2o9i:A (GLU321) to (LEU428) CRYSTAL STRUCTURE OF THE HUMAN PREGNANE X RECEPTOR LBD IN COMPLEX WITH AN SRC-1 COACTIVATOR PEPTIDE AND T0901317 | NUCLEAR RECEPTOR, PREGNANE X RECEPTOR, PXR, T0901317, TRANSCRIPTION
2o9i:B (PRO1322) to (PHE1429) CRYSTAL STRUCTURE OF THE HUMAN PREGNANE X RECEPTOR LBD IN COMPLEX WITH AN SRC-1 COACTIVATOR PEPTIDE AND T0901317 | NUCLEAR RECEPTOR, PREGNANE X RECEPTOR, PXR, T0901317, TRANSCRIPTION
1n83:A (GLU397) to (PHE511) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN THE ORPHAN NUCLEAR HORMONE RECEPTOR ROR(ALPHA)-LBD AND CHOLESTEROL | THREE-LAYERED ALPHA HELICAL SANDWICH, RECEPTOR, TRANSCRIPTION REGULATION, NUCLEAR PROTEIN, DNA BINDING, LIPID BINDING PROTEIN
2ao6:A (MET780) to (SER888) CRYSTAL STRUCTURE OF THE HUMAN ANDROGEN RECEPTOR LIGAND BINDING DOMAIN BOUND WITH TIF2(III) 740-753 PEPTIDE AND R1881 | CRYSTAL STRUCTURE; HUMAN ANDROGEN RECEPTOR LIGAND BINDING DOMAIN; TRANSCRIPTIONAL INTERMEDIARY FACTOR 2 740-753; R188
2ath:A (LYS358) to (TYR473) CRYSTAL STRUCTURE OF THE LIGAND BINDING DOMAIN OF HUMAN PPAR-GAMMA IM COMPLEX WITH AN AGONIST | PPAR, TRANSCRIPTION
2om9:A (ARG357) to (TYR473) AJULEMIC ACID, A SYNTHETIC CANNABINOID BOUND TO PPAR GAMMA | PPAR GAMMA, AJULEMIC ACID, CANNABINOID, PARTIAL AGONIST, TRANSCRIPTION
2om9:B (MET364) to (TYR473) AJULEMIC ACID, A SYNTHETIC CANNABINOID BOUND TO PPAR GAMMA | PPAR GAMMA, AJULEMIC ACID, CANNABINOID, PARTIAL AGONIST, TRANSCRIPTION
2om9:C (ARG357) to (TYR473) AJULEMIC ACID, A SYNTHETIC CANNABINOID BOUND TO PPAR GAMMA | PPAR GAMMA, AJULEMIC ACID, CANNABINOID, PARTIAL AGONIST, TRANSCRIPTION
2om9:D (MET364) to (TYR473) AJULEMIC ACID, A SYNTHETIC CANNABINOID BOUND TO PPAR GAMMA | PPAR GAMMA, AJULEMIC ACID, CANNABINOID, PARTIAL AGONIST, TRANSCRIPTION
2awh:A (LYS358) to (TYR473) HUMAN NUCLEAR RECEPTOR-LIGAND COMPLEX 1 | NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, PPAR, GENE REGULATION
2awh:B (LYS358) to (TYR473) HUMAN NUCLEAR RECEPTOR-LIGAND COMPLEX 1 | NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, PPAR, GENE REGULATION
2b1v:A (MET421) to (ARG548) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH OBCP-1M AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
2b1v:B (MET421) to (ASP545) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH OBCP-1M AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
2b1z:A (MET421) to (ARG548) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH 17METHYL-17ALPHA-DIHYDROEQUILENIN AND A GLUCOC INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
2b1z:B (MET421) to (LEU544) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH 17METHYL-17ALPHA-DIHYDROEQUILENIN AND A GLUCOC INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
2b23:A (MET421) to (ARG548) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN AND A GLUCOCORTICOID RECEPTOR-INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
2b23:B (GLU419) to (ALA546) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN AND A GLUCOCORTICOID RECEPTOR-INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
1nrl:A (GLU321) to (LEU428) CRYSTAL STRUCTURE OF THE HUMAN PXR-LBD IN COMPLEX WITH AN SRC-1 COACTIVATOR PEPTIDE AND SR12813 | NUCLEAR RECEPTOR, COACTIVATOR, PXR, XENOBIOTIC, SRC-1, LIGAND BINDING DOMAIN, TRANSCRIPTION
2b50:A (LYS358) to (TYR473) HUMAN NUCLEAR RECEPTOR-LIGAND COMPLEX 2 | NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, PPAR, GENE REGULATION
2b50:B (LYS358) to (TYR473) HUMAN NUCLEAR RECEPTOR-LIGAND COMPLEX 2 | NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, PPAR, GENE REGULATION
2ouz:A (MET421) to (MET543) CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR ALPHA-LASOFOXIFENE COMPLEX | NUCLEAR RECEPTOR, SERM, ESTROGEN, HORMONE-GROWTH FACTOR COMPLEX
1nuo:A (VAL348) to (PHE459) TWO RTH MUTANTS WITH IMPAIRED HORMONE BINDING | ALPHA HELIX, NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
2oz7:A (TYR781) to (GLN902) CRYSTAL STRUCTURE OF THE HUMAN ANDROGEN RECEPTOR T877A MUTANT LIGAND- BINDING DOMAIN WITH CYPROTERONE ACETATE | ANDROGEN RECEPTOR, ANTI-ANDROGEN, PROSTATE CANCER, HORMONE RECEPTOR
2p15:A (MET421) to (LEU544) CRYSTAL STRUCTURE OF THE ER ALPHA LIGAND BINDING DOMAIN WITH THE AGONIST ORTHO-TRIFLUOROMETHYLPHENYLVINYL ESTRADIOL | NULEAR RECEPTOR, LIGAND BINDING DOMAIN, HELIX 12, HORMONE RECEPTOR
2p15:B (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ER ALPHA LIGAND BINDING DOMAIN WITH THE AGONIST ORTHO-TRIFLUOROMETHYLPHENYLVINYL ESTRADIOL | NULEAR RECEPTOR, LIGAND BINDING DOMAIN, HELIX 12, HORMONE RECEPTOR
1nyx:B (ARG357) to (LYS474) LIGAND BINDING DOMAIN OF THE HUMAN PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR GAMMA IN COMPLEX WITH AN AGONIST | PPAR, NUCLEAR RECEPTOR, TRANSCRIPTION, GENE REGULATION, AGONIST COMPLEX
2baw:A (LYS358) to (TYR473) HUMAN NUCLEAR RECEPTOR-LIGAND COMPLEX 1 | NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, PPAR, TRANSCRIPTION
2baw:B (PHE360) to (TYR473) HUMAN NUCLEAR RECEPTOR-LIGAND COMPLEX 1 | NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, PPAR, TRANSCRIPTION
3erd:A (MET421) to (LEU549) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DIETHYLSTILBESTROL AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ESTROGEN, AGONIST, COACTIVATOR
3erd:B (MET421) to (ARG548) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DIETHYLSTILBESTROL AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ESTROGEN, AGONIST, COACTIVATOR
2p4y:A (PHE360) to (TYR473) CRYSTAL STRUCTURE OF HUMAN PPAR-GAMMA-LIGAND BINDING DOMAIN COMPLEXED WITH AN INDOLE-BASED MODULATOR | NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, LBD, ALPHA HELIX SANDWICH, PPAR-HOMODIMER, SPPARGM, PARTIAL AGONIST, TRANSCRIPTION
2p54:A (LYS349) to (TYR464) A CRYSTAL STRUCTURE OF PPAR ALPHA BOUND WITH SRC1 PEPTIDE AND GW735 | PPAR ALPHA GW735 SRC1 AGONIST HDLC, TRANSCRIPTION
3et0:A (ARG357) to (TYR473) STRUCTURE OF PPARGAMMA WITH 3-(5-METHOXY-1H-INDOL-3-YL)- PROPIONIC ACID | PPAR, PPARG, PPARGAMMA, DRUG DISCOVERY, DIABETES, ADIPONECTIN, METABOLIC DISEASE, FRAGMENT-BASED DRUG DISCOVERY, SCAFFOLD-BASED DRUG DISCOVERY, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
3et1:A (ARG348) to (ARG465) STRUCTURE OF PPARALPHA WITH 3-[5-METHOXY-1-(4-METHOXY- BENZENESULFONYL)-1H-INDOL-3-YL]-PROPIONIC ACID | PPAR, PPARA, PPARALPHA, DRUG DISCOVERY, DIABETES, ADIPONECTIN, METABOLIC DISEASE, FRAGMENT-BASED DRUG DISCOVERY, SCAFFOLD-BASED DRUG DISCOVERY, ACTIVATOR, DNA- BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACYLTRANSFERASE, ALTERNATIVE SPLICING, CHROMOSOMAL REARRANGEMENT, PHOSPHOPROTEIN, PROTO-ONCOGENE, TRANSFERASE, UBL CONJUGATION, TRANSCRIPTION/TRANSFERASE COMPLEX
3et1:B (GLU356) to (TYR464) STRUCTURE OF PPARALPHA WITH 3-[5-METHOXY-1-(4-METHOXY- BENZENESULFONYL)-1H-INDOL-3-YL]-PROPIONIC ACID | PPAR, PPARA, PPARALPHA, DRUG DISCOVERY, DIABETES, ADIPONECTIN, METABOLIC DISEASE, FRAGMENT-BASED DRUG DISCOVERY, SCAFFOLD-BASED DRUG DISCOVERY, ACTIVATOR, DNA- BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACYLTRANSFERASE, ALTERNATIVE SPLICING, CHROMOSOMAL REARRANGEMENT, PHOSPHOPROTEIN, PROTO-ONCOGENE, TRANSFERASE, UBL CONJUGATION, TRANSCRIPTION/TRANSFERASE COMPLEX
3et2:A (ILE328) to (LYS438) STRUCTURE OF PPARDELTA WITH 3-[5-METHOXY-1-(4-METHOXY- BENZENESULFONYL)-1H-INDOL-3-YL]-PROPIONIC ACID | PPAR, PPARD, PPARDELTA, DRUG DISCOVERY, DIABETES, ADIPONECTIN, METABOLIC DISEASE, FRAGMENT-BASED DRUG DISCOVERY, SCAFFOLD-BASED DRUG DISCOVERY, ACTIVATOR, ALTERNATIVE SPLICING, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, K.ZHANG, WED OCT 1 17:27:09 2008 ON NOD
3et2:B (ILE328) to (LYS438) STRUCTURE OF PPARDELTA WITH 3-[5-METHOXY-1-(4-METHOXY- BENZENESULFONYL)-1H-INDOL-3-YL]-PROPIONIC ACID | PPAR, PPARD, PPARDELTA, DRUG DISCOVERY, DIABETES, ADIPONECTIN, METABOLIC DISEASE, FRAGMENT-BASED DRUG DISCOVERY, SCAFFOLD-BASED DRUG DISCOVERY, ACTIVATOR, ALTERNATIVE SPLICING, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, K.ZHANG, WED OCT 1 17:27:09 2008 ON NOD
3et3:A (ARG357) to (TYR473) STRUCTURE OF PPARGAMMA WITH 3-[5-METHOXY-1-(4-METHOXY- BENZENESULFONYL)-1H-INDOL-3-YL]-PROPIONIC ACID | PPAR, PPARG, PPARGAMMA, DRUG DISCOVERY, DIABETES, ADIPONECTIN, METABOLIC DISEASE, FRAGMENT-BASED DRUG DISCOVERY, SCAFFOLD-BASED DRUG DISCOVERY, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACYLTRANSFERASE, CHROMOSOMAL REARRANGEMENT, PROTO-ONCOGENE, TRANSFERASE, UBL CONJUGATION
4x1g:A (GLU321) to (LEU428) CRYSTAL STRUCTURE OF THE HPXR-LBD IN COMPLEX WITH THE SYNTHETIC ESTROGEN 17ALPHA-ETHINYLESTRADIOL AND THE PESTICIDE TRANS-NONACHLOR | HORMONE RECEPTOR, ESTROGEN, PESTICIDE, GENE REGULATION
3f7d:A (SER343) to (ALA459) SF-1 LBD BOUND BY PHOSPHATIDYLCHOLINE | NUCLEAR RECEPTOR, COACTIVATOR PEPTIDE, LIGAND, PHOSPHOLIPID, PHOSPHATIDYLCHOLINE, TRANSCRIPTIONAL REGULATION, DNA-BINDING, METAL- BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER, ACTIVATOR, RNA-BINDING
3s9s:A (ARG357) to (TYR473) LIGAND BINDING DOMAIN OF PPARGAMMA COMPLEXED WITH A BENZIMIDAZOLE PARTIAL AGONIST | PPAR, NUCLEAR RECEPTOR, TRANSCRIPTION
3fal:D (GLN330) to (TRP441) HUMANRXR ALPHA & MOUSE LXR ALPHA COMPLEXED WITH RETENOIC ACID AND GSK2186 | NUCLEAR HORMONE RECEPTOR NONSTEROIDAL LXR AGONIST CHOLOESTOROL METABOLISM, DNA-BINDING, HOST-VIRUS INTERACTION, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, UBL CONJUGATION, ZINC, ZINC-FINGER, SIGNALING PROTEIN
4xao:A (PRO322) to (PHE429) CRYSTAL STRUCTURE OF THE HPXR-LBD OBTAINED IN PRESENCE OF THE PESTICIDE TRANS-NONACHLOR | HORMONE RECEPTOR, PESTICIDE, GENE REGULATION
3fc6:D (GLN330) to (TRP441) HRXRALPHA & MLXRALPHA WITH AN INDOLE PHARMACOPHORE, SB786875 | LIVER X RECEPTOR, NUCLEAR HORMONE RECEPTORS, AGONISTS, EPOXYCHOLESTEROL, DNA-BINDING, HOST-VIRUS INTERACTION, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, UBL CONJUGATION, ZINC, ZINC-FINGER
2piq:A (MET780) to (SER888) ANDROGEN RECEPTOR LBD WITH SMALL MOLECULE | ANDROGEN RECEPTOR, INHIBITORS COACTIVATOR BINDING AF-2, HORMONE RECEPTOR
2piw:A (TYR781) to (SER888) ANDROGEN RECEPTOR WITH SMALL MOLECULE | ANDROGEN RECEPTOR INHIBITORS COACTIVATOR BINDING, HORMONE RECEPTOR
3fei:A (ARG348) to (TYR464) DESIGN AND BIOLOGICAL EVALUATION OF NOVEL, BALANCED DUAL PPARA/G AGONISTS | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, DIABETES, ACTIVATOR, DNA-BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
2pob:A (GLU365) to (TYR473) PPARGAMMA LIGAND BINDING DOMAIN COMPLEXED WITH A FARGLITAZAR ANALOGUE GW4709 | PPARG, NUCLEAR RECEPTOR,PPAR, GENE REGULATION
2pog:A (VAL422) to (MET543) BENZOPYRANS AS SELECTIVE ESTROGEN RECEPTOR B AGONISTS (SERBAS). PART 2: STRUCTURE ACTIVITY RELATIONSHIP STUDIES ON THE BENZOPYRAN SCAFFOLD. | NUCLEAR RECEPTOR, LIGAND-BINDING, LIPID BINDING PROTEIN
3sp9:A (LYS322) to (TYR437) STRUCTURAL BASIS FOR ILOPROST AS A DUAL PPARALPHA/DELTA AGONIST | NUCLEAR RECEPTOR LBD, NUCLEAR RECEPTOR FOLD, LIGAND BINDING, GENE TRANSCRIPTION, DRUG BINDING, TRANSCRIPTION
3sp9:B (LYS322) to (THR427) STRUCTURAL BASIS FOR ILOPROST AS A DUAL PPARALPHA/DELTA AGONIST | NUCLEAR RECEPTOR LBD, NUCLEAR RECEPTOR FOLD, LIGAND BINDING, GENE TRANSCRIPTION, DRUG BINDING, TRANSCRIPTION
2q3y:A (TYR109) to (GLY237) ANCESTRAL CORTICIOD RECEPTOR IN COMPLEX WITH DOC | NUCLEAR RECEPTOR, MINERALOCOTICIOD, LIGAND BINDING DOMAIN, DOC, CORTISOL, EVOLUTION, TRANSCRIPTION
3fur:A (MET364) to (TYR477) CRYSTAL STRUCTURE OF PPARG IN COMPLEX WITH INT131 | NUCLEAR RECEPTOR, PPARGAMMA, X-RAY, CRYSTAL STRUCTURE, PARTIAL AGONIST, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, INT131, TRANSCRIPTION/TRANSCRIPTION REGULATOR COMPLEX
2q59:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA LBD BOUND TO FULL AGONIST MRL20 | PROTEIN-LIGAND COMPLEX, LIGAND BINDING PROTEIN
2q5g:A (LYS358) to (LYS474) LIGAND BINDING DOMAIN OF PPAR DELTA RECEPTOR IN COMPLEX WITH A PARTIAL AGONIST | PPAR DELTA, TRANSCRIPTION
2q5s:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA BOUND TO PARTIAL AGONIST NTZDPA | PROTEIN-LIGAND COMPLEX, LIGAND BINDING PROTEIN
2q61:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN BOUND TO PARTIAL AGONIST SR145 | PROTEIN-LIGAND COMPLEX, LIGAND BINDING PROTEIN
2q61:B (LYS358) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN BOUND TO PARTIAL AGONIST SR145 | PROTEIN-LIGAND COMPLEX, LIGAND BINDING PROTEIN
2q6s:A (ARG357) to (ILE472) 2.4 ANGSTROM CRYSTAL STRUCTURE OF PPAR GAMMA COMPLEXED TO BVT.13 WITHOUT CO-ACTIVATOR PEPTIDES | PROTEIN-LIGAND COMPLEX, LIGAND BINDING PROTEIN
2q7i:A (MET780) to (GLN902) THE WILD TYPE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN BOUND WITH TESTOSTERONE AND AN AR 20-30 PEPTIDE | ANDROGEN RECEPTOR STEROID NUCLEAR RECEPTOR LIGAND BINDING DOMAIN, TESTOSETERONE, N-TERMINAL AR PEPTIDE, TIF2 BOXIII COACTIVATOR PEPTIDE, HORMONE
2q7j:A (MET780) to (SER888) THE WILD TYPE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN BOUND WITH TESTOSTERONE AND A TIF2 BOX 3 COACTIVATOR PEPTIDE 740-753 | ANDROGEN RECEPTOR STEROID NUCLEAR RECEPTOR LIGAND BINDING DOMAIN, TESTOSETERONE, TIF2 BOXIII COACTIVATOR PEPTIDE, HORMONE
2q8s:A (ARG357) to (LYS474) X-RAY CRYSTAL STRUCTURE OF THE NUCLEAR HORMONE RECEPTOR PPAR-GAMMA IN A COMPLEX WITH A PPAR GAMMA/ALPHA DUAL AGONIST | LIGAND-BOUND COMPLEX, HORMONE RECEPTOR
2qa6:A (MET421) to (LEU549) CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR ALPHA MUTANT 537S COMPLEXED WITH 4-(6-HYDROXY-1H-INDAZOL-3-YL)BENZENE-1,3-DIOL | PROTEIN-LIGAND COMPLEX, TRANSCRIPTION
2qa8:A (GLY442) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN MUTANT 537S COMPLEXED WITH GENISTEIN | PROTEIN-LIGAND COMPLEX, TRANSCRIPTION
3sz1:A (ARG357) to (TYR473) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH LUTEOLIN AND MYRISTIC ACID | PPAR GAMMA, NUCLEAR RECEPTOR, LUTEOLIN, TRANSCRIPTION
3t03:A (LYS386) to (TYR501) CRYSTAL STRUCTURE OF PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A NOVEL PARTIAL AGONIST GQ-16 | PROTEIN-DRUG COMPLEX, THIAZOLIDINEDIONES, LIGAND BINDING PROTEIN, TRANSCRIPTION FACTOR, NUCLEUS RECEPTOR, TRANSCRIPTION-TRANSCRIPTION REGULATOR COMPLEX
3t03:B (ARG385) to (TYR501) CRYSTAL STRUCTURE OF PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A NOVEL PARTIAL AGONIST GQ-16 | PROTEIN-DRUG COMPLEX, THIAZOLIDINEDIONES, LIGAND BINDING PROTEIN, TRANSCRIPTION FACTOR, NUCLEUS RECEPTOR, TRANSCRIPTION-TRANSCRIPTION REGULATOR COMPLEX
1p8d:B (GLN346) to (TRP457) X-RAY CRYSTAL STRUCTURE OF LXR LIGAND BINDING DOMAIN WITH 24(S),25- EPOXYCHOLESTEROL | LXR, EPOXYCHOLESTEROL, NUCLEAR RECEPTOR, STEROID RECEPTOR, LIVER X RECEPTOR, TRANSCRIPTION, MEMBRANE PROTEIN-PROTEIN BINDING COMPLEX
1db1:A (SER306) to (GLY423) CRYSTAL STRUCTURE OF THE NUCLEAR RECEPTOR FOR VITAMIN D COMPLEXED TO VITAMIN D | COMPLEX, GENE REGULATION
2qgt:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED TO AN ETHER ESTRADIOL COMPOUND | PROTEIN-LIGAND COMPLEX, TRANSCRIPTION
2qh6:B (MET421) to (HIS547) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED WITH AN OXABICYCLIC DIARYLETHYLENE COMPOUND | PROTEIN-LIGAND COMPLEX, TRANSCRIPTION
3g8i:A (LYS349) to (TYR464) ALEGLITAZAR, A NEW, POTENT, AND BALANCED PPAR ALPHA/GAMMA AGONIST FOR THE TREATMENT OF TYPE II DIABETES | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, DIABETES, ACTIVATOR, DNA-BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACYLTRANSFERASE, ALTERNATIVE SPLICING, CHROMOSOMAL REARRANGEMENT, PHOSPHOPROTEIN, PROTO- ONCOGENE, TRANSFERASE, UBL CONJUGATION, TRANSCRIPTION/TRANSFERASE COMPLEX
3g9e:A (LYS358) to (TYR473) ALEGLITAAR. A NEW. POTENT, AND BALANCED DUAL PPARA/G AGONIST FOR THE TREATMENT OF TYPE II DIABETES | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, DIABETES, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACYLTRANSFERASE, CHROMOSOMAL REARRANGEMENT, PROTO-ONCOGENE, TRANSFERASE, UBL CONJUGATION, TRANSCRIPTION/TRANSFERASE COMPLEX
3gbk:A (LYS358) to (TYR473) CRYSTAL STRUCTURE OF HUMAN PPAR-GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH A POTENT AND SELECTIVE AGONIST | PPAR AGANISTS, X-RAY CO-CRYSTAL ANALYSIS, STRUCTURE-BASED DRUG DESIGN, SELECTIVE, TYPE II DIABETES, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, LIGAND BINDING PROTEIN
3gbk:B (GLU365) to (TYR473) CRYSTAL STRUCTURE OF HUMAN PPAR-GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH A POTENT AND SELECTIVE AGONIST | PPAR AGANISTS, X-RAY CO-CRYSTAL ANALYSIS, STRUCTURE-BASED DRUG DESIGN, SELECTIVE, TYPE II DIABETES, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, LIGAND BINDING PROTEIN
4xum:A (GLU365) to (TYR473) PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH INDOMETHACIN | PPARGAMMA, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, NSAIDS, INDOMETHACIN, TRANSLATION
4xum:B (LYS358) to (TYR473) PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH INDOMETHACIN | PPARGAMMA, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, NSAIDS, INDOMETHACIN, TRANSLATION
4is8:A (GLU421) to (ALA538) DIVERGENT SEQUENCE TUNES LIGAND SENSITIVITY IN PHOSPHOLIPID-REGULATED HORMONE RECEPTORS | LIGAND BINDING DOMAIN, TRANSCRIPTION
4is8:B (VAL422) to (ALA538) DIVERGENT SEQUENCE TUNES LIGAND SENSITIVITY IN PHOSPHOLIPID-REGULATED HORMONE RECEPTORS | LIGAND BINDING DOMAIN, TRANSCRIPTION
2qpy:A (MET780) to (SER888) AR LBD WITH SMALL MOLECULE | ANDROGEN RECEPTOR DHT COACTIVATOR, DNA-BINDING, LIPID- BINDING, METAL-BINDING, NUCLEUS, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, UBL CONJUGATION, ZINC, ZINC-FINGER, DNA BINDING PROTEIN
4itf:A (SER306) to (PHE422) CRYSTAL STRUCTURE OF THE HUMAN VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH 1ALPHA,25-DIHYDROXY-2ALPHA-[2-(1H-TETRAZOLE-1- YL)ETHYL]VITAMIN D3 | HORMONE RECEPTOR, TRANSCRIPTION
4iu7:B (MET421) to (LEU549) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH CONSTRAINED WAY-DERIVATIVE, 2B | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, NUCLEUS, TRANSCRIPTION
2qr9:A (MET421) to (LEU549) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED WITH AN OXABICYCLIC DERIVATIVE COMPOUND | PROTEIN-LIGAND COMPLEX, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
2qr9:B (VAL422) to (ALA546) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED WITH AN OXABICYCLIC DERIVATIVE COMPOUND | PROTEIN-LIGAND COMPLEX, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3t58:B (PHE406) to (HIS538) C76A/C455S MUTANT OF MOUSE QSOX1 CONTAINING AN INTERDOMAIN DISULFIDE | OXIDOREDUCTASE
3t58:C (GLY405) to (ILE544) C76A/C455S MUTANT OF MOUSE QSOX1 CONTAINING AN INTERDOMAIN DISULFIDE | OXIDOREDUCTASE
3t58:D (GLY405) to (ILE544) C76A/C455S MUTANT OF MOUSE QSOX1 CONTAINING AN INTERDOMAIN DISULFIDE | OXIDOREDUCTASE
4iui:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DYNAMIC WAY DERIVATIVE, 4A | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, NUCLEUS, TRANSCRIPTION
4iui:B (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DYNAMIC WAY DERIVATIVE, 4A | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, NUCLEUS, TRANSCRIPTION
3t59:B (GLY405) to (ILE544) C76A/C455S MUTANT OF MOUSE QSOX1 CONTAINING AN INTERDOMAIN DISULFIDE | OXIDOREDUCTASE
4iv2:B (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DYNAMIC WAY-DERIVATIVE, 5A | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4iv4:B (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH CONSTRAINED WAY-DERIVATIVE, 5B | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4ivw:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH CONSTRAINED WAY-DERIVATIVE, 6B | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4ivw:B (MET421) to (ALA546) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH CONSTRAINED WAY-DERIVATIVE, 6B | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4ivy:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DYNAMIC WAY-DERIVATIVE, 7A | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4ivy:B (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DYNAMIC WAY-DERIVATIVE, 7A | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
2qse:A (MET421) to (ASN532) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED WITH BURNED MEAT COMPOUND 4-OH-PHIP | PROTEIN-LIGAND COMPLEX, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
2qse:B (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED WITH BURNED MEAT COMPOUND 4-OH-PHIP | PROTEIN-LIGAND COMPLEX, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
4iw6:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH CONSTRAINED WAY-DERIVATIVE, 7B | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4iw6:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH CONSTRAINED WAY-DERIVATIVE, 7B | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4iw8:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DYNAMIC WAY-DERIVATIVE, 9A | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4iwc:A (GLY420) to (ALA546) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DYNAMIC THIOPHENE-DERIVATIVE | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4iwc:B (MET421) to (LEU549) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DYNAMIC THIOPHENE-DERIVATIVE | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4iwf:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DYNAMIC OXIME-DERIVATIVE | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
1pq6:B (VAL347) to (TRP457) HUMAN LXR BETA HORMONE RECEPTOR / GW3965 COMPLEX | LXRB+KB043546/WAY207380/GW3965, TRANSCRIPTION REGULATION
1prg:A (ARG357) to (TYR473) LIGAND BINDING DOMAIN OF THE HUMAN PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR GAMMA | THIAZOLIDINEDIONE, LIGAND-BINDING DOMAIN, NUCLEAR RECEPTOR, APO, TRANSCRIPTION FACTOR, ORPHAN RECEPTOR, GENE REGULATION
2qw4:B (TRP151) to (ASP263) HUMAN NR4A1 LIGAND-BINDING DOMAIN | NUCLEAR RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, DNA-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC- FINGER, HORMONE RECEPTOR
2qw4:D (ILE152) to (ASP263) HUMAN NR4A1 LIGAND-BINDING DOMAIN | NUCLEAR RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, DNA-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC- FINGER, HORMONE RECEPTOR
4y29:A (ARG357) to (TYR473) IDENTIFICATION OF A NOVEL PPARG LIGAND THAT REGULATES METABOLISM | AF-2 HELIX, LIGAND BINDING POCKET, THREE-LAYER HELICAL SANDWICH, TRANSCRIPTION REGULATOR PPARG, NR1C3, PEROXISOME PROLIFERATOR- ACTIVATED RECEPTOR GAMMA, NHR, NUCLEAR RECEPTOR, COACTIVATOR, TRANSCRIPTION FACTOR, DNA BINDING PROTEIN-TRANSCRIPTION COMPLEX
2qxm:A (MET421) to (LEU549) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED TO BURNED MEAT COMPOUND PHIP | PROTEIN-LIGAND COMPLEX, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
2qxm:B (VAL422) to (ALA546) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED TO BURNED MEAT COMPOUND PHIP | PROTEIN-LIGAND COMPLEX, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
2qzo:A (VAL422) to (LEU549) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED WITH WAY-169916 | PROTEIN-LIGAND COMPLEX, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
2qzo:B (VAL422) to (ASP545) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED WITH WAY-169916 | PROTEIN-LIGAND COMPLEX, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
2r40:D (MET413) to (TRP526) CRYSTAL STRUCTURE OF 20E BOUND ECR/USP | NUCLEAR RECEPTOR LIGAND-BINDING DOMAIN, ANTI-PARALLEL ALPHA-HELICAL SANDWICH, ECDYSONE RECEPTOR, ECR, GENE REGULATION
1pzl:A (SER253) to (GLY367) CRYSTAL STRUCTURE OF HNF4A LBD IN COMPLEX WITH THE LIGAND AND THE COACTIVATOR SRC-1 PEPTIDE | TRANSCRIPTION
4j5w:A (MET323) to (PHE429) CRYSTAL STRUCTURE OF THE APO-PXR/RXRALPHA LBD HETEROTETRAMER COMPLEX | PREGNANE X RECEPTOR, RETINOID X RECEPTOR ALPHA, LIGAND BINDING DOMAIN, NUCLEAR RECEPTOR, ALPHA HELICAL SANDWICH, UNIQUE INTERMOLECULAR BETA-SHEET DIMERIZATION, XENOBIOTIC SENSING, UPREGULATION OF DRUG METABOLISM ENZYMES, RETINOIC ACID-BINDING PROTEIN
4j5w:B (MET323) to (PHE429) CRYSTAL STRUCTURE OF THE APO-PXR/RXRALPHA LBD HETEROTETRAMER COMPLEX | PREGNANE X RECEPTOR, RETINOID X RECEPTOR ALPHA, LIGAND BINDING DOMAIN, NUCLEAR RECEPTOR, ALPHA HELICAL SANDWICH, UNIQUE INTERMOLECULAR BETA-SHEET DIMERIZATION, XENOBIOTIC SENSING, UPREGULATION OF DRUG METABOLISM ENZYMES, RETINOIC ACID-BINDING PROTEIN
4j5x:C (GLY343) to (GLU456) CRYSTAL STRUCTURE OF THE SR12813-BOUND PXR/RXRALPHA LBD HETEROTETRAMER COMPLEX | PREGNANE X RECEPTOR, RETINOID X RECEPTOR ALPHA, LIGAND BINDING DOMAIN, NUCLEAR RECEPTOR, SR12813, ALPHA HELICAL SANDWICH, UNIQUE INTERMOLECULAR BETA-SHEET DIMERIZATION, XENOBIOTIC SENSING, UPREGULATION OF DRUG METABOLISM ENZYMES, RETINOIC ACID-BINDING PROTEIN
4j5x:A (PRO322) to (PHE429) CRYSTAL STRUCTURE OF THE SR12813-BOUND PXR/RXRALPHA LBD HETEROTETRAMER COMPLEX | PREGNANE X RECEPTOR, RETINOID X RECEPTOR ALPHA, LIGAND BINDING DOMAIN, NUCLEAR RECEPTOR, SR12813, ALPHA HELICAL SANDWICH, UNIQUE INTERMOLECULAR BETA-SHEET DIMERIZATION, XENOBIOTIC SENSING, UPREGULATION OF DRUG METABOLISM ENZYMES, RETINOIC ACID-BINDING PROTEIN
4j5x:B (GLU321) to (PHE429) CRYSTAL STRUCTURE OF THE SR12813-BOUND PXR/RXRALPHA LBD HETEROTETRAMER COMPLEX | PREGNANE X RECEPTOR, RETINOID X RECEPTOR ALPHA, LIGAND BINDING DOMAIN, NUCLEAR RECEPTOR, SR12813, ALPHA HELICAL SANDWICH, UNIQUE INTERMOLECULAR BETA-SHEET DIMERIZATION, XENOBIOTIC SENSING, UPREGULATION OF DRUG METABOLISM ENZYMES, RETINOIC ACID-BINDING PROTEIN
2r6w:A (MET421) to (MET543) ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN COMPLEXED TO A SERM | ESTROGEN RECEPTOR, LIGAND-BINDING DOMAIN, ALTERNATIVE SPLICING, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, POLYMORPHISM, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
2r6w:B (MET421) to (ALA546) ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN COMPLEXED TO A SERM | ESTROGEN RECEPTOR, LIGAND-BINDING DOMAIN, ALTERNATIVE SPLICING, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, POLYMORPHISM, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
4jaz:B (ARG357) to (TYR473) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN PPARGAMMA LBD AND TRANS- RESVERATROL | BUNDLE OF ALPHA-HELICES, SMALL FOUR-STRNDED BETA-SHEET, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, NUCLEUS, OBESITY, PHOSPHORYLATION, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION
3tkc:A (SER306) to (GLY423) DESIGN, SYNTHESIS, EVALUATION AND STRUCTURE OF VITAMIN D ANALOGUES WITH FURAN SIDE CHAINS | ALPHA-HELICAL SANDWICH, TRANSCRIPTION, CALCITRIOL, PHOSPHORYLATION, NUCLEUS
3tkm:A (LYS322) to (TYR437) CRYSTAL STRUCTURE PPAR DELTA BINDING GW0742 | NUCLEAR RECEPTOR, TRANSCRIPTION, TRANSCRIPTION-TRANSCRIPTION ACTIVATOR COMPLEX
3gyu:A (LYS634) to (PHE749) NUCLEAR RECEPTOR DAF-12 FROM PARASITIC NEMATODE STRONGYLOIDES STERCORALIS IN COMPLEX WITH ITS PHYSIOLOGICAL LIGAND DAFACHRONIC ACID DELTA 7 | NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, DAFACHRONIC ACID, SRC1, NEMATODE, STRONGYLOIDES STERCORALIS, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
3gz9:A (LYS358) to (TYR473) CRYSTAL STRUCTURE OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DELTA (PPARD) IN COMPLEX WITH A FULL AGONIST | PPAR, PPAR DELTA, TRANSCRIPTION, NUCLEAR RECEPTOR FOLD, TRANSCRIPTION REGULATION, HORMONE, GROWTH FACTOR RECEPTOR, COMPLEX, ACTIVATOR, ALTERNATIVE SPLICING, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, ZINC, ZINC-FINGER
3h0a:D (MET364) to (TYR473) CRYSTAL STRUCTURE OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA (PPARG) AND RETINOIC ACID RECEPTOR ALPHA (RXRA) IN COMPLEX WITH 9-CIS RETINOIC ACID, CO-ACTIVATOR PEPTIDE, AND A PARTIAL AGONIST | PPAR, TRANSCRIPTION, NUCLEAR RECEPTOR FOLD, TRANSCRIPTION REGULATION, HORMONE, GROWTH FACTOR RECEPTOR, COMPLEX, DNA-BINDING, HOST-VIRUS INTERACTION, ISOPEPTIDE BOND, METAL-BINDING, NUCLEUS, RECEPTOR, ZINC-FINGER, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, OBESITY, PHOSPHOPROTEIN, ACYLTRANSFERASE, PROTO-ONCOGENE, TRANSFERASE
2rew:A (MET355) to (TYR464) CRYSTAL STRUCTURE OF PPARALPHA LIGAND BINDING DOMAIN WITH BMS-631707 | ALPHA HELICAL, ACTIVATOR, DNA-BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
1ere:C (MET421) to (ARG548) HUMAN ESTROGEN RECEPTOR LIGAND-BINDING DOMAIN IN COMPLEX WITH 17BETA-ESTRADIOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, STEROID, AGONIST
1ere:D (MET421) to (ARG548) HUMAN ESTROGEN RECEPTOR LIGAND-BINDING DOMAIN IN COMPLEX WITH 17BETA-ESTRADIOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, STEROID, AGONIST
1ere:F (MET421) to (ARG548) HUMAN ESTROGEN RECEPTOR LIGAND-BINDING DOMAIN IN COMPLEX WITH 17BETA-ESTRADIOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, STEROID, AGONIST
1qkn:A (ILE328) to (ALA452) RAT OESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN IN COMPLEX WITH ANTAGONIST RALOXIFENE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ANTAGONIST
4jl4:B (ARG357) to (TYR473) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN PPARGAMMA LBD AND THE LIGAND LJ570 [(2S)-3-(BIPHENYL-4-YL)-2-(BIPHENYL-4-YLOXY)PROPANOIC ACID] | BUNDLE OF ALPHA-HELICES, SMALL FOUR-STRNDED BETA-SHEET, TRANSCRIPTION FACTOR, RXR, TRANSCRIPTION-AGONIST COMPLEX
1exa:A (ASP309) to (GLU417) ENANTIOMER DISCRIMINATION ILLUSTRATED BY CRYSTAL STRUCTURES OF THE HUMAN RETINOIC ACID RECEPTOR HRARGAMMA LIGAND BINDING DOMAIN: THE COMPLEX WITH THE ACTIVE R-ENANTIOMER BMS270394. | ENANTIOMER DISCRIMINATION, RETINOID LIGAND COMPLEXES, ANTIPARALLEL ALPHA-HELICAL SANDWICH FOLD, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS, GENE REGULATION
1exx:A (GLY305) to (GLU417) ENANTIOMER DISCRIMINATION ILLUSTRATED BY CRYSTAL STRUCTURES OF THE HUMAN RETINOIC ACID RECEPTOR HRARGAMMA LIGAND BINDING DOMAIN: THE COMPLEX WITH THE INACTIVE S-ENANTIOMER BMS270395. | ENANTIOMER DISCRIMINATION, RETINOID LIGAND COMPLEXES, ANTIPARALLEL ALPHA-HELICAL SANDWICH FOLD, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS, GENE REGULATION
3tx7:B (ALA422) to (ALA538) CRYSTAL STRUCTURE OF LRH-1/BETA-CATENIN COMPLEX | LRH-1, BETA-CATENIN, ARMADILLO REPEAT, NUCLEAR RECEPTOR LIGAND BINDING DOMAIN, PROTEIN BINDING
3ty0:A (ARG357) to (TYR473) STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH (R)-5-(3- ((3-(6-METHOXYBENZO[D]ISOXAZOL-3-YL)-2-OXO-2,3-DIHYDRO-1H- BENZO[D]IMIDAZOL-1-YL)METHYL)PHENYL)-5-METHYLOXAZOLIDINE-2,4-DIONE | NUCLEAR RECEPTOR LIGAND BINDING DOMAIN, TRANSCRIPTION REGULATOR
3ty0:B (GLU865) to (TYR973) STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH (R)-5-(3- ((3-(6-METHOXYBENZO[D]ISOXAZOL-3-YL)-2-OXO-2,3-DIHYDRO-1H- BENZO[D]IMIDAZOL-1-YL)METHYL)PHENYL)-5-METHYLOXAZOLIDINE-2,4-DIONE | NUCLEAR RECEPTOR LIGAND BINDING DOMAIN, TRANSCRIPTION REGULATOR
1r1k:D (MET413) to (TRP526) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE HETERODIMER ECR/USP BOUND TO PONASTERONE A | NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, HETERODIMER, ALPHA-HELICAL SANDWICH, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
3hc6:A (ASP359) to (TRP469) FXR WITH SRC1 AND GSK088 | FXR, NUCLEAR RECEPTOR, GW4064, ALPHA-HELICAL SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DNA-BINDING, METAL- BINDING, NUCLEUS, RECEPTOR, REPRESSOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
1fby:B (LEU1353) to (GLU1456) CRYSTAL STRUCTURE OF THE HUMAN RXR ALPHA LIGAND BINDING DOMAIN BOUND TO 9-CIS RETINOIC ACID | NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, RETINOID RECEPTOR, TRANSCRIPTION
1r20:D (MET413) to (TRP526) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE HETERODIMER ECR/USP BOUND TO THE SYNTHETIC AGONIST BYI06830 | NUCLEAR RECEPTOR, HETERODIMER, ALPHA-HELICAL SANDWICH, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
4jyh:B (LEU298) to (MET407) CRYSTAL STRUCTURE OF RARBETA LBD IN COMPLEX WITH SELECTIVE AGONIST BMS948 [4-{[(8-PHENYLNAPHTHALEN-2-YL)CARBONYL]AMINO}BENZOIC ACID] | LIGAND BINDING DOMAIN, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION- AGONIST COMPLEX
1fd0:A (ASP309) to (GLU417) ISOTYPE SELECTIVITY OF THE HUMAN RETINOIC ACID NUCLEAR RECEPTOR HRAR: THE COMPLEX WITH THE RARGAMMA-SELECTIVE RETINOID SR11254 | ISOTYPE SELECTIVITY, RETINOID LIGAND COMPLEXES, DRUG DESIGN, ANTIPARALLEL ALPHA-HELICAL SANDWICH FOLD, CH...O HYDROGEN BOND, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS, GENE REGULATION
3u9q:A (MET364) to (TYR473) LIGAND BINDING DOMAIN OF PPARGAMMA COMPLEXED WITH DECANOIC ACID AND PGC-1A PEPTIDE | NUCLEAR RECEPTOR, ADIPOGENESIS, RXRA, NUCLEUS, TRANSCRIPTION
1r5k:A (MET421) to (ASP545) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH GW5638 | ALPHA HELIX, HELICAL SANDWICH, DNA BINDING PROTEIN
2v0v:A (ASP481) to (LYS576) CRYSTAL STRUCTURE OF REV-ERB BETA | ZINC, RECEPTOR, REPRESSOR, ZINC-FINGER, DNA-BINDING, CONSTITUTIVE REPRESSION, TRANSCRIPTION REGULATION, ORPHAN RECEPTOR, A-HELICAL SANDWICH, TRANSCRIPTION, METAL-BINDING, NUCLEAR PROTEIN
1fm9:D (ARG357) to (TYR473) THE 2.1 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE HETERODIMER OF THE HUMAN RXRALPHA AND PPARGAMMA LIGAND BINDING DOMAINS RESPECTIVELY BOUND WITH 9-CIS RETINOIC ACID AND GI262570 AND CO-ACTIVATOR PEPTIDES. | THE HETERODIMER OF THE NUCLEAR RECEPTOR LIGAND BINDING DOMAINS OF RXRALPHA AND PPARGAMMA BOUND RESPECTIVELY WITH 9-CIS RETINOIC ACID AND GI262570 AND CO-ACTIVATOR PEPTIDES, TRANSCRIPTION
2ewp:A (LEU343) to (ILE438) CRYSTAL STRUCTURE OF ESTROGEN RELATED RECEPTOR-3 (ERR-GAMMA) LIGAND BINDING DOMAIND WITH TAMOXIFEN ANALOG GSK5182 | TAMOXIFEN, ERR, ESTROGEN RELATED RECEPTOR, ORPHAN RECEPTOR, TRANSCRIPTION
4yt1:A (ARG357) to (TYR473) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A GAMMMA SELECTIVE SYNTHETIC PARTIAL AGONIST MEKT76 | NUCLEAR RECEPTOR, TRANSCRIPTION
4yt1:B (LYS358) to (TYR473) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A GAMMMA SELECTIVE SYNTHETIC PARTIAL AGONIST MEKT76 | NUCLEAR RECEPTOR, TRANSCRIPTION
3hlv:A (VAL422) to (ARG548) CRYSTAL STRUCTURE OF HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE AND 16-ALPHA-HYDROXY-ESTRONE ((8S,9R,13S,14R, 16R)-3,16-DIHYDROXY-13-METHYL-7,8,9,11,12,14,15, 16-OCTAHYDRO-6H- CYCLOPENTA[A]PHENANTHREN-17-ONE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HYDROXY-ESTRONE, ALTERNATIVE SPLICING, DNA-BINDING, GLYCOPROTEIN, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACTIVATOR, HORMONE, NUCLEAR RECEPTOR
3hm1:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE AND ESTRONE ((8R,9S,13S,14S)-3-HYDROXY-13-METHYL- 7,8,9,11,12,14,15,16-OCTAHYDRO-6H-CYCLOPENTA[A]PHENANTHREN-17-ONE) | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, ESTRONE, ALTERNATIVE SPLICING, DNA-BINDING, GLYCOPROTEIN, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACTIVATOR, HORMONE, NUCLEAR RECEPTOR
3hm1:B (VAL422) to (ALA546) CRYSTAL STRUCTURE OF HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE AND ESTRONE ((8R,9S,13S,14S)-3-HYDROXY-13-METHYL- 7,8,9,11,12,14,15,16-OCTAHYDRO-6H-CYCLOPENTA[A]PHENANTHREN-17-ONE) | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, ESTRONE, ALTERNATIVE SPLICING, DNA-BINDING, GLYCOPROTEIN, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACTIVATOR, HORMONE, NUCLEAR RECEPTOR
1rdt:D (ARG357) to (TYR473) CRYSTAL STRUCTURE OF A NEW REXINOID BOUND TO THE RXRALPHA LIGAND BINDING DOAMIN IN THE RXRALPHA/PPARGAMMA HETERODIMER | HORMONE, RECEPTOR, POLYMORPHISM, HORMONE/GROWTH FACTOR COMPLEX
2f4b:A (LYS358) to (TYR473) CRYSTAL STRUCTURE OF THE LIGAND BINDING DOMAIN OF HUMAN PPAR-GAMMA IN COMPLEX WITH AN AGONIST | PPAR, TRANSCRIPTION ACTIVATOR
2f4b:B (ARG357) to (TYR473) CRYSTAL STRUCTURE OF THE LIGAND BINDING DOMAIN OF HUMAN PPAR-GAMMA IN COMPLEX WITH AN AGONIST | PPAR, TRANSCRIPTION ACTIVATOR
3ho0:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF THE PPARGAMMA-LBD COMPLEXED WITH A NEW ARYLOXY-3PHENYLPROPANOIC ACID | BUNDLE OF ALPHA-HELICES, SMALL FOUR-STRANDED BETA-SHEET, TRANSCRIPTION, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
3ho0:B (ARG357) to (LYS474) CRYSTAL STRUCTURE OF THE PPARGAMMA-LBD COMPLEXED WITH A NEW ARYLOXY-3PHENYLPROPANOIC ACID | BUNDLE OF ALPHA-HELICES, SMALL FOUR-STRANDED BETA-SHEET, TRANSCRIPTION, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
1g1u:D (GLY343) to (GLY443) THE 2.5 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE RXRALPHA LIGAND BINDING DOMAIN IN TETRAMER IN THE ABSENCE OF LIGAND | CRYSTAL STRUCTURE, RXRALPHA LIGAND BINDING DOMAIN, TETRAMER, ABSENCE OF LIGAND, TRANSCRIPTION
2fai:A (VAL422) to (ARG548) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH OBCP-2M AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
2fai:B (MET421) to (ARG548) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH OBCP-2M AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
3hod:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF THE PPARGAMMA-LBD COMPLEXED WITH A NEW ARYLOXY-3PHENYLPROPANOIC ACID | BUNDLE OF ALPHA-HELICES, SMALL FOUR-STRANDED BETA-SHEET, TRANSCRIPTION, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
3up0:A (HIS583) to (PHE682) NUCLEAR RECEPTOR DAF-12 FROM HOOKWORM ANCYLOSTOMA CEYLANICUM IN COMPLEX WITH (25S)-DELTA7-DAFACHRONIC ACID | NEMATODE, STEROID BINDING PROTEIN-TRANSCRIPTION COMPLEX
3up0:B (HIS583) to (PHE682) NUCLEAR RECEPTOR DAF-12 FROM HOOKWORM ANCYLOSTOMA CEYLANICUM IN COMPLEX WITH (25S)-DELTA7-DAFACHRONIC ACID | NEMATODE, STEROID BINDING PROTEIN-TRANSCRIPTION COMPLEX
3uu7:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BISPHENOL-A | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
3uua:A (MET421) to (ALA546) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BISPHENOL-AF | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
3uua:B (GLY442) to (ARG548) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BISPHENOL-AF | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
3uuc:A (MET421) to (LEU544) CRYSTAL STRUCTURE OF HERA-LBD (WT) IN COMPLEX WITH BISPHENOL-C | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
3uuc:B (VAL422) to (MET543) CRYSTAL STRUCTURE OF HERA-LBD (WT) IN COMPLEX WITH BISPHENOL-C | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
3uuc:C (MET421) to (ASP545) CRYSTAL STRUCTURE OF HERA-LBD (WT) IN COMPLEX WITH BISPHENOL-C | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
3uuc:D (MET421) to (GLU542) CRYSTAL STRUCTURE OF HERA-LBD (WT) IN COMPLEX WITH BISPHENOL-C | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
1s0x:A (ASP398) to (ARG500) CRYSTAL STRUCTURE OF THE HUMAN RORALPHA LIGAND BINDING DOMAIN IN COMPLEX WITH CHOLESTEROL SULFATE AT 2.2A | THREE-LAYERED ALPHA HELICAL SANDWICH, NUCLEAR HORMONE RECEPTOR, ORPHAN RECEPTOR, LIGAND BINDING DOMAIN, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
3hv0:A (ASN481) to (ASN579) TRYPTOPHANYL-TRNA SYNTHETASE FROM CRYPTOSPORIDIUM PARVUM | TRNA-LIGASE, ATP-BINDING, AMINOACYL-TRNA SYNTHETASE, LIGASE, NUCLEOTIDE-BINDING, PROTEIN BIOSYNTHESIS, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP
3hv0:B (ASN481) to (ASN579) TRYPTOPHANYL-TRNA SYNTHETASE FROM CRYPTOSPORIDIUM PARVUM | TRNA-LIGASE, ATP-BINDING, AMINOACYL-TRNA SYNTHETASE, LIGASE, NUCLEOTIDE-BINDING, PROTEIN BIOSYNTHESIS, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP
3hvl:A (MET323) to (PHE429) TETHERED PXR-LBD/SRC-1P COMPLEXED WITH SR-12813 | PXR, SRC-1, TETHERED, ENGINEERED, DRUG-DRUG INTERACTIONS, DNA- BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER, TRANSFERASE
1s9p:D (LEU343) to (GLY442) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAIN OF THE ESTROGEN-RELATED RECEPTOR GAMMA IN COMPLEX WITH DIETHYLSTILBESTROL | LIGAND-BINDING DOMAIN, ANTAGONIST COMPLEX, TRANSCRIPTION
1s9q:A (LEU343) to (GLY442) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAIN OF THE ESTROGEN-RELATED RECEPTOR GAMMA IN COMPLEX WITH 4-HYDROXYTAMOXIFEN | LIGAND-BINDING DOMAIN, ANTAGONIST COMPLEX, TRANSCRIPTION
3v3e:B (TRP151) to (LEU265) CRYSTAL STRUCTURE OF THE HUMAN NUR77 LIGAND-BINDING DOMAIN | ORPHAN NUCLEAR RECEPTOR, TRANSCRIPTION
3v49:A (TYR781) to (SER888) STRUCTURE OF AR LBD WITH ACTIVATOR PEPTIDE AND SARM INHIBITOR 1 | DIARYLHYDANTOIN, SYNTHESIS, SARM, ANTIANDROGEN, LIGAND BINDING DOMAIN, TESTOSTERONE, DIHYDROTESTOSTERONE, TRANSCRIPTION, SARM (SELECTIVE ANDROGEN RECEPTOR MODULATOR)
3v4a:A (MET780) to (SER888) STRUCTURE OF AR LBD WITH ACTIVATOR PEPTIDE AND SARM INHIBITOR 2 | DIARYLHYDANTOIN, SYNTHESIS, ANTIANDROGEN, ANDROGEN RECEPTOR, TESTOSTERONE, SELECTIVE ANDROGEN RECEPTOR MODULATOR, DIHYDROTESTOSTERONE, TRANSCRIPTION
2fvj:A (MET364) to (TYR473) A NOVEL ANTI-ADIPOGENIC PARTIAL AGONIST OF PEROXISOME PROLIFERATOR- ACTIVATED RECEPTOR-GAMMA (PPARG) RECRUITS PPARG-COACTIVATOR-1 ALPHA (PGC1A) BUT POTENTIATES INSULIN SIGNALING IN VITRO | NUCLEAR RECEPTOR LBD, ALPHA HELICAL SANDWICH, SIGNALING PROTEIN
3v7o:A (SER41) to (TYR124) CRYSTAL STRUCTURE OF THE C-TERMINAL DOMAIN OF EBOLA VIRUS VP30 (STRAIN RESTON-89) | EBOLA, VP30, SSGCID, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, SMT, NUCLEOPROTEIN, TRANSCRIPTION
2g0g:A (ARG357) to (TYR473) STRUCTURE-BASED DRUG DESIGN OF A NOVEL FAMILY OF PPAR PARTIAL AGONISTS: VIRTUAL SCREENING, X-RAY CRYSTALLOGRAPHY AND IN VITRO/IN VIVO BIOLOGICAL ACTIVITIES | PPAR, TRANSCRIPTION ACTIVATOR
2g0g:B (ARG357) to (LYS474) STRUCTURE-BASED DRUG DESIGN OF A NOVEL FAMILY OF PPAR PARTIAL AGONISTS: VIRTUAL SCREENING, X-RAY CRYSTALLOGRAPHY AND IN VITRO/IN VIVO BIOLOGICAL ACTIVITIES | PPAR, TRANSCRIPTION ACTIVATOR
2g0h:A (ARG357) to (LYS474) STRUCTURE-BASED DRUG DESIGN OF A NOVEL FAMILY OF PPAR PARTIAL AGONISTS: VIRTUAL SCREENING, X-RAY CRYSTALLOGRAPHY AND IN VITRO/IN VIVO BIOLOGICAL ACTIVITIES | PPAR, TRANSCRIPTION ACTIVATOR
2g0h:B (GLU365) to (TYR473) STRUCTURE-BASED DRUG DESIGN OF A NOVEL FAMILY OF PPAR PARTIAL AGONISTS: VIRTUAL SCREENING, X-RAY CRYSTALLOGRAPHY AND IN VITRO/IN VIVO BIOLOGICAL ACTIVITIES | PPAR, TRANSCRIPTION ACTIVATOR
2g44:A (VAL422) to (ARG548) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH OBCP-1M-G AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
2g44:B (VAL422) to (LEU544) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH OBCP-1M-G AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
3v9t:A (PHE360) to (TYR473) CRYSTAL STRUCTURE OF THE PPARGAMMA-LBD COMPLEXED WITH A CERCOSPORAMIDE DERIVATIVE MODULATOR | THREE-LAYERED ALPHA-HELICAL SANDWICH, TRANSCRIPTION REGULATION, TRANSCRIPTION-TRANSCRIPTION REGULATOR COMPLEX
3v9v:A (LYS358) to (TYR473) CRYSTAL STRUCTURE OF THE PPARGAMMA-LBD COMPLEXED WITH A CERCOSPORAMIDE DERIVATIVE MODULATOR | THREE-LAYERED ALPHA-HELICAL SANDWICH, TRANSCRIPTION REGULATION, TRANSCRIPTION-TRANSCRIPTION REGULATOR COMPLEX
3v9y:A (LYS358) to (TYR473) CRYSTAL STRUCTURE OF THE PPARGAMMA-LBD COMPLEXED WITH A CERCOSPORAMIDE DERIVATIVE MODULATOR | THREE-LAYERED ALPHA-HELICAL SANDWICH, TRANSCRIPTION REGULATION, TRANSCRIPTION-TRANSCRIPTION REGULATOR COMPLEX
2g5o:A (MET421) to (ALA546) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH 2- (BUT-1-ENYL)-17BETA-ESTRADIOL AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
2g5o:B (MET421) to (ASP545) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH 2- (BUT-1-ENYL)-17BETA-ESTRADIOL AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
2vsr:A (ARG357) to (TYR473) HPPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH 9-(S)-HODE | TRANSCRIPTION REGULATION, ALTERNATIVE SPLICING, LIGAND BINDING DOMAIN, NUCLEAR RECEPTOR, DIABETES MELLITUS, ZINC-FINGER, DNA-BINDING, POLYMORPHISM, TRANSCRIPTION, ZINC, OBESITY, NUCLEUS, RECEPTOR, ACTIVATOR, OXIDISED FATTY ACID, TRANSCRIPTION FACTOR, METAL-BINDING, PHOSPHOPROTEIN, DISEASE MUTATION
2vst:A (ARG357) to (TYR473) HPPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH 13-(S)- HODE | TRANSCRIPTION REGULATION, ALTERNATIVE SPLICING, LIGAND BINDING DOMAIN, NUCLEAR RECEPTOR, DIABETES MELLITUS, ZINC-FINGER, DNA-BINDING, POLYMORPHISM, TRANSCRIPTION, ZINC, OBESITY, NUCLEUS, RECEPTOR, ACTIVATOR, OXIDISED FATTY ACID, TRANSCRIPTION FACTOR, METAL-BINDING, PHOSPHOPROTEIN, DISEASE MUTATION
2vv2:A (ARG357) to (LYS474) HPPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH 5-HEPA | TRANSCRIPTION REGULATION, ALTERNATIVE SPLICING, LIGAND BINDING DOMAIN, NUCLEAR RECEPTOR, DIABETES MELLITUS, ZINC-FINGER, DNA-BINDING, POLYMORPHISM, TRANSCRIPTION, ZINC, OBESITY, NUCLEUS, RECEPTOR, ACTIVATOR, OXIDISED FATTY ACID, TRANSCRIPTION FACTOR, METAL-BINDING, PHOSPHOPROTEIN, DISEASE MUTATION
2vv4:A (ARG357) to (TYR473) HPPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH 6-OXOOTE | RECEPTOR, NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, OXIDISED FATTY ACID, TRANSCRIPTION FACTOR
1gwq:A (MET421) to (ALA546) HUMAN OESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH RALOXIFENE CORE AND TIF2 NRBOX2 PEPTIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, TRANSACTIVATION, AGONIST, AF2 COACTIVATOR , RECEPTOR, ACTIVATOR, TRANSCRIPTI REGULATION, DNA-BINDING, NUCLEAR PROTEIN, ZINC FINGER, STER BINDING, PHOSPHORYLATION, POLYMORPHISM, ALTERNATIVE SPLICIN
1gwq:B (MET421) to (ALA546) HUMAN OESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH RALOXIFENE CORE AND TIF2 NRBOX2 PEPTIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, TRANSACTIVATION, AGONIST, AF2 COACTIVATOR , RECEPTOR, ACTIVATOR, TRANSCRIPTI REGULATION, DNA-BINDING, NUCLEAR PROTEIN, ZINC FINGER, STER BINDING, PHOSPHORYLATION, POLYMORPHISM, ALTERNATIVE SPLICIN
1gwx:A (LYS358) to (TYR473) MOLECULAR RECOGNITION OF FATTY ACIDS BY PEROXISOME PROLIFERATOR-ACTIVATED RECEPTORS | PPAR, FATTY ACIDS, TRANSCRIPTION, NUCLEAR RECEPTOR FOLD
1gwx:B (ARG357) to (TYR473) MOLECULAR RECOGNITION OF FATTY ACIDS BY PEROXISOME PROLIFERATOR-ACTIVATED RECEPTORS | PPAR, FATTY ACIDS, TRANSCRIPTION, NUCLEAR RECEPTOR FOLD
3ia6:A (ARG357) to (TYR473) X-RAY CRYSTAL STRUCTURE OF THE NUCLEAR HORMONE RECEPTOR PPAR-GAMMA IN A COMPLEX WITH A PPAR GAMMA/ALPHA DUAL AGONIST | PROTEIN-LIGAND COMPLEX, DUAL SPECIFICITY, INHIBITOR, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
3vhw:A (SER306) to (GLY423) CRYSTAL STRUCTURE OF THE HUMAN VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH 4-MP | HORMONE RECEPTOR, TRANSCRIPTION
3vi8:A (LYS349) to (ARG465) HUMAN PPAR ALPHA LIGAND BINDING DOMAIN IN COMPLEX WITH A SYNTHETIC AGONIST APHM13 | NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, PPAR, TRANSCRIPTION
3vji:A (ARG357) to (TYR473) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH JKPL53 | TRANSCRIPTION FACTOR, TRANSCRIPTION
3vji:B (LYS358) to (TYR473) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH JKPL53 | TRANSCRIPTION FACTOR, TRANSCRIPTION
4l36:A (ALA138) to (LEU227) CRYSTAL STRUCTURE OF THE CYTOCHROME P450 ENZYME TXTE | CYTOCHROME P450, DIRECT NITRATION, INDOLYL, L-TRYPTOPHAN, L-4- NITROTRYPTOPHAN, HEME, OXIDOREDUCTASE
3vjs:A (THR302) to (LEU410) VITAMIN D RECEPTOR COMPLEX WITH A CARBORANE COMPOUND | NUCLEAR RECEPTOR, SYNTHETIC AGONIST, CARBORANE, TRANSCRIPTION
1t65:A (TYR781) to (SER888) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN WITH DHT AND A PEPTIDE DERIVED FORM ITS PHYSIOLOGICAL COACTIVATOR GRIP1 NR BOX 2 BOUND IN A NON- HELICAL CONFORMATION | ANDROGEN RECEPTOR LIGAND BINDING DOMAIN GRIP1 NR BOX2 COACTIVATORS CRYSTAL STRUCTURE NON-HELICAL, HORMONE/GROWTH FACTOR COMPLEX
1t63:A (MET780) to (SER888) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN WITH DHT AND A PEPTIDE DERIVED FROM ITS PHYSIOLOGICAL COACTIVATOR GRIP1 NR BOX3 | ANDROGEN RECEPTOR LIGAND BINDING DOMAIN GRIP1 NR BOXES COACTIVATORS DHT CRYSTAL STRUCTURE, HORMONE/GROWTH FACTOR COMPLEX
4zn9:A (MET421) to (VAL533) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH OXABICYCLIC HEPTENE SULFONATE (OBHS) | PROTEIN LIGAND COMPLEX, TRANSCRIPTION
4zns:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH A 3-FLUORO-SUBSTITUTED OBHS DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4znt:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH A 3-BROMO-SUBSTITUTED OBHS DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4znt:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH A 3-BROMO-SUBSTITUTED OBHS DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4znv:A (VAL422) to (ASN532) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH A 2-METHOXY-SUBSTITUTED OBHS DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4znv:B (MET421) to (ASN532) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH A 2-METHOXY-SUBSTITUTED OBHS DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4znw:A (VAL422) to (VAL533) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH A 4-BROMO-SUBSTITUTED OBHS DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
2gp7:D (ASP344) to (LYS457) ESTROGEN RELATED RECEPTOR-GAMMA LIGAND BINDING DOMAIN | ESTROGEN RELATED RECEPTOR, ERR, ERRG, ESRRG, NUCLEAR RECEPTOR, STEROID RECEPTOR, TRANSCRIPTION
1t7f:A (TYR781) to (SER888) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH A LXXLL MOTIF | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING DOMAIN, AF-2, ANDROGEN, TESTOSTERONE, DHT, ALPHA-HELICAL SANDWICH, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
2gpo:A (LEU343) to (VAL458) ESTROGEN RELATED RECEPTOR-GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH A SYNTHETIC PEPTIDE FROM RIP140 | ESTROGEN RELATED RECEPTOR, ERR, ERRG, ESRRG, NUCLEAR RECEPTOR, STEROID RECEPTOR, RIP140, TRANSCRIPTION
2gpu:A (LEU343) to (LEU454) ESTROGEN RELATED RECEPTOR-GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH 4-HYDROXY-TAMOXIFEN | ESTROGEN RELATED RECEPTOR, ERR, ERRG, ESRRG, NUCLEAR RECEPTOR, STEROID RECEPTOR, TRANSCRIPTION
2gpv:A (LEU343) to (GLY442) ESTROGEN RELATED RECEPTOR-GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH 4-HYDROXY-TAMOXIFEN AND A SMRT PEPTIDE | ESTROGEN RELATED RECEPTOR, ERR, ERRG, ESRRG, NUCLEAR RECEPTOR, STEROID RECEPTOR, SMRT, TAMOXIFEN, TRANSCRIPTION
1t7t:A (TYR781) to (GLN902) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH 5-ALPHA DIHYDROTESTOSTERONE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING DOMAIN, AF-2, ANDROGEN, TESTOSTERONE, DHT, ALPHA-HELICAL SANDWICH, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
2gtk:A (ARG357) to (TYR473) STRUCTURE-BASED DESIGN OF INDOLE PROPIONIC ACIDS AS NOVEL PPARAG CO-AGONISTS | NUCLEAR RECEPTOR, TRANSCRIPTION REGULATOR
4lbd:A (LEU307) to (GLU417) LIGAND-BINDING DOMAIN OF THE HUMAN RETINOIC ACID RECEPTOR GAMMA BOUND TO THE SYNTHETIC AGONIST BMS961 | NUCLEAR RECEPTOR, RETINOIC ACID RECEPTOR, ALL-TRANS RETINOIC ACID, LIGAND-BINDING DOMAIN, COMPLEX, HOLO FORM, TRANSCRIPTION REGULATION, LIGAND-DEPENDENT, ACTIVE CONFORMATION, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS
2gwx:A (LYS358) to (TYR473) MOLECULAR RECOGNITION OF FATTY ACIDS BY PEROXISOME PROLIFERATOR-ACTIVATED RECEPTORS | PPAR, FATTY ACIDS, TRANSCRIPTION, NUCLEAR RECEPTOR FOLD
2gwx:B (ARG357) to (MET476) MOLECULAR RECOGNITION OF FATTY ACIDS BY PEROXISOME PROLIFERATOR-ACTIVATED RECEPTORS | PPAR, FATTY ACIDS, TRANSCRIPTION, NUCLEAR RECEPTOR FOLD
3ipu:A (VAL333) to (TRP443) X-RAY STRUCTURE OF BENZISOXAZOLE UREA SYNTHETIC AGONIST BOUND TO THE LXR-ALPHA | NUCLEAR RECEPTOR, LXR HOMODIMER, LXR SIGNALING, ALTERNATIVE SPLICING, DNA-BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACTIVATOR, ACYLTRANSFERASE, CHROMOSOMAL REARRANGEMENT, ISOPEPTIDE BOND, PHOSPHOPROTEIN, PROTO-ONCOGENE, TRANSFERASE, UBL CONJUGATION
3ipu:B (VAL333) to (TRP443) X-RAY STRUCTURE OF BENZISOXAZOLE UREA SYNTHETIC AGONIST BOUND TO THE LXR-ALPHA | NUCLEAR RECEPTOR, LXR HOMODIMER, LXR SIGNALING, ALTERNATIVE SPLICING, DNA-BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACTIVATOR, ACYLTRANSFERASE, CHROMOSOMAL REARRANGEMENT, ISOPEPTIDE BOND, PHOSPHOPROTEIN, PROTO-ONCOGENE, TRANSFERASE, UBL CONJUGATION
1hg4:A (SER383) to (ALA497) ULTRASPIRACLE LIGAND BINDING DOMAIN FROM DROSOPHILA MELANOGASTER | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING
1hg4:B (SER383) to (ALA497) ULTRASPIRACLE LIGAND BINDING DOMAIN FROM DROSOPHILA MELANOGASTER | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING
1hg4:F (SER383) to (ALA497) ULTRASPIRACLE LIGAND BINDING DOMAIN FROM DROSOPHILA MELANOGASTER | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING
2ham:A (SER306) to (GLY423) CRYSTAL STRUCTURE OF VDR LBD COMPLEXED TO 2ALPHA-PROPYL- CALCITRIOL | ALPHA-HELICAL SANDWICH, GENE REGULATION
2har:A (SER306) to (GLY423) CRYSTAL STRUCTURE OF VDR LBD IN COMPLEX WITH 2 ALPHA-(3- HYDROXY-1-PROPOXY) CALCITRIOL | ALPHA HELICAL SANDWICH, GENE REGULATION
3vn2:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA COMPLEXED WITH TELMISARTAN | SIGNALING PROTEIN
2hc4:A (THR334) to (LEU440) CRYSTAL STRUCTURE OF THE LBD OF VDR OF DANIO RERIO IN COMPLEX WITH CALCITRIOL | ALPHA HELICAL SANDWICH, GENE REGULATION
2hfp:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF PPAR GAMMA WITH N-SULFONYL-2-INDOLE CARBOXAMIDE LIGANDS | PPAR PPARGAMMA LBD, TRANSCRIPTION
3ixp:D (MET413) to (TRP526) CRYSTAL STRUCTURE OF THE ECDYSONE RECEPTOR BOUND TO BYI08346 | ANTI-PARALLEL ALPHA-HELICES, TRANSCRIPTION, TRANSCRIPTION REGULATION
3vso:A (ARG357) to (TYR473) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A GAMMA SELECTIVE AGONIST MEKT21 | MAINLY ALPHA, NUCLEAR RECEPTOR, TRANSCRIPTION
3vsp:A (ARG357) to (TYR473) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A GAMMA SELECTIVE AGONIST MEKT28 | MAINLY ALPHA, NUCLEAR RECEPTOR, TRANSCRIPTION
3vt3:A (THR302) to (LEU410) CRYSTAL STRUCTURES OF RAT VDR-LBD WITH R270L MUTATION | TRANSCRIPTION, HORMONE RECEPTOR
3vt4:A (THR302) to (THR411) CRYSTAL STRUCTURES OF RAT VDR-LBD WITH R270L MUTATION | TRANSCRIPTION, HORMONE RECEPTOR
3vt5:A (THR302) to (LEU410) CRYSTAL STRUCTURES OF RAT VDR-LBD WITH R270L MUTATION | TRANSCRIPTION, HORMONE RECEPTOR
3vt6:A (THR302) to (LEU410) CRYSTAL STRUCTURE OF RAT VDR-LBD WITH 2-SUBSTITUTED-16-ENE-22-THIA- 1ALPHA,25-DIHYDROXY-26,27-DIMETHYL-19-NORVITAMIN D3 | TRANSCRIPTION, HORMONE RECEPTOR
3vt8:A (THR302) to (LEU410) CRYSTAL STRUCTURES OF RAT VDR-LBD WITH W282R MUTATION | TRANSCRIPTION, HORMONE RECEPTOR
3vtb:A (THR302) to (THR411) CRYSTAL STRUCTURE OF RAT VITAMIN D RECEPTOR BOUND TO A PARTIAL AGONIST 25-ADAMANTYL-23-YNE-19-NORVITAMMIN D ADTK1 | TRANSCRIPTION, HORMONE RECEPTOR
3w0a:A (SER306) to (GLY423) CRYSTAL STRUCTURE ANALYSIS OF VITAMIN D RECEPTOR | VITAMIN D RECEPTOR, HORMONE RECEPTOR
3w0c:A (SER306) to (GLY423) CRYSTAL STRUCTURE ANALYSIS OF VITAMIN D RECEPTOR | VITAMIN D RECEPTOR, HORMONE RECEPTOR
3w0g:A (THR302) to (THR411) CRYSTAL STRUCTURE OF RAT VDR LIGAND BINDING DOMAIN IN COMPLEX WITH NOVEL NONSECOSTEROIDAL LIGANDS | GENE REGULATION, TRANSCRIPTION
3w0i:A (THR302) to (THR411) CRYSTAL STRUCTURE OF RAT VDR LIGAND BINDING DOMAIN IN COMPLEX WITH NOVEL NONSECOSTEROIDAL LIGANDS | GENE REGULATION, TRANSCRIPTION
3w0y:A (SER306) to (GLY423) CRYSTAL STRUCTURE ANALYSIS OF VITAMIN D RECEPTOR | VITAMIN D RECEPTOR, HORMONE RECEPTOR
4lto:A (ALA151) to (SER285) BACTERIAL SODIUM CHANNEL IN HIGH CALCIUM, I222 SPACE GROUP | CATION CHANNEL FOLD, COILED COIL SODIUM CHANNEL, PLASMA MEMBRANE, TRANSPORT PROTEIN
4lto:C (GLY149) to (SER285) BACTERIAL SODIUM CHANNEL IN HIGH CALCIUM, I222 SPACE GROUP | CATION CHANNEL FOLD, COILED COIL SODIUM CHANNEL, PLASMA MEMBRANE, TRANSPORT PROTEIN
4ltp:A (GLY149) to (ARG284) BACTERIAL SODIUM CHANNEL IN HIGH CALCIUM, I222 SPACE GROUP, CRYSTAL 2 | CATION CHANNEL FOLD, COILED COIL SODIUM CHANNEL, PLASMA MEMBRANE, TRANSPORT PROTEIN
4ltq:A (ILE150) to (ARG284) BACTERIAL SODIUM CHANNEL IN LOW CALCIUM, P42 SPACE GROUP | CATION CHANNEL FOLD, COILED COIL SODIUM CHANNEL, PLASMA MEMBRANE, TRANSPORT PROTEIN
4ltq:B (ILE150) to (SER285) BACTERIAL SODIUM CHANNEL IN LOW CALCIUM, P42 SPACE GROUP | CATION CHANNEL FOLD, COILED COIL SODIUM CHANNEL, PLASMA MEMBRANE, TRANSPORT PROTEIN
4ltq:C (ILE150) to (SER285) BACTERIAL SODIUM CHANNEL IN LOW CALCIUM, P42 SPACE GROUP | CATION CHANNEL FOLD, COILED COIL SODIUM CHANNEL, PLASMA MEMBRANE, TRANSPORT PROTEIN
4ltq:D (ILE150) to (SER285) BACTERIAL SODIUM CHANNEL IN LOW CALCIUM, P42 SPACE GROUP | CATION CHANNEL FOLD, COILED COIL SODIUM CHANNEL, PLASMA MEMBRANE, TRANSPORT PROTEIN
4ltq:H (ILE150) to (SER285) BACTERIAL SODIUM CHANNEL IN LOW CALCIUM, P42 SPACE GROUP | CATION CHANNEL FOLD, COILED COIL SODIUM CHANNEL, PLASMA MEMBRANE, TRANSPORT PROTEIN
4ltq:I (ILE150) to (SER285) BACTERIAL SODIUM CHANNEL IN LOW CALCIUM, P42 SPACE GROUP | CATION CHANNEL FOLD, COILED COIL SODIUM CHANNEL, PLASMA MEMBRANE, TRANSPORT PROTEIN
4ltq:J (ILE150) to (SER285) BACTERIAL SODIUM CHANNEL IN LOW CALCIUM, P42 SPACE GROUP | CATION CHANNEL FOLD, COILED COIL SODIUM CHANNEL, PLASMA MEMBRANE, TRANSPORT PROTEIN
4ltq:K (ILE150) to (SER285) BACTERIAL SODIUM CHANNEL IN LOW CALCIUM, P42 SPACE GROUP | CATION CHANNEL FOLD, COILED COIL SODIUM CHANNEL, PLASMA MEMBRANE, TRANSPORT PROTEIN
2hvc:A (TYR781) to (SER888) THE CRYSTAL STRUCTURE OF LIGAND-BINDING DOMAIN (LBD) OF HUMAN ANDROGEN RECEPTOR IN COMPLEX WITH A SELECTIVE MODULATOR LGD2226 | COMPLEXED WITH LGD2226, DNA-BINDING, STEROID-BINDING, LIGAND BINDING PROTEIN
1i7g:A (ARG348) to (TYR468) CRYSTAL STRUCTURE OF THE LIGAND BINDING DOMAIN FROM HUMAN PPAR-ALPHA IN COMPLEX WITH THE AGONIST AZ 242 | ANTI PARALLEL HELIX SANDWICH, TRANSCRIPTION
2hwq:A (ARG357) to (TYR473) STRUCTURAL BASIS FOR THE STRUCTURE-ACTIVITY RELATIONSHIPS OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONISTS | PPAR, LIGAND BINDING PROTEIN
2hwr:A (LYS358) to (TYR473) STRUCTURAL BASIS FOR THE STRUCTURE-ACTIVITY RELATIONSHIPS OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONISTS | PPAR, LIGAND BINDING PROTEIN
1i7i:A (ARG357) to (LYS474) CRYSTAL STRUCTURE OF THE LIGAND BINDING DOMAIN OF HUMAN PPAR-GAMMA IN COMPLEX WITH THE AGONIST AZ 242 | ANTI PARALLEL HELIX SANDWICH, TRANSCRIPTION
1i7i:B (LYS358) to (TYR473) CRYSTAL STRUCTURE OF THE LIGAND BINDING DOMAIN OF HUMAN PPAR-GAMMA IN COMPLEX WITH THE AGONIST AZ 242 | ANTI PARALLEL HELIX SANDWICH, TRANSCRIPTION
1ie8:A (SER306) to (GLY423) CRYSTAL STRUCTURE OF THE NUCLEAR RECEPTOR FOR VITAMIN D LIGAND BINDING DOMAIN BOUND TO KH1060 | VDR, KH1060, GENE REGULATION
3w5p:A (THR302) to (THR411) CRYSTAL STRUCTURE OF COMPLEXES OF VITAMIN D RECEPTOR LIGAND BINDING DOMAIN WITH LITHOCHOLIC ACID DERIVATIVES | ZINC-FINGER, NUCLEAR RECEPTOR-AGONIST COMPLEX, TRANSCRIPTION, RECEPTOR,TRANSCRIPTION REGULATION, ACTIVATOR, DNA-BINDING, METAL- BINDING, PHOSPHOPROTEIN, NUCLEUS
3w5t:A (THR302) to (THR411) CRYSTAL STRUCTURE OF COMPLEXES OF VITAMIN D RECEPTOR LIGAND BINDING DOMAIN WITH LITHOCHOLIC ACID DERIVATIVES | ZINC-FINGER, NUCLEAR RECEPTOR-AGONIST COMPLEX, TRANSCRIPTION, RECEPTOR, TRANSCRIPTION REGULATION, ACTIVATOR, DNA-BINDING, METAL- BINDING, PHOSPHOPROTEIN, NUCLEUS
3w5r:A (THR302) to (THR411) CRYSTAL STRUCTURE OF COMPLEXES OF VITAMIN D RECEPTOR LIGAND BINDING DOMAIN WITH LITHOCHOLIC ACID DERIVATIVES | ZINC-FINGER, NUCLEAR RECEPTOR-AGONIST COMPLEX, TRANSCRIPTION, RECEPTOR, TRANSCRIPTION REGULATION, ACTIVATOR ,DNA-BINDING, METAL- BINDING, PHOSPHOPROTEIN, NUCLEUS
2i4j:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN PPARGAMMA AND THE AGONIST LT160 (UREIDOFIBRATE DERIVATIVE) | BUNDLE OF ALPHA-HELICES AND A SMALL FOUR-STRANDED BETA- SHEET, TRANSCRIPTION
1uhl:B (GLU334) to (TRP443) CRYSTAL STRUCTURE OF THE LXRALFA-RXRBETA LBD HETERODIMER | LIGAND-BINDING DOMAIN, DNA BINDING PROTEIN
2i4p:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN PPARGAMMA AND THE PARTIAL AGONIST LT127 (UREIDOFIBRATE DERIVATIVE). STRUCTURE OBTAINED FROM CRYSTALS OF THE APO-FORM SOAKED FOR 30 DAYS. | BUNDLE OF ALPHA-HELICES AND A SMALL FOUR-STRANDED BETA- SHEET, TRANSCRIPTION
2i4z:A (ARG357) to (LYS474) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN PPARGAMMA AND THE PARTIAL AGONIST LT127 (UREIDOFIBRATE DERIVATIVE). THIS STRUCTURE HAS BEEN OBTAINED FROM CRYSTALS SOAKED FOR 6 HOURS. | BUNDLE OF ALPHA-HELICES AND A SMALL FOUR-STRANDED BETA- SHEET, TRANSCRIPTION
5a86:A (PRO322) to (LEU428) STRUCTURE OF PREGNANE X RECEPTOR IN COMPLEX WITH A SPHINGOSINE 1-PHOSPHATE RECEPTOR 1 ANTAGONIST | SIGNALING PROTEIN, PXR LIGAND, PXR AGONIST, CYP3A4 INDUCTION, NUCLEAR RECEPTOR
5a86:B (PRO322) to (LEU428) STRUCTURE OF PREGNANE X RECEPTOR IN COMPLEX WITH A SPHINGOSINE 1-PHOSPHATE RECEPTOR 1 ANTAGONIST | SIGNALING PROTEIN, PXR LIGAND, PXR AGONIST, CYP3A4 INDUCTION, NUCLEAR RECEPTOR
1ilg:A (PRO322) to (PHE429) CRYSTAL STRUCTURE OF APO HUMAN PREGNANE X RECEPTOR LIGAND BINDING DOMAIN | NUCLEAR RECEPTOR, MULTIPLE BINDING MODES, XENOBIOTIC, PROMISCUOUS, APO, GENE REGULATION
1upv:A (GLN346) to (TRP457) CRYSTAL STRUCTURE OF THE HUMAN LIVER X RECEPTOR BETA LIGAND BINDING DOMAIN IN COMPLEX WITH A SYNTHETIC AGONIST | RECEPTOR, NUCLEAR HORMONE RECEPTOR, LIGAND BINDING DOMAIN, LIVER X RECEPTOR, CRYSTAL STRUCTURE, TRANSCRIPTION FACTOR
4mg5:A (VAL422) to (ALA546) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH CHLORDECONE | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mg5:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH CHLORDECONE | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mg6:A (VAL422) to (ALA546) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BENZYLBUTYLPHTALATE | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mg6:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BENZYLBUTYLPHTALATE | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mg7:A (MET421) to (ALA546) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH FERUTININE | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mg8:B (VAL422) to (ALA546) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH ALPHA-ZEARALANOL | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mg9:A (VAL422) to (ALA546) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BUTYLPARABEN | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mg9:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BUTYLPARABEN | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mga:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH 4-TERT- OCTYLPHENOL | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mgb:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH TCBPA | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mgb:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH TCBPA | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
2iog:A (VAL422) to (MET543) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH COMPOUND 11F | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ER-ALPHA, ANTAGONIST, HORMONE
4mgc:A (MET421) to (ALA546) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BENZOPHENONE-2 | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mgc:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BENZOPHENONE-2 | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mgd:A (VAL422) to (ALA546) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH HPTE | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mgd:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH HPTE | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
3wj4:A (PRO366) to (LYS474) CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH TRIBUTYLTIN | PROTEIN-LIGAND COMPLEX, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION
3wj4:B (LYS358) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH TRIBUTYLTIN | PROTEIN-LIGAND COMPLEX, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION
3wj5:A (ARG357) to (LYS474) CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH TRIPHENYLTIN | PROTEIN-LIGAND COMPLEX, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION
3wj5:B (LYS358) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH TRIPHENYLTIN | PROTEIN-LIGAND COMPLEX, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION
2j14:A (LYS322) to (TYR437) 3,4,5-TRISUBSTITUTED ISOXAZOLES AS NOVEL PPARDELTA AGONISTS: PART2 | TRANSCRIPTION, NUCLEAR RECEPTOR FOLD, TRANSCRIPTION REGULATION, PPAR, ZINC, RECEPTOR, ACTIVATOR, FATTY ACIDS, NUCLEAR PROTEIN, ALTERNATIVE SPLICING, ZINC-FINGER, DNA-BINDING, METAL-BINDING
2j14:B (LYS322) to (LYS438) 3,4,5-TRISUBSTITUTED ISOXAZOLES AS NOVEL PPARDELTA AGONISTS: PART2 | TRANSCRIPTION, NUCLEAR RECEPTOR FOLD, TRANSCRIPTION REGULATION, PPAR, ZINC, RECEPTOR, ACTIVATOR, FATTY ACIDS, NUCLEAR PROTEIN, ALTERNATIVE SPLICING, ZINC-FINGER, DNA-BINDING, METAL-BINDING
5avi:A (VAL333) to (TRP443) CRYSTAL STRUCTURE OF LXRALPHA IN COMPLEX WITH TERT-BUTYL BENZOATE ANALOG, COMPOUND 4 | AGONIST, COMPLEX, TRANSCRIPTION
5avi:C (VAL333) to (TRP443) CRYSTAL STRUCTURE OF LXRALPHA IN COMPLEX WITH TERT-BUTYL BENZOATE ANALOG, COMPOUND 4 | AGONIST, COMPLEX, TRANSCRIPTION
5avl:A (VAL333) to (TRP443) CRYSTAL STRUCTURE OF LXRALPHA IN COMPLEX WITH TERT-BUTYL BENZOATE ANALOG, COMPOUND 32B | AGONIST, COMPLEX
2xhs:A (LEU912) to (ALA1023) CRYSTAL STRUCTURE OF THE LIGAND BINDING DOMAIN OF FUSHI TARAZU FACTOR 1 OF DROSOPHILA MELANOGASTER. | TRANSCRIPTION
2j7x:A (ILE328) to (ASN451) STRUCTURE OF ESTRADIOL-BOUND ESTROGEN RECEPTOR BETA LBD IN COMPLEX WITH LXXLL MOTIF FROM NCOA5 | ZINC-FINGER, NUCLEAR RECEPTOR, PHOSPHORYLATION, STEROID-BINDING, GLYCOPROTEIN, TRANSCRIPTION REGULATION, TRANSCRIPTION,
2xkw:A (ARG357) to (TYR473) LIGAND BINDING DOMAIN OF HUMAN PPAR-GAMMA IN COMPLEX WITH THE AGONIST PIOGLITAZONE | TRANSCRIPTION, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, GENE REGULATION, THIAZOLIDINEDIONE
3wwr:A (PRO312) to (GLY423) CRYSTAL STRUCTURE OF THE HUMAN VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH 1-((((1S,2R,6R,Z)-2,6-DIHYDROXY-4-((E)-2-((1R, 3AS,7AR)-1-((R)-6-HYDROXY-6-METHYLHEPTAN-2-YL)-7A-METHYLHEXAHYDRO-1H- INDEN-4(2H)-YLIDENE)ETHYLIDENE)-3-METHYLENECYCLOHEXYL)OXY)METHYL) CYCLOPROPANECARBONITRILE | HORMONE RECEPTOR, TRANSCRIPTION
5azt:A (LYS349) to (TYR464) TERNARY COMPLEX OF HPPARALPHA LIGAND BINDING DOMAIN, 17-OXODHA AND A SRC1 PEPTIDE | NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, LIGAND BINDING DOMAIN, ZINC-FINGER, DNA BINDING, TRANSCRIPTION, OBESITY, NUCLEUS, RECEPTOR, ACTIVATOR, OXIDIZED FATTY ACID, TRANSCRIPTION FACTOR, AGONIST, DUAL AGONIST, COVALENT, PPRE, NUCLEAR, CO-ACTIVATOR, DNA BINDING PROTEIN
5azt:B (LYS349) to (TYR464) TERNARY COMPLEX OF HPPARALPHA LIGAND BINDING DOMAIN, 17-OXODHA AND A SRC1 PEPTIDE | NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, LIGAND BINDING DOMAIN, ZINC-FINGER, DNA BINDING, TRANSCRIPTION, OBESITY, NUCLEUS, RECEPTOR, ACTIVATOR, OXIDIZED FATTY ACID, TRANSCRIPTION FACTOR, AGONIST, DUAL AGONIST, COVALENT, PPRE, NUCLEAR, CO-ACTIVATOR, DNA BINDING PROTEIN
5azv:A (GLU365) to (TYR473) CRYSTAL STRUCTURE OF HPPARGAMMA LIGAND BINDING DOMAIN COMPLEXED WITH 17-OXODHA | NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, LIGAND BINDING DOMAIN, ZINC-FINGER, DNA BINDING, TRANSCRIPTION, OBESITY, NUCLEUS, RECEPTOR, ACTIVATOR, OXIDIZED FATTY ACID, TRANSCRIPTION FACTOR, AGONIST, DUAL AGONIST, COVALENT, PPRE, NUCLEAR, DNA BINDING PROTEIN
3x1h:B (ARG357) to (LYS474) HPPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH 5-OXO- TRICOSAHEXAENOIC ACID | NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, LIGAND BINDING DOMAIN, DIABETES MELLITUS, ZINC-FINGER, DNA-BINDING, TRANSCRIPTION, OBESITY
3x1i:A (LYS358) to (TYR473) HPPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH 6-OXO- TETRACOSAHEXAENOIC ACID | NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, LIGAND BINDING DOMAIN, DIABETES MELLITUS, ZINC-FINGER, DNA-BINDING, TRANSCRIPTION, OBESITY
3x1i:B (LYS358) to (TYR473) HPPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH 6-OXO- TETRACOSAHEXAENOIC ACID | NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, LIGAND BINDING DOMAIN, DIABETES MELLITUS, ZINC-FINGER, DNA-BINDING, TRANSCRIPTION, OBESITY
3x31:A (SER306) to (GLY423) CRYSTAL STRUCTURE OF THE HUMAN VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH 7,8-CIS-14-EPI-1A,25-DIHYDROXY-19-NORVITAMIN D3 | HORMONE RECEPTOR, TRANSCRIPTION
3x36:A (SER306) to (GLY423) CRYSTAL STRUCTURE OF THE HUMAN VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH 7,8-CIS-1A,25-DIHYDROXY-19-NORVITAMIN D3 | TRANSCRIPTION, HORMONE RECEPTOR
2xyj:A (ARG321) to (MET440) NOVEL SULFONYLTHIADIAZOLES WITH AN UNUSUAL BINDING MODE AS PARTIAL DUAL PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR (PPAR) GAMMA-DELTA AGONISTS WITH HIGH POTENCY AND IN-VIVO EFFICACY | TRANSCRIPTION
2xyj:B (ARG321) to (MET440) NOVEL SULFONYLTHIADIAZOLES WITH AN UNUSUAL BINDING MODE AS PARTIAL DUAL PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR (PPAR) GAMMA-DELTA AGONISTS WITH HIGH POTENCY AND IN-VIVO EFFICACY | TRANSCRIPTION
2xyw:A (LYS322) to (TYR437) NOVEL SULFONYLTHIADIAZOLES WITH AN UNUSUAL BINDING MODE AS PARTIAL DUAL PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR (PPAR) GAMMA-DELTA AGONISTS WITH HIGH POTENCY AND IN-VIVO EFFICACY | DNA-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, RECEPTOR, ACTIVATOR, ZINC-FINGER
2xyw:B (LYS322) to (LYS438) NOVEL SULFONYLTHIADIAZOLES WITH AN UNUSUAL BINDING MODE AS PARTIAL DUAL PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR (PPAR) GAMMA-DELTA AGONISTS WITH HIGH POTENCY AND IN-VIVO EFFICACY | DNA-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, RECEPTOR, ACTIVATOR, ZINC-FINGER
2xyx:A (ILE328) to (TYR437) NOVEL SULFONYLTHIADIAZOLES WITH AN UNUSUAL BINDING MODE AS PARTIAL DUAL PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR (PPAR) GAMMA-DELTA AGONISTS WITH HIGH POTENCY AND IN-VIVO EFFICACY | DNA-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, RECEPTOR, ACTIVATOR, ZINC-FINGER
2xyx:B (ILE328) to (MET440) NOVEL SULFONYLTHIADIAZOLES WITH AN UNUSUAL BINDING MODE AS PARTIAL DUAL PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR (PPAR) GAMMA-DELTA AGONISTS WITH HIGH POTENCY AND IN-VIVO EFFICACY | DNA-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, RECEPTOR, ACTIVATOR, ZINC-FINGER
1k4w:A (SER335) to (THR440) X-RAY STRUCTURE OF THE ORPHAN NUCLEAR RECEPTOR ROR BETA LIGAND-BINDING DOMAIN IN THE ACTIVE CONFORMATION | LIGAND-BINDING DOMAIN, ALPHA-HELICAL SANDWICH, TRANSCRIPTIONALLY ACTIVE CONFORMATION, HORMONE/GROWTH FACTOR COMPLEX
1k74:D (PRO359) to (TYR473) THE 2.3 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE HETERODIMER OF THE HUMAN PPARGAMMA AND RXRALPHA LIGAND BINDING DOMAINS RESPECTIVELY BOUND WITH GW409544 AND 9-CIS RETINOIC ACID AND CO-ACTIVATOR PEPTIDES. | THE HETERODIMER OF THE NUCLEAR RECEPTOR LIGAND BINDING DOMAINS OF RXRALPHA AND PPARGAMMA BOUND RESPECTIVELY WITH 9-CIS RETINOIC ACID AND GW409544 AND COACTIVATOR PEPTIDES, TRANSCRIPTION
1k7l:A (MET355) to (ARG465) THE 2.5 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE HUMAN PPARALPHA LIGAND BINDING DOMAIN BOUND WITH GW409544 AND A CO-ACTIVATOR PEPTIDE. | THE 2.5 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE HUMAN PPARALPHA LIGAND BINDING DOMAIN BOUND WITH GW409544 AND A COACTIVATOR PEPTIDE, TRANSCRIPTION
1k7l:C (ARG348) to (TYR464) THE 2.5 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE HUMAN PPARALPHA LIGAND BINDING DOMAIN BOUND WITH GW409544 AND A CO-ACTIVATOR PEPTIDE. | THE 2.5 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE HUMAN PPARALPHA LIGAND BINDING DOMAIN BOUND WITH GW409544 AND A COACTIVATOR PEPTIDE, TRANSCRIPTION
1k7l:E (MET355) to (ARG465) THE 2.5 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE HUMAN PPARALPHA LIGAND BINDING DOMAIN BOUND WITH GW409544 AND A CO-ACTIVATOR PEPTIDE. | THE 2.5 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE HUMAN PPARALPHA LIGAND BINDING DOMAIN BOUND WITH GW409544 AND A COACTIVATOR PEPTIDE, TRANSCRIPTION
3zqt:A (MET780) to (GLN902) TARGETING THE BINDING FUNCTION 3 SITE OF THE ANDROGEN RECEPTOR THROUGH IN SILICO MOLECULAR MODELING | TRANSCRIPTION, SMALL MOLECULE INHIBITOR
2yat:A (ASP426) to (ALA546) CRYSTAL STRUCTURE OF ESTRADIOL DERIVED METAL CHELATE AND ESTROGEN RECEPTOR-LIGAND BINDING DOMAIN COMPLEX | TRANSCRIPTION
1kkq:A (LYS349) to (TYR468) CRYSTAL STRUCTURE OF THE HUMAN PPAR-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH AN ANTAGONIST GW6471 AND A SMRT COREPRESSOR MOTIF | NUCLEAR COREPRESSOR NUCLEAR HORMONE RECEPTORS ANTAGONIST, TRANSCRIPTION
1kkq:C (LYS349) to (MET467) CRYSTAL STRUCTURE OF THE HUMAN PPAR-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH AN ANTAGONIST GW6471 AND A SMRT COREPRESSOR MOTIF | NUCLEAR COREPRESSOR NUCLEAR HORMONE RECEPTORS ANTAGONIST, TRANSCRIPTION
1kkq:D (PHE351) to (TYR468) CRYSTAL STRUCTURE OF THE HUMAN PPAR-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH AN ANTAGONIST GW6471 AND A SMRT COREPRESSOR MOTIF | NUCLEAR COREPRESSOR NUCLEAR HORMONE RECEPTORS ANTAGONIST, TRANSCRIPTION
2lvj:A (ARG10) to (PHE77) SOLUTION STRUCTURE OF HEMI-MG-BOUND PHL P 7 | EF-HAND PROTEIN, MAGNESIUM-BINDING PROTEIN, ALLERGEN
1knu:A (ARG357) to (TYR473) LIGAND BINDING DOMAIN OF THE HUMAN PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR GAMMA IN COMPLEX WITH A SYNTHETIC AGONIST | PPAR, NUCLEAR RECEPTOR, TRANSCRIPTION, GENE REGULATION, AGONIST COMPLEX, DNA BINDING PROTEIN
1knu:B (ARG357) to (TYR473) LIGAND BINDING DOMAIN OF THE HUMAN PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR GAMMA IN COMPLEX WITH A SYNTHETIC AGONIST | PPAR, NUCLEAR RECEPTOR, TRANSCRIPTION, GENE REGULATION, AGONIST COMPLEX, DNA BINDING PROTEIN
1x7r:A (MET421) to (ALA546) CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR ALPHA COMPLEXED WITH GENISTEIN | ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN RECEPTOR ALPHA, ER-ALPHA, ESTROGEN, NUCLEAR RECEPT TRANSCRIPTION FACTOR, AGONIST
2npa:A (MET355) to (ARG465) THE CRYSTAL STRUCTURE OF THE HUMAN PPARAPLPHA LIGAND BINDING DOMAIN IN COMPLEX WITH A A-HYDROXYIMINO PHENYLPROPANOIC ACID | PROTEIN-AGONIST COMPLEX, TRANSCRIPTION
2npa:C (MET355) to (ARG465) THE CRYSTAL STRUCTURE OF THE HUMAN PPARAPLPHA LIGAND BINDING DOMAIN IN COMPLEX WITH A A-HYDROXYIMINO PHENYLPROPANOIC ACID | PROTEIN-AGONIST COMPLEX, TRANSCRIPTION
2yja:B (MET421) to (LEU549) STAPLED PEPTIDES BINDING TO ESTROGEN RECEPTOR ALPHA. | HORMONE RECEPTOR-PEPTIDE COMPLEX
1l2i:A (MET421) to (ALA546) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH (R,R)-5,11-CIS-DIETHYL-5,6,11,12- TETRAHYDROCHRYSENE-2,8-DIOL AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ESTROGEN, AGONIST, COACTIVATOR, TRANSCRIPTION RECEPTOR/COACTIVATOR COMPLEX
1l2i:B (MET421) to (HIS547) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH (R,R)-5,11-CIS-DIETHYL-5,6,11,12- TETRAHYDROCHRYSENE-2,8-DIOL AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ESTROGEN, AGONIST, COACTIVATOR, TRANSCRIPTION RECEPTOR/COACTIVATOR COMPLEX
2ylp:A (TYR781) to (SER888) TARGETING THE BINDING FUNCTION 3 SITE OF THE ANDROGEN RECEPTOR THROUGH IN SILICO MOLECULAR MODELING | HORMONE RECEPTOR, BINDING FUNCTION 3
2nv7:B (ILE373) to (ALA497) CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-555 | ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
2nxx:A (LEU296) to (GLY403) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE T.CASTANEUM (COLEOPTERA) HETERODIMER ECRUSP BOUND TO PONASTERONE A | HORMONE RECEPTOR, APO AND HOLO LIGAND BINDING POCKET, HORMONE/GROWTH FACTOR COMPLEX
2nxx:B (TYR292) to (GLU402) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE T.CASTANEUM (COLEOPTERA) HETERODIMER ECRUSP BOUND TO PONASTERONE A | HORMONE RECEPTOR, APO AND HOLO LIGAND BINDING POCKET, HORMONE/GROWTH FACTOR COMPLEX
2nxx:C (LEU296) to (GLY403) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE T.CASTANEUM (COLEOPTERA) HETERODIMER ECRUSP BOUND TO PONASTERONE A | HORMONE RECEPTOR, APO AND HOLO LIGAND BINDING POCKET, HORMONE/GROWTH FACTOR COMPLEX
2nxx:D (TYR292) to (GLY403) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE T.CASTANEUM (COLEOPTERA) HETERODIMER ECRUSP BOUND TO PONASTERONE A | HORMONE RECEPTOR, APO AND HOLO LIGAND BINDING POCKET, HORMONE/GROWTH FACTOR COMPLEX
1xj7:A (MET780) to (SER888) COMPLEX ANDROGEN RECEPTOR LBD AND RAC3 PEPTIDE | ANDROGEN RECEPTOR COACTIVATORS LXXLL MOTIF, HORMONE/GROWTH FACTOR COMPLEX
4a4v:A (ARG357) to (TYR473) LIGAND BINDING DOMAIN OF HUMAN PPAR GAMMA IN COMPLEX WITH AMORFRUTIN 2 | RECEPTOR, AGONIST, DIABETES, INSULIN RESISTANCE
4oj4:A (ARG357) to (TYR477) CRYSTAL STRUCTURE OF V290M PPARGAMMA MUTANT IN COMPLEX WITH DICLOFENAC | MAINLY ALPHA HELIX, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, RXR, TRANSCRIPTION
1xnn:A (TYR781) to (SER888) CRYSTAL STRUCTURE OF THE RAT ANDROGEN RECEPTOR LIGAND BINDING DOMAIN T877A MUTANT COMPLEX WITH (3A-ALPHA-,4- ALPHA 7-ALPHA-,7A-ALPHA-)-3A,4,7,7A-TETRAHYDRO-2-(4-NITRO- 1-NAPHTHALENYL)-4,7-ETHANO-1H-ISOINDOLE-1,3(2H)-DIONE. | ANDROGEN RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, LIGAND-BINDING DOMAIN, HORMONE/GROWTH FACTOR COMPLEX
1m13:A (PRO322) to (PHE429) CRYSTAL STRUCTURE OF THE HUMAN PREGANE X RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH HYPERFORIN, A CONSTITUENT OF ST. JOHN'S WORT | NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, PROTEIN-LIGAND COMPLEX, TRANSCRIPTION
4okx:A (TYR781) to (SER888) CRYSTAL STRUCTURE OF W741L-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE | ALPHA-HELIX, HORMONE/GROWTH FACTOR RECEPTOR, PHOSPHORYLATION, HORMONE RECEPTOR-PEPTIDE COMPLEX, SIGNAL TRANSDUCTION
1xp1:A (MET421) to (MET543) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH COMPOUND 15 | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ER-ALPHA, ANTAGONIST, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
1xp6:A (MET421) to (MET543) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH COMPOUND 16 | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ER-ALPHA, ANTAGONIST, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
1xpc:A (MET421) to (MET543) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH COMPOUND 19 | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ER-ALPHA, ANTAGONIST, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
1xq3:A (TYR781) to (GLY909) CRYSTAL STRUCTURE OF THE HUMAN ANDROGEN RECEPTOR LIGAND BINDING DOMAIN BOUND WITH R1881 | CRYSTAL STRUCTURE; HUMAN ANDROGEN RECEPTOR LIGAND BINDING DOMAIN; R1881, TRANSCRIPTION
4oni:B (ALA422) to (ALA538) STRUCTURE OF HUMAN ORPHAN RECEPTOR LRH1 BOUND TO TWO BACTERIAL PHOSPHOLIPIDS | ALPHA HELICAL SANDWICH FOLD, NUCLEAR RECEPTOR, CO-FACTOR BINDING, NUCLEAR PROTEIN
2zk0:A (ARG357) to (TYR473) HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA LIGAND BINDING DOMAIN | ANTI PARALLEL HELIX SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
2zk0:B (ARG357) to (TYR473) HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA LIGAND BINDING DOMAIN | ANTI PARALLEL HELIX SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
2zk1:A (ARG357) to (TYR473) HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH 15-DEOXY-DELTA12,14- PROSTAGLANDIN J2 | ANTI PARALLEL HELIX SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
2zk2:A (ARG357) to (TYR473) HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH GLUTATHION CONJUGATED 15-DEOXY-DELTA12,14-PROSTAGLANDIN J2 | ANTI PARALLEL HELIX SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
2zk2:B (MET364) to (TYR473) HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH GLUTATHION CONJUGATED 15-DEOXY-DELTA12,14-PROSTAGLANDIN J2 | ANTI PARALLEL HELIX SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
2zk3:A (ARG357) to (TYR473) HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH 8-OXO- EICOSATETRAENOIC ACID | ANTI PARALLEL HELIX SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
2zk3:B (PRO359) to (TYR473) HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH 8-OXO- EICOSATETRAENOIC ACID | ANTI PARALLEL HELIX SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
2zk5:A (GLU365) to (TYR473) HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH NITRO-233 | ANTI PARALLEL HELIX SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
2zk5:B (PRO359) to (TYR473) HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH NITRO-233 | ANTI PARALLEL HELIX SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
2zk6:A (GLU365) to (TYR473) HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH C8-BODIPY | ANTI PARALLEL HELIX SANDWICH, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
2zk6:B (PRO359) to (TYR473) HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH C8-BODIPY | ANTI PARALLEL HELIX SANDWICH, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3kdt:A (LYS349) to (ARG465) CRYSTAL STRUCTURE OF PEROXISOME PROLIFERATOR-ACTIVATEDECEPTOR ALPHA (PPARALPHA) COMPLEX WITH N-3-((2-(4-CHLOROPHENYL)-5-METHYL-1,3- OXAZOL-4-YL)METHOXY)BENZYL)-N-(METHOXYCARBONYL)GLYCINE | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION REGULATION, ACTIVATOR, DNA- BINDING, LIPID-BINDING, RECEPTOR, TRANSCRIPTION, HORMONE RECEPTOR
3kdu:A (MET355) to (ARG465) CRYSTAL STRUCTURE OF PEROXISOME PROLIFERATOR-ACTIVATEDECEPTOR ALPHA (PPARALPHA) COMPLEX WITH N-3-((2-(4-CHLOROPHENYL)-5-METHYL-1,3- OXAZOL-4-YL)METHOXY)BENZYL)-N-((4-METHYLPHENOXY)CARBONYL)GLYCINE | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION REGULATION, ACTIVATOR, DNA- BINDING, LIPID-BINDING, RECEPTOR, TRANSCRIPTION, HORMONE RECEPTOR
3kdu:B (MET355) to (TYR464) CRYSTAL STRUCTURE OF PEROXISOME PROLIFERATOR-ACTIVATEDECEPTOR ALPHA (PPARALPHA) COMPLEX WITH N-3-((2-(4-CHLOROPHENYL)-5-METHYL-1,3- OXAZOL-4-YL)METHOXY)BENZYL)-N-((4-METHYLPHENOXY)CARBONYL)GLYCINE | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION REGULATION, ACTIVATOR, DNA- BINDING, LIPID-BINDING, RECEPTOR, TRANSCRIPTION, HORMONE RECEPTOR
3kfc:A (VAL347) to (ASP458) COMPLEX STRUCTURE OF LXR WITH AN AGONIST | NUCLEAR RECEPTOR, LXR, LIVER X RECEPTOR, LXR AGONIST, LXR LIGAND, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3kfc:B (GLN346) to (TRP457) COMPLEX STRUCTURE OF LXR WITH AN AGONIST | NUCLEAR RECEPTOR, LXR, LIVER X RECEPTOR, LXR AGONIST, LXR LIGAND, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3kfc:D (GLN346) to (TRP457) COMPLEX STRUCTURE OF LXR WITH AN AGONIST | NUCLEAR RECEPTOR, LXR, LIVER X RECEPTOR, LXR AGONIST, LXR LIGAND, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
2zmh:A (THR302) to (LEU410) CRYSTAL STRUCTURE OF RAT VITAMIN D RECEPTOR BOUND TO ADAMANTYL VITAMIN D ANALOGS: STRUCTURAL BASIS FOR VITAMIN D RECEPTOR ANTAGONISM AND/OR PARTIAL AGONISM | NUCLEAR RECEPTOR-ANTAGONIST COMPLEX, DNA-BINDING, METAL- BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACTIVATOR
2znn:A (LYS349) to (ARG465) HUMAN PPAR ALPHA LIGAND BINDING DOMAIN IN COMPLEX WITH A SYNTHETIC AGONIST TIPP703 | NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, PPAR, ACTIVATOR, DNA- BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
2znp:A (PHE374) to (TYR473) HUMAN PPAR DELTA LIGAND BINDING DOMAIN IN COMPLEX WITH A SYNTHETIC AGONIST TIPP204 | NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, PPAR, ACTIVATOR, DNA- BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
2znp:B (LYS358) to (TYR473) HUMAN PPAR DELTA LIGAND BINDING DOMAIN IN COMPLEX WITH A SYNTHETIC AGONIST TIPP204 | NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, PPAR, ACTIVATOR, DNA- BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
2zno:A (ARG357) to (LYS474) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A SYNTHETIC AGONIST TIPP703 | NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, PPAR, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
1m7w:D (SER253) to (GLY367) HNF4A LIGAND BINDING DOMAIN WITH BOUND FATTY ACID | TRANSCRIPTION FACTOR
1xvp:D (GLU237) to (PRO341) CRYSTAL STRUCTURE OF CAR/RXR HETERODIMER BOUND WITH SRC1 PEPTIDE, FATTY ACID AND CITCO | CAR, RXR, CITCO, SRC1, DNA BINDING PROTEIN
1y0s:A (LYS358) to (TYR473) CRYSTAL STRUCTURE OF PPAR DELTA COMPLEXED WITH GW2331 | PPAR, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
1y0s:B (LYS358) to (TYR473) CRYSTAL STRUCTURE OF PPAR DELTA COMPLEXED WITH GW2331 | PPAR, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
2zvt:A (ASP362) to (LYS474) CYS285SER MUTANT PPARGAMMA LIGAND-BINDING DOMAIN COMPLEXED WITH 15-DEOXY-DELTA12,14-PROSTAGLANDIN J2 | ANTI PARALLEL HELIX SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
2zvt:B (LYS358) to (TYR473) CYS285SER MUTANT PPARGAMMA LIGAND-BINDING DOMAIN COMPLEXED WITH 15-DEOXY-DELTA12,14-PROSTAGLANDIN J2 | ANTI PARALLEL HELIX SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
4ozt:E (GLY406) to (ASP517) CRYSTAL STRUCTURE OF THE LIGAND BINDING DOMAINS OF THE BOVICOLA OVIS ECDYSONE RECEPTOR ECR/USP HETERODIMER (PONA CRYSTAL) | ECDYSONE RECEPTOR, USP, PONA, TRANSCRIPTION
2zxm:A (THR302) to (THR411) A NEW CLASS OF VITAMIN D RECEPTOR LIGANDS THAT INDUCE STRUCTURAL REARRANGEMENT OF THE LIGAND-BINDING POCKET | NUCLEAR RECEPTOR-ANTAGONIST COMPLEX, TRANSCRIPTION, DNA- BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACTIVATOR
2zxn:A (THR302) to (LEU410) A NEW CLASS OF VITAMIN D RECEPTOR LIGANDS THAT INDUCE STRUCTURAL REARRANGEMENT OF THE LIGAND-BINDING POCKET | NUCLEAR RECEPTOR-AGONIST COMPLEX, TRANSCRIPTION, DNA- BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACTIVATOR
3kmg:A (GLU365) to (TYR473) THE X-RAY CRYSTAL STRUCTURE OF PPAR-GAMMA IN COMPLEX WITH AN INDOLE DERIVATIVE MODULATOR, GSK538, AND AN SRC-1 PEPTIDE | PPAR-GAMMA, PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR, TELMISARTAN, DIABETES, MODULATOR, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3kmg:D (GLU365) to (TYR473) THE X-RAY CRYSTAL STRUCTURE OF PPAR-GAMMA IN COMPLEX WITH AN INDOLE DERIVATIVE MODULATOR, GSK538, AND AN SRC-1 PEPTIDE | PPAR-GAMMA, PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR, TELMISARTAN, DIABETES, MODULATOR, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3kpz:A (SER306) to (VAL421) CRYSTAL STRUCTURE OF A NOVEL VITAMIN D3 ANALOGUE, ZK203278 SHOWING DISSOCIATED PROFILE | NUCLEAR RECEPTOR, AGONIST, DNA-BINDING, TRANSCRIPTION REGULATION, TRANSCRIPTION-HORMONE COMPLEX
3a2j:A (SER306) to (GLY423) CRYSTAL STRUCTURE OF THE HUMAN VITAMIN D RECEPTOR (H305F/H397F) LIGAND BINDING DOMAIN COMPLEXED WITH TEI-9647 | HORMONE/GROWTH FACTOR RECEPTOR, DNA-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC- FINGER, ACTIVATOR, DISEASE MUTATION, RECEPTOR, HORMONE RECEPTOR
3a3z:X (SER306) to (GLY423) CRYSTAL STRUCTURE OF THE HUMAN VDR LIGAND BINDING DOMAIN BOUND TO THE SYNTHETIC AGONIST COMPOUND 2ALPHA-METHYL-AMCR277A(C23S) | TRANSCRIPTION, STRUCTURAL GENOMICS, SPINE2, STRUCTURAL PROTEOMICS IN EUROPE 2, GENE REGULATION
3a40:X (SER306) to (GLY423) CRYSTAL STRUCTURE OF THE HUMAN VDR LIGAND BINDING DOMAIN BOUND TO THE SYNTHETIC AGONIST COMPOUND 2ALPHA-METHYL-AMCR277B(C23R) | TRANSCRIPTION, STRUCTURAL GENOMICS, SPINE2, STRUCTURAL PROTEOMICS IN EUROPE 2, GENE REGULATION
1yim:A (VAL422) to (LEU544) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH COMPOUND 4 | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ER-ALPHA, ANTAGONIST, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
3a78:A (SER306) to (GLY423) CRYSTAL STRUCTURE OF THE HUMAN VDR LIGAND BINDING DOMAIN BOUND TO THE NATURAL METABOLITE 1ALPHA,25-DIHYDROXY-3-EPI-VITAMIN D3 | TRANSCRIPTION, GENE REGULATION, DISEASE MUTATION, DNA-BINDING, METAL- BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION REGULATION, ZINC-FINGER
1yje:A (TRP481) to (ASP593) CRYSTAL STRUCTURE OF THE RNGFI-B LIGAND-BINDING DOMAIN | NGFI-B, NUR77, NUCLEAR RECEPTOR, LIGAND-BINDING DOMAIN, NOVEL COREGULATOR INTERFACE, CELL-SPECIFIC, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS, TRANSCRIPTION
1mzn:A (ALA344) to (GLU456) CRYSTAL STRUCTURE AT 1.9 ANGSTROEMS RESOLUTION OF THE HOMODIMER OF HUMAN RXR ALPHA LIGAND BINDING DOMAIN BOUND TO THE SYNTHETIC AGONIST COMPOUND BMS 649 AND A COACTIVATOR PEPTIDE | TRANSCRIPTION, NUCLEAR RECEPTOR, RETINOIC ACID RECEPTORS, AGONIST
1ymt:A (SER343) to (ALA459) MOUSE SF-1 LBD | NUCLEAR RECEPTOR, SF-1, LIGAND-BINDING DOMAIN, LIGAND, PHOSPHATIDYL GLYCEROL, CO-REPRESSOR PEPTIDE, TRANSCRIPTION
1yok:A (ALA422) to (HIS537) CRYSTAL STRUCTURE OF HUMAN LRH-1 BOUND WITH TIF-2 PEPTIDE AND PHOSPHATIDYLGLYCEROL | LRH-1, TIF-1, PHOSPHATIDYLGLYCEROL, TRANSCRIPTION
1yow:A (LEU343) to (GLN457) HUMAN STEROIDOGENIC FACTOR 1 LBD WITH BOUND CO-FACTOR PEPTIDE | STEROIDOGENIC FACTOR 1, SF1, PHOSPHOLIPID, PHOSPHATIDYL ETHANOLAMINE, PHOSPHATIDYL GLYCEROL, TRANSCRIPTION
1yp0:A (LEU345) to (ALA459) STRUCTURE OF THE STEROIDOGENIC FACTOR-1 LIGAND BINDING DOMAIN BOUND TO PHOSPHOLIPID AND A SHP PEPTIDE MOTIF | LIGAND DEPENDENT NUCLEAR RECEPTOR, STEROIDOGENIC FACTOR-1, NR5A1, HELICAL SANDWICH FOLD, LBD FOLD, TRANSCRIPTION
3l03:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE AND ESTETROL (ESTRA-1,3,5(10)-TRIENE-3,15 ALPHA, 16ALPHA,17BETA-TETROL) | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, ESTETROL, DNA-BINDING, GLYCOPROTEIN, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER, ACTIVATOR
3l03:B (VAL422) to (ALA546) CRYSTAL STRUCTURE OF HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE AND ESTETROL (ESTRA-1,3,5(10)-TRIENE-3,15 ALPHA, 16ALPHA,17BETA-TETROL) | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, ESTETROL, DNA-BINDING, GLYCOPROTEIN, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER, ACTIVATOR
3l0e:A (VAL347) to (ASP458) X-RAY CRYSTAL STRUCTURE OF A POTENT LIVER X RECEPTOR MODULATOR | HLXR-BETA, HUMAN LIVER X RECEPTOR-BETA, SULFONAMIDE MODULATOR, DNA- BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER, ACTIVATOR, PHOSPHOPROTEIN
1n4h:A (ASP129) to (THR233) CHARACTERIZATION OF LIGANDS FOR THE ORPHAN NUCLEAR RECEPTOR RORBETA | ALPHA-HELICAL SANDWICH, PROTEIN-PEPTIDE-LIGAND COMPLEX, HORMONE/GROWTH FACTOR COMPLEX
3l1b:A (SER362) to (TRP473) COMPLEX STRUCTURE OF FXR LIGAND-BINDING DOMAIN WITH A TETRAHYDROAZEPINOINDOLE COMPOUND | NUCLEAR RECEPTOR, FXR AGONIST, FXR LIGAND-BINDING DOMAIN, NUCLEUS, RECEPTOR, TRANSCRIPTION REGULATION, TRANSCRIPTION
3ads:A (ARG357) to (TYR473) HUMAN PPARGAMMA LIGAND-BINDING DOMAIN IN COMPLEX WITH INDOMETHACIN | NUCLEAR RECEPTOR, LIGAND-DEPENDENT TRANSCRIPTION FACTOR, LIGAND- BINDING DOMAIN, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, DNA- BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3ads:B (PRO359) to (TYR473) HUMAN PPARGAMMA LIGAND-BINDING DOMAIN IN COMPLEX WITH INDOMETHACIN | NUCLEAR RECEPTOR, LIGAND-DEPENDENT TRANSCRIPTION FACTOR, LIGAND- BINDING DOMAIN, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, DNA- BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3adu:A (GLU365) to (TYR473) HUMAN PPARGAMMA LIGAND-BINDING DOMAIN IN COMPLEX WITH 5-METHOXY-INDOLE ACETATE | NUCLEAR RECEPTOR, LIGAND-DEPENDENT TRANSCRIPTION FACTOR, LIGAND- BINDING DOMAIN, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, DNA- BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3adv:A (ARG357) to (LYS474) HUMAN PPARGAMMA LIGAND-BINDING DOMAIN IN COMPLEX WITH SEROTONIN | NUCLEAR RECEPTOR, LIGAND-DEPENDENT TRANSCRIPTION FACTOR, LIGAND- BINDING DOMAIN, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, DNA- BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3adw:A (MET364) to (TYR473) HUMAN PPARGAMMA LIGAND-BINDING DOMAIN IN COMPLEX WITH 5-METHOXY-INDOLE ACETATE AND 15-OXO-EICOSATETRAENOIC ACID | NUCLEAR RECEPTOR, LIGAND-DEPENDENT TRANSCRIPTION FACTOR, LIGAND- BINDING DOMAIN, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, DNA- BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3adw:B (PRO359) to (TYR473) HUMAN PPARGAMMA LIGAND-BINDING DOMAIN IN COMPLEX WITH 5-METHOXY-INDOLE ACETATE AND 15-OXO-EICOSATETRAENOIC ACID | NUCLEAR RECEPTOR, LIGAND-DEPENDENT TRANSCRIPTION FACTOR, LIGAND- BINDING DOMAIN, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, DNA- BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3adx:A (ARG357) to (TYR473) HUMAN PPARGAMMA LIGAND-BINDING DOMAIN IN COMPLEX WITH INDOMETHACIN AND NITRO-233 | NUCLEAR RECEPTOR, LIGAND-DEPENDENT TRANSCRIPTION FACTOR, LIGAND- BINDING DOMAIN, ACTIVATOR, DIABETES MELLITUS, DISEASE MUTATION, DNA- BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3l3z:A (TYR781) to (SER888) CRYSTAL STRUCTURE OF DHT-BOUND ANDROGEN RECEPTOR IN COMPLEX WITH THE THIRD MOTIF OF STEROID RECEPTOR COACTIVATOR 3 | ANDROGEN RECEPTOR, LIGAND BINDING DOMAIN, STEROID RECEPTOR COACTIVATOR 3, 5-ALPHA-DIHYDROTESTOSTERONE (DHT), PROSTATE CANCER, PROTEIN BINDING
5did:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DIFLUORO-SUBSTITUTED A-CD RING ESTROGEN DERIVATIVE (1S,3AR,5S, 7AS)-5-(2,3-DIFLUORO-4-HYDROXYPHENYL)-7A-METHYLOCTAHYDRO-1H-INDEN-1- OL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5die:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A TRIFLUORO-SUBSTITUTED A-CD RING ESTROGEN DERIVATIVE (1S,3AR, 5S,7AS)-7A-METHYL-5-(2,3,5-TRIFLUORO-4-HYDROXYPHENYL)OCTAHYDRO-1H- INDEN-1-OL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dig:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A TRIFLUOROMETHYL-SUBSTITUTED A-CD RING ESTROGEN DERIVATIVE (1S, 3AR,5S,7AS)-5-[4-HYDROXY-2-(TRIFLUOROMETHYL)PHENYL]-7A- METHYLOCTAHYDRO-1H-INDEN-1-OL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
1yuc:B (ALA422) to (ALA538) HUMAN NUCLEAR RECEPTOR LIVER RECEPTOR HOMOLOGUE-1, LRH-1, BOUND TO PHOSPHOLIPID AND A FRAGMENT OF HUMAN SHP | LIVER RECEPTOR HOMOLOGUE 1; NUCLEAR RECEPTOR LIGAND BINDING DOMAIN; LRH-1; PHOSPHOLIPID; SHP; SMALL HETERODIMER PARTNER, TRANSCRIPTION REGULATION
5dk9:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A PHENYLAMINO-SUBSTITUTED ETHYL TRIARYL-ETHYLENE DERIVATIVE 4, 4'-{2-[3-(PHENYLAMINO)PHENYL]BUT-1-ENE-1,1-DIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dkg:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A T-BUTYL-SUBSTITUTED, METHYL, TRIARYL-ETHYLENE DERIVATIVE 4,4'- [2-(4-TERT-BUTYLPHENYL)PROP-1-ENE-1,1-DIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dkg:B (MET421) to (LEU549) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A T-BUTYL-SUBSTITUTED, METHYL, TRIARYL-ETHYLENE DERIVATIVE 4,4'- [2-(4-TERT-BUTYLPHENYL)PROP-1-ENE-1,1-DIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dks:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 2-NAPHTHYLAMINO-SUBSTITUTED, ETHYL, TRIARYL-ETHYLENE DERIVATIVE 4,4'-{2-[3-(NAPHTHALEN-1-YLAMINO)PHENYL]BUT-1-ENE-1,1- DIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dks:B (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 2-NAPHTHYLAMINO-SUBSTITUTED, ETHYL, TRIARYL-ETHYLENE DERIVATIVE 4,4'-{2-[3-(NAPHTHALEN-1-YLAMINO)PHENYL]BUT-1-ENE-1,1- DIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dl4:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A PHENYLAMINO-SUBSTITUTED, METHYL, TRIARYL-ETHYLENE DERIVATIVE 4,4'-{2-[3-(PHENYLAMINO)PHENYL]PROP-1-ENE-1,1-DIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dl4:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A PHENYLAMINO-SUBSTITUTED, METHYL, TRIARYL-ETHYLENE DERIVATIVE 4,4'-{2-[3-(PHENYLAMINO)PHENYL]PROP-1-ENE-1,1-DIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4ple:A (ALA422) to (ALA538) HUMAN NUCLEAR RECEPTOR LIVER RECEPTOR HOMOLOGUE-1, LRH-1, BOUND TO AN E. COLI PHOSPHOLIPID AND A FRAGMENT OF TIF-2 | NUCLEAR RECEPTOR, PHOSPHOLIPID, TRANSCRIPTION
4ple:C (ALA422) to (ALA538) HUMAN NUCLEAR RECEPTOR LIVER RECEPTOR HOMOLOGUE-1, LRH-1, BOUND TO AN E. COLI PHOSPHOLIPID AND A FRAGMENT OF TIF-2 | NUCLEAR RECEPTOR, PHOSPHOLIPID, TRANSCRIPTION
4ple:E (ALA422) to (HIS537) HUMAN NUCLEAR RECEPTOR LIVER RECEPTOR HOMOLOGUE-1, LRH-1, BOUND TO AN E. COLI PHOSPHOLIPID AND A FRAGMENT OF TIF-2 | NUCLEAR RECEPTOR, PHOSPHOLIPID, TRANSCRIPTION
4ple:G (ALA422) to (ALA538) HUMAN NUCLEAR RECEPTOR LIVER RECEPTOR HOMOLOGUE-1, LRH-1, BOUND TO AN E. COLI PHOSPHOLIPID AND A FRAGMENT OF TIF-2 | NUCLEAR RECEPTOR, PHOSPHOLIPID, TRANSCRIPTION
5dlr:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A TRIARYL-ETHYLENE COMPOUND 4,4'-(2-PHENYLETHENE-1,1-DIYL) DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dlr:B (GLY420) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A TRIARYL-ETHYLENE COMPOUND 4,4'-(2-PHENYLETHENE-1,1-DIYL) DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dmc:A (MET421) to (HIS547) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A NITRILE-SUBSTITUTED TRIARYL-ETHYLENE DERIVATIVE 3,3-BIS(4- HYDROXYPHENYL)-2-PHENYLPROP-2-ENENITRILE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dmc:B (VAL422) to (HIS547) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A NITRILE-SUBSTITUTED TRIARYL-ETHYLENE DERIVATIVE 3,3-BIS(4- HYDROXYPHENYL)-2-PHENYLPROP-2-ENENITRILE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dmf:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 4-FLUOROPHENYLAMINO-SUBSTITUTED, METHYL TRIARYL-ETHYLENE DERIVATIVE 4,4'-(2-{3-[(4-FLUOROPHENYL)AMINO]PHENYL}PROP-1-ENE-1,1- DIYL)DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4pp6:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH RESVERATROL | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, NUCLEUS, PROTEIN BINDING
4prg:A (ARG357) to (TYR473) 0072 PARTIAL AGONIST PPAR GAMMA COCRYSTAL | THIAZOLIDINONE, LIGAND-BINDING DOMAIN, NUCLEAR RECEPTOR, ORPHAN RECEPTOR
4prg:B (PHE374) to (TYR473) 0072 PARTIAL AGONIST PPAR GAMMA COCRYSTAL | THIAZOLIDINONE, LIGAND-BINDING DOMAIN, NUCLEAR RECEPTOR, ORPHAN RECEPTOR
4prg:C (ARG357) to (TYR473) 0072 PARTIAL AGONIST PPAR GAMMA COCRYSTAL | THIAZOLIDINONE, LIGAND-BINDING DOMAIN, NUCLEAR RECEPTOR, ORPHAN RECEPTOR
4ami:A (ASN204) to (PRO321) TURKEY BETA1 ADRENERGIC RECEPTOR WITH STABILISING MUTATIONS AND BOUND BIASED AGONIST BUCINDOLOL | MEMBRANE PROTEIN, 7TMR BETA1-ADRENOCEPTOR, STABILISING MUTATIONS, BIASED AGONIST
5dp0:A (GLU419) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 4-FLUOROPHENYLAMINO-SUBSTITUTED TRIARYL-ETHYLENE DERIVATIVE 4, 4'-(2-{3-[(4-FLUOROPHENYL)AMINO]PHENYL}ETHENE-1,1-DIYL)DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dp0:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 4-FLUOROPHENYLAMINO-SUBSTITUTED TRIARYL-ETHYLENE DERIVATIVE 4, 4'-(2-{3-[(4-FLUOROPHENYL)AMINO]PHENYL}ETHENE-1,1-DIYL)DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5drj:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DICHLORO-SUBSTITUTED, 3-METHYL 2,5-DIARYLTHIOPHENE-CORE LIGAND 4,4'-(3-METHYLTHIENE-2,5-DIYL)BIS(3-CHLOROPHENOL) | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5drj:B (MET421) to (LEU549) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DICHLORO-SUBSTITUTED, 3-METHYL 2,5-DIARYLTHIOPHENE-CORE LIGAND 4,4'-(3-METHYLTHIENE-2,5-DIYL)BIS(3-CHLOROPHENOL) | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5drm:A (MET421) to (ALA546) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DICHLORO-SUBSTITUTED, 2,5-DIARYLTHIOPHENE-CORE LIGAND 4,4'- THIENE-2,5-DIYLBIS(3-CHLOROPHENOL) | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5drm:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DICHLORO-SUBSTITUTED, 2,5-DIARYLTHIOPHENE-CORE LIGAND 4,4'- THIENE-2,5-DIYLBIS(3-CHLOROPHENOL) | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dsh:A (LYS358) to (TYR473) HUMAN PPARGAMMA LIGAND BINDING DMAIN COMPLEXED WITH SB1406 IN A COVALENT BONDED FORM | PPARGAMMA, ANTAGONIST, TRANSCRIPTION-TRANSFERASE COMPLEX
4pwl:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN PPARGAMMA-LBD AND THE S ENANTIOMER OF MBX-102 (METAGLIDASEN) | ALPHA-HELICES, SMALL FOUR-STRANDED BETA-SHEET, ACTIVATOR, DNA- BINDING, NUCLEUS, OBESITY, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION X-RAY DIFFRACTION, TRANSCRIPTION FACTOR, RXR-ALPHA
4pwl:B (ARG357) to (TYR473) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN PPARGAMMA-LBD AND THE S ENANTIOMER OF MBX-102 (METAGLIDASEN) | ALPHA-HELICES, SMALL FOUR-STRANDED BETA-SHEET, ACTIVATOR, DNA- BINDING, NUCLEUS, OBESITY, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION X-RAY DIFFRACTION, TRANSCRIPTION FACTOR, RXR-ALPHA
1zdt:A (GLY341) to (ALA458) THE CRYSTAL STRUCTURE OF HUMAN STEROIDOGENIC FACTOR-1 | STEROIDOGENIC FACTOR-1, NUCLEAR RECEPTOR, PHOLPHOLIPID, PHOSPHATIDYLETHANOLAMINE, TRANSCRIPTION
5dtv:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DIMETHYL-SUBSTITUTED, 3,4-DIARYLTHIOPHENE DIOXIDE CORE LIGAND | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
3an3:A (ARG357) to (TYR473) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A GAMMA SELECTIVE AGONIST MO3S | MAINLY ALPHA, NUCLEAR RECEPTOR, TRANSCRIPTION
3an3:B (PRO359) to (ILE472) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A GAMMA SELECTIVE AGONIST MO3S | MAINLY ALPHA, NUCLEAR RECEPTOR, TRANSCRIPTION
3an4:A (ARG357) to (LYS474) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A GAMMA SELECTIVE AGONIST MO4R | MAINLY ALPHA, NUCLEAR RECEPTOR, TRANSCRIPTION
3an4:B (LYS358) to (TYR473) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A GAMMA SELECTIVE AGONIST MO4R | MAINLY ALPHA, NUCLEAR RECEPTOR, TRANSCRIPTION
5due:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A PARA-HYDROXYL-SUBSTITUTED, SULFOXIDE-BRIDGED OXABICYCLIC HEPTENE SULFONATE (SOBHS)-2 ANALOG 4-HYDROXYPHENYL (1S,2S,4S,5S,6R, 7S)-5,6-BIS(4-HYDROXY-2-METHYLPHENYL)-7-THIABICYCLO[2.2.1]HEPTANE-2- SULFONATE 7-OXIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5due:B (MET421) to (LEU549) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A PARA-HYDROXYL-SUBSTITUTED, SULFOXIDE-BRIDGED OXABICYCLIC HEPTENE SULFONATE (SOBHS)-2 ANALOG 4-HYDROXYPHENYL (1S,2S,4S,5S,6R, 7S)-5,6-BIS(4-HYDROXY-2-METHYLPHENYL)-7-THIABICYCLO[2.2.1]HEPTANE-2- SULFONATE 7-OXIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
1zgy:A (ARG357) to (TYR473) STRUCTURAL AND BIOCHEMICAL BASIS FOR SELECTIVE REPRESSION OF THE ORPHAN NUCLEAR RECEPTOR LRH-1 BY SHP | PROTEIN-PEPTIDE COMPLEX, TRANSCRIPTION
5duh:A (VAL418) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A SULFOXIDE-BRIDGED OXABICYCLIC HEPTENE SULFONATE (SOBHS)-3 ANALOG PHENYL (1S,2S,4S,7S)-5,6-BIS(4-HYDROXY-3-METHYLPHENYL)-7- THIABICYCLO[2.2.1]HEPT-5-ENE-2-SULFONATE 7-OXIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5duh:B (MET421) to (ASN532) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A SULFOXIDE-BRIDGED OXABICYCLIC HEPTENE SULFONATE (SOBHS)-3 ANALOG PHENYL (1S,2S,4S,7S)-5,6-BIS(4-HYDROXY-3-METHYLPHENYL)-7- THIABICYCLO[2.2.1]HEPT-5-ENE-2-SULFONATE 7-OXIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dv3:A (LYS358) to (LYS474) HUMAN PPARGAMMA LIGAND BINDING DMAIN COMPLEXED WITH SB1405 IN A COVALENT BONDED FORM | PPARGAMMA, ANTAGONIST, TRANSCRIPTION-TRANSFERASE COMPLEX
5dv6:A (LYS358) to (TYR473) HUMAN PPARGAMMA LIGAND BINDING DMAIN COMPLEXED WITH SB1404 IN A COVALENT BONDED FORM | PPARGAMMA, ANTAGONIST, TRANSCRIPTION-TRANSFERASE COMPLEX
5dv8:A (MET364) to (TYR473) HUMAN PPARGAMMA LIGAND BINDING DMAIN COMPLEXED WITH SB1451 IN A COVALENT BONDED FORM | PPARGAMMA, ANTAGONIST, TRANSCRIPTION-TRANSFERASE COMPLEX
5dvc:A (LYS358) to (TYR473) HUMAN PPARGAMMA LIGAND BINDING DMAIN COMPLEXED WITH SB1453 IN A COVALENT BONDED FORM | PPARGAMMA, ANTAGONIST, TRANSCRIPTION-TRANSFERASE COMPLEX
5dwe:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 2-CHLORO-SUBSTITUTED TRIARYL-IMINE ANALOG 4,4'-[(2- CHLOROPHENYL)CARBONIMIDOYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dwe:B (GLY420) to (LEU549) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 2-CHLORO-SUBSTITUTED TRIARYL-IMINE ANALOG 4,4'-[(2- CHLOROPHENYL)CARBONIMIDOYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dwj:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A RESORCINYL 4-FLUORO-SUBSTITUTED DIARYL-IMINE ANALOG 4-[(E)- [(4-FLUOROPHENYL)IMINO](4-HYDROXYPHENYL)METHYL]BENZENE-1,3-DIOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dwj:B (MET421) to (LEU549) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A RESORCINYL 4-FLUORO-SUBSTITUTED DIARYL-IMINE ANALOG 4-[(E)- [(4-FLUOROPHENYL)IMINO](4-HYDROXYPHENYL)METHYL]BENZENE-1,3-DIOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dwl:A (LYS358) to (TYR473) HUMAN PPARGAMMA LIGAND BINDING DMAIN IN COMPLEX WITH SR1664 | PPARGAMMA, ANTAGONIST, TRANSCRIPTION-TRANSFERASE COMPLEX
3lmp:A (LYS358) to (TYR473) CRYSTAL STRUCTURE OF THE PPARGAMMA-LBD COMPLEXED WITH A CERCOSPORAMIDE DERIVATIVE MODULATOR | THREE-LAYERED ALPHA-HELICAL SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
5dxg:A (MET421) to (ARG548) ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN Y537S MUTANT IN COMPLEX WITH STAPLED PEPTIDE SRC2-P5 | ESTROGEN RECEPTOR, HORMONE, STAPLED PEPTIDE, PEPTIDE MIMETIC, BREAST CANCER, HORMONE RECEPTOR-PEPTIDE COMPLEX
5dxg:B (MET421) to (ARG548) ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN Y537S MUTANT IN COMPLEX WITH STAPLED PEPTIDE SRC2-P5 | ESTROGEN RECEPTOR, HORMONE, STAPLED PEPTIDE, PEPTIDE MIMETIC, BREAST CANCER, HORMONE RECEPTOR-PEPTIDE COMPLEX
1zky:A (MET421) to (ARG548) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH OBCP-3M AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
1zky:B (MET421) to (ALA546) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH OBCP-3M AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
5dxb:A (VAL422) to (ARG548) ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN Y537S MUTANT IN COMPLEX WITH STAPLED PEPTIDE SRC2-P1 AND ESTRADIOL | ESTROGEN RECEPTOR ALPHA, SOMATIC MUTATAION, STAPLED PEPTIDE, PEPTIDE MIMETIC, HORMONE RECEPTOR, BREAST CANCER, HORMONE RECEPTOR-PEPTIDE COMPLEX
5dxb:B (MET421) to (ARG548) ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN Y537S MUTANT IN COMPLEX WITH STAPLED PEPTIDE SRC2-P1 AND ESTRADIOL | ESTROGEN RECEPTOR ALPHA, SOMATIC MUTATAION, STAPLED PEPTIDE, PEPTIDE MIMETIC, HORMONE RECEPTOR, BREAST CANCER, HORMONE RECEPTOR-PEPTIDE COMPLEX
5dxe:A (MET421) to (ASP545) ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN Y537S MUTANT IN COMPLEX WITH STAPLED PEPTIDE SRC2-P4 AND ESTRADIOL | ESTROGEN RECEPTOR ALPHA, STAPLED PEPTIDE, PEPTIDE MIMETIC, BREAST CANCER, HORMONE, SOMATIC MUTATION, HORMONE RECEPTOR-PEPTIDE COMPLEX
5dxe:B (MET421) to (ARG548) ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN Y537S MUTANT IN COMPLEX WITH STAPLED PEPTIDE SRC2-P4 AND ESTRADIOL | ESTROGEN RECEPTOR ALPHA, STAPLED PEPTIDE, PEPTIDE MIMETIC, BREAST CANCER, HORMONE, SOMATIC MUTATION, HORMONE RECEPTOR-PEPTIDE COMPLEX
5dxk:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(9S)-BICYCLO[3.3.1]NON-9- YLMETHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dxk:B (VAL422) to (ALA546) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(9S)-BICYCLO[3.3.1]NON-9- YLMETHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dxm:A (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 3-[(E)-(1S,5S)-BICYCLO[3.3.1]NON-9- YLIDENE(4-HYDROXYPHENYL)METHYL]PHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dxp:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4-[(E)-(1S,5S)-BICYCLO[3.3.1]NON-9- YLIDENE(PHENYL)METHYL]PHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dxq:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(1S,5S)-BICYCLO[3.3.1]NON-9- YLIDENEMETHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dxq:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(1S,5S)-BICYCLO[3.3.1]NON-9- YLIDENEMETHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dy8:B (MET421) to (LEU549) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-{[(3S)-3- ETHYLCYCLOHEXYLIDENE]METHANEDIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dz0:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(4-METHYLCYCLOHEXYLIDENE) METHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dz0:B (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(4-METHYLCYCLOHEXYLIDENE) METHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dz1:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(4-ETHYLCYCLOHEXYLIDENE) METHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dz1:B (GLY420) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(4-ETHYLCYCLOHEXYLIDENE) METHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dz3:B (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-{[4-(FLUOROMETHYL) CYCLOHEXYLIDENE]METHANEDIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dzh:A (VAL422) to (VAL533) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-{[4-(2-HYDROXYETHYL) CYCLOHEXYLIDENE]METHANEDIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dzh:B (GLU419) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-{[4-(2-HYDROXYETHYL) CYCLOHEXYLIDENE]METHANEDIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dzi:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-{[(3S)-3-(2-HYDROXYETHYL) CYCLOHEXYLIDENE]METHANEDIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5e15:A (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-{[4-(2-HYDROXYETHYL) CYCLOHEXYLIDENE]METHANEDIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5e15:B (MET421) to (LEU549) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-{[4-(2-HYDROXYETHYL) CYCLOHEXYLIDENE]METHANEDIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4q50:A (VAL422) to (ASP545) THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN D538G MUTANT IN COMPLEX WITH 4-HYDROXYTAMOXIFEN | ACQUIRED SERM-RESISTANCE, BREAST CANCER, ACTIVATING MUTATION, SERM-ER STRUCTURE, ALPHA HELIX, NUCLEAR HORMONE RECEPTOR, HORMONE BINDING PROTEIN
4q50:B (MET421) to (ASP545) THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN D538G MUTANT IN COMPLEX WITH 4-HYDROXYTAMOXIFEN | ACQUIRED SERM-RESISTANCE, BREAST CANCER, ACTIVATING MUTATION, SERM-ER STRUCTURE, ALPHA HELIX, NUCLEAR HORMONE RECEPTOR, HORMONE BINDING PROTEIN
4q50:D (VAL422) to (ASP545) THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN D538G MUTANT IN COMPLEX WITH 4-HYDROXYTAMOXIFEN | ACQUIRED SERM-RESISTANCE, BREAST CANCER, ACTIVATING MUTATION, SERM-ER STRUCTURE, ALPHA HELIX, NUCLEAR HORMONE RECEPTOR, HORMONE BINDING PROTEIN
4q50:E (MET421) to (ASP545) THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN D538G MUTANT IN COMPLEX WITH 4-HYDROXYTAMOXIFEN | ACQUIRED SERM-RESISTANCE, BREAST CANCER, ACTIVATING MUTATION, SERM-ER STRUCTURE, ALPHA HELIX, NUCLEAR HORMONE RECEPTOR, HORMONE BINDING PROTEIN
4q50:H (MET421) to (LEU544) THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN D538G MUTANT IN COMPLEX WITH 4-HYDROXYTAMOXIFEN | ACQUIRED SERM-RESISTANCE, BREAST CANCER, ACTIVATING MUTATION, SERM-ER STRUCTURE, ALPHA HELIX, NUCLEAR HORMONE RECEPTOR, HORMONE BINDING PROTEIN
5e19:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE METHYL {4-[BIS(4-HYDROXYPHENYL) METHYLIDENE]CYCLOHEXYL}ACETATE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5e1c:A (GLY420) to (LEU549) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE DIMETHYL {(1S)-3-[BIS(4- HYDROXYPHENYL)METHYLIDENE]CYCLOHEXYL}PROPANEDIOATE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5e1c:B (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE DIMETHYL {(1S)-3-[BIS(4- HYDROXYPHENYL)METHYLIDENE]CYCLOHEXYL}PROPANEDIOATE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
3aun:A (THR302) to (LEU410) CRYSTAL STRUCTURE OF THE RAT VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH YR335 AND A SYNTHETIC PEPTIDE CONTAINING THE NR2 BOX OF DRIP 205 | BINDING SITES, BIPHENYL COMPOUNDS, PROTEIN BINDING, TERTIARY, RATS, RECEPTORS, CALCITRIOL, VITAMIN D, TRANSCRIPTION
3auq:A (SER306) to (PHE422) CRYSTAL STRUCTURE OF THE HUMAN VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH YNE-DIENE TYPE ANALOG OF ACTIVE 14-EPI-2ALPHA- METHYL-19-NORVITAMIN D3 | HORMONE RECEPTOR, TRANSCRIPTION
4qe6:A (SER358) to (ILE468) FXR WITH CDCA AND NCOA-2 PEPTIDE | RECEPTOR, BILE ACID RECEPTOR DNA, TRANSCRIPTION
4qe8:A (ASP359) to (TRP469) FXR WITH DM175 AND NCOA-2 PEPTIDE | RECEPTOR, BILE ACID RECEPTOR DNA, TRANSCRIPTION
3az1:A (SER306) to (GLY423) CRYSTAL STRUCTURE ANALYSIS OF VITAMIN D RECEPTOR | VITAMIN D RECEPTOR, HORMONE RECEPTOR
3az3:A (SER306) to (GLY423) CRYSTAL STRUCTURE ANALYSIS OF VITAMIN D RECEPTOR | VITAMIN D RECEPTOR, HORMONE RECEPTOR
3b0q:A (ARG357) to (TYR473) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH MCC555 | NUCLEAR RECEPTOR, TRANSCRIPTION
3b0q:B (LYS358) to (TYR473) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH MCC555 | NUCLEAR RECEPTOR, TRANSCRIPTION
3b0t:A (SER306) to (GLY423) HUMAN VDR LIGAND BINDING DOMAIN IN COMPLEX WITH MAXACALCITOL | NUCLEAR RECEPTOR, TRANSCRIPTION, GENE REGULATION
3b1m:A (LYS358) to (TYR473) CRYSTAL STRUCTURE OF THE PPARGAMMA-LBD COMPLEXED WITH A CERCOSPORAMIDE DERIVATIVE MODULATOR CERCO-A | TRANSCRIPTION
3m7r:A (SER306) to (GLY423) CRYSTAL STRUCTURE OF VDR H305Q MUTANT | LIGAND BINDING DOMAIN, TRANSCRIPTION, STRUCTURAL GENOMICS, SPINE, STRUCTURAL PROTEOMICS IN EUROPE
3b3k:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN PPARGAMMA AND THE FULL AGONIST LT175 | BUNDLE OF ALPHA-HELICES, SMALL FOUR-STRNDED BETA-SHEET, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHORYLATION, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
5ehj:A (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(4AR,8AR)-OCTAHYDRONAPHTHALEN- 2(1H)-YLIDENEMETHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5ehj:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(4AR,8AR)-OCTAHYDRONAPHTHALEN- 2(1H)-YLIDENEMETHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
2acl:B (VAL331) to (TRP441) LIVER X-RECEPTOR ALPHA LIGAND BINDING DOMAIN WITH SB313987 | NUCLEAR HORMONE RECEPTOR LIGAND BINDING DOMAIN TRANSCRIPTION FACTOR THREE LAYERED A-HELIX FOLD
2acl:D (VAL331) to (TRP441) LIVER X-RECEPTOR ALPHA LIGAND BINDING DOMAIN WITH SB313987 | NUCLEAR HORMONE RECEPTOR LIGAND BINDING DOMAIN TRANSCRIPTION FACTOR THREE LAYERED A-HELIX FOLD
2acl:F (VAL331) to (TRP441) LIVER X-RECEPTOR ALPHA LIGAND BINDING DOMAIN WITH SB313987 | NUCLEAR HORMONE RECEPTOR LIGAND BINDING DOMAIN TRANSCRIPTION FACTOR THREE LAYERED A-HELIX FOLD
4qjr:A (SER342) to (ALA458) CRYSTAL STRUCTURE OF HUMAN NUCLEAR RECEPTOR SF-1 (NR5A1) BOUND TO ITS HORMONE PIP3 AT 2.4 A RESOLUTION | NUCLEAR HORMONE RECEPTOR, NR5A1, SF-1 LIGAND BINDINGNUCLEAR DOMAIN, REGULATORY LIGANDS, TRANSCRIPTION, TRANSCRIPTION REGULATION, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, PARTNERSHIP FOR STEM CELL BIOLOGY, PIP3, PIP2, NUCLEUS, NUCLEAR PHOSPHATIDYLINOSITOL PHOSPHATES, TRANSCRIPTION FACTOR-HORMONE COMPLEX
4qk4:A (SER342) to (ALA458) CRYSTAL STRUCTURE OF HUMAN NUCLEAR RECEPTOR SF-1 (NR5A1) BOUND TO PIP2 AT 2.8 A RESOLUTION | NUCLEAR HORMONE RECEPTOR, NR5A1, SF-1 LIGAND BINDING DOMAIN, REGULATORY LIGANDS, TRANSCRIPTION, TRANSCRIPTION REGULATION, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, PARTNERSHIP FOR STEM CELL BIOLOGY, PIP3, PIP2, NUCLEUS, NUCLEAR PHOSPHATIDYLINOSITOL PHOSPHATES, TRANSCRIPTION FACTOR-HORMONE COMPLEX
4bcr:A (LYS349) to (TYR464) STRUCTURE OF PPARALPHA IN COMPLEX WITH WY14643 | TRANSCRIPTION, NUCLEAR RECEPTOR, PPAR, FIBRATE
4bcr:B (LYS349) to (TYR464) STRUCTURE OF PPARALPHA IN COMPLEX WITH WY14643 | TRANSCRIPTION, NUCLEAR RECEPTOR, PPAR, FIBRATE
3bej:A (ASP359) to (TRP469) STRUCTURE OF HUMAN FXR IN COMPLEX WITH MFA-1 AND CO- ACTIVATOR PEPTIDE | FXR, BAR, NR1H4, BILE ACID RECEPTOR, NHR, NUCLEAR RECEPTOR, ACTIVATOR, ALTERNATIVE SPLICING, DNA-BINDING, METAL-BINDING, NUCLEUS, REPRESSOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACYLTRANSFERASE, CHROMOSOMAL REARRANGEMENT, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, TRANSFERASE, UBL CONJUGATION, TRANSCRIPTION/TRANSFERASE COMPLEX, TRANSCRIPTION REGULATOR
5f9b:A (ARG357) to (TYR473) X-RAY CRYSTAL STRUCTURE OF PPARGAMMA IN THE COMPLEX WITH CAULOPHYLLOGENIN | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, DIABETES, BUNDLE OF ALPHA- HELICES, TRANSCRIPTION
4r06:A (GLU365) to (TYR473) CRYSTAL STRUCTURE OF SR2067 BOUND TO PPARGAMMA | NUCLEAR RECEPTOR, LIGAND BINDING PROTEIN, TRANSCRIPTION
4r2u:D (GLU365) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA IN COMPLEX WITH SR1664 | NUCLEAR RECEPTOR LIGAND BINDING DOMAIN, TRANSCRIPTION
4r6s:A (LYS358) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMMA IN COMPLEX WITH SR1663 | NUCLEAR RECEPTOR LIGAND BINDING DOMAIN, TRANSCRIPTION
4r6s:B (LYS358) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMMA IN COMPLEX WITH SR1663 | NUCLEAR RECEPTOR LIGAND BINDING DOMAIN, TRANSCRIPTION
4rak:B (GLN346) to (TRP457) CRYSTAL STRUCTURE OF NUCLEAR RECEPTOR SUBFAMILY 1, GROUP H, MEMBER 2 (LXRB) COMPLEXED WITH PARTIAL AGONIST | NHR, NR1H2, LXR-B, LXRB, UNR, NER-I, RIP15, NER, LIGAND BINDING DOMAIN, NUCLEAR HORMONE RECEPTOR, RXR, TRANSCRIPTION-AGONIST COMPLEX
3cds:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN PPAR-GAMMA AND THE AGONIST LT248 (CLOFIBRIC ACID ANALOGUE) | BUNDLE OF ALPHA-HELICES AND A SMALL FOUR-STRANDED BETA- SHEET, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
3cjw:A (MET289) to (LEU381) CRYSTAL STRUCTURE OF THE HUMAN COUP-TFII LIGAND BINDING DOMAIN | COUP-TFII, NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, ORPHAN RECEPTOR, THREE-LAYERED HELICAL SANDWICH, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
3noa:A (PRO359) to (TYR473) CRYSTAL STRUCTURE OF HUMAN PPAR-GAMMA LIGAND BINDING DOMAIN COMPLEX WITH A POTENCY IMPROVED AGONIST | HYPOGLYCEMIC AGENTS, MODELS, MOLECULAR, PPAR ALPHA, PPAR GAMMA, PROTEIN ISOFORMS, QUINOLINES, STRUCTURE-ACTIVITY RELATIONSHIP, THIAZOLIDINEDIONES, TRANSCRIPTION
5fqp:A (MET421) to (LEU544) SELECTIVE ESTROGEN RECEPTOR DOWNREGULATOR ANTAGONISTS: TETRAHYDROISOQUINOLINE PHENOLS 1. | SIGNALING PROTEIN, BREAST CANCER, ESTROGEN RECEPTOR DOWNREGULATOR, FULVESTRANT, THIQ, NUCLEAR HORMONE RECEPTOR
5fqs:A (MET421) to (LEU544) SELECTIVE ESTROGEN RECEPTOR DOWNREGULATOR ANTAGONISTS: TETRAHYDROISOQUINOLINE PHENOLS 3. | SIGNALING PROTEIN, BREAST CANCER, ESTROGEN RECEPTOR DOWNREGULATOR, FULVESTRANT, THIQ, NUCLEAR HORMONE RECEPTOR
5fqt:A (MET421) to (LEU544) SELECTIVE ESTROGEN RECEPTOR DOWNREGULATOR ANTAGONISTS: TETRAHYDROISOQUINOLINE PHENOLS 4. | SIGNALING PROTEIN, BREAST CANCER, ESTROGEN RECEPTOR DOWNREGULATOR, FULVESTRANT, THIQ, NUCLEAR HORMONE RECEPTOR
3cs4:A (SER306) to (GLY423) STRUCTURE-BASED DESIGN OF A SUPERAGONIST LIGAND FOR THE VITAMIN D NUCLEAR RECEPTOR | VDR, SUPERAGONIST, DISEASE MUTATION, DNA-BINDING, METAL- BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, GENE REGULATION
3cs8:A (MET364) to (TYR473) STRUCTURAL AND BIOCHEMICAL BASIS FOR THE BINDING SELECTIVITY OF PPARG TO PGC-1A | COACTIVATOR, NUCLEAR RECEPTOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL- BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, RNA-BINDING, NUCLEAR PROTEIN
4ci4:A (LYS349) to (TYR464) STRUCTURAL BASIS FOR GL479 A DUAL PEROXISOME PROLIFERATOR- ACTIVATED RECEPTOR ALPHA AGONIST | TRANSFERASE, DUAL AGONIST, PPAR, NUCLEAR RECEPTOR, GL479
4ci5:A (MET364) to (TYR473) STRUCTURAL BASIS FOR GL479 A DUAL PEROXISOME PROLIFERATOR- ACTIVATED RECEPTOR GAMMA AGONIST | NUCLEAR PROTEIN, DUAL AGONIST, NUCLEAR RECEPTOR
3o1e:A (THR334) to (LEU440) STRUCTURE-FUNCTION OF GEMINI DERIVATIVES WITH TWO DIFFERENT SIDE CHAINS AT C-20, GEMINI-0072 AND GEMINI-0097. | TRANSCRIPTION FACTOR, VITAMIN D, NUCLEUS, TRANSCRIPTION-TRANSCRIPTION ACTIVATOR COMPLEX
3cwd:A (ARG357) to (TYR473) MOLECULAR RECOGNITION OF NITRO-FATTY ACIDS BY PPAR GAMMA | PPAR GAMMA, NUCLEAR RECEPTOR, SRC1-2 MOTIF, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
4rwv:A (ALA422) to (ALA538) CRYSTAL STRUCTURE OF PIP3 BOUND HUMAN NUCLEAR RECEPTOR LRH-1 (LIVER RECEPTOR HOMOLOG 1, NR5A2) IN COMPLEX WITH A CO-REGULATOR DAX-1 (NR0B1) PEPTIDE AT 1.86 A RESOLUTION | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, PF00104 FAMILY, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, PARTNERSHIP FOR STEM CELL BIOLOGY, TRANSCRIPTION
4rzg:B (TRP151) to (LEU265) CRYSTAL STRUCTURE ANALYSIS OF THE DNPA-BOUNDED NUR77 LIGAND BINDING DOMAIN | NUR77-LBD AND DNPA COMPLEX, TRANSCRIPTION
4s0t:A (PRO322) to (PHE429) STRUCTURE OF HUMAN PREGNANE X RECEPTOR LIGAND BINDING DOMAIN BOUND WITH ADNECTIN-1 AND COMPOUND-1 | NUCLEAR RECEPTOR, MULTIPLE BINDING MODES, XENOBIOTIC, PROMISCUOUS, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION
4s15:A (ASP398) to (THR512) CRYSTAL STRUCTURE OF THE ORPHAN NUCLEAR RECEPTOR RORALPHA LIGAND- BINDING DOMAIN IN COMPLEX WITH 4ALPHA-CABOXYL, 4BETA-METHYL- ZYMOSTEROL (4ACD8) | TRANSCRIPTION FACTOR, TRANSCRIPTION
4s15:B (ASP398) to (ARG500) CRYSTAL STRUCTURE OF THE ORPHAN NUCLEAR RECEPTOR RORALPHA LIGAND- BINDING DOMAIN IN COMPLEX WITH 4ALPHA-CABOXYL, 4BETA-METHYL- ZYMOSTEROL (4ACD8) | TRANSCRIPTION FACTOR, TRANSCRIPTION
3d57:B (VAL348) to (GLU460) TR VARIANT D355R | THYROID HORMONE RECEPTOR, LIGAND BINDING DOMAIN, D355R MUTANT, HOMODIMER, ALTERNATIVE SPLICING, DEAFNESS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, HORMONE, TRANSCRIPTION RECEPTOR
3d5f:A (LYS358) to (LYS474) CRYSTAL STRUCTURE OF PPAR-DELTA COMPLEX | NUCLEAR RECEPTOR, ACTIVATOR, ALTERNATIVE SPLICING, DNA- BINDING, METAL-BINDING, NUCLEUS, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
3d5f:B (LYS358) to (TYR473) CRYSTAL STRUCTURE OF PPAR-DELTA COMPLEX | NUCLEAR RECEPTOR, ACTIVATOR, ALTERNATIVE SPLICING, DNA- BINDING, METAL-BINDING, NUCLEUS, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
3dct:A (ASP359) to (TRP469) FXR WITH SRC1 AND GW4064 | FXR, NUCLEAR RECEPTOR, GW4064, ALPHA-HELICAL SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, REPRESSOR, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACYLTRANSFERASE, CHROMOSOMAL REARRANGEMENT, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, TRANSFERASE, UBL CONJUGATION, TRANSCRIPTION/TRANSCRIPTION ACTIVATOR COMPLEX
3ogt:A (SER306) to (GLY423) DESIGN, CHEMICAL SYNTHESIS, FUNCTIONAL CHARACTERIZATION AND CRYSTAL STRUCTURE OF THE SIDECHAIN ANALOGUE OF 1,25-DIHYDROXYVITAMIN D3. | TRANSCRIPTION FACTOR, VITAMIN D, NUCLEUS, TRANSCRIPTION
4tv1:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH PROPYLPARABEN | NUCLEAR HORMONE RECEPTOR, LIGAND BINDING DOMAIN, ENDOCRINE DISRUPTOR, ENVIRONMENTAL COMPOUND, HORMONE RECEPTOR
3oki:C (SER362) to (TRP458) CRYSTAL STRUCTURE OF HUMAN FXR IN COMPLEX WITH (2S)-2-[2-(4- CHLOROPHENYL)-1H-BENZIMIDAZOL-1-YL]-N,2-DICYCLOHEXYLETHANAMIDE | NUCLEAR RECEPTOR, CHOLESTEROL, BILE ACID, DNA-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, LIGAND BINDING DOMAIN TRANSCRIPTION REGULATION, COACTIVATOR, FXR ALTERNATIVE SPLICING, HORMONE RECEPTOR
3omk:A (SER362) to (SER457) CRYSTAL STRUCTURE OF HUMAN FXR IN COMPLEX WITH (2S)-2-[2-(4- CHLOROPHENYL)-5,6-DIFLUORO-1H-BENZIMIDAZOL-1-YL]-2-CYCLOHEXYL-N-(2- METHYLPHENYL)ETHANAMIDE | NUCLEAR RECEPTOR, CHOLESTEROL, BILE ACID, DNA-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, LIGAND BINDING DOMAIN TRANSCRIPTION REGULATION, COACTIVATOR, FXR ALTERNATIVE SPLICING, HORMONE RECEPTOR
3omm:C (SER362) to (TRP458) CRYSTAL STRUCTURE OF HUMAN FXR IN COMPLEX WITH 4-({(2S)-2-[2-(4- CHLOROPHENYL)-5,6-DIFLUORO-1H-BENZIMIDAZOL-1-YL]-2- CYCLOHEXYLACETYL}AMINO)-3-FLUOROBENZOIC ACID | NUCLEAR RECEPTOR, CHOLESTEROL, BILE ACID, DNA-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, LIGAND BINDING DOMAIN TRANSCRIPTION REGULATION, COACTIVATOR, FXR ALTERNATIVE SPLICING, HORMONE RECEPTOR
5gt4:A (SER306) to (PHE422) CRYSTAL STRUCTURE OF THE HUMAN VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH (1R,2S,3R,5Z,7E,14BETA,17ALPHA)-2-CYANOPROPOXY- 9,10-SECOCHOLESTA-5,7,10-TRIENE-1,3,25-TRIOL | NUCLEAR HORMONE RECEPTOR FULL AGONIST LIGAND COMPLEX, TRANSCRIPTION
3oof:A (ASP363) to (TRP458) CRYSTAL STRUCTURE OF HUMAN FXR IN COMPLEX WITH 4-({(2S)-2-[2-(4- CHLOROPHENYL)-5,6-DIFLUORO-1H-BENZIMIDAZOL-1-YL]-2- CYCLOHEXYLACETYL}AMINO)BENZOIC ACID | NUCLEAR RECEPTOR, CHOLESTEROL, BILE ACID, DNA-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, LIGAND BINDING DOMAIN TRANSCRIPTION REGULATION, COACTIVATOR, FXR ALTERNATIVE SPLICING, HORMONE RECEPTOR
3oof:C (SER362) to (SER457) CRYSTAL STRUCTURE OF HUMAN FXR IN COMPLEX WITH 4-({(2S)-2-[2-(4- CHLOROPHENYL)-5,6-DIFLUORO-1H-BENZIMIDAZOL-1-YL]-2- CYCLOHEXYLACETYL}AMINO)BENZOIC ACID | NUCLEAR RECEPTOR, CHOLESTEROL, BILE ACID, DNA-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, LIGAND BINDING DOMAIN TRANSCRIPTION REGULATION, COACTIVATOR, FXR ALTERNATIVE SPLICING, HORMONE RECEPTOR
3os8:A (VAL418) to (LEU544) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3os8:B (VAL418) to (LEU544) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3os8:C (VAL422) to (ALA546) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3os8:D (VAL422) to (ALA546) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3osi:A (GLU365) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH TETRACHLORO-BISPHENOL A (TCBPA) | TRANSCRIPTION, LIGAND BINDING PROTEIN
3os9:A (VAL422) to (ASP545) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3os9:B (VAL422) to (ASP545) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3os9:C (VAL422) to (ASP545) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3os9:D (VAL422) to (LEU544) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3osa:C (MET421) to (ALA546) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3osa:D (MET421) to (ALA546) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
5hbh:B (ASP187) to (MET257) CDK8-CYCC IN COMPLEX WITH 5-{5-CHLORO-4-[1-(2-METHOXY-ETHYL)-1,8- DIAZA-SPIRO[4.5]DEC-8-YL]-PYRIDIN-3-YL}-1-METHYL-1,3-DIHYDRO- BENZO[C]ISOTHIAZOLE 2,2-DIOXIDE | CDK8 KINASE / CYCLIN C, TRANSFERASE
3osw:A (LYS358) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH TETRABROMO-BISPHENOL A (TBBPA) | TRANSCRIPTION, LIGAND BINDING PROTEIN
3oz0:A (LYS358) to (TYR473) PPAR DELTA IN COMPLEX WITH AZPPARD02 | TRANSCRIPTION FACTOR, TRANSCRIPTION, NUCLEAR RECEPTOR FOLD, TRANSCRIPTION REGULATION, TRANSCRIPTION-TRANSCRIPTION REGULATOR COMPLEX
3dy6:A (LYS358) to (TYR473) PPARDELTA COMPLEXED WITH AN ANTHRANILIC ACID PARTIAL AGONIST | PPAR, NULEAR RECEPTOR, ACTIVATOR, DNA-BINDING, METAL-BINDING, NUCLEUS, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3dy6:B (LYS358) to (TYR473) PPARDELTA COMPLEXED WITH AN ANTHRANILIC ACID PARTIAL AGONIST | PPAR, NULEAR RECEPTOR, ACTIVATOR, DNA-BINDING, METAL-BINDING, NUCLEUS, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3p0u:B (VAL487) to (LEU580) CRYSTAL STRUCTURE OF THE LIGAND BINDING DOMAIN OF HUMAN TESTICULAR RECEPTOR 4 | LIGAND BINDING DOMAIN, ORPHAN NUCLEAR RECEPTOR, TESTICULAR RECEPTOR 4, SIGNALING PROTEIN
4dk8:C (GLN346) to (TRP457) CRYSTAL STRUCTURE OF LXR LIGAND BINDING DOMAIN IN COMPLEX WITH PARTIAL AGONIST 5 | LIGAND BINDING DOMAIN, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION- PEPTIDE-AGONIST COMPLEX
5hjs:B (VAL169) to (TRP279) IDENTIFICATION OF LXRBETA SELECTIVE AGONISTS FOR THE TREATMENT OF ALZHEIMER'S DISEASE | AGONIST, ALZHEIMER'S, SIGNALING PROTEIN
5hk7:C (ILE150) to (SER285) BACTERIAL SODIUM CHANNEL PORE, 2.95 ANGSTROM RESOLUTION | BACTERIAL SODIUM CHANNEL PORE, TRANSPORT PROTEIN
5hk7:D (ILE150) to (ARG283) BACTERIAL SODIUM CHANNEL PORE, 2.95 ANGSTROM RESOLUTION | BACTERIAL SODIUM CHANNEL PORE, TRANSPORT PROTEIN
4dma:A (VAL422) to (LEU549) CRYSTAL STRUCTURE OF ERA LBD IN COMPLEX WITH RU100132 | TRANSCRIPTION, NUCLEAR RECEPTOR, ER, ESTROGEN RECEPTOR, ALPHA HELICAL SANDWICH, TRANSCRIPTION FACTOR, ESTRADIOL, TRANSCRIPTION-PROTEIN BINDING-AGONIST COMPLEX
4dor:A (ALA422) to (ALA538) HUMAN NUCLEAR RECEPTOR LIVER RECEPTOR HOMOLOGUE-1, LRH-1, IN ITS APO STATE BOUND TO A FRAGMENT OF HUMAN SHP BOX1 | NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, PHOSPHOLIPIDS, NR5A, DIABETES, PHOSPHATIDYLCHOLINE, TRANSCRIPTION
4dor:B (ALA422) to (ALA538) HUMAN NUCLEAR RECEPTOR LIVER RECEPTOR HOMOLOGUE-1, LRH-1, IN ITS APO STATE BOUND TO A FRAGMENT OF HUMAN SHP BOX1 | NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, PHOSPHOLIPIDS, NR5A, DIABETES, PHOSPHATIDYLCHOLINE, TRANSCRIPTION
4dos:A (ALA422) to (ALA538) HUMAN NUCLEAR RECEPTOR LIVER RECEPTOR HOMOLOGUE-1, LRH-1, BOUND TO DLPC AND A FRAGMENT OF TIF-2 | NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, PHOSPHOLIPIDS, NR5A, DIABETES, PHOSPHATIDYLCHOLINE, DLPC, TRANSCRIPTION
3p8x:A (SER306) to (PHE422) SYNTHESIS, STRUCTURE, AND BIOLOGICAL ACTIVITY OF DES-SIDE CHAIN ANALOGUES OF 1ALPHA,25-DIHYDROXYVITAMIN D3 WITH SUBSTITUENTS AT C-18 | HELICES SANDWICH, TRANSCRIPTION REGULATION, VITAMIN D, TRANSCRIPTION REGULATOR
4dqm:A (LEU308) to (LEU414) REVEALING A MARINE NATURAL PRODUCT AS A NOVEL AGONIST FOR RETINOIC ACID RECEPTORS WITH A UNIQUE BINDING MODE AND ANTITUMOR ACTIVITY | NUCLEAR RECEPTOR TRANSCRIPTION FACTOR, LIGAND BINDING DOMAIN, TRANSCRIPTION REGULATION, NUCLEUS, TRANSCRIPTION-TRANSFERASE COMPLEX
4dqm:C (THR306) to (LEU414) REVEALING A MARINE NATURAL PRODUCT AS A NOVEL AGONIST FOR RETINOIC ACID RECEPTORS WITH A UNIQUE BINDING MODE AND ANTITUMOR ACTIVITY | NUCLEAR RECEPTOR TRANSCRIPTION FACTOR, LIGAND BINDING DOMAIN, TRANSCRIPTION REGULATION, NUCLEUS, TRANSCRIPTION-TRANSFERASE COMPLEX
3pba:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH MONOSULFATE TETRABROMO-BISPHENOL A (MONOTBBPA) | TRANSCRIPTION, LIGAND BINDING PROTEIN
3pba:B (LYS358) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH MONOSULFATE TETRABROMO-BISPHENOL A (MONOTBBPA) | TRANSCRIPTION, LIGAND BINDING PROTEIN
5hyr:B (MET421) to (ASP545) ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN Y537S MUTANT IN COMPLEX WITH STAPLED PEPTIDE SRC2-SP2 AND ESTRADIOL | BREAST CANCER, ESTROGEN RECEPTOR, SYNTHETIC PEPTIDE, STAPLED PEPTIDE, ENDOCRINE, HORMONE, GENE REGULATION
5hzc:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF THE COMPLEX PPARGAMMA/AL26-29 | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, DIABETES, BUNDLE OF ALPHA- HELICES, TRANSCRIPTION
3plz:A (ALA422) to (ALA538) HUMAN LRH1 LBD BOUND TO GR470 | ALPHA HELICAL SANDWHICH, NUCLEAR RECEPTOR, FAMILY FIVE, TRANSCRIPTION FACTOR, CO-ACTIVATOR, TRANSCRIPTION-RECEPTOR-AGONIST COMPLEX
3po9:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH TRIPROPYLTIN | TRANSCRIPTION, LIGAND BINDING DOMAIN
4e4k:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA WITH THE LIGAND JO21 | BUNDLE OF ALPHA-HELICES AND A SMALL FOUR-STRANDED BETA-SHEET, TRANSCRIPTION FACTOR, TRANSCRIPTION
4e4k:B (PHE360) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA WITH THE LIGAND JO21 | BUNDLE OF ALPHA-HELICES AND A SMALL FOUR-STRANDED BETA-SHEET, TRANSCRIPTION FACTOR, TRANSCRIPTION
4e4q:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA WITH THE LIGAND FS214 | BUNDLE OF ALPHA-HELICES AND A SMALL FOUR-STRANDED BETA-SHEET, TRANSCRIPTION FACTOR, TRANSCRIPTION
3prg:A (ARG357) to (LYS474) LIGAND BINDING DOMAIN OF HUMAN PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR | THIAZOLIDINEDIONE, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ADIPOCYTE DIFFERENTIATION
4em9:A (MET364) to (TYR473) HUMAN PPAR GAMMA IN COMPLEX WITH NONANOIC ACIDS | NUCLEAR RECEPTOR, RETINOIC ACID RECEPTOR, NUCLEUS, TRANSCRIPTION
5iwn:B (ALA151) to (SER285) BACTERIAL SODIUM CHANNEL PORE DOMAIN, HIGH BROMIDE | BACTERIAL SODIUM CHANNEL, LOW BR, TRANSPORT PROTEIN
5iwn:C (ILE150) to (SER285) BACTERIAL SODIUM CHANNEL PORE DOMAIN, HIGH BROMIDE | BACTERIAL SODIUM CHANNEL, LOW BR, TRANSPORT PROTEIN
5iwo:A (ALA151) to (GLY286) BACTERIAL SODIUM CHANNEL PORE DOMAIN, LOW BROMIDE | BACTERIAL SODIUM CHANNEL, HIGH BR, TRANSPORT PROTEIN
3q95:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF HUMAN ESTROGEN RECEPTOR ALPHA LBD IN COMPLEX WITH GRIP PEPTIDE AND ESTRIOL | TRANSCRIPTIONAL REGULATOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATOR
3q97:A (MET421) to (ALA546) CRYSTAL STRUCTURE OF HUMAN ESTROGEN RECEPTOR ALPHA LBD IN COMPLEX WITH GRIP PEPTIDE AND TWO ISOMERS OF ETHOXY TRIPHENYLETHYLENE | TRANSCRIPTIONAL REGULATOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATOR
3q97:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF HUMAN ESTROGEN RECEPTOR ALPHA LBD IN COMPLEX WITH GRIP PEPTIDE AND TWO ISOMERS OF ETHOXY TRIPHENYLETHYLENE | TRANSCRIPTIONAL REGULATOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATOR
4f9m:A (PHE360) to (TYR473) CRYSTAL STRUCTURE OF THE PPARGAMMA-LBD COMPLEXED WITH A CERCOSPORAMIDE DERIVATIVE MODULATOR | THREE-LAYERED ALPHA-HELICAL SANDWICH, TRANSCRIPTION REGULATION, TRANSCRIPTION-TRANSCRIPTION REGULATOR COMPLEX
3qt0:A (MET364) to (TYR473) REVEALING A STEROID RECEPTOR LIGAND AS A UNIQUE PPARGAMMA AGONIST | PPAR GAMMA LBD DOMAIN, TRANSCRIPTION
4fgy:A (MET392) to (TYR501) IDENTIFICATION OF A UNIQUE PPAR LIGAND WITH AN UNEXPECTED BINDING MODE AND ANTIBETIC ACTIVITY | PPAR LBD, NUCLEAR RECEPTOR FOLD, LIGAND BINDING, GENE TRANSCRIPTION, TRANSCRIPTION-TRANSFERASE-ANTIBIOTIC COMPLEX
4fhh:A (THR334) to (LEU440) DEVELOPMENT OF SYNTHETICALLY ACCESSIBLE NON-SECOSTEROIDAL HYBRID MOLECULES COMBINING VITAMIN D RECEPTOR AGONISM AND HISTONE DEACETYLASE INHIBITION | LIGAND BINDING DOMAIN, APHA HELICAL SANDWICH, ALPHA HELICAL SANDWICH, TRANSCRIPTION FACTOR, ADN COREGULATORS, PHOSPHORYLATION AND HDAC INHIBITOR, NUCLEUS, TRANSCRIPTION-PROTEIN BINDING-INHIBITOR COMPLEX
3r29:B (VAL354) to (MET454) CRYSTAL STRUCTURE OF RXRALPHA LIGAND-BINDING DOMAIN COMPLEXED WITH COREPRESSOR SMRT2 | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING DOMAIN, TRANSCRIPTION
3r8a:B (LYS358) to (LYS474) X-RAY CRYSTAL STRUCTURE OF THE NUCLEAR HORMONE RECEPTOR PPAR-GAMMA IN A COMPLEX WITH A COMPOUND WITH DUAL PPAR GAMMA AGONISM AND ANGIOTENSIN II TYPE I RECEPTOR ANTAGONISM ACTIVITY | NUCLEAR HORMONE ACTIVATOR, ANGIOTENSIN II TYPE I RECEPTOR ANTAGONIST, LIGAND BOUND STRUCTURE, DIABETES MELLITUS, METABOLIC SYNDROME, OBESITY, NUCLEAR PROTEIN
3r8i:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA WITH AN ACHIRAL UREIDOFIBRATE DERIVATIVE (RT86) | PROTEIN-DNA COMPLEX, BUNDLE OF ALPHA-HELICES, SMALL FOUR-STRANDED BETA-SHEET, TRANSCRIPTION, ACTIVATOR, DIABETES MELLITUS, OBESITY, TRANSCRIPTION REGULATION, DNA BINDING, PHOSPHORYLATION, NUCLEUS
4g1d:A (THR334) to (LEU440) STRUCTURAL BASIS FOR THE ACCOMMODATION OF BIS- AND TRIS-AROMATIC DERIVATIVES IN VITAMIN D NUCLEAR RECEPTOR | TRANSCRIPTION REGULATION, VDR, VITAMIN D, ALPHA HELICAL SANDWICH, TRANSCRIPTION, LIGAND, ADN, PHOSPHORYLATION, NUCLEUS, TRANSCRIPTION- TRANSCRIPTION INHIBITOR COMPLEX
4g1y:A (THR334) to (THR441) STRUCTURAL BASIS FOR THE ACCOMMODATION OF BIS- AND TRIS-AROMATIC DERIVATIVES IN VITAMIN D NUCLEAR RECEPTOR | VDR, TRANSCRIPTION REGULATION, NUCLEAR RECEPTOR, ALPHA HELICAL SANDWICH, LIGAND, DNA, PHOSPHORYLATION, NUCLEUS, TRANSCRIPTION- TRANSCRIPTION INHIBITOR COMPLEX
4g1z:A (THR334) to (PRO434) STRUCTURAL BASIS FOR THE ACCOMMODATION OF BIS- AND TRIS-AROMATIC DERIVATIVES IN VITAMIN D NUCLEAR RECEPTOR | VDR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, ALPHA HELICAL SANDWICH, LIGAND, DNA, PHOSPHORYLATION, NUCLEUS, TRANSCRIPTION- TRANSCRIPTION INHIBITOR COMPLEX
4g2i:A (SER306) to (GLY423) STRUCTURAL BASIS FOR THE ACCOMMODATION OF BIS- AND TRIS-AROMATIC DERIVATIVES IN VITAMIN D NUCLEAR RECEPTOR | VDR, TRANSCRIPTION REGULATION, NUCLEAR RECEPTOR, ALPHA HELICAL SANDWICH, LIGAND, DNA, PHOSPHORYLATION, NUCLEUS, TRANSCRIPTION- TRANSCRIPTION INHIBITOR COMPLEX
5kce:B (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-METHYL, 2-CHLOROBENZYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, SIGNALING PROTEIN, TRANSCRIPTION
5kcf:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-ETHYL, 4-METHOXYBENZYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5kcf:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-ETHYL, 4-METHOXYBENZYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5kct:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-ETHYL, 4-CHLOROBENZYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5kcu:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-ETHYL, ALPHA-NAPHTHYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5kcu:B (MET421) to (LEU544) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-ETHYL, ALPHA-NAPHTHYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5kcw:A (GLY420) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-TRIFLUOROETHYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5kcw:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-TRIFLUOROETHYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5kd9:A (VAL422) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-TRIFLUOROETHYL 4-CHLOROBENZYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5lga:A (THR334) to (LEU440) STRUCTURAL ANALYSIS AND BIOLOGICAL ACTIVITIES OF BXL0124, A GEMINI ANALOG OF VITAMIN D | VITAMIN D NUCLEAR RECEPTOR, AGONIST, GEMINI, TRANSCRIPTION
5syz:A (ALA422) to (ALA538) HUMAN LIVER RECEPTOR HOMOLOGUE-1 (LRH-1) BOUND TO A RJW100 STEREOISOMER AND A FRAGMENT OF TIF-2 | NUCLEAR RECEPTOR, AGONIST, COACTIVATOR, NUCLEAR PROTEIN
5t3t:F (SER182) to (VAL265) EBOLA VIRUS VP30 CTD BOUND TO NUCLEOPROTEIN | TRANSCRIPTION, REPLICATION, REGULATOR, CO-FACTOR, VIRAL PROTEIN
5t3t:G (SER182) to (VAL265) EBOLA VIRUS VP30 CTD BOUND TO NUCLEOPROTEIN | TRANSCRIPTION, REPLICATION, REGULATOR, CO-FACTOR, VIRAL PROTEIN
5t3t:J (SER182) to (VAL265) EBOLA VIRUS VP30 CTD BOUND TO NUCLEOPROTEIN | TRANSCRIPTION, REPLICATION, REGULATOR, CO-FACTOR, VIRAL PROTEIN
2ocf:A (VAL422) to (ARG548) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH ESTRADIOL AND THE E2#23 FN3 MONOBODY | ESTROGEN RECEPTOR, LBD, MONOBODY, ESTRADIOL, HORMONE-GROWTH FACTOR COMPLEX
3s27:B (LEU203) to (VAL275) THE CRYSTAL STRUCTURE OF SUCROSE SYNTHASE-1 FROM ARABIDOPSIS THALIANA AND ITS FUNCTIONAL IMPLICATIONS. | GLYCOSYLTRANSFERASE, SUCROSE METABOLISM, SUGAR ACCEPTOR COMPLEX, ROSSMANN FOLD, GT-B FOLD, UDP, FRUCTOSE, CYTOSOL, TRANSFERASE
4hee:X (ARG357) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA IN COMPLEX WITH COMPOUND 13 | PPARGAMMA, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
3s29:B (ASN202) to (VAL275) THE CRYSTAL STRUCTURE OF SUCROSE SYNTHASE-1 FROM ARABIDOPSIS THALIANA AND ITS FUNCTIONAL IMPLICATIONS. | GLYCOSYLTRANSFERASE, SUCROSE METABOLISM, SUGAR ACCEPTOR COMPLEX, ROSSMANN FOLD, GT-B FOLD, UDP, FRUCTOSE, CYTOSOL, TRANSFERASE
2pin:B (VAL348) to (GLU460) THYROID RECEPTOR BETA IN COMPLEX WITH INHIBITOR | THYROID RECEPTOR BETA, NUCLEAR RECEPTORS, INHIBITORS, PROTEIN-PROTEIN INTERACTIONS, COREGULATOR BINDING, AF-2 POCKET, AROMATIC-BETA-AMINO KETONES, STRUCTURE-BASED DRUG DESIGN, SURFACE INTERACTING DRUGS, HORMONE RECEPTOR
2pip:L (MET780) to (SER888) ANDROGEN RECEPTOR LBD WITH SMALL MOLECULE | ANDROGEN RECEPTOR, COACTIVATORS, AF-2 POCKET, INHIBITORS, HORMONE RECEPTOR
2pit:A (MET780) to (SER888) ANDROGEN RECEPTOR LBD WITH SMALL MOLECULE | ANDROGEN RECEPTOR COACTIVATOR BINDING INHIBITORS AF-2, HORMONE RECEPTOR
3fej:A (ARG357) to (TYR473) DESIGN AND BIOLOGICAL EVALUATION OF NOVEL, BALANCED DUAL PPARA/G AGONISTS | NUCLEAR RECPETOR,TRANSCRIPTION FACTOR, DIABETES, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
4xhd:A (PRO322) to (LEU428) STRUCTURE OF HUMAN PREGNANE X RECEPTOR LIGAND BINDING DOMAIN WITH COMPOUND-1 | PREGNANE X RECEPTOR, PXR, LIGAND BINDING DOMAIN, STEROID RECEPTOR COACTIVATOR-1; CCR1, CHEMOKINE RECEPTOR-1; ADNECTIN NR, NUCLEAR RECEPTOR; AF, ACTIVATION FUNCTION; CYP, CYTOCHROME P450; MDR1, MULTI-DRUG RESISTANCE GENE-1., TRANSCRIPTION
2prg:A (ARG357) to (TYR473) LIGAND-BINDING DOMAIN OF THE HUMAN PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR GAMMA | COMPLEX (THIAZOLIDINEDIONE/RECEPTOR), LIGAND-BINDING DOMAIN, NUCLEAR RECEPTOR, APO, TRANSCRIPTION FACTOR, ORPHAN RECEPTOR
2prg:B (ARG357) to (TYR473) LIGAND-BINDING DOMAIN OF THE HUMAN PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR GAMMA | COMPLEX (THIAZOLIDINEDIONE/RECEPTOR), LIGAND-BINDING DOMAIN, NUCLEAR RECEPTOR, APO, TRANSCRIPTION FACTOR, ORPHAN RECEPTOR
1osh:A (ASP363) to (ILE472) A CHEMICAL, GENETIC, AND STRUCTURAL ANALYSIS OF THE NUCLEAR BILE ACID RECEPTOR FXR | NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, TRANSCRIPTION
2q5p:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA BOUND TO PARTIAL AGONIST MRL24 | PROTEIN-LIGAND COMPLEX, LIGAND BINDING PROTEIN
2q5p:B (ARG357) to (TYR473) CRYSTAL STRUCTURE OF PPARGAMMA BOUND TO PARTIAL AGONIST MRL24 | PROTEIN-LIGAND COMPLEX, LIGAND BINDING PROTEIN
4xuh:A (GLU365) to (TYR473) PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH SULINDAC SULFIDE | NUCLEAR RECEPTOR, PPARGAMMA, SULINDAC SULFIDE, NSAIDS, TRANSLATION
4ite:A (SER306) to (GLY423) CRYSTAL STRUCTURE OF THE HUMAN VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH 1ALPHA,25-DIHYDROXY-2ALPHA-[2-(2H-TETRAZOL-2- YL)ETHYL]VITAMIN D3 | HORMONE RECEPTOR, TRANSCRIPTION
1pqc:A (GLN346) to (TRP457) HUMAN LXR BETA HORMONE RECEPTOR COMPLEXED WITH T0901317 | LXRB+T0901317, TRANSCRIPTION REGULATION
3gyt:A (ARG630) to (PHE749) NUCLEAR RECEPTOR DAF-12 FROM PARASITIC NEMATODE STRONGYLOIDES STERCORALIS IN COMPLEX WITH ITS PHYSIOLOGICAL LIGAND DAFACHRONIC ACID DELTA 4 | NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, DAFACHRONIC ACID, SRC1, NEMATODE, STRONGYLOIDES STERCORALIS, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
1err:B (GLY420) to (HIS550) HUMAN ESTROGEN RECEPTOR LIGAND-BINDING DOMAIN IN COMPLEX WITH RALOXIFENE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, STEROID, ANTAGONIST
1fcz:A (THR308) to (GLU417) ISOTYPE SELECTIVITY OF THE HUMAN RETINOIC ACID NUCLEAR RECEPTOR HRAR: THE COMPLEX WITH THE PANAGONIST RETINOID BMS181156 | ISOTYPE SELECTIVITY, RETINOID LIGAND COMPLEXES, DRUG DESIGN, ANTIPARALLEL ALPHA-HELICAL SANDWICH FOLD, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS, GENE REGULATION
1fm6:D (LYS358) to (TYR473) THE 2.1 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE HETERODIMER OF THE HUMAN RXRALPHA AND PPARGAMMA LIGAND BINDING DOMAINS RESPECTIVELY BOUND WITH 9-CIS RETINOIC ACID AND ROSIGLITAZONE AND CO-ACTIVATOR PEPTIDES. | THE HETERODIMER OF THE NUCLEAR RECEPTOR LIGAND BINDING DOMAINS OF RXRALPHA AND PPARGAMMA BOUND RESPECTIVELY WITH 9-CIS RETINOIC ACID AND ROSIGLITAZONE AND CO-ACTIVATOR PEPTIDES, TRANSCRIPTION
1fm6:X (GLU365) to (TYR473) THE 2.1 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE HETERODIMER OF THE HUMAN RXRALPHA AND PPARGAMMA LIGAND BINDING DOMAINS RESPECTIVELY BOUND WITH 9-CIS RETINOIC ACID AND ROSIGLITAZONE AND CO-ACTIVATOR PEPTIDES. | THE HETERODIMER OF THE NUCLEAR RECEPTOR LIGAND BINDING DOMAINS OF RXRALPHA AND PPARGAMMA BOUND RESPECTIVELY WITH 9-CIS RETINOIC ACID AND ROSIGLITAZONE AND CO-ACTIVATOR PEPTIDES, TRANSCRIPTION
2vix:A (MET250) to (TYR349) METHYLATED SHIGELLA FLEXNERI MXIC | TRANSPORT PROTEIN, SECRETION REGULATION, T3SS, VIRULENCE, TYPE THREE SECRETION SYSTEM
2vix:B (MET250) to (TYR349) METHYLATED SHIGELLA FLEXNERI MXIC | TRANSPORT PROTEIN, SECRETION REGULATION, T3SS, VIRULENCE, TYPE THREE SECRETION SYSTEM
1sj0:A (MET421) to (MET543) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE ANTAGONIST LIGAND 4-D | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ER-ALPHA, ANTAGONIST, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
2vv0:B (LYS358) to (TYR473) HPPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH DHA | NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, ALTERNATIVE SPLICING, LIGAND BINDING DOMAIN, DIABETES MELLITUS, ZINC-FINGER, DNA-BINDING, POLYMORPHISM, TRANSCRIPTION, ZINC, OBESITY, NUCLEUS, RECEPTOR, ACTIVATOR, OXIDISED FATTY ACID, TRANSCRIPTION FACTOR, METAL-BINDING, PHOSPHOPROTEIN, DISEASE MUTATION
3vdx:C (LEU279) to (ASN368) STRUCTURE OF A 16 NM PROTEIN CAGE DESIGNED BY FUSING SYMMETRIC OLIGOMERIC DOMAINS | PROTEIN DESIGN, BIONANOTECHNOLOGY, PROTEIN ASSEMBLY, SYMMETRY, BIOMATERIALS, DE NOVO PROTEIN
3vjh:A (ARG357) to (TYR473) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH JKPL35 | TRANSCRIPTION
3vjt:A (THR302) to (LEU410) VITAMIN D RECEPTOR COMPLEX WITH A CARBORANE COMPOUND | NUCLEAR RECEPTOR, SYNTHETIC AGONIST, CARBORANE, TRANSCRIPTION
4zn7:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH DIETHYLSTILBESTROL | NUCLEAR RECEPTOR TRANSCRIPTION FACTOR NUCLEUS PROTEIN-LIGAND COMPLEX, TRANSCRIPTION
4zn7:B (MET421) to (ALA546) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH DIETHYLSTILBESTROL | NUCLEAR RECEPTOR TRANSCRIPTION FACTOR NUCLEUS PROTEIN-LIGAND COMPLEX, TRANSCRIPTION
4znu:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH A 2-METHYL-SUBSTITUTED OBHS DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4l96:A (PRO359) to (ASP475) STRUCTURE OF THE COMPLEX BETWEEN THE F360L PPARGAMMA MUTANT AND THE LIGAND LT175 (SPACE GROUP I222) | TRANSCRIPTION FACTOR, RXRALPHA, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
3ipq:A (VAL333) to (TRP443) X-RAY STRUCTURE OF GW3965 SYNTHETIC AGONIST BOUND TO THE LXR-ALPHA | NUCLEAR RECEPTOR, LXR HOMODIMER, LXR SIGNALING, ALTERNATIVE SPLICING, DNA-BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACTIVATOR, ACYLTRANSFERASE, CHROMOSOMAL REARRANGEMENT, ISOPEPTIDE BOND, PHOSPHOPROTEIN, PROTO-ONCOGENE, TRANSFERASE, UBL CONJUGATION
2hb8:A (SER306) to (PHE422) CRYSTAL STRUCTURE OF VDR LBD IN COMPLEX WITH 2ALPHA-METHYL CALCITRIOL | ALPHA HELICAL SANDWICH, GENE REGULATION
2hbh:A (THR334) to (LEU440) CRYSTAL STRUCTURE OF VITAMIN D NUCLEAR RECEPTOR LIGAND BINDING DOMAIN BOUND TO A LOCKED SIDE-CHAIN ANALOG OF CALCITRIOL AND SRC-1 PEPTIDE | ALPHA HELICAL SANDWICH, GENE REGULATION
4ltr:C (ILE150) to (SER285) BACTERIAL SODIUM CHANNEL, HIS245GLY MUTANT, I222 SPACE GROUP | CATION CHANNEL FOLD, COILED COIL SODIUM CHANNEL, PLASMA MEMBRANE, TRANSPORT PROTEIN
1ie9:A (SER306) to (GLY423) CRYSTAL STRUCTURE OF THE NUCLEAR RECEPTOR FOR VITAMIN D LIGAND BINDING DOMAIN BOUND TO MC1288 | VDR, MC1288, GENE REGULATION
1ulh:A (ALA318) to (THR415) A SHORT PEPTIDE INSERTION CRUCIAL FOR ANGIOSTATIC ACTIVITY OF HUMAN TRYPTOPHANYL-TRNA SYNTHETASE | AMINOACYLATION, ANGIOSTATIC CYTOKINE, APOPTOSIS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, STRUCTURAL GENOMICS, LIGASE
5aav:A (MET421) to (HIS550) OPTIMIZATION OF A NOVEL BINDING MOTIF TO TO (E)-3-(3,5- DIFLUORO-4-((1R,3R)-2-(2-FLUORO-2-METHYLPROPYL)-3-METHYL-2, 3,4,9-TETRAHYDRO-1H-PYRIDO(3,4-B)INDOL-1-YL)PHENYL)ACRYLIC ACID (AZD9496), A POTENT AND ORALLY BIOAVAILABLE SELECTIVE ESTROGEN RECEPTOR DOWNREGULATOR AND ANTAGONIST | SIGNALING PROTEIN, BREAST CANCER, ESTROGEN RECEPTOR DOWNREGULATOR, FULVESTRANT, AZD9496, NUCLEAR HORMONE RECEPTOR
5aav:B (VAL422) to (ASP545) OPTIMIZATION OF A NOVEL BINDING MOTIF TO TO (E)-3-(3,5- DIFLUORO-4-((1R,3R)-2-(2-FLUORO-2-METHYLPROPYL)-3-METHYL-2, 3,4,9-TETRAHYDRO-1H-PYRIDO(3,4-B)INDOL-1-YL)PHENYL)ACRYLIC ACID (AZD9496), A POTENT AND ORALLY BIOAVAILABLE SELECTIVE ESTROGEN RECEPTOR DOWNREGULATOR AND ANTAGONIST | SIGNALING PROTEIN, BREAST CANCER, ESTROGEN RECEPTOR DOWNREGULATOR, FULVESTRANT, AZD9496, NUCLEAR HORMONE RECEPTOR
5acc:A (MET421) to (LEU544) A NOVEL ORAL SELECTIVE ESTROGEN RECEPTOR DOWN-REGULATOR, AZD9496, DRIVES TUMOUR GROWTH INHIBITION IN ESTROGEN RECEPTOR POSITIVE AND ESR1 MUTANT MODELS | SIGNALING PROTEIN, SERD, METASTATIC BREAST CANCER, ER MUTATION, ESR1 MUTATION, COMBINATION THERAPY
3wgp:A (SER306) to (GLY423) CRYSTAL STRUCTURE ANALYSIS OF VITAMIN D RECEPTOR | STEROID HORMON RECEPTOR FAMILY MEMBER, HORMONE RECEPTOR
5ak2:A (GLU423) to (HIS550) OXYPHENYLPROPENOIC ACIDS AS ORAL SELECTIVE ESTROGEN RECEPTOR DOWN-REGULATORS. | SIGNALING PROTEIN
3wmh:A (LYS358) to (LYS474) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A GAMMMA SELECTIVE SYNTHETIC PARTIAL AGONIST MEKT75 | MAINLY ALPHA, NUCLEAR RECEPTOR, TRANSCRIPTION
3wmh:B (LYS358) to (TYR473) HUMAN PPAR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A GAMMMA SELECTIVE SYNTHETIC PARTIAL AGONIST MEKT75 | MAINLY ALPHA, NUCLEAR RECEPTOR, TRANSCRIPTION
2lbd:A (THR308) to (GLU417) LIGAND-BINDING DOMAIN OF THE HUMAN RETINOIC ACID RECEPTOR GAMMA BOUND TO ALL-TRANS RETINOIC ACID | NUCLEAR RECEPTOR, RETINOIC ACID RECEPTOR, ALL-TRANS RETINOIC ACID, LIGAND-BINDING DOMAIN, COMPLEX, HOLO FORM, TRANSCRIPTION REGULATION, LIGAND-DEPENDENT, ACTIVE CONFORMATION, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS
2yfe:A (ARG357) to (TYR473) LIGAND BINDING DOMAIN OF HUMAN PPAR GAMMA IN COMPLEX WITH AMORFRUTIN 1 | RECEPTOR, AGONIST, DIABETES, INSULIN RESISTANCE
1x76:A (ILE373) to (ALA497) CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-697 | ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST
2ylo:A (TYR781) to (GLN902) TARGETING THE BINDING FUNCTION 3 SITE OF THE ANDROGEN RECEPTOR THROUGH IN SILICO MOLECULAR MODELING | HORMONE RECEPTOR, BINDING FUNCTION 3
2yly:A (GLU371) to (ALA497) SULFONAMIDES AS SELECTIVE ESTROGEN RECEPTOR BETA AGONISTS. | RECEPTOR
2o4r:A (THR302) to (LEU410) CRYSTAL STRUCTURE OF RAT VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH VITIII 17-20E AND THE NR2 BOX OF DRIP 205 | NUCLEAR RECEPTOR-LIGAND COMPLEX, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
4a4w:A (ARG357) to (TYR473) LIGAND BINDING DOMAIN OF HUMAN PPAR GAMMA IN COMPLEX WITH AMORFRUTIN 2 | RECEPTOR, AGONIST, DIABETES, INSULIN RESISTANCE
1xp9:A (MET421) to (MET543) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH COMPOUND 18 | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ER-ALPHA, ANTAGONIST, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
2zmj:A (THR302) to (LEU410) CRYSTAL STRUCTURE OF RAT VITAMIN D RECEPTOR BOUND TO ADAMANTYL VITAMIN D ANALOGS: STRUCTURAL BASIS FOR VITAMIN D RECEPTOR ANTAGONISM AND/OR PARTIAL AGONISM | NUCLEAR RECEPTOR-ANTAGONIST COMPLEX, DNA-BINDING, METAL- BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACTIVATOR
2znq:A (LYS358) to (TYR473) HUMAN PPAR DELTA LIGAND BINDING DOMAIN IN COMPLEX WITH A SYNTHETIC AGONIST TIPP401 | NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, PPAR, ACTIVATOR, DNA- BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
2znq:B (LYS358) to (TYR473) HUMAN PPAR DELTA LIGAND BINDING DOMAIN IN COMPLEX WITH A SYNTHETIC AGONIST TIPP401 | NUCLEAR RECEPTOR, PROTEIN-LIGAND COMPLEX, PPAR, ACTIVATOR, DNA- BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
1yye:A (ILE373) to (LEU500) CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-202196 | ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, AGONIST
4ppp:A (GLN441) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH FLUORO-RESVERATROL | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, PROTEIN BINDING
4ppp:B (GLN441) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH FLUORO-RESVERATROL | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, PROTEIN BINDING
4pps:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH AN A-CD RING ESTROGEN DERIVATIVE | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, PROTEIN BINDING
4pvu:A (PRO359) to (TYR473) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN PPARGAMMA-LBD AND THE R ENANTIOMER OF MBX-102 (METAGLIDASEN) | ALPHA-HELICES, SMALL FOUR-STRANDED BETA-SHEET, ACTIVATOR, TDNA- BINDING, NUCLEUS, OBESITY, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION
4pvu:B (PRO359) to (TYR473) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN PPARGAMMA-LBD AND THE R ENANTIOMER OF MBX-102 (METAGLIDASEN) | ALPHA-HELICES, SMALL FOUR-STRANDED BETA-SHEET, ACTIVATOR, TDNA- BINDING, NUCLEUS, OBESITY, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION
5dvs:A (MET421) to (ALA546) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 2-METHYL-SUBSTITUTED TRIARYL-IMINE 4,4'-[(2-METHYLPHENYL) CARBONIMIDOYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dvs:B (VAL422) to (ALA546) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 2-METHYL-SUBSTITUTED TRIARYL-IMINE 4,4'-[(2-METHYLPHENYL) CARBONIMIDOYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dx3:A (MET421) to (ASP545) ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN Y537S MUTANT IN COMPLEX WITH STAPLED PEPTIDE SRC2-P3 AND ESTRADIOL | SYNTHETIC PEPTIDE, STAPLED PEPTIDE, ESTROGEN RECEPTOR ALPHA, SOMATIC MUTATION, PEPTIDE MIMETIC, AF-2 BINDING, HORMONE RECEPTOR-PEPTIDE COMPLEX
5dyb:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-(3,4-DIHYDRONAPHTHALEN-2(1H)- YLIDENEMETHANEDIYL)DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dyb:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-(3,4-DIHYDRONAPHTHALEN-2(1H)- YLIDENEMETHANEDIYL)DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5e0x:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-{[(3S)-3-(4-METHOXYPHENYL) CYCLOHEXYLIDENE]METHANEDIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5e0x:B (VAL422) to (VAL533) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-{[(3S)-3-(4-METHOXYPHENYL) CYCLOHEXYLIDENE]METHANEDIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
3aur:A (SER306) to (GLY423) CRYSTAL STRUCTURE OF THE HUMAN VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH YNE-DIENE TYPE ANALOG OF ACTIVE 14-EPI-2BETA- METHYL-19-NORVITAMIN D3 | HORMONE RECEPTOR, TRANSCRIPTION
3ax8:A (SER306) to (GLY423) CRYSTAL STRUCTURE OF THE HUMAN VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH 15ALPHA-METHOXY-1ALPHA,25-DIHYDROXYVITAMIN D3 | HORMONE RECEPTOR, TRANSCRIPTION
3az2:A (SER306) to (GLY423) CRYSTAL STRUCTURE ANALYSIS OF VITAMIN D RECEPTOR | VITAMIN D RECEPTOR, HORMONE RECEPTOR
3b0r:A (ARG357) to (TYR473) HUMAN PPAR GAMMA LIGAND BINDING DMAIN COMPLEXED WITH GW9662 IN A COVALENT BONDED FORM | NUCLEAR RECEPTOR, TRANSCRIPTION
3b5r:A (TYR781) to (SER888) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH SARM C-31 | ANDROGEN RECEPTOR, NONSTEROIDAL, SARM, DISEASE MUTATION, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRIPLET REPEAT EXPANSION, UBL CONJUGATION, ZINC, ZINC-FINGER
4rbn:D (ILE189) to (ILE261) THE CRYSTAL STRUCTURE OF NITROSOMONAS EUROPAEA SUCROSE SYNTHASE: INSIGHTS INTO THE EVOLUTIONARY ORIGIN OF SUCROSE METABOLISM IN PROKARYOTES | SUCROSE SYNTHASE, ROSSMANN FOLD, GLUCOSYLTRANSFERASE, NDP-GLUCOSE, D- FRUCTOSE, NDP, SUCROSE, CYTOSOL, TRANSFERASE
5fqv:A (MET421) to (LEU544) SELECTIVE ESTROGEN RECEPTOR DOWNREGULATOR ANTAGONISTS: TETRAHYDROISOQUINOLINE PHENOLS 5. | SIGNALING PROTEIN, BREAST CANCER, ESTROGEN RECEPTOR DOWNREGULATOR, FULVESTRANT, THIQ, NUCLEAR HORMONE RECEPTOR
3nsp:A (GLY341) to (GLY443) CRYSTAL STRUCTURE OF TETRAMERIC RXRALPHA-LBD | NUCLEAR RECEPTOR RETINOIC X RECEPOR ALPHA LIGAND BINDING DOMAIN, TRANSCRIPTION
3cs6:A (SER306) to (PHE422) STRUCTURE-BASED DESIGN OF A SUPERAGONIST LIGAND FOR THE VITAMIN D NUCLEAR RECEPTOR | VDR, AGONIST, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, GENE REGULATION
3d6d:A (ARG357) to (TYR473) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN PPARGAMMA LBD AND THE LT175(R-ENANTIOMER) | BUNDLE OF ALPHA-HELICES AND A SMALL FOUR-STRANDED BETA- SHEET, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
3peq:A (LYS358) to (TYR473) PPARD COMPLEXED WITH A PHENOXYACETIC ACID PARTIAL AGONIST | PPAR NUCLEAR RECEPTOR, TRANSCRIPTION-TRANSCRIPTION AGONIST COMPLEX
3peq:B (LYS358) to (MET476) PPARD COMPLEXED WITH A PHENOXYACETIC ACID PARTIAL AGONIST | PPAR NUCLEAR RECEPTOR, TRANSCRIPTION-TRANSCRIPTION AGONIST COMPLEX
4ema:A (ARG357) to (TYR473) HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA IN COMPLEX WITH ROSIGLITAZONE | NUCLEAR RECEPTOR, RETINOIC ACID RECEPTOR, NUCLEUS, TRANSCRIPTION
4ema:B (LYS358) to (TYR473) HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA IN COMPLEX WITH ROSIGLITAZONE | NUCLEAR RECEPTOR, RETINOIC ACID RECEPTOR, NUCLEUS, TRANSCRIPTION
4g2h:A (THR334) to (LEU440) STRUCTURAL BASIS FOR THE ACCOMMODATION OF BIS- AND TRIS-AROMATIC DERIVATIVES IN VITAMIN D NUCLEAR RECEPTOR | VDR, TRANSCRIPTION REGULATION, NUCLEAR RECEPTOR, ALPHA HELICAL SANDWICH, TRASNCRIPTION REGULATION, LIGAND, DNA, PHOSPHORYLATION, NUCLEUS, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
5kcd:A (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-METHYL SUBSTITUTED OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5kcd:B (MET421) to (ARG548) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-METHYL SUBSTITUTED OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION