED PAK1 KINASE DOMAIN | KINASE DOMAIN, SIGNALLING PATHWAY, TRANSFERASE
3q53:A (GLY442) to (HIS518) STRUCTURE OF PHOSPHORYLATED PAK1 KINASE DOMAIN IN COMPLEX WITH ATP | KINASE DOMAIN, SIGNALLING PATHWAY, TRANSFERASE
4fg7:A (ALA198) to (HIS273) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE I 1-293 IN COMPLEX WITH ATP | CAMK, CALMODULIN, AUTOINHIBITION, REGULATION MECHANISM, KINASE, TRANSFERASE
4fg8:A (SER196) to (HIS273) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE I 1-315 IN COMPLEX WITH ATP | CAMK, CALMODULIN, AUTOINHIBITION, REGULATION MECHANISM, KINASE, TRANSFERASE
4fg8:B (SER196) to (HIS273) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE I 1-315 IN COMPLEX WITH ATP | CAMK, CALMODULIN, AUTOINHIBITION, REGULATION MECHANISM, KINASE, TRANSFERASE
4fg9:A (SER196) to (HIS273) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE I 1-320 IN COMPLEX WITH ATP | CAMK, CALMODULIN, AUTOINHIBITION, REGULATION MECHANISM, KINASE, TRANSFERASE
4fg9:B (SER196) to (HIS273) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE I 1-320 IN COMPLEX WITH ATP | CAMK, CALMODULIN, AUTOINHIBITION, REGULATION MECHANISM, KINASE, TRANSFERASE
4fgb:A (ALA198) to (HIS273) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE I APO FORM | CAMK, CALMODULIN, AUTOINHIBITION, REGULATION MECHANISM, KINASE, TRANSFERASE
4fif:A (GLY493) to (HIS569) CATALYTIC DOMAIN OF HUMAN PAK4 WITH RPKPLVDP PEPTIDE | SERINE/THREONINE-PROTEIN KINASE PAK4, KINASE DOMAIN, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-PEPTIDE COMPLEX
4fih:A (GLY493) to (HIS569) CATALYTIC DOMAIN OF HUMAN PAK4 WITH QKFTGLPRQW PEPTIDE | SERINE/THREONINE-PROTEIN KINASE PAK4, KINASE DOMAIN, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
4fii:A (GLY493) to (HIS569) CATALYTIC DOMAIN OF HUMAN PAK4 WITH RPKPLVDP PEPTIDE | SERINE/THREONINE-PROTEIN KINASE PAK4, KINASE DOMAIN, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-PEPTIDE COMPLEX
5jms:A (ASP228) to (HIS305) CRYSTAL STRUCTURE OF TGCDPK1 BOUND TO CGP060476 | KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, HYDROLASE
5jzj:A (ASP569) to (HIS644) CRYSTAL STRUCTURE OF DCLK1-KD IN COMPLEX WITH AMPPN | KINASE, DOUBLECORTIN, TRANSFERASE
5jzj:B (ASP569) to (HIS644) CRYSTAL STRUCTURE OF DCLK1-KD IN COMPLEX WITH AMPPN | KINASE, DOUBLECORTIN, TRANSFERASE
5kbq:A (GLY442) to (HIS518) PAK1 IN COMPLEX WITH BIS-ANILINO PYRIMIDINE INHIBITOR | SERINE/THREONINE-PROTEIN KINASE PAK1, KINASE, TRANSFERASE
5t6a:A (ASP228) to (HIS305) CRYSTAL STRUCTURE OF TGCDPK1 FROM TOXOPLASMA GONDII COMPLEXED WITH 5GA | STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPKS, SERINE/THREONINE PROTEIN KINASE, NUCLEOTIDE-BINDING, TRANSFERASE
5t6i:A (CYS231) to (HIS305) CRYSTAL STRUCTURE OF TGCDPK1 FROM TOXOPLASMA GONDII COMPLEXED WITH 5GB | STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPKS, SERINE/THREONINE PROTEIN KINASE, NUCLEOTIDE-BINDING, TRANSFERASE
5t6k:A (ASP228) to (HIS305) CRYSTAL STRUCTURE OF TGCDPK1 FROM TOXOPLASMA GONDII COMPLEXED WITH GW780159X | STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPKS, SERINE/THREONINE PROTEIN KINASE, NUCLEOTIDE-BINDING, TRANSFERASE
4wg5:A (LYS230) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1647 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1nxk:A (TYR240) to (HIS322) CRYSTAL STRUCTURE OF STAUROSPORINE BOUND TO MAP KAP KINASE 2 | PROTEIN KINASE, MK2, PHOSPHORYLATION, STAUROSPORINE, TRANSFERASE
1nxk:B (TYR240) to (HIS322) CRYSTAL STRUCTURE OF STAUROSPORINE BOUND TO MAP KAP KINASE 2 | PROTEIN KINASE, MK2, PHOSPHORYLATION, STAUROSPORINE, TRANSFERASE
1nxk:D (TYR240) to (HIS322) CRYSTAL STRUCTURE OF STAUROSPORINE BOUND TO MAP KAP KINASE 2 | PROTEIN KINASE, MK2, PHOSPHORYLATION, STAUROSPORINE, TRANSFERASE
3sxf:A (CYS231) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH BUMPED KINASE INHIBITOR, RM-1-89 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4jg6:A (ALA586) to (HIS676) RSK2 CTD BOUND TO 2-CYANO-3-(1H-INDAZOL-5-YL)ACRYLAMIDE | PROTEIN KINASE, PHOSPHORYLATION, COVALENT INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4yga:A (CYS231) to (HIS305) CDPK1, FROM TOXOPLASMA GONDII, BOUND TO INHIBITORY VHH-1B7 | SERINE/THREONINE PROTEIN KINASE, VHH DOMAIN, INHIBITOR, METAL BINDING PROTEIN
4yga:C (CYS231) to (HIS305) CDPK1, FROM TOXOPLASMA GONDII, BOUND TO INHIBITORY VHH-1B7 | SERINE/THREONINE PROTEIN KINASE, VHH DOMAIN, INHIBITOR, METAL BINDING PROTEIN
4yga:E (ASP228) to (HIS305) CDPK1, FROM TOXOPLASMA GONDII, BOUND TO INHIBITORY VHH-1B7 | SERINE/THREONINE PROTEIN KINASE, VHH DOMAIN, INHIBITOR, METAL BINDING PROTEIN
3upx:A (ASP228) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1300 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3i79:A (ASP228) to (HIS305) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) | PROTEIN KINASE, CALMODULIN, EF HAND, BUMPED KINASE INHIBITOR, ATP- BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, TRANSFERASE
2vz6:A (PRO193) to (HIS268) STRUCTURE OF HUMAN CALCIUM CALMODULIN DEPENDENT PROTEIN KINASE TYPE II ALPHA (CAMK2A) IN COMPLEX WITH INDIRUBIN E804 | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, CELL JUNCTION, CELL MEMBRANE, LONG TERM POTENTIATION, BRAIN, KINASE, SYNAPSE, MEMBRANE, NMDA RECEPTOR SIGNALLING, PHOSPHOPROTEIN, CALMODULIN-BINDING, NUCLEOTIDE-BINDING
2vz6:B (PRO193) to (HIS268) STRUCTURE OF HUMAN CALCIUM CALMODULIN DEPENDENT PROTEIN KINASE TYPE II ALPHA (CAMK2A) IN COMPLEX WITH INDIRUBIN E804 | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, CELL JUNCTION, CELL MEMBRANE, LONG TERM POTENTIATION, BRAIN, KINASE, SYNAPSE, MEMBRANE, NMDA RECEPTOR SIGNALLING, PHOSPHOPROTEIN, CALMODULIN-BINDING, NUCLEOTIDE-BINDING
2w4o:A (GLY219) to (HIS297) CRYSTAL STRUCTURE OF HUMAN CAMK4 IN COMPLEX WITH 4-AMINO( SULFAMOYL-PHENYLAMINO)-TRIAZOLE-CARBOTHIOIC ACID (2,6- DIFLUORO-PHENYL)-AMIDE) | CALMODULIN-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHOPROTEIN, KINASE, NUCLEUS, TRANSFERASE
4lg4:B (CYS200) to (HIS275) STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5 | HIPPO, MST AUTOACTIVATION, DIMERIZATION, SIGNALING PROTEIN
4lg4:D (ASN199) to (HIS275) STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5 | HIPPO, MST AUTOACTIVATION, DIMERIZATION, SIGNALING PROTEIN
4lg4:F (ASN199) to (HIS275) STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5 | HIPPO, MST AUTOACTIVATION, DIMERIZATION, SIGNALING PROTEIN
4zy6:A (GLY442) to (HIS518) CRYSTAL STRUCTURE OF P21-ACTIVATED KINASE 1 IN COMPLEX WITH AN INHIBITOR COMPOUND 29 | PAK1, KINASE, INHIBITOR, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4zy6:B (GLY442) to (HIS518) CRYSTAL STRUCTURE OF P21-ACTIVATED KINASE 1 IN COMPLEX WITH AN INHIBITOR COMPOUND 29 | PAK1, KINASE, INHIBITOR, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2hy8:1 (GLY442) to (HIS518) PAK1 COMPLEX WITH ST2001 | TYPICAL FOLD OF SER/THR KINASES. INHIBITOR IS BOUND BETWEEN THE N-TERMINAL AND C-TERMINAL DOMAINS., TRANSFERASE
4m97:A (ASP227) to (HIS304) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM NEOSPORA CANINUM | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING
2x7o:A (GLU394) to (GLY500) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH AN INDOLINONE INHIBITOR | KINASE, TRANSFERASE, GLYCOPROTEIN
2x7o:B (GLU394) to (GLY500) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH AN INDOLINONE INHIBITOR | KINASE, TRANSFERASE, GLYCOPROTEIN
2x7o:D (GLU394) to (GLN497) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH AN INDOLINONE INHIBITOR | KINASE, TRANSFERASE, GLYCOPROTEIN
2x7o:E (GLU394) to (GLY500) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH AN INDOLINONE INHIBITOR | KINASE, TRANSFERASE, GLYCOPROTEIN
3kc3:A (TYR240) to (HIS322) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:B (TYR240) to (HIS322) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:D (TYR240) to (HIS322) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:E (TYR240) to (HIS322) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:F (TYR240) to (HIS322) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:G (TYR240) to (HIS322) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:H (CYS244) to (HIS322) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:I (TYR240) to (HIS322) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:J (TYR240) to (HIS322) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3kc3:L (TYR240) to (HIS322) MK2 COMPLEXED TO INHIBITOR N4-(7-(BENZOFURAN-2-YL)-1H-INDAZOL-5-YL) PYRIMIDINE-2,4-DIAMINE | MAPKAP-K2, MK2, TNFALPHA, DIAMINOPYRIMIDINE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:A (SER243) to (HIS322) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:B (TYR240) to (HIS322) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:C (TYR240) to (HIS322) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:D (TYR240) to (HIS322) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:F (TYR240) to (HIS322) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:G (TYR240) to (HIS322) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:I (TYR240) to (HIS322) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:J (SER243) to (HIS322) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3a2c:L (TYR240) to (HIS322) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR COMPLEX BOUND TO MAPKAP KINASE-2 (MK2) | GLY-RICH LOOP FORMED, AIPHA-HELIX, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4pds:A (SER387) to (HIS463) CRYSTAL STRUCTURE OF RAD53 KINASE DOMAIN AND SCD2 IN COMPLEX WITH AMPPNP | KINASE DOMAIN, ANP, C-LOBE, ACTIVATION SEGMENT EXCHANGE, TRANSFERASE
4pds:B (ASN383) to (HIS463) CRYSTAL STRUCTURE OF RAD53 KINASE DOMAIN AND SCD2 IN COMPLEX WITH AMPPNP | KINASE DOMAIN, ANP, C-LOBE, ACTIVATION SEGMENT EXCHANGE, TRANSFERASE
5dey:A (VAL445) to (HIS518) CRYSTAL STRUCTURE OF PAK1 IN COMPLEX WITH AN INHIBITOR COMPOUND G-5555 | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5e8x:A (GLU394) to (GLU499) TGF-BETA RECEPTOR TYPE 1 KINASE DOMAIN (T204D,I211V,Y249F,S280T, Y282F,S287N,A350C,L352F) IN COMPLEX WITH STAUROSPORINE | ALK5, KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3mfs:A (PRO199) to (HIS273) CASK-4M CAM KINASE DOMAIN, AMPPNP | CATALYTIC MECHANISM, KINASE CATALYSIS, MG2+-MEDIATED PHOSPHATE TRANSFER, PROTEIN KINASE, TRANSFERASE
4qox:A (ASP248) to (HIS325) CRYSTAL STRUCTURE OF CDPK4 FROM PLASMODIUM FALCIPARUM, PF3D7_0717500 | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPK, PLASMODIUM, MALARIA, TRANSFERASE
3bhh:A (PRO194) to (HIS269) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE IIB ISOFORM 1 (CAMK2B) | CAMK2B, CAM2, CAMK2, CAM KINASE II BETA CHAIN, CAMK II BETA SUBUNIT, CALCIUM/CALMODULION DEPENDENT PROTEIN KINASE II BETA, EC:2.7.1.123, MGC29528, PROLINE RICH CALMODULIN DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, CALMODULIN- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
3bhh:B (PRO194) to (HIS269) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE IIB ISOFORM 1 (CAMK2B) | CAMK2B, CAM2, CAMK2, CAM KINASE II BETA CHAIN, CAMK II BETA SUBUNIT, CALCIUM/CALMODULION DEPENDENT PROTEIN KINASE II BETA, EC:2.7.1.123, MGC29528, PROLINE RICH CALMODULIN DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, CALMODULIN- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
3bhh:C (PRO194) to (HIS269) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE IIB ISOFORM 1 (CAMK2B) | CAMK2B, CAM2, CAMK2, CAM KINASE II BETA CHAIN, CAMK II BETA SUBUNIT, CALCIUM/CALMODULION DEPENDENT PROTEIN KINASE II BETA, EC:2.7.1.123, MGC29528, PROLINE RICH CALMODULIN DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, CALMODULIN- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
3bhh:D (PRO194) to (HIS269) CRYSTAL STRUCTURE OF HUMAN CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE IIB ISOFORM 1 (CAMK2B) | CAMK2B, CAM2, CAMK2, CAM KINASE II BETA CHAIN, CAMK II BETA SUBUNIT, CALCIUM/CALMODULION DEPENDENT PROTEIN KINASE II BETA, EC:2.7.1.123, MGC29528, PROLINE RICH CALMODULIN DEPENDENT PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, CALMODULIN- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
4daw:A (VAL445) to (HIS518) CRYSTAL STRUCTURE OF PAK1 KINASE DOMAIN WITH THE RUTHENIUM PHTHALIMIDE COMPLEX | SERINE/THREONINE KINASE, PHOSPHORYLATION, ATP-BINDING, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5ig1:A (ALA197) to (HIS272) CRYSTAL STRUCTURE OF S. ROSETTA CAMKII KINASE DOMAIN | CA2+/CAM-DEPENDENT KINASE, CHOANOFLAGELLATE, TRANSFERASE
3r2b:A (TYR240) to (HIS322) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:B (TYR240) to (HIS322) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:C (TYR240) to (HIS322) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:D (TYR240) to (HIS322) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:E (TYR240) to (HIS322) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:F (TYR240) to (HIS322) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:G (TYR240) to (HIS322) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:H (SER243) to (HIS322) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:I (TYR240) to (HIS322) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:J (TYR240) to (HIS322) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:K (TYR240) to (HIS322) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2b:L (TYR240) to (HIS322) MK2 KINASE BOUND TO COMPOUND 5B | KINASE DOMAIN WITH BOUND INHIBITOR, KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r2y:A (ASP241) to (HIS322) MK2 KINASE BOUND TO COMPOUND 1 | KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5jzn:A (ASP569) to (HIS644) CRYSTAL STRUCTURE OF DCLK1-KD IN COMPLEX WITH NVP-TAE684 | KINASE, DOUBLECORTIN, TRANSFERASE
5jzn:B (ASP569) to (HIS644) CRYSTAL STRUCTURE OF DCLK1-KD IN COMPLEX WITH NVP-TAE684 | KINASE, DOUBLECORTIN, TRANSFERASE