1n7v:A (GLY224) to (TYR330) THE RECEPTOR-BINDING PROTEIN P2 OF BACTERIOPHAGE PRD1: CRYSTAL FORM III | BACTERIOPHAGE PRD1, VIRAL RECEPTOR-BINDING, BETA-PROPELLER, PROLINE-RICH, ANTIBIOTIC-RESISTANCE, VIRAL PROTEIN
2aid:A (GLY52) to (GLY78) STRUCTURE OF A NON-PEPTIDE INHIBITOR COMPLEXED WITH HIV-1 PROTEASE: DEVELOPING A CYCLE OF STRUCTURE-BASED DRUG DESIGN | ASPARTYL PROTEASE, HIV, NON-PEPTIDE INHIBITOR, DRUG DESIGN
1a30:B (ARG57) to (GLY78) HIV-1 PROTEASE COMPLEXED WITH A TRIPEPTIDE INHIBITOR | ASPARTIC PROTEASE, HIV PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1n93:X (ARG97) to (ALA116) CRYSTAL STRUCTURE OF THE BORNA DISEASE VIRUS NUCLEOPROTEIN | RNA VIRUS NUCLEOPROTEIN TETRAMER, VIRAL PROTEIN
2akk:A (ASP17) to (GLY42) SOLUTION STRUCTURE OF PHNA-LIKE PROTEIN RP4479 FROM RHODOPSEUDOMONAS PALUSTRIS | BETA-STRAND PROTEIN; STRUCTURAL GENOMICS; PSI; PROTEIN STRUCTURE INITIATIVE; NORTHEAST STRUCTURAL GENOMICS CONSORTIUM; NESG; ONTARIO CENTRE FOR STRUCTURAL PROTEOMICS; OCSP, STRUCTURAL GENOMICS, UNKNOWN FUNCTION
2akl:A (THR60) to (ASN84) SOLUTION STRUCTURE FOR PHN-A LIKE PROTEIN PA0128 FROM PSEUDOMONAS AERUGINOSA | TWO DOMAINS; ZN BINDING PROTEIN; BETA-STRAND PROTEIN, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM; NESG; ONTARIO CENTRE FOR STRUCTURAL PROTEOMICS; OCSP, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, UNKNOWN FUNCTION
2akq:D (GLY17) to (THR49) THE STRUCTURE OF BOVINE B-LACTOGLOBULIN A IN CRYSTALS GROWN AT VERY LOW IONIC STRENGTH | B-LACTOGLBULIN, X-RAY, CRYSTAL LATTICE, LOW IONIC STRENGTH, PSEUDO-MEROHEDRAL TWINNING, TRANSPORT PROTEIN
4wfn:H (VAL75) to (ASN100) CRYSTAL STRUCTURE OF THE LARGE RIBOSOMAL SUBUNIT (50S) OF DEINOCOCCUS RADIODURANS CONTAINING A THREE RESIDUE INSERTION IN L22 IN COMPLEX WITH ERYTHROMYCIN | RIBOSOME, ANTIBIOTICS, RRESISTANCE, ERYTHROMYCIN
4gwa:A (LYS110) to (LEU131) CRYSTAL STRUCTURE OF A GH7 FAMILY CELLOBIOHYDROLASE FROM LIMNORIA QUADRIPUNCTATA | CELLOBIOHYDROLASE, GLYCOSYL HYDROLASE, HYDROLASE
4gwa:B (LYS110) to (LEU131) CRYSTAL STRUCTURE OF A GH7 FAMILY CELLOBIOHYDROLASE FROM LIMNORIA QUADRIPUNCTATA | CELLOBIOHYDROLASE, GLYCOSYL HYDROLASE, HYDROLASE
1a8k:A (ARG57) to (GLY78) CRYSTALLOGRAPHIC ANALYSIS OF HUMAN IMMUNODEFICIENCY VIRUS 1 PROTEASE WITH AN ANALOG OF THE CONSERVED CA-P2 SUBSTRATE: INTERACTIONS WITH FREQUENTLY OCCURRING GLUTAMIC ACID RESIDUE AT P2' POSITION OF SUBSTRATES | HUMAN IMMUNODEFICIENCY VIRUS PROTEASE, PROTON-MEDIATED INTERACTION, VIRAL MATURATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1a94:A (ARG57) to (GLY78) STRUCTURAL BASIS FOR SPECIFICITY OF RETROVIRAL PROTEASES | HUMAN IMMUNODEFICIENCY VIRUS PROTEASE, ROUS SARCOMA VIRUS PROTEASE, PROTEIN-MEDIATED INTERACTION, VIRAL MATURATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1a94:D (ARG57) to (GLY78) STRUCTURAL BASIS FOR SPECIFICITY OF RETROVIRAL PROTEASES | HUMAN IMMUNODEFICIENCY VIRUS PROTEASE, ROUS SARCOMA VIRUS PROTEASE, PROTEIN-MEDIATED INTERACTION, VIRAL MATURATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2aoc:B (ARG157) to (GLY178) CRYSTAL STRUCTURE ANALYSIS OF HIV-1 PROTEASE MUTANT I84V WITH A SUBSTRATE ANALOG P2-NC | HIV-1 PROTEASE, MUTANT, DIMER, SUBSTRATE ANALOG, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2aod:B (ARG157) to (GLY178) CRYSTAL STRUCTURE ANALYSIS OF HIV-1 PROTEASE WITH A SUBSTRATE ANALOG P2-NC | HIV-1 PROTEASE, MUTANT, DIMER, SUBSTRATE ANALOG, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2aoe:B (ARG157) to (GLY178) CRYSTAL STRUCTURE ANALYSIS OF HIV-1 PROTEASE MUTANT V82A WITH A SUBSTRATE ANALOG CA-P2 | HIV-1 PROTEASE, SUBSTRATE ANALOG, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2aof:B (ARG157) to (GLY178) CRYSTAL STRUCTURE ANALYSIS OF HIV-1 PROTEASE MUTANT V82A WITH A SUBSTRATE ANALOG P1-P6 | HIV-1 PROTEASE, MUTANT, DIMER, SUBSTRATE ANALOG, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2aog:B (ARG157) to (GLY178) CRYSTAL STRUCTURE ANALYSIS OF HIV-1 PROTEASE MUTANT V82A WITH A SUBSTRATE ANALOG P2-NC | HIV-1 PROTEASE, MUTANT, DIMER, SUBSTRATE ANALOG, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2aoi:B (GLY152) to (GLY178) CRYSTAL STRUCTURE ANALYSIS OF HIV-1 PROTEASE WITH A SUBSTRATE ANALOG P1-P6 | HIV-1 PROTEASE, MUTANT, DIMER, SUBSTRATE ANALOG, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1a9m:A (ARG57) to (GLY78) G48H MUTANT OF HIV-1 PROTEASE IN COMPLEX WITH A PEPTIDIC INHIBITOR U-89360E | ASPARTYL PROTEASE, DRUG RESISTANT, MUTATION
2aoj:B (ARG157) to (GLY178) CRYSTAL STRUCTURE ANALYSIS OF HIV-1 PROTEASE WITH A SUBSTRATE ANALOG P6-PR | HIV-1 PROTEASE, MUTANT, DIMER, SUBSTRATE ANALOG, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2avq:B (ARG57) to (GLY78) KINETICS, STABILITY, AND STRUCTURAL CHANGES IN HIGH RESOLUTION CRYSTAL STRUCTURES OF HIV-1 PROTEASE WITH DRUG RESISTANT MUTATIONS L24I, I50V, AND G73S | HIV-1 PROTEASE, DRUG RESISTANT, SUBSTRATE ANALOG, NON-ACTIVE SITE MUTANTS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2avv:A (GLY52) to (GLY78) KINETICS, STABILITY, AND STRUCTURAL CHANGES IN HIGH RESOLUTION CRYSTAL STRUCTURES OF HIV-1 PROTEASE WITH DRUG RESISTANT MUTATIONS L24I, I50V, AND G73S | DRUG RESISTANCE, HIV-1 PROTEASE,INDINAVIR, SUBSTRATE ANALOG, NON-ACTIVE SITE MUTANTS., HYDROLASE
2avv:E (GLY52) to (GLY78) KINETICS, STABILITY, AND STRUCTURAL CHANGES IN HIGH RESOLUTION CRYSTAL STRUCTURES OF HIV-1 PROTEASE WITH DRUG RESISTANT MUTATIONS L24I, I50V, AND G73S | DRUG RESISTANCE, HIV-1 PROTEASE,INDINAVIR, SUBSTRATE ANALOG, NON-ACTIVE SITE MUTANTS., HYDROLASE
4gzf:A (ARG57) to (GLY78) MULTI-DRUG RESISTANT HIV-1 PROTEASE 769 VARIANT WITH REDUCED LRF PEPTIDE | MULTI-DRUG RESISTANCE, PROTEASE INHIBITOR, DRUG RESISTANCE, SUBSTRATE PEPTIDES, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2awn:D (SER3) to (GLU28) CRYSTAL STRUCTURE OF THE ADP-MG-BOUND E. COLI MALK (CRYSTALLIZED WITH ATP-MG) | ATP-BINDING CASSETTE, TRANSPORT PROTEIN
4gzy:D (TYR132) to (THR154) CRYSTAL STRUCTURES OF BACTERIAL RNA POLYMERASE PAUSED ELONGATION COMPLEXES | RNA POLYMERASE, TRANSCRIPTION, PAUSED TRANSCRIPTION ELONGATION COMPLEX, TRANSCRIPTIONAL PAUSING, DNA DIRECTED RNA TRANSCRIPTION, TRANSCRIPTION-DNA-RNA COMPLEX
4gzz:D (TYR132) to (THR154) CRYSTAL STRUCTURES OF BACTERIAL RNA POLYMERASE PAUSED ELONGATION COMPLEXES | RNA POLYMERASE, TRANSCRIPTION, PAUSED TRANSCRIPTION ELONGATION COMPLEX, TRANSCRIPTIONAL PAUSING, DNA DIRECTED RNA TRANSCRIPTION', TRANSCRIPTION-DNA-RNA HYBRID COMPLEX
1ajv:B (ARG57) to (GLY78) HIV-1 PROTEASE IN COMPLEX WITH THE CYCLIC SULFAMIDE INHIBITOR AHA006 | PROTEASE, ASPARTYL PROTEASE, NON-PEPTIDE INHIBITOR, DRUG DESIGN, HIV-1
1ajx:B (ARG57) to (GLY78) HIV-1 PROTEASE IN COMPLEX WITH THE CYCLIC UREA INHIBITOR AHA001 | PROTEASE, ASPARTYL PROTEASE, NON-PEPTIDE INHIBITOR, DRUG DESIGN, HIV-1
3eif:A (GLY985) to (ASP1014) 1.9 ANGSTROM CRYSTAL STRUCTURE OF THE ACTIVE FORM OF THE C5A PEPTIDASE FROM STREPTOCOCCUS PYOGENES (SCPA) | SUBTILISIN-LIKE CELL ENVELOPE PROTEASE, MULTI-DOMAIN, PA DOMAIN, FIBRONECTIN TYPE III DOMAINS, HYDROLASE
1npa:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE-HUP | PROTEASE, HIV, ASPARTYL PROTEASE, HYDROLASE
1npw:B (ARG257) to (GLY278) CRYSTAL STRUCTURE OF HIV PROTEASE COMPLEXED WITH LGZ479 | PROTEASE, HYDROLASE
3ekq:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF INHIBITOR SAQUINAVIR (SQV) IN COMPLEX WITH MULTI- DRUG RESISTANT HIV-1 PROTEASE (L63P/V82T/I84V) (REFERRED TO AS ACT IN PAPER) | PROTEASE INHIBITOR, DRUG RESISTANCE, ENTROPY ENTHALPY COMPENSATION, AIDS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX, PROTEASE
3ekt:D (ARG57) to (GLY78) CRYSTAL STRUCTURE OF THE INHIBITOR DARUNAVIR (DRV) IN COMPLEX WITH A MULTI-DRUG RESISTANT HIV-1 PROTEASE VARIANT (L10F/G48V/I54V/V64I/V82A) (REFER: FLAP+ IN CITATION.) | HIV-1, PROTEASE, MULTI-DRUG RESISTANCE, DARUNAVIR, AIDS, HYDROLASE
3ekw:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF THE INHIBITOR ATAZANAVIR (ATV) IN COMPLEX WITH A MULTI-DRUG RESISTANCE HIV-1 PROTEASE VARIANT (L10I/G48V/I54V/V64I/V82A) REFER: FLAP+ IN CITATION. | HIV-1, PROTEASE, MULTI-DRUG RESISTANCE, ATAZANAVIR, AIDS, HYDROLASE
2b60:A (ARG57) to (GLY78) STRUCTURE OF HIV-1 PROTEASE MUTANT BOUND TO RITONAVIR | HIV-1 PROTEASE, PROTEASE INHIBITORS, RITONAVIR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3em4:V (ARG57) to (GLY78) CRYSTAL STRUCTURE OF ATAZANAVIR (ATV) IN COMPLEX WITH I50L/A71V DRUG- RESISTANT HIV-1 PROTEASE | DRUG RESISTANCE, HYPERSUSCEPTIBILITY, PROTEASE INHIBITOR, HIV, ATAZANAVIR, AIDS, HYDROLASE, PROTEASE
3em6:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF I50L/A71V MUTANT OF HIV-1 PROTEASE IN COMPLEX WITH INHIBITOR DARUNAVIR | PROTEASE INHIBITOR, HYPER SUSCEPTIBILITY, DRUG RESISTANCE, HIV, DARUNAVIR, AIDS, HYDROLASE, PROTEASE
2oxv:A (ASN214) to (GLN240) STRUCTURE OF THE A138T PROMISCUOUS MUTANT OF THE ECORI RESTRICTION ENDONUCLEASE BOUND TO ITS COGNATE RECOGNITION SITE. | ECORI, TYPE II RESTRICTION ENDONUCLEASE, PROTEIN-DNA INTERACTIONS, PROMISCUOUS MUTANT, RELAXED SPECIFICITY MUTANT, HYDROLASE/DNA COMPLEX
3eoj:A (ASP93) to (TYR122) FMO PROTEIN FROM PROSTHECOCHLORIS AESTUARII 2K AT 1.3A RESOLUTION | EXCITATION ENERGY TRANSFER, BETA SHEET, GAMMA-TURNS, BACTERIOCHLOROPHYLL, CHLOROPHYLL, CHROMOPHORE, ELECTRON TRANSPORT, MAGNESIUM, METAL-BINDING, PHOTOSYNTHESIS, REACTION CENTER, TRANSPORT
1axa:A (ARG57) to (GLY78) ACTIVE-SITE MOBILITY IN HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 PROTEASE AS DEMONSTRATED BY CRYSTAL STRUCTURE OF A28S MUTANT | HIV PROTEASE, MUTANT, X-RAY, ASPARTIC PROTEASE, HYDROLASE, ACID PROTEINASE, ASPARTYL PROTEASE
2b7z:A (ARG57) to (GLY78) STRUCTURE OF HIV-1 PROTEASE MUTANT BOUND TO INDINAVIR | HIV-1, PROTEASE, INDINAVIR, DRUG RESISTANCE, ACTIVE SITE MUTATIONS, NON-ACTIVE SITE MUTATIONS,VIRAL PROTEIN, VIRAL PROTEIN
1nvm:B (GLN248) to (GLY279) CRYSTAL STRUCTURE OF A BIFUNCTIONAL ALDOLASE-DEHYDROGENASE : SEQUESTERING A REACTIVE AND VOLATILE INTERMEDIATE | SEQUESTERED TUNNEL, SUBSTRATE CHANNELING, BIFUNCTIONAL ENZYME, LYASE- OXIDOREDUCTASE COMPLEX
1nvm:D (GLN248) to (GLY279) CRYSTAL STRUCTURE OF A BIFUNCTIONAL ALDOLASE-DEHYDROGENASE : SEQUESTERING A REACTIVE AND VOLATILE INTERMEDIATE | SEQUESTERED TUNNEL, SUBSTRATE CHANNELING, BIFUNCTIONAL ENZYME, LYASE- OXIDOREDUCTASE COMPLEX
1nvm:F (GLN248) to (GLY279) CRYSTAL STRUCTURE OF A BIFUNCTIONAL ALDOLASE-DEHYDROGENASE : SEQUESTERING A REACTIVE AND VOLATILE INTERMEDIATE | SEQUESTERED TUNNEL, SUBSTRATE CHANNELING, BIFUNCTIONAL ENZYME, LYASE- OXIDOREDUCTASE COMPLEX
1nvm:H (GLN248) to (GLY279) CRYSTAL STRUCTURE OF A BIFUNCTIONAL ALDOLASE-DEHYDROGENASE : SEQUESTERING A REACTIVE AND VOLATILE INTERMEDIATE | SEQUESTERED TUNNEL, SUBSTRATE CHANNELING, BIFUNCTIONAL ENZYME, LYASE- OXIDOREDUCTASE COMPLEX
4hap:A (LYS110) to (LEU131) CRYSTAL STRUCTURE OF A GH7 FAMILY CELLOBIOHYDROLASE FROM LIMNORIA QUADRIPUNCTATA IN COMPLEX WITH CELLOBIOSE | CELLOBIOHYDROLASE, HYDROLASE
4hap:B (LYS110) to (LEU131) CRYSTAL STRUCTURE OF A GH7 FAMILY CELLOBIOHYDROLASE FROM LIMNORIA QUADRIPUNCTATA IN COMPLEX WITH CELLOBIOSE | CELLOBIOHYDROLASE, HYDROLASE
4haq:A (LYS110) to (LEU131) CRYSTAL STRUCTURE OF A GH7 FAMILY CELLOBIOHYDROLASE FROM LIMNORIA QUADRIPUNCTATA IN COMPLEX WITH CELLOBIOSE AND CELLOTRIOSE | CELLOBIOHYDROLASE, HYDROLASE
2b9k:A (ASN9) to (TYR30) SOLUTION STRUCTURE OF LCI, AN AMP FROM BACILLUS SUBTILIS | BETA-STRANDED PROTEIN, AMP, ANTIBIOTIC
2p37:A (TRP88) to (ASN118) CRYSTAL STRUCTURE OF A LECTIN FROM CANAVALIA MARITIMA SEEDS (CML) IN COMPLEX WITH MAN1-3MAN-OME | CANAVALIA GLADIATA LECTIN, DIMANNOSIDE, SUGAR BINDING PROTEIN
4wwn:A (PHE473) to (LEU529) CRYSTAL STRUCTURE OF HUMAN PI3K-GAMMA IN COMPLEX WITH (S)-N-(1-(7- FLUORO-2-(PYRIDIN-2-YL)QUINOLIN-3-YL)ETHYL)-9H-PURIN-6-AMINE AMG319 INHIBITOR | KINASE, PHOSPHOTRANSFER, PIP2
4hdb:B (ARG157) to (GLY178) CRYSTAL STRUCTURE OF HIV-1 PROTEASE MUTANTS D30N COMPLEXED WITH INHIBITOR GRL-0519 | ASPARTIC ACID PROTEASE, DRUG RESISTANCE, HIV-1 PROTEASE INHIBITOR GRL-0519, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3ers:X (VAL63) to (ALA86) CRYSTAL STRUCTURE OF E. COLI TRBP111 | OLIGONUCLEOTIDE-OLIGOSACCHARIDE BINDING FOLD, RNA-BINDING, TRNA-BINDING, RNA BINDING PROTEIN
3s2a:A (PHE473) to (LEU529) CRYSTAL STRUCTURE OF PI3K-GAMMA IN COMPLEX WITH A QUINOLINE INHIBITOR | P110-GAMMA, KINASE, PHOSPHOTRANSFER, P101, P84, LEUKOCYTES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1beb:A (GLY17) to (THR49) BOVINE BETA-LACTOGLOBULIN, LATTICE X | LIPOCALIN, MILK WHEY PROTEIN, BOVINE, RETINOL-BINDING
1beb:B (GLY17) to (THR49) BOVINE BETA-LACTOGLOBULIN, LATTICE X | LIPOCALIN, MILK WHEY PROTEIN, BOVINE, RETINOL-BINDING
3s43:B (ARG157) to (GLY178) HIV-1 PROTEASE TRIPLE MUTANTS V32I, I47V, V82I WITH ANTIVIRAL DRUG AMPRENAVIR | AMPRENAVIR, HIV/AIDS, DRUG RESISTANCE, ASPARTIC PROTEASE, MOLECULAR RECOGNITION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4x1v:A (LYS110) to (ASP136) CRYSTAL STRUCTURE OF THE 2ND SH3 DOMAIN FROM HUMAN CD2AP (CMS) IN COMPLEX WITH A PROLINE-RICH PEPTIDE (AA 76-91) FROM HUMAN ARAP1 | ENDOCYTOSIS ADAPTOR PROTEIN, PROTEIN-PEPTIDE BINARY COMPLEX, KIDNEY, SIGNALING PROTEIN, STRUCTURAL GENOMICS CONSORTIUM, SGC
1bim:A (PHE83) to (THR105) CRYSTALLOGRAPHIC STUDIES ON THE BINDING MODES OF P2-P3 BUTANEDIAMIDE RENIN INHIBITORS | ASPARTIC PROTEINASE, ASPARTYL PROTEASE, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, ZYMOGEN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2pf5:D (VAL57) to (TYR78) CRYSTAL STRUCTURE OF THE HUMAN TSG-6 LINK MODULE | LINK MODULE; HYALURONAN-BINDING DOMAIN; ALPHA/BETA DOMAIN, CELL ADHESION
3s54:B (ARG57) to (GLY78) HIV-1 PROTEASE TRIPLE MUTANTS V32I, I47V, V82I WITH ANTIVIRAL DRUG DARUNAVIR IN SPACE GROUP P21212 | DARUNAVIR,HIV/AIDS, DRUG RESISTANCE, ASPARTIC PROTEASE, MOLECULAR RECOGNITION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2bpw:B (ARG57) to (GLY78) HIV-1 PROTEASE-INHIBITOR COMPLEX | ACID PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2bpy:B (ARG57) to (GLY78) HIV-1 PROTEASE-INHIBITOR COMPLEX | ACID PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2bpz:B (ARG57) to (GLY78) HIV-1 PROTEASE-INHIBITOR COMPLEX | ACID PROTEASE, HYDROLASE-HYDROLASE COMPLEX
2bqv:B (ARG157) to (GLY178) HIV-1 PROTEASE IN COMPLEX WITH INHIBITOR AHA455 | HYDROLASE/INHIBITOR, HYDROLASE/INHIBITOR COMPLEX, HIV-1 PROTEASE, INHIBITOR, DRUG DESIGN, HYDROLASE COMPLEX
3s85:D (ARG57) to (GLY78) DISCOVERY OF NEW HIV PROTEASE INHIBITORS WITH POTENTIAL FOR CONVENIENT DOSING AND REDUCED SIDE EFFECTS: A-790742 AND A-792611. | BETA BARREL, ACID PROTEASE, ASPARTIC-TYPE ENDOPEPIDASE ACTIVITY, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2bsd:A (ASN52) to (LYS77) STRUCTURE OF LACTOCOCCAL BACTERIOPHAGE P2 RECEPTOR BINDING PROTEIN | LACTOCOCCUS LACTIS, PHAGE, LLAMA VHH, RECEPTOR BINDING PROTEIN, RECEPTOR
2bsd:B (ASN52) to (LYS77) STRUCTURE OF LACTOCOCCAL BACTERIOPHAGE P2 RECEPTOR BINDING PROTEIN | LACTOCOCCUS LACTIS, PHAGE, LLAMA VHH, RECEPTOR BINDING PROTEIN, RECEPTOR
2pk6:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE (Q7K, L33I, L63I) IN COMPLEX WITH KNI-10033 | PROTEASE COMPLEX, VIRAL PROTEIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2plf:A (TYR51) to (ALA94) THE STRUCTURE OF AIF2GAMMA SUBUNIT FROM THE ARCHAEON SULFOLOBUS SOLFATARICUS IN THE NUCLEOTIDE-FREE FORM. | AIF2, INITIATION FACTOR 2 GAMMA SUBUNIT, INITIATION OF THE TRANSLATION, NUCLEOTIDE BINDING
3fg1:A (PRO453) to (ILE480) CRYSTAL STRUCTURE OF DELTA413-417:GS LOX | LIPOXYGENASE, ARICHIDONIC METABOLISM, DIOXYGENASE, FATTY ACID BIOSYNTHESIS, HEME, IRON, LIPID SYNTHESIS, LYASE, MEMBRANE, METAL- BINDING, MULTIFUNCTIONAL ENZYME, OXIDOREDUCTASE, OXYLIPIN BIOSYNTHESIS
3fg1:D (PRO453) to (ILE480) CRYSTAL STRUCTURE OF DELTA413-417:GS LOX | LIPOXYGENASE, ARICHIDONIC METABOLISM, DIOXYGENASE, FATTY ACID BIOSYNTHESIS, HEME, IRON, LIPID SYNTHESIS, LYASE, MEMBRANE, METAL- BINDING, MULTIFUNCTIONAL ENZYME, OXIDOREDUCTASE, OXYLIPIN BIOSYNTHESIS
3fg3:A (PRO453) to (ILE480) CRYSTAL STRUCTURE OF DELTA413-417:GS I805W LOX | LIPOXYGENASE, ARICHIDONIC METABOLISM, DIOXYGENASE, FATTY ACID BIOSYNTHESIS, HEME, IRON, LIPID SYNTHESIS, LYASE, MEMBRANE, METAL- BINDING, MULTIFUNCTIONAL ENZYME, OXIDOREDUCTASE, OXYLIPIN BIOSYNTHESIS
3fg3:C (PRO453) to (ILE480) CRYSTAL STRUCTURE OF DELTA413-417:GS I805W LOX | LIPOXYGENASE, ARICHIDONIC METABOLISM, DIOXYGENASE, FATTY ACID BIOSYNTHESIS, HEME, IRON, LIPID SYNTHESIS, LYASE, MEMBRANE, METAL- BINDING, MULTIFUNCTIONAL ENZYME, OXIDOREDUCTASE, OXYLIPIN BIOSYNTHESIS
3fg3:D (PRO453) to (ILE480) CRYSTAL STRUCTURE OF DELTA413-417:GS I805W LOX | LIPOXYGENASE, ARICHIDONIC METABOLISM, DIOXYGENASE, FATTY ACID BIOSYNTHESIS, HEME, IRON, LIPID SYNTHESIS, LYASE, MEMBRANE, METAL- BINDING, MULTIFUNCTIONAL ENZYME, OXIDOREDUCTASE, OXYLIPIN BIOSYNTHESIS
2pny:A (ILE128) to (LYS157) STRUCTURE OF HUMAN ISOPENTENYL-DIPHOSPHATE DELTA-ISOMERASE 2 | CAROTENOID BIOSYNTHESIS, CHOLESTEROL BIOSYNTHESIS, ISOMERASE, ISOPRENE BIOSYNTHESIS, LIPID SYNTHESIS, PEROXISOME, STEROID BIOSYNTHESIS, STEROL BIOSYNTHESIS, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
2c11:C (GLU536) to (ASN592) CRYSTAL STRUCTURE OF THE 2-HYDRAZINOPYRIDINE OF SEMICARBAZIDE-SENSITIVE AMINE OXIDASE | OXIDOREDUCTASE, ADHESION PROTEIN-1, 2-HYDROXYPYRIDINE, METAL-BINDING, CELL ADHESION, GLYCOPROTEIN, SIGNAL-ANCHOR, TPQ, TRANSMEMBRANE
3fhh:A (MET605) to (TRP640) CRYSTAL STRUCTURE OF THE HEME/HEMOGLOBIN OUTER MEMBRANE TRANSPORTER SHUA FROM SHIGELLA DYSENTERIAE | MEMBRANE PROTEIN, TRANSPORTER, TONB-DEPENDENT TRANSPORTER, MEMBRANE, RECEPTOR, TONB BOX
1ohr:A (ARG57) to (GLY78) VIRACEPT (R) (NELFINAVIR MESYLATE, AG1343): A POTENT ORALLY BIOAVAILABLE INHIBITOR OF HIV-1 PROTEASE | ASPARTYL PROTEASE, HYDROLASE, HIV-I PROTEASE
4i35:A (GLY131) to (ASN155) THE CRYSTAL STRUCTURE OF SERRALYSIN | AMINO ACID SEQUENCE, BINDING SITES, CALCIUM,X-RAY CRYSTALLOGRAPHY, METALLOENDOPEPTIDASES, PROTEIN STRUCTURE, 1. ZINCIN LIKE 2. SINGLE- STRANDED RIGHT-HANDED BETA-HELIX, HYDROLASE, METAL ION BINDING, EXTRACELLULAR
3fiq:A (GLY14) to (GLY45) ODORANT BINDING PROTEIN OBP1 | LIPOCALIN, ODERANT-BINDING PROTEIN, TRANSPORT PROTEIN
4xiw:A (MET137) to (ALA163) CARBONIC ANHYDRASE CAH3 FROM CHLAMYDOMONAS REINHARDTII IN COMPLEX WITH ACETAZOLAMIDE | LYASE, ACETAZOLAMIDE, PHOTOSYSTEM II-ASSOCIATED
4xiw:B (MET137) to (ALA163) CARBONIC ANHYDRASE CAH3 FROM CHLAMYDOMONAS REINHARDTII IN COMPLEX WITH ACETAZOLAMIDE | LYASE, ACETAZOLAMIDE, PHOTOSYSTEM II-ASSOCIATED
4xiw:C (MET137) to (ALA163) CARBONIC ANHYDRASE CAH3 FROM CHLAMYDOMONAS REINHARDTII IN COMPLEX WITH ACETAZOLAMIDE | LYASE, ACETAZOLAMIDE, PHOTOSYSTEM II-ASSOCIATED
4xiw:D (MET137) to (ALA163) CARBONIC ANHYDRASE CAH3 FROM CHLAMYDOMONAS REINHARDTII IN COMPLEX WITH ACETAZOLAMIDE | LYASE, ACETAZOLAMIDE, PHOTOSYSTEM II-ASSOCIATED
4xix:A (MET137) to (ALA163) CARBONIC ANHYDRASE CAH3 FROM CHLAMYDOMONAS REINHARDTII IN COMPLEX WITH PHOSPHATE. | PHOTOSYSTEM II-ASSOCIATED, LYASE
4xix:C (MET137) to (ALA163) CARBONIC ANHYDRASE CAH3 FROM CHLAMYDOMONAS REINHARDTII IN COMPLEX WITH PHOSPHATE. | PHOTOSYSTEM II-ASSOCIATED, LYASE
4xix:E (MET137) to (ALA163) CARBONIC ANHYDRASE CAH3 FROM CHLAMYDOMONAS REINHARDTII IN COMPLEX WITH PHOSPHATE. | PHOTOSYSTEM II-ASSOCIATED, LYASE
1olp:A (ASP336) to (GLY363) ALPHA TOXIN FROM CLOSTRIDIUM ABSONUM | ZINC PHOSPHOLIPASE C, GAS GANGRENE DETERMINANT, MEMBRANE BINDING, CALCIUM BINDING, HYDROLASE
1olp:D (ASP336) to (GLY363) ALPHA TOXIN FROM CLOSTRIDIUM ABSONUM | ZINC PHOSPHOLIPASE C, GAS GANGRENE DETERMINANT, MEMBRANE BINDING, CALCIUM BINDING, HYDROLASE
2puk:B (ARG6) to (GLU34) CRYSTAL STRUCTURE OF THE BINARY COMPLEX BETWEEN FERREDOXIN: THIOREDOXIN REDUCTASE AND THIOREDOXIN M | THIOREDOXIN, PROTEIN-PROTEIN COMPLEX, REDOX, IRON-SULFUR, ELECTRON TRANSPORT
2puk:F (ARG6) to (GLU34) CRYSTAL STRUCTURE OF THE BINARY COMPLEX BETWEEN FERREDOXIN: THIOREDOXIN REDUCTASE AND THIOREDOXIN M | THIOREDOXIN, PROTEIN-PROTEIN COMPLEX, REDOX, IRON-SULFUR, ELECTRON TRANSPORT
2pva:B (VAL29) to (GLY56) OXIDIZED PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE
2pva:D (VAL29) to (GLY56) OXIDIZED PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE
2pvo:B (ASP5) to (GLU34) CRYSTAL SRTUCTURE OF THE TERNARY COMPLEX BETWEEN THIOREDOXIN F, FERREDOXIN, AND FERREDOXIN: THIOREDOXIN REDUCTASE | THIOREDOXIN, FERREDOXIN. REDOX, IRON-SULFUR CLUSTER, PROTEIN-PROTEIN COMPLEX, ELECTRON TRANSPORT
2pwc:B (ARG57) to (GLY78) HIV-1 PROTEASE IN COMPLEX WITH A AMINO DECORATED PYRROLIDINE-BASED INHIBITOR | PROTEIN-LIGAND COMPLEX, HYDROLASE
2pwr:B (ARG57) to (GLY78) HIV-1 PROTEASE IN COMPLEX WITH A CARBAMOYL DECORATED PYRROLIDINE-BASED INHIBITOR | PROTEIN-LIGAND COMPLEX, HYDROLASE
4ian:A (ARG676) to (GLY694) CRYSTAL STRUCTURE OF APO HUMAN PRPF4B KINASE DOMAIN | KINASE, TRANSFERASE
4ian:B (ARG676) to (VAL697) CRYSTAL STRUCTURE OF APO HUMAN PRPF4B KINASE DOMAIN | KINASE, TRANSFERASE
3sq5:B (LYS454) to (THR502) CRYSTAL STRUCTURE ANALYSIS OF THE YEAST TYROSYL-DNA PHOSPHODIESTERASE H432N MUTANT | PHOSPHODIESTERASE, DNA BINDING, NUCLEAR, HYDROLASE
3sq7:D (LYS454) to (THR502) CRYSTAL STRUCTURE ANALYSIS OF THE YEAST TYROSYL-DNA PHOSPHODIESTERASE H432N_GLU MUTANT | PHOSPHODIESTERASE, DNA BINDING, NUCLEAR, HYDROLASE
4ib7:A (GLY17) to (THR49) BOVINE BETA-LACTOGLOBULIN (ISOFORM A) IN COMPLEX WITH DODECYLTRIMETHYLAMMONIUM (DTAC) | LIPOCALIN, TRANSPORT PROTEIN
4iba:A (GLY17) to (THR49) BOVINE BETA-LACTOGLOBULIN (ISOFORM B) IN COMPLEX WITH DODECYL SULPHATE (SDS) | LIPOCALIN, TRANSPORT PROTEIN
2q2p:A (GLY17) to (PRO50) BETA-LACTOGLOBULIN (REVERSE NATIVE) | LIPOCALIN, VARIANT A, TRANSPORT PROTEIN
2q3k:B (GLY52) to (GLY78) CRYSTAL STRUCTURE OF LYSINE SULFONAMIDE INHIBITOR REVEALS THE DISPLACEMENT OF THE CONSERVED FLAP WATER MOLECULE IN HIV-1 PROTEASE | DRUG DESIGN, HIV-1 PROTEASE, PROTEASE INHIBITORS, VIRAL PROTEIN
1cvm:A (GLY309) to (HIS342) CADMIUM INHIBITED CRYSTAL STRUCTURE OF PHYTASE FROM BACILLUS AMYLOLIQUEFACIENS | THERMOSTABLE BACILLUS PHYTASE PHYTATE PHOSPHATASE CADMIUM CALCIUM, HYDROLASE
1cwo:A (ILE89) to (GLU120) HUMAN CYCLOPHILIN A COMPLEXED WITH THR2, LEU5, D-HIV8, LEU10 CYCLOSPORIN | ISOMERASE-IMMUNOSUPPRESSANT COMPLEX, CYCLOPHILIN-CYCLOSPORIN COMPLEX, CYCLOSPORIN C, IMMUNOSUPPRESSANT
1p49:A (ILE463) to (SER506) STRUCTURE OF HUMAN PLACENTAL ESTRONE/DHEA SULFATASE | STEROID BIOSYNTHESIS, STEROID SULFATASE, ESTRONE SULFATE, DEHYDROEPIANDROSTERONE SULFATE, HUMAN PLACENTAL ENZYME, ENDOPLASMIC RETICULUM MEMBRANE-BOUND, HYDROLASE
2cem:B (ARG157) to (GLY178) P1' EXTENDED HIV-1 PROTEASE INHIBITORS ENCOMPASSING A TERTIARY ALCOHOL IN THE TRANSITION-STATE MIMICKING SCAFFOLD | HIV-1, PROTEASE, INHIBITOR, ASPARTYL PROTEASE, HYDROLASE
4xoa:E (ALA115) to (THR158) CRYSTAL STRUCTURE OF A FIMH*DSG COMPLEX FROM E.COLI K12 IN SPACE GROUP P1 | TYPE I PILUS, CATCH-BOND, CELL ADHESION, LECTIN, UPEC, BACTERIAL ADHESIN, UTI, MANNOSE, ISOMERASE
2qci:B (ARG157) to (GLY178) HIV-1 PROTEASE MUTANT D30N WITH POTENT ANTIVIRAL INHIBITOR GRL-98065 | HIV-1, MUTANT D30N, PROTEASE INHIBITOR, HYDROLASE
1d4h:B (ARG157) to (GLY178) HIV-1 PROTEASE IN COMPLEX WITH THE INHIBITOR BEA435 | DIMER, HYDROLASE
1d4i:B (ARG157) to (GLY178) HIV-1 PROTEASE IN COMPLEX WITH THE INHIBITOR BEA425 | DIMER, HYDROLASE
1d4j:B (ARG157) to (GLY178) HIV-1 PROTEASE IN COMPLEX WITH THE INHIBITOR MSL370 | DIMER, HYDROLASE
1d4y:B (ARG57) to (GLY78) HIV-1 PROTEASE TRIPLE MUTANT/TIPRANAVIR COMPLEX | HYDROLASE, ACID PROTEASE, ASPARTYL PROTEASE
3g1j:A (GLN17) to (ARG40) STRUCTURE FROM THE MOBILE METAGENOME OF VIBRIO CHOLERAE. INTEGRON CASSETTE PROTEIN VCH_CASS4. | NOVEL, INTEGRON CASSETTE PROTEIN, VIBRIO CHOLERAE, OYSTER POND, WOODSHOLE, USA, STRUCTURAL GENOMICS, UNKNOWN FUNCTION, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG
2qd6:B (ARG157) to (GLY178) HIV-1 PROTEASE MUTANT I50V WITH POTENT ANTIVIRAL INHIBITOR GRL-98065 | HIV-1 PROTEASE MUTANT I50V, PROTEASE INHIBITOR, HYDROLASE
2qd7:B (ARG157) to (GLY178) HIV-1 PROTEASE MUTANT V82A WITH POTENT ANTIVIRAL INHIBITOR GRL-98065 | HIV-1 PROTEASE MUTANT V82A, PROTEASE INHIBITOR, HYDROLASE
2qd8:B (ARG157) to (GLY178) HIV-1 PROTEASE MUTANT I84V WITH POTENT ANTIVIRAL INHIBITOR GRL-98065 | HIV-1 PROTEASE MUTANT I84V, PROTEASE INHIBITOR, HYDROLASE
1daz:C (ARG57) to (GLY78) STRUCTURAL AND KINETIC ANALYSIS OF DRUG RESISTANT MUTANTS OF HIV-1 PROTEASE | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX, REDUCED PEPTIDE INHIBITOR
1daz:D (ARG157) to (GLY178) STRUCTURAL AND KINETIC ANALYSIS OF DRUG RESISTANT MUTANTS OF HIV-1 PROTEASE | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX, REDUCED PEPTIDE INHIBITOR
2qi0:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF PROTEASE INHIBITOR, MIT-1-KK80 IN COMPLEX WITH WILD TYPE HIV-1 PROTEASE | DRUG DESIGN, HIV-1 PROTEASE, PROTEASE INHIBITORS, HYDROLASE
1df3:A (GLY17) to (LEU48) SOLUTION STRUCTURE OF A RECOMBINANT MOUSE MAJOR URINARY PROTEIN | LIPOCALIN, CARRIER PROTEIN, PHEROMONE, 8-STRANDED BETA- BARREL, BINDING POCKET, DISULFIDE BRIDGE (64-157), SIGNALING PROTEIN, TRANSPORT PROTEIN
3g7g:C (GLY34) to (ARG66) CRYSTAL STRUCTURE OF THE PROTEIN WITH UNKNOWN FUNCTION FROM CLOSTRIDIUM ACETOBUTYLICUM ATCC 824 | PROTEIN WITH UNKNOWN FUCTION, STRUCTURAL GENOMICS, PSI, MCSG, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, UNKNOWN FUNCTION
3g7g:F (GLY34) to (ARG66) CRYSTAL STRUCTURE OF THE PROTEIN WITH UNKNOWN FUNCTION FROM CLOSTRIDIUM ACETOBUTYLICUM ATCC 824 | PROTEIN WITH UNKNOWN FUCTION, STRUCTURAL GENOMICS, PSI, MCSG, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, UNKNOWN FUNCTION
3g7g:G (GLY34) to (ARG66) CRYSTAL STRUCTURE OF THE PROTEIN WITH UNKNOWN FUNCTION FROM CLOSTRIDIUM ACETOBUTYLICUM ATCC 824 | PROTEIN WITH UNKNOWN FUCTION, STRUCTURAL GENOMICS, PSI, MCSG, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, UNKNOWN FUNCTION
3g7g:H (GLY34) to (ARG66) CRYSTAL STRUCTURE OF THE PROTEIN WITH UNKNOWN FUNCTION FROM CLOSTRIDIUM ACETOBUTYLICUM ATCC 824 | PROTEIN WITH UNKNOWN FUCTION, STRUCTURAL GENOMICS, PSI, MCSG, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, UNKNOWN FUNCTION
1pfp:A (THR72) to (ASP114) CATHELIN-LIKE MOTIF OF PROTEGRIN-3 | PG-3, SEMET, SECYS, DISELENIDE, ANTIMICROBIAL PROTEIN
1dj7:B (ARG6) to (GLU34) CRYSTAL STRUCTURE OF FERREDOXIN THIOREDOXIN REDUCTASE | 4FE-4S CLUSTER BINDING FOLD WITH CXCX16CXCX8CXC BINDING MOTIF, ELECTRON TRANSPORT
4ipm:A (LYS110) to (LEU131) CRYSTAL STRUCTURE OF A GH7 FAMILY CELLOBIOHYDROLASE FROM LIMNORIA QUADRIPUNCTATA IN COMPLEX WITH THIOCELLOBIOSE | THIOCELLOBIOSE, CELLOBIOHYDROLASE, HYDROLASE
2qmp:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE COMPLEXED WITH PL-100 | HIV-1 PROTEASE, ASPARTYL PROTEASE, HYDROLASE, MULTIFUNCTIONAL ENZYME, NUCLEOTIDYLTRANSFERASE, RNA- DIRECTED DNA POLYMERASE, TRANSFERASE
2qnn:B (GLY52) to (GLY78) HIV-1 PROTEASE IN COMPLEX WITH A MULTIPLE DECORATED PYRROLIDINE-BASED INHIBITOR | PROTEIN-LIGAND COMPLEX, AIDS, ASPARTYL PROTEASE, CAPSID MATURATION, CORE PROTEIN, DNA INTEGRATION, DNA RECOMBINATION, DNA-DIRECTED DNA POLYMERASE, ENDONUCLEASE, HYDROLASE, LIPOPROTEIN, MAGNESIUM, MEMBRANE, METAL-BINDING, MULTIFUNCTIONAL ENZYME, MYRISTATE, NUCLEASE, NUCLEOTIDYLTRANSFERASE, PHOSPHORYLATION, PROTEASE, RNA- BINDING, RNA-DIRECTED DNA POLYMERASE, TRANSFERASE, VIRAL NUCLEOPROTEIN, VIRION, ZINC-FINGER
2cws:A (ASN274) to (SER307) CRYSTAL STRUCTURE AT 1.0 A OF ALGINATE LYASE A1-II', A MEMBER OF POLYSACCHARIDE LYASE FAMILY-7 | ALGINATE LYASE, POLYSACCHARIDE LYASE FAMILY-7, LYASE
1pnz:A (LEU699) to (PHE741) CRYSTAL STRUCTURE OF FERRIC CITRATE TRANSPORTER FECA IN THE UNLIGANDED FORM | OUTER MEMBRANE PROTEIN, BETA BARREL, TONB-DEPENDENT TRANSPORT
1po0:A (LEU699) to (PHE741) CRYSTAL STRUCTURE OF FERRIC CITRATE TRANSPORTER FECA IN COMPLEX WITH IRON-FREE CITRATE | OUTER MEMBRANE PROTEIN, BETA BARREL, TONB-DEPENDENT TRANSPORT, CITRATE, SIDEROPHORE
1po3:A (LEU699) to (LYS740) CRYSTAL STRUCTURE OF FERRIC CITRATE TRANSPORTER FECA IN COMPLEX WITH FERRIC CITRATE | OUTER MEMBRANE PROTEIN, BETA BARREL, TONB-DEPENDENT TRANSPORT, CITRATE, SIDEROPHORE, IRON
1pp1:X (ARG97) to (ALA116) CRYSTAL STRUCTURE OF THE BORNA DISEASE VIRUS NUCLEOPROTEIN | RNA VIRUS NUCLEOPROTEIN TETRAMER, VIRAL PROTEIN
1dw6:C (ARG57) to (GLY78) STRUCTURAL AND KINETIC ANALYSIS OF DRUG RESISTANT MUTANTS OF HIV-1 PROTEASE | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1dw6:D (ARG157) to (GLY178) STRUCTURAL AND KINETIC ANALYSIS OF DRUG RESISTANT MUTANTS OF HIV-1 PROTEASE | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2quy:A (VAL29) to (GLY56) TRUNCATED MUTANT ASN175ALA OF PENICILLIN V ACYLASE FROM BACILLUS SPHAERICUS | PENICILLIN, AUTOPROTEOLYSIS, NTN, OXY-ANION HOLE, ANTIBIOTIC RESISTANCE, HYDROLASE, ZYMOGEN
2quy:C (VAL29) to (GLY56) TRUNCATED MUTANT ASN175ALA OF PENICILLIN V ACYLASE FROM BACILLUS SPHAERICUS | PENICILLIN, AUTOPROTEOLYSIS, NTN, OXY-ANION HOLE, ANTIBIOTIC RESISTANCE, HYDROLASE, ZYMOGEN
2quy:D (VAL29) to (GLY56) TRUNCATED MUTANT ASN175ALA OF PENICILLIN V ACYLASE FROM BACILLUS SPHAERICUS | PENICILLIN, AUTOPROTEOLYSIS, NTN, OXY-ANION HOLE, ANTIBIOTIC RESISTANCE, HYDROLASE, ZYMOGEN
2quy:E (VAL29) to (GLY56) TRUNCATED MUTANT ASN175ALA OF PENICILLIN V ACYLASE FROM BACILLUS SPHAERICUS | PENICILLIN, AUTOPROTEOLYSIS, NTN, OXY-ANION HOLE, ANTIBIOTIC RESISTANCE, HYDROLASE, ZYMOGEN
4y0r:A (GLY17) to (THR49) BOVINE BETA-LACTOGLOBULIN COMPLEX WITH PRAMOCAINE CRYSTALLIZED FROM AMMONIUM SULPHATE (BLG-PRM2) | TRANSPORT, LIGAND BINDING
3ta4:E (GLN114) to (ASP145) SMALL LACCASE FROM AMYCOLATOPSIS SP. ATCC 39116 COMPLEXED WITH 1-(3,4- DIMETHOXYPHENYL)-2-(2-METHOXYPHENOXY)-1,3-DIHYDROXYPROPANE | 2-DOMAIN COPPER OXIDASE, OXIDOREDUCTASE, SECRETED
3gn5:B (GLY14) to (GLY34) STRUCTURE OF THE E. COLI PROTEIN MQSA (YGIT/B3021) | ZN-BINDING PROTEIN, HTH-XRE DNA BINDING MOTIF, DNA-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, DNA BINDING PROTEIN
2r3w:B (ARG57) to (GLY78) I84V HIV-1 PROTEASE IN COMPLEX WITH A AMINO DECORATED PYRROLIDINE-BASED INHIBITOR | PROTEIN-LIGAND COMPLEX, HYDROLASE
2r4i:A (ASN82) to (LEU106) CRYSTAL STRUCTURE OF A NTF2-LIKE PROTEIN (CHU_1428) FROM CYTOPHAGA HUTCHINSONII ATCC 33406 AT 1.60 A RESOLUTION | NTF2-LIKE PROTEIN, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, UNKNOWN FUNCTION
2r73:A (ARG26) to (GLU57) CRYSTAL STRUCTURE OF THE POSSUM MILK WHEY LIPOCALIN TRICHOSURIN AT PH 8.2 | LIPOCALIN, BETA BARREL, MILK WHEY LIPOCALIN, DIMER, GLYCOPROTEIN, MILK PROTEIN, SECRETED, TRANSPORT, TRANSPORT PROTEIN
2dl5:A (THR15) to (GLU39) SOLUTION STRUCTURE OF THE FIRST SH3 DOMAIN OF HUMAN KIAA0769 PROTEIN | SH3 DOMAIN, KIAA0769, FCHSD2, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, UNKNOWN FUNCTION
1ebw:B (ARG157) to (GLY178) HIV-1 PROTEASE IN COMPLEX WITH THE INHIBITOR BEA322 | DIMER, PROTEIN-INHIBITOR COMPLEX, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1ec0:B (ARG157) to (GLY178) HIV-1 PROTEASE IN COMPLEX WITH THE INHIBITOR BEA403 | DIMER, PROTEIN-INHIBITOR COMPLEX, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1ec1:B (ARG157) to (GLY178) HIV-1 PROTEASE IN COMPLEX WITH THE INHIBITOR BEA409 | DIMER, PROTEIN-INHIBITOR COMPLEX, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1ec3:B (ARG157) to (GLY178) HIV-1 PROTEASE IN COMPLEX WITH THE INHIBITOR MSA367 | DIMER, PROTEIN-INHIBITOR COMPLEX, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
3tkg:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV MODEL PROTEASE PRECURSOR/SAQUINAVIR COMPLEX | HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3tkw:B (GLY52) to (GLY78) CRYSTAL STRUCTURE OF HIV PROTEASE MODEL PRECURSOR/DARUNAVIR COMPLEX | HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1edq:A (THR36) to (ASN70) CRYSTAL STRUCTURE OF CHITINASE A FROM S. MARCESCENS AT 1.55 ANGSTROMS | BETA-ALPHA (TIM) BARREL, HYDROLASE
3tl9:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV PROTEASE MODEL PRECURSOR/SAQUINAVIR COMPLEX | HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3tof:B (ARG57) to (GLY78) HIV-1 PROTEASE - EPOXYDIC INHIBITOR COMPLEX (PH 6 - ORTHOROMBIC CRYSTAL FORM P212121) | HIV PR, EPOXIDE, IN-CRYSTAL REACTION, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3tog:A (GLY52) to (GLY78) HIV-1 PROTEASE - EPOXYDIC INHIBITOR COMPLEX (PH 9 - MONOCLINIC CRYSTAL FORM P21) | HIV PR, EPOXIDE, IN-CRYSTAL REACTION, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3tog:C (ARG57) to (GLY78) HIV-1 PROTEASE - EPOXYDIC INHIBITOR COMPLEX (PH 9 - MONOCLINIC CRYSTAL FORM P21) | HIV PR, EPOXIDE, IN-CRYSTAL REACTION, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3tog:D (GLY52) to (GLY78) HIV-1 PROTEASE - EPOXYDIC INHIBITOR COMPLEX (PH 9 - MONOCLINIC CRYSTAL FORM P21) | HIV PR, EPOXIDE, IN-CRYSTAL REACTION, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3toh:B (ARG57) to (GLY78) HIV-1 PROTEASE - EPOXYDIC INHIBITOR COMPLEX (PH 9 - ORTHOROMBIC CRYSTAL FORM P212121) | HIV PR, EPOXIDE, IN-CRYSTAL REACTION, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1ehn:A (THR36) to (ASN70) CRYSTAL STRUCTURE OF CHITINASE A MUTANT E315Q COMPLEXED WITH OCTA-N- ACETYLCHITOOCTAOSE (NAG)8. | TIM BARREL, PROTEIN-OLIGOSACCHARIDE COMPLEX, HYDROLASE
4jhn:A (LYS55) to (LYS82) THE CRYSTAL STRUCTURE OF THE RPGR RCC1-LIKE DOMAIN | RCC1, BETA PROPELLAR, SEVEN BLADED-PROPELLER, UNKNOWN FUNCTION
4jhn:B (LYS55) to (LYS82) THE CRYSTAL STRUCTURE OF THE RPGR RCC1-LIKE DOMAIN | RCC1, BETA PROPELLAR, SEVEN BLADED-PROPELLER, UNKNOWN FUNCTION
4jhn:D (LYS55) to (LYS82) THE CRYSTAL STRUCTURE OF THE RPGR RCC1-LIKE DOMAIN | RCC1, BETA PROPELLAR, SEVEN BLADED-PROPELLER, UNKNOWN FUNCTION
1eib:A (THR36) to (ASN70) CRYSTAL STRUCTURE OF CHITINASE A MUTANT D313A COMPLEXED WITH OCTA-N- ACETYLCHITOOCTAOSE (NAG)8. | TIM BARREL, PROTEIN-OLIGOSACCHARIDE COMPLEX, HYDROLASE
1qc9:A (ASN214) to (GLN240) THE CRYSTALLOGRAPHIC STRUCTURE OF RESTRICTION ENDONUCLEASE ECO RI AT 3.3 A IN THE ABSENSE OF DNA | PROTEIN, RESTRICTION ENDONUCLEASE, APOENZYME, ENDONUCLEASE
1qc9:B (ASN214) to (GLN240) THE CRYSTALLOGRAPHIC STRUCTURE OF RESTRICTION ENDONUCLEASE ECO RI AT 3.3 A IN THE ABSENSE OF DNA | PROTEIN, RESTRICTION ENDONUCLEASE, APOENZYME, ENDONUCLEASE
1qc9:C (ASN214) to (GLN240) THE CRYSTALLOGRAPHIC STRUCTURE OF RESTRICTION ENDONUCLEASE ECO RI AT 3.3 A IN THE ABSENSE OF DNA | PROTEIN, RESTRICTION ENDONUCLEASE, APOENZYME, ENDONUCLEASE
2duo:B (GLY156) to (ASN182) CRYSTAL STRUCTURE OF VIP36 EXOPLASMIC/LUMENAL DOMAIN, CA2+- BOUND FORM | BETA SANDWICH, CARBOHYDRATE BINDING PROTEIN, CARGO RECEPTOR, PROTEIN TRANSPORT
2dur:A (GLY156) to (ASN182) CRYSTAL STRUCTURE OF VIP36 EXOPLASMIC/LUMENAL DOMAIN, CA2+/MAN2-BOUND FORM | BETA SANDWICH, CARBOHYDRATE BINDING PROTEIN, CARGO RECEPTOR, PROTEIN TRANSPORT
3tsu:A (GLY494) to (ARG519) CRYSTAL STRUCTURE OF E. COLI HYPF WITH AMP-PNP AND CARBAMOYL PHOSPHATE | ZN FINGER, NUCLEOTIDE BINDING, HYDROGENASE MATURATION FACTOR, TRANSFERASE
3ttf:A (GLY494) to (ARG519) CRYSTAL STRUCTURE OF E. COLI HYPF WITH AMP AND CARBAMOYL PHOSPHATE | ZN FINGER, NUCLEOTIDE BINDING, HYDROGENASE MATURATION FACTOR, HYPE, TRANSFERASE
2rnm:B (SER257) to (GLY282) STRUCTURE OF THE HET-S(218-289) PRION IN ITS AMYLOID FORM OBTAINED BY SOLID-STATE NMR | HET-S(218-289), BETA-SOLENOID, PRION, AMYLOID FIBRIL, PARALLEL BETA- SHEETS, HYDROPHOBIC CORE, SALT BRIDGES, ASPARAGINE LADDERS, BETA- HELIX, PROTEIN FIBRIL
3h4l:B (GLY257) to (SER298) CRYSTAL STRUCTURE OF N TERMINAL DOMAIN OF A DNA REPAIR PROTEIN | PMS1, ATP BINDING, DNA REPAIR, DNA DAMAGE, NUCLEUS, PHOSPHOPROTEIN, DNA BINDING PROTEIN, PROTEIN BINDING
3h5b:B (ARG157) to (GLY178) CRYSTAL STRUCTURE OF WILD TYPE HIV-1 PROTEASE WITH NOVEL P1'-LIGAND GRL-02031 | HIV-1, WILD TYPE PROTEASE, PROTEASE INHIBITOR, P1'-LIGAND, AIDS, HYDROLASE
2e6v:A (GLY156) to (ASN183) CRYSTAL STRUCTURE OF VIP36 EXOPLASMIC/LUMENAL DOMAIN, CA2+/MAN3GLCNAC-BOUND FORM | BETA SANDWICH, CARBOHYDRATE BINDING PROTEIN, CARGO RECEPTOR, PROTEIN TRANSPORT
2e6v:C (GLY156) to (ASN182) CRYSTAL STRUCTURE OF VIP36 EXOPLASMIC/LUMENAL DOMAIN, CA2+/MAN3GLCNAC-BOUND FORM | BETA SANDWICH, CARBOHYDRATE BINDING PROTEIN, CARGO RECEPTOR, PROTEIN TRANSPORT
2e9x:C (GLU1030) to (PRO1069) THE CRYSTAL STRUCTURE OF HUMAN GINS CORE COMPLEX | GINS COMPLEX, EUKARYOTIC DNA REPLICATION
2e9x:G (GLU30) to (GLU67) THE CRYSTAL STRUCTURE OF HUMAN GINS CORE COMPLEX | GINS COMPLEX, EUKARYOTIC DNA REPLICATION
1f7a:A (ARG57) to (GLY78) HOW DOES A SYMMETRIC DIMER RECOGNIZE AN ASYMMETRIC SUBSTRATE? A SUBSTRATE COMPLEX OF HIV-1 PROTEASE. | CAPSID, SUBSTRATE RECOGNITION, HYDROLASE
3u4k:A (SER144) to (SER175) CRYSTAL STRUCTURE OF THE RECEPTOR BINDING DOMAIN OF PLASMID-BORN ADHESIN MRKD1P OF KLEBSIELLA PNEUMONIAE | PILI ADHESION, COLLAGEN V BINDER, PATHOGENICITY, JELLY-ROLL BETA BARREL FOLD, CELL ADHESION
2uxz:A (ARG57) to (GLY78) TWO-CARBON-ELONGATED HIV-1 PROTEASE INHIBITORS WITH A TERTIARY-ALCOHOL-CONTAINING TRANSITION-STATE MIMIC | HIV-1, PROTEASE, HYDROLASE, INHIBITOR, ASPARTYL PROTEASE
2uy0:A (ARG57) to (GLY78) TWO-CARBON-ELONGATED HIV-1 PROTEASE INHIBITORS WITH A TERTIARY-ALCOHOL-CONTAINING TRANSITION-STATE MIMIC | HIV-1, PROTEASE, HYDROLASE, INHIBITOR, ASPARTYL PROTEASE
1fej:D (ARG157) to (GLY178) STRUCTURAL IMPLICATIONS OF DRUG RESISTANT MUTANTS OF HIV-1 PROTEASE: HIGH RESOLUTION CRYSTAL STRUCTURES OF THE MUTANT PROTEASE/SUBSTRATE ANALOG COMPLEXES | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1ff0:C (ARG57) to (GLY78) STRUCTURAL IMPLICATIONS OF DRUG RESISTANT MUTANTS OF HIV-1 PROTEASE: HIGH RESOLUTION CRYSTAL STRUCTURES OF THE MUTANT PROTEASE/SUBSTRATE ANALOG COMPLEXES. | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1ff0:D (ARG157) to (GLY178) STRUCTURAL IMPLICATIONS OF DRUG RESISTANT MUTANTS OF HIV-1 PROTEASE: HIGH RESOLUTION CRYSTAL STRUCTURES OF THE MUTANT PROTEASE/SUBSTRATE ANALOG COMPLEXES. | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1fff:D (ARG157) to (GLY178) STRUCTURAL IMPLICATIONS OF DRUG RESISTANT MUTANTS OF HIV-1 PROTEASE : HIGH RESOLUTION CRYSTAL STRUCTURES OF THE MUTANT PROTEASE/SUBSTRATE ANALOG COMPLEXES. | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1ffi:D (ARG157) to (GLY178) STRUCTURAL IMPLICATIONS OF DRUG RESISTANT MUTANTS OF HIV-1 PROTEASE: HIGH RESOLUTION CRYSTAL STRUCTURES OF THE MUTANT PROTEASE/SUBSTRATE ANALOG COMPLEXES | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1fg6:D (ARG157) to (GLY178) STRUCTURAL IMPLICATIONS OF DRUG RESISTANT MUTANTS OF HIV-1 PROTEASE: HIGH RESOLUTION CRYSTAL STRUCTURES OF THE MUTANT PROTEASE/SUBSTRATE ANALOG COMPLEXES | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1fgc:D (ARG157) to (GLY178) STRUCTURAL IMPLICATIONS OF DRUG RESISTANT MUTANTS OF HIV-1 PROTEASE: HIGH RESOLUTION CRYSTAL STRUCTURES OF THE MUTANT PROTEASE/SUBSTRATE ANALOG COMPLEXES | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1r5n:A (SER492) to (ASP515) CRYSTAL STRUCTURE ANALYSIS OF SUP35 COMPLEXED WITH GDP | TRANSLATION TERMINATION, PEPTIDE RELEASE, GTPASE
1fiv:A (THR66) to (ASP94) STRUCTURE OF AN INHIBITOR COMPLEX OF PROTEINASE FROM FELINE IMMUNODEFICIENCY VIRUS | ACID PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1r77:B (ALA285) to (LYS317) CRYSTAL STRUCTURE OF THE CELL WALL TARGETING DOMAIN OF PEPTIDYLGLYCAN HYDROLASE ALE-1 | SH3B DOMAIN, CELL WALL TARGETING DOMAIN, LYSOSTAPHIN, PEPTIDOGLYCAN HYDROLASE, GLYCYLGLYCINE ENDOPEPTIDASE
1fl0:A (VAL207) to (ALA230) CRYSTAL STRUCTURE OF THE EMAP2/RNA-BINDING DOMAIN OF THE P43 PROTEIN FROM HUMAN AMINOACYL-TRNA SYNTHETASE COMPLEX | RNA-BINDING DOMAIN, OB-FOLD, TRNA SYNTHETASE COMPLEX, RNA BINDING PROTEIN
3uex:A (GLY17) to (THR49) BOVINE BETA-LACTOGLOBULIN COMPLEX WITH STEARIC ACID | BETA PROTEIN, BETA BARREL, LIPOCALIN, BOVINE MILK, TRANSPORT PROTEIN
2eul:B (GLY131) to (GLY156) STRUCTURE OF THE TRANSCRIPTION FACTOR GFH1. | GFH1, TRANSCRIPTION FACTOR, RNA POLYMERASE, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, STRUCTURAL GENOMICS, TRANSCRIPTION
2eul:D (GLY131) to (GLY156) STRUCTURE OF THE TRANSCRIPTION FACTOR GFH1. | GFH1, TRANSCRIPTION FACTOR, RNA POLYMERASE, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, STRUCTURAL GENOMICS, TRANSCRIPTION
4k4p:A (ARG57) to (GLY78) TL-3 INHIBITED TRP6ALA HIV PROTEASE | FRAGMENT BINDING, EXOSITE, PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4k4q:A (ARG57) to (GLY78) TL-3 INHIBITED TRP6ALA HIV PROTEASE WITH 3-BROMO-2,6-DIMETHOXYBENZOIC ACID BOUND IN FLAP SITE | FRAGMENT BINDING, EXOSITE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4k4r:A (ARG57) to (GLY78) TL-3 INHIBITED TRP6ALA HIV PROTEASE WITH 1-BROMO-2-NAPTHOIC ACID BOUND IN EXOSITE | FRAGMENT BINDING, EXOSITE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1foc:A (TYR52) to (PHE72) CYTOCHROME C557: IMPROPERLY FOLDED THERMUS THERMOPHILUS C552 | CYTOCHROME C, THERMUS THERMOPHILUS, HEME INVERSION, ELECTRON TRANSPORT
1fq8:A (TRP190) to (THR216) X-RAY STRUCTURE OF DIFLUOROSTATINE INHIBITOR CP81,198 BOUND TO SACCHAROPEPSIN | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2ez7:A (PHE66) to (TRP97) CARBONIC ANHYDRASE ACTIVATORS. ACTIVATION OF ISOZYMES I, II, IV, VA, VII AND XIV WITH L- AND D-HISTIDINE AND CRYSTALLOGRAPHIC ANALYSIS OF THEIR ADDUCTS WITH ISOFORM II: ENGINEERING PROTON TRANSFER PROCESSES WITHIN THE ACTIVE SITE OF AN ENZYME | CARBONIC ANHYDRASE II, ACTIVATORS, LYASE
2vat:A (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE IN COMPLEX WITH COENZYME A | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vat:C (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE IN COMPLEX WITH COENZYME A | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vat:D (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE IN COMPLEX WITH COENZYME A | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vat:E (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE IN COMPLEX WITH COENZYME A | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vat:G (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE IN COMPLEX WITH COENZYME A | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vat:H (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE IN COMPLEX WITH COENZYME A | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vat:J (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE IN COMPLEX WITH COENZYME A | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vat:K (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE IN COMPLEX WITH COENZYME A | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vat:L (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE IN COMPLEX WITH COENZYME A | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vav:A (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE (DAC-SOAK) | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vav:C (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE (DAC-SOAK) | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vav:D (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE (DAC-SOAK) | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vav:E (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE (DAC-SOAK) | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vav:G (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE (DAC-SOAK) | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vav:H (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE (DAC-SOAK) | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vav:K (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE (DAC-SOAK) | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vav:L (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE (DAC-SOAK) | ACETYL TRANSFERASE, A/B- HYDROLASE FOLD, TRANSFERASE, ACYLTRANSFERASE, ACETYL COENZYME A, ANTIBIOTIC BIOSYNTHESIS, CEPHALOSPORIN BIOSYNTHESIS
2vax:A (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE (CEPHALOSPORIN C-SOAK) | DEACETYLCEPHALOSPORIN C, CEPHALOSPORIN BIOSYNTHESIS, A/B- HYDROLASE FOLD, ANTIBIOTIC BIOSYNTHESIS, TRANSFERASE, ACYLTRANSFERASE, ACETYL TRANSFERASE
2vax:D (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE (CEPHALOSPORIN C-SOAK) | DEACETYLCEPHALOSPORIN C, CEPHALOSPORIN BIOSYNTHESIS, A/B- HYDROLASE FOLD, ANTIBIOTIC BIOSYNTHESIS, TRANSFERASE, ACYLTRANSFERASE, ACETYL TRANSFERASE
2vax:E (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE (CEPHALOSPORIN C-SOAK) | DEACETYLCEPHALOSPORIN C, CEPHALOSPORIN BIOSYNTHESIS, A/B- HYDROLASE FOLD, ANTIBIOTIC BIOSYNTHESIS, TRANSFERASE, ACYLTRANSFERASE, ACETYL TRANSFERASE
2vax:G (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE (CEPHALOSPORIN C-SOAK) | DEACETYLCEPHALOSPORIN C, CEPHALOSPORIN BIOSYNTHESIS, A/B- HYDROLASE FOLD, ANTIBIOTIC BIOSYNTHESIS, TRANSFERASE, ACYLTRANSFERASE, ACETYL TRANSFERASE
2vax:H (ASP17) to (GLY43) CRYSTAL STRUCTURE OF DEACETYLCEPHALOSPORIN C ACETYLTRANSFERASE (CEPHALOSPORIN C-SOAK) | DEACETYLCEPHALOSPORIN C, CEPHALOSPORIN BIOSYNTHESIS, A/B- HYDROLASE FOLD, ANTIBIOTIC BIOSYNTHESIS, TRANSFERASE, ACYLTRANSFERASE, ACETYL TRANSFERASE
4yx7:D (LEU8) to (CYS46) COMPLEX OF SPAO(SPOA1,2) AND ORGB(APAR)::T4LYSOZYME FUSION PROTEIN | TYPE III SECRETION SYSTEM, PROTEIN TRANSPORT
4kb9:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF WILD-TYPE HIV-1 PROTEASE WITH NOVEL TRICYCLIC P2- LIGANDS GRL-0739A | SPARTIC ACID PROTEASE, HIV-1 PROTEASE INHIBITOR GRL-0739A, A NOVEL TRICYCLIC P2-LIGAND,, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2f81:B (ARG157) to (GLY178) HIV-1 PROTEASE MUTANT L90M COMPLEXED WITH INHIBITOR TMC114 | HIV-1 PROTEASE-INHIBITOR COMPLEX, HYDROLASE
2f8g:B (ARG157) to (GLY178) HIV-1 PROTEASE MUTANT I50V COMPLEXED WITH INHIBITOR TMC114 | HIV-1 PROTEASE-INHIBITOR COMPLEX, HYDROLASE
1g2k:B (ARG57) to (GLY78) HIV-1 PROTEASE WITH CYCLIC SULFAMIDE INHIBITOR, AHA047 | HIV, PROTEASE INHIBITORS, HYDROLASE
1g35:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE IN COMPLEX WITH INHIBITOR, AHA024 | PROTEIN-INHIBITOR COMPLEX, HYDROLASE
2fde:A (ARG57) to (GLY78) WILD TYPE HIV PROTEASE BOUND WITH GW0385 | HIV PROTEASE, INHIBITOR, GW0385, HYDROLASE
2vdd:B (LEU61) to (SER96) CRYSTAL STRUCTURE OF THE OPEN STATE OF TOLC OUTER MEMBRANE COMPONENT OF MUTLIDRUG EFFLUX PUMPS | BETA BARREL, ALPHA HELICAL BARREL, MULTIDRUG EFFLUX PUMP, INTEGRAL MEMBRANE PROTEIN, OUTER MEMBRANE, MEMBRANE, TRANSPORT, TRANSMEMBRANE, TRANSPORT PROTEIN
2vdd:C (LEU61) to (SER96) CRYSTAL STRUCTURE OF THE OPEN STATE OF TOLC OUTER MEMBRANE COMPONENT OF MUTLIDRUG EFFLUX PUMPS | BETA BARREL, ALPHA HELICAL BARREL, MULTIDRUG EFFLUX PUMP, INTEGRAL MEMBRANE PROTEIN, OUTER MEMBRANE, MEMBRANE, TRANSPORT, TRANSMEMBRANE, TRANSPORT PROTEIN
1sdt:B (GLY152) to (GLY178) CRYSTAL STRUCTURES OF HIV PROTEASE V82A AND L90M MUTANTS REVEAL CHANGES IN INDINAVIR BINDING SITE. | DRUG RESISTANCE; HIV-1, HYDROLASE
1sdu:A (ARG57) to (GLY78) CRYSTAL STRUCTURES OF HIV PROTEASE V82A AND L90M MUTANTS REVEAL CHANGES IN INDINAVIR BINDING SITE. | DRUG RESISTANCE HIV-1 PROTEASE, HYDROLASE
1sdu:B (ARG157) to (GLY178) CRYSTAL STRUCTURES OF HIV PROTEASE V82A AND L90M MUTANTS REVEAL CHANGES IN INDINAVIR BINDING SITE. | DRUG RESISTANCE HIV-1 PROTEASE, HYDROLASE
2fxe:A (ARG57) to (GLY78) X-RAY CRYSTAL STRUCTURE OF HIV-1 PROTEASE CRM MUTANT COMPLEXED WITH ATAZANAVIR (BMS-232632) | HUMAN IMMUNODEFICIENCY VIRUS (HIV), HIV-1 PROTEASE, REYATAZ, ATAZANAVIR, BMS-232632, HYDROLASE
2fxe:B (ARG57) to (GLY78) X-RAY CRYSTAL STRUCTURE OF HIV-1 PROTEASE CRM MUTANT COMPLEXED WITH ATAZANAVIR (BMS-232632) | HUMAN IMMUNODEFICIENCY VIRUS (HIV), HIV-1 PROTEASE, REYATAZ, ATAZANAVIR, BMS-232632, HYDROLASE
1gnh:A (ALA131) to (ASP163) HUMAN C-REACTIVE PROTEIN | PENTRAXIN, ACUTE-PHASE REACTANT, ACUTE-PHASE PROTEIN
1gnh:C (ALA131) to (ASP163) HUMAN C-REACTIVE PROTEIN | PENTRAXIN, ACUTE-PHASE REACTANT, ACUTE-PHASE PROTEIN
1gnh:E (ALA131) to (ASP163) HUMAN C-REACTIVE PROTEIN | PENTRAXIN, ACUTE-PHASE REACTANT, ACUTE-PHASE PROTEIN
1gs0:A (THR491) to (VAL537) CRYSTAL STRUCTURE OF THE CATALYTIC FRAGMENT OF MURINE POLY (ADP-RIBOSE) POLYMERASE-2 | TRANSFERASE, CRYSTAL STRUCTURE, CATALYTIC FRAGMENT, POLYMERASE TRANSFERASE, NUCLEAR PROTEIN, DNA-BINDING
3i6o:B (ARG157) to (GLY178) CRYSTAL STRUCTURE OF WILD TYPE HIV-1 PROTEASE WITH MACROCYCLIC INHIBITOR GRL-0216A | HIV-1, WILD TYPE PROTEASE, PROTEASE INHIBITOR, MACROCYCLIC LIGAND, AIDS, ASPARTYL PROTEASE, HYDROLASE
3i7e:A (ARG57) to (GLY78) CO-CRYSTAL STRUCTURE OF HIV-1 PROTEASE BOUND TO A MUTANT RESISTANT INHIBITOR UIC-98038 | AIDS, HIV, HIV PRTEASE, HIV-PROTEASE INHIBITOR, DRUG DESIGN, ASPARTIC PROTEASE, ACID PROTEASE, STRUCTURE BASED DRUG DESIGN, ASPARTYL PROTEASE, HYDROLASE, PROTEASE
2vxm:A (GLU241) to (THR287) SCREENING A LIMITED STRUCTURE-BASED LIBRARY IDENTIFIES UDP- GALNAC-SPECIFIC MUTANTS OF ALPHA-1,3 GALACTOSYLTRANSFERASE | GLYCOSYLTRANSFERASE, 3 GALACTOSYLTRANSFERASE, TRANSMEMBRANE, GOLGI APPARATUS, ENZYME MECHANISM, GLYCOPROTEIN, METAL-BINDING, SIGNAL-ANCHOR, ALPHA-1, MEMBRANE, MANGANESE, TRANSFERASE, GLYCOSYLTRANSFERASE GALACTOSYLTRANSFERASE, TRANSFERASE SUBSTRATE SPECIFICITY
2vxm:B (GLU241) to (THR287) SCREENING A LIMITED STRUCTURE-BASED LIBRARY IDENTIFIES UDP- GALNAC-SPECIFIC MUTANTS OF ALPHA-1,3 GALACTOSYLTRANSFERASE | GLYCOSYLTRANSFERASE, 3 GALACTOSYLTRANSFERASE, TRANSMEMBRANE, GOLGI APPARATUS, ENZYME MECHANISM, GLYCOPROTEIN, METAL-BINDING, SIGNAL-ANCHOR, ALPHA-1, MEMBRANE, MANGANESE, TRANSFERASE, GLYCOSYLTRANSFERASE GALACTOSYLTRANSFERASE, TRANSFERASE SUBSTRATE SPECIFICITY
1gx9:A (GLY17) to (THR49) BOVINE BETA-LACTOGLOBULIN COMPLEXED WITH RETINOIC ACID, TRIGONAL LATTICE Z | LIPOCALIN, MILK , WHEY TRANSPORT, BOVINE, RETINOL-BINDING ALLERGEN, SIGNAL, 3D-STRUCTURE, RETINOIC ACID-BINDING
1gyg:A (PHE334) to (GLY363) R32 CLOSED FORM OF ALPHA-TOXIN FROM CLOSTRIDIUM PERFRINGENS STRAIN CER89L43 | ZINC PHOSPHOLIPASE C, GANGRENE DETERMINANT, C2 DOMAIN, CA AND MEMBRANE BINDING, HYDROLASE
4zjn:A (LYS173) to (PRO194) CRYSTAL STRUCTURE OF THE BACTERIOPHAGE G20C PORTAL PROTEIN | BACTERIOPHAGE PORTAL PROTEIN, TRANSPORT PROTEIN
3vf5:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE MUTANT I47V WITH NOVEL P1'-LIGANDS GRL-02031 | PROTEASE INHIBITOR,P1'-LIGAND, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3vfb:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE MUTANT N88D WITH NOVEL P1'-LIGANDS GRL-02031 | PROTEASE INHIBITOR,P1'-LIGAND, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2vzo:A (ASP772) to (LEU792) CRYSTAL STRUCTURE OF AMYCOLATOPSIS ORIENTALIS EXO- CHITOSANASE CSXA | GH2, CSXA, PNP-GLUCOSAMINE, GLYCOSIDE HYDROLASE, EXO-BETA-D-GLUCOSAMINIDASE, HYDROLASE
2vzo:B (ASP772) to (LEU792) CRYSTAL STRUCTURE OF AMYCOLATOPSIS ORIENTALIS EXO- CHITOSANASE CSXA | GH2, CSXA, PNP-GLUCOSAMINE, GLYCOSIDE HYDROLASE, EXO-BETA-D-GLUCOSAMINIDASE, HYDROLASE
4zls:B (ARG57) to (GLY78) HIV-1 WILD TYPE PROTEASE WITH GRL-096-13A (A BOC-DERIVATIVE P2-LIGAND, 3,-5-DIMETHYLBIPHENYL P1-LIGAND) | MULTIDRUG-RESISTANT STRAINS, HYDROLASE INHIBITOR COMPLEX, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
2vzt:A (ASP772) to (LEU792) COMPLEX OF AMYCOLATOPSIS ORIENTALIS EXO-CHITOSANASE CSXA E541A WITH PNP-BETA-D-GLUCOSAMINE | GH2, CSXA, PNP-GLUCOSAMINE, GLYCOSIDE HYDROLASE, EXO-BETA-D-GLUCOSAMINIDASE, HYDROLASE
2w2j:A (LEU70) to (GLY101) CRYSTAL STRUCTURE OF THE HUMAN CARBONIC ANHYDRASE RELATED PROTEIN VIII | LYASE, METAL-BINDING
3imn:A (TYR351) to (LEU377) CRYSTAL STRUCTURE OF HEPARIN LYASE I FROM BACTEROIDES THETAIOTAOMICRON | JELLY ROLL, LYASE
4lh8:A (MET1) to (ASP28) TRIAZINE HYDROLASE FROM ARTHOBACTER AURESCENS MODIFIED FOR MAXIMUM EXPRESSION IN E.COLI | AMIDOHYDROLASE, HYDROLASES TRIAZINE HERBICIDES, HYDROLASE
3vkh:A (PHE4637) to (THR4670) X-RAY STRUCTURE OF A FUNCTIONAL FULL-LENGTH DYNEIN MOTOR DOMAIN | AAA+ PROTEIN, MOLECULAR MOTOR, MICROTUBLES, MOTOR PROTEIN
2wb7:B (GLU319) to (THR359) PT26-6P | EXTRA CHROMOSOMAL ELEMENTS, UNKNOWN FUNCTION
3itq:B (ILE143) to (PHE181) CRYSTAL STRUCTURE OF A PROLYL 4-HYDROXYLASE FROM BACILLUS ANTHRACIS | PROLYL 4-HYDROXYLASE, DOUBLE-STRANDED BETA HELIX, ALPHA-KETOGLUTARATE DEPENDENT NON-HEME IRON OXYGENASE, OXIDOREDUCTASE
2hah:A (GLY61) to (ASP94) THE STRUCTURE OF FIV 12S PROTEASE IN COMPLEX WITH TL-3 | RETROVIRAL, PROTEASE, ASPARTYL, FELINE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2hb3:B (ARG57) to (GLY78) WILD-TYPE HIV-1 PROTEASE IN COMPLEX WITH POTENT INHIBITOR GRL06579 | ACTIVE-SITE CAVITY PROTEASE INHIBITOR CATALYTIC ASPARTIC ACID, HYDROLASE
2hc0:A (ARG1057) to (GLY1078) STRUCTURE OF HIV PROTEASE 6X MUTANT IN COMPLEX WITH AB-2. | HIV, PROTEASE, MUTANT, ASPARTYL, HYDROLASE
4lmf:D (THR40) to (SER73) C1S CUB1-EGF-CUB2 | CUB DOMAIN, EGF-LIKE DOMAIN, COMPLEMENT C1S, HYDROLASE
1hvh:A (GLY52) to (GLY78) NONPEPTIDE CYCLIC CYANOGUANIDINES AS HIV PROTEASE INHIBITORS | HYDROLASE, ACID PROTEASE
1hvi:A (ARG57) to (GLY78) INFLUENCE OF STEREOCHEMISTRY ON ACTIVITY AND BINDING MODES FOR C2 SYMMETRY-BASED DIOL INHIBITORS OF HIV-1 PROTEASE | HYDROLASE(ACID PROTEASE)
1hvj:A (ARG57) to (GLY78) INFLUENCE OF STEREOCHEMISTRY ON ACTIVITY AND BINDING MODES FOR C2 SYMMETRY-BASED DIOL INHIBITORS OF HIV-1 PROTEASE | HYDROLASE(ACID PROTEASE)
1hvk:A (ARG57) to (GLY78) INFLUENCE OF STEREOCHEMISTRY ON ACTIVITY AND BINDING MODES FOR C2 SYMMETRY-BASED DIOL INHIBITORS OF HIV-1 PROTEASE | HYDROLASE(ACID PROTEASE)
1hvs:A (ARG57) to (GLY78) STRUCTURAL BASIS OF DRUG RESISTANCE FOR THE V82A MUTANT OF HIV-1 PROTEASE: BACKBONE FLEXIBILITY AND SUBSITE REPACKING | HYDROLASE (ACID PROTEASE)
1hxd:A (GLU110) to (GLN141) CRYSTAL STRUCTURE OF E. COLI BIOTIN REPRESSOR WITH BOUND BIOTIN | LIGASE, REPRESSOR, BIOTIN, DNA-BINDING
2wkz:B (ARG157) to (GLY178) HIV-1 PROTEASE INHIBITORS CONTAINING A TERTIARY ALCOHOL IN THE TRANSITION-STATE MIMIC WITH IMPROVED CELL-BASED ANTIVIRAL ACTIVITY | TRANSITION-STATE MIMIC, INHIBITOR, HYDROLASE
2wl0:A (ARG57) to (GLY78) HIV-1 PROTEASE INHIBITORS CONTAINING A TERTIARY ALCOHOL IN THE TRANSITION-STATE MIMIC WITH IMPROVED CELL-BASED ANTIVIRAL ACTIVITY | TRANSITION-STATE MIMIC, INHIBITOR, HYDROLASE
3vvm:A (ARG10) to (GLY37) CRYSTAL STRUCTURE OF G52A-P55G MUTANT OF L-SERINE-O-ACETYLTRANSFERASE FOUND IN D-CYCLOSERINE BIOSYNTHETIC PATHWAY | D-CYCLOSERINE, ALPHA/BETA HYDROLASE DOMAIN, L-SERINE-O- ACETYLTRANSFERASE, TRANSFERASE
2wly:A (THR36) to (ASN70) CHITINASE A FROM SERRATIA MARCESCENS ATCC990 IN COMPLEX WITH CHITOTRIO-THIAZOLINE. | HYDROLASE, THIAZOLINES, CHITINASE A, GLYCOSIDASE, CHITIN HYDROLYSIS, CHITIN DEGRADATION, POLYSACCHARIDE DEGRADATION, FAMILY 18 CHITINASES, CARBOHYDRATE METABOLISM
2wm0:A (THR36) to (ASN70) CHITINASE A FROM SERRATIA MARCESCENS ATCC990 IN COMPLEX WITH CHITOBIO-THIAZOLINE THIOAMIDE. | HYDROLASE, CHITIN HYDROLYSIS, CHITIN DEGRADATION, POLYSACCHARIDE DEGRADATION, CARBOHYDRATE METABOLISM
1i2m:D (LEU36) to (PRO66) RAN-RCC1-SO4 COMPLEX | BETA-PROPELLER, G FOLD OR GTPASE FOLD, CELL CYCLE
2hs2:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF M46L MUTANT OF HIV-1 PROTEASE COMPLEXED WITH TMC114 (DARUNAVIR) | ASPARTIC PROTEASE ACTIVE SITE SURFACE BINDING SITE, HYDROLASE
1u2x:A (ASP177) to (GLU215) CRYSTAL STRUCTURE OF A HYPOTHETICAL ADP-DEPENDENT PHOSPHOFRUCTOKINASE FROM PYROCOCCUS HORIKOSHII OT3 | ADP-PFK, PYROCOCCUS, MIDWEST CENTER FOR STRUCTURAL GENOMICS, APC5054, PROTEIN STRUCTURE INITIATIVE, PSI, MCSG, TRANSFERASE
1u2x:B (PRO178) to (GLU215) CRYSTAL STRUCTURE OF A HYPOTHETICAL ADP-DEPENDENT PHOSPHOFRUCTOKINASE FROM PYROCOCCUS HORIKOSHII OT3 | ADP-PFK, PYROCOCCUS, MIDWEST CENTER FOR STRUCTURAL GENOMICS, APC5054, PROTEIN STRUCTURE INITIATIVE, PSI, MCSG, TRANSFERASE
1uai:A (TYR189) to (THR222) CRYSTAL STRUCTURE OF THE ALGINATE LYASE FROM CORYNEBACTERIUM SP. | JELLYROLL BETA-SANDWICH, LYASE
4m00:A (ASN466) to (THR492) CRYSTAL STRUCTURE OF THE LIGAND BINDING REGION OF STAPHYLOCOCCAL ADHESION SRAP | ALL BETA, ADHESION, CARBOHYDRATE/SUGAR BINDING, CELL ADHESION
1ufg:A (ASP61) to (ALA91) SOLUTION STRUCTURE OF IMMUNOGLOBULIN LIKE DOMAIN OF MOUSE NUCLEAR LAMIN | IMMUNOGLOBULIN LIKE FOLD, NUCLEAR LAMIN, STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, STRUCTURAL PROTEIN
2i4u:B (ARG257) to (GLY278) HIV-1 PROTEASE WITH TMC-126 | PROTEIN INHIBITOR COMPLEX, HYDROLASE
2i4v:B (ARG257) to (GLY278) HIV-1 PROTEASE I84V, L90M WITH TMC126 | HIV-1 PROTEIN INHIBITOR MUTANT, HYDROLASE
2i4w:B (ARG257) to (GLY278) HIV-1 PROTEASE WT WITH GS-8374 | HIV-1 PROTEASE INHIBITOR, HYDROLASE
2i4x:B (ARG257) to (GLY278) HIV-1 PROTEASE I84V, L90M WITH GS-8374 | HIV-1 PROTEASE I84VL90M INHIBITOR, HYDROLASE
2wxf:A (ASP430) to (PHE485) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH PIK-39. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
2wxg:A (ASP430) to (PHE485) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH SW13. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
2wxh:A (ASP430) to (PHE485) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH SW14. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER, NUCLEOTIDE-BINDING
1uoj:D (GLY23) to (ILE69) CRYSTAL STRUCTURE OF PSEUDOMONAS AERUGINOSA LECTIN 1 IN THE CALCIUM-FREE STATE | SUGAR BINDING PROTEIN, GALACTOSE BINDING
2wxq:A (ASP430) to (PHE485) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH AS15. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
2idw:B (ARG157) to (GLY178) CRYSTAL STRUCTURE ANALYSIS OF HIV-1 PROTEASE MUTANT V82A WITH A POTENT NON-PEPTIDE INHIBITOR (UIC-94017) | HIV-1 PROTEASE, MUTANT, DIMER, INHIBITOR, UIC-94017, HYDROLASE
2ieo:B (ARG157) to (GLY178) CRYSTAL STRUCTURE ANALYSIS OF HIV-1 PROTEASE MUTANT I84V WITH A POTENT NON-PEPTIDE INHIBITOR (UIC-94017) | HIV-1 PROTEASE, MUTANT, I84V, DIMER, INHIBITOR, UIC-94017, TMC114, DARUNAVIR, HYDROLASE
2wzp:A (ASN52) to (LYS77) STRUCTURES OF LACTOCOCCAL PHAGE P2 BASEPLATE SHED LIGHT ON A NOVEL MECHANISM OF HOST ATTACHMENT AND ACTIVATION IN SIPHOVIRIDAE | BASEPLATE, VIRAL PROTEIN
2wzp:B (ASN52) to (LYS77) STRUCTURES OF LACTOCOCCAL PHAGE P2 BASEPLATE SHED LIGHT ON A NOVEL MECHANISM OF HOST ATTACHMENT AND ACTIVATION IN SIPHOVIRIDAE | BASEPLATE, VIRAL PROTEIN
2wzp:C (ASN52) to (LYS77) STRUCTURES OF LACTOCOCCAL PHAGE P2 BASEPLATE SHED LIGHT ON A NOVEL MECHANISM OF HOST ATTACHMENT AND ACTIVATION IN SIPHOVIRIDAE | BASEPLATE, VIRAL PROTEIN
2wzp:G (ASN52) to (LYS77) STRUCTURES OF LACTOCOCCAL PHAGE P2 BASEPLATE SHED LIGHT ON A NOVEL MECHANISM OF HOST ATTACHMENT AND ACTIVATION IN SIPHOVIRIDAE | BASEPLATE, VIRAL PROTEIN
2wzp:H (ASN52) to (LYS77) STRUCTURES OF LACTOCOCCAL PHAGE P2 BASEPLATE SHED LIGHT ON A NOVEL MECHANISM OF HOST ATTACHMENT AND ACTIVATION IN SIPHOVIRIDAE | BASEPLATE, VIRAL PROTEIN
2wzp:I (ASN52) to (LYS77) STRUCTURES OF LACTOCOCCAL PHAGE P2 BASEPLATE SHED LIGHT ON A NOVEL MECHANISM OF HOST ATTACHMENT AND ACTIVATION IN SIPHOVIRIDAE | BASEPLATE, VIRAL PROTEIN
4mb8:C (GLY22) to (THR50) EVOLUTIONARY HISTORY AND METABOLIC INSIGHTS OF ANCIENT MAMMALIAN URICASES | URIC ACID OXIDASE, LYSOZOME, OXIDOREDUCTASE
1izh:B (ARG57) to (GLY78) INHIBITOR OF HIV PROTEASE WITH UNUSUAL BINDING MODE POTENTLY INHIBITING MULTI-RESISTANT PROTEASE MUTANTS | HIV-1 PROTEINASE, POTENT INHIBITOR, SUBSITE BINDING, HYDROLASE
5ah7:B (ARG157) to (GLY178) DISUBSTITUTED BIS-THF MOIETIES AS NEW P2 LIGANDS IN NON-PEPTIDAL HIV-1 PROTEASE INHIBITORS (II) | HYDROLASE, RATIONAL DRUG DESIGN, BIS-THF BIS-DIOL
5ah8:A (GLY52) to (GLY78) DISUBSTITUTED BIS-THF MOIETIES AS NEW P2 LIGANDS IN NON-PEPTIDAL HIV-1 PROTEASE INHIBITORS (II) | HYDROLASE, RATIONAL DRUG DESIGN, BIS-THF BIS-DIOL
5ah9:B (ARG157) to (GLY178) DISUBSTITUTED BIS-THF MOIETIES AS NEW P2 LIGANDS IN NON- PEPTIDAL HIV-1 PROTEASE INHIBITORS (II) | HYDROLASE, INHIBITOR, RATIONAL DRUG DESIGN, BIS-THF BIS-DIOL
5aha:A (GLY52) to (GLY78) DISUBSTITUTED BIS-THF MOIETIES AS NEW P2 LIGANDS IN NON- PEPTIDAL HIV-1 PROTEASE INHIBITORS (II) | HYDROLASE, INHIBITOR, RATIONAL DRUG DESIGN, BIS-THF BIS-DIOL
5ahb:A (ARG57) to (GLY78) DISUBSTITUTED BIS-THF MOIETIES AS NEW P2 LIGANDS IN NON-PEPTIDAL HIV-1 PROTEASE INHIBITORS (II) | HYDROLASE, INHIBITOR, RATIONAL DRUG DESIGN, BIS-THF BIS-DIOL
2iou:A (ALA73) to (ALA102) MAJOR TROPISM DETERMINANT P1 (MTD-P1) VARIANT COMPLEXED WITH BORDETELLA BROCHISEPTICA VIRULENCE FACTOR PERTACTIN EXTRACELLULAR DOMAIN (PRN-E). | MTD; PRN; PERTACTIN, VIRAL PROTEIN-MEMBRANE PROTEIN COMPLEX
2iou:C (ALA73) to (ALA102) MAJOR TROPISM DETERMINANT P1 (MTD-P1) VARIANT COMPLEXED WITH BORDETELLA BROCHISEPTICA VIRULENCE FACTOR PERTACTIN EXTRACELLULAR DOMAIN (PRN-E). | MTD; PRN; PERTACTIN, VIRAL PROTEIN-MEMBRANE PROTEIN COMPLEX
2iou:E (ALA73) to (ALA102) MAJOR TROPISM DETERMINANT P1 (MTD-P1) VARIANT COMPLEXED WITH BORDETELLA BROCHISEPTICA VIRULENCE FACTOR PERTACTIN EXTRACELLULAR DOMAIN (PRN-E). | MTD; PRN; PERTACTIN, VIRAL PROTEIN-MEMBRANE PROTEIN COMPLEX
2x53:A (ASN52) to (LYS77) STRUCTURE OF THE PHAGE P2 BASEPLATE IN ITS ACTIVATED CONFORMATION WITH SR | BASEPLATE, VIRAL PROTEIN
2x53:B (ASN52) to (ALA75) STRUCTURE OF THE PHAGE P2 BASEPLATE IN ITS ACTIVATED CONFORMATION WITH SR | BASEPLATE, VIRAL PROTEIN
2x53:C (ASN52) to (LYS77) STRUCTURE OF THE PHAGE P2 BASEPLATE IN ITS ACTIVATED CONFORMATION WITH SR | BASEPLATE, VIRAL PROTEIN
2x53:D (ASN52) to (LYS77) STRUCTURE OF THE PHAGE P2 BASEPLATE IN ITS ACTIVATED CONFORMATION WITH SR | BASEPLATE, VIRAL PROTEIN
2x53:E (ASN52) to (ALA75) STRUCTURE OF THE PHAGE P2 BASEPLATE IN ITS ACTIVATED CONFORMATION WITH SR | BASEPLATE, VIRAL PROTEIN
2x53:G (ASN52) to (LYS77) STRUCTURE OF THE PHAGE P2 BASEPLATE IN ITS ACTIVATED CONFORMATION WITH SR | BASEPLATE, VIRAL PROTEIN
2x53:H (ASN52) to (ALA75) STRUCTURE OF THE PHAGE P2 BASEPLATE IN ITS ACTIVATED CONFORMATION WITH SR | BASEPLATE, VIRAL PROTEIN
2x53:J (ASN52) to (LYS77) STRUCTURE OF THE PHAGE P2 BASEPLATE IN ITS ACTIVATED CONFORMATION WITH SR | BASEPLATE, VIRAL PROTEIN
2x53:K (ASN52) to (ALA75) STRUCTURE OF THE PHAGE P2 BASEPLATE IN ITS ACTIVATED CONFORMATION WITH SR | BASEPLATE, VIRAL PROTEIN
2x53:M (ASN52) to (LYS77) STRUCTURE OF THE PHAGE P2 BASEPLATE IN ITS ACTIVATED CONFORMATION WITH SR | BASEPLATE, VIRAL PROTEIN
2x53:N (ASN52) to (ALA75) STRUCTURE OF THE PHAGE P2 BASEPLATE IN ITS ACTIVATED CONFORMATION WITH SR | BASEPLATE, VIRAL PROTEIN
2x53:P (ASN52) to (LYS77) STRUCTURE OF THE PHAGE P2 BASEPLATE IN ITS ACTIVATED CONFORMATION WITH SR | BASEPLATE, VIRAL PROTEIN
2x53:Q (ASN52) to (ALA75) STRUCTURE OF THE PHAGE P2 BASEPLATE IN ITS ACTIVATED CONFORMATION WITH SR | BASEPLATE, VIRAL PROTEIN
3wod:D (TYR132) to (THR154) RNA POLYMERASE-GP39 COMPLEX | RNA POLYMERASE, TRANSCRIPTION, TRANSFERASE-TRANSCRIPTION COMPLEX
1vav:A (TYR193) to (SER221) CRYSTAL STRUCTURE OF ALGINATE LYASE PA1167 FROM PSEUDOMONAS AERUGINOSA AT 2.0 A RESOLUTION | BETA-SANDWICH, STRUCTURAL GENOMICS, LYASE
1vav:B (TYR193) to (SER221) CRYSTAL STRUCTURE OF ALGINATE LYASE PA1167 FROM PSEUDOMONAS AERUGINOSA AT 2.0 A RESOLUTION | BETA-SANDWICH, STRUCTURAL GENOMICS, LYASE
5anb:E (VAL79) to (VAL101) MECHANISM OF EIF6 RELEASE FROM THE NASCENT 60S RIBOSOMAL SUBUNIT | TRANSLATION, RIBOSOMOPATHY, GTPASE, RIBOSOME BIOGENESIS
5anc:E (LYS72) to (VAL101) MECHANISM OF EIF6 RELEASE FROM THE NASCENT 60S RIBOSOMAL SUBUNIT | TRANSLATION, RIBOSOMOPATHY, EFL1, GTPASE, RIBOSOME BIOGENESIS
1vcd:A (ARG54) to (GLY85) CRYSTAL STRUCTURE OF A T.THERMOPHILUS HB8 AP6A HYDROLASE NDX1 | NUDIX PROTEIN, DIADENOSINE POLYPHOSPHATE, AP6A, THERMUS THERMOPHILUS HB8, HYDROLASE, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, STRUCTURAL GENOMICS
3wp4:A (ARG77) to (SER105) THE CRYSTAL STRUCTURE OF NATIVE CDBFV FROM NEOCALLIMASTIX PATRICIARUM | XYLANASE, REGULATORY N-TERMINAL REGION, DISULFIDE BOND, INDUSTRIAL ENZYME, BETA-JELLYROLL FOLD, HYDROLASE
3wp6:A (ARG77) to (SER105) THE COMPLEX STRUCTURE OF CDBFV E109A WITH XYLOTRIOSE | XYLANASE, REGULATORY N-TERMINAL REGION, DISULFIDE BOND, INDUSTRIAL ENZYME, BETA-JELLYROLL FOLD, HYDROLASE
1jld:A (LYS57) to (GLY78) POTENT HIV PROTEASE INHIBITORS CONTAINING A NOVEL (HYDROXYETHYL)AMIDE ISOSTERE | POLYPROTEIN, HIV-2 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX, AIDS
1jmu:B (TRP333) to (VAL368) CRYSTAL STRUCTURE OF THE REOVIRUS MU1/SIGMA3 COMPLEX | PROTEIN-PROTEIN COMPLEX, JELLY ROLL, ZINC FINGER, VIRAL PROTEIN
1jmu:D (TRP333) to (VAL368) CRYSTAL STRUCTURE OF THE REOVIRUS MU1/SIGMA3 COMPLEX | PROTEIN-PROTEIN COMPLEX, JELLY ROLL, ZINC FINGER, VIRAL PROTEIN
1jmu:F (TRP333) to (VAL368) CRYSTAL STRUCTURE OF THE REOVIRUS MU1/SIGMA3 COMPLEX | PROTEIN-PROTEIN COMPLEX, JELLY ROLL, ZINC FINGER, VIRAL PROTEIN
4mwf:A (ALA88) to (THR110) STRUCTURE OF HEPATITIS C VIRUS ENVELOPE GLYCOPROTEIN E2 CORE BOUND TO BROADLY NEUTRALIZING ANTIBODY AR3C | IMMUNOGLOBULIN FOLD, HCV E2, IMMUNE SYSTEM
5ayj:C (MET9) to (GLY55) HYPERTHERMOSTABLE MUTANT OF BACILLUS SP. TB-90 URATE OXIDASE - R298C | DISULFIDE BOND, THERMOSTABILITY, PROTEIN ENGINEERING, OXIDASE, SUBUNIT-SUBUNIT INTERACTION, OXIDOREDUCTASE
1w5w:B (ARG57) to (GLY78) HIV-1 PROTEASE IN COMPLEX WITH FLUORO SUBSTITUTED DIOL- BASED C2-SYMMETRIC INHIBITOR | HYDROLASE/HYDROLASE INHIBITOR, HYDROLASE, DIMER, PROTEIN-INHIBITOR COMPLEX
1w5x:B (ARG57) to (GLY78) HIV-1 PROTEASE IN COMPLEX WITH FLUORO SUBSTITUTED DIOL- BASED C2-SYMMETRIC INHIBITOR | HYDROLASE/HYDROLASE INHIBITOR, HYDROLASE, DIMER, PROTEIN-INHIBITOR COMPLEX
4n75:B (GLY781) to (TRP810) STRUCTURAL BASIS OF BAMA-MEDIATE OUTER MEMBRANE PROTEIN BIOGENESIS | BARREL, OUTER MEMBRANE PROTEIN BIOGENESIS, MEMBRANE PROTEIN, OMP85, YAET
1w6h:A (LYS68) to (ASP89) NOVEL PLASMEPSIN II-INHIBITOR COMPLEX | MALARIA, DRUG, ASPARTIC PROTEASE, PLASMEPSIN, HYDROLASE, GLYCOPROTEIN
2jg8:A (PHE95) to (GLU119) CRYSTALLOGRAPHIC STRUCTURE OF HUMAN C1Q GLOBULAR HEADS COMPLEXED TO PHOSPHATIDYL-SERINE | POLYMORPHISM, GLYCOPROTEIN, PHAGOCYTOSIS, DISEASE MUTATION, COMPLEMENT PATHWAY, IMMUNE SYSTEM, CELL SURFACE MOLECULE, PYRROLIDONE CARBOXYLIC ACID, HYDROXYLATION, INNATE IMMUNITY, IMMUNE RESPONSE, COLLAGEN, TOLERANCE, APOPOTOSIS, COMPLEMENT
2jg8:D (GLN90) to (GLU119) CRYSTALLOGRAPHIC STRUCTURE OF HUMAN C1Q GLOBULAR HEADS COMPLEXED TO PHOSPHATIDYL-SERINE | POLYMORPHISM, GLYCOPROTEIN, PHAGOCYTOSIS, DISEASE MUTATION, COMPLEMENT PATHWAY, IMMUNE SYSTEM, CELL SURFACE MOLECULE, PYRROLIDONE CARBOXYLIC ACID, HYDROXYLATION, INNATE IMMUNITY, IMMUNE RESPONSE, COLLAGEN, TOLERANCE, APOPOTOSIS, COMPLEMENT
1w8l:A (ILE89) to (GLU120) ENZYMATIC AND STRUCTURAL CHARACTERIZATION OF NON PEPTIDE LIGAND CYCLOPHILIN COMPLEXES | 3D-STRUCTURE, COMPLEX (ISOMERASE/IMMUNOSUPPRESSANT), NON- PEPTIDE LIGAND, ISOMERASE, MULTIGENE FAMILY, ROTAMASE
2jit:A (GLU711) to (PRO733) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN T790M MUTATION | EGFR, T790M, KINASE, RECEPTOR, CELL CYCLE, PHOSPHORYLATION, DISEASE MUTATION, NUCLEOTIDE-BINDING, TYROSINE-PROTEIN KINASE, ANTI-ONCOGENE, EPIDERMAL GROWTH FACTOR, ATP-BINDING, TRANSFERASE
1k1t:B (ARG157) to (GLY178) COMBINING MUTATIONS IN HIV-1 PROTEASE TO UNDERSTAND MECHANISMS OF RESISTANCE | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1k1u:A (ARG57) to (GLY78) COMBINING MUTATIONS IN HIV-1 PROTEASE TO UNDERSTAND MECHANISMS OF RESISTANCE | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1k1u:B (ARG157) to (GLY178) COMBINING MUTATIONS IN HIV-1 PROTEASE TO UNDERSTAND MECHANISMS OF RESISTANCE | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5bry:B (ARG57) to (GLY78) HIV-1 WILD TYPE PROTEASE WITH GRL-011-11A (A METHYLAMINE BIS- TETRAHYDROFURAN P2-LIGAND, SULFONAMIDE ISOSTERE DERIVATE) | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1k2b:B (ARG57) to (GLY78) COMBINING MUTATIONS IN HIV-1 PROTEASE TO UNDERSTAND MECHANISMS OF RESISTANCE | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1k2c:B (ARG57) to (GLY78) COMBINING MUTATIONS IN HIV-1 PROTEASE TO UNDERSTAND MECHANISMS OF RESISTANCE | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5bs4:B (ARG57) to (GLY78) HIV-1 WILD TYPE PROTEASE WITH GRL-047-11A (A METHYLAMINE BIS- TETRAHYDROFURAN P2-LIGAND, 4-AMINO SULFONAMIDE DERIVATIVE) | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1wbk:B (ARG57) to (GLY78) HIV-1 PROTEASE IN COMPLEX WITH ASYMMETRIC INHIBITOR, BEA568 | HYDROLASE/INHIBITOR, HYDROLASE/INHIBITOR COMPLEX, AIDS, ASPARTYL PROTEASE, DIMER, HYDROLASE, HYDROLASE/HYDROLASE INHIBITOR, PROTEIN-INHIBITOR COMPLEX
1wbm:B (ARG57) to (GLY78) HIV-1 PROTEASE IN COMPLEX WITH SYMMETRIC INHIBITOR, BEA450 | HYDROLASE/INHIBITOR, HYDROLASE/INHIBITOR COMPLEX, AIDS, ASPARTYL PROTEASE, DIMER, HYDROLASE, HYDROLASE/HYDROLASE INHIBITOR, PROTEIN-INHIBITOR COMPLEX
2xye:A (ARG57) to (GLY78) HIV-1 INHIBITORS WITH A TERTIARY-ALCOHOL-CONTAINING TRANSITION-STATE MIMIC AND VARIOUS P2 AND P1 PRIME SUBSTITUENTS | HYDROLASE, AIDS
2xye:B (ARG157) to (GLY178) HIV-1 INHIBITORS WITH A TERTIARY-ALCOHOL-CONTAINING TRANSITION-STATE MIMIC AND VARIOUS P2 AND P1 PRIME SUBSTITUENTS | HYDROLASE, AIDS
2xyf:A (ARG57) to (GLY78) HIV-1 INHIBITORS WITH A TERTIARY-ALCOHOL-CONTAINING TRANSITION-STATE MIMIC AND VARIOUS P2 AND P1 PRIME SUBSTITUENTS | HYDROLASE, AIDS
1k6c:A (ARG57) to (GLY78) LACK OF SYNERGY FOR INHIBITORS TARGETING A MULTI-DRUG RESISTANT HIV-1 PROTEASE | INDINAVIR, INHIBITOR RECOGNITION, DRUG RESISTANCE, HIV-1 PROTEASE, HYDROLASE
1k6c:B (ARG57) to (GLY78) LACK OF SYNERGY FOR INHIBITORS TARGETING A MULTI-DRUG RESISTANT HIV-1 PROTEASE | INDINAVIR, INHIBITOR RECOGNITION, DRUG RESISTANCE, HIV-1 PROTEASE, HYDROLASE
1k6p:A (ARG57) to (GLY78) LACK OF SYNERGY FOR INHIBITORS TARGETING A MULTI-DRUG RESISTANT HIV-1 PROTEASE | INDINAVIR, INHIBITOR RECOGNITION, DRUG RESISTANCE, HIV-1 PROTEASE, HYDROLASE
1k6t:A (ARG57) to (GLY78) LACK OF SYNERGY FOR INHIBITORS TARGETING A MULTI-DRUG RESISTANT HIV-1 PROTEASE | INDINAVIR, INHIBITOR RECOGNITION, HIV-1 PROTEASE, DRUG RESISTANCE, HYDROLASE
1k6t:B (ARG57) to (GLY78) LACK OF SYNERGY FOR INHIBITORS TARGETING A MULTI-DRUG RESISTANT HIV-1 PROTEASE | INDINAVIR, INHIBITOR RECOGNITION, HIV-1 PROTEASE, DRUG RESISTANCE, HYDROLASE
1k6v:A (ARG57) to (GLY78) LACK OF SYNERGY FOR INHIBITORS TARGETING A MULTI-DRUG RESISTANT HIV-1 PROTEASE | INDINAVIR, INHIBITOR RECOGNITION, DRUG RESISTANCE, HIV-1 PROTEASE, HYDROLASE
1k6v:B (ARG57) to (GLY78) LACK OF SYNERGY FOR INHIBITORS TARGETING A MULTI-DRUG RESISTANT HIV-1 PROTEASE | INDINAVIR, INHIBITOR RECOGNITION, DRUG RESISTANCE, HIV-1 PROTEASE, HYDROLASE
4nfx:B (VAL6) to (ALA40) STRUCTURE AND ATYPICAL HYDROLYSIS MECHANISM OF THE NUDIX HYDROLASE ORF153 (YMFB) FROM ESCHERICHIA COLI | NUDIX HYDROLASE; YMFB; NUCLEOSIDE TRIPHOSPHATASE; METAL IONS-BASED CATALYSIS, NUDIX MOTIF, PHOSPHATASE, HYDROLASE
4nfx:C (VAL6) to (ALA40) STRUCTURE AND ATYPICAL HYDROLYSIS MECHANISM OF THE NUDIX HYDROLASE ORF153 (YMFB) FROM ESCHERICHIA COLI | NUDIX HYDROLASE; YMFB; NUCLEOSIDE TRIPHOSPHATASE; METAL IONS-BASED CATALYSIS, NUDIX MOTIF, PHOSPHATASE, HYDROLASE
1wgb:A (PRO113) to (ARG143) CRYSTAL STRUCTURE OF A PROBABLE FLAVOPROTEIN FROM THERMUS THERMOPHILUS HB8 | FLAVOPROTEIN, HB8, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, STRUCTURAL GENOMICS, OXIDOREDUCTASE
2kpw:A (GLN35) to (ALA65) NMR SOLUTION STRUCTURE OF LAMIN-B1 PROTEIN FROM HOMO SAPIENS: NORTHEAST STRUCTURAL GENOMICS CONSORTIUM MEGA TARGET, HR5546A (439-549) | PSI-2, NESG, HR5546A, LAMIN-B1, GFT, ACETYLATION, CHROMOSOMAL REARRANGEMENT, COILED COIL, INTERMEDIATE FILAMENT, LEUKODYSTROPHY, LIPOPROTEIN, MEMBRANE, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, PRENYLATION, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM
4nli:A (GLY17) to (THR49) CRYSTAL STRUCTURE OF SHEEP BETA-LACTOGLOBULIN (SPACE GROUP P3121) | LIPOCALIN, TRANSPORT, MILK, TRANSPORT PROTEIN
4nlj:B (GLY17) to (THR49) CRYSTAL STRUCTURE OF SHEEP BETA-LACTOGLOBULIN (SPACE GROUP P1) | LIPOCALIN, TRANSPORT, MILK, TRANSPORT PROTEIN
2kzb:A (SER283) to (ILE314) SOLUTION STRUCTURE OF ALPHA-MANNOSIDASE BINDING DOMAIN OF ATG19 | SELECTIVE AUTOPHAGY, ATG19, ALPHA-MANNOSIDASE, PROTEIN TRANSPORT
3zps:B (ARG157) to (GLY178) DESIGN AND SYNTHESIS OF P1-P3 MACROCYCLIC TERTIARY ALCOHOL COMPRISING HIV-1 PROTEASE INHIBITORS | HYDROLASE, PROTEASE INHIBITOR, RATIONAL DRUG DESIGN,
3zpt:B (ARG157) to (GLY178) DESIGN AND SYNTHESIS OF P1-P3 MACROCYCLIC TERTIARY ALCOHOL COMPRISING HIV-1 PROTEASE INHIBITORS | HYDROLASE, RATIONAL DRUG DESIGN, MACROCYCLIC TERTIARY ALCOHOL
3zpu:B (ARG157) to (GLY178) DESIGN AND SYNTHESIS OF P1-P3 MACROCYCLIC TERTIARY ALCOHOL COMPRISING HIV-1 PROTEASE INHIBITORS | HYDROLASE, PROTEASE INHIBITOR, RATIONAL DRUG DESIGN
3zpy:A (TYR414) to (ASN446) CRYSTAL STRUCTURE OF THE MARINE PL7 ALGINATE LYASE ALYA1 FROM ZOBELLIA GALACTANIVORANS | LYASE, POLYSACCHARIDASES, MARINE BACTERIAL ENZYME
3zpy:B (TYR414) to (ASN446) CRYSTAL STRUCTURE OF THE MARINE PL7 ALGINATE LYASE ALYA1 FROM ZOBELLIA GALACTANIVORANS | LYASE, POLYSACCHARIDASES, MARINE BACTERIAL ENZYME
1kj7:A (ARG57) to (GLY78) SUBSTRATE SHAPE DETERMINES SPECIFICITY OF RECOGNITION RECOGNITION FOR HIV-1 PROTEASE: ANALYSIS OF CRYSTAL STRUCTURES OF SIX SUBSTRATE COMPLEXES | P2-NUCLEOCAPSID, SUBSTRATE RECOGNITION, HYDROLASE
1kjh:A (ARG57) to (GLY78) SUBSTRATE SHAPE DETERMINES SPECIFICITY OF RECOGNITION RECOGNITION FOR HIV-1 PROTEASE: ANALYSIS OF CRYSTAL STRUCTURES OF SIX SUBSTRATE COMPLEXES | RNASE H, INTEGRASE, SUBSTRATE RECOGNITION, HYDROLASE
1kmo:A (ASP698) to (PHE741) CRYSTAL STRUCTURE OF THE OUTER MEMBRANE TRANSPORTER FECA | MEMBRANE PROTEIN, IRON TRANSPORTER, TONB-DEPENDENT RECEPTOR, SIDEROPHORE
1kmp:A (LEU699) to (PHE741) CRYSTAL STRUCTURE OF THE OUTER MEMBRANE TRANSPORTER FECA COMPLEXED WITH FERRIC CITRATE | INTEGRAL OUTER MEMBRANE PROTEIN, TONB-DEPENDENT RECEPTOR, SIDEROPHORE, IRON, MEMBRANE PROTEIN
4nwv:C (LYS273) to (LEU304) CRYSTAL STRUCTURE OF ORSAY VIRUS-LIKE PARTICLE | BETA BARREL, VIRUS
4nww:C (LYS273) to (LEU304) CRYSTAL STRUCTURE OF AN N-TERMINALLY TRUNCATED CAPSID PROTEIN MUTANT OF ORSAY VIRUS | BETA BARREL, VIRUS
3jcm:W (ASN50) to (ARG74) CRYO-EM STRUCTURE OF THE SPLICEOSOMAL U4/U6.U5 TRI-SNRNP | U4/U6.U5 TRI-SNRNP, PRE-MRNA, TRANSCRIPTION
3jcm:X (VAL38) to (ARG64) CRYO-EM STRUCTURE OF THE SPLICEOSOMAL U4/U6.U5 TRI-SNRNP | U4/U6.U5 TRI-SNRNP, PRE-MRNA, TRANSCRIPTION
3jcm:Z (ASN50) to (ARG74) CRYO-EM STRUCTURE OF THE SPLICEOSOMAL U4/U6.U5 TRI-SNRNP | U4/U6.U5 TRI-SNRNP, PRE-MRNA, TRANSCRIPTION
3jcm:a (VAL38) to (ARG64) CRYO-EM STRUCTURE OF THE SPLICEOSOMAL U4/U6.U5 TRI-SNRNP | U4/U6.U5 TRI-SNRNP, PRE-MRNA, TRANSCRIPTION
1kwi:A (THR72) to (ASP114) CRYSTAL STRUCTURE ANALYSIS OF THE CATHELICIDIN MOTIF OF PROTEGRINS | PROTEGRIN, CATHELICIDIN MOTIF, DISULFIDE, MAD, SELENOCYSTINE, ANTIMICROBIAL PROTEIN
3zyp:A (GLY188) to (ALA211) CELLULOSE INDUCED PROTEIN, CIP1 | METAL BINDING PROTEIN, CALCIUM-BINDING, CBM-CONTAINING, BETA SANDWICH JELLY ROLL, CARBOHYDRATE-BINDING
2nmz:B (ARG157) to (GLY178) CRYSTAL STRUCTURE ANALYSIS OF HIV-1 PROTEASE MUTANT V82A WITH A INHIBITOR SAQUINAVIR | HIV-1 PROTEASE, MUTANT, V82A, DIMER, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5c9b:B (ASN176) to (LEU201) CRYSTAL STRUCTURE OF A RETROPEPSIN-LIKE ASPARTIC PROTEASE FROM RICKETTSIA CONORII | PEPSIN, APRICK, HYDROLASE
5c9d:A (ALA179) to (LEU201) CRYSTAL STRUCTURE OF A RETROPEPSIN-LIKE ASPARTIC PROTEASE FROM RICKETTSIA CONORII | PEPSIN, APRICK, HYDROLASE
5c9f:B (ALA179) to (LEU201) CRYSTAL STRUCTURE OF A RETROPEPSIN-LIKE ASPARTIC PROTEASE FROM RICKETTSIA CONORII | PEPSIN, APRICK, HYDROLASE
5c9f:C (ALA179) to (LEU201) CRYSTAL STRUCTURE OF A RETROPEPSIN-LIKE ASPARTIC PROTEASE FROM RICKETTSIA CONORII | PEPSIN, APRICK, HYDROLASE
2nnk:B (ARG157) to (GLY178) CRYSTAL STRUCTURE ANALYSIS OF HIV-1 PROTEASE MUTANT I84V WITH A INHIBITOR SAQUINAVIR | HIV-1 PROTEASE, MUTANT, I84V, DIMER, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2nnp:B (ARG157) to (GLY178) CRYSTAL STRUCTURE ANALYSIS OF HIV-1 PROTEASE MUTANT I84V WITH A INHIBITOR SAQUINAVIR | HIV-1 PROTEASE, MUTANT, I84V, DIMER, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3zzu:A (GLY333) to (SER371) CRYSTAL STRUCTURE OF STAPHYLOCOCCUS AUREUS ELONGATION FACTOR G WITH MUTATIONS M16I AND F88L | TRANSLATION
5cas:A (GLU711) to (PRO733) EGFR KINASE DOMAIN MUTANT "TMLR" WITH COMPOUND 41A | PROTEIN KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2nq3:A (MET111) to (GLU145) CRYSTAL STRUCTURE OF THE C2 DOMAIN OF HUMAN ITCHY HOMOLOG E3 UBIQUITIN PROTEIN LIGASE | C2 DOMAIN, LIGASE, UBL CONJUGATION PATHWAY, STRUCTURAL GENOMICS CONSORTIUM, SGC
1l2l:A (CYS177) to (GLY203) CRYSTAL STRUCTURE OF ADP-DEPENDENT GLUCOKINASE FROM A PYROCOCCUS HORIKOSHII | ADP GLUCOKINASE APO, TRANSFERASE
3jvy:B (ARG157) to (GLY178) HIV-1 PROTEASE MUTANT G86A WITH DARUNAVIR | HIV-1 PROTEASE, MUTANT G86A, INHIBITOR, DARUNAVIR, AIDS, ASPARTYL PROTEASE, HYDROLASE, METAL-BINDING
3jw2:B (ARG157) to (GLY178) HIV-1 PROTEASE MUTANT G86S WITH DARUNAVIR | HIV-1 PROTEASE, MUTANT G86S, INHIBITOR, DARUNAVIR, AIDS, ASPARTYL PROTEASE, METAL-BINDING, HYDROLASE
4obh:A (GLY52) to (GLY78) CRYSTAL STRUCTURE OF INACTIVE HIV-1 PROTEASE IN COMPLEX WITH THE P1-P6 SUBSTRATE VARIANT (L449F) | CO-EVOLUTION, RESISTANCE, HYDROLASE
4obh:C (GLY52) to (GLY78) CRYSTAL STRUCTURE OF INACTIVE HIV-1 PROTEASE IN COMPLEX WITH THE P1-P6 SUBSTRATE VARIANT (L449F) | CO-EVOLUTION, RESISTANCE, HYDROLASE
4obh:D (ARG57) to (GLY78) CRYSTAL STRUCTURE OF INACTIVE HIV-1 PROTEASE IN COMPLEX WITH THE P1-P6 SUBSTRATE VARIANT (L449F) | CO-EVOLUTION, RESISTANCE, HYDROLASE
2nxl:B (ARG57) to (GLY78) STRUCTURE OF HIV-1 PROTEASE D25N COMPLEXED WITH THE RT-RH ANALOGUE PEPTIDE GLY-ALA-GLU-VAL-PHE*TYR-VAL-ASP-GLY-ALA | PEPTIDE DESIGN; MOLECULAR DYNAMICS; HIV PROTEASE; SUBSTRATE RECOGNITION; CALORIMETRY, HYDROLASE/HYDROLASE SUBSTRATE COMPLEX
2nxm:A (ARG57) to (GLY78) STRUCTURE OF HIV-1 PROTEASE D25N COMPLEXED WITH THE RT-RH ANALOGUE PEPTIDE GLY-ALA-GLN-THR-PHE*TYR-VAL-ASP-GLY-ALA | PEPTIDE DESIGN; MOLECULAR DYNAMICS; HIV PROTEASE; SUBSTRATE RECOGNITION; CALORIMETRY, HYDROLASE/HYDROLASE SUBSTRATE COMPLEX
2nzh:B (VAL64) to (GLY87) CRYSTAL STRUCTURE OF A SECRETION CHAPERONE CSAA FROM BACILLUS SUBTILIS IN THE SPACE GROUP P 4 21 2 | BETA BARREL, OLIGONUCLEOTIDE/OLIGOSACCHARIDE BINDING FOLD, HOMODIMER, CHAPERONE
3k3s:A (ALA17) to (ARG40) CRYSTAL STRUCTURE OF ALTRONATE HYDROLASE (FRAGMENT 1-84) FROM SHIGELLA FLEXNERI. | ALTRONATE HYDROLASE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, HYDROLASE
3k48:D (SER107) to (GLY136) CRYSTAL STRUCTURE OF APRIL BOUND TO A PEPTIDE | CYTOKINE, TNFSF, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISULFIDE BOND, GLYCOPROTEIN, IMMUNE RESPONSE, SECRETED
2z4o:B (ARG157) to (GLY178) WILD TYPE HIV-1 PROTEASE WITH POTENT ANTIVIRAL INHIBITOR GRL-98065 | HIV-1, WILD TYPE PROTEASE, PROTEASE INHIBITOR, HYDROLASE
3k4v:B (GLY52) to (GLY78) NEW CRYSTAL FORM OF HIV-1 PROTEASE/SAQUINAVIR STRUCTURE REVEALS CARBAMYLATION OF N-TERMINAL PROLINE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX, CARBAMYLATION, AIDS, ASPARTYL PROTEASE, CAPSID MATURATION, CAPSID PROTEIN,
3k4v:C (ARG57) to (GLY78) NEW CRYSTAL FORM OF HIV-1 PROTEASE/SAQUINAVIR STRUCTURE REVEALS CARBAMYLATION OF N-TERMINAL PROLINE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX, CARBAMYLATION, AIDS, ASPARTYL PROTEASE, CAPSID MATURATION, CAPSID PROTEIN,
3k4v:D (GLY52) to (GLY78) NEW CRYSTAL FORM OF HIV-1 PROTEASE/SAQUINAVIR STRUCTURE REVEALS CARBAMYLATION OF N-TERMINAL PROLINE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX, CARBAMYLATION, AIDS, ASPARTYL PROTEASE, CAPSID MATURATION, CAPSID PROTEIN,
5cou:A (GLY78) to (PRO97) STRUCTURE AND MECHANISM OF A EUKARYAL NICK-SEALING RNA LIGASE K170M+ATP | RNA REPAIR, ADENYLYLTRANSFERASE, LIGASE
2o4k:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE (Q7K) IN COMPLEX WITH ATAZANAVIR | PROTEASE COMPLEX, VIRAL PROTEIN
2o4l:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE (Q7K, I50V) IN COMPLEX WITH TIPRANAVIR | PROTEASE, VIRAL PROTEIN
2o4n:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE (TRM MUTANT) IN COMPLEX WITH TIPRANAVIR | PROTEASE, VIRAL PROTEIN
2o4n:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE (TRM MUTANT) IN COMPLEX WITH TIPRANAVIR | PROTEASE, VIRAL PROTEIN
2o4p:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE (Q7K) IN COMPLEX WITH TIPRANAVIR | PROTEASE, VIRAL PROTEIN
4a4q:A (ARG57) to (GLY78) STEREOSELECTIVE SYNTHESIS, X-RAY ANALYSIS, AND BIOLOGICAL EVALUATION OF A NEW CLASS OF LACTAM BASED HIV-1 PROTEASE INHIBITORS | HYDROLASE, GAMMA-BUTYROL-LACTAM, INHIBITOR
4a4q:B (ARG157) to (GLY178) STEREOSELECTIVE SYNTHESIS, X-RAY ANALYSIS, AND BIOLOGICAL EVALUATION OF A NEW CLASS OF LACTAM BASED HIV-1 PROTEASE INHIBITORS | HYDROLASE, GAMMA-BUTYROL-LACTAM, INHIBITOR
2za9:A (ASN274) to (SER307) CRYSTAL STRUCTURE OF ALGINATE LYASE A1-II' N141C/N199C | ALGINATE LYASE, POLYSACCHARIDE LYASE FAMILY 7, N141C/N199C, LYASE
2zaa:A (ASN274) to (ASN308) CRYSTAL STRUCTURE OF FAMILY 7 ALGINATE LYASE A1-II' H191N/Y284F IN COMPLEX WITH SUBSTRATE (GGMG) | ALGINATE LYASE, POLYSACCHARIDE LYASE FAMILY 7, Y284F_TETRASACCHRIDE COMPLEX, LYASE
2zab:A (ASN274) to (SER307) CRYSTAL STRUCTURE OF FAMILY 7 ALGINATE LYASE A1-II' Y284F IN CMPLEX WITH PRODUCT (GGG) | ALGINATE LYASE, POLYSACCHARIDE LYASE FAMILY 7, Y284F, COMPLEX, LYASE
2zac:A (ASN274) to (SER307) CRYSTAL STRUCTURE OF FAMILY 7 ALGINATE LYASE A1-II' Y284F IN COMPLEX WITH PRODUCT (MMG) | ALGINATE, POLYSACCHARIDE LYASE FAMILY 7, Y284F_MMG COMPLEX, LYASE
4a6b:A (ARG57) to (GLY78) STEREOSELECTIVE SYNTHESIS, X-RAY ANALYSIS, AND BIOLOGICAL EVALUATION OF A NEW CLASS OF LACTAM BASED HIV-1 PROTEASE INHIBITORS | HYDROLASE, GAMMA-BUTYROL-LACTAM
4a6c:B (ARG157) to (GLY178) STEREOSELECTIVE SYNTHESIS, X-RAY ANALYSIS, AND BIOLOGICAL EVALUATION OF A NEW CLASS OF LACTAM BASED HIV-1 PROTEASE INHIBITORS | HYDROLASE, GAMMA-BUTYROL-LACTAM
4oju:A (TYR60) to (LYS83) CRYSTAL STRUCTURE OF A LEUCINE-RICH REPEAT PROTEIN (BACCAP_00569) FROM BACTEROIDES CAPILLOSUS ATCC 29799 AT 2.00 A RESOLUTION | LEUCINE RICH REPEATS,PF13306 FAMILY PROTEIN, PUTATIVE PROTEIN BINDING, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, UNKNOWN FUNCTION
4oju:B (TYR60) to (LYS83) CRYSTAL STRUCTURE OF A LEUCINE-RICH REPEAT PROTEIN (BACCAP_00569) FROM BACTEROIDES CAPILLOSUS ATCC 29799 AT 2.00 A RESOLUTION | LEUCINE RICH REPEATS,PF13306 FAMILY PROTEIN, PUTATIVE PROTEIN BINDING, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, UNKNOWN FUNCTION
4oju:C (TYR60) to (LYS83) CRYSTAL STRUCTURE OF A LEUCINE-RICH REPEAT PROTEIN (BACCAP_00569) FROM BACTEROIDES CAPILLOSUS ATCC 29799 AT 2.00 A RESOLUTION | LEUCINE RICH REPEATS,PF13306 FAMILY PROTEIN, PUTATIVE PROTEIN BINDING, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, UNKNOWN FUNCTION
4oju:D (TYR60) to (LYS83) CRYSTAL STRUCTURE OF A LEUCINE-RICH REPEAT PROTEIN (BACCAP_00569) FROM BACTEROIDES CAPILLOSUS ATCC 29799 AT 2.00 A RESOLUTION | LEUCINE RICH REPEATS,PF13306 FAMILY PROTEIN, PUTATIVE PROTEIN BINDING, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, UNKNOWN FUNCTION
1m14:A (GLU687) to (PRO709) TYROSINE KINASE DOMAIN FROM EPIDERMAL GROWTH FACTOR RECEPTOR | TRANSFERASE, TYROSINE KINASE DOMAIN
4omw:A (GLY17) to (PRO50) CRYSTAL STRUCTURE OF GOAT BETA-LACTOGLOBULIN (ORTHORHOMBIC FORM) | LIPOCALIN, TRANSPORT, TRANSPORT PROTEIN
4omw:B (GLY17) to (PRO50) CRYSTAL STRUCTURE OF GOAT BETA-LACTOGLOBULIN (ORTHORHOMBIC FORM) | LIPOCALIN, TRANSPORT, TRANSPORT PROTEIN
4omw:C (GLY17) to (PRO50) CRYSTAL STRUCTURE OF GOAT BETA-LACTOGLOBULIN (ORTHORHOMBIC FORM) | LIPOCALIN, TRANSPORT, TRANSPORT PROTEIN
4omw:D (GLY17) to (THR49) CRYSTAL STRUCTURE OF GOAT BETA-LACTOGLOBULIN (ORTHORHOMBIC FORM) | LIPOCALIN, TRANSPORT, TRANSPORT PROTEIN
1xq7:A (LYS91) to (PRO121) CYCLOPHILIN FROM TRYPANOSOMA CRUZI BOUND TO CYCLOSPORIN A | ISOMERASE-IMMUNOSUPPRESSANT COMPLEX, CYCLOPHILIN-CYCLOSPORIN COMPLEX, CYCLOSPORIN A, IMMUNOSUPPRESSANT, CYCLOPHILIN, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, PSI, STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA CONSORTIUM, SGPP
1xq7:B (LYS91) to (PRO121) CYCLOPHILIN FROM TRYPANOSOMA CRUZI BOUND TO CYCLOSPORIN A | ISOMERASE-IMMUNOSUPPRESSANT COMPLEX, CYCLOPHILIN-CYCLOSPORIN COMPLEX, CYCLOSPORIN A, IMMUNOSUPPRESSANT, CYCLOPHILIN, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, PSI, STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA CONSORTIUM, SGPP
1xq7:C (LYS91) to (PRO121) CYCLOPHILIN FROM TRYPANOSOMA CRUZI BOUND TO CYCLOSPORIN A | ISOMERASE-IMMUNOSUPPRESSANT COMPLEX, CYCLOPHILIN-CYCLOSPORIN COMPLEX, CYCLOSPORIN A, IMMUNOSUPPRESSANT, CYCLOPHILIN, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, PSI, STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA CONSORTIUM, SGPP
3kdb:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE (Q7K, L33I, L63I) IN COMPLEX WITH KNI-10006 | VIRAL PROTEIN, HYDROLASE, PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3kdd:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE (Q7K, L33I, L63I) IN COMPLEX WITH KNI-10265 | VIRAL PROTEIN, HYDROLASE, PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3kf0:B (ARG57) to (GLY78) HIV PROTEASE WITH FRAGMENT 4D9 BOUND | PROTEASE, TL-3 INHIBITOR, FRAGMENT HIT, ASPARTYL PROTEASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3kff:A (GLY17) to (GLU49) MAJOR MOUSE URINARY PROTEIN IV COMPLEXED WITH 2-SEC-BUTYL-4,5- DIHYDROTHIAZOLE | PHEROMONE, MAJOR URINARY PROTEIN, LIPOCALIN, BETA BARREL, DISULFIDE BOND, PHEROMONE-BINDING, SECRETED, TRANSPORT, TRANSPORT PROTEIN
3kfn:B (ARG57) to (GLY78) HIV PROTEASE (PR) WITH INHIBITOR TL-3 AND FRAGMENT HIT 4D9 BY SOAKING | HIV-1, PROTEASE, EXO SITE, ASPARTYL PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3kfr:A (ARG57) to (GLY78) HIV PROTEASE (PR) DIMER WITH INHIBITOR TL-3 BOUND AND FRAGMENT 1F1 IN THE OUTSIDE/TOP OF FLAP | HIV-1, PROTEASE, ASPARTYL PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5czi:A (GLU711) to (PRO733) EGFR L858R MUTANT IN COMPLEX WITH A SHC PEPTIDE SUBSTRATE | EGFR, L858R, KINASE, EGF, TRANSFERASE
4ozx:A (GLY270) to (GLY304) CRYSTAL STRUCTURE OF THE ALGINATE LYASE FROM KLEBSIELLA PNEUMONIAE | BETA-JELLY ROLL FOLD, ALGINATE, MANNURONATE, GULURONATE, POLYSACCHARIDE LYASE
1miq:A (ILE14) to (THR35) CRYSTAL STRUCTURE OF PROPLASMEPSIN FROM THE HUMAN MALARIAL PATHOGEN PLASMODIUM VIVAX | ASPARTIC PROTEINASE ZYMOGEN, DOMAIN OPENING, HYDROLASE
1y88:A (GLU21) to (ASP44) CRYSTAL STRUCTURE OF PROTEIN OF UNKNOWN FUNCTION AF1548 | AF1548, APC5567, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, PSI, MIDWEST CENTER FOR STRUCTURAL GENOMICS CENTER, MCSG, UNKNOWN FUNCTION
1mrx:B (ARG57) to (GLY78) STRUCTURE OF HIV PROTEASE (MUTANT Q7K L33I L63I V82F I84V ) COMPLEXED WITH KNI-577 | HIV, KNI-577, PROTEASE, DRUG TARGET, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5d5d:A (HIS218) to (GLY261) IN MESO IN SITU SERIAL X-RAY CRYSTALLOGRAPHY STRUCTURE OF ALGE AT 100 K | BETA-BARREL MEMBRANE PROTEINS, ALGE ALGINATE EXPORT PROTEIN, TRANSPORT PROTEIN
1msn:B (ARG57) to (GLY78) THE HIV PROTEASE (MUTANT Q7K L33I L63I V82F I84V) COMPLEXED WITH KNI- 764 (AN INHIBITOR) | HIV, KNI-764, PROTEASE, DRUG TARGET, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1msm:B (ARG57) to (GLY78) THE HIV PROTEASE (MUTANT Q7K L33I L63I) COMPLEXED WITH KNI-764 (AN INHIBITOR) | HIV, KNI-764, PROTEASE, DRUG TARGET, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1ybh:A (GLN644) to (GLY666) CRYSTAL STRUCTURE OF ARABIDOPSIS THALIANA ACETOHYDROXYACID SYNTHASE IN COMPLEX WITH A SULFONYLUREA HERBICIDE CHLORIMURON ETHYL | ACETOHYDROXYACID SYNTHASE, ACETOLACTATE SYNTHASE, HERBICIDE, SULFONYLUREA, THIAMIN DIPHOSPHATE, FAD, INHIBITOR, CYSTEINE-S- DIOXIDE, CHES, TRANSFERASE
4p9a:A (CYS541) to (SER571) X-RAY CRYSTAL STRUCTURE OF PA PROTEIN FROM INFLUENZA STRAIN H7N9 | PA PROTEIN INFLUENZA H7N9 POLYMERASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, SSGCID, VIRAL PROTEIN
1mt8:A (ARG57) to (GLY78) VIABILITY OF A DRUG-RESISTANT HIV-1 PROTEASE MUTANT: STRUCTURAL INSIGHTS FOR BETTER ANTIVIRAL THERAPY | MATRIX, CAPSID, GAG CLEAVAGE, DRUG RESISTANCE, SUBSTRATE RECOGNITION, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1mt9:A (ARG57) to (GLY78) VIABILITY OF A DRUG-RESISTANT HIV-1 PROTEASE MUTANT: STRUCTURAL INSIGHTS FOR BETTER ANTIVIRAL THERAPY | MATRIX, CAPSID, GAG CLEAVAGE, DRUG RESISTANCE, SUBSTRATE RECOGNITION, HYDROLASE
1mt9:B (ARG57) to (GLY78) VIABILITY OF A DRUG-RESISTANT HIV-1 PROTEASE MUTANT: STRUCTURAL INSIGHTS FOR BETTER ANTIVIRAL THERAPY | MATRIX, CAPSID, GAG CLEAVAGE, DRUG RESISTANCE, SUBSTRATE RECOGNITION, HYDROLASE
1mtb:A (ARG57) to (GLY78) VIABILITY OF A DRUG-RESISTANT HIV-1 PROTEASE MUTANT: STRUCTURAL INSIGHTS FOR BETTER ANTIVIRAL THERAPY | HIV-1 PROTEASE, DRUG RESISTANCE, SUBSTRATE RECOGNITION, INHIBITOR BINDING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5d7w:A (GLY131) to (ASN155) CRYSTAL STRUCTURE OF SERRALYSIN | PROTEASE, METALLOPROTEASE, HYDROLASE
1yge:A (VAL105) to (ASN133) LIPOXYGENASE-1 (SOYBEAN) AT 100K | DIOXYGENASE, LIPOXYGENASE, METALLOPROTEIN, FATTY ACIDS
1yhz:A (GLN644) to (GLY666) CRYSTAL STRUCTURE OF ARABIDOPSIS THALIANA ACETOHYDROXYACID SYNTHASE IN COMPLEX WITH A SULFONYLUREA HERBICIDE, CHLORSULFURON | ACETOHYDROXYACID SYNTHASE, ACETOLACTATE SYNTHASE, HERBICIDE, SULFONYLUREA, THIAMIN DIPHOSPHATE, FAD, INHIBITOR, CYSTEINE-S- DIOXIDE, CHES, CHLORSULFURON, TRANSFERASE
1ykf:A (MET1) to (PRO24) NADP-DEPENDENT ALCOHOL DEHYDROGENASE FROM THERMOANAEROBIUM BROCKII | OXIDOREDUCTASE
1ykf:B (MET1) to (PRO24) NADP-DEPENDENT ALCOHOL DEHYDROGENASE FROM THERMOANAEROBIUM BROCKII | OXIDOREDUCTASE
3kyg:A (GLY88) to (GLN116) CRYSTAL STRUCTURE OF VCA0042 (L135R) COMPLEXED WITH C-DI-GMP | C-DI-GMP, PILZ DOMAIN, PP4397, VCA0042, UNKNOWN FUNCTION
3kyg:B (GLU138) to (ARG165) CRYSTAL STRUCTURE OF VCA0042 (L135R) COMPLEXED WITH C-DI-GMP | C-DI-GMP, PILZ DOMAIN, PP4397, VCA0042, UNKNOWN FUNCTION
3kza:A (GLY17) to (THR49) CRYSTAL STRUCTURE OF GYUBA, A PATCHED CHIMERA OF B-LACTGLOBULIN | ARTIFICIAL PROTEIN, CHIMERA PROTEIN, DISULFIDE BOND, MILK PROTEIN, RETINOL-BINDING, SECRETED, TRANSPORT, TRANSPORT PROTEIN
3kza:B (GLY17) to (THR49) CRYSTAL STRUCTURE OF GYUBA, A PATCHED CHIMERA OF B-LACTGLOBULIN | ARTIFICIAL PROTEIN, CHIMERA PROTEIN, DISULFIDE BOND, MILK PROTEIN, RETINOL-BINDING, SECRETED, TRANSPORT, TRANSPORT PROTEIN
3abz:A (TRP810) to (TRP842) CRYSTAL STRUCTURE OF SE-MET LABELED BETA-GLUCOSIDASE FROM KLUYVEROMYCES MARXIANUS | GLYCOSIDE HYDROLASE FAMILY3 BETA-GLUCOSIDASE, PA14 DOMAIN, HYDROLASE
3abz:B (TRP810) to (TRP842) CRYSTAL STRUCTURE OF SE-MET LABELED BETA-GLUCOSIDASE FROM KLUYVEROMYCES MARXIANUS | GLYCOSIDE HYDROLASE FAMILY3 BETA-GLUCOSIDASE, PA14 DOMAIN, HYDROLASE
3abz:C (TRP810) to (TRP842) CRYSTAL STRUCTURE OF SE-MET LABELED BETA-GLUCOSIDASE FROM KLUYVEROMYCES MARXIANUS | GLYCOSIDE HYDROLASE FAMILY3 BETA-GLUCOSIDASE, PA14 DOMAIN, HYDROLASE
3abz:D (TRP810) to (TRP842) CRYSTAL STRUCTURE OF SE-MET LABELED BETA-GLUCOSIDASE FROM KLUYVEROMYCES MARXIANUS | GLYCOSIDE HYDROLASE FAMILY3 BETA-GLUCOSIDASE, PA14 DOMAIN, HYDROLASE
5df0:A (ARG29) to (ASN63) CRYSTAL STRUCTURE OF ACMNPV CHITINASE A IN COMPLEX WITH CHITOTRIO- THIAZOLINE DITHIOAMIDE | CHITINASE, ACMNPV, CHITIN, GLYCOSIDASE, HYDROLASE
5df0:B (ARG29) to (ASN63) CRYSTAL STRUCTURE OF ACMNPV CHITINASE A IN COMPLEX WITH CHITOTRIO- THIAZOLINE DITHIOAMIDE | CHITINASE, ACMNPV, CHITIN, GLYCOSIDASE, HYDROLASE
4phv:B (ARG57) to (GLY78) X-RAY CRYSTAL STRUCTURE OF THE HIV PROTEASE COMPLEX WITH L- 700,417, AN INHIBITOR WITH PSEUDO C2 SYMMETRY | HYDROLASE(ASPARTIC PROTEINASE)
5dgu:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE INHIBITORS CONTAINING SUBSTITUTED FUSED-TETRAHYDROPYRANYL TETRAHYDROFURAN AS P2-LIGAND GRL-004-11A | HIV-1 PROTEASE, ENZYME, HYDROLASE, HYDROLASE INHIBITOR
5dgw:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE INHIBITOR GRL-105-11A CONTAINING SUBSTITUTED FUSED-TETRAHYDROPYRANYL TETRAHYDROFURAN AS P2-LIGAND | HIV-1 PROTEASE, ENZYME, HYDROLASE, HYDROLASE INHIBITOR
1yu1:A (ALA73) to (PRO101) MAJOR TROPISM DETERMINANT P3C VARIANT | C-TYPE LECTIN, BETA SANDWICH, BETA PRISM, VARIABILITY, DIVERSITY- GENERATING RETROELEMENT, VIRAL PROTEIN
1yu2:A (ALA73) to (ALA102) MAJOR TROPISM DETERMINANT M1 VARIANT | C-TYPE LECTIN, BETA SANDWICH, BETA PRISM, VARIABILITY, DIVERSITY- GENERATING RETROELEMENT, VIRAL PROTEIN
1yu3:A (ALA73) to (PRO101) MAJOR TROPISM DETERMINANT I1 VARIANT | C-TYPE LECTIN, BETA SANDWICH, BETA PRISM, VARIABILITY, DIVERSITY- GENERATING RETROELEMENT, VIRAL PROTEIN
1yup:B (GLY17) to (PRO50) REINDEER BETA-LACTOGLOBULIN | TRANSPORT PROTEIN
1yup:E (GLY17) to (THR49) REINDEER BETA-LACTOGLOBULIN | TRANSPORT PROTEIN
1yup:H (GLY17) to (PRO50) REINDEER BETA-LACTOGLOBULIN | TRANSPORT PROTEIN
5dl7:A (ASP301) to (LEU341) CRYSTAL STRUCTURE OF ACINETOBACTER BAUMANNII OCCAB3 | OUTER MEMBRANE PROTEIN, BETA-BARREL, ANTIBIOTIC UPTAKE, ACINETOBACTER BAUMANNII, MEMBRANE PROTEIN
5dm6:H (VAL75) to (ASN100) CRYSTAL STRUCTURE OF THE 50S RIBOSOMAL SUBUNIT FROM DEINOCOCCUS RADIODURANS | PROTEIN SYNTHESIS, PEPTIDYLTRANSFERASE, RIBOZYME, RIBONUCLEOPROTEIN, RIBOSOME
5dma:A (GLY672) to (ARG693) CRYSTAL STRUCTURE OF C-TERMINAL TUDOR DOMAIN IN PCRA/UVRD HELICASE | RNA POLYMERASE, PCRA/UVRD HELICASE, TUDOR DOMAIN, TRANSCRIPTION, HYDROLASE
5dmp:A (THR88) to (ASN113) STRUCTURE OF THE ARCHAEAL NHEJ PHOSPHOESTERASE FROM METHANOCELLA PALUDICOLA. | ARCHAEAL PROTEINS, BIOCATALYSIS, DNA REPAIR ENZYMES, PHOSPHORIC DIESTER HYDROLASES, PHOSPHORIC MONOESTER HYDROLASES, HYDROLASE
4akm:A (SER336) to (PHE363) CRYSTAL STRUCTURE OF THE HUMAN LYSOSOME-ASSOCIATED MEMBRANE PROTEIN LAMP-3 (AKA DC-LAMP) | MEMBRANE PROTEIN, GLYCOSYLATION, BETA PRISM
4akm:B (SER336) to (PHE363) CRYSTAL STRUCTURE OF THE HUMAN LYSOSOME-ASSOCIATED MEMBRANE PROTEIN LAMP-3 (AKA DC-LAMP) | MEMBRANE PROTEIN, GLYCOSYLATION, BETA PRISM
3aic:E (GLU966) to (LYS1001) CRYSTAL STRUCTURE OF GLUCANSUCRASE FROM STREPTOCOCCUS MUTANS | BETA-ALPHA-BARRELS, TRANSFERASE
5dpk:A (GLU295) to (HIS323) MUTY ADENINE GLYCOSYLASE BOUND TO A TRANSITION STATE ANALOG (1N) PAIRED WITH D(8-OXOG) IN DUPLEXED DNA TO 2.2 A | PROTEIN-DNA COMPLEX, DNA REPAIR, GLYCOSYLASE, TRANSITION STATE ANALOG, HYDROLASE-DNA COMPLEX
3lix:A (PRO11) to (THR33) CRYSTAL STRUCTURE OF HTLV PROTEASE COMPLEXED WITH THE INHIBITOR KNI- 10729 | HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3ams:A (GLY281) to (HIS314) CRYSTAL STRUCTURES OF BACILLUS SUBTILIS ALKALINE PHYTASE IN COMPLEX WITH CA2+, CD2+, CO2+, NI2+, MG2+ AND MYO-INOSITOL HEXASULFATE | BETA-PROPELLER, PHYTASE, PHYTATE, MYO-INOSITOL HEXASULFATE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1zhs:B (GLN30) to (VAL54) CRYSTAL STRUCTURE OF MVL BOUND TO MAN3GLCNAC2 | MVL, HIV-1, CARBOHYDRATE BINDING, SUGAR BINDING PROTEIN
1zhs:C (GLN30) to (VAL54) CRYSTAL STRUCTURE OF MVL BOUND TO MAN3GLCNAC2 | MVL, HIV-1, CARBOHYDRATE BINDING, SUGAR BINDING PROTEIN
1zhs:F (GLN30) to (VAL54) CRYSTAL STRUCTURE OF MVL BOUND TO MAN3GLCNAC2 | MVL, HIV-1, CARBOHYDRATE BINDING, SUGAR BINDING PROTEIN
1zkf:B (ILE89) to (GLU120) CYRSTAL STRUCTURE OF HUMAN CYCLOPHILIN-A IN COMPLEX WITH SUC-AGPF-PNA | CYPA, CYCLOPHILIN-A, CYCLOPHILIN, PPIASE, PROLYL-ISOMERASE, ISOMERASE, ISOMERASE-ISOMERASE SUBSTRATE COMPLEX
5e16:A (TYR94) to (GLY122) CO-CRYSTAL STRUCTURE OF THE N-TERMIAL CGMP BINDING DOMAIN OF PLASMODIUM FALCIPARUM PKG WITH CGMP | KINASE, CGMP BINDING DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
1zsf:A (GLY52) to (GLY78) CRYSTAL STRUCTURE OF COMPLEX OF A HYDROXYETHYLAMINE INHIBITOR WITH HIV-1 PROTEASE AT 2.0A RESOLUTION | HIV, PROTEASE, PEPTIDOMIMETIC INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4ax3:A (LEU400) to (MET421) STRUCTURE OF THREE-DOMAIN HEME-CU NITRITE REDUCTASE FROM RALSTONIA PICKETTII AT 1.6 A RESOLUTION | THREE-DOMAIN HEME-CU NITRITE REDUCTASE, ELECTRON TRANSFER, OXIDOREDUCTASE, PROTON CHANNEL, DENITRIFICATION
4ax3:C (LEU400) to (MET421) STRUCTURE OF THREE-DOMAIN HEME-CU NITRITE REDUCTASE FROM RALSTONIA PICKETTII AT 1.6 A RESOLUTION | THREE-DOMAIN HEME-CU NITRITE REDUCTASE, ELECTRON TRANSFER, OXIDOREDUCTASE, PROTON CHANNEL, DENITRIFICATION
4ax3:D (GLY402) to (MET421) STRUCTURE OF THREE-DOMAIN HEME-CU NITRITE REDUCTASE FROM RALSTONIA PICKETTII AT 1.6 A RESOLUTION | THREE-DOMAIN HEME-CU NITRITE REDUCTASE, ELECTRON TRANSFER, OXIDOREDUCTASE, PROTON CHANNEL, DENITRIFICATION
3ary:A (LEU36) to (SER71) CRYSTAL STRUCTURE ANALYSIS OF CHITINASE A FROM VIBRIO HARVEYI WITH NOVEL INHIBITORS - COMPLEX STRUCTURE WITH 2-(IMIDAZOLIN-2-YL)-5- ISOTHIOCYANATOBENZOFURAN | TIM BARREL, INHIBITOR COMPLEX, GLYCOSIDASE, HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
5e5u:C (VAL124) to (TRP152) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN CARBONIC ANHYDRASE-LIKE DOMAIN OF PTPRG AND IMMUNOGLOBULIN DOMAINS 2-3 OF CNTN6 | NEURAL CELL ADHESION MOLECULE, RECEPTOR-TYPE PROTEIN TYROSINE PHOSPHATASE, IMMUNOGLOBULIN DOMAINS, CARBONIC ANHYDRASE-LIKE DOMAIN, CELL ADHESION-HYDROLASE COMPLEX
1zyr:D (TYR132) to (THR154) STRUCTURE OF THERMUS THERMOPHILUS RNA POLYMERASE HOLOENZYME IN COMPLEX WITH THE ANTIBIOTIC STREPTOLYDIGIN | RNA POLYMERASE; STREPTOLYDIGIN; TRANSCRIPTION; HOLOENZYME, TRANSCRIPTION,TRANSFERASE
1zyr:N (TYR132) to (THR154) STRUCTURE OF THERMUS THERMOPHILUS RNA POLYMERASE HOLOENZYME IN COMPLEX WITH THE ANTIBIOTIC STREPTOLYDIGIN | RNA POLYMERASE; STREPTOLYDIGIN; TRANSCRIPTION; HOLOENZYME, TRANSCRIPTION,TRANSFERASE
4b0b:B (LEU138) to (THR166) CRYSTAL STRUCTURE OF 3-HYDROXYDECANOYL-ACYL CARRIER PROTEIN DEHYDRATASE (FABA) FROM PSEUDOMONAS AERUGINOSA IN COMPLEX WITH 3-(PYRIDIN-2-YLOXY)ANILINE | LYASE, FATTY ACID BIOSYNTHESIS, BACTERIAL VIRULENCE, DRUG DISCOVERY
2a3x:F (PRO129) to (ASP161) DECAMERIC CRYSTAL STRUCTURE OF HUMAN SERUM AMYLOID P-COMPONENT BOUND TO BIS-1,2-{[(Z)-2CARBOXY- 2-METHYL-1,3-DIOXANE]- 5-YLOXYCARBONYL}- PIPERAZINE | MULTIVALENT LIGAND, SERUM AMYLOID, METAL BINDING PROTEIN
2a4z:A (PHE473) to (ALA528) CRYSTAL STRUCTURE OF HUMAN PI3KGAMMA COMPLEXED WITH AS604850 | PROTEIN-INHIBITOR COMPLEX, PI3KG, TRANSFERASE
3azq:B (GLY142) to (ASP169) CRYSTAL STRUCTURE OF PUROMYCIN HYDROLASE S511A MUTANT COMPLEXED WITH PGG | POP FAMILY, HYDROLASE
3m4p:A (LYS218) to (PRO248) ENTAMOEBA HISTOLYTICA ASPARAGINYL-TRNA SYNTHETASE (ASNRS) IN COMPLEX WITH ASPARAGINYL-ADENYLATE | AMINOACYL-TRNA SYNTHETASE, TRNA LIGASE, AARS, ASNRS, TRANSLATION, ATP-BINDING, NUCLEOTIDE-BINDING, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, LIGASE, PROTEIN BIOSYNTHESIS
3m4p:B (LYS218) to (PRO248) ENTAMOEBA HISTOLYTICA ASPARAGINYL-TRNA SYNTHETASE (ASNRS) IN COMPLEX WITH ASPARAGINYL-ADENYLATE | AMINOACYL-TRNA SYNTHETASE, TRNA LIGASE, AARS, ASNRS, TRANSLATION, ATP-BINDING, NUCLEOTIDE-BINDING, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, LIGASE, PROTEIN BIOSYNTHESIS
3m4p:C (LYS218) to (PRO248) ENTAMOEBA HISTOLYTICA ASPARAGINYL-TRNA SYNTHETASE (ASNRS) IN COMPLEX WITH ASPARAGINYL-ADENYLATE | AMINOACYL-TRNA SYNTHETASE, TRNA LIGASE, AARS, ASNRS, TRANSLATION, ATP-BINDING, NUCLEOTIDE-BINDING, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, LIGASE, PROTEIN BIOSYNTHESIS
3m4p:D (LYS218) to (PRO248) ENTAMOEBA HISTOLYTICA ASPARAGINYL-TRNA SYNTHETASE (ASNRS) IN COMPLEX WITH ASPARAGINYL-ADENYLATE | AMINOACYL-TRNA SYNTHETASE, TRNA LIGASE, AARS, ASNRS, TRANSLATION, ATP-BINDING, NUCLEOTIDE-BINDING, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, LIGASE, PROTEIN BIOSYNTHESIS
5eed:B (GLY17) to (THR49) OVINE LACTOGLOBULIN COMPLEX WITH DECANOL | TRANSPORT PROTEIN, LIGAND BINDING
3ma2:C (LEU334) to (PRO364) COMPLEX MEMBRANE TYPE-1 MATRIX METALLOPROTEINASE (MT1-MMP) WITH TISSUE INHIBITOR OF METALLOPROTEINASE-1 (TIMP-1) | PROTEIN - PROTEIN COMPLEX, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISULFIDE BOND, MEMBRANE, METAL-BINDING, METALLOPROTEASE, PROTEASE, TRANSMEMBRANE, ZYMOGEN, ERYTHROCYTE MATURATION, GLYCOPROTEIN, METALLOENZYME INHIBITOR, METALLOPROTEASE INHIBITOR, SECRETED, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4qj9:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF INACTIVE HIV-1 PROTEASE IN COMPLEX WITH P1-P6 SUBSTRATE VARIANT (R452S) | CO-EVOLUTION, PROTEASE, HYDROLASE
4qj9:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF INACTIVE HIV-1 PROTEASE IN COMPLEX WITH P1-P6 SUBSTRATE VARIANT (R452S) | CO-EVOLUTION, PROTEASE, HYDROLASE
3b7v:B (ARG157) to (GLY178) HIV-1 PROTEASE COMPLEXED WITH GEM-DIOL-AMINE TETRAHEDRAL INTERMEDIATE NLLTQI | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3b80:B (ARG157) to (GLY178) HIV-1 PROTEASE MUTANT I54V COMPLEXED WITH GEM-DIOL-AMINE INTERMEDIATE NLLTQI | HYDROLASE-HYDROLASE SUBSTRATE COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4bcl:A (ASP93) to (TYR122) FMO PROTEIN FROM PROSTHECOCHLORIS AESTUARII 2K AT ROOM TEMPERATURE | ELECTRON TRANSPORT, EXCITATION ENERGY TRANSFER, REACTION CENTER
3bb9:C (ASP102) to (ALA135) CRYSTAL STRUCTURE OF A PUTATIVE KETOSTEROID ISOMERASE (SFRI_1973) FROM SHEWANELLA FRIGIDIMARINA NCIMB 400 AT 1.80 A RESOLUTION | STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, UNKNOWN FUNCTION
3mji:B (VAL32) to (GLY59) ACTIVATION OF CATALYTIC CYSTEINE WITHOUT A BASE IN A MUTANT PENICILLIN ACYLASE PRECURSOR | ZYMOGEN, HYDROLASE, PENICILLIN, AUTOPROTEOLYSIS, ANTIBIOTIC RESISTANCE, CATALYSIS, PENICILLIN V ACYLASE, AMIDASE
3bhe:A (GLY52) to (GLY78) HIV-1 PROTEASE IN COMPLEX WITH A THREE ARMED PYRROLIDINE DERIVATIVE | PROTEIN-LIGAND COMPLEX, HYDROLASE
4qwt:B (PRO80) to (ILE107) ANAEROBIC CRYSTAL STRUCTURE OF DELTA413-417:GS LOX IN COMPLEX WITH ARACHIDONATE | IRON BINDING, MEMBRANE-ASSOCIATED, OXIDOREDUCTASE
4qwt:D (PRO80) to (ILE107) ANAEROBIC CRYSTAL STRUCTURE OF DELTA413-417:GS LOX IN COMPLEX WITH ARACHIDONATE | IRON BINDING, MEMBRANE-ASSOCIATED, OXIDOREDUCTASE
3mxd:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE INHIBITOR KC53 IN COMPLEX WITH WILD-TYPE PROTEASE | DRUG DESIGN, HIV-1 PROTEASE, PROTEASE INHIBITORS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3bva:B (ARG57) to (GLY78) CYSTAL STRUCTURE OF HIV-1 ACTIVE SITE MUTANT D25N AND P2-NC ANALOG INHIBITOR | DRUG RESISTANCE, HIV-1, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3bvb:B (ARG57) to (GLY78) CYSTAL STRUCTURE OF HIV-1 ACTIVE SITE MUTANT D25N AND INHIBITOR DARUNAVIR | DRUG RESISTANCE; HIV-1; D25N, MUTANT, AIDS, ASPARTYL PROTEASE, CAPSID MATURATION, CORE PROTEIN, DNA INTEGRATION, DNA RECOMBINATION, DNA- DIRECTED DNA POLYMERASE, ENDONUCLEASE, HYDROLASE, LIPOPROTEIN, MAGNESIUM, MEMBRANE, METAL-BINDING, MULTIFUNCTIONAL ENZYME, MYRISTATE, NUCLEASE, NUCLEOTIDYLTRANSFERASE, NUCLEUS, PHOSPHOPROTEIN, PROTEASE, RNA-BINDING, RNA-DIRECTED DNA POLYMERASE, TRANSFERASE, VIRAL NUCLEOPROTEIN, VIRION, ZINC-FINGER
4r1j:A (VAL62) to (ASP88) CRYSTAL STRUCTURE OF ARC1P-C | EMAP, TRNA BINDING, TRNA, RNA BINDING PROTEIN
3cc2:K (VAL74) to (ASP99) THE REFINED CRYSTAL STRUCTURE OF THE HALOARCULA MARISMORTUI LARGE RIBOSOMAL SUBUNIT AT 2.4 ANGSTROM RESOLUTION WITH RRNA SEQUENCE FOR THE 23S RRNA AND GENOME-DERIVED SEQUENCES FOR R-PROTEINS | GENOMIC SEQUNECE FOR R-PROTEINS, RIBONUCLEOPROTEIN, RIBOSOMAL PROTEIN, RNA-BINDING, RRNA-BINDING, TRNA-BINDING, METAL-BINDING, ZINC-FINGER, RIBOSOME
3cc4:K (VAL74) to (ASP99) CO-CRYSTAL STRUCTURE OF ANISOMYCIN BOUND TO THE 50S RIBOSOMAL SUBUNIT | WILD TYPE, LARGE RIBOSOMAL SUBUNIT, HALOARCULA MARISMORTUI, CO- CRYSTAL, ANISOMYCIN, RIBOSOME
3cc7:K (VAL74) to (ASP99) STRUCTURE OF ANISOMYCIN RESISTANT 50S RIBOSOMAL SUBUNIT: 23S RRNA MUTATION C2487U | ANISOMYCIN RESISTANCE, C2487U, LARGE RIBOSOMAL SUBUNIT, 23S RRNA, RIBONUCLEOPROTEIN, RIBOSOMAL PROTEIN, RNA-BINDING, RRNA-BINDING, TRNA-BINDING, METAL-BINDING, ZINC-FINGER, RIBOSOME
3ccl:K (VAL74) to (ASP99) STRUCTURE OF ANISOMYCIN RESISTANT 50S RIBOSOMAL SUBUNIT: 23S RRNA MUTATION U2535C. DENSITY FOR ANISOMYCIN IS VISIBLE BUT NOT INCLUDED IN MODEL. | U2535C MUTATION, 23S RRNA, LARGE RIBOSOMAL SUBUNIT, RIBOSOME
3ccq:K (VAL74) to (ASP99) STRUCTURE OF ANISOMYCIN RESISTANT 50S RIBOSOMAL SUBUNIT: 23S RRNA MUTATION A2488U | GENOMIC SEQUNECE FOR R-PROTEINS, RIBOSOME
3ccs:K (VAL74) to (ASP99) STRUCTURE OF ANISOMYCIN RESISTANT 50S RIBOSOMAL SUBUNIT: 23S RRNA MUTATION G2482A | G2482A MUTATION, 23S RRNA, LARGE RIBOSOMAL SUBUNIT, RIBOSOME
3cd6:K (LEU69) to (ASP99) CO-CYSTAL OF LARGE RIBOSOMAL SUBUNIT MUTANT G2616A WITH CC-PUROMYCIN | G2616A MUTATION, 23S RRNA, LARGE RIBOSOMAL SUBUNIT, CC-PUROMYCIN, RIBOSOME
3ndt:C (ARG57) to (GLY78) HIV-1 PROTEASE SAQUINAVIR:RITONAVIR 1:1 COMPLEX STRUCTURE | HYDROLASE, AIDS, ASPARTYL PROTEASE, CARBAMYLATION, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3ndu:A (GLY53) to (GLY79) HIV-1 PROTEASE SAQUINAVIR:RITONAVIR 1:5 COMPLEX STRUCTURE | HIV-1 PROTEASE, HYDROLASE, AIDS, ASPARTYL PROTEASE, SAQUINAVIR, CARBAMYLATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3ndu:B (GLY53) to (GLY79) HIV-1 PROTEASE SAQUINAVIR:RITONAVIR 1:5 COMPLEX STRUCTURE | HIV-1 PROTEASE, HYDROLASE, AIDS, ASPARTYL PROTEASE, SAQUINAVIR, CARBAMYLATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3ndu:C (ARG57) to (GLY78) HIV-1 PROTEASE SAQUINAVIR:RITONAVIR 1:5 COMPLEX STRUCTURE | HIV-1 PROTEASE, HYDROLASE, AIDS, ASPARTYL PROTEASE, SAQUINAVIR, CARBAMYLATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3ndu:D (GLY52) to (GLY78) HIV-1 PROTEASE SAQUINAVIR:RITONAVIR 1:5 COMPLEX STRUCTURE | HIV-1 PROTEASE, HYDROLASE, AIDS, ASPARTYL PROTEASE, SAQUINAVIR, CARBAMYLATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3ndw:A (ARG57) to (GLY78) HIV-1 PROTEASE SAQUINAVIR:RITONAVIR 1:15 COMPLEX STRUCTURE | HIV-1 PROTEASE, HYDROLASE, AIDS, ASPARTYL PROTEASE, SAQUINAVIR, CARBAMYLATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3ndw:B (ARG57) to (GLY78) HIV-1 PROTEASE SAQUINAVIR:RITONAVIR 1:15 COMPLEX STRUCTURE | HIV-1 PROTEASE, HYDROLASE, AIDS, ASPARTYL PROTEASE, SAQUINAVIR, CARBAMYLATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3ndx:B (ARG57) to (GLY78) HIV-1 PROTEASE SAQUINAVIR:RITONAVIR 1:50 COMPLEX STRUCTURE | HIV-1 PROTEASE, HYDROLASE, AIDS, ASPARTYL PROTEASE, SAQUINAVIR, CARBAMYLATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3cm8:A (CYS541) to (SER571) A RNA POLYMERASE SUBUNIT STRUCTURE FROM VIRUS | PROTEIN-PEPTIDE COMPLEX, NUCLEOTIDE-BINDING, NUCLEOTIDYLTRANSFERASE, RNA REPLICATION, RNA-DIRECTED RNA POLYMERASE, TRANSFERASE, RNA BINDING PROTEIN/TRANSFERASE COMPLEX
3cma:K (VAL74) to (ASP99) THE STRUCTURE OF CCA AND CCA-PHE-CAP-BIO BOUND TO THE LARGE RIBOSOMAL SUBUNIT OF HALOARCULA MARISMORTUI | RIBOSOME 50S, PROTEIN-PROTEIN COMPLEX, RNA-RNA COMPLEX, PROTEIN-RNA COMPLEX, PEPTIDYL-TRNA HYDROLYSIS, RIBOSOME
4riy:B (GLU687) to (PRO709) CRYSTAL STRUCTURE OF AN EGFR/HER3 KINASE DOMAIN HETERODIMER CONTAINING THE CANCER-ASSOCIATED HER3-E909G MUTATION | RECEPTOR TYROSINE KINASE, PSEUDOKINASE, KINASE, ATP BINDING, MEMBRANE, TRANSFERASE
5fr8:B (GLN689) to (PHE730) CRYSTAL STRUCTURE OF THE SIDEROPHORE RECEPTOR PIRA FROM ACINETOBACTER BAUMANNII | TRANSPORT PROTEIN, TONB-DEPENDENT RECEPTOR, OUTER-MEMBRANE PROTEIN
3nqk:A (GLY182) to (TYR212) CRYSTAL STRUCTURE OF A STRUCTURAL GENOMICS, UNKNOWN FUNCTION (BACOVA_03322) FROM BACTEROIDES OVATUS AT 2.61 A RESOLUTION | STRUCTURAL GENOMICS, UNKNOWN FUNCTION, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2
3nqk:A (TYR283) to (ASN327) CRYSTAL STRUCTURE OF A STRUCTURAL GENOMICS, UNKNOWN FUNCTION (BACOVA_03322) FROM BACTEROIDES OVATUS AT 2.61 A RESOLUTION | STRUCTURAL GENOMICS, UNKNOWN FUNCTION, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2
4rny:B (SER241) to (ALA265) STRUCTURE OF HELICOBACTER PYLORI CSD3 FROM THE ORTHORHOMBIC CRYSTAL | M23B METALLOPEPTIDASE, METALLOPEPTIDASE, PEPTIDOGLYCAN, HYDROLASE
3nu9:B (ARG157) to (GLY178) CRYSTAL STRUCTURE OF HIV-1 PROTEASE MUTANT I84V WITH ANTIVIRAL DRUG AMPRENAVIR | ENZYME INHIBITION, ASPARTIC PROTEASE, HIV/AIDS, CONFORMATIONAL CHANGE, AMPRENAVIR, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5fu7:F (VAL477) to (CYS504) DROSOPHILA NANOS NBR PEPTIDE BOUND TO THE NOT MODULE OF THE HUMAN CCR4-NOT COMPLEX | GENE REGULATION, DEADENYLATION, MRNA DECAY, CCR4-NOT, TRANSCRIPTION, TRANSLATIONAL REPRESSION
3nuo:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE MUTANT L90M WITH ANTIVIRAL DRUG AMPRENAVIR | ENZYME INHIBITION, ASPARTIC PROTEASE, HIV/AIDS, CONFORMATIONAL CHANGE, AMPRENAVIR, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3nwa:B (VAL574) to (THR626) GLYCOPROTEIN B FROM HERPES SIMPLEX VIRUS TYPE 1, W174R MUTANT, LOW-PH | COILED-COIL, ENVELOPE GLYCOPROTEIN, MEMBRANE FUSION, VIRAL PROTEIN, GLYCOPROTEIN B, HERPESVIRUS 1, HSV-1, MEMBRANE
4ck4:A (GLY17) to (THR49) OVINE BETA-LACTOGLOBULIN AT ATOMIC RESOLUTION | TRANSPORT PROTEIN, OVINE-LACTOGLOBULIN, HIGH RESOLUTION
4ck4:B (GLY17) to (THR49) OVINE BETA-LACTOGLOBULIN AT ATOMIC RESOLUTION | TRANSPORT PROTEIN, OVINE-LACTOGLOBULIN, HIGH RESOLUTION
3cyx:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 MUTANT I50V AND INHIBITOR SAQUINAVIRA | DRUG RESISTANCE; HIV-1, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4coe:B (ARG157) to (GLY178) MACROCYCLIC TRANSITION-STATE MIMICKING HIV-1 PROTEASE INHIBITORS ENCOMPASSING A TERTIARY ALCOHOL | HYDROLASE, INHIBITOR, RATIONAL DRUG DESIGN, ENZYME
3d1x:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 MUTANT I54M AND INHIBITOR SAQUINAVIR | DRUG RESISTANCE, HIV-1, I54M, FLAP MUTANT, AIDS, ASPARTYL PROTEASE, CAPSID MATURATION, CAPSID PROTEIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX, VIRAL NUCLEOPROTEIN
3d1z:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 MUTANT I54M AND INHIBITOR DARUNAVIR | DRUG RESISTANCE; HIV-1, FLAP MUTANT, I54M, DARUNAVIR, HYDROLASE
3d20:B (ARG157) to (GLY178) CRYSTAL STRUCTURE OF HIV-1 MUTANT I54V AND INHIBITOR DARUNAVIA | DRUG RESISTANCE; HIV-1, I54V, FLAP MUTANT, AIDS, ASPARTYL PROTEASE, CAPSID MATURATION, CAPSID PROTEIN, DNA INTEGRATION, DNA RECOMBINATION, DNA-DIRECTED DNA POLYMERASE, ENDONUCLEASE, HYDROLASE, LIPOPROTEIN, MAGNESIUM, MEMBRANE, METAL-BINDING, MULTIFUNCTIONAL ENZYME, MYRISTATE, NUCLEASE, NUCLEOTIDYLTRANSFERASE, NUCLEUS, PHOSPHOPROTEIN, PROTEASE, RNA-BINDING, RNA-DIRECTED DNA POLYMERASE, TRANSFERASE, VIRAL NUCLEOPROTEIN, VIRION, ZINC-FINGER
4cpr:B (ARG157) to (GLY178) MACROCYCLIC TRANSITION-STATE MIMICKING HIV-1 PROTEASE INHIBITORS ENCOMPASSING A TERTIARY ALCOHOL | HYDROLASE, INHIBITOR, RATIONAL DRUG DESIGN
4cps:B (ARG157) to (GLY178) MACROCYCLIC TRANSITION-STATE MIMICKING HIV-1 PROTEASE INHIBITORS ENCOMPASSING A TERTIARY ALCOHOL | HYDROLASE, INHIBITOR, RATIONAL DRUG DESIGN
4cpx:A (ARG57) to (GLY78) MACROCYCLIC TRANSITION-STATE MIMICKING HIV-1 PROTEASE INHIBITORS ENCOMPASSING A TERTIARY ALCOHOL | HYDROLASE, INHIBITOR, RATIONAL DRUG DESIGN
4cpx:B (ARG157) to (GLY178) MACROCYCLIC TRANSITION-STATE MIMICKING HIV-1 PROTEASE INHIBITORS ENCOMPASSING A TERTIARY ALCOHOL | HYDROLASE, INHIBITOR, RATIONAL DRUG DESIGN
4cpt:B (ARG157) to (GLY178) MACROCYCLIC TRANSITION-STATE MIMICKING HIV-1 PROTEASE INHIBITORS ENCOMPASSING A TERTIARY ALCOHOL | HYDROLASE, HIV-1 PROTEASE, INHIBITOR, RATIONAL DRUG DESIGN, ENZYME
4cpu:B (ARG157) to (GLY178) MACROCYCLIC TRANSITION-STATE MIMICKING HIV-1 PROTEASE INHIBITORS ENCOMPASSING A TERTIARY ALCOHOL | HYDROLASE, HIV-1 PROTEASE, INHIBITOR, RATIONAL DRUG DESIGN
4cpw:B (ARG157) to (GLY178) MACROCYCLIC TRANSITION-STATE MIMICKING HIV-1 PROTEASE INHIBITORS ENCOMPASSING A TERTIARY ALCOHOL | HYDROLASE, INHIBITOR, RATIONAL DRUG DESIGN
3o9h:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF WILD-TYPE HIV-1 PROTEASE IN COMPLEX WITH KD26 | HIV-1 PROTEASE, DRUG RESISTANCE, DRUG DESIGN, PROTEASE INHIBITORS, AIDS, ASPARTYL PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3o9h:B (GLY52) to (GLY78) CRYSTAL STRUCTURE OF WILD-TYPE HIV-1 PROTEASE IN COMPLEX WITH KD26 | HIV-1 PROTEASE, DRUG RESISTANCE, DRUG DESIGN, PROTEASE INHIBITORS, AIDS, ASPARTYL PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3dk1:B (ARG157) to (GLY178) WILD TYPE HIV-1 PROTEASE WITH POTENT ANTIVIRAL INHIBITOR GRL-0105A | HIV-1, WILD TYPE PROTEASE, PROTEASE INHIBITOR, HYDROLASE, AIDS, ASPARTYL PROTEASE, CAPSID MATURATION, CAPSID PROTEIN, CYTOPLASM, DNA INTEGRATION, DNA RECOMBINATION, DNA-DIRECTED DNA POLYMERASE, ENDONUCLEASE, LIPOPROTEIN, MAGNESIUM, METAL- BINDING, MULTIFUNCTIONAL ENZYME, MYRISTATE, NUCLEASE, NUCLEOTIDYLTRANSFERASE, NUCLEUS, PHOSPHOPROTEIN, PROTEASE, RIBOSOMAL FRAMESHIFTING, RNA-BINDING, RNA-DIRECTED DNA POLYMERASE, TRANSFERASE, VIRAL NUCLEOPROTEIN, VIRION, ZINC, ZINC-FINGER
4tvg:B (ARG57) to (GLY78) HIV PROTEASE (PR) DIMER IN CLOSED FORM WITH PEPSTATIN IN ACTIVE SITE AND FRAGMENT AK-2097 IN THE OUTSIDE/TOP OF FLAP | APO PROTEASE, ALLOSTERY, FRAGMENT BINDING
4tvh:B (ARG57) to (GLY78) HIV PROTEASE (PR) DIMER IN CLOSED FORM WITH TL-3 IN ACTIVE SITE AND FRAGMENT AK-2097 IN THE OUTSIDE/TOP OF FLAP | HIV PROTEASE, ALLOSTERY, FRAGMENT BINDING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3doi:A (LYS122) to (HIS153) CRYSTAL STRUCTURE OF A THERMOSTABLE ESTERASE COMPLEX WITH PARAOXON | ALPHA-BETA HYDROLASE, BETA SHEET
3dte:A (LYS190) to (PRO214) CRYSTAL STRUCTURE OF THE IRRE PROTEIN, A CENTRAL REGULATOR OF DNA DAMAGE REPAIR IN DEINOCOCCACEAE | DEINOCOCCUS, RADIOTOLERANCE, GENE REGULATION, METALLOPEPTIDASE, IRRE
5hc1:C (ALA156) to (VAL178) STRUCTURE OF EAV NSP11 H141A MUTANT AT 3.10A | NSP11, EQUINE ARTERITIS VIRUS, ENDORIBONUCLEASE, NONSTRUCTURAL PROTEIN 11, NIDOVIRUS, NF-KAPPAB, HYDROLASE
3oxw:C (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 I50V, A71V PROTEASE IN COMPLEX WITH THE PROTEASE INHIBITOR DARUNAVIR | HIV-1 PROTEASE, INHIBITOR RESISTANCE, AIDS, ASPARTYL PROTEASE, DRUG RESISTANCE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4dfg:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF WILD-TYPE HIV-1 PROTEASE WITH CYCLOPENTYLTETRAHYDRO- FURANYL URETHANES AS P2-LIGAND, GRL-0249A | ASPARTIC ACID PROTEASE, HIV-1 PROTEASE INHIBITOR GRL-0249A, CYCLOPENTYLTETRAHYDRO- FURANYL URETHANES P2-LIGANDS, WILD-TYPE HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4djo:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF WILD-TYPE HIV-1 PROTEASE IN COMPLEX WITH MKP56 | HIV-1 PROTEASE, DRUG RESISTANCE, DRUG DESIGN, PROTEASE INHIBITORS, AIDS, ASPARTYL PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4djo:B (GLY52) to (GLY78) CRYSTAL STRUCTURE OF WILD-TYPE HIV-1 PROTEASE IN COMPLEX WITH MKP56 | HIV-1 PROTEASE, DRUG RESISTANCE, DRUG DESIGN, PROTEASE INHIBITORS, AIDS, ASPARTYL PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4u67:H (VAL75) to (ASN100) CRYSTAL STRUCTURE OF THE LARGE RIBOSOMAL SUBUNIT (50S) OF DEINOCOCCUS RADIODURANS CONTAINING A THREE RESIDUE INSERTION IN L22 | RIBOSOME, ANTIBIOTICS, RESISTANCE, ERYTHROMYCIN
3p27:B (SER429) to (GLY453) CRYSTAL STRUCTURE OF S. CEREVISIAE HBS1 PROTEIN (GDP-BOUND FORM), A TRANSLATIONAL GTPASE INVOLVED IN RNA QUALITY CONTROL PATHWAYS AND INTERACTING WITH DOM34/PELOTA | GDP/GTP BINDING DOMAIN, BETA-BARREL, TRANSLATIONAL GTPASE, STRUCTURAL GENOMICS, PARIS-SUD YEAST STRUCTURAL GENOMICS, YSG, SIGNALING PROTEIN
3p56:C (ARG66) to (LEU134) THE STRUCTURE OF THE HUMAN RNASE H2 COMPLEX DEFINES KEY INTERACTION INTERFACES RELEVANT TO ENZYME FUNCTION AND HUMAN DISEASE | RNASE H FOLD, TRIPLE BETA-BARREL, NUCLEASE THAT CLEAVES RNA/DNA HYBRIDS, PROLIFERATING CELL NUCLEAR ANTIGEN (PCNA) AND RNA/DNA HYBRIDS, NUCLEUS, HYDROLASE-REPLICATION COMPLEX
3p56:F (ARG66) to (LEU134) THE STRUCTURE OF THE HUMAN RNASE H2 COMPLEX DEFINES KEY INTERACTION INTERFACES RELEVANT TO ENZYME FUNCTION AND HUMAN DISEASE | RNASE H FOLD, TRIPLE BETA-BARREL, NUCLEASE THAT CLEAVES RNA/DNA HYBRIDS, PROLIFERATING CELL NUCLEAR ANTIGEN (PCNA) AND RNA/DNA HYBRIDS, NUCLEUS, HYDROLASE-REPLICATION COMPLEX
3p5j:C (ARG66) to (LEU136) THE STRUCTURE OF THE HUMAN RNASE H2 COMPLEX DEFINES KEY INTERACTION INTERFACES RELEVANT TO ENZYME FUNCTION AND HUMAN DISEASE | RNASE H2 FOLD, TRIPLE BETA-BARREL, NUCLEASE THAT CLEAVES RNA/DNA HYBRIDS, PROLIFERATING CELL NUCLEAR ANTIGEN (PCNA) AND RNA/DNA HYBRIDS, NUCLEUS, HYDROLASE-REPLICATION COMPLEX
4dqb:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF WILD-TYPE HIV-1 PROTEASE IN COMPLEX WITH DRV | HIV-1 PROTEASE, DRUG RESISTANCE, DRUG DESIGN, PROTEASE INHIBITORS, AIDS, ASPARTYL PROTEASE, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5htd:A (GLY17) to (THR49) RECOMBINANT BOVINE BETA-LACTOGLOBULIN VARIANT L1A/I2S WITH ENDOGENOUS LIGAND (SBLGB#1) | LIPOCALIN, TRANSPORT PROTEIN
5hv0:A (ALA139) to (PHE181) STRUCTURAL ANALYSIS OF COFACTOR BINDING OF A PROLYL 4-HYDROXYLASE FROM THE PATHOGENIC BACTERIUM BACILLUS ANTHRACIS | P4H, DIOXYGENASE, CUPIN, FE(II)/ALPHA-KETOGLUTARATE, OXIDOREDUCTASE
5hv0:B (ALA139) to (PHE181) STRUCTURAL ANALYSIS OF COFACTOR BINDING OF A PROLYL 4-HYDROXYLASE FROM THE PATHOGENIC BACTERIUM BACILLUS ANTHRACIS | P4H, DIOXYGENASE, CUPIN, FE(II)/ALPHA-KETOGLUTARATE, OXIDOREDUCTASE
5hx2:D (ASN121) to (LYS157) IN VITRO ASSEMBLED STAR-SHAPED HUBLESS T4 BASEPLATE | T4, BASEPLATE, COMPLEX, VIRAL PROTEIN
3ph5:A (GLY33) to (THR65) BOVINE BETA LACTOGLOBULIN CRYSTALLIZED THROUGH LIGANDATION OF YTTRIUM CATIONS | TRANSPORT PROTEIN
3ph6:A (GLY33) to (THR65) BOVINE BETA LACTOGLOBULIN CRYTSALLIZED THROUGH LIGANDATION OF YTTRIUM | TRANSPORT PROTEIN
3ph6:B (GLY33) to (THR65) BOVINE BETA LACTOGLOBULIN CRYTSALLIZED THROUGH LIGANDATION OF YTTRIUM | TRANSPORT PROTEIN
4unm:B (PRO165) to (PRO192) STRUCTURE OF GALACTOSE OXIDASE HOMOLOGUE FROM STREPTOMYCES LIVIDANS | METAL BINDING PROTEIN, COPPER OXIDASE
5i9y:A (VAL613) to (THR634) CRYSTAL STRUCTURE OF EPHRIN A2 (EPHA2) RECEPTOR PROTEIN KINASE WITH DASATINIB | TRANSFERASE, TYROSINE-PROTEIN KINASE, RECEPTOR, ATP-BINDING
5iat:B (SER144) to (PHE181) MECHANISTIC AND STRUCTURAL ANALYSIS OF SUBSTRATE RECOGNITION AND COFACTOR BINDING BY AN UNUSUAL BACTERIAL PROLYL HYDROXYLASE - APO- BAP4H | P4H, DIOXYGENASE, CUPIN, FE(II)/ALPHA-KETOGLUTARATE, OXIDOREDUCTASE
3pp9:A (ASP21) to (LEU55) 1.6 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF PUTATIVE STREPTOTHRICIN ACETYLTRANSFERASE FROM BACILLUS ANTHRACIS STR. AMES IN COMPLEX WITH ACETYL COENZYME A | PUTATIVE STREPTOTHRICIN ACETYLTRANSFERASE, TOXIN PRODUCTION AND RESISTANCE, INFECTIOUS DISEASES, STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES (CSGID), TRANSFERASE
3pp9:C (ASN15) to (LEU55) 1.6 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF PUTATIVE STREPTOTHRICIN ACETYLTRANSFERASE FROM BACILLUS ANTHRACIS STR. AMES IN COMPLEX WITH ACETYL COENZYME A | PUTATIVE STREPTOTHRICIN ACETYLTRANSFERASE, TOXIN PRODUCTION AND RESISTANCE, INFECTIOUS DISEASES, STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES (CSGID), TRANSFERASE
3puf:C (GLU71) to (LEU134) CRYSTAL STRUCTURE OF HUMAN RNASE H2 COMPLEX | RNASE H FOLD, TRIPLE BARREL FOLD, HYDROLASE, RNASE H
3puf:I (GLU71) to (LEU134) CRYSTAL STRUCTURE OF HUMAN RNASE H2 COMPLEX | RNASE H FOLD, TRIPLE BARREL FOLD, HYDROLASE, RNASE H
3puf:O (GLU71) to (LEU134) CRYSTAL STRUCTURE OF HUMAN RNASE H2 COMPLEX | RNASE H FOLD, TRIPLE BARREL FOLD, HYDROLASE, RNASE H
3puf:R (GLU71) to (LEU134) CRYSTAL STRUCTURE OF HUMAN RNASE H2 COMPLEX | RNASE H FOLD, TRIPLE BARREL FOLD, HYDROLASE, RNASE H
3pva:A (VAL29) to (GLY56) PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE, HYDROLASE
3pva:B (VAL29) to (GLY56) PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE, HYDROLASE
3pva:C (VAL29) to (GLY56) PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE, HYDROLASE
3pva:D (VAL29) to (GLY56) PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE, HYDROLASE
3pva:E (VAL29) to (GLY56) PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE, HYDROLASE
3pva:F (VAL29) to (GLY56) PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE, HYDROLASE
3pva:G (VAL29) to (GLY56) PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE, HYDROLASE
3pva:H (VAL29) to (GLY56) PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE, HYDROLASE
3pvo:D (ALA131) to (ASP163) MONOCLINIC FORM OF HUMAN C-REACTIVE PROTEIN | PENTRAXIN FAMILY, IMMUNE SYSTEM
3pvo:H (ALA131) to (ASP163) MONOCLINIC FORM OF HUMAN C-REACTIVE PROTEIN | PENTRAXIN FAMILY, IMMUNE SYSTEM
3pvo:I (ALA131) to (ASP163) MONOCLINIC FORM OF HUMAN C-REACTIVE PROTEIN | PENTRAXIN FAMILY, IMMUNE SYSTEM
3pvo:S (ALA131) to (ASP163) MONOCLINIC FORM OF HUMAN C-REACTIVE PROTEIN | PENTRAXIN FAMILY, IMMUNE SYSTEM
3pwr:B (ARG157) to (GLY178) HIV-1 PROTEASE MUTANT L76V COMPLEXED WITH SAQUINAVIR | HIV-1, PROTEASE, MUTATION L76V, SAQUINAVIR, HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
5io7:A (GLY17) to (THR49) BOVINE BETA-LACTOGLOBULIN COMPLEX WITH DODECANE AT HIGH PRESSURE (0.43 GPA) | BETA-LACTOGLOBULIN, LIPOCALIN, TRANSPORT PROTEIN
4ejk:B (ARG57) to (GLY78) HIV PROTEASE (PR) DIMER IN CLOSED FORM WITH PEPSTATIN IN ACTIVE SITE AND FRAGMENT 1F1-N IN THE OUTSIDE/TOP OF FLAP | APO PROTEASE, ALLOSTERY, FRAGMENT BINDING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3q2r:A (TYR147) to (PRO177) CRYSTAL STRUCTURE OF SGLIPR1 SOAKED WITH ZINC CHLORIDE | GLIOMA, CRISP, HUMAN GLIOMA PATHOGENESIS-RELATED PROTEIN 1 (GLIPR1), RTVP1, MEMBRANE PROTEIN
4epj:A (GLY152) to (GLY178) CRYSTAL STRUCTURE OF INACTIVE SINGLE CHAIN WILD-TYPE HIV-1 PROTEASE IN COMPLEX WITH THE SUBSTRATE P2-NC | HIV-1 PROTEASE, SPECIFICITY DESIGN, DRUG DESIGN, PROTEASE INHIBITORS, AIDS, ASPARTYL PROTEASE, HYDROLASE, HYDROLASE-HYDROLASE SUBSTRATE COMPLEX
5ivt:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV PROTEASE COMPLEXED WITH [(1S)-1-[(S)-(4- CHLOROPHENYL)-(3,5-DIFLUOROPHENYL)METHYL]-2-[[5-FLUORO-4-[2-[(2R,5S)- 5-(2,2,2-TRIFLUOROETHYLCARBAMOYLOXYMETHYL)MORPHOLIN-4-IUM-2- YL]ETHYL]PYRIDIN-1-IUM-3-YL]AMINO]-2-OXO-ETHYL]AMMONIUM | HIV, PROTEASE, HYDROLASE-INHIBITOR COMPLEX
5iy7:N (LYS348) to (TRP376) HUMAN HOLO-PIC IN THE OPEN STATE | INITIATION, RNA POLYMERASE II, HUMAN, TRANSCRIPTION, TRANSFERASE-DNA COMPLEX
5iy8:N (LYS348) to (TRP376) HUMAN HOLO-PIC IN THE INITIAL TRANSCRIBING STATE | INITIATION, RNA POLYMERASE II, HUMAN, TRANSCRIPTION, TRANSFERASE-DNA COMPLEX
4f07:C (MET118) to (PRO147) STRUCTURE OF THE STYRENE MONOOXYGENASE FLAVIN REDUCTASE (SMOB) FROM PSEUDOMONAS PUTIDA S12 | NADH-DEPENDENTFLAVIN REDUCTASE, SMOA, OXIDOREDUCTASE
5iyb:N (LYS348) to (TRP376) HUMAN CORE-PIC IN THE OPEN STATE | INITIATION, RNA POLYMERASE II, HUMAN, TRANSCRIPTION, TRANSFERASE-DNA COMPLEX
4f1s:A (PHE473) to (HIS532) CRYSTAL STRUCTURE OF HUMAN PI3K-GAMMA IN COMPLEX WITH A PYRIDYL- TRIAZINE-SULFONAMIDE INHIBITOR | PHOSPHOTRANSFERASE, LIPID KINASE, P85, TRANSFERASE-INHIBITOR COMPLEX
4f8b:B (TYR42) to (GLU74) CRYSTAL STRUCTURE OF THE COVALENT THIOIMIDE INTERMEDIATE OF UNIMODULAR NITRILE REDUCTASE QUEF | BETA BARREL, PROTEIN THIOIMIDE COMPLEX, PTERIN BINDING FOLD, TUNNEL FOLD, TRNA MODIFICATION ENZYME, 7-CYANO-7-DEAZAGUANINE, NADPH, OXIDOREDUCTASE
4f8b:C (TYR42) to (GLU74) CRYSTAL STRUCTURE OF THE COVALENT THIOIMIDE INTERMEDIATE OF UNIMODULAR NITRILE REDUCTASE QUEF | BETA BARREL, PROTEIN THIOIMIDE COMPLEX, PTERIN BINDING FOLD, TUNNEL FOLD, TRNA MODIFICATION ENZYME, 7-CYANO-7-DEAZAGUANINE, NADPH, OXIDOREDUCTASE
4faf:B (ARG57) to (GLY78) SUBSTRATE CA/P2 IN COMPLEX WITH A HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 PROTEASE VARIANT | PROTEASE, VIRAL PROTEIN
4v0i:A (ASP430) to (PHE485) WATER NETWORK DETERMINES SELECTIVITY FOR A SERIES OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS OVER PI3K-DELTA | TRANSFERASE, PI3K, KINASE SELECTIVITY
4v0i:B (ASP430) to (PHE485) WATER NETWORK DETERMINES SELECTIVITY FOR A SERIES OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS OVER PI3K-DELTA | TRANSFERASE, PI3K, KINASE SELECTIVITY
3qp0:B (ARG57) to (GLY78) HIV-1 PROTEASE (MUTANT Q7K L33I L63I) IN COMPLEX WITH A NOVEL INHIBITOR | ASPARTYL PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3qpj:B (ARG57) to (GLY78) HIV-1 PROTEASE (MUTANT Q7K L33I L63I) IN COMPLEX WITH A THREE-ARMED PYRROLIDINE-BASED INHIBITOR | ASPARTYL PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3qrm:B (ARG57) to (GLY78) HIV-1 PROTEASE (MUTANT Q7K L33I L63I) IN COMPLEX WITH A THREE-ARMED PYRROLIDINE-BASED INHIBITOR | ASPARTYL PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3qro:B (ARG57) to (GLY78) HIV-1 PROTEASE (MUTANT Q7K L33I L63I) IN COMPLEX WITH A THREE-ARMED PYRROLIDINE-BASED INHIBITOR | ASPARTYL PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3qtd:A (ASP386) to (ALA412) CRYSTAL STRUCTURE OF PUTATIVE MODULATOR OF GYRASE (PMBA) FROM PSEUDOMONAS AERUGINOSA PAO1 | PUTATIVE MODULATOR OF GYRASE (PMBA), STRUCTURAL GENOMICS, PSI- BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, GENE REGULATION
3qtd:B (ASP386) to (ALA412) CRYSTAL STRUCTURE OF PUTATIVE MODULATOR OF GYRASE (PMBA) FROM PSEUDOMONAS AERUGINOSA PAO1 | PUTATIVE MODULATOR OF GYRASE (PMBA), STRUCTURAL GENOMICS, PSI- BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, GENE REGULATION
3qtd:C (ASP386) to (ALA412) CRYSTAL STRUCTURE OF PUTATIVE MODULATOR OF GYRASE (PMBA) FROM PSEUDOMONAS AERUGINOSA PAO1 | PUTATIVE MODULATOR OF GYRASE (PMBA), STRUCTURAL GENOMICS, PSI- BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, GENE REGULATION
3qtd:D (ASP386) to (ALA412) CRYSTAL STRUCTURE OF PUTATIVE MODULATOR OF GYRASE (PMBA) FROM PSEUDOMONAS AERUGINOSA PAO1 | PUTATIVE MODULATOR OF GYRASE (PMBA), STRUCTURAL GENOMICS, PSI- BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, GENE REGULATION
4fgc:A (TYR42) to (GLU74) CRYSTAL STRUCTURE OF ACTIVE SITE MUTANT C55A OF NITRILE REDUCTASE QUEF, BOUND TO SUBSTRATE PREQ0 | BETA BARREL, PTERIN BINDING FOLD, TUNNEL FOLD, TRNA MODIFICATION ENZYME, 7-CYANO-7-DEAZAGUANINE (PREQ0) BINDING, NADPH BINDING, OXIDOREDUCTASE
4fgc:B (TYR42) to (GLU74) CRYSTAL STRUCTURE OF ACTIVE SITE MUTANT C55A OF NITRILE REDUCTASE QUEF, BOUND TO SUBSTRATE PREQ0 | BETA BARREL, PTERIN BINDING FOLD, TUNNEL FOLD, TRNA MODIFICATION ENZYME, 7-CYANO-7-DEAZAGUANINE (PREQ0) BINDING, NADPH BINDING, OXIDOREDUCTASE
3r4b:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF WILD-TYPE HIV-1 PROTEASE IN COMPLEX WITH TMC310911 | DRUG RESISTANCE, DRUG DESIGN, PROTEASE INHIBITORS, AIDS, ASPARTYL PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4fl8:B (ARG57) to (GLY78) HIV-1 PROTEASE COMPLEXED WITH GEM-DIOL-AMINE TETRAHEDRAL INTERMEDIATE | HYDROLASE, CATALYTIC MECHANISM, DRUG RESISTANCE, ASPARTIC PROTEASE
4flg:A (ARG57) to (GLY78) HIV-1 PROTEASE MUTANT I47V COMPLEXED WITH REACTION INTERMEDIATE | HYDROLASE, CATALYTIC MECHANISM, DRUG RESISTANCE, ASPARTIC PROTEASE
4fm6:A (ARG57) to (GLY78) HIV-1 PROTEASE MUTANT V32I COMPLEXED WITH REACTION INTERMEDIATE | HYDROLASE, CATALYTIC MECHANISM, DRUG RESISTANCE, ASPARTIC PROTEASE
5jfp:B (ARG57) to (GLY78) HIV-1 WILD TYPE PROTEASE WITH GRL-097-13A (A ADAMANTANE P1-LIGAND WITH BIS-THF IN P2 AND ISOBUTYLAMINE IN P1') | ADAMANTANE, HIV-1 PROTEASE INHIBITOR GRL-097-13A, DARUNAVIR, MULTIDRUG-RESISTANT, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5jfu:B (ARG57) to (GLY78) HIV-1 WILD TYPE PROTEASE WITH GRL-007-14A (A ADAMANTANE P1-LIGAND WITH BIS-THF IN P2 AND BENZYLAMINE IN P1') | ADAMANTANE, HIV-1 PROTEASE INHIBITOR GRL-007-14A, DARUNAVIR, MULTIDRUG-RESISTANT, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4frt:B (LEU143) to (GLY189) CRYSTAL STRUCTURE OF PSEUDOMONAS AERUGINOSA OCCK7 (OPDD) | BETA-BARREL, TRANSPORTER (PORIN), OUTER MEMBRANE, TRANSPORT PROTEIN
5jp0:A (TRP750) to (TRP776) BACTEROIDES OVATUS XYLOGLUCAN PUL GH3B WITH BOUND GLUCOSE | GLYCOSIDE HYDROLASE, GH3, HYDROLASE
5jp0:B (TRP750) to (TRP776) BACTEROIDES OVATUS XYLOGLUCAN PUL GH3B WITH BOUND GLUCOSE | GLYCOSIDE HYDROLASE, GH3, HYDROLASE
5jsz:B (ILE3) to (GLU31) FOLATE ECF TRANSPORTER: APO STATE | ECF TRANSPORTER, FOLATE, MEMBRANE PROTEIN, VITAMIN TRANSPORT, TRANSPORT PROTEIN
5k6l:A (PHE375) to (GLU408) STRUCTURE OF A GH3 B-GLUCOSIDASE FROM COW RUMEN METAGENOME | GLYCOSIDE HYDROLASE, METAGENOME, B-GLICOSIDASE, FUNCTIONAL FOOD, PREBIOTICS, MICROBIOTA, HYDROLASE
4gb2:B (ARG57) to (GLY78) HIV-1 PROTEASE (MUTANT Q7K L33I L63I) IN COMPLEX WITH A BICYCLIC PYRROLIDINE INHIBITOR | DIMER, ASPARTYL PROTEASE, INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4gny:A (GLY17) to (THR49) BOVINE BETA-LACTOGLOBULIN COMPLEX WITH DODECYL SULFATE | BETA PROTEIN, LIPOCALIN, MILK PROTEIN, TRANSPORT PROTEIN
5kov:A (GLN449) to (HIS485) CRYSTAL STRUCTURE OF THE HUMAN ASTROVIRUS 2 CAPSID PROTEIN SPIKE IN COMPLEX WITH A SINGLE CHAIN VARIABLE FRAGMENT OF AN ASTROVIRUS NEUTRALIZING ANTIBODY AT 3.24-A RESOLUTION | VIRAL PROTEIN, CAPSID PROTEIN, ICOSAHEDRAL VIRUS, SINGLE CHAIN VARIABLE FRAGMENT.
5kov:B (GLN449) to (HIS485) CRYSTAL STRUCTURE OF THE HUMAN ASTROVIRUS 2 CAPSID PROTEIN SPIKE IN COMPLEX WITH A SINGLE CHAIN VARIABLE FRAGMENT OF AN ASTROVIRUS NEUTRALIZING ANTIBODY AT 3.24-A RESOLUTION | VIRAL PROTEIN, CAPSID PROTEIN, ICOSAHEDRAL VIRUS, SINGLE CHAIN VARIABLE FRAGMENT.
5kov:H (GLN449) to (HIS485) CRYSTAL STRUCTURE OF THE HUMAN ASTROVIRUS 2 CAPSID PROTEIN SPIKE IN COMPLEX WITH A SINGLE CHAIN VARIABLE FRAGMENT OF AN ASTROVIRUS NEUTRALIZING ANTIBODY AT 3.24-A RESOLUTION | VIRAL PROTEIN, CAPSID PROTEIN, ICOSAHEDRAL VIRUS, SINGLE CHAIN VARIABLE FRAGMENT.
5kov:N (GLN449) to (HIS485) CRYSTAL STRUCTURE OF THE HUMAN ASTROVIRUS 2 CAPSID PROTEIN SPIKE IN COMPLEX WITH A SINGLE CHAIN VARIABLE FRAGMENT OF AN ASTROVIRUS NEUTRALIZING ANTIBODY AT 3.24-A RESOLUTION | VIRAL PROTEIN, CAPSID PROTEIN, ICOSAHEDRAL VIRUS, SINGLE CHAIN VARIABLE FRAGMENT.
5kov:S (GLN449) to (HIS485) CRYSTAL STRUCTURE OF THE HUMAN ASTROVIRUS 2 CAPSID PROTEIN SPIKE IN COMPLEX WITH A SINGLE CHAIN VARIABLE FRAGMENT OF AN ASTROVIRUS NEUTRALIZING ANTIBODY AT 3.24-A RESOLUTION | VIRAL PROTEIN, CAPSID PROTEIN, ICOSAHEDRAL VIRUS, SINGLE CHAIN VARIABLE FRAGMENT.
5kr0:B (ARG57) to (GLY78) PROTEASE E35D-APV | HIV-1 PROTEASE, E35D, SALT-BRIDGE INTERACTION, NATURAL POLYMORPHISM, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5kr1:B (LYS57) to (GLY78) PROTEASE PR5-DRV | HIV-1 PROTEASE, E35D, SALT-BRIDGE INTERACTION, NATURAL POLYMORPHISM, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1a3y:B (GLY14) to (ASP46) ODORANT BINDING PROTEIN FROM NASAL MUCOSA OF PIG | LIPOCALIN, OLFACTION
2avs:A (ARG57) to (GLY78) KINETICS, STABILITY, AND STRUCTURAL CHANGES IN HIGH RESOLUTION CRYSTAL STRUCTURES OF HIV-1 PROTEASE WITH DRUG RESISTANT MUTATIONS L24I, I50V, AND G73S | DRUG RESISTANCE, HIV-1 PROTEASE,INDINAVIR, SUBSTRATE ANALOG, NON-ACTIVE SITE MUTANTS., HYDROLASE
2avs:B (ARG57) to (GLY78) KINETICS, STABILITY, AND STRUCTURAL CHANGES IN HIGH RESOLUTION CRYSTAL STRUCTURES OF HIV-1 PROTEASE WITH DRUG RESISTANT MUTATIONS L24I, I50V, AND G73S | DRUG RESISTANCE, HIV-1 PROTEASE,INDINAVIR, SUBSTRATE ANALOG, NON-ACTIVE SITE MUTANTS., HYDROLASE
2azc:B (ARG57) to (GLY78) HIV-1 PROTEASE NL4-3 6X MUTANT | HIV, PROTEASE, INHIBITOR, TL-3, 6X, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3ekx:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF THE WILD-TYPE HIV-1 PROTEASE WITH THE INHIBITOR, NELFINAVIR | HIV PROTEASE, PROTEASE INHIBITORS, DRUG RESISTANCE, AMPRENAVIR, AIDS, PROTEASE, HYDROLASE
3el4:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF INHIBITOR SAQUINAVIR (SQV) COMPLEXED WITH THE MULTIDRUG HIV-1 PROTEASE VARIANT L63P/V82T/I84V | PROTEASE INHIBITOR, DRUG RESISTANCE, HIV PROTEASE, ENTROPY-ENTHALPY COMPENSATION, AIDS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX, PROTEASE
3el4:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF INHIBITOR SAQUINAVIR (SQV) COMPLEXED WITH THE MULTIDRUG HIV-1 PROTEASE VARIANT L63P/V82T/I84V | PROTEASE INHIBITOR, DRUG RESISTANCE, HIV PROTEASE, ENTROPY-ENTHALPY COMPENSATION, AIDS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX, PROTEASE
2b7f:D (PRO11) to (THR33) CRYSTAL STRUCTURE OF HUMAN T-CELL LEUKEMIA VIRUS PROTEASE, A NOVEL TARGET FOR ANTI-CANCER DESIGN | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3s53:A (ARG57) to (GLY78) HIV-1 PROTEASE TRIPLE MUTANTS V32I, I47V, V82I WITH ANTIVIRAL DRUG DARUNAVIR IN SPACE GROUP P212121 | DARUNAVIR,HIV/AIDS, DRUG RESISTANCE, ASPARTIC PROTEASE, MOLECULAR RECOGNITION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3fg4:B (PRO453) to (ILE480) CRYSTAL STRUCTURE OF DELTA413-417:GS I805A LOX | LIPOXYGENASE, ARICHIDONIC METABOLISM, DIOXYGENASE, FATTY ACID BIOSYNTHESIS, HEME, IRON, LIPID SYNTHESIS, LYASE, MEMBRANE, METAL- BINDING, MULTIFUNCTIONAL ENZYME, OXIDOREDUCTASE, OXYLIPIN BIOSYNTHESIS
3fg4:D (PRO453) to (ILE480) CRYSTAL STRUCTURE OF DELTA413-417:GS I805A LOX | LIPOXYGENASE, ARICHIDONIC METABOLISM, DIOXYGENASE, FATTY ACID BIOSYNTHESIS, HEME, IRON, LIPID SYNTHESIS, LYASE, MEMBRANE, METAL- BINDING, MULTIFUNCTIONAL ENZYME, OXIDOREDUCTASE, OXYLIPIN BIOSYNTHESIS
2pu9:B (ARG6) to (GLU34) CRYSTAL SRTUCTURE OF THE BINARY COMPLEX BETWEEN FERREDOXIN: THIOREDOXIN REDUCTASE AND THIOREDOXIN F | THIOREDOXIN, PROTEIN-PROTEIN COMPLEX, REDOX, IRON-SULFUR, ELECTRON TRANSPORT
2puo:B (ARG6) to (GLU34) CRYSTAL SRTUCTURE OF THE NEM MODIFIED FERREDOXIN:THIOREDOXIN REDUCTASE | THIOREDOXIN, REDOX, IRON-SULFUR, ELECTRON TRANSPORT
2pvg:B (ASP5) to (GLU34) CRYSTAL SRTUCTURE OF THE BINARY COMPLEX BETWEEN FERREDOXIN AND FERREDOXIN:THIOREDOXIN REDUCTASE | THIOREDOXIN, FERREDOXIN. REDOX, IRON-SULFUR, ELECTRON TRANSPORT
3st5:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF WILD-TYPE HIV-1 PROTEASE WITH C3-SUBSTITUTED HEXAHYDROCYCLOPENTAFURANYL URETHANE AS P2-LIGAND, GRL-0489A | ASPARTIC ACID PROTEASE, HIV-1 PROTEASE INHIBITOR GRL-0489A, C3- SUBSTITUTED HEXAHYDROCYCLOPENTAFURANYL URETHANE AS P2-LIGANDS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1cwf:A (ILE89) to (GLU120) HUMAN CYCLOPHILIN A COMPLEXED WITH 2-VAL CYCLOSPORIN | ISOMERASE-IMMUNOSUPPRESSANT COMPLEX, CYCLOPHILIN-CYCLOSPORIN COMPLEX, CYCLOSPORIN D, IMMUNOSUPPRESSANT, CYCLOPHILIN
2cen:B (ARG157) to (GLY178) P1' EXTENDED HIV-1 PROTEASE INHIBITORS ENCOMPASSING A TERTIARY ALCOHOL IN THE TRANSITION-STATE MIMICKING SCAFFOLD | HIV-1, PROTEASE, INHIBITOR, ASPARTYL PROTEASE, HYDROLASE
1d4s:B (ARG57) to (GLY78) HIV-1 PROTEASE V82F/I84V DOUBLE MUTANT/TIPRANAVIR COMPLEX | HYDROLASE, ACID PROTEASE, ASPARTYL PROTEASE
1p9u:C (SER59) to (TYR81) CORONAVIRUS MAIN PROTEINASE (3CLPRO) STRUCTURE: BASIS FOR DESIGN OF ANTI-SARS DRUGS | SARS-COV, HCOV, TGEV, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4iuj:A (CYS541) to (SER571) STRUCTURE OF POLYMERASE ACID PROTEIN (PA) FROM INFLUENZAVIRUS A INFLUENZA A VIRUS A, WILSON-SMITH/1933 (H1N1) | SSGCID, INFLUENZA, H1N1, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, TRANSCRIPTION
1dt1:A (GLY53) to (PHE72) THERMUS THERMOPHILUS CYTOCHROME C552 SYNTHESIZED BY ESCHERICHIA COLI | CYTOCHROME C552, THERMUS THERMOPHILUS, OXIDOREDUCTASE
1ebz:B (ARG157) to (GLY178) HIV-1 PROTEASE IN COMPLEX WITH THE INHIBITOR BEA388 | DIMER, PROTEIN-INHIBITOR COMPLEX, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1ec2:B (ARG157) to (GLY178) HIV-1 PROTEASE IN COMPLEX WITH THE INHIBITOR BEA428 | DIMER, PROTEIN-INHIBITOR COMPLEX, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1qg5:A (GLY17) to (THR49) HIGH RESOLUTION CRYSTAL STRUCTURE OF THE BOVINE BETA- LACTOGLOBULIN (ISOFORM A) | LIPOCALIN, ISOFORM A, TRANSPORT PROTEIN
3ttd:A (GLY494) to (ARG519) CRYSTAL STRUCTURE OF E. COLI HYPF WITH AMP-CPP AND CARBAMOYL PHOSPHATE | ZN FINGER, NUCLEOTIDE BINDING, HYDROGENASE MATURATION FACTOR, HYPE, TRANSFERASE
3tto:B (GLN2491) to (ASN2518) CRYSTAL STRUCTURE OF LEUCONOSTOC MESENTEROIDES NRRL B-1299 N- TERMINALLY TRUNCATED DEXTRANSUCRASE DSR-E IN TRICLINIC FORM | (BETA/ALPHA)8 BARREL, SUCROSE/DEXTRAN/GLUCO-OLIGOSACCHARIDE BINDING, ALPHA-1,2 BRANCHING DEXTRANSUCRASE, TRANSFERASE
3u23:A (ARG111) to (GLU139) ATOMIC RESOLUTION CRYSTAL STRUCTURE OF THE 2ND SH3 DOMAIN FROM HUMAN CD2AP (CMS) IN COMPLEX WITH A PROLINE-RICH PEPTIDE FROM HUMAN RIN3 | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, BETA- BARREL, ADAPTOR PROTEIN, PROTEIN BINDING
1fg8:D (ARG157) to (GLY178) STRUCTURAL IMPLICATIONS OF DRUG RESISTANT MUTANTS OF HIV-1 PROTEASE: HIGH RESOLUTION CRYSTAL STRUCTURES OF THE MUTANT PROTEASE/SUBSTRATE ANALOG COMPLEXES | HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1rd6:A (THR36) to (ASN70) CRYSTAL STRUCTURE OF S. MARCESCENS CHITINASE A MUTANT W167A | CHITINASE A, HYDROLASE
2f80:B (ARG57) to (GLY78) HIV-1 PROTEASE MUTANT D30N COMPLEXED WITH INHIBITOR TMC114 | PROTEIN-INHIBITOR COMPLEX, HYDROLASE
4kgq:A (ASN93) to (ARG124) CRYSTAL STRUCTURE OF A HUMAN LIGHT LOOP MUTANT IN COMPLEX WITH DCR3 | LIGHT, DCR3, TNF, TNFR, TNF14, STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW HVEM, N-GLYCOSYLATION, MEMBRANE, SECRETED PROTEIN, CYTOKINE, IFN, JELLY-ROLL FOLD, BIND TNF RECEPTOR HVEM AND LTBR, LTBR, PROTEIN STRUCTURE INITIATIVE, ATOMS-TO-ANIMALS: THE IMMUNE FUNCTION NETWORK, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, IMMUNE SYSTEM
3i3t:C (VAL480) to (GLY512) CRYSTAL STRUCTURE OF COVALENT UBIQUITIN-USP21 COMPLEX | UBIQUITIN-SPECIFIC PROTEASE ACTIVITY, HYDROLASE, UBIQUITIN BIOLOGY, STRUCTURAL GENOMICS CONSORTIUM, SGC, ACTIVATOR, CHROMATIN REGULATOR, NUCLEUS, PROTEASE, THIOL PROTEASE, TRANSCRIPTION, TRANSCRIPTION REGULATION, UBL CONJUGATION PATHWAY, ISOPEPTIDE BOND, PHOSPHOPROTEIN
1srp:A (GLY131) to (ASN155) STRUCTURAL ANALYSIS OF SERRATIA PROTEASE | HYDROLASE (METALLOPROTEASE)
2vzu:B (ASP772) to (LEU792) COMPLEX OF AMYCOLATOPSIS ORIENTALIS EXO-CHITOSANASE CSXA D469A WITH PNP-BETA-D-GLUCOSAMINE | GH2, CSXA, PNP-GLUCOSAMINE, GLYCOSIDE HYDROLASE, EXO-BETA-D-GLUCOSAMINIDASE, HYDROLASE
2vzv:A (ASP772) to (LEU792) SUBSTRATE COMPLEX OF AMYCOLATOPSIS ORIENTALIS EXO- CHITOSANASE CSXA E541A WITH CHITOSAN | EXO-BETA-D-GLUCOSAMINIDASE, GH2, CSXA, CHITOSAN, GLYCOSIDE HYDROLASE, HYDROLASE
2vzv:B (ASP772) to (LEU792) SUBSTRATE COMPLEX OF AMYCOLATOPSIS ORIENTALIS EXO- CHITOSANASE CSXA E541A WITH CHITOSAN | EXO-BETA-D-GLUCOSAMINIDASE, GH2, CSXA, CHITOSAN, GLYCOSIDE HYDROLASE, HYDROLASE
1t77:B (SER2079) to (SER2101) CRYSTAL STRUCTURE OF THE PH-BEACH DOMAINS OF HUMAN LRBA/BGL | PH-BEACH DOMAINS; VESICLE TRAFFICKING; SIGNAL TRANSDUCTION, SIGNALING PROTEIN
1t77:D (SER2079) to (SER2101) CRYSTAL STRUCTURE OF THE PH-BEACH DOMAINS OF HUMAN LRBA/BGL | PH-BEACH DOMAINS; VESICLE TRAFFICKING; SIGNAL TRANSDUCTION, SIGNALING PROTEIN
1t7j:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF INHIBITOR AMPRENAVIR IN COMPLEX WITH A MULTI-DRUG RESISTANT VARIANT OF HIV-1 PROTEASE (L63P/V82T/I84V) | HIV-1 PROTEASE, DRUG RESITANCE, THERMODYNAMICS, SUBSTRATE ENVELOPE, HYDROLASE
1hiv:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF A COMPLEX OF HIV-1 PROTEASE WITH A DIHYDROETHYLENE-CONTAINING INHIBITOR: COMPARISONS WITH MOLECULAR MODELING | ACID PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1hvl:A (ARG57) to (GLY78) INFLUENCE OF STEREOCHEMISTRY ON ACTIVITY AND BINDING MODES FOR C2 SYMMETRY-BASED DIOL INHIBITORS OF HIV-1 PROTEASE | HYDROLASE(ACID PROTEASE)
4lzu:A (GLY17) to (THR49) BOVINE BETA-LACTOGLOBULIN CRYSTALLIZED IN THE PRESENCE OF 2 MM ZINC CHLORIDE | TRANSPORT PROTEIN
2i4d:B (ARG257) to (GLY278) CRYSTAL STRUCTURE OF WT HIV-1 PROTEASE WITH GS-8373 | HIV-1 PROTEASE, HYDROLASE
1iiq:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE COMPLEXED WITH A HYDROXYETHYLAMINE PEPTIDOMIMETIC INHIBITOR | HIV PROTEASE, PEPTIDOMIMETICS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2wxo:A (ASP430) to (PHE485) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH AS5. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
2ien:B (ARG157) to (GLY178) CRYSTAL STRUCTURE ANALYSIS OF HIV-1 PROTEASE WITH A POTENT NON-PEPTIDE INHIBITOR (UIC-94017) | HIV-1 PROTEASE, DIMER, INHIBITOR, UIC-94017, TMC114, DARUNAVIR, HYDROLASE
2x05:A (ASP772) to (LEU792) INHIBITION OF THE EXO-BETA-D-GLUCOSAMINIDASE CSXA BY A GLUCOSAMINE-CONFIGURED CASTANOSPERMINE AND AN AMINO- AUSTRALINE ANALOGUE | EXO-BETA-D-GLUCOSAMINIDASE, GLYCOSIDE HYDROLASE, GH2, CSXA, HYDROLASE, GLYCOSIDASE
2x38:A (ASP430) to (PHE485) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH IC87114. | PHOSPHOINOSITIDE 3-KINASE, ISOFORM-SPECIFIC INHIBITORS, CANCER, TRANSFERASE
5ahc:A (ARG57) to (GLY78) DISUBSTITUTED BIS-THF MOIETIES AS NEW P2 LIGANDS IN NON- PEPTIDAL HIV-1 PROTEASE INHIBITORS (II) | HYDROLASE, INHIBITOR, RATIONAL DRUG DESIGN BIS-THF BIS-DIOL
5ahc:B (ARG157) to (GLY178) DISUBSTITUTED BIS-THF MOIETIES AS NEW P2 LIGANDS IN NON- PEPTIDAL HIV-1 PROTEASE INHIBITORS (II) | HYDROLASE, INHIBITOR, RATIONAL DRUG DESIGN BIS-THF BIS-DIOL
3wn7:A (LEU373) to (ASN397) CRYSTAL STRUCTURE OF KEAP1 IN COMPLEX WITH THE N-TERMINAL REGION OF THE NRF2 TRANSCRIPTION FACTOR | BETA-PROPELLER, KELCH MOTIF,DEGRON, TRANSCRIPTION
2iwm:B (VAL32) to (GLY59) PRECURSOR MUTANT CYS1SER OF PENICILLIN V ACYLASE FROM BACILLUS SPHAERICUS | ZYMOGEN, HYDROLASE, PRECURSOR, PENICILLIN, AUTOPROTEOLYSIS, ANTIBIOTIC RESISTANCE
2iwm:D (VAL32) to (GLY59) PRECURSOR MUTANT CYS1SER OF PENICILLIN V ACYLASE FROM BACILLUS SPHAERICUS | ZYMOGEN, HYDROLASE, PRECURSOR, PENICILLIN, AUTOPROTEOLYSIS, ANTIBIOTIC RESISTANCE
1vdn:A (LYS87) to (PRO118) CRYSTAL STRUCTURE OF YEAST CYCLOPHILIN A COMPLEXED WITH ACE-ALA-ALA- PRO-ALA-7-AMINO-4-METHYLCOUMARIN | BETA BARREL, ISOMERASE-ISOMERASE INHIBITOR COMPLEX, ROTAMASE
4n1r:A (ILE89) to (GLU120) STRUCTURE OF CYCLOPHILIN A IN COMPLEX WITH BENZENESULFONOHYDRAZIDE. | LIGAND COMPLEX, BETA BARREL, PROLYL CIS/TRANS ISOMERASE, CYTOSOLIC, ISOMERASE
1w5v:B (ARG57) to (GLY78) HIV-1 PROTEASE IN COMPLEX WITH FLUORO SUBSTITUTED DIOL- BASED C2-SYMMETRIC INHIBITOR | HYDROLASE/HYDROLASE INHIBITOR, HYDROLASE, DIMER, PROTEIN-INHIBITOR COMPLEX
1k4n:A (ARG79) to (PRO103) STRUCTURAL GENOMICS, PROTEIN EC4020 | STRUCTURAL GENOMICS, A NEW FOLD OF PROTEIN, PSI, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, UNKNOWN FUNCTION
1kiu:N (ALA119) to (VAL156) FIMH ADHESIN Q133N MUTANT-FIMC CHAPERONE COMPLEX WITH METHYL-ALPHA-D-MANNOSE | ADHESIN-CHAPERONE COMPLEX, MANNOSE-BOUND, CHAPERONE/CELL ADHESION COMPLEX
1kiu:P (ALA119) to (VAL156) FIMH ADHESIN Q133N MUTANT-FIMC CHAPERONE COMPLEX WITH METHYL-ALPHA-D-MANNOSE | ADHESIN-CHAPERONE COMPLEX, MANNOSE-BOUND, CHAPERONE/CELL ADHESION COMPLEX
1kjf:B (ARG57) to (GLY78) SUBSTRATE SHAPE DETERMINES SPECIFICITY OF RECOGNITION RECOGNITION FOR HIV-1 PROTEASE: ANALYSIS OF CRYSTAL STRUCTURES OF SIX SUBSTRATE COMPLEXES | P1-P6, SUBSTRATE RECOGNITION, HYDROLASE
2mly:A (ASP162) to (GLY190) NMR STRUCTURE OF E. COLI TRIGGER FACTOR IN COMPLEX WITH UNFOLDED PHOA1-150 | MOLECULAR CHAPERONE, UNFOLDED PROTEIN, CHAPERONE
1xf1:A (GLY985) to (ASP1014) STRUCTURE OF C5A PEPTIDASE- A KEY VIRULENCE FACTOR FROM STREPTOCOCCUS | C5A PEPTIDASE, HYDROLASE
1xf1:B (GLY985) to (ASP1014) STRUCTURE OF C5A PEPTIDASE- A KEY VIRULENCE FACTOR FROM STREPTOCOCCUS | C5A PEPTIDASE, HYDROLASE
2nr4:A (ILE116) to (ASN145) CRYSTAL STRUCTURE OF FMN-BOUND PROTEIN MM1853 FROM METHANOSARCINA MAZEI, PFAM DUF447 | STRUCTURAL GENOMICS, UNKNOWN FUNCTION, FLAVOPROTEIN, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
2z42:A (ASN274) to (SER307) CRYSTAL STRUTURE OF FAMILY 7 ALGINATE LYASE A1-II' FROM SPHINGOMONAS SP. A1 | ALGINATE LYASE, POLYSACCHARIDE LYASE FAMILY 7, LYASE
3kdc:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE (Q7K, L33I, L63I) IN COMPLEX WITH KNI-10074 | VIRAL PROTEIN, HYDROLASE, PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3kfs:A (ARG57) to (GLY78) HIV PROTEASE (PR) DIMER WITH INHIBITOR TL-3 BOUND AND FRAGMENT 2F4 IN THE OUTSIDE/TOP OF FLAP | HIV-1, PROTEASE, ASPARTYL PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1yhy:A (GLN644) to (GLY666) CRYSTAL STRUCTURE OF ARABIDOPSIS THALIANA ACETOHYDROXYACID SYNTHASE IN COMPLEX WITH A SULFONYLUREA HERBICIDE, METSULFURON METHYL | ACETOHYDROXYACID SYNTHASE, ACETOLACTATE SYNTHASE, HERBICIDE, SULFONYLUREA, THIAMIN DIPHOSPHATE, FAD, INHIBITOR, CYSTEINE-S- DIOXIDE, CHES, METSULFURON METHYL, TRANSFERASE
1yi0:A (GLN644) to (GLY666) CRYSTAL STRUCTURE OF ARABIDOPSIS THALIANA ACETOHYDROXYACID SYNTHASE IN COMPLEX WITH A SULFONYLUREA HERBICIDE, SULFOMETURON METHYL | ACETOHYDROXYACID SYNTHASE, ACETOLACTATE SYNTHASE, HERBICIDE, SULFONYLUREA, THIAMIN DIPHOSPHATE, FAD, INHIBITOR, CYSTEINE-S- DIOXIDE, CHES, SULFOMETURON METHYL, TRANSFERASE
3ac0:A (TRP810) to (TRP842) CRYSTAL STRUCTURE OF BETA-GLUCOSIDASE FROM KLUYVEROMYCES MARXIANUS IN COMPLEX WITH GLUCOSE | GLYCOSIDE HYDROLASE FAMILY3 BETA-GLUCOSIDASE, PA14 DOMAIN, HYDROLASE
3ac0:B (TRP810) to (TRP842) CRYSTAL STRUCTURE OF BETA-GLUCOSIDASE FROM KLUYVEROMYCES MARXIANUS IN COMPLEX WITH GLUCOSE | GLYCOSIDE HYDROLASE FAMILY3 BETA-GLUCOSIDASE, PA14 DOMAIN, HYDROLASE
3ac0:C (TRP810) to (TRP842) CRYSTAL STRUCTURE OF BETA-GLUCOSIDASE FROM KLUYVEROMYCES MARXIANUS IN COMPLEX WITH GLUCOSE | GLYCOSIDE HYDROLASE FAMILY3 BETA-GLUCOSIDASE, PA14 DOMAIN, HYDROLASE
3ac0:D (TRP810) to (TRP842) CRYSTAL STRUCTURE OF BETA-GLUCOSIDASE FROM KLUYVEROMYCES MARXIANUS IN COMPLEX WITH GLUCOSE | GLYCOSIDE HYDROLASE FAMILY3 BETA-GLUCOSIDASE, PA14 DOMAIN, HYDROLASE
1yu4:B (ALA73) to (PRO101) MAJOR TROPISM DETERMINANT U1 VARIANT | C-TYPE LECTIN, BETA SANDWICH, BETA PRISM, VARIABILITY, DIVERSITY-GENERATING RETROELEMENT, VIRAL PROTEIN
1yu4:C (ALA73) to (ALA102) MAJOR TROPISM DETERMINANT U1 VARIANT | C-TYPE LECTIN, BETA SANDWICH, BETA PRISM, VARIABILITY, DIVERSITY-GENERATING RETROELEMENT, VIRAL PROTEIN
3aos:A (PRO42) to (GLY69) CRYSTAL STRUCTURE OF JUVENILE HORMONE BINDING PROTEIN FROM SILKWORM IN COMPLEX WITH JH II | BETA-BARREL, JUVENILE HORMONE, HEMOLYMPH, HORMONE BINDING PROTEIN
1zru:A (ASN52) to (ALA75) STRUCTURE OF THE LACTOPHAGE P2 RECEPTOR BINDING PROTEIN IN COMPLEX WITH GLYCEROL | 3 DOMAINS: BETA BARREL, BETA PRISM, BETA BARREL, STRUCTURAL GENOMICS, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, VIRAL PROTEIN
1zru:C (ASN52) to (LYS77) STRUCTURE OF THE LACTOPHAGE P2 RECEPTOR BINDING PROTEIN IN COMPLEX WITH GLYCEROL | 3 DOMAINS: BETA BARREL, BETA PRISM, BETA BARREL, STRUCTURAL GENOMICS, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, VIRAL PROTEIN
3lwn:G (PHE9) to (GLY32) SHIGELLA IPGB2 IN COMPLEX WITH HUMAN RHOA, GDP AND MG2+ (COMPLEX B) | IPGB2, RHOA, GTPASE, GEF, GEF-GTPASE-COMPLEX, WXXXE, TTSS EFFECTOR PROTEIN, BACTERIAL GEF, CYTOSKELETON DYNAMICS, SIGNALING PROTEIN- RHOA-BINDING PROTEIN COMPLEX
3mtn:C (VAL480) to (GLY512) USP21 IN COMPLEX WITH A UBIQUITIN-BASED, USP21-SPECIFIC INHIBITOR | UBIQUITIN-SPECIFIC PROTEASE ACTIVITY, HYDROLASE, UBIQUITIN BIOLOGY, STRUCTURAL GENOMICS CONSORTIUM, SGC, ACTIVATOR, CHROMATIN REGULATOR, NUCLEUS, PROTEASE, THIOL PROTEASE, TRANSCRIPTION, TRANSCRIPTION REGULATION, UBL CONJUGATION PATHWAY, ISOPEPTIDE BOND, PHOSPHOPROTEIN, INHIBITOR
3ccr:K (VAL74) to (ASP99) STRUCTURE OF ANISOMYCIN RESISTANT 50S RIBOSOMAL SUBUNIT: 23S RRNA MUTATION A2488C. DENSITY FOR ANISOMYCIN IS VISIBLE BUT NOT INCLUDED IN THE MODEL. | A2488C MUTATION, 23S RRNA, LARGE RIBOSOMAL SUBUNIT, RIBOSOME
3nls:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF HIV-1 PROTEASE IN COMPLEX WITH KNI-10772 | PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3nu3:B (GLY152) to (GLY178) WILD TYPE HIV-1 PROTEASE WITH ANTIVIRAL DRUG AMPRENAVIR | ENZYME INHIBITION, ASPARTIC PROTEASE, HIV/AIDS, CONFORMATIONAL CHANGE, AMPRENAVIR, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3nu4:B (ARG157) to (GLY178) CRYSTAL STRUCTURE OF HIV-1 PROTEASE MUTANT V32I WITH ANTIVIRAL DRUG AMPRENAVIR | ENZYME INHIBITION, ASPARTIC PROTEASE, HIV/AIDS, CONFORMATIONAL CHANGE, AMPRENAVIR, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3o5k:D (ASP51) to (SER80) FK1 DOMAIN OF FKBP51, CRYSTAL FORM VIII | FK-506 BINDING DOMAIN, HSP90 COCHAPERONE, IMMUNOPHILINE, PEPTIDYL- PROLYL ISOMERASE, ISOMERASE
4cp7:B (ARG157) to (GLY178) MACROCYCLIC TRANSITION-STATE MIMICKING HIV-1 PROTEASE INHIBITORS ENCOMPASSING A TERTIARY ALCOHOL | HYDROLASE, INHIBITOR, RATIONAL DRUG DESIGN, ENZYME
3d1y:B (ARG157) to (GLY178) CRYSTAL STRUCTURE OF HIV-1 MUTANT I54V AND INHIBITOR SAQUINA | DRUG RESISTANCE, HIV-1, I54V, FLAP MUTANT, AIDS, ASPARTYL PROTEASE, CAPSID MATURATION, CAPSID PROTEIN, PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4cpq:B (ARG157) to (GLY178) MACROCYCLIC TRANSITION-STATE MIMICKING HIV-1 PROTEASE INHIBITORS ENCOMPASSING A TERTIARY ALCOHOL | HYDROLASE, INHIBITOR, RATIONAL DRUG DESIGN
3ok9:A (ARG57) to (GLY78) CRYSTAL STRUCTURE OF WILD-TYPE HIV-1 PROTEASE WITH NEW OXATRICYCLIC DESIGNED INHIBITOR GRL-0519A | ASPARTIC ACID PROTEASE, HIV-1 PROTEASE INHIBITOR GRL-0519A, OXATRICYCLIC LIGANDS, MULTIDRUG-RESISTANT HIV STRAINS, WILD-TYPE HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3dku:D (VAL6) to (ALA40) CRYSTAL STRUCTURE OF NUDIX HYDROLASE ORF153, YMFB, FROM ESCHERICHIA COLI K-1 | NUDIX HYDROLASE, ORF153, YMFB, NUCLEOSIDE TRIPHOSPHATASE
4u02:D (ILE4) to (ALA28) CRYSTAL STRUCTURE OF APO-TTHA1159 | ATP BINDING PROTEIN, ABC AMINO ACID TRANSPORTER, NUCLEOTIDE BINDING DOMAIN, TRANSPORT PROTEIN
3oxc:B (ARG157) to (GLY178) WILD TYPE HIV-1 PROTEASE WITH ANTIVIRAL DRUG SAQUINAVIR | ENZYME INHIBITION, ASPARTIC PROTEASE, HIV/AIDS, SAQUINAVIR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4dgu:A (GLN212) to (LEU240) CRYSTAL STRUCTURE OF A PUTATIVE CELL ADHESION PROTEIN (BT0320) FROM BACTEROIDES THETAIOTAOMICRON VPI-5482 AT 2.37 A RESOLUTION | CELL ADHESION PROTEIN, FIMBRIAL RELATED PROTEIN, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, CELL ADHESION
4dqc:A (GLY52) to (GLY78) CRYSTAL STRUCTURE OF (G16C/L38C) HIV-1 PROTEASE IN COMPLEX WITH DRV | HIV-1 PROTEASE, DRUG RESISTANCE, DRUG DESIGN, PROTEASE INHIBITORS, AIDS, ASPARTYL PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4dqc:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF (G16C/L38C) HIV-1 PROTEASE IN COMPLEX WITH DRV | HIV-1 PROTEASE, DRUG RESISTANCE, DRUG DESIGN, PROTEASE INHIBITORS, AIDS, ASPARTYL PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4dqh:B (ARG57) to (GLY78) CRYSTAL STRUCTURE OF (R14C/E65C) HIV-1 PROTEASE IN COMPLEX WITH DRV | HIV-1 PROTEASE, DRUG RESISTANCE, DRUG DESIGN, PROTEASE INHIBITORS, AIDS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4e43:B (ARG57) to (GLY78) HIV PROTEASE (PR) DIMER WITH ACETATE IN EXO SITE AND PEPTIDE IN ACTIVE SITE | HIV-1 PROTEASE, EXO SITE, ASPARTYL PROTEASE, FRAGMENT SCREEN, HYDROLASE
3pwm:B (ARG157) to (GLY178) HIV-1 PROTEASE MUTANT L76V WITH DARUNAVIR | HIV-1, PROTEASE, MUTATION L76V, DARUNAVIR, HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4ejl:A (ARG57) to (GLY78) APO HIV PROTEASE (PR) DIMER IN CLOSED FORM WITH FRAGMENT 1F1-N IN THE OUTSIDE/TOP OF FLAP | APO PROTEASE, ALLOSTERY, FRAGMENT BINDING, HYDROLASE
3qaa:B (ARG157) to (GLY178) HIV-1 WILD TYPE PROTEASE WITH A SUBSTITUTED BIS-TETRAHYDROFURAN INHIBITOR, GRL-044-10A | ASPARTIC ACID PROTEASE, HIV-1 PROTEASE INHIBITOR GRL-044-10A, SUBSTITUTED BIS-TETRAHYDROFURAN INHIBITOR, WILD-TYPE HIV-1 PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5iyc:N (LYS348) to (TRP376) HUMAN CORE-PIC IN THE INITIAL TRANSCRIBING STATE | INITIATION, RNA POLYMERASE II, HUMAN, TRANSCRIPTION, TRANSFERASE-DNA COMPLEX
4g9i:B (GLY505) to (TYR529) CRYSTAL STRUCTURE OF T.KODAKARENSIS HYPF | ZINC FINGER, HYDROGENASE MATURATION, ATP BINDING, CARBAMOYLATION, TRANSFERASE
5kqz:B (ARG57) to (GLY78) PROTEASE E35D-CAP2 | HIV-1 PROTEASE, E35D, SALT-BRIDGE INTERACTION, NATURAL POLYMORPHISM, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5lkh:A (SER1314) to (SER1346) CRYO-EM STRUCTURE OF THE TC TOXIN TCDA1 IN ITS PORE STATE (OBTAINED BY FLEXIBLE FITTING) | NANODISC, TOXIN, INJECTION, PORE-FORMING
5lkh:B (SER1314) to (SER1346) CRYO-EM STRUCTURE OF THE TC TOXIN TCDA1 IN ITS PORE STATE (OBTAINED BY FLEXIBLE FITTING) | NANODISC, TOXIN, INJECTION, PORE-FORMING
5lkh:C (SER1314) to (SER1346) CRYO-EM STRUCTURE OF THE TC TOXIN TCDA1 IN ITS PORE STATE (OBTAINED BY FLEXIBLE FITTING) | NANODISC, TOXIN, INJECTION, PORE-FORMING
5lkh:D (SER1314) to (SER1346) CRYO-EM STRUCTURE OF THE TC TOXIN TCDA1 IN ITS PORE STATE (OBTAINED BY FLEXIBLE FITTING) | NANODISC, TOXIN, INJECTION, PORE-FORMING
5lkh:E (SER1314) to (SER1346) CRYO-EM STRUCTURE OF THE TC TOXIN TCDA1 IN ITS PORE STATE (OBTAINED BY FLEXIBLE FITTING) | NANODISC, TOXIN, INJECTION, PORE-FORMING
5lne:B (VAL118) to (MET156) E. COLI F9 PILUS ADHESIN FMLH BOUND TO THE THOMSEN-FRIEDENREICH (TF) ANTIGEN | FIMBRIAL ADHESIN, LECTIN, O-GLYCAN, CELL ADHESION