1n7q:A (ALA757) to (GLU814) STREPTOCOCCUS PNEUMONIAE HYALURONATE LYASE W291A/W292A DOUBLE MUTANT COMPLEX WITH HYALURONAN HEXASACCHRIDE | PROTEIN MUTANT, LYASE
3rkl:A (ILE4) to (GLU50) THE CRYSTAL STRUCTURE OF A81 FROM SULFOLOBUS TURRETED ICOSAHEDRAL VIRUS | 4-HELIX BUNDLE, HYPERTHERMOPHILIC VIRAL PROTEIN, VIRAL PROTEIN
3rkl:B (ILE4) to (SER47) THE CRYSTAL STRUCTURE OF A81 FROM SULFOLOBUS TURRETED ICOSAHEDRAL VIRUS | 4-HELIX BUNDLE, HYPERTHERMOPHILIC VIRAL PROTEIN, VIRAL PROTEIN
3rkl:C (ILE4) to (SER47) THE CRYSTAL STRUCTURE OF A81 FROM SULFOLOBUS TURRETED ICOSAHEDRAL VIRUS | 4-HELIX BUNDLE, HYPERTHERMOPHILIC VIRAL PROTEIN, VIRAL PROTEIN
3rkl:D (ILE4) to (GLU50) THE CRYSTAL STRUCTURE OF A81 FROM SULFOLOBUS TURRETED ICOSAHEDRAL VIRUS | 4-HELIX BUNDLE, HYPERTHERMOPHILIC VIRAL PROTEIN, VIRAL PROTEIN
1n7r:A (ALA757) to (LEU813) STREPTOCOCCUS PNEUMONIAE HYALURONATE LYASE W291A/W292A/F343V MUTANT COMPLEX WITH HEXASACCHARIDE HYALURONAN | PROTEIN MUTANT, LYASE
3e7v:A (ILE490) to (LEU545) CRYSTAL STRUCTURE OF HUMAN HASPIN WITH A PYRAZOLO-PYRIMIDINE LIGAND | HASPIN, GERM CELL ASSOCIATED 2 (HASPIN), HAPLOID GERM CELL SPECIFIC NUCLEAR PROTEIN KINASE, SGC, STRUCTURAL GENOMICS CONSORTIUM, ATP- BINDING, CELL CYCLE, CHROMATIN REGULATOR, KINASE, MAGNESIUM, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
1a6e:A (VAL340) to (ASP401) THERMOSOME-MG-ADP-ALF3 COMPLEX | THERMOPLASMA ACIDOPHILUM, GROUP II CHAPERONIN, CCT, TRIC, PROTEIN FOLDING, ATPASE, TRANSITION STATE COMPLEX, ATP HYDROLYSIS, CHAPERONIN
2ogr:D (TYR91) to (LYS140) CRYSTAL STRUCTURE OF YELLOW FLUORESCENT PROTEIN FROM ZOANTHUS SP. AT 1.8 A RESOLUTION | GFP-LIKE PROTEINS, YELLOW FLUORESCENT PROTEIN, ZOANTHUS SP., CHROMOPHORE STRUCTURE, TETRAMER STRUCTURE, INTERMONOMER INTERFACES
3roi:A (LYS138) to (LEU179) 2.20 ANGSTROM RESOLUTION STRUCTURE OF 3-PHOSPHOSHIKIMATE 1- CARBOXYVINYLTRANSFERASE (AROA) FROM COXIELLA BURNETII | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, TRANSFERASE
2ant:I (PHE258) to (LEU299) THE 2.6 A STRUCTURE OF ANTITHROMBIN INDICATES A CONFORMATIONAL CHANGE AT THE HEPARIN BINDING SITE | SERPIN, HEPARIN, INHIBITOR
3rps:B (ARG43) to (ARG89) STRUCTURE OF HUMAN CK2ALPHA IN COMPLEX WITH THE ATP-COMPETITIVE INHIBITOR 3-(4,5,6,7-TETRABROMO-1H-BENZOTRIAZOL-1-YL)PROPAN-1-OL | EUKARYOTIC PROTEIN KINASE FOLD, ATP CK2BETA, PHOSPHORYLATION, CYTOPLASM NUCLEUS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2arq:A (LEU241) to (ILE286) HUMAN PLASMINOGEN ACTIVATOR INHIBITOR-2.[LOOP (66-98) DELETION MUTANT] COMPLEXED WITH PEPTIDE N-ACETYL-TEAAAGDGGVMTGR-OH | SERPIN, PEPTIDE BINDING, INHIBITOR, HYDROLASE INHIBITOR-PEPTIDE COMPLEX
2ol2:B (HIS224) to (LEU263) HIGH RESOLUTION STRUCTURE OF NATIVE PCI IN SPACE GROUP P21 | SERPIN, HYDROLASE INHIBITOR
3rrs:A (ASN237) to (ALA299) CRYSTAL STRUCTURE ANALYSIS OF CELLOBIOSE PHOSPHORYLASE FROM CELLULOMONAS UDA | GH94, ALPHA BARREL, CELLOBIOSE PHOSPHORYLASE, DISACCHARIDE PHOSPHORYLASE, TRANSFERASE
3rsy:A (ASN237) to (ALA299) CELLOBIOSE PHOSPHORYLASE FROM CELLULOMONAS UDA IN COMPLEX WITH SULFATE AND GLYCEROL | GH94, ALPHA BARREL, CELLOBIOSE PHOSPHORYLASE, DISACCHARIDE PHOSPHORYLASE, TRANSFERASE
3efr:A (ASN95) to (LYS169) BIOTIN PROTEIN LIGASE R40G MUTANT FROM AQUIFEX AEOLICUS IN COMPLEX WITH BIOTIN | PROTEIN BIOTIN COMPLEX, LIGASE
3efr:B (ASN95) to (LYS169) BIOTIN PROTEIN LIGASE R40G MUTANT FROM AQUIFEX AEOLICUS IN COMPLEX WITH BIOTIN | PROTEIN BIOTIN COMPLEX, LIGASE
3efy:A (LYS152) to (HIS204) STRUCTURE OF THE CYCLOMODULIN CIF FROM PATHOGENIC ESCHERICHIA COLI | CIF, CELL CYCLE, BACTERIA, VIRULENCE FACTOR, TYPE III SECRETION, E. COLI, PLASMID
3efy:B (CYS151) to (HIS204) STRUCTURE OF THE CYCLOMODULIN CIF FROM PATHOGENIC ESCHERICHIA COLI | CIF, CELL CYCLE, BACTERIA, VIRULENCE FACTOR, TYPE III SECRETION, E. COLI, PLASMID
3eg9:B (LYS726) to (CYS781) CRYSTAL STRUCTURE OF THE MAMMALIAN COPII-COAT PROTEIN SEC23/24 BOUND TO THE TRANSPORT SIGNAL SEQUENCE OF MEMBRIN | COPII COAT, VESICLE TRANSPORT, TRANSPORT SIGNAL SEQUENCE, DISEASE MUTATION, ENDOPLASMIC RETICULUM, ER-GOLGI TRANSPORT, GOLGI APPARATUS, MEMBRANE, PROTEIN TRANSPORT, TRANSPORT
1nkg:A (ASN192) to (ASP245) RHAMNOGALACTURONAN LYASE FROM ASPERGILLUS ACULEATUS | POLYSACCHARIDE LYASE, CARBOHYDRATE ACTIVE ENZYME, PECTIN, LYASE
3egx:A (ALA162) to (LEU204) CRYSTAL STRUCTURE OF THE MAMMALIAN COPII-COAT PROTEIN SEC23A/24A COMPLEXED WITH THE SNARE PROTEIN SEC22B AND BOUND TO THE TRANSPORT SIGNAL SEQUENCE OF THE SNARE PROTEIN BET1 | COPII COAT PROTEIN, VESICLE TRANSPORT, TRANSPORT SIGNAL SEQUENCE, DISEASE MUTATION, ENDOPLASMIC RETICULUM, ER-GOLGI TRANSPORT, GOLGI APPARATUS, MEMBRANE, PROTEIN TRANSPORT, TRANSPORT, PHOSPHOPROTEIN, TRANSMEMBRANE
3egx:B (ALA783) to (ALA838) CRYSTAL STRUCTURE OF THE MAMMALIAN COPII-COAT PROTEIN SEC23A/24A COMPLEXED WITH THE SNARE PROTEIN SEC22B AND BOUND TO THE TRANSPORT SIGNAL SEQUENCE OF THE SNARE PROTEIN BET1 | COPII COAT PROTEIN, VESICLE TRANSPORT, TRANSPORT SIGNAL SEQUENCE, DISEASE MUTATION, ENDOPLASMIC RETICULUM, ER-GOLGI TRANSPORT, GOLGI APPARATUS, MEMBRANE, PROTEIN TRANSPORT, TRANSPORT, PHOSPHOPROTEIN, TRANSMEMBRANE
3eh2:B (LYS460) to (CYS515) CRYSTAL STRUCTURE OF THE HUMAN COPII-COAT PROTEIN SEC24C | COPII-COAT PROTEIN, VESICLE TRANSPORT, CYTOPLASM, ENDOPLASMIC RETICULUM, ER-GOLGI TRANSPORT, GOLGI APPARATUS, MEMBRANE, PHOSPHOPROTEIN, PROTEIN TRANSPORT, TRANSPORT
3eh2:C (LYS460) to (CYS515) CRYSTAL STRUCTURE OF THE HUMAN COPII-COAT PROTEIN SEC24C | COPII-COAT PROTEIN, VESICLE TRANSPORT, CYTOPLASM, ENDOPLASMIC RETICULUM, ER-GOLGI TRANSPORT, GOLGI APPARATUS, MEMBRANE, PHOSPHOPROTEIN, PROTEIN TRANSPORT, TRANSPORT
1aiz:A (LYS18) to (GLY67) STRUCTURE OF APO-AZURIN FROM ALCALIGENES DENITRIFICANS AT 1.8 ANGSTROMS RESOLUTION | ELECTRON TRANSPORT(CADMIUM BINDING)
3rwa:H (PHE158) to (LYS205) CRYSTAL STRUCTURE OF CIRCULAR-PERMUTATED MKATE | GFP-LIKE FLUORESENT PROTEINS, MKATE, CIRCULAR PERMUTATED, FLUORESCENT PROTEIN
1ant:L (PHE258) to (LEU299) BIOLOGICAL IMPLICATIONS OF A 3 ANGSTROMS STRUCTURE OF DIMERIC ANTITHROMBIN | SERINE PROTEASE INHIBITOR
1ant:I (PHE258) to (LEU299) BIOLOGICAL IMPLICATIONS OF A 3 ANGSTROMS STRUCTURE OF DIMERIC ANTITHROMBIN | SERINE PROTEASE INHIBITOR
3eit:B (LYS198) to (ARG250) THE 2.6 ANGSTROM CRYSTAL STRUCTURE OF CHBP, THE CIF HOMOLOGUE FROM BURKHOLDERIA PSEUDOMALLEI | PAPAIN-LIKE FOLD,APAIN SUPERFAMILY, HYDROLYTIC ENZYME, UNKNOWN FUNCTION
3rzf:A (LYS18) to (LYS67) CRYSTAL STRUCTURE OF INHIBITOR OF KAPPAB KINASE BETA (I4122) | KINASE ULD, KINASE UBIQUITIN-LIKE DOMAIN SCAFFOLD HELIX, KINASE, I KAPPA B ALPHA, PHOSPHORYLATION, IMMUNE SYSTEM, SIGNALING PROTEIN
4h58:B (GLN460) to (THR507) BRAF IN COMPLEX WITH COMPOUND 3 | PROTEIN KINASE, STRUCTURE BASED DRUG DISCOVERY, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
1ath:A (PHE258) to (GLU298) THE INTACT AND CLEAVED HUMAN ANTITHROMBIN III COMPLEX AS A MODEL FOR SERPIN-PROTEINASE INTERACTIONS | HUMAN ANTITHROMBIN-III
2owb:A (ARG57) to (LEU108) STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN POLO-LIKE KINASE 1 | CATALYTIC DOMAIN, PLK1, POLO-LIKE KINASE1, KINASE, TRANSFERASE
1ntd:A (PRO71) to (THR112) STRUCTURE OF ALCALIGENES FAECALIS NITRITE REDUCTASE MUTANT M150E THAT CONTAINS ZINC | OXIDOREDUCTASE, FLAVOPROTEIN, FAD, NITRATE ASSIMILATION, OXIDOREDUCTASE (NITRIC OXIDE(A))
3emg:A (LEU377) to (LEU427) DISCOVERY AND SAR OF NOVEL 4-THIAZOLYL-2- PHENYLAMINOPYRIMIDINES AS POTENT INHIBITORS OF SPLEEN TYROSINE KINASE (SYK) | KINASE, SYK, ALTERNATIVE SPLICING, ATP-BINDING, HOST-VIRUS INTERACTION, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE, UBL CONJUGATION
3epc:R (VAL141) to (GLN188) CRYOEM STRUCTURE OF POLIOVIRUS RECEPTOR BOUND TO POLIOVIRUS TYPE 1 | CD155 STRUCTURE IMMUNOGLOBULIN SUPERFAMILY, POLIOVIRUS CAPSID JELLY ROLE, CELL ADHESION, CELL MEMBRANE, GLYCOPROTEIN, HOST-VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, RECEPTOR, SECRETED, TRANSMEMBRANE, VIRAL PROTEIN
3epf:R (ALA143) to (GLN188) CRYOEM STRUCTURE OF POLIOVIRUS RECEPTOR BOUND TO POLIOVIRUS TYPE 2 | CD155 STRUCTURE IMMUNOGLOBULIN SUPERFAMILY, POLIOVIRUS CAPSID JELLY ROLE, CELL ADHESION, CELL MEMBRANE, GLYCOPROTEIN, HOST-VIRUS INTERACTION, IMMUNOGLOBULIN DOMAIN, MEMBRANE, RECEPTOR, SECRETED, TRANSMEMBRANE, VIRAL PROTEIN
1azu:A (ASN18) to (GLY67) STRUCTURAL FEATURES OF AZURIN AT 2.7 ANGSTROMS RESOLUTION | ELECTRON TRANSPORT (COPPER BINDING)
2p3g:X (TYR63) to (ALA111) CRYSTAL STRUCTURE OF A PYRROLOPYRIDINE INHIBITOR BOUND TO MAPKAP KINASE-2 | KINASE DOMAIN, ATP-BINDING, SERINE/THREONINE KINASE, MAP KINASES, MK-2, MK2, TRANSFERASE
4hcp:A (ASN199) to (ARG250) CRYSTAL STRUCTURE OF BURKHOLDERIA PSEUDOMALLEI EFFECTOR PROTEIN CHBP IN COMPLEX WITH NEDD8 | DEAMIDASE, ALPHA/BETA/ALPHA FOLD, DEAMIDATION, NEDD8/UBIQUITIN, BACTERIAL CYTOSOL, PROTEIN BINDING
3s1y:A (TYR286) to (ASN314) AMP-C BETA-LACTAMASE (PSEUDOMONAS AERUGINOSA) IN COMPLEX WITH A BETA- LACTAMASE INHIBITOR | HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1o07:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN Q120L/Y150E MUTANT OF AMPC AND A BETA-LACTAM INHIBITOR (MXG) | ENZYME INHIBITOR COMPLEX, BETA-LACTAMASE BETA-LACTAM COMPLEX, HYDROLASE
4wz4:A (TYR286) to (ASN314) CRYSTAL STRUCTURE OF P. AERUGINOSA AMPC | BETA LACTAMASE, INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2p9k:F (PRO50) to (ALA98) CRYSTAL STRUCTURE OF BOVINE ARP2/3 COMPLEX CO-CRYSTALLIZED WITH ATP AND CROSSLINKED WITH GLUTARALDEHYDE | COMPLEX, ACTIN, WD REPEAT, STRUCTURAL PROTEIN
2p9i:F (PRO50) to (ALA98) CRYSTAL STRUCTURE OF BOVINE ARP2/3 COMPLEX CO-CRYSTALLIZED WITH ADP AND CROSSLINKED WITH GLUTERALDEHYDE | COMPLEX, WD REPEAT, ACTIN, STRUCTURAL PROTEIN
2p9l:F (PRO50) to (ALA98) CRYSTAL STRUCTURE OF BOVINE ARP2/3 COMPLEX | ACTIN, WD REPEAT, COMPLEX, STRUCTURAL PROTEIN
2bha:A (LEU352) to (VAL423) E. COLI AMINOPEPTIDASE P IN COMPLEX WITH SUBSTRATE | HYDROLASE, HYDROLASE/SUBSTRATE COMPLEX, PROLINE-SPECIFIC PEPTIDASE, SUBSTRATE COMPLEX, METALLOENZYME, PITA-BREAD FOLD, DINUCLEAR HYDROLASE
2p9n:F (PRO50) to (ALA98) CRYSTAL STRUCTURE OF BOVINE ARP2/3 COMPLEX CO-CRYSTALLIZED WITH ADP | ACTIN, WD REPEAT, COMPLEX, STRUCTURAL PROTEIN
2bhc:A (LEU352) to (VAL423) NA SUBSTITUTED E. COLI AMINOPEPTIDASE P | HYDROLASE, PROLINE-SPECIFIC PEPTIDASE, METALLOENZYME, PITA-BREAD FOLD, DINUCLEAR HYDROLASE
2p9s:F (PRO50) to (ALA98) STRUCTURE OF BOVINE ARP2/3 COMPLEX CO-CRYSTALLIZED WITH ATP/MG2+ | ACTIN, WD REPEAT, COMPLEX, STRUCTURAL PROTEIN
2p9u:F (PRO50) to (ALA98) CRYSTAL STRUCTURE OF BOVINE ARP2/3 COMPLEX CO-CRYSTALLIZED WITH AMP-PNP AND CALCIUM | ACTIN, WD REPEAT, COMPLEX, STRUCTURAL PROTEIN
2p9v:B (TYR259) to (ASP288) STRUCTURE OF AMPC BETA-LACTAMASE WITH CROSS-LINKED ACTIVE SITE AFTER EXPOSURE TO SMALL MOLECULE INHIBITOR | BETA-LACTAMASE, CROSS-LINK, HYDROLASE
2bil:B (TYR38) to (VAL96) THE HUMAN PROTEIN KINASE PIM1 IN COMPLEX WITH ITS CONSENSUS PEPTIDE PIMTIDE | PIM1, KINASE, CANCER, LEUKEMIA, TRANSFERASE
3s4a:A (ASN237) to (ALA299) CELLOBIOSE PHOSPHORYLASE FROM CELLULOMONAS UDA IN COMPLEX WITH CELLOBIOSE | GH94, ALPHA BARREL, CELLOBIOSE PHOSPHORYLASE, DISACCHARIDE PHOSPHORYLASE, TRANSFERASE
3s4a:B (ASN237) to (ALA299) CELLOBIOSE PHOSPHORYLASE FROM CELLULOMONAS UDA IN COMPLEX WITH CELLOBIOSE | GH94, ALPHA BARREL, CELLOBIOSE PHOSPHORYLASE, DISACCHARIDE PHOSPHORYLASE, TRANSFERASE
4x2j:A (ILE211) to (THR251) SELECTION OF FRAGMENTS FOR KINASE INHIBITOR DESIGN: DECORATION IS KEY | TRANSFERASE, PROTEIN KINASE, INHIBITOR COMPLEX
4x2k:A (ILE211) to (THR251) SELECTION OF FRAGMENTS FOR KINASE INHIBITOR DESIGN: DECORATION IS KEY | TRANSFERASE, PROTEIN KINASE, INHIBITOR COMPLEX
3s4c:A (ASN237) to (SER301) LACTOSE PHOSPHORYLASE IN COMPLEX WITH SULFATE | GH94, ALPHA BARREL, LACTOSE PHOSPHORYLASE, DISACCHARIDE PHOSPHORYLASE, TRANSFERASE
1bib:A (ASP176) to (GLY257) THE E. COLI BIOTIN HOLOENZYME SYNTHETASE(SLASH)BIO REPRESSOR CRYSTAL STRUCTURE DELINEATES THE BIOTIN AND DNA- BINDING DOMAINS | TRANSCRIPTION REGULATION
2bls:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE FROM ESCHERICHIA COLI | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE
2bls:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE FROM ESCHERICHIA COLI | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE
3f2a:A (ASP108) to (GLY137) CRYSTAL STRUCTURE OF HUMAN PIM-1 IN COMPLEX WITH DAPPA | POTEIN KINASE FOLD, ALTERNATIVE INITIATION, ATP-BINDING, CELL MEMBRANE, CYTOPLASM, KINASE, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3f5n:E (GLY226) to (VAL271) STRUCTURE OF NATIVE HUMAN NEUROSERPIN | NEUROSERPIN, SERPIN, CLEAVED FORM, FENIB, HUMAN, TISSUE PLASMINOGEN ACTIVATOR, HYDROLASE INHIBITOR
2brg:A (LEU15) to (LEU62) STRUCTURE-BASED DESIGN OF NOVEL CHK1 INHIBITORS: INSIGHTS INTO HYDROGEN BONDING AND PROTEIN-LIGAND AFFINITY | DRUG DESIGN, FURANOPYRIMIDINE, MOLECULAR RECOGNITION, ONCOLOGY, PYRROLOPYRIMIDINE, ATP-BINDING, CELL CYCLE, DNA DAMAGE, KINASE, NUCLEAR PROTEIN, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2brm:A (LEU15) to (LEU62) STRUCTURE-BASED DESIGN OF NOVEL CHK1 INHIBITORS: INSIGHTS INTO HYDROGEN BONDING AND PROTEIN-LIGAND AFFINITY | DRUG DESIGN, FURANOPYRIMIDINE, MOLECULAR RECOGNITION, ONCOLOGY, PYRROLOPYRIMIDINE, ATP-BINDING, CELL CYCLE, DNA DAMAGE, KINASE, NUCLEAR PROTEIN, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2brv:X (ALA757) to (LEU813) CRYSTAL STRUCTURE OF STREPTOCOCCUS PNEUMONIAE HYALURONATE LYASE FROM 70PERCENT SATURATED MALONATE. | (ALFA5/ALFA5) BARREL, CELL WALL, LYASE, PEPTIDOGLYCAN-ANCHOR
1br8:L (PHE258) to (LEU299) IMPLICATIONS FOR FUNCTION AND THERAPY OF A 2.9A STRUCTURE OF BINARY-COMPLEXED ANTITHROMBIN | SERPINS, ANTITHROMBIN, BINARY-COMPLEX, CRYSTAL STRUCTURE, HEPARIN, POLYMERISATION, THROMBOSIS, EMPHYSEMA, CIRRHOSIS, BLOOD CLOTTING
1br8:I (ARG259) to (LEU299) IMPLICATIONS FOR FUNCTION AND THERAPY OF A 2.9A STRUCTURE OF BINARY-COMPLEXED ANTITHROMBIN | SERPINS, ANTITHROMBIN, BINARY-COMPLEX, CRYSTAL STRUCTURE, HEPARIN, POLYMERISATION, THROMBOSIS, EMPHYSEMA, CIRRHOSIS, BLOOD CLOTTING
3s87:A (LYS423) to (ILE485) STRUCTURE OF YEAST RIBONUCLEOTIDE REDUCTASE 1 WITH DGTP AND ADP | DNTP REGULATION, ALLOSTERY, OXIDOREDUCTASE
3f7z:A (ILE62) to (LEU104) X-RAY CO-CRYSTAL STRUCTURE OF GLYCOGEN SYNTHASE KINASE 3BETA IN COMPLEX WITH AN INHIBITOR | ENZYME, PROTEIN KINASE, INHIBITOR CO-CRYSTAL STRUCTURE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
3f7z:B (ILE62) to (LEU104) X-RAY CO-CRYSTAL STRUCTURE OF GLYCOGEN SYNTHASE KINASE 3BETA IN COMPLEX WITH AN INHIBITOR | ENZYME, PROTEIN KINASE, INHIBITOR CO-CRYSTAL STRUCTURE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
3s8c:A (LYS423) to (ASN488) STRUCTURE OF YEAST RIBONUCLEOTIDE REDUCTASE 1 R293A WITH AMPPNP AND CDP | DNTP REGULATION, ALLOSTERY, OXIDOREDUCTASE
4x7q:A (LEU38) to (VAL90) PIM2 KINASE IN COMPLEX WITH COMPOUND 1S | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2btj:C (TYR87) to (LYS134) FLUORESCENT PROTEIN EOSFP - RED FORM | PHOTO-INDUCED PROTEIN CLEAVAGE, GREEN-TO-RED CONVERSION, FLUORESCENT PROTEIN, LUMINESCENT PROTEIN
4hrv:A (VAL109) to (SER178) CRYSTAL STRUCTURE OF LIPOPROTEIN GNA1162 FROM NEISSERIA MENINGITIDIS | DUF799, LIPID BINDING PROTEIN
4hrv:B (TYR117) to (SER178) CRYSTAL STRUCTURE OF LIPOPROTEIN GNA1162 FROM NEISSERIA MENINGITIDIS | DUF799, LIPID BINDING PROTEIN
3say:A (ILE62) to (LEU104) CRYSTAL STRUCTURE OF HUMAN GLYCOGEN SYNTHASE KINASE 3 BETA (GSK3B) IN COMPLEX WITH INHIBITOR 142 | KINASE, ATP HYDROLYSIS, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4xba:A (ILE52) to (VAL84) HNT3 | GMP, NUCLEOTIDYL TRANSFERASE, HYDROLASE
1byg:A (GLY202) to (ALA237) KINASE DOMAIN OF HUMAN C-TERMINAL SRC KINASE (CSK) IN COMPLEX WITH INHIBITOR STAUROSPORINE | PROTEIN KINASE, C-TERMINAL SRC KINASE, PHOSPHORYLATION, STAUROSPORINE, TRANSFERASE
4hvi:A (LEU828) to (LEU878) JAK3 KINASE DOMAIN IN COMPLEX WITH 2-CYCLOPROPYL-5H-PYRROLO[2,3- B]PYRAZINE-7-CARBOXYLIC ACID ((R)-1-METHYL-2-OXO-2-PIPERIDIN-1-YL- ETHYL)-AMIDE | KINASE-INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4hvm:B (SER382) to (ASP457) CRYSTAL STRUCTURE OF TALLYSOMYCIN BIOSYNTHESIS PROTEIN TLMII | PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, NATURAL PRODUCT BIOSYNTHESIS, NATPRO, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NONRIBOSOMAL PEPTIDE SYNTHETASES, BIOSYNTHETIC PROTEIN, GO.119753
2bwu:A (LEU352) to (VAL423) ASP271ALA ESCHERICHIA COLI AMINOPEPTIDASE P | AMINOPEPTIDASE P, METALLOENZYME, 'PITA-BREAD' ENZYME, PROLINE-SPECIFIC ENZYME, MANGANESE ENZYME, HYDROLASE
2pl0:A (LEU251) to (GLN294) LCK BOUND TO IMATINIB | KINASE PHOSPHORYLATION, TRANSFERASE
4xd7:H (PHE67) to (ASN125) STRUCTURE OF THERMOPHILIC F1-ATPASE INHIBITED BY EPSILON SUBUNIT | F1-ATPASE, ATP SYNTHASE, ROTARY MOTOR PROTEIN, ROTATIONAL CATALYSIS, BACILLUS PS3, THERMOPHILIC, HYDROLASE
1c3b:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE FROM E. COLI COMPLEXED WITH INHIBITOR, BENZO(B) THIOPHENE-2-BORONIC ACID (BZB) | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, HYDROLASE
1c3b:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE FROM E. COLI COMPLEXED WITH INHIBITOR, BENZO(B) THIOPHENE-2-BORONIC ACID (BZB) | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, HYDROLASE
1c4f:A (TYR92) to (GLY134) GREEN FLUORESCENT PROTEIN S65T AT PH 4.6 | GREENFLUORESCENT PROTEIN, BIOLUMINESCENCE, PHOTOACTIVE PROTEIN, FLUORESCENT TAG, PH TITRATION, SIGNALING PROTEIN
4xg4:A (LEU377) to (LEU427) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4xg9:A (LEU377) to (GLN425) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4xg9:B (LEU377) to (GLN425) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
2ppa:C (PRO71) to (THR112) ANAEROBICALLY MANIPULATED WILD TYPE OXIDIZED AFNIR BOUND TO NITROUS OXIDE | NITRITE REDUCTASE, DENITRIFICATION, NITROUS OXIDE, BACTERIA, OXIDOREDUCTASE
4i2v:A (LEU44) to (LEU84) X-RAY STRUCTURE OF THE UNLIGANDED URIDINE PHOSPHORYLASE FROM YERSINIA PSEUDOTUBERCULOSIS AT 2.12A RESOLUTION | ROSSMANN FOLD, TRANSFERASE, PYRIMIDINE METABOLISM
4i41:A (ASP108) to (ARG136) CRYSTAL STRUCTURE OF HUMAN SER/THR KINASE PIM1 IN COMPLEX WITH MITOXANTRONE | SER/THR KINASE, MITOXANTRONE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3fkv:B (TYR259) to (ASP288) AMPC K67R MUTANT COMPLEXED WITH BENZO(B)THIOPHENE-2-BORONIC ACID (BZB) | AMPC, K67R, BETA-LACTAMASE, GENERAL BASE, ANTIBIOTIC RESISTANCE, PERIPLASM, HYDROLASE
3fkw:B (TYR259) to (ASP288) AMPC K67R MUTANT APO STRUCTURE | AMPC, K67R, BETA-LACTAMASE, GENERAL BASE, ANTIBIOTIC RESISTANCE, PERIPLASM, HYDROLASE
4xjx:A (ASN132) to (SER184) STRUCTURE OF MUTANT (E165H) OF THE HSDR SUBUNIT OF THE ECOR124I RESTRICTION ENZYME IN COMPLEX WITH ATP | RESTRICTION ENZYME, ATP, HYDROLASE
4xjx:B (ASN132) to (ILE180) STRUCTURE OF MUTANT (E165H) OF THE HSDR SUBUNIT OF THE ECOR124I RESTRICTION ENZYME IN COMPLEX WITH ATP | RESTRICTION ENZYME, ATP, HYDROLASE
2pu4:A (TYR259) to (ASP288) AMPC BETA-LACAMASE WITH BOUND COVALENT OXADIAZOLE INHIBITOR | AMPC BETA-LACTAMASE OXADIAZOLE, HYDROLASE
2pu4:B (TYR259) to (ASP288) AMPC BETA-LACAMASE WITH BOUND COVALENT OXADIAZOLE INHIBITOR | AMPC BETA-LACTAMASE OXADIAZOLE, HYDROLASE
3fmd:A (ILE490) to (GLU548) CRYSTAL STRUCTURE OF HUMAN HASPIN WITH AN ISOQUINOLINE LIGAND | HASPIN, GERM CELL ASSOCIATED 2, HAPLOID GERM CELL SPECIFIC NUCLEAR PROTEIN KINASE, ATP-BINDING, CELL CYCLE, CHROMATIN REGULATOR, KINASE, MAGNESIUM, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE,STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
1onh:A (TYR262) to (ASP291) GC1 BETA-LACTAMASE WITH A PENEM INHIBITOR | MIXED ALPHA/BETA, CEPHALOSPORINASE, INHIBITION, CLASS C BETA- LACTAMASE, HYDROLASE
4xli:B (THR289) to (LYS337) CRYSTAL STRUCTURE OF ABL2/ARG KINASE IN COMPLEX WITH DASATINIB | TRANSFERASE, INHIBITOR, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4i6q:A (LEU828) to (LEU878) JAK3 KINASE DOMAIN IN COMPLEX WITH 2-PHENOXY-5H-PYRROLO[2,3- B]PYRAZINE-7-CARBOXYLIC ACID ((S)-1-CYCLOPROPYL-ETHYL)-AMIDE | KINASE-INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2pxs:A (TYR91) to (LYS140) CRYSTAL STRUCTURE OF N66D MUTANT OF GREEN FLUORESCENT PROTEIN FROM ZOANTHUS SP. AT 2.2 A RESOLUTION (MATURE STATE) | ZOANTHUS FAMILY, RED FLUORESCENT PROTEIN, GREEN FLUORESCENT PROTEIN, CHROMOPHORE STRUCTURE
2pxw:A (TYR91) to (LYS140) CRYSTAL STRUCTURE OF N66D MUTANT OF GREEN FLUORESCENT PROTEIN FROM ZOANTHUS SP. AT 2.4 A RESOLUTION (TRANSITION STATE) | ZOANTHUS FAMILY, RED FLUORESCENT PROTEIN, GREEN FLUORESCENT PROTEIN, CHROMOPHORE STRUCTURE
1ckj:B (GLY19) to (GLN63) CASEIN KINASE I DELTA TRUNCATION MUTANT CONTAINING RESIDUES 1-317 COMPLEX WITH BOUND TUNGSTATE | PROTEIN KINASE, PHOSPHOTRANSFERASE
3sp4:A (ILE52) to (VAL84) CRYSTAL STRUCTURE OF APRATAXIN ORTHOLOG HNT3 FROM SCHIZOSACCHAROMYCES POMBE | HIT DOMAIN, ZINC FINGER, DNA-BINDING PROTEIN, DNA DEADENYLASE, HYDROLASE
3fqe:A (LEU377) to (GLN425) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH YM193306 | SYK, SPLEEN TYPROSINE KINASE, KINASE INHIBITOR, PYRIMIDINE-5- CARBOXAMIDE, ATP-BINDING, HOST-VIRUS INTERACTION, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3spd:A (ILE52) to (VAL84) CRYSTAL STRUCTURE OF APRATAXIN ORTHOLOG HNT3 IN COMPLEX WITH DNA | HIT DOMAIN, ZINC FINGER, DNA DEADENYLASE, DNA BINDING, HYDROLASE-DNA COMPLEX
3spd:B (ILE52) to (VAL84) CRYSTAL STRUCTURE OF APRATAXIN ORTHOLOG HNT3 IN COMPLEX WITH DNA | HIT DOMAIN, ZINC FINGER, DNA DEADENYLASE, DNA BINDING, HYDROLASE-DNA COMPLEX
3spd:C (ILE52) to (VAL84) CRYSTAL STRUCTURE OF APRATAXIN ORTHOLOG HNT3 IN COMPLEX WITH DNA | HIT DOMAIN, ZINC FINGER, DNA DEADENYLASE, DNA BINDING, HYDROLASE-DNA COMPLEX
3spd:D (ILE52) to (VAL84) CRYSTAL STRUCTURE OF APRATAXIN ORTHOLOG HNT3 IN COMPLEX WITH DNA | HIT DOMAIN, ZINC FINGER, DNA DEADENYLASE, DNA BINDING, HYDROLASE-DNA COMPLEX
3frk:B (HIS162) to (TYR214) X-RAY STRUCTURE OF QDTB FROM T. THERMOSACCHAROLYTICUM IN COMPLEX WITH A PLP:TDP-3-AMINOQUINOVOSE ALDIMINE | AMINOTRANSFERASE, SUGAR-MODIFICATION, NATURAL PORDUCT
4iaa:A (ASP108) to (GLU135) CRYSTAL STRUCTURE OF SER/THR KINASE PIM1 IN COMPLEX WITH THIORIDAZINE | PIM1 KINASE/ONCOGENE/THIORIDAZINE, SER/THR KINASE, THIORIDAZINE, TRANSFERASE
1ova:C (ARG228) to (ILE266) CRYSTAL STRUCTURE OF UNCLEAVED OVALBUMIN AT 1.95 ANGSTROMS RESOLUTION | SERPIN
4ifc:A (TYR690) to (ASP743) CRYSTAL STRUCTURE OF ADP-BOUND HUMAN PRPF4B KINASE DOMAIN | KINASE, TRANSFERASE
4ifc:B (TYR690) to (ASP743) CRYSTAL STRUCTURE OF ADP-BOUND HUMAN PRPF4B KINASE DOMAIN | KINASE, TRANSFERASE
3ssa:A (ASP125) to (ARG165) CRYSTAL STRUCTURE OF SUBUNIT B MUTANT N157T OF THE A1AO ATP SYNTHASE | HYDROLASE, ATP BINDING
2c9i:C (GLY87) to (LYS135) STRUCTURE OF THE FLUORESCENT PROTEIN ASFP499 FROM ANEMONIA SULCATA | FLUORESCENT PROTEIN, BETA-BARREL, BIOLUMINESCENCE, LUMINESCENCE, LUMINESCENT PROTEIN
2c9i:E (GLY87) to (LYS135) STRUCTURE OF THE FLUORESCENT PROTEIN ASFP499 FROM ANEMONIA SULCATA | FLUORESCENT PROTEIN, BETA-BARREL, BIOLUMINESCENCE, LUMINESCENCE, LUMINESCENT PROTEIN
2c9i:H (GLY87) to (LYS135) STRUCTURE OF THE FLUORESCENT PROTEIN ASFP499 FROM ANEMONIA SULCATA | FLUORESCENT PROTEIN, BETA-BARREL, BIOLUMINESCENCE, LUMINESCENCE, LUMINESCENT PROTEIN
2ccw:A (LYS18) to (GLY67) CRYSTAL STRUCTURE OF AZURIN II AT ATOMIC RESOLUTION (1.13 ANGSTROM) | ELECTRON TRANSPORT (CUPROPROTEIN), AZURIN II, ALCALIGENES XYLOSOXIDANS, ELECTRON TRANSFER, CUPREDOXIN, ELECTRON TRANSPORT, CUPROPROTEIN, COPPER, METAL- BINDING, PERIPLASMIC
2q9m:A (TYR259) to (ASP288) 4-SUBSTITUTED TRINEMS AS BROAD SPECTRUM-LACTAMASE INHIBITORS: STRUCTURE-BASED DESIGN, SYNTHESIS AND BIOLOGICAL ACTIVITY | BETA-LACTAMASE INHIBITOR, TRICYCLIC CARBAPENEM, HYDROLASE
4iij:C (GLY43) to (GLY81) CRYSTAL STRUCTURE OF TUBULIN-STATHMIN-TTL-APO COMPLEX | ALPHA-TUBULIN, BETA-TUBULIN, LIGASE, GTPASE, MICROTUBULE, STATHMIN, CELL CYCLE
4iir:B (TYR690) to (ASP743) CRYSTAL STRUCTURE OF AMPPNP-BOUND HUMAN PRPF4B KINASE DOMAIN | KINASE, TRANSFERASE
4ikf:A (GLN27) to (LEU64) PFV INTASOME WITH INHIBITOR MB-76 | INTEGRASE ZINC BINDING, CORE AND DNA-BINDING DOMAINS, DNA INTEGRATION, INHIBITOR, NUCLEUS, VIRAL PROTEIN-DNA-INHIBITOR COMPLEX, ENDONUCLEASE, NUCLEOTIDYLTRANSFERASE, RECOMBINATION, HHCC MOTIF, DDE MOTIF
2qg7:B (SER110) to (ASN165) PLASMODIUM VIVAX ETHANOLAMINE KINASE PV091845 | MALARIA, ETHANOLAMINE KINASE, PV091845, SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSFERASE
2qg7:E (SER110) to (ASN165) PLASMODIUM VIVAX ETHANOLAMINE KINASE PV091845 | MALARIA, ETHANOLAMINE KINASE, PV091845, SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSFERASE
1pcs:A (SER17) to (LEU55) THE 2.15 A CRYSTAL STRUCTURE OF A TRIPLE MUTANT PLASTOCYANIN FROM THE CYANOBACTERIUM SYNECHOCYSTIS SP. PCC 6803 | ELECTRON TRANSPORT, PLASTOCYANIN
3g6g:B (GLU270) to (LYS315) EQUALLY POTENT INHIBITION OF C-SRC AND ABL BY COMPOUNDS THAT RECOGNIZE INACTIVE KINASE CONFORMATIONS | CANCER, IMATINIB RESISTANCE, DSA COMPOUNDS, KINASE, DFG-ASP-OUT, ATP- BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE
2cnv:A (ALA16) to (LEU68) SAICAR-SYNTHASE FROM SACCHAROMYCES CEREVISIAE COMPLEXED SAICAR | LIGASE, PHOSPHORIBOSYLAMINOIMIDAZOLESUCCINOCARBOXAMIDE (SAICAR) SYN LIGASE, SYNTHETASE, ACETYLATION, ATPBINDING PROTEIN, PURINE BIOSYNTHESIS
3t2c:A (ARG203) to (ALA256) FRUCTOSE-1,6-BISPHOSPHATE ALDOLASE/PHOSPHATASE FROM THERMOPROTEUS NEUTROPHILUS, DHAP-BOUND FORM | (BETA/ALPHA)8 TIM BARREL, FBP, F6P, DHAP, GAP, PHOSPHORYLATION, LYASE, HYDROLASE
3t2b:A (ARG203) to (ALA256) FRUCTOSE-1,6-BISPHOSPHATE ALDOLASE/PHOSPHATASE FROM THERMOPROTEUS NEUTROPHILUS, LIGAND FREE | (BETA/ALPHA)8 TIM BARREL, FBP, F6P, DHAP, GAP, PHOSPHORYLATION, LYASE, HYDROLASE
3t2e:A (LYS204) to (ALA256) FRUCTOSE-1,6-BISPHOSPHATE ALDOLASE/PHOSPHATASE FROM THERMOPROTEUS NEUTROPHILUS, F6P-BOUND FORM | (BETA/ALPHA)8 TIM BARREL, FBP, F6P, DHAP, GAP, PHOSPHORYLATION, LYASE, HYDROLASE
3t2g:A (LYS204) to (ALA254) FRUCTOSE-1,6-BISPHOSPHATE ALDOLASE/PHOSPHATASE FROM THERMOPROTEUS NEUTROPHILUS, Y229F VARIANT WITH DHAP | (BETA/ALPHA)8 TIM BARREL, FBP, F6P, DHAP, GAP, PHOSPHORYLATION, LYASE, HYDROLASE
2cqs:A (ASP237) to (ARG297) CRYSTAL STRUCTURE OF CELLVIBRIO GILVUS CELLOBIOSE PHOSPHORYLASE CRYSTALLIZED FROM AMMONIUM SULFATE | BETA-SANDWICH, (ALPHA/ALPHA)6 BARREL, TRANSFERASE
2qlr:C (ALA345) to (LEU425) CRYSTAL STRUCTURE OF HUMAN KYNURENINE AMINOTRANSFERASE II | ALPHA & BETA PROTEIN, PLP-DEPENDENT TRANSFERASE, AMINOTRANSFERASE, MITOCHONDRION, MULTIFUNCTIONAL ENZYME, PYRIDOXAL PHOSPHATE, TRANSIT PEPTIDE, TRANSFERASE
4iq6:B (GLY63) to (LEU104) GSK-3BETA WITH INHIBITOR 6-CHLORO-N-CYCLOHEXYL-4-(1H-PYRROLO[2,3- B]PYRIDIN-3-YL)PYRIDIN-2-AMINE | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2qmj:A (ALA240) to (GLY282) CRYSTRAL STRUCTURE OF THE N-TERMINAL SUBUNIT OF HUMAN MALTASE- GLUCOAMYLASE IN COMPLEX WITH ACARBOSE | HYDROLASE, GLYCOSYL HYDROLASE FAMILY 31, GLYCOPROTEIN, GLYCOSIDASE, MEMBRANE, MULTIFUNCTIONAL ENZYME, SIGNAL-ANCHOR, SULFATION, TRANSMEMBRANE
1pi4:B (TYR259) to (ASP288) STRUCTURE OF N289A MUTANT OF AMPC IN COMPLEX WITH SM3, A PHENYLGLYCLBORONIC ACID BEARING THE CEPHALOTHIN R1 SIDE CHAIN | CRYSTAL STRUCTURE, ENZYME INHIBITOR COMPLEX, BETA-LACTAMASE, HYDROLASE
1pi5:B (TYR259) to (ASP288) STRUCTURE OF N289A MUTANT OF AMPC IN COMPLEX WITH SM2, CARBOXYPHENYLGLYCYLBORONIC ACID BEARING THE CEPHALOTHIN R1 SIDE CHAIN | CRYSTAL STRUCTURE, ENZYME INHIBITOR COMPLEX, BETA-LACTAMASE, HYDROLASE
1pj5:A (PHE632) to (GLY677) CRYSTAL STRUCTURE OF DIMETHYLGLYCINE OXIDASE OF ARTHROBACTER GLOBIFORMIS IN COMPLEX WITH ACETATE | CHANNELLING, FAD BINDING, FOLATE BINDING, AMINE OXIDASE, OXIDOREDUCTASE
1pj6:A (PHE632) to (GLY677) CRYSTAL STRUCTURE OF DIMETHYLGLYCINE OXIDASE OF ARTHROBACTER GLOBIFORMIS IN COMPLEX WITH FOLIC ACID | CHANNELLING, FOLATE BINDING, FAD BINDING, AMINE OXIDATION, OXIDOREDUCTASE
1pj7:A (PHE632) to (GLY677) STRUCTURE OF DIMETHYLGLYCINE OXIDASE OF ARTHROBACTER GLOBIFORMIS IN COMPLEX WITH FOLINIC ACID | CHANNELLING, FAD BINDING, FOLINIC ACID, FOLATE BINDING, AMINE OXIDATION, OXIDOREDUCTASE
1dmr:A (GLY6) to (SER48) OXIDIZED DMSO REDUCTASE FROM RHODOBACTER CAPSULATUS | OXIDOREDUCTASE, REDUCTASE, DMSO, MOLYBDOPTERIN
4xux:A (TYR279) to (ASP308) STRUCTURE OF AMPC BOUND TO RPX-7009 AT 1.75 A | HYDROLASE-ANTIBIOTIC COMPLEX
4xv2:B (GLN461) to (ASN500) B-RAF KINASE V600E ONCOGENIC MUTANT IN COMPLEX WITH DABRAFENIB | B-RAF, BRAF, PROTO-ONCOGENE, V600E, KINASE, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4ivb:B (GLY882) to (LEU932) JAK1 KINASE (JH1 DOMAIN) IN COMPLEX WITH THE INHIBITOR TRANS-4-{2- [(1R)-1-HYDROXYETHYL]IMIDAZO[4,5-D]PYRROLO[2,3-B]PYRIDIN-1(6H)- YL}CYCLOHEXANECARBONITRILE | PROTEIN KINASE, PHOSPHOTRANSFER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2qt8:A (ASN86) to (GLY157) COPROPORPHYRINOGEN III OXIDASE FROM LEISHMANIA MAJOR | HEME METABOLISM, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA CONSORTIUM, SGPP, HEME BIOSYNTHESIS, OXIDOREDUCTASE, PORPHYRIN BIOSYNTHESIS
4ix5:B (GLY179) to (ASN226) CRYSTAL STRUCTURE OF A STT7 HOMOLOG FROM MICROMONAS ALGAE IN COMPLEX WITH AMP-PNP | PROTEIN KINASE, CANONICAL PROTEIN KINASE FOLD, ATP BINDING, TRANSFERASE
1dyz:A (LYS18) to (GLY67) OXIDISED AZURIN II FROM ALCALIGENES XYLOSOXIDANS | ELECTRON TRANSPORT, CUPREDOXIN, CUPROPROTEIN
1dz0:A (LYS18) to (GLY67) REDUCED AZURIN II FROM ALCALIGENES XYLOSOXIDANS | ELECTRON TRANSPORT, CUPREDOXIN, CUPROPROTEIN
1dzg:I (PHE258) to (GLU298) N135Q-S380C-ANTITHROMBIN-III | BLOOD CLOTTING, SERPIN
1e05:L (PHE258) to (LEU299) PLASMA ALPHA ANTITHROMBIN-III | BLOOD CLOTTING, SERPIN
1e18:A (GLY6) to (SER48) TUNGSTEN-SUSBSTITUTED DMSO REDUCTASE FROM RHODOBACTER CAPSULATUS | OXIDOREDUCTASE, REDUCTASE, DMSO, MOLYBDOPTERIN, MOLYBDENUM, TUNGSTEN
4j1r:A (ILE62) to (LEU104) CRYSTAL STRUCTURE OF GSK3B IN COMPLEX WITH INHIBITOR 15R | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, KINASE, PHOSPHORYLATION, TRANSFERASE
4j1r:B (ILE62) to (LEU104) CRYSTAL STRUCTURE OF GSK3B IN COMPLEX WITH INHIBITOR 15R | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, KINASE, PHOSPHORYLATION, TRANSFERASE
4j1r:C (ILE62) to (LEU104) CRYSTAL STRUCTURE OF GSK3B IN COMPLEX WITH INHIBITOR 15R | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, KINASE, PHOSPHORYLATION, TRANSFERASE
4j1r:D (ILE62) to (LEU104) CRYSTAL STRUCTURE OF GSK3B IN COMPLEX WITH INHIBITOR 15R | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, KINASE, PHOSPHORYLATION, TRANSFERASE
3tb9:A (LYS423) to (ASN488) STRUCTURE OF YEAST RIBONUCLEOTIDE REDUCTASE 1 Q288A WITH AMPPNP AND CDP | EUKARYOTIC, RIBONUCLEOTIDE REDUCTASE, DNTP REGULATION, OXIDOREDUCTASE
3gqb:B (GLN129) to (ARG169) CRYSTAL STRUCTURE OF THE A3B3 COMPLEX FROM V-ATPASE | A3B3, V-ATPASE, ATP SYNTHESIS, ATP-BINDING, HYDROGEN ION TRANSPORT, HYDROLASE, ION TRANSPORT, NUCLEOTIDE-BINDING, TRANSPORT
3gqm:B (LYS132) to (ARG184) CRYSTAL STRUCTURE OF CELL INHIBITING FACTOR (CIF) FROM BURKHOLDERIA PSEUDOMALLEI (CIFBP) | CELL INHIBITING FACTOR, CIF, CIFBP, UNKNOWN FUNCTION
3gqz:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT-BASED INHIBITOR | HYDROLASE, LACTAMASE, FRAGMENT, ANTIBIOTIC RESISTANCE, PERIPLASM, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
3gr2:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT-BASED INHIBITOR | HYDROLASE, AMPC, LACTAMASE, FRAGMENT, ANTIBIOTIC RESISTANCE, PERIPLASM, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
3grj:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT-BASED INHIBITOR | HYDROLASE/HYDROLASE INHIBITOR, ANTIBIOTIC RESISTANCE, HYDROLASE, PERIPLASM
1e61:A (GLY6) to (SER48) OXIDIZED DMSO REDUCTASE EXPOSED TO HEPES - STRUCTURE II BUFFER | OXIDOREDUCTASE, REDUCTASE, DMSO, MOLYBDOPTERIN
1e61:C (GLY6) to (SER48) OXIDIZED DMSO REDUCTASE EXPOSED TO HEPES - STRUCTURE II BUFFER | OXIDOREDUCTASE, REDUCTASE, DMSO, MOLYBDOPTERIN
3gsi:A (PHE632) to (GLY677) CRYSTAL STRUCTURE OF D552A DIMETHYLGLYCINE OXIDASE MUTANT OF ARTHROBACTER GLOBIFORMIS IN COMPLEX WITH TETRAHYDROFOLATE | OXIDOREDUCTASE, CHANNELLING, FAD BINDING, FOLINIC ACID, FOLATE BINDING, AMINE OXIDATION
2dd9:B (TYR81) to (ASP128) A MUTANT OF GFP-LIKE PROTEIN FROM CHIRIDIUS POPPEI | GFP-LIKE PROTEIN, FLUORESCENT PROTEIN, LUMINESCENT PROTEIN
3gtc:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT-BASED INHIBITOR | HYDROLASE, ANTIBIOTIC RESISTANCE, PERIPLASM, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
3gtc:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT-BASED INHIBITOR | HYDROLASE, ANTIBIOTIC RESISTANCE, PERIPLASM, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
4j71:A (ILE62) to (LEU104) CRYSTAL STRUCTURE OF GSK3B IN COMPLEX WITH INHIBITOR 1R | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, KINASE, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
1q2q:A (TYR262) to (ASP291) ENTEROBACTER CLOACAE GC1 CLASS C BETA-LACTAMASE COMPLEXED WITH PENEM WAY185229 | HYDROLASE, INHIBITION, BETA-LACTAM ANTIBIOTICS, DRUG DESIGN
3tgw:A (ASP125) to (ARG165) CRYSTAL STRUCTURE OF SUBUNIT B MUTANT H156A OF THE A1AO ATP SYNTHASE | HYDROLASE, ATP SYNTHESIS, HYDROGEN ION TRANSPORT
3tgx:C (ASP3) to (GLU42) IL-21:IL21R COMPLEX | CLASS I CYTOKINE, CLASS I CYTOKINE RECEPTOR, SUGARBRIDGE, FIBRONECTIN DOMAIN, SIGNALING, CYTOKINE-CYTOKINE RECEPTOR COMPLEX
3tgx:K (ASP3) to (GLU42) IL-21:IL21R COMPLEX | CLASS I CYTOKINE, CLASS I CYTOKINE RECEPTOR, SUGARBRIDGE, FIBRONECTIN DOMAIN, SIGNALING, CYTOKINE-CYTOKINE RECEPTOR COMPLEX
3tgx:O (ASP3) to (GLU42) IL-21:IL21R COMPLEX | CLASS I CYTOKINE, CLASS I CYTOKINE RECEPTOR, SUGARBRIDGE, FIBRONECTIN DOMAIN, SIGNALING, CYTOKINE-CYTOKINE RECEPTOR COMPLEX
1q3w:A (ILE62) to (LEU104) GSK-3 BETA COMPLEXED WITH ALSTERPAULLONE | KINASE, INSULIN PATHWAY, ALSTERPAULLONE, TRANSFERASE
1q41:A (ILE62) to (LEU104) GSK-3 BETA COMPLEXED WITH INDIRUBIN-3'-MONOXIME | KINASE, INSULIN PATHWAY, INDIRUBIN-3'-MONOXIME, TRANSFERASE
3tiv:A (ASP125) to (ARG165) CRYSTAL STRUCTURE OF SUBUNIT B MUTANT N157A OF THE A1AO ATP SYNTHASE | HYDROLASE, ATP SYNTHESIS, HYDROGEN ION TRANSPORT
4jd2:F (PRO50) to (ALA98) CRYSTAL STRUCTURE OF BOS TAURUS ARP2/3 COMPLEX BINDING WITH MUS MUSCULUS GMF | ACTIN FILAMENT POLYMERIZATION AND BRANCHING, STRUCTURAL PROTEIN
3gvb:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT-BASED INHIBITOR | HYDROLASE, ANTIBIOTIC RESISTANCE, PERIPLASM, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1q8z:A (GLY165) to (ASP213) THE APOENZYME STRUCTURE OF THE YEAST SR PROTEIN KINASE, SKY1P | DISALLOWED, KINASE, TRANSFERASE
1ef7:A (GLY186) to (ASN228) CRYSTAL STRUCTURE OF HUMAN CATHEPSIN X | PAPAIN-LIKE, CYSTEINE PROTEASE, CARBOXYPEPTIDASE, CATHEPSIN, HYDROLASE
1ef7:B (GLY186) to (ASN228) CRYSTAL STRUCTURE OF HUMAN CATHEPSIN X | PAPAIN-LIKE, CYSTEINE PROTEASE, CARBOXYPEPTIDASE, CATHEPSIN, HYDROLASE
1q99:A (GLY165) to (ASP213) CRYSTAL STRUCTURE OF THE SACCHAROMYCES CEREVISIAE SR PROTEIN KINSAE, SKY1P, COMPLEXED WITH THE NON-HYDROLYZABLE ATP ANALOGUE, AMP-PNP | PROTEIN KINASE, TRANSFERASE
2r9w:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE WITH BOUND PHTHALAMIDE INHIBITOR | AMPC BETA LACTAMASE, PTHALAMIDE, ANTIBIOTIC RESISTANCE, HYDROLASE
2r9w:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE WITH BOUND PHTHALAMIDE INHIBITOR | AMPC BETA LACTAMASE, PTHALAMIDE, ANTIBIOTIC RESISTANCE, HYDROLASE
2r9x:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE WITH BOUND PHTHALAMIDE INHIBITOR | AMPC BETA-LACTAMASE, PTHALAMIDE, ANTIBIOTIC RESISTANCE, HYDROLASE
2r9x:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE WITH BOUND PHTHALAMIDE INHIBITOR | AMPC BETA-LACTAMASE, PTHALAMIDE, ANTIBIOTIC RESISTANCE, HYDROLASE
3ton:A (ALA1192) to (ILE1233) CRYSTRAL STRUCTURE OF THE C-TERMINAL SUBUNIT OF HUMAN MALTASE- GLUCOAMYLASE | HYDROLASE, CARBOHYDRATE/SUGAR BINDING, MEMBRANE
3ton:B (ALA1192) to (ILE1233) CRYSTRAL STRUCTURE OF THE C-TERMINAL SUBUNIT OF HUMAN MALTASE- GLUCOAMYLASE | HYDROLASE, CARBOHYDRATE/SUGAR BINDING, MEMBRANE
3top:A (ALA1192) to (ILE1233) CRYSTRAL STRUCTURE OF THE C-TERMINAL SUBUNIT OF HUMAN MALTASE- GLUCOAMYLASE IN COMPLEX WITH ACARBOSE | MEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3top:B (ALA1192) to (ILE1233) CRYSTRAL STRUCTURE OF THE C-TERMINAL SUBUNIT OF HUMAN MALTASE- GLUCOAMYLASE IN COMPLEX WITH ACARBOSE | MEMBRANE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4jhn:C (TYR299) to (PHE349) THE CRYSTAL STRUCTURE OF THE RPGR RCC1-LIKE DOMAIN | RCC1, BETA PROPELLAR, SEVEN BLADED-PROPELLER, UNKNOWN FUNCTION
2rcx:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH (1R)-1-(2-THIOPHEN-2-YL- ACETYLAMINO)-1-(3-(2-CARBOXYVINYL)-PHENYL) METHYLBORONIC ACID | AMPC, BETA-LACTAMASE, CEPHALOSPORINASE, SERINE HYDROLASE, ANTIBIOTIC RESISTANCE, PERIPLASM
2rcx:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH (1R)-1-(2-THIOPHEN-2-YL- ACETYLAMINO)-1-(3-(2-CARBOXYVINYL)-PHENYL) METHYLBORONIC ACID | AMPC, BETA-LACTAMASE, CEPHALOSPORINASE, SERINE HYDROLASE, ANTIBIOTIC RESISTANCE, PERIPLASM
2rfs:A (GLY1085) to (PHE1134) X-RAY STRUCTURE OF SU11274 BOUND TO C-MET | C-MET, RECEPTOR TYROSINE KINASE, SU11274, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE
1emm:A (TYR92) to (GLY134) GREEN FLUORESCENT PROTEIN FROM AEQUOREA VICTORIA, MUTANT | FLUORESCENT PROTEIN, BETA-BARREL, BIOLUMINESCENCE, LUMINESCENCE
1etj:C (ASN18) to (GLY67) AZURIN MUTANT WITH MET 121 REPLACED BY GLU | ELECTRON TRANSPORT, COPPER, PERIPLASMIC
1eu1:A (GLY6) to (SER48) THE CRYSTAL STRUCTURE OF RHODOBACTER SPHAEROIDES DIMETHYLSULFOXIDE REDUCTASE REVEALS TWO DISTINCT MOLYBDENUM COORDINATION ENVIRONMENTS. | MOLYBDENUM, MOLYBDENUM COFACTOR, DMSO, REDUCTASE, MOLYBDOPTERIN, MGD, OXIDOREDUCTASE
2rk9:A (GLU39) to (ALA95) THE CRYSTAL STRUCTURE OF A GLYOXALASE/BLEOMYCIN RESISTANCE PROTEIN/DIOXYGENASE SUPERFAMILY MEMBER FROM VIBRIO SPLENDIDUS 12B01 | 11005R, GLYOXALASE/BLEOMYCIN RESISTANCE PROTEIN/DIOXYGENASE SUPERFAMILY, NYSGXRC, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE II, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, PSI-2, OXIDOREDUCTASE
2rk9:B (GLU39) to (ALA95) THE CRYSTAL STRUCTURE OF A GLYOXALASE/BLEOMYCIN RESISTANCE PROTEIN/DIOXYGENASE SUPERFAMILY MEMBER FROM VIBRIO SPLENDIDUS 12B01 | 11005R, GLYOXALASE/BLEOMYCIN RESISTANCE PROTEIN/DIOXYGENASE SUPERFAMILY, NYSGXRC, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE II, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, PSI-2, OXIDOREDUCTASE
4jpq:A (VAL120) to (MSE164) CRYSTAL STRUCTURE OF A PUTATIVE CARBOHYDRATE-BINDING PROTEIN (BACUNI_03838) FROM BACTEROIDES UNIFORMIS ATCC 8492 AT 2.70 A RESOLUTION | CARBOHYDRATE-BINDING FAMILY 9, PF16011, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, UNKNOWN FUNCTION
4jpq:B (VAL120) to (MSE164) CRYSTAL STRUCTURE OF A PUTATIVE CARBOHYDRATE-BINDING PROTEIN (BACUNI_03838) FROM BACTEROIDES UNIFORMIS ATCC 8492 AT 2.70 A RESOLUTION | CARBOHYDRATE-BINDING FAMILY 9, PF16011, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, UNKNOWN FUNCTION
4jq7:A (LEU694) to (VAL745) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN IN COMPLEX WITH COMPOUND 2A | TRANSFERASE, TYROSINE KINASE DOMAIN, ATP-BINDING DOMAIN, AUTOPHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jq8:A (LEU694) to (VAL745) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN IN COMPLEX WITH COMPOUND 4B | TRANSFERASE, TYROSINE KINASE DOMAIN, ATP-BINDING DOMAIN, AUTOPHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jqe:A (GLY47) to (SER90) CRYSTAL STRUCTURE OF SCCK2 ALPHA IN COMPLEX WITH AMPPN | PROTEIN KINASE, PROTEIN PHOSPHORYLATION, TRANSFERASE
3h4f:C (PRO71) to (THR112) MET62LEU VARIANT OF NITRITE REDUCTASE FROM ALCALIGENES FAECLIS | NITRITE REDUCTASE, NIR, HIGH-THROUGHPUT SCREENING, OXIDASE, COPPER, FAD, FLAVOPROTEIN, METAL-BINDING, NITRATE ASSIMILATION, OXIDOREDUCTASE, PERIPLASM, PYRROLIDONE CARBOXYLIC ACID
2tsa:B (ASN18) to (GLY67) AZURIN MUTANT M121A | ELECTRON TRANSPORT
4jrv:A (LEU694) to (VAL745) CRYSTAL STRUCTURE OF EGFR KINASE DOMAIN IN COMPLEX WITH COMPOUND 4C | TRANSFERASE, TYROSINE KINASE DOMAIN, ATP-BINDING DOMAIN, AUTOPHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2e5a:A (LYS252) to (ILE306) CRYSTAL STRUCTURE OF BOVINE LIPOYLTRANSFERASE IN COMPLEX WITH LIPOYL-AMP | LIPOYLTRANSFERASE, LIPOYL-AMP, LIGASE
4jt5:B (ALA2226) to (LYS2258) MTORDELTAN-MLST8-PP242 COMPLEX | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jt5:A (ALA2226) to (LYS2258) MTORDELTAN-MLST8-PP242 COMPLEX | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2e9o:A (LEU15) to (LEU62) STRUCTURE OF H-CHK1 COMPLEXED WITH AA582939 | PROTEIN-INHIBITOR COMPLEX, TRANSFERASE
1r1l:L (ARG259) to (LEU299) STRUCTURE OF DIMERIC ANTITHROMBIN COMPLEXED WITH A P14-P9 REACTIVE LOOP PEPTIDE AND AN EXOGENOUS TRIPEPTIDE (FORMYL-NORLEUCINE-LF) | SERPIN, LOOP-SHEET POLYMER, BETA-BARREL, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4jx7:A (ASP108) to (GLU135) CRYSTAL STRUCTURE OF PIM1 KINASE IN COMPLEX WITH INHIBITOR 2-[(TRANS- 4-AMINOCYCLOHEXYL)AMINO]-4-{[3-(TRIFLUOROMETHYL) PHENYL]AMINO}PYRIDO[4,3-D]PYRIMIDIN-5(6H)-ONE | SERINE/THREONINE-PROTEIN KINASES, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jxg:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH OXACILLIN | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, ACYL-ENZYME COMPLEX, HYDROLASE-ANTIBIOTIC COMPLEX
4jxg:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH OXACILLIN | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, ACYL-ENZYME COMPLEX, HYDROLASE-ANTIBIOTIC COMPLEX
4jxs:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH A NON-COVALENT INHIBITOR 3-[(4-CARBOXYBENZYL) SULFAMOYL]THIOPHENE-2-CARBOXYLIC ACID (COMPOUND 4) | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, BETA-LACTAMASE INHIBITOR COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4jxv:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH A NON-COVALENT INHIBITOR 3-{[2-(4-CARBOXYPHENYL) ETHYL]SULFAMOYL}THIOPHENE-2-CARBOXYLIC ACID (COMPOUND 5) | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4jxw:A (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH A NON-COVALENT INHIBITOR 3-{[3-(4-CARBOXYPHENYL) PROPYL]SULFAMOYL}THIOPHENE-2-CARBOXYLIC ACID (COMPOUND 6) | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4jxw:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH A NON-COVALENT INHIBITOR 3-{[3-(4-CARBOXYPHENYL) PROPYL]SULFAMOYL}THIOPHENE-2-CARBOXYLIC ACID (COMPOUND 6) | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1fcm:B (TYR256) to (ASP285) CRYSTAL STRUCTURE OF THE E.COLI AMPC BETA-LACTAMASE MUTANT Q120L/Y150E COVALENTLY ACYLATED WITH THE INHIBITORY BETA-LACTAM, CLOXACILLIN | BETA-LACTAMASE BETA-LACTAM COMPLEX, ENZYME INHIBITOR COMPLEX, HYDROLASE-ANTIBIOTIC COMPLEX
1fcn:B (TYR256) to (ASP285) CRYSTAL STRUCTURE OF THE E. COLI AMPC BETA-LACTAMASE MUTANT Q120L/Y150E COVALENTLY ACYLATED WITH THE SUBSTRATE BETA-LACTAM LORACARBEF | BETA-LACTAMASE BETA-LACTAM COMPLEX, ENZYME INHIBITOR COMPLEX, HYDROLASE
1fco:B (TYR256) to (ASP285) CRYSTAL STRUCTURE OF THE E. COLI AMPC BETA-LACTAMASE COVALENTLY ACYLATED WITH THE INHIBITORY BETA-LACTAM, MOXALACTAM | BETA-LACTAMASE BETA-LACTAM COMPLEX, ENZYME INHIBITOR COMPLEX, HYDROLASE
3u8a:B (PHE88) to (LYS135) CRYSTAL STRUCTURE OF MONOMERIC REVERSIBLY PHOTOSWITCHABLE RED FLUORESCENT PROTEIN RSTAGRFP IN THE OFF STATE | BETA-BARREL, FLUORESCENT PROTEIN, LIGHT INDUCED REVERSIBLE PHOTOSWITCHING, REVERSIBLY PHOTOSWITCHABLE FLUORESCENT PROTEIN, CIS- TRANS ISOMERIZATION
3u8c:B (PHE88) to (LYS135) CRYSTAL STRUCTURE OF MONOMERIC REVERSIBLY PHOTOSWITCHABLE RED FLUORESCENT PROTEIN RSTAGRFP IN THE ON STATE | BETA BARREL, FLUORESCENT PROTEIN, LIGHT INDUCED REVERSIBLE PHOTOSWITCHING, REVERSIBLY PHOTOSWITCHABLE FLUORESCENT PROTEIN, CIS- TRANS ISOMERIZATION
3u8c:C (PHE88) to (LYS135) CRYSTAL STRUCTURE OF MONOMERIC REVERSIBLY PHOTOSWITCHABLE RED FLUORESCENT PROTEIN RSTAGRFP IN THE ON STATE | BETA BARREL, FLUORESCENT PROTEIN, LIGHT INDUCED REVERSIBLE PHOTOSWITCHING, REVERSIBLY PHOTOSWITCHABLE FLUORESCENT PROTEIN, CIS- TRANS ISOMERIZATION
2ejf:A (ASP104) to (LYS173) CRYSTAL STRUCTURE OF THE BIOTIN PROTEIN LIGASE (MUTATIONS R48A AND K111A) AND BIOTIN CARBOXYL CARRIER PROTEIN COMPLEX FROM PYROCOCCUS HORIKOSHII OT3 | BIOTINYLATION, DIMER, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, LIGASE
2emn:A (VAL93) to (GLY134) GREEN FLUORESCENT PROTEIN FROM AEQUOREA VICTORIA, MUTANT | FLUORESCENT PROTEIN, BETA-BARREL, BIOLUMINESCENCE, LUMINESCENCE
4k1b:A (ASP108) to (ARG136) STRUCTURE OF PIM-1 KINASE BOUND TO N-(5-(2-FLUOROPHENYL)-1H-PYRROLO[2, 3-B]PYRIDIN-3-YL)-5-((((3R,4R)-3-FLUOROPIPERIDIN-4-YL)METHYL)AMINO) PYRAZOLO[1,5-A]PYRIMIDINE-3-CARBOXAMIDE | PIM-1, KINASE DOMAIN, SER/THR KINASE, ATP-COMPETITIVE, STRUCTURE- BASED DRUG DESIGN, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yr8:C (ASN28) to (CYS79) CRYSTAL STRUCTURE OF JNK IN COMPLEX WITH A REGULATOR PROTEIN | KINASE DOMAIN, CATALYTIC DOMAIN, TRANSFERASE-HYDROLASE COMPLEX
2euf:B (GLU14) to (GLU69) X-RAY STRUCTURE OF HUMAN CDK6-VCYCLIN IN COMPLEX WITH THE INHIBITOR PD0332991 | INHIBITOR COMPLEX OF HUMAN CYCLIN-DEPENDENT KINASE 6, CELL CYCLE- TRANSFERASE COMPLEX
4ysd:A (PRO72) to (ILE111) ROOM TEMPERATURE STRUCTURE OF COPPER NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS | NITRITE, COPPER, REDUCTASE, OXIDOREDUCTASE
4yso:A (PRO72) to (ILE111) COPPER NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS - 0.064 MGY | NITRITE, COPPER, REDUCTASE, OXIDOREDUCTASE
4ysp:A (PRO72) to (ILE111) STRUCTURE OF COPPER NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS - 8.32 MGY | NITRITE, COPPER, REDUCTASE, OXIDOREDUCTASE
4ysu:A (PRO72) to (ILE111) STRUCTURE OF COPPER NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS - 25.0 MGY | NITRITE, COPPER, REDUCTASE, OXIDOREDUCTASE
4ysr:A (PRO72) to (ILE111) STRUCTURE OF COPPER NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS - 16.6 MGY | NITRITE, COPPER, REDUCTASE, OXIDOREDUCTASE
4yss:A (PRO72) to (ILE111) STRUCTURE OF COPPER NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS - 16.7 MGY | NITRITE, COPPER, REDUCTASE, OXIDOREDUCTASE
4yst:A (PRO72) to (ILE111) STRUCTURE OF COPPER NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS - 24.9 MGY | NITRITE, COPPER, REDUCTASE, OXIDOREDUCTASE
1fr1:A (TYR259) to (ASP288) REFINED CRYSTAL STRUCTURE OF BETA-LACTAMASE FROM CITROBACTER FREUNDII INDICATES A MECHANISM FOR BETA-LACTAM HYDROLYSIS | HYDROLASE, ANTIBIOTIC RESISTANCE, CLASS C BETA-LACTAMASE
1fr1:B (TYR259) to (ASP288) REFINED CRYSTAL STRUCTURE OF BETA-LACTAMASE FROM CITROBACTER FREUNDII INDICATES A MECHANISM FOR BETA-LACTAM HYDROLYSIS | HYDROLASE, ANTIBIOTIC RESISTANCE, CLASS C BETA-LACTAMASE
1fr6:A (TYR259) to (ASP288) REFINED CRYSTAL STRUCTURE OF BETA-LACTAMASE FROM CITROBACTER FREUNDII INDICATES A MECHANISM FOR BETA-LACTAM HYDROLYSIS | HYDROLASE, ANTIBIOTIC RESISTANCE, CLASS C BETA-LACTAMASE, MONOBACTUM
1fr6:B (TYR259) to (ASP288) REFINED CRYSTAL STRUCTURE OF BETA-LACTAMASE FROM CITROBACTER FREUNDII INDICATES A MECHANISM FOR BETA-LACTAM HYDROLYSIS | HYDROLASE, ANTIBIOTIC RESISTANCE, CLASS C BETA-LACTAMASE, MONOBACTUM
1fsw:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE FROM E. COLI COMPLEXED WITH INHIBITOR CEPHALOTHINBORONIC ACID | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, HYDROLASE
1fsw:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE FROM E. COLI COMPLEXED WITH INHIBITOR CEPHALOTHINBORONIC ACID | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, HYDROLASE
1fsy:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE FROM E. COLI COMPLEXED WITH INHIBITOR CLOXACILLINBORONIC ACID | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, HYDROLASE
1fsy:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE FROM E. COLI COMPLEXED WITH INHIBITOR CLOXACILLINBORONIC ACID | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, HYDROLASE
1rgz:A (TYR262) to (ASP291) ENTEROBACTER CLOACAE GC1 CLASS C BETA-LACTAMASE COMPLEXED WITH TRANSITION-STATE ANALOG OF CEFOTAXIME | HYDROLASE, CEPHALOSPORINASE, ENZYME INHIBITION, PHOSPHONATE, BETA- LACTAM ANTIBIOTICS, DRUG DESIGN
2f2h:A (GLN214) to (THR258) STRUCTURE OF THE YICI THIOSUGAR MICHAELIS COMPLEX | BETA8ALPHA8 BARREL, HYDROLASE
2f2h:B (GLN214) to (THR258) STRUCTURE OF THE YICI THIOSUGAR MICHAELIS COMPLEX | BETA8ALPHA8 BARREL, HYDROLASE
2f2h:C (GLN214) to (THR258) STRUCTURE OF THE YICI THIOSUGAR MICHAELIS COMPLEX | BETA8ALPHA8 BARREL, HYDROLASE
2f2h:D (GLN214) to (THR258) STRUCTURE OF THE YICI THIOSUGAR MICHAELIS COMPLEX | BETA8ALPHA8 BARREL, HYDROLASE
2f2h:E (GLN214) to (THR258) STRUCTURE OF THE YICI THIOSUGAR MICHAELIS COMPLEX | BETA8ALPHA8 BARREL, HYDROLASE
2f2h:F (GLN214) to (THR258) STRUCTURE OF THE YICI THIOSUGAR MICHAELIS COMPLEX | BETA8ALPHA8 BARREL, HYDROLASE
3ukr:F (PRO50) to (ALA98) CRYSTAL STRUCTURE OF BOS TAURUS ARP2/3 COMPLEX WITH BOUND INHIBITOR CK-666 | BETA-PROPELLER ACTIN FOLD, STRUCTURAL PROTEIN, ATP BINDING
3ule:F (PRO50) to (ALA98) STRUCTURE OF BOS TAURUS ARP2/3 COMPLEX WITH BOUND INHIBITOR CK-869 AND ATP | BETA-PROPELLOR, STRUCTURAL PROTEIN, ACTIN FILAMENT NUCLEATOR
4kbk:B (GLY16) to (GLN60) CK1D IN COMPLEX WITH (3S)-3-{4-[3-(4-FLUOROPHENYL)-1-METHYL-1H- PYRAZOL-4-YL]PYRIDIN-2-YL}MORPHOLINE INHIBITOR | SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3umx:A (ASP108) to (GLU135) CRYSTAL STRUCTURE OF PIM1 KINASE IN COMPLEX WITH INHIBITOR (Z)-2-[(1H- INDOL-3-YL)METHYLENE]-7-(AZEPAN-1-YLMETHYL)-6-HYDROXYBENZOFURAN- 3(2H)-ONE | PIM-1, KINASE, P-LOOP, KINASE INHIBITOR, RATIONAL DRUG DESIGN, TRANSFERASE-INHIBITOR COMPLEX
3hmm:A (GLY12) to (THR51) STRUCTURE OF ALK5 + GW855857 | TGF-BETA, ALK5, KINASE, INHIBITOR, QUINAZOLINE, AORTIC ANEURYSM, ATP-BINDING, CRANIOSYNOSTOSIS, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, MAGNESIUM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN POLYMORPHISM, RECEPTOR, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSMEMBRANE
3hnc:A (LYS424) to (ILE481) CRYSTAL STRUCTURE OF HUMAN RIBONUCLEOTIDE REDUCTASE 1 BOUND TO THE EFFECTOR TTP | OXIDOREDUCTASE, RIBONUCLEOTIDE REDUCTASE, ALLOSTERIC ENZYME, ATP- BINDING, DNA REPLICATION, NUCLEOTIDE-BINDING
3hnc:B (LYS424) to (ILE481) CRYSTAL STRUCTURE OF HUMAN RIBONUCLEOTIDE REDUCTASE 1 BOUND TO THE EFFECTOR TTP | OXIDOREDUCTASE, RIBONUCLEOTIDE REDUCTASE, ALLOSTERIC ENZYME, ATP- BINDING, DNA REPLICATION, NUCLEOTIDE-BINDING
3hnd:A (LYS424) to (ILE481) CRYSTAL STRUCTURE OF HUMAN RIBONUCLEOTIDE REDUCTASE 1 BOUND TO THE EFFECTOR TTP AND SUBSTRATE GDP | OXIDOREDUCTASE, RIBONUCLEOTIDE REDUCTASE, ALLOSTERIC ENZYME, ATP- BINDING, DNA REPLICATION, NUCLEOTIDE-BINDING
3hnd:B (LYS424) to (ILE481) CRYSTAL STRUCTURE OF HUMAN RIBONUCLEOTIDE REDUCTASE 1 BOUND TO THE EFFECTOR TTP AND SUBSTRATE GDP | OXIDOREDUCTASE, RIBONUCLEOTIDE REDUCTASE, ALLOSTERIC ENZYME, ATP- BINDING, DNA REPLICATION, NUCLEOTIDE-BINDING
3hne:A (LYS424) to (ILE483) CRYSTAL STRUCTURE OF HUMAN RIBONUCLEOTIDE REDUCTASE 1 BOUND TO THE EFFECTORS TTP AND ATP | OXIDOREDUCTASE, RIBONUCLEOTIDE REDUCTASE, ALLOSTERIC ENZYME, ATP- BINDING, DNA REPLICATION, NUCLEOTIDE-BINDING
3hne:B (LYS424) to (ASN484) CRYSTAL STRUCTURE OF HUMAN RIBONUCLEOTIDE REDUCTASE 1 BOUND TO THE EFFECTORS TTP AND ATP | OXIDOREDUCTASE, RIBONUCLEOTIDE REDUCTASE, ALLOSTERIC ENZYME, ATP- BINDING, DNA REPLICATION, NUCLEOTIDE-BINDING
3hnf:B (LYS424) to (ASN484) CRYSTAL STRUCTURE OF HUMAN RIBONUCLEOTIDE REDUCTASE 1 BOUND TO THE EFFECTORS TTP AND DATP | OXIDOREDUCTASE, RIBONUCLEOTIDE REDUCTASE, ALLOSTERIC ENZYME, ATP- BINDING, DNA REPLICATION, NUCLEOTIDE-BINDING
4ken:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE N152G MUTANT IN COMPLEX WITH CEFOXITIN | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, ACYL-ENZYME COMPLEX, HYDROLASE-ANTIBIOTIC COMPLEX
2fbl:A (ARG80) to (PHE125) THE CRYSTAL STRUCTURE OF THE HYPOTHETICAL PROTEIN NE1496 | APC5855, NE1496, PSI, PROTEIN STRUCTURE INITIATIVE, MCSG, MIDWEST CENTER FOR STRUCTURAL GENOMICS, STRUCTURAL GENOMICS, UNKNOWN FUNCTION
2fbl:B (ARG80) to (PHE125) THE CRYSTAL STRUCTURE OF THE HYPOTHETICAL PROTEIN NE1496 | APC5855, NE1496, PSI, PROTEIN STRUCTURE INITIATIVE, MCSG, MIDWEST CENTER FOR STRUCTURAL GENOMICS, STRUCTURAL GENOMICS, UNKNOWN FUNCTION
4kg5:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE N152G MUTANT IN COMPLEX WITH CEFOTAXIME | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, ACYL-ENZYME COMPLEX, HYDROLASE-ANTIBIOTIC COMPLEX
4kg5:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE N152G MUTANT IN COMPLEX WITH CEFOTAXIME | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, ACYL-ENZYME COMPLEX, HYDROLASE-ANTIBIOTIC COMPLEX
4kg5:C (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE N152G MUTANT IN COMPLEX WITH CEFOTAXIME | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, ACYL-ENZYME COMPLEX, HYDROLASE-ANTIBIOTIC COMPLEX
4kg5:D (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE N152G MUTANT IN COMPLEX WITH CEFOTAXIME | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, ACYL-ENZYME COMPLEX, HYDROLASE-ANTIBIOTIC COMPLEX
4kg2:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH CEFOTAXIME | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, ACYL-ENZYME COMPLEX, HYDROLASE-ANTIBIOTIC COMPLEX
4kg2:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH CEFOTAXIME | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, ACYL-ENZYME COMPLEX, HYDROLASE-ANTIBIOTIC COMPLEX
4kg6:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE N152G MUTANT FROM E. COLI | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, HYDROLASE
4kg6:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE N152G MUTANT FROM E. COLI | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, HYDROLASE
4kg6:C (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE N152G MUTANT FROM E. COLI | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, HYDROLASE
4kg6:D (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE N152G MUTANT FROM E. COLI | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, HYDROLASE
4kgf:A (PHE88) to (LYS135) CRYSTAL STRUCTURE OF NEAR-INFRARED FLUORESCENT PROTEIN WITH AN EXTENDED STOKES SHIFT, PH 8.0 | STRUCTURAL GENOMICS, PROTEINSTRUCTURE INITIATIVE, NEW YORK STRUCTURAL GENOMIX RESEARCHCONSORTIUM, HYDROLASE, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, FLUORESCENT PROTEIN
1rwh:A (GLU586) to (LEU640) CRYSTAL STRUCTURE OF ARTHROBACTER AURESCENS CHONDROITIN AC LYASE IN COMPLEX WITH CHONDROITIN TETRASACCHARIDE | CHONDROITINASE, CHONDROITIN, CHONDROITIN LYASE, LYASE
2ffy:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE N289A MUTANT IN COMPLEX WITH A BORONIC ACID DEACYLATION TRANSITION STATE ANALOG COMPOUND SM3 | AMPC; BETA-LACTAMASE; DEACYLATION; TRANSITION STATE; BORONIC ACID, HYDROLASE
4kio:A (VAL366) to (LEU413) KINASE DOMAIN MUTANT OF HUMAN ITK IN COMPLEX WITH A COVALENTLY-BINDING INHIBITOR | KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1ga0:A (TYR262) to (ASP291) STRUCTURE OF THE E. CLOACAE GC1 BETA-LACTAMASE WITH A CEPHALOSPORIN SULFONE INHIBITOR | MIXED ALPHA/BETA, CEPHALOSPORINASE, INHIBITION, CONFORMATIONAL CHANGE, CLASS C BETA-LACTAMASE, HYDROLASE
1ga9:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI COMPLEXED WITH NON-BETA-LACTAMASE INHIBITOR (2, 3-(4- BENZENESULFONYL-THIOPHENE-2-SULFONYLAMINO)-PHENYLBORONIC ACID) | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE
1ga9:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI COMPLEXED WITH NON-BETA-LACTAMASE INHIBITOR (2, 3-(4- BENZENESULFONYL-THIOPHENE-2-SULFONYLAMINO)-PHENYLBORONIC ACID) | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE
1gce:A (TYR262) to (GLY289) STRUCTURE OF THE BETA-LACTAMASE OF ENTEROBACTER CLOACAE GC1 | BETA-LACTAM HYDROLASE, CEPHALOSPORINASE, DRUG DESIGN, EXTENDED- SPECTRUM BETA- LACTAMASE, HYDROLASE
4kmq:A (SER335) to (ASP380) 1.9 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF UNCHARACTERIZED PROTEIN LMO2446 FROM LISTERIA MONOCYTOGENES EGD-E | UNCHARACTERIZED PROTEIN, VIRULENCE, PATHOGENESIS, CSGID, STRUCTURAL GENOMICS, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, TIM-BARREL, UNKNOWN FUNCTION
3uwx:A (ILE4) to (LEU40) CRYSTAL STRUCTURE OF UVRA-UVRB COMPLEX | UVRA, UVRB, NUCLEOTIDE EXCISION REPAIR, DNA REPAIR, ABC ATPASE, ATP BINDING, DNA BINDING, DNA BINDING PROTEIN
3huf:B (GLY90) to (GLY137) STRUCTURE OF THE S. POMBE NBS1-CTP1 COMPLEX | NBS1, FHA DOMAIN, BRCT DOMAIN, PHOSPHOPROTEIN BINDING, PHOSPHOSERINE BINDING, DNA REPAIR, CTP1, CHROMOSOMAL PROTEIN, DNA DAMAGE, NUCLEUS, PHOSPHOPROTEIN, TELOMERE, MEIOSIS, CELL CYCLE
1s6r:A (TYR259) to (ASP288) 908R CLASS C BETA-LACTAMASE BOUND TO IODO-ACETAMIDO-PHENYL BORONIC ACID | HYDROLASE
2fta:A (ASN18) to (GLY67) STRUCTURE OF CU(II)AZURIN WITH THE METAL-BINDING LOOP SEQUENCE "CTFPGHSALM" REPLACED WITH "CTPHPFM" | BLUE COPPER-BINDING PROTEIN, GREEK-KEY BETA-BARREL, ELECTRON TRANSPORT
4knu:A (PRO59) to (GLU99) COPPER NITRITE REDUCTASE FROM NITROSOMONAS EUROPAEA AT PH 6.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
4knu:B (PRO59) to (GLU99) COPPER NITRITE REDUCTASE FROM NITROSOMONAS EUROPAEA AT PH 6.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
4knu:C (PRO59) to (GLU99) COPPER NITRITE REDUCTASE FROM NITROSOMONAS EUROPAEA AT PH 6.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
4knu:D (PRO59) to (GLU99) COPPER NITRITE REDUCTASE FROM NITROSOMONAS EUROPAEA AT PH 6.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
4knu:E (PRO59) to (GLU99) COPPER NITRITE REDUCTASE FROM NITROSOMONAS EUROPAEA AT PH 6.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
4knu:F (PRO59) to (GLU99) COPPER NITRITE REDUCTASE FROM NITROSOMONAS EUROPAEA AT PH 6.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
2fw3:A (LEU234) to (ASP279) CRYSTAL STRUCTURE OF RAT CARNITINE PALMITOYLTRANSFERASE 2 IN COMPLEX WITH ANTIDIABETIC DRUG ST1326 | CENTRAL SIX-STRANDED BETA-SHEET, TRANSFERASE
1gng:B (ILE62) to (LEU104) GLYCOGEN SYNTHASE KINASE-3 BETA (GSK3) COMPLEX WITH FRATTIDE PEPTIDE | TRANSFERASE, PROTEIN KINASE, GSK3/FRATTIDE COMPLEX, PHOSPHORYLATED, ACTIVE
3v7b:A (GLY43) to (ALA86) DIP2269 PROTEIN FROM CORYNEBACTERIUM DIPHTHERIAE | STRUCTURAL GENOMICS, PSI-BIOLOGY, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, UNKNOWN FUNCTION
3v7b:B (GLY43) to (ALA87) DIP2269 PROTEIN FROM CORYNEBACTERIUM DIPHTHERIAE | STRUCTURAL GENOMICS, PSI-BIOLOGY, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, UNKNOWN FUNCTION
4kr8:A (GLY19) to (ASN74) SALMONELLA TYPHI OMPF COMPLEX WITH DAUNOMYCIN | BETA BARREL, TRANSPORT, OUTER MEMBRANE, MEMBRANE PROTEIN
2g3o:A (TYR83) to (ASP130) THE 2.1A CRYSTAL STRUCTURE OF COPGFP | BETA-BARREL, CHROMOPHORE, GFP, LUMINESCENT PROTEIN
2g3o:B (TYR83) to (ASP130) THE 2.1A CRYSTAL STRUCTURE OF COPGFP | BETA-BARREL, CHROMOPHORE, GFP, LUMINESCENT PROTEIN
2g3o:C (GLY81) to (ASP130) THE 2.1A CRYSTAL STRUCTURE OF COPGFP | BETA-BARREL, CHROMOPHORE, GFP, LUMINESCENT PROTEIN
2g3o:D (GLY81) to (ASP130) THE 2.1A CRYSTAL STRUCTURE OF COPGFP | BETA-BARREL, CHROMOPHORE, GFP, LUMINESCENT PROTEIN
2g3o:E (GLY81) to (ASP130) THE 2.1A CRYSTAL STRUCTURE OF COPGFP | BETA-BARREL, CHROMOPHORE, GFP, LUMINESCENT PROTEIN
2g3o:F (GLY81) to (ASP130) THE 2.1A CRYSTAL STRUCTURE OF COPGFP | BETA-BARREL, CHROMOPHORE, GFP, LUMINESCENT PROTEIN
4ktr:B (MET1) to (PHE33) CRYSTAL STRUCTURE OF 2-O-ALPHA-GLUCOSYLGLYCEROL PHOSPHORYLASE IN COMPLEX WITH ISOFAGOMINE AND GLYCEROL | (ALPHA/ALPHA)6 BARREL, PHOSPHORYLASE, TRANSFERASE
1gs8:A (PRO65) to (THR106) CRYSTAL STRUCTURE OF MUTANT D92N ALCALIGENES XYLOSOXIDANS NITRITE REDUCTASE | OXIDOREDUCTASE, MULTICOPPER, PERIPLASMIC
3vbt:A (ASP108) to (GLY137) EXPLOITATION OF HYDROGEN BONDING CONSTRAINTS AND FLAT HYDROPHOBIC ENERGY LANDSCAPES IN PIM-1 KINASE NEEDLE SCREENING AND INHIBITOR DESIGN | PIM1, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3vbv:A (ASP108) to (GLY137) EXPLOITATION OF HYDROGEN BONDING CONSTRAINTS AND FLAT HYDROPHOBIC ENERGY LANDSCAPES IN PIM-1 KINASE NEEDLE SCREENING AND INHIBITOR DESIGN | PIM1, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3vbw:A (ASP108) to (GLY137) EXPLOITATION OF HYDROGEN BONDING CONSTRAINTS AND FLAT HYDROPHOBIC ENERGY LANDSCAPES IN PIM-1 KINASE NEEDLE SCREENING AND INHIBITOR DESIGN | PIM1, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3vc4:A (GLN37) to (VAL96) EXPLOITATION OF HYDROGEN BONDING CONSTRAINTS AND FLAT HYDROPHOBIC ENERGY LANDSCAPES IN PIM-1 KINASE NEEDLE SCREENING AND INHIBITOR DESIGN | PIM1, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2g6x:A (TYR83) to (ASP130) CRYSTAL STRUCTURE OF A NOVEL GREEN FLUORESCENT PROTEIN FROM MARINE COPEPOD PONTELLINA PLUMATA | GREEN FLUORESCENT PROTEIN, NATURAL CHROMOPHORE, RAPID MATURATION, BETA CAN, LUMINESCENT PROTEIN
2g6x:B (TYR83) to (ASP130) CRYSTAL STRUCTURE OF A NOVEL GREEN FLUORESCENT PROTEIN FROM MARINE COPEPOD PONTELLINA PLUMATA | GREEN FLUORESCENT PROTEIN, NATURAL CHROMOPHORE, RAPID MATURATION, BETA CAN, LUMINESCENT PROTEIN
2g6x:C (THR84) to (ASP130) CRYSTAL STRUCTURE OF A NOVEL GREEN FLUORESCENT PROTEIN FROM MARINE COPEPOD PONTELLINA PLUMATA | GREEN FLUORESCENT PROTEIN, NATURAL CHROMOPHORE, RAPID MATURATION, BETA CAN, LUMINESCENT PROTEIN
2g6x:D (TYR83) to (ASP130) CRYSTAL STRUCTURE OF A NOVEL GREEN FLUORESCENT PROTEIN FROM MARINE COPEPOD PONTELLINA PLUMATA | GREEN FLUORESCENT PROTEIN, NATURAL CHROMOPHORE, RAPID MATURATION, BETA CAN, LUMINESCENT PROTEIN
2g6y:A (THR84) to (ASP130) CRYSTAL STRUCTURE OF THE NOVEL GREEN FLUORESCENT PROTEIN FROM MARINE COPEPOD PONTELLINA PLUMATA | GREEN FLUORESCENT PROTEIN, NATURAL CHROMOPHORE, RAPID MATURATION, BETA-CAN, LUMINESCENT PROTEIN
2g6y:B (TYR83) to (ASP130) CRYSTAL STRUCTURE OF THE NOVEL GREEN FLUORESCENT PROTEIN FROM MARINE COPEPOD PONTELLINA PLUMATA | GREEN FLUORESCENT PROTEIN, NATURAL CHROMOPHORE, RAPID MATURATION, BETA-CAN, LUMINESCENT PROTEIN
2g6y:C (TYR83) to (ASP130) CRYSTAL STRUCTURE OF THE NOVEL GREEN FLUORESCENT PROTEIN FROM MARINE COPEPOD PONTELLINA PLUMATA | GREEN FLUORESCENT PROTEIN, NATURAL CHROMOPHORE, RAPID MATURATION, BETA-CAN, LUMINESCENT PROTEIN
2g6y:D (TYR83) to (ASP130) CRYSTAL STRUCTURE OF THE NOVEL GREEN FLUORESCENT PROTEIN FROM MARINE COPEPOD PONTELLINA PLUMATA | GREEN FLUORESCENT PROTEIN, NATURAL CHROMOPHORE, RAPID MATURATION, BETA-CAN, LUMINESCENT PROTEIN
2g7j:A (THR26) to (ALA63) SOLUTION NMR STRUCTURE OF THE PUTATIVE CYTOPLASMIC PROTEIN YGAC FROM SALMONELLA TYPHIMURIUM. NORTHEAST STRUCTURAL GENOMICS TARGET STR72. | STR72, AUTOSTRUCTURE, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, NESG, UNKNOWN FUNCTION
1sr5:A (PHE258) to (LEU299) ANTITHROMBIN-ANHYDROTHROMBIN-HEPARIN TERNARY COMPLEX STRUCTURE | SERINE PROTEINASE INHIBITOR, ANTITHROMBIN ACTIVATION BY HEP ANHYDROTHROMBIN, PROTEIN-PROTEIN INTERACTIONS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4kwu:A (SER335) to (THR382) 1.9 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF UNCHARACTERIZED PROTEIN LMO2446 FROM LISTERIA MONOCYTOGENES EGD-E IN COMPLEX WITH ALPHA-D- GLUCOSE, BETA-D-GLUCOSE, MAGNESIUM AND CALCIUM | CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, STRUCTURAL GENOMICS, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, TIM-BARREL, BETA-FOLD, UNKNOWN FUNCTION
2ga9:D (LYS334) to (LEU373) CRYSTAL STRUCTURE OF THE HETERODIMERIC VACCINIA VIRUS POLYADENYLATE POLYMERASE WITH BOUND ATP-GAMMA-S | POLYADENYLATE POLYMERASE, NUCLEOTIDYLTRANSFERASE, POXVIRUS, HETERODIMER, PROCESSIVITY, TRANSFERASE
2gag:A (MET757) to (GLY803) HETEROTETERAMERIC SARCOSINE: STRUCTURE OF A DIFLAVIN METALOENZYME AT 1.85 A RESOLUTION | SARCOSINE OXIDASE, FLAVOENZYME, ELECTRON TRANSFER, FOLATE-METHYLATING ENZYME, OXIDOREDUCTASE
2gag:C (ASN151) to (SER198) HETEROTETERAMERIC SARCOSINE: STRUCTURE OF A DIFLAVIN METALOENZYME AT 1.85 A RESOLUTION | SARCOSINE OXIDASE, FLAVOENZYME, ELECTRON TRANSFER, FOLATE-METHYLATING ENZYME, OXIDOREDUCTASE
2gah:A (MSE757) to (GLY803) HETEROTETRAMERIC SARCOSINE: STRUCTURE OF A DIFLAVIN METALOENZYME AT 1.85 A RESOLUTION | SARCOSINE OXIDASE, FLAVOENZYME, ELECTRON TRANSFER, FOLATE- METHYLATING ENZYME, OXIDOREDUCTASE
2gah:C (ASN151) to (SER198) HETEROTETRAMERIC SARCOSINE: STRUCTURE OF A DIFLAVIN METALOENZYME AT 1.85 A RESOLUTION | SARCOSINE OXIDASE, FLAVOENZYME, ELECTRON TRANSFER, FOLATE- METHYLATING ENZYME, OXIDOREDUCTASE
3i7f:A (PHE431) to (GLY489) ASPARTYL TRNA SYNTHETASE FROM ENTAMOEBA HISTOLYTICA | TRNA LIGASE, APO, ATP-BINDING, AMINOACYL-TRNA SYNTHETASE, LIGASE, NUCLEOTIDE-BINDING, PROTEIN BIOSYNTHESIS, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP
3i7h:A (ALA956) to (HIS991) CRYSTAL STRUCTURE OF DDB1 IN COMPLEX WITH THE H-BOX MOTIF OF HBX | DDB1, HBV, X PROTEIN, H-BOX MOTIF, CYTOPLASM, DNA DAMAGE, DNA REPAIR, DNA-BINDING, HOST-VIRUS INTERACTION, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, UBL CONJUGATION, UBL CONJUGATION PATHWAY, ACTIVATOR, APOPTOSIS, MITOCHONDRION, TRANSCRIPTION, TRANSCRIPTION REGULATION, PROTEIN BINDING/VIRAL PROTEIN COMPLEX
2vwe:C (SER52) to (THR85) CRYSTAL STRUCTURE OF VASCULAR ENDOTHELIAL GROWTH FACTOR-B IN COMPLEX WITH A NEUTRALIZING ANTIBODY FAB FRAGMENT | IMMUNE SYSTEM, GLYCOPROTEIN, CYSTEINE-KNOT, GROWTH FACTOR, VEGF-B, MITOGEN, SECRETED, ANGIOGENESIS, NEUTRALIZING ANTIBODY, HEPARIN-BINDING, ALTERNATIVE SPLICING
2gcd:A (ILE34) to (LEU83) TAO2 KINASE DOMAIN-STAUROSPORINE STRUCTURE | TAO2, MAP3K, INHIBITOR, STAUROSPORINE, CRYSTAL STRUCTURE, TRANSFERASE
4kz4:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 60 (2-[(PROPYLSULFONYL)AMINO]BENZOIC ACID) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4kz4:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 60 (2-[(PROPYLSULFONYL)AMINO]BENZOIC ACID) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4kz5:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 5 (N-{[3-(2-CHLOROPHENYL)-5-METHYL-1,2-OXAZOL-4-YL]CARBONYL}GLYCINE) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4kz7:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 16 ((1R,4S)-4,7,7-TRIMETHYL-3-OXO-2-OXABICYCLO[2.2.1]HEPTANE-1- CARBOXYLIC ACID) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4kz7:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 16 ((1R,4S)-4,7,7-TRIMETHYL-3-OXO-2-OXABICYCLO[2.2.1]HEPTANE-1- CARBOXYLIC ACID) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4kz8:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 20 (1,3-DIETHYL-2-THIOXODIHYDROPYRIMIDINE-4,6(1H,5H)-DIONE) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4kz8:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 20 (1,3-DIETHYL-2-THIOXODIHYDROPYRIMIDINE-4,6(1H,5H)-DIONE) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4kz9:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 41 ((4R,4AS,8AS)-4-PHENYLDECAHYDROQUINOLIN-4-OL) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE
4kza:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 48 (3-(CYCLOPROPYLSULFAMOYL)THIOPHENE-2-CARBOXYLIC ACID) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4kza:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 48 (3-(CYCLOPROPYLSULFAMOYL)THIOPHENE-2-CARBOXYLIC ACID) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
2gfg:B (GLY119) to (SER172) CRYSTAL STRUCTURE OF A PUTATIVE ADENYLATE CYCLASE (BH2851) FROM BACILLUS HALODURANS AT 2.12 A RESOLUTION | ANTIPARALLEL BARREL, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, UNKNOWN FUNCTION
4kzs:A (TYR231) to (SER283) CRYSTAL STRUCTURE OF THE SECRETED PROTEIN HP1454 FROM THE HUMAN PATHOGEN HELICOBACTER PYLORI | HELICOBACTER PYLORI, SECRETED PROTEINS, OUTER MEMBRANE, TOL-PAL SYSTEM, THREE-HELIX BUNDLE, UNKNOWN FUNCTION
3vf9:A (LEU377) to (LEU427) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE SYK CATALYTIC DOMAIN WITH THIENOPYRAZOLYLINDOLE INHIBITOR 027 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4zk3:A (HIS220) to (LYS260) PSORIASIS PATHOGENESIS - PSO P27 CONSTITUTE A COMPACT STRUCTURE FORMING LARGE AGGREGATES. LOW PH STRUCTURE | IMMUNE SYSTEM, AUTOIMMUNITY, PATHOGENESIS, PSO P27, PSO P27-COMPLEX, PSORIASIS, SCCA1, SERPINB3, HYDROLASE INHIBITOR
4zk8:A (PRO72) to (ILE111) COPPER-CONTAINING NITRITE REDUCTASE FROM THERMOPHILIC BACTERIUM GEOBACILLUS THERMODENITRIFICANS (RE-REFINED) | COPPER, OXIDOREDUCTASE, DENITRIFICATION, ELECTRON TRANSFER, NITRITE
1h24:A (ASN3) to (LEU58) CDK2/CYCLIN A IN COMPLEX WITH A 9 RESIDUE RECRUITMENT PEPTIDE FROM E2F | TRANSFERASE, CELL CYCLE, PROTEIN KINASE, CYCLIN, CDK2, RECRUITMENT, PEPTIDE SPECIFICITY, SERINE/THREONINE-PROTEIN KINASE, ATP- BINDING, CELL DIVISION, MITOSIS, PHOSPHORYLATION
4zlf:A (CYS242) to (LYS287) CELLOBIONIC ACID PHOSPHORYLASE - CELLOBIONIC ACID COMPLEX | (ALPHA/ALPHA)6 BARREL, GLYCOSIDE HYDROLASE FAMILY 94, OXIDATIVE CELLULOSE DEGRADATION SYSTEM, INTRACELLULAR ENZYME, TRANSFERASE
4zli:A (CYS242) to (LYS287) CELLOBIONIC ACID PHOSPHORYLASE - 3-O-BETA-D-GLUCOPYRANOSYL-ALPHA-D- GLUCOPYRANURONIC ACID COMPLEX | (ALPHA/ALPHA)6 BARREL, GLYCOSIDE HYDROLASE FAMILY 94, OXIDATIVE CELLULOSE DEGRADATION SYSTEM, INTRACELLULAR ENZYME, TRANSFERASE
2w00:A (ASN132) to (ILE180) CRYSTAL STRUCTURE OF THE HSDR SUBUNIT OF THE ECOR124I RESTRICTION ENZYME IN COMPLEX WITH ATP | ATP-BINDING, DNA-BINDING, RESTRICTION SYSTEM, HELICASE, HYDROLASE, R.ECOR124I, NUCLEOTIDE-BINDING, TYPE I RESTRICTION-MODIFICATION ENZYME
2w00:B (ASN132) to (ILE180) CRYSTAL STRUCTURE OF THE HSDR SUBUNIT OF THE ECOR124I RESTRICTION ENZYME IN COMPLEX WITH ATP | ATP-BINDING, DNA-BINDING, RESTRICTION SYSTEM, HELICASE, HYDROLASE, R.ECOR124I, NUCLEOTIDE-BINDING, TYPE I RESTRICTION-MODIFICATION ENZYME
4znj:A (GLU95) to (ALA139) THERMUS PHAGE P74-26 LARGE TERMINASE ATPASE DOMAIN MUTANT R139A (I 2 3 SPACE GROUP) | DNA TRANSLOCATION, VIRAL PROTEIN
3iie:A (GLU247) to (ALA285) 1-DEOXY-D-XYLULOSE 5-PHOSPHATE REDUCTOISOMERASE FROM YERSINIA PESTIS. | STRUCTURAL GENOMICS, IDP00499, XYLULOSE, REDUCTOISOMERASE, ISOPRENE BIOSYNTHESIS, METAL-BINDING, NADP, OXIDOREDUCTASE, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID
1tb6:I (PHE258) to (GLU298) 2.5A CRYSTAL STRUCTURE OF THE ANTITHROMBIN-THROMBIN-HEPARIN TERNARY COMPLEX | HEPARIN, HYDROLASE-BLOOD CLOTTING COMPLEX
3imh:B (ILE19) to (GLU61) CRYSTAL STRUCTURE OF GALACTOSE 1-EPIMERASE FROM LACTOBACILLUS ACIDOPHILUS NCFM | STRUCTURAL GENOMICS, PSI-2, EPIMERASE, GALACTOSE, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ISOMERASE
3io5:A (ASP219) to (GLY280) CRYSTAL STRUCTURE OF A DIMERIC FORM OF THE UVSX RECOMBINASE CORE DOMAIN FROM ENTEROBACTERIA PHAGE T4 | STORAGE DIMER, INACTIVE CONFORMATION, RECA LIKE CORE DOMAIN, ATP- BINDING, DNA DAMAGE, DNA RECOMBINATION, DNA REPAIR, DNA REPLICATION, NUCLEOTIDE-BINDING, DNA BINDING PROTEIN
3io5:B (ASP219) to (GLY280) CRYSTAL STRUCTURE OF A DIMERIC FORM OF THE UVSX RECOMBINASE CORE DOMAIN FROM ENTEROBACTERIA PHAGE T4 | STORAGE DIMER, INACTIVE CONFORMATION, RECA LIKE CORE DOMAIN, ATP- BINDING, DNA DAMAGE, DNA RECOMBINATION, DNA REPAIR, DNA REPLICATION, NUCLEOTIDE-BINDING, DNA BINDING PROTEIN
4lfi:B (VAL46) to (SER90) CRYSTAL STRUCTURE OF SCCK2 ALPHA IN COMPLEX WITH GMPPNP | PROTEIN KINASE, PROTEIN PHOSPHORYLATION, TRANSFERASE
3iq7:A (ILE490) to (LEU545) CRYSTAL STRUCTURE OF HUMAN HASPIN IN COMPLEX WITH 5-IODOTUBERCIDIN | HASPIN, GERM CELL ASSOCIATED 2, HAPLOID GERM CELL SPECIFIC NUCLEAR PROTEIN KINASE, SGC, STRUCTURAL GENOMICS CONSORTIUM, ATP-BINDING, CELL CYCLE, CHROMATIN REGULATOR, KINASE, MAGNESIUM, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2h4t:A (LEU234) to (ASP279) CRYSTAL STRUCTURE OF RAT CARNITINE PALMITOYLTRANSFERASE II | CARNITINE ACYLTRANSFERASE
4ljb:B (TYR87) to (LYS134) STRUCTURE OF A PHOTOBLEACHED STATE OF IRISFP UNDER HIGH INTENSITY LASER-LIGHT | FLUORESCENT PROTEIN, PHOTOBLEACHING, BETA-BARREL, DECARBOXYLATION
1hn0:A (GLU833) to (GLU895) CRYSTAL STRUCTURE OF CHONDROITIN ABC LYASE I FROM PROTEUS VULGARIS AT 1.9 ANGSTROMS RESOLUTION | CHONDROITINASE ABC I, CHONROITIN DIGESTION, MECHANISM, LYASE
3iwi:B (TYR262) to (ASP291) X-RAY CRYSTAL STRUCTURE OF THE EXTENDED-SPECTRUM AMPC OMEGA LOOP INSERTION (H210AAA) MUTANT BETA-LACTAMASE AT 1.64 ANGSTROM RESOLUTION | SERINE HYDROLASE, BETA-LACTAMASE, CEPHALOSPORINASE, EXTENDED-SPECTRUM ANTIBIOTIC RESISTANCE, ANTIBIOTIC RESISTANCE, HYDROLASE, PERIPLASM
2hdq:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH 2-CARBOXYTHIOPHENE | FRAGMENT-BASED BETA-LACTAMASE AMPC DRUG DESIGN, HYDROLASE
2hdr:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH 4-AMINO-3- HYDROXYBENZOIC ACID | AMPC FRAGMENT-BASED DRUG DESIGN BETA-LACTAMASE, HYDROLASE
2hdu:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH 2-ACETAMIDOTHIOPHENE-3- CARBOXYLIC ACID | AMPC BETA-LACTAMASE FRAGMENT-BASED DRUG DESIGN, HYDROLASE
4zy5:A (ILE276) to (ASN322) CRYSTAL STRUCTURE OF P21-ACTIVATED KINASE 1 IN COMPLEX WITH AN INHIBITOR COMPOUND 17 | KINASE, INHIBITOR, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3iwo:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF THE EXTENDED-SPECTRUM AMPC Y221G MUTANT BETA-LACTAMASE AT 1.90 ANGSTROM RESOLUTION | SERINE HYDROLASE, BETA-LACTAMASE, CEPHALOSPORINASE, EXTENDED-SPECTRUM ANTIBIOTIC RESISTANCE, ANTIBIOTIC RESISTANCE, HYDROLASE, PERIPLASM
3iwq:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF THE EXTENDED-SPECTRUM AMPC E219K MUTANT BETA-LACTAMASE AT 1.84 ANGSTROM RESOLUTION | SERINE HYDROLASE, BETA-LACTAMASE, CEPHALOSPORINASE, EXTENDED-SPECTRUM ANTIBIOTIC RESISTANCE, ANTIBIOTIC RESISTANCE, HYDROLASE, PERIPLASM
3ixb:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF THE EXTENDED-SPECTRUM AMPC E219K MUTANT BETA-LACTAMASE COMPLEXED WITH BENZO(B)THIOPHENE-2- BORONIC ACID (BZB) AT 1.63 ANGSTROM RESOLUTION | SERINE HYDROLASE, BETA-LACTAMASE, CEPHALOSPORINASE, EXTENDED-SPECTRUM ANTIBIOTIC RESISTANCE, ANTIBIOTIC RESISTANCE, HYDROLASE, PERIPLASM
3ixh:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF THE EXTENDED-SPECTRUM AMPC Y221G MUTANT BETA-LACTAMASE IN COMPLEX WITH CEFOTAXIME AT 2.3 ANGSTROM RESOLUTION | SERINE HYDROLASE, BETA-LACTAMASE, CEPHALOSPORINASE, EXTENDED-SPECTRUM ANTIBIOTIC RESISTANCE, ANTIBIOTIC RESISTANCE, HYDROLASE
2hij:I (PHE258) to (LEU299) CRYSTAL STRUCTURE OF P14 ALANINE VARIANT OF ANTITHROMBIN | THROMBIN, INHIBITION, HEPARIN ANALOGUE, SERINE PROTEASE 2 INHIBITOR, BLOOD CLOTTING- HYDROLASE INHIBITOR COMPLEX
2hij:L (PHE258) to (LEU299) CRYSTAL STRUCTURE OF P14 ALANINE VARIANT OF ANTITHROMBIN | THROMBIN, INHIBITION, HEPARIN ANALOGUE, SERINE PROTEASE 2 INHIBITOR, BLOOD CLOTTING- HYDROLASE INHIBITOR COMPLEX
4lna:A (ASP40) to (GLY102) CRYSTAL STRUCTURE OF PURINE NUCLEOSIDE PHOSPHORYLASE I FROM SPIROSOMA LINGUALE DSM 74, NYSGRC TARGET 029362 | STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, NYSGRC,, PSI- BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, TRANSFERASE
3vsk:A (LYS52) to (ILE113) CRYSTAL STRUCTURE OF PENICILLIN-BINDING PROTEIN 3 (PBP3) FROM METHICILIN-RESISTANT STAPHYLOCOCCUS AUREUS IN THE APO FORM. | PENICILLIN-BINDING DOMAIN, TRANSPEPTIDASE, PENICILLIN-BINDING PROTEIN
3vsk:B (LYS52) to (ILE113) CRYSTAL STRUCTURE OF PENICILLIN-BINDING PROTEIN 3 (PBP3) FROM METHICILIN-RESISTANT STAPHYLOCOCCUS AUREUS IN THE APO FORM. | PENICILLIN-BINDING DOMAIN, TRANSPEPTIDASE, PENICILLIN-BINDING PROTEIN
3vsk:B (GLY617) to (LYS678) CRYSTAL STRUCTURE OF PENICILLIN-BINDING PROTEIN 3 (PBP3) FROM METHICILIN-RESISTANT STAPHYLOCOCCUS AUREUS IN THE APO FORM. | PENICILLIN-BINDING DOMAIN, TRANSPEPTIDASE, PENICILLIN-BINDING PROTEIN
3vsl:A (LYS52) to (ILE113) CRYSTAL STRUCTURE OF PENICILLIN-BINDING PROTEIN 3 (PBP3) FROM METHICILIN-RESISTANT STAPHYLOCOCCUS AUREUS IN THE CEFOTAXIME BOUND FORM. | PENICILLIN-BINDING DOMAIN, TRANSPEPTIDASE, PENICILLIN-BINDING PROTEIN
1txn:B (ASP107) to (ASP182) CRYSTAL STRUCTURE OF COPROPORPHYRINOGEN III OXIDASE | STRUCTURAL GENOMICS, DIMER, NOVEL FOLD, PSI, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, OXIDOREDUCTASE
1tyq:F (PRO50) to (ALA98) CRYSTAL STRUCTURE OF ARP2/3 COMPLEX WITH BOUND ATP AND CALCIUM | STRUCTURAL PROTEIN
1i09:B (ASP58) to (LEU104) STRUCTURE OF GLYCOGEN SYNTHASE KINASE-3 (GSK3B) | KINASE, BETA BARREL, TRANSFERASE
3vw6:B (GLY687) to (LEU732) CRYSTAL STRUCTURE OF HUMAN APOPTOSIS SIGNAL-REGULATING KINASE 1 (ASK1) WITH IMIDAZOPYRIDINE INHIBITOR | TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1u1z:E (MSE1) to (ASP78) THE STRUCTURE OF (3R)-HYDROXYACYL-ACP DEHYDRATASE (FABZ) | DEHYDRATASE; FATTY ACID BIOSYNTHESIS; HOT DOG FOLD, LYASE
2wou:A (GLN208) to (THR251) ALK5 IN COMPLEX WITH 4-((4-((2,6-DIMETHYL-3-PYRIDYL)OXY)-2- PYRIDYL)AMINO)BENZENESULFONAMIDE | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ALK, ATP-BINDING, KINASE INHIBITOR, NUCLEOTIDE-BINDING, TGF BETA TYPE I RECEPTOR
1u2v:F (PRO50) to (ALA98) CRYSTAL STRUCTURE OF ARP2/3 COMPLEX WITH BOUND ADP AND CALCIUM | STRUCTURAL PROTEIN
1u4f:B (ASN198) to (ILE261) CRYSTAL STRUCTURE OF CYTOPLASMIC DOMAINS OF IRK1 (KIR2.1) CHANNEL | CYTOPLASMIC DOMAIN, KIR2.1, IRK1, INWARDLY RECTIFYING K CHANNEL, RECTIFICATION, ALLERGEN
1i5q:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF THE E. COLI AMPC BETA-LACTAMASE MUTANT N152A COVALENTLY ACYLATED WITH THE INHIBITORY BETA-LACTAM, MOXALACTAM | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, HYDROLASE
4lv0:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH M-AMINOPHENYL BORONIC ACID | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, BORONIC ACID, COVALENT INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4lv0:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH M-AMINOPHENYL BORONIC ACID | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, BORONIC ACID, COVALENT INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4lv2:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH [1-(6-CHLOROPYRIMIDIN-4-YL)-1H- PYRAZOL-4-YL] BORONIC ACID | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, BORONIC ACID, COVALENT INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4lv2:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH [1-(6-CHLOROPYRIMIDIN-4-YL)-1H- PYRAZOL-4-YL] BORONIC ACID | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, BORONIC ACID, COVALENT INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4lv1:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH [1-(3-CHLOROPHENYL)-1H-PYRAZOL-4- YL] BORONIC ACID | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, BORONIC ACID, COVALENT INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4lv1:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH [1-(3-CHLOROPHENYL)-1H-PYRAZOL-4- YL] BORONIC ACID | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, BORONIC ACID, COVALENT INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4lv3:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH (3,5-DI-TERT-BUTYLPHENYL) BORONIC ACID | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, BORONIC ACID, COVALENT INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3w37:A (LEU743) to (THR775) SUGAR BEET ALPHA-GLUCOSIDASE WITH ACARBOSE | ALPHA-GLUCOSIDASE, GLYCOSIDE HYDROLASE FAMILY 31, (BETA/ALPHA)8- BARREL, ACARBOSE, HYDROLASE, CARBOHYDRATE
3w38:A (LEU743) to (THR775) SUGAR BEET ALPHA-GLUCOSIDASE | ALPHA-GLUCOSIDASE, GLYCOSIDE HYDROLASE FAMILY 31, (BETA/ALPHA)8- BARREL, HYDROLASE, CARBOHYDRATE
5a4t:B (ILE165) to (THR215) DYRK1A IN COMPLEX WITH NITRILE BENZOTHIAZOLE FRAGMENT | TRANSFERASE
2hz4:B (THR243) to (GLU292) ABL KINASE DOMAIN UNLIGATED AND IN COMPLEX WITH TETRAHYDROSTAUROSPORINE | TYROSINE KINASE, TRANSFERASE
2hzm:A (GLY127) to (PHE163) STRUCTURE OF THE MEDIATOR HEAD SUBCOMPLEX MED18/20 | BETA BARREL, CHANNEL, TRANSCRIPTION
2i26:P (VAL56) to (ASP101) CRYSTAL STRUCTURE ANALYSIS OF THE NURSE SHARK NEW ANTIGEN RECEPTOR ANCESTRAL VARIABLE DOMAIN IN COMPLEX WITH LYSOZYME | IMMUNOGLOBULIN FOLD, PROTEIN-PROTEIN COMPLEX, IMMUNE SYSTEM
1iel:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH CEFTAZIDIME | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE
5a65:A (LYS114) to (LEU182) CRYSTAL STRUCTURE OF MOUSE THIAMINE TRIPHOSPHATASE IN COMPLEX WITH THIAMINE DIPHOSPHATE, ORTHOPHOSPHATE AND MAGNESIUM IONS. | TRIPHOSPHATE TUNNEL METALLOENZYME, HYDROLASE
5a65:B (LYS114) to (LEU182) CRYSTAL STRUCTURE OF MOUSE THIAMINE TRIPHOSPHATASE IN COMPLEX WITH THIAMINE DIPHOSPHATE, ORTHOPHOSPHATE AND MAGNESIUM IONS. | TRIPHOSPHATE TUNNEL METALLOENZYME, HYDROLASE
1uhg:A (ARG218) to (LEU252) CRYSTAL STRUCTURE OF S-OVALBUMIN AT 1.9 ANGSTROM RESOLUTION | ALLERGEN, EGG WHITE PROTEIN, SERPIN
3w7w:B (GLN204) to (ARG250) CRYSTAL STRUCTURE OF E. COLI YGJK E727A COMPLEXED WITH 2-O-ALPHA-D- GLUCOPYRANOSYL-ALPHA-D-GALACTOPYRANOSE | GH63, PROCESSING ALPHA-GLUCOSIDASE I, ALPHA/ALPHA BARREL, HYDROLASE
2i6l:A (MET21) to (LEU72) CRYSTAL STRUCTURE OF HUMAN MITOGEN ACTIVATED PROTEIN KINASE 6 (MAPK6) | MAPK6, ERK3, MITOGEN ACTIVATED PROTEIN KINASE 6, EXTRACELLULAR SIGNAL REGULATED KINASE 3, SERINE PHOSPHORYLATION, THREONINE PHOSPHORYLATION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
4m4r:H (TYR48) to (CYS90) EPHA4 ECTODOMAIN COMPLEX WITH EPHRIN A5 | EPH RECEPTOR EPHRIN COMPLEX, TRANSFERASE
1umg:A (ARG204) to (ALA256) CRYSTAL STRUCURE OF FRUCTOSE-1,6-BISPHOSPHATASE | FRUCTOSE-1,6-BISPHOSPHATASE, HYPERTHERMOPHILIC ARCHAEA, ALPHA-BETA- BETA-ALPHA FOUR LAYER SANDWICH, MAGNESIUM ION, PHOSPHATASE, OCTAMER, THREE METAL-ASSISTED MECHANISM, HYDROLASE
1un9:A (ARG207) to (LEU248) CRYSTAL STRUCTURE OF THE DIHYDROXYACETONE KINASE FROM C. FREUNDII IN COMPLEX WITH AMP-PNP AND MG2+ | KINASE, GLYCERONE KINASE, DHA KINASE, DIHYDROXYACETONE KINASE
1un9:B (ARG207) to (LEU248) CRYSTAL STRUCTURE OF THE DIHYDROXYACETONE KINASE FROM C. FREUNDII IN COMPLEX WITH AMP-PNP AND MG2+ | KINASE, GLYCERONE KINASE, DHA KINASE, DIHYDROXYACETONE KINASE
2wxi:A (CYS749) to (GLY805) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH SW30. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
2wxi:A (TYR813) to (LEU839) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH SW30. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
2wxm:A (TYR813) to (LEU839) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH DL06. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
4m67:A (LEU209) to (PHE257) CRYSTAL STRUCTURE OF THE HUMAN MLKL KINASE-LIKE DOMAIN | KINASE-LIKE, A SUBSTRATE OF RIP3, RIP3, SIGNALING PROTEIN
2icr:C (TYR91) to (LYS140) RED FLUORESCENT PROTEIN ZRFP574 FROM ZOANTHUS SP. | RED FLUORESCENT PROTEIN, ZRFP574, ZOANTHUS SP., CHROMOPHORE STRUCTURE, CYS-PHE LINK
2wxx:A (PHE286) to (ILE327) CRYSTAL STRUCTURE OF MOUSE ANGIOTENSINOGEN IN THE OXIDISED FORM | GLYCOPROTEIN, HYPERTENSION, VASOCONSTRICTOR, RENIN, SERPINS, VASOACTIVE, ANGIOTENSIN, HORMONE
2wxx:B (PHE286) to (LEU326) CRYSTAL STRUCTURE OF MOUSE ANGIOTENSINOGEN IN THE OXIDISED FORM | GLYCOPROTEIN, HYPERTENSION, VASOCONSTRICTOR, RENIN, SERPINS, VASOACTIVE, ANGIOTENSIN, HORMONE
2wxx:C (PHE286) to (ILE327) CRYSTAL STRUCTURE OF MOUSE ANGIOTENSINOGEN IN THE OXIDISED FORM | GLYCOPROTEIN, HYPERTENSION, VASOCONSTRICTOR, RENIN, SERPINS, VASOACTIVE, ANGIOTENSIN, HORMONE
2wxx:D (PHE286) to (LEU326) CRYSTAL STRUCTURE OF MOUSE ANGIOTENSINOGEN IN THE OXIDISED FORM | GLYCOPROTEIN, HYPERTENSION, VASOCONSTRICTOR, RENIN, SERPINS, VASOACTIVE, ANGIOTENSIN, HORMONE
2wxz:A (PHE286) to (HIS330) CRYSTAL STRUCTURE OF RAT ANGIOTENSINOGEN IN C2 SPACE GROUP | HORMONE, ANGIOTENSINOGEN, RENIN, ANGIOTENSIN, HYPERTENSION, GLYCOPROTEIN, VASOCONSTRICTOR, VASOACTIVE
2wxz:C (PHE286) to (HIS330) CRYSTAL STRUCTURE OF RAT ANGIOTENSINOGEN IN C2 SPACE GROUP | HORMONE, ANGIOTENSINOGEN, RENIN, ANGIOTENSIN, HYPERTENSION, GLYCOPROTEIN, VASOCONSTRICTOR, VASOACTIVE
2wy1:A (PHE286) to (HIS330) CRYSTAL STRUCTURE OF RAT ANGIOTENSINOGEN IN P321 SPACE GROUP | HORMONE, RENIN, ANGIOTENSIN, HYPERTENSION, GLYCOPROTEIN, VASOCONSTRICTOR, VASOACTIVE
2wy1:B (PHE286) to (HIS330) CRYSTAL STRUCTURE OF RAT ANGIOTENSINOGEN IN P321 SPACE GROUP | HORMONE, RENIN, ANGIOTENSIN, HYPERTENSION, GLYCOPROTEIN, VASOCONSTRICTOR, VASOACTIVE
2wyh:A (ASN739) to (GLU801) STRUCTURE OF THE STREPTOCOCCUS PYOGENES FAMILY GH38 ALPHA- MANNOSIDASE | HYDROLASE, GLYCOSIDASE, GLYCOSIDE HYDROLASE
4mbi:A (GLN37) to (VAL96) DISCOVERY OF PYRAZOLO[1,5A]PYRIMIDINE-BASED PIM1 INHIBITORS | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2x03:A (LEU588) to (ASP650) THE X-RAY STRUCTURE OF THE STREPTOMYCES COELICOLOR A3 CHONDROITIN AC LYASE Y253 MUTANT | HYALURONATE LYASE, LYASE, CHONDROITIN LYASE, FAMILY 8
1uv5:A (ILE62) to (LEU104) GLYCOGEN SYNTHASE KINASE 3 BETA COMPLEXED WITH 6-BROMOINDIRUBIN-3'-OXIME | TRANSFERASE, KINASE, INSULIN PATHWAY , WNT SIGNALING PATHWAY, TRANSFERASE SERINE/THREONINE-PROTEIN KINASE
3we8:A (TYR38) to (VAL96) PIM-1 KINASE IN COMPLEX WITH RUTHENIUM-BASED INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3we8:A (ASP108) to (GLU135) PIM-1 KINASE IN COMPLEX WITH RUTHENIUM-BASED INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3wel:A (THR739) to (THR775) SUGAR BEET ALPHA-GLUCOSIDASE WITH ACARVIOSYL-MALTOTRIOSE | ALPHA-GLUCOSIDASE, GLYCOSIDE HYDROLASE FAMILY 31, (BETA/ALPHA)8- BARREL, ACARBOSE DERIVATIVE, HYDROLASE
3wem:A (THR739) to (THR775) SUGAR BEET ALPHA-GLUCOSIDASE WITH ACARVIOSYL-MALTOTETRAOSE | ALPHA-GLUCOSIDASE, GLYCOSIDE HYDROLASE FAMILY 31, (BETA/ALPHA)8- BARREL, ACARBOSE DERIVATIVE, HYDROLASE
3wen:A (THR739) to (THR775) SUGAR BEET ALPHA-GLUCOSIDASE WITH ACARVIOSYL-MALTOPENTAOSE | ALPHA-GLUCOSIDASE, GLYCOSIDE HYDROLASE FAMILY 31, (BETA/ALPHA)8- BARREL, ACARBOSE DERIVATIVE, HYDROLASE
3weo:A (MET272) to (ILE311) SUGAR BEET ALPHA-GLUCOSIDASE WITH ACARVIOSYL-MALTOHEXAOSE | ALPHA-GLUCOSIDASE, GLYCOSIDE HYDROLASE FAMILY 31, (BETA/ALPHA)8- BARREL, ACARBOSE DERIVATIVE, HYDROLASE
5aeg:A (TYR202) to (LEU243) A BACTERIAL PROTEIN STUCTURE IN GLYCOSIDE HYDROLASE FAMILY 31. | HYDROLASE, GH31, ALPHA-SULFOQUINOVOSIDASE
5aeg:B (TYR202) to (LEU243) A BACTERIAL PROTEIN STUCTURE IN GLYCOSIDE HYDROLASE FAMILY 31. | HYDROLASE, GH31, ALPHA-SULFOQUINOVOSIDASE
4mf1:A (ILE369) to (LEU413) ITK KINASE DOMAIN IN COMPLEX WITH BENZOTHIAZOLE INHIBITOR 12B (1S,2S)- 2-{4-[(DIMETHYLAMINO)METHYL]PHENYL}-N-[6-(1H-PYRAZOL-4-YL)-1,3- BENZOTHIAZOL-2-YL]CYCLOPROPANECARBOXAMIDE | PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1j1b:A (ILE62) to (LEU104) BINARY COMPLEX STRUCTURE OF HUMAN TAU PROTEIN KINASE I WITH AMPPNP | COMPLEX, TAU, KINASE, AMPPNP, TRANSFERASE
1j1c:A (GLY63) to (LEU104) BINARY COMPLEX STRUCTURE OF HUMAN TAU PROTEIN KINASE I WITH ADP | COMPLEX, TAU, KINASE, ADP, TRANSFERASE
3wi9:A (PRO72) to (ILE111) CRYSTAL STRUCTURE OF COPPER NITRITE REDUCTASE FROM GEOBACILLUS KAUSTOPHILUS | CUPREDOXIN-FOLD, TRIMER, NITRITE REDUCTION, OXIDOREDUCTASE
3wia:A (PRO72) to (ILE111) CRYSTAL STRUCTURE OF THE N-TERMINAL 1-37 RESIDUES DELETED MUTANT OF GEOBACILLUS COPPER NITRITE REDUCTASE | CUPREDOXIN-FOLD, TRIMER, NITRITE REDUCTION, OXIDOREDUCTASE
3wia:B (PRO72) to (ILE111) CRYSTAL STRUCTURE OF THE N-TERMINAL 1-37 RESIDUES DELETED MUTANT OF GEOBACILLUS COPPER NITRITE REDUCTASE | CUPREDOXIN-FOLD, TRIMER, NITRITE REDUCTION, OXIDOREDUCTASE
3wia:C (PRO72) to (ILE111) CRYSTAL STRUCTURE OF THE N-TERMINAL 1-37 RESIDUES DELETED MUTANT OF GEOBACILLUS COPPER NITRITE REDUCTASE | CUPREDOXIN-FOLD, TRIMER, NITRITE REDUCTION, OXIDOREDUCTASE
3wia:D (PRO72) to (ILE111) CRYSTAL STRUCTURE OF THE N-TERMINAL 1-37 RESIDUES DELETED MUTANT OF GEOBACILLUS COPPER NITRITE REDUCTASE | CUPREDOXIN-FOLD, TRIMER, NITRITE REDUCTION, OXIDOREDUCTASE
3wia:E (PRO72) to (ILE111) CRYSTAL STRUCTURE OF THE N-TERMINAL 1-37 RESIDUES DELETED MUTANT OF GEOBACILLUS COPPER NITRITE REDUCTASE | CUPREDOXIN-FOLD, TRIMER, NITRITE REDUCTION, OXIDOREDUCTASE
3wia:F (PRO72) to (ILE111) CRYSTAL STRUCTURE OF THE N-TERMINAL 1-37 RESIDUES DELETED MUTANT OF GEOBACILLUS COPPER NITRITE REDUCTASE | CUPREDOXIN-FOLD, TRIMER, NITRITE REDUCTION, OXIDOREDUCTASE
3wia:G (PRO72) to (ILE111) CRYSTAL STRUCTURE OF THE N-TERMINAL 1-37 RESIDUES DELETED MUTANT OF GEOBACILLUS COPPER NITRITE REDUCTASE | CUPREDOXIN-FOLD, TRIMER, NITRITE REDUCTION, OXIDOREDUCTASE
3wia:H (PRO72) to (ILE111) CRYSTAL STRUCTURE OF THE N-TERMINAL 1-37 RESIDUES DELETED MUTANT OF GEOBACILLUS COPPER NITRITE REDUCTASE | CUPREDOXIN-FOLD, TRIMER, NITRITE REDUCTION, OXIDOREDUCTASE
3wia:I (PRO72) to (ILE111) CRYSTAL STRUCTURE OF THE N-TERMINAL 1-37 RESIDUES DELETED MUTANT OF GEOBACILLUS COPPER NITRITE REDUCTASE | CUPREDOXIN-FOLD, TRIMER, NITRITE REDUCTION, OXIDOREDUCTASE
3wiq:A (PHE215) to (GLU271) CRYSTAL STRUCTURE OF KOJIBIOSE PHOSPHORYLASE COMPLEXED WITH KOJIBIOSE | (ALPHA/ALPHA)6 BARREL, PHOSPHORYLASE, TRANSFERASE
3wir:A (PHE215) to (GLU271) CRYSTAL STRUCTURE OF KOJIBIOSE PHOSPHORYLASE COMPLEXED WITH GLUCOSE | (ALPHA/ALPHA)6 BARREL, PHOSPHORYLASE, TRANSFERASE
3wir:B (PHE215) to (GLU271) CRYSTAL STRUCTURE OF KOJIBIOSE PHOSPHORYLASE COMPLEXED WITH GLUCOSE | (ALPHA/ALPHA)6 BARREL, PHOSPHORYLASE, TRANSFERASE
3wir:C (PHE215) to (GLU271) CRYSTAL STRUCTURE OF KOJIBIOSE PHOSPHORYLASE COMPLEXED WITH GLUCOSE | (ALPHA/ALPHA)6 BARREL, PHOSPHORYLASE, TRANSFERASE
3wir:D (PHE215) to (GLU271) CRYSTAL STRUCTURE OF KOJIBIOSE PHOSPHORYLASE COMPLEXED WITH GLUCOSE | (ALPHA/ALPHA)6 BARREL, PHOSPHORYLASE, TRANSFERASE
1j4g:D (ASP57) to (ALA92) CRYSTAL STRUCTURE ANALYSIS OF THE TRICHOSANTHIN DELTA C7 | ANTIVIRAL, PROTEIN SYNTHESIS INHIBITOR, HYDROLASE
3wkp:A (PRO72) to (ILE111) C135A MUTANT OF GEOBACILLUS THERMODENITRIFICANS COPPER-CONTAINING NITRITE REDUCTASE IN COMPLEX WITH NITRITE | GREEK KEY BETA BARREL, NITRITE REDUCTASE, OXIDOREDUCTASE
3wkq:A (PRO72) to (ILE111) COPPER-CONTAINING NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS IN COMPLEX WITH FORMATE | GREEK KEY BETA BARREL, NITRITE REDUCTASE, OXIDOREDUCTASE
2x8e:A (LEU15) to (LEU62) DISCOVERY OF A NOVEL CLASS OF TRIAZOLONES AS CHECKPOINT KINASE INHIBITORS - HIT TO LEAD EXPLORATION | NUCLEOTIDE-BINDING, CYTOSKELETON, PHOSPHOPROTEIN, ISOPEPTIDE BOND, CELL CYCLE, TRANSFERASE, DNA DAMAGE, DNA REPAIR
3wni:A (PRO72) to (ILE111) 1.50 A RESOLUTION CRYSTAL STRUCTURE OF DIOXYGEN BOUND COPPER- CONTAINING NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS | GREEK KEY BETA BARREL, DISSIMILATORY NITRITE REDUCTASE, PERIPLASM- LIKE SPACE, OXIDOREDUCTASE
3wnj:A (PRO72) to (ILE111) 1.20 A RESOLUTION CRYSTAL STRUCTURE OF DIOXYGEN BOUND COPPER- CONTAINING NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS | GREEK KEY BETA BARREL, DISSIMILATORY NITRITE REDUCTASE, PERIPLASM- LIKE SPACE, OXIDOREDUCTASE
1v8c:A (VAL53) to (GLY109) CRYSTAL STRUCTURE OF MOAD RELATED PROTEIN FROM THERMUS THERMOPHILUS HB8 | MOAD RELATED PROTEIN, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, STRUCTURAL GENOMICS, PROTEIN BINDING
2xa4:B (GLN853) to (LEU905) INHIBITORS OF JAK2 KINASE DOMAIN | KINASE, MEMBRANE, TRANSFERASE, ATP-BINDING, PROTO-ONCOGENE, PHOSPHOPROTEIN
2j0l:A (GLY429) to (PHE468) CRYSTAL STRUCTURE OF A THE ACTIVE CONFORMATION OF THE KINASE DOMAIN OF FOCAL ADHESION KINASE WITH A PHOSPHORYLATED ACTIVATION LOOP. | FOCAL ADHESION, CELL MIGRATION, PHOSPHORYLATION, FERM, KINASE, TRANSFERASE, ATP-BINDING, INTEGRIN SIGNALING, NUCLEOTIDE-BINDING, TYROSINE-PROTEIN KINASE
4mq1:B (ARG158) to (HIS213) THE CRYSTAL STRUCTURE OF DYRK1A WITH A BOUND PYRIDO[2,3-D]PYRIMIDINE INHIBITOR | DYRK1A, DYRK1B, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ws1:A (HIS260) to (GLY289) N288Q-N321Q MUTANT BETA-LACTAMASE DERIVED FROM CHROMOHALOBACTER SP.560 (CONDITION-1B) | CEPHALOSPORINASE, HYDROLASE
3ws2:A (HIS260) to (GLN288) N288Q-N321Q MUTANT BETA-LACTAMASE DERIVED FROM CHROMOHALOBACTER SP.560 (CONDITION-1C) | CEPHALOSPORINASE, HYDROLASE
1vjy:A (GLY212) to (THR251) CRYSTAL STRUCTURE OF A NAPHTHYRIDINE INHIBITOR OF HUMAN TGF- BETA TYPE I RECEPTOR | TRANSFERASE, PROTEIN KINASE, INHIBITOR COMPLEX
1vla:B (HIS-1) to (CYS49) CRYSTAL STRUCTURE OF HYDROPEROXIDE RESISTANCE PROTEIN OSMC (TM0919) FROM THERMOTOGA MARITIMA AT 1.80 A RESOLUTION | TM0919, HYDROPEROXIDE RESISTANCE PROTEIN OSMC, STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI, JOINT CENTER FOR STRUCTURAL GENOMICS, OXIDOREDUCTASE
1jow:B (GLN12) to (GLU69) CRYSTAL STRUCTURE OF A COMPLEX OF HUMAN CDK6 AND A VIRAL CYCLIN | CDK-CYCLIN COMPLEX, CYCLIN FOLD, CELL CYCLE/TRANSFERASE COMPLEX
1vly:A (GLN142) to (LEU177) CRYSTAL STRUCTURE OF A PUTATIVE AMINOMETHYLTRANSFERASE (YGFZ) FROM ESCHERICHIA COLI AT 1.30 A RESOLUTION | STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI, TRANSFERASE
2xiz:A (TYR38) to (VAL96) PROTEIN KINASE PIM-1 IN COMPLEX WITH FRAGMENT-3 FROM CRYSTALLOGRAPHIC FRAGMENT SCREEN | PHOSPHORYLATION, TRANSFERASE
2xiz:A (ASP108) to (GLU135) PROTEIN KINASE PIM-1 IN COMPLEX WITH FRAGMENT-3 FROM CRYSTALLOGRAPHIC FRAGMENT SCREEN | PHOSPHORYLATION, TRANSFERASE
5awg:H (ASP6) to (GLY49) CRYSTAL STRUCTURE OF HG-BOUND SUFB-SUFC-SUFD COMPLEX FROM ESCHERICHIA COLI | IRON-SULFUR CLUSTERS, IRON-SULFUR PROTEINS, ABC PROTEINS, ABC ATPASE, TRANSPORT PROTEIN-PROTEIN BINDING COMPLEX
1jrr:A (LEU241) to (ILE286) HUMAN PLASMINOGEN ACTIVATOR INHIBITOR-2.[LOOP (66-98) DELETIONMUTANT] COMPLEXED WITH PEPTIDE MIMICKING THE REACTIVE CENTER LOOP | SERPIN, PEPTIDE BINDING, PEPTIDE BINDING PROTEIN
1vrq:A (MET756) to (GLY802) CRYSTAL STRUCTURE OF HETEROTETRAMERIC SARCOSINE OXIDASE FROM CORYNEBACTERIUM SP. U-96 IN COMPLEX WITH FOLINIC ACID | HETEROTETRAMERIC SARCOSINE OXIDASE, FLAVOENZYME, OXIDOREDUCTASE
4mxz:B (LEU273) to (LEU308) SRC M314L T338M DOUBLE MUTANT BOUND TO KINASE INHIBITOR BOSUTINIB | KINASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3j7x:B (MET51) to (VAL148) CAPSID EXPANSION MECHANISM OF BACTERIOPHAGE T7 REVEALED BY MULTI-STATE ATOMIC MODELS DERIVED FROM CRYO-EM RECONSTRUCTIONS | MATURATION, DNA PACKAGING, PROCAPSID, NON-COVALENT TOPOLOGICAL LINKING, VIRUS
4myh:A (ASP435) to (ARG484) STRUCTURE OF THE GLUTATHIONE BOUND MITOCHONDRIAL ABC TRANSPORTER, ATM1 | ABC TRANSPORTER, MEMBRANE TRANSPORT, MITOCHONDRIAL INNER MEMBRANE, GLUTATHIONE, TRANSPORT PROTEIN
1vz7:B (LYS154) to (VAL212) ORNITHINE ACETYLTRANSFERASE (ORF6 GENE PRODUCT - CLAVULANIC ACID BIOSYNTHESIS) FROM STREPTOMYCES CLAVULIGERUS | TRANSFERASE, ORNITHINE ACETYLTRANSFERASE, CLAVULANIC ACID, N-ACETYL- ORNITHINE, N-ACETYL-GLUTAMATE, ANTIBIOTIC
1jvq:L (PHE258) to (LEU299) CRYSTAL STRUCTURE AT 2.6A OF THE TERNARY COMPLEX BETWEEN ANTITHROMBIN, A P14-P8 REACTIVE LOOP PEPTIDE, AND AN EXOGENOUS TETRAPEPTIDE | LOOP-SHEET POLYMER, BETA-BARREL, BLOOD CLOTTING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1jxf:A (SER19) to (LEU56) SOLUTION STRUCTURE OF REDUCED CU(I) PLASTOCYANIN FROM SYNECHOCYSTIS PCC6803 | COPPER PROTEIN BETA BARREL ELECTRON TRANSFER, PROTON TRANSPORT
3x1e:A (PRO72) to (ILE111) STRUCTURE OF COPPER-CONTAINING NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS WITHOUT CHLORIDE | BETA BARREL, NITRITE REDUCTION, OXIDOREDUCTASE
3x1f:A (PRO72) to (ILE111) H294M MUTANT OF COPPER-CONTAINING NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS | BETA BARREL, NITRITE REDUCTION, OXIDOREDUCTASE
3x1g:A (PRO72) to (ILE111) H294M MUTANT OF COPPER-CONTAINING NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS SHOWING TWO COORDINATION GEOMETRIES AT THE T2CU SITE | BETA BARREL, NITRITE REDUCTION, OXIDOREDUCTASE
2jam:A (LEU29) to (LYS75) CRYSTAL STRUCTURE OF HUMAN CALMODULIN-DEPENDENT PROTEIN KINASE I G | TRANSFERASE, KINASE, MEMBRANE, ATP-BINDING, PRENYLATION, SERINE/THREONINE-PROTEIN KINASE, ALTERNATIVE SPLICING, PROTEIN SERINE/THREONINE KINASE, CALMODULIN BINDING, CALMODULIN-BINDING, NUCLEOTIDE BINDING, NUCLEOTIDE-BINDING, LIPOPROTEIN, POLYMORPHISM, GOLGI APPARATUS, PHOSPHORYLATION, ALLOSTERIC ENZYME
2jam:B (LEU29) to (LYS74) CRYSTAL STRUCTURE OF HUMAN CALMODULIN-DEPENDENT PROTEIN KINASE I G | TRANSFERASE, KINASE, MEMBRANE, ATP-BINDING, PRENYLATION, SERINE/THREONINE-PROTEIN KINASE, ALTERNATIVE SPLICING, PROTEIN SERINE/THREONINE KINASE, CALMODULIN BINDING, CALMODULIN-BINDING, NUCLEOTIDE BINDING, NUCLEOTIDE-BINDING, LIPOPROTEIN, POLYMORPHISM, GOLGI APPARATUS, PHOSPHORYLATION, ALLOSTERIC ENZYME
1w2m:F (LEU352) to (VAL423) CA-SUBSTITUTED FORM OF E. COLI AMINOPEPTIDASE P | HYDROLASE, PROLINE-SPECIFIC PEPTIDASE, METALLOENZYME, PITA- BREAD FOLD, METALLOPROTEASE
3zc6:C (GLY829) to (LEU878) CRYSTAL STRUCTURE OF JAK3 KINASE DOMAIN IN COMPLEX WITH AN INDAZOLE SUBSTITUTED PYRROLOPYRAZINE INHIBITOR | TRANSFERASE, SCID, SEVERE COMBINED IMMUNODEFICIENCY, STAT5, STAT6, INTERLEUKIN-2, COMMON-GAMMA CHAIN, ATP SITE KINASE INHIBITOR, CANCER
2xsg:A (THR227) to (VAL268) STRUCTURE OF THE GH92 FAMILY GLYCOSYL HYDROLASE CCMAN5 | HYDROLASE, MANNOSIDASE
2xsg:B (THR227) to (VAL268) STRUCTURE OF THE GH92 FAMILY GLYCOSYL HYDROLASE CCMAN5 | HYDROLASE, MANNOSIDASE
3zdi:A (ASP58) to (LEU104) GLYCOGEN SYNTHASE KINASE 3 BETA COMPLEXED WITH AXIN PEPTIDE AND INHIBITOR 7D | TRANSFERASE-PEPTIDE COMPLEX, INSULIN PATHWAY, WNT SIGNALING PATHWAY, TRANSFERASE SERINE/THREONINE-PROTEIN KINASE, INHIBITOR
4naa:A (MET228) to (SER276) CRYSTAL STRUCTURE OF UVB PHOTORECEPTOR UVR8 FROM ARABIDOPSIS THALIANA AND UV-INDUCED STRUCTURAL CHANGES AT 120K | 7-BLADE BETA-PROPELLER, SIGNALING PROTEIN
4naa:B (MET228) to (SER276) CRYSTAL STRUCTURE OF UVB PHOTORECEPTOR UVR8 FROM ARABIDOPSIS THALIANA AND UV-INDUCED STRUCTURAL CHANGES AT 120K | 7-BLADE BETA-PROPELLER, SIGNALING PROTEIN
4naa:C (MET228) to (SER276) CRYSTAL STRUCTURE OF UVB PHOTORECEPTOR UVR8 FROM ARABIDOPSIS THALIANA AND UV-INDUCED STRUCTURAL CHANGES AT 120K | 7-BLADE BETA-PROPELLER, SIGNALING PROTEIN
4naa:D (MET228) to (SER276) CRYSTAL STRUCTURE OF UVB PHOTORECEPTOR UVR8 FROM ARABIDOPSIS THALIANA AND UV-INDUCED STRUCTURAL CHANGES AT 120K | 7-BLADE BETA-PROPELLER, SIGNALING PROTEIN
5brl:A (ALA48) to (ILE86) CRYSTAL STRUCTURE OF L124D STARD4 | LIPID BINDING PROTEIN, ALPHA HELIX GRIP
5brl:B (ALA48) to (ILE86) CRYSTAL STRUCTURE OF L124D STARD4 | LIPID BINDING PROTEIN, ALPHA HELIX GRIP
4nc4:A (MET228) to (SER276) CRYSTAL STRUCTURE OF PHOTORECEPTOR ATUVR8 MUTANT W285F AND LIGHT- INDUCED STRUCTURAL CHANGES AT 120K | 7-BLADE BETA-PROPELLER, SIGNALING PROTEIN
4nc4:B (MET228) to (SER276) CRYSTAL STRUCTURE OF PHOTORECEPTOR ATUVR8 MUTANT W285F AND LIGHT- INDUCED STRUCTURAL CHANGES AT 120K | 7-BLADE BETA-PROPELLER, SIGNALING PROTEIN
4nc4:C (MET228) to (SER276) CRYSTAL STRUCTURE OF PHOTORECEPTOR ATUVR8 MUTANT W285F AND LIGHT- INDUCED STRUCTURAL CHANGES AT 120K | 7-BLADE BETA-PROPELLER, SIGNALING PROTEIN
4nc4:D (MET228) to (SER276) CRYSTAL STRUCTURE OF PHOTORECEPTOR ATUVR8 MUTANT W285F AND LIGHT- INDUCED STRUCTURAL CHANGES AT 120K | 7-BLADE BETA-PROPELLER, SIGNALING PROTEIN
1k32:A (THR637) to (GLU668) CRYSTAL STRUCTURE OF THE TRICORN PROTEASE | PROTEIN DEGRADATION, SUBSTRATE GATING, SERINE PROTEASE, BETA PROPELLER, PROTEASOME, HYDROLASE
1k32:C (THR637) to (GLU668) CRYSTAL STRUCTURE OF THE TRICORN PROTEASE | PROTEIN DEGRADATION, SUBSTRATE GATING, SERINE PROTEASE, BETA PROPELLER, PROTEASOME, HYDROLASE
1k32:F (THR637) to (GLU668) CRYSTAL STRUCTURE OF THE TRICORN PROTEASE | PROTEIN DEGRADATION, SUBSTRATE GATING, SERINE PROTEASE, BETA PROPELLER, PROTEASOME, HYDROLASE
1k3s:A (LEU22) to (SER66) TYPE III SECRETION CHAPERONE SIGE | TYPE III, SECRETION, CHAPERONE, SIGE
2jld:B (ASP58) to (LEU104) EXTREMELY TIGHT BINDING OF RUTHENIUM COMPLEX TO GLYCOGEN SYNTHASE KINASE 3 | WNT SIGNALING PATHWAY, SERINE/THREONINE-PROTEIN KINASE, RUTHENIUM GLYCOGEN SYNTHASE KINASE PICOMOLAR, NUCLEOTIDE-BINDING, ALTERNATIVE SPLICING, KINASE, TRANSFERASE, ATP-BINDING, PHOSPHOPROTEIN
5bvk:A (GLY617) to (LEU679) FRAGMENT-BASED DISCOVERY OF POTENT AND SELECTIVE DDR1/2 INHIBITORS | DDR1, TRANSFERASE
5bvw:A (LYS613) to (LEU679) FRAGMENT-BASED DISCOVERY OF POTENT AND SELECTIVE DDR1/2 INHIBITORS | DDR1, FRAGMENTS, TRANSFERASE
1k8k:F (PRO50) to (ALA98) CRYSTAL STRUCTURE OF ARP2/3 COMPLEX | BETA-PROPELLER, STRUCTURAL PROTEIN
1we5:A (GLN214) to (PHE257) CRYSTAL STRUCTURE OF ALPHA-XYLOSIDASE FROM ESCHERICHIA COLI | TIM BARREL, GLYCOSIDE HYDROLASE, GH FAMILY 31
1we5:B (GLN214) to (THR258) CRYSTAL STRUCTURE OF ALPHA-XYLOSIDASE FROM ESCHERICHIA COLI | TIM BARREL, GLYCOSIDE HYDROLASE, GH FAMILY 31
1we5:C (GLN214) to (THR258) CRYSTAL STRUCTURE OF ALPHA-XYLOSIDASE FROM ESCHERICHIA COLI | TIM BARREL, GLYCOSIDE HYDROLASE, GH FAMILY 31
1we5:D (GLN214) to (THR258) CRYSTAL STRUCTURE OF ALPHA-XYLOSIDASE FROM ESCHERICHIA COLI | TIM BARREL, GLYCOSIDE HYDROLASE, GH FAMILY 31
1we5:E (GLN214) to (THR258) CRYSTAL STRUCTURE OF ALPHA-XYLOSIDASE FROM ESCHERICHIA COLI | TIM BARREL, GLYCOSIDE HYDROLASE, GH FAMILY 31
1we5:F (GLN214) to (THR258) CRYSTAL STRUCTURE OF ALPHA-XYLOSIDASE FROM ESCHERICHIA COLI | TIM BARREL, GLYCOSIDE HYDROLASE, GH FAMILY 31
1k9a:D (LEU195) to (THR241) CRYSTAL STRUCTURE ANALYSIS OF FULL-LENGTH CARBOXYL-TERMINAL SRC KINASE AT 2.5 A RESOLUTION | CARBOXYL-TERMINAL SRC KINASE, COOH-TERMINAL SRC KINASE, CSK, SRC, SFK, SIGNAL TRANSDUCTION, SH2, SH3, SRC HOMOLOGY, TYROSINE KINASE, CYTOPLASMIC TYROSINE KINASE, CBP, ONCOGENE, CANCER, TRANSFERASE
1wlr:A (LEU352) to (VAL423) APO AMINOPEPTIDASE P FROM E. COLI | PROLINE-SPECIFIC PEPTIDASE, METALLOENZYME, PITA-BREAD FOLD, HYDROLASE
2kew:A (THR72) to (GLY129) THE SOLUTION STRUCTURE OF BACILLUS SUBTILIS SR211 START DOMAIN BY NMR SPECTROSCOPY | BACILLUS SUBTILIS, PROTEIN YNDB, START DOMAIN, NMR RESONANCE ASSIGNMENTS, LIPID BINDING, STRUCTURAL GENOMICS, UNKNOWN FUNCTION, PSI-2, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, NESG
2y3a:A (TYR833) to (GLU881) CRYSTAL STRUCTURE OF P110BETA IN COMPLEX WITH ICSH2 OF P85BETA AND THE DRUG GDC-0941 | TRANSFERASE, PHOSPHOINOSITIDE 3-KINASE, RTK
4nk3:A (TYR286) to (ASN314) AMP-C BETA-LACTAMASE (PSEUDOMONAS AERUGINOSA) IN COMPLEX WITH MK-7655 | HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1kds:A (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH THE INHIBITOR 3-NITROPHENYLBORONIC ACID | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, PHENYLBORONIC ACID INHIBITOR COMPLEX
1kds:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH THE INHIBITOR 3-NITROPHENYLBORONIC ACID | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, PHENYLBORONIC ACID INHIBITOR COMPLEX
1kdw:A (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH THE INHIBITOR 4-CARBOXYPHENYLBORONIC ACID | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, PHENYLBORONIC ACID INHIBITOR
1kdw:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH THE INHIBITOR 4-CARBOXYPHENYLBORONIC ACID | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, PHENYLBORONIC ACID INHIBITOR
1ke3:A (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH THE INHIBITOR 4,4'-BIPHENYLDIBORONIC ACID | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, PHENYLBORONIC ACID INHIBITOR
1ke3:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH THE INHIBITOR 4,4'-BIPHENYLDIBORONIC ACID | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, PHENYLBORONIC ACID INHIBITOR
1ke4:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE
1wop:A (TYR169) to (ILE217) CRYSTAL STRUCTURE OF T-PROTEIN OF THE GLYCINE CLEAVAGE SYSTEM | AMINOMETHYLTRANSFERASE, T-PROTEIN, FOLINIC ACID
1wor:A (TYR169) to (ILE217) CRYSTAL STRUCTURE OF T-PROTEIN OF THE GLYCINE CLEAVAGE SYSTEM | AMINOMETHYLTRANSFERASE, T-PROTEIN, DIHYDROLIPOIC ACID
1wos:A (TYR169) to (ILE217) CRYSTAL STRUCTURE OF T-PROTEIN OF THE GLYCINE CLEAVAGE SYSTEM | AMINOMETHYLTRANSFERASE, T-PROTEIN
1wq7:A (ASP104) to (ASN174) CRYSTAL STRUCTURE OF BIOTIN-(ACETYL-COA-CARBOXYLASE) LIGASE FROM PYROCOCCUS HORIKOSHII OT3 | BIOTIN BIOSYNTHESIS, DIMER, STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, LIGASE
2y6o:A (ILE627) to (PHE667) CRYSTAL STRUCTURE OF EPHA4 KINASE DOMAIN IN COMPLEX WITH DASATINIB. | SIGNALLING PROTEIN, TRANSFERASE
1wsr:B (MET177) to (LYS221) CRYSTAL STRUCTURE OF HUMAN T-PROTEIN OF GLYCINE CLEAVAGE SYSTEM | GLYCINE-CLEAVAGE SYTEM, AMINOMETHYL TRANSFERASE
1wsv:A (MET177) to (LYS221) CRYSTAL STRUCTURE OF HUMAN T-PROTEIN OF GLYCINE CLEAVAGE SYSTEM | GLYCINE-CLEAVAGE SYTEM, AMINOMETHYL TRANSFERASE
1wsv:B (MET177) to (LYS221) CRYSTAL STRUCTURE OF HUMAN T-PROTEIN OF GLYCINE CLEAVAGE SYSTEM | GLYCINE-CLEAVAGE SYTEM, AMINOMETHYL TRANSFERASE
2l8o:A (ASP78) to (LEU137) SOLUTION STRUCTURE OF CHR148 FROM CYTOPHAGA HUTCHINSONII, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM TARGET CHR148 | MIXED ALPHA-BETA PROTEIN, PSI-BIOLOGY, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, NESG, UNKNOWN FUNCTION
3jbh:A (ASN559) to (LYS596) TWO HEAVY MEROMYOSIN INTERACTING-HEADS MOTIFS FLEXIBLE DOCKED INTO TARANTULA THICK FILAMENT 3D-MAP ALLOWS IN DEPTH STUDY OF INTRA- AND INTERMOLECULAR INTERACTIONS | MYOSIN INTERACTING-HEADS MOTIF, CRYO-EM, THICK FILAMENT, FLEXIBLE DOCKING, SINGLE PARTICLE RECONSTRUCTION, ITERATIVE HELICAL REAL SPACE RECONSTRUCTION (IHRSR), INTER- AND INTRAMOLECULAR INTERACTIONS, MYOSIN REGULATION, SUPER-RELAXATION, STRIATED MUSCLE, TARANTULA, CONTRACTILE PROTEIN
5c26:A (LEU377) to (LEU427) CRYSTAL STRUCTURE OF SYK IN COMPLEX WITH COMPOUND 1 | SPLEEN TYROSINE KINASE, INHIBITOR, TRANSFERASE-INHIBITOR COMPLEX
5c27:A (LEU377) to (LEU427) CRYSTAL STRUCTURE OF SYK IN COMPLEX WITH COMPOUND 2 | SPLEEN TYROSINE KINASE, INHIBITOR, TRANSFERASE-INHIBITOR COMPLEX
3zrk:A (ILE62) to (LEU104) IDENTIFICATION OF 2-(4-PYRIDYL)THIENOPYRIDINONES AS GSK-3BETA INHIBITORS | TRANSFERASE-PEPTIDE COMPLEX, KINASE
3zrk:B (ILE62) to (LEU104) IDENTIFICATION OF 2-(4-PYRIDYL)THIENOPYRIDINONES AS GSK-3BETA INHIBITORS | TRANSFERASE-PEPTIDE COMPLEX, KINASE
3zrl:B (ILE62) to (LEU104) IDENTIFICATION OF 2-(4-PYRIDYL)THIENOPYRIDINONES AS GSK-3BETA INHIBITORS | TRANSFERASE-PEPTIDE COMPLEX, KINASE
2m2w:A (SER75) to (PHE116) TERNARY COMPLEX OF ASFV POL X WITH DNA AND MGDGTP | DNA POLYMERASE, ASFV POL X, NUCLEOTIDYL TRANSFERASE, TRANSFERASE-DNA COMPLEX
1x2g:C (ASP122) to (TYR211) CRYSTAL STRUCTURE OF LIPATE-PROTEIN LIGASE A FROM ESCHERICHIA COLI | LIPOATE-PROTEIN LIGASE, LIPOIC ACID, PROTEIN ACYLATION, POST-TRANSLATIONAL MODIFICATION
1x2h:C (ASP122) to (GLY212) CRYSTAL STRUCTURE OF LIPATE-PROTEIN LIGASE A FROM ESCHERICHIA COLI COMPLEXED WITH LIPOIC ACID | LIPOATE-PROTEIN LIGASE, LIPOIC ACID, PROTEIN ACYLATION, POST-TRANSLATIONAL MODIFICATION
1x31:A (MET756) to (GLY802) CRYSTAL STRUCTURE OF HETEROTETRAMERIC SARCOSINE OXIDASE FROM CORYNEBACTERIUM SP. U-96 | HETEROTETRAMERIC SARCOSINE OXIDASE, FLAVOENZYME, OXIDOREDUCTASE
1x31:C (ASN149) to (ALA196) CRYSTAL STRUCTURE OF HETEROTETRAMERIC SARCOSINE OXIDASE FROM CORYNEBACTERIUM SP. U-96 | HETEROTETRAMERIC SARCOSINE OXIDASE, FLAVOENZYME, OXIDOREDUCTASE
1x8b:A (ILE305) to (ALA351) STRUCTURE OF HUMAN WEE1A KINASE: KINASE DOMAIN COMPLEXED WITH INHIBITOR PD0407824 | KINASE, CELL CYCLE, WEE1, TRANSFERASE
1xbb:A (LEU377) to (LEU427) CRYSTAL STRUCTURE OF THE SYK TYROSINE KINASE DOMAIN WITH GLEEVEC | GLEEVEC, STI-571, IMATINIB, SYK, SPLEEN TYPROSINE KINASE, ACTIVE CONFORMATION, STRUCTURAL GENOMICS, STRUCTURAL GENOMIX, TRANSFERASE
1kvl:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC S64G MUTANT BETA-LACTAMASE IN COMPLEX WITH SUBSTRATE AND PRODUCT FORMS OF CEPHALOTHIN | AMIDE HYDROLASE, BETA-LACTAMASE, CEPHALOTHIN, SUBSTRATE- ENZYME COMPLEX, PRODUCT-ENZYME COMPLEX
1kvm:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC WT BETA-LACTAMASE IN COMPLEX WITH COVALENTLY BOUND CEPHALOTHIN | AMIDE HYDROLASE, BETA-LACTAMASE, CEPHALOTHIN, ACYL-ENZYME COMPLEX
5c98:A (VAL223) to (ILE266) 1.45A RESOLUTION STRUCTURE OF SRPN18 FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE, INSECT IMMUNITY, ENZYME INHIBITOR, UNKNOWN FUNCTION
5c98:B (VAL223) to (ILE266) 1.45A RESOLUTION STRUCTURE OF SRPN18 FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE, INSECT IMMUNITY, ENZYME INHIBITOR, UNKNOWN FUNCTION
1l0d:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC S64D MUTANT BETA-LACTAMASE | AMIDE HYDROLASE, BETA-LACTAMASE, MUTANT ENZYME
1l0e:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC K67Q MUTANT BETA-LACTAMASE | AMIDE HYDROLASE, BETA-LACTAMASE, MUTANT ENZYME
1l0f:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC N152H MUTANT BETA-LACTAMASE | AMIDE HYDROLASE, BETA-LACTAMASE, MUTANT ENZYME
1l0g:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC S64G MUTANT BETA-LACTAMASE | AMIDE HYDROLASE, BETA-LACTAMASE, MUTANT ENZYME
5ca0:C (GLY43) to (THR80) CRYSTAL STRUCTURE OF T2R-TTL-LEXIBULIN COMPLEX | INHIBITOR, COMPLEX, TUBULIN, STRUCTURAL PROTEIN
2npl:X (GLY4) to (PRO46) NMR STRUCTURE OF CARD D2 DOMAIN | COXSAKIEVIRUS AND ADENOVIRUS RECEPTOR, CELL ADHESION
2nq2:D (ALA4) to (GLY53) AN INWARD-FACING CONFORMATION OF A PUTATIVE METAL-CHELATE TYPE ABC TRANSPORTER. | PUTATIVE IRON CHELATIN ABC TRANSPORTER, ATP-BINDING PROTEIN, NUCLEOTIDE BINDING DOMAIN, TRANSMEMBRANE DOMAIN, METAL TRANSPORT
5cb4:C (GLY43) to (GLY81) CRYSTAL STRUCTURE OF T2R-TTL-TIVANTINIB COMPLEX | INHIBITOR, COMPLEX, TUBULIN, STRUCTURAL PROTEIN
1l2s:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH A DOCK-PREDICTED NON-COVALENT INHIBITOR | BETA-LACTAMASE/INHIBITOR COMPLEX, CEPHALOSPORINASE, HYDROLASE
1xgi:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH 3-(3-NITRO- PHENYLSULFAMOYL)-THIOPHENE-2-CARBOXYLIC ACID | AMPC, BETA-LACTAMASE, CEPHALOSPORINASE, SERINE HYDROLASE
2nut:A (ALA162) to (LEU204) CRYSTAL STRUCTURE OF THE HUMAN SEC23A/24A HETERODIMER, COMPLEXED WITH THE SNARE PROTEIN SEC22B | HUMAN COPII SEC23/24 COMPLEXED WITH SEC22, PROTEIN TRANSPORT
5cdz:A (TYR200) to (LEU239) CRYSTAL STRUCTURE OF CONSERPIN IN THE LATENT STATE | SERINE PROTEASE INHIBITOR, AGGREGATION RESISTANT, CONSENSUS DESIGN, STABILITY, LATENT STATE, HYDROLASE, HYDROLASE INHIBITOR
5cf8:A (GLY856) to (LEU905) CRYSTAL STRUCTURE OF JANUS KINASE 2 IN COMPLEX WITH N,N-DICYCLOPROPYL- 10-ETHYL-7-[(3-METHOXYPROPYL)AMINO] -3-METHYL-3,5,8,10- TETRAAZATRICYCLO[7.3.0.0,6] DODECA-1(9),2(6),4,7,11-PENTAENE-11- CARBOXAMIDE | KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5cf8:B (GLY856) to (LEU905) CRYSTAL STRUCTURE OF JANUS KINASE 2 IN COMPLEX WITH N,N-DICYCLOPROPYL- 10-ETHYL-7-[(3-METHOXYPROPYL)AMINO] -3-METHYL-3,5,8,10- TETRAAZATRICYCLO[7.3.0.0,6] DODECA-1(9),2(6),4,7,11-PENTAENE-11- CARBOXAMIDE | KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5chm:A (PHE258) to (ASN286) CRYSTAL STRUCTURE OF FOX-4 CEPHAMYCINASE COMPLEXED WITH CEFTAZIDIME BATSI (LP06) | BETA-LACTAMASE, HYDROLASE
1lf6:A (ASP224) to (GLU267) CRYSTAL STRUCTURE OF BACTERIAL GLUCOAMYLASE | (ALPHA/ALPHA) BARREL, 6 ALPHA-HELICAL HAIRPIN TORROID, SUPER BETA SANDWICH, CARBOHYDRASE FAMILY GH15, HYDROLASE
1lf6:B (ASP224) to (GLU267) CRYSTAL STRUCTURE OF BACTERIAL GLUCOAMYLASE | (ALPHA/ALPHA) BARREL, 6 ALPHA-HELICAL HAIRPIN TORROID, SUPER BETA SANDWICH, CARBOHYDRASE FAMILY GH15, HYDROLASE
1lf9:B (ASP224) to (GLU267) CRYSTAL STRUCTURE OF BACTERIAL GLUCOAMYLASE COMPLEXED WITH ACARBOSE | (ALPHA/ALPHA) BARREL, 6 ALPHA-HELICAL HAIRPIN TORROID, SUPER BETA SANDWICH, CARBOHYDRASE FAMILY GH15, ACARBOSE, HYDROLASE
1ll5:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC WT BETA-LACTAMASE IN COMPLEX WITH COVALENTLY BOUND IMIPENEM | BETA-LACTAMASE, CARBAPENEM, IMIPENEM, HYDROLASE
1ll9:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH AMOXICILLIN | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE, HYDROLASE
1ll9:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH AMOXICILLIN | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE, HYDROLASE
1llb:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH ATMO-PENICILLIN | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE, HYDROLASE
1llb:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH ATMO-PENICILLIN | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE, HYDROLASE
5cnt:A (ILE430) to (TYR495) CRYSTAL STRUCTURE OF THE DATP INHIBITED E. COLI CLASS IA RIBONUCLEOTIDE REDUCTASE COMPLEX BOUND TO UDP AND DATP AT 3.25 ANGSTROMS RESOLUTION | ALLOSTERY, SUBSTRATE SPECIFICITY, RIBONUCLEOTIDE REDUCTASE, NUCLEOTIDE METABOLISM, OXIDOREDUCTASE
5cnt:B (ILE430) to (ASP494) CRYSTAL STRUCTURE OF THE DATP INHIBITED E. COLI CLASS IA RIBONUCLEOTIDE REDUCTASE COMPLEX BOUND TO UDP AND DATP AT 3.25 ANGSTROMS RESOLUTION | ALLOSTERY, SUBSTRATE SPECIFICITY, RIBONUCLEOTIDE REDUCTASE, NUCLEOTIDE METABOLISM, OXIDOREDUCTASE
5cnu:A (ILE430) to (TYR495) CRYSTAL STRUCTURE OF THE DATP INHIBITED E. COLI CLASS IA RIBONUCLEOTIDE REDUCTASE COMPLEX BOUND TO ADP AND DGTP AT 3.40 ANGSTROMS RESOLUTION | ALLOSTERY, SUBSTRATE SPECIFICITY, RIBONUCLEOTIDE REDUCTASE, NUCLEOTIDE METABOLISM, OXIDOREDUCTASE
5cnu:B (ILE430) to (ASP494) CRYSTAL STRUCTURE OF THE DATP INHIBITED E. COLI CLASS IA RIBONUCLEOTIDE REDUCTASE COMPLEX BOUND TO ADP AND DGTP AT 3.40 ANGSTROMS RESOLUTION | ALLOSTERY, SUBSTRATE SPECIFICITY, RIBONUCLEOTIDE REDUCTASE, NUCLEOTIDE METABOLISM, OXIDOREDUCTASE
5cnu:D (ILE430) to (ASP494) CRYSTAL STRUCTURE OF THE DATP INHIBITED E. COLI CLASS IA RIBONUCLEOTIDE REDUCTASE COMPLEX BOUND TO ADP AND DGTP AT 3.40 ANGSTROMS RESOLUTION | ALLOSTERY, SUBSTRATE SPECIFICITY, RIBONUCLEOTIDE REDUCTASE, NUCLEOTIDE METABOLISM, OXIDOREDUCTASE
5cnv:D (ILE430) to (TYR495) CRYSTAL STRUCTURE OF THE DATP INHIBITED E. COLI CLASS IA RIBONUCLEOTIDE REDUCTASE COMPLEX BOUND TO GDP AND TTP AT 3.20 ANGSTROMS RESOLUTION | ALLOSTERY, SUBSTRATE SPECIFICITY, RIBONUCLEOTIDE REDUCTASE, NUCLEOTIDE METABOLISM, OXIDOREDUCTASE
4a55:A (CYS769) to (GLY828) CRYSTAL STRUCTURE OF P110ALPHA IN COMPLEX WITH ISH2 OF P85ALPHA AND THE INHIBITOR PIK-108 | TRANSFERASE, ONCOGENE, LIPID KINASE, MEMBRANE BINDING, CANCER MUTATIONS, TUMOURS, GROWTH FACTOR SIGNALLING, PI3-KINASE INHIBITOR, NON-ATP COMPETITIVE LIGAND BINDING SITE, STRUCTURE-ACTIVITY RELATIONSHIP, ENZYME REGULATION
2zau:C (PHE29) to (GLY88) CRYSTAL STRUCTURE OF AN N-TERMINALLY TRUNCATED SELENOPHOSPHATE SYNTHETASE FROM AQUIFEX AEOLICUS | INTRAMOLECULAR S-S BOND, TRIMER OF DIMERS, ATP-BINDING, KINASE, MAGNESIUM, NUCLEOTIDE-BINDING, SELENIUM, SELENOCYSTEINE, TRANSFERASE, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
2o5k:A (ILE62) to (LEU104) CRYSTAL STRUCTURE OF GSK3BETA IN COMPLEX WITH A BENZOIMIDAZOL INHIBITOR | GSK3BETA, BENZOIMIDAZOL INHIBITOR, TRANSFERASE
2zbe:A (GLU482) to (CYS525) CALCIUM PUMP CRYSTAL STRUCTURE WITH BOUND BEF3 IN THE ABSENCE OF CALCIUM AND TG | MEMBRANE PROTEIN, P-TYPE ATPASE, HAD FOLD, ALTERNATIVE SPLICING, ATP-BINDING, CALCIUM, CALCIUM TRANSPORT, ENDOPLASMIC RETICULUM, HYDROLASE, ION TRANSPORT, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, SARCOPLASMIC RETICULUM, TRANSMEMBRANE, TRANSPORT
2zbe:B (GLU482) to (CYS525) CALCIUM PUMP CRYSTAL STRUCTURE WITH BOUND BEF3 IN THE ABSENCE OF CALCIUM AND TG | MEMBRANE PROTEIN, P-TYPE ATPASE, HAD FOLD, ALTERNATIVE SPLICING, ATP-BINDING, CALCIUM, CALCIUM TRANSPORT, ENDOPLASMIC RETICULUM, HYDROLASE, ION TRANSPORT, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, SARCOPLASMIC RETICULUM, TRANSMEMBRANE, TRANSPORT
2o65:A (ASP108) to (ARG136) CRYSTAL STRUCTURE OF PIM1 WITH PENTAHYDROXYFLAVONE | PIM1, PENTAHYDROXYFLAVONE, TRANSFERASE
1lxm:A (LYS854) to (SER910) CRYSTAL STRUCTURE OF STREPTOCOCCUS AGALACTIAE HYALURONATE LYASE COMPLEXED WITH HEXASACCHARIDE UNIT OF HYALURONAN | STREPTOCOCCUS AGALACTIAE, PROTEIN-CARBOHYDRATE COMPLEX, HYALURONAN, LYASE
2zc7:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF CLASS C BETA-LACTAMASE ACT-1 | TWO-DOMAIN STRUCTURE, HYDROLASE
4okp:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH THE PRODUCT FORM OF 7-AMINO-DESACETOXYCEPHALOSPORANIC ACID | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE
4old:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH THE PRODUCT FORM OF (6R,7R)-7-AMINO-8-OXO-5-THIA-1-AZABICYCLO[4.2.0]OCT-2-ENE-2- CARBOXYLIC ACID | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE
4olg:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH COVALENTLY BOUND N-FORMYL 7-AMINOCEPHALOSPORANIC ACID | AMPC BETA-LACTAMASE, CLASS, CEPHALOSPORINASE, HYDROLASE
1m27:A (GLY49) to (GLN88) CRYSTAL STRUCTURE OF SAP/FYNSH3/SLAM TERNARY COMPLEX | SH2-SH3 INTERACTION, SIGNALING PROTEIN, TRANSFERASE
1m2r:A (VAL45) to (LEU88) CRYSTAL STRUCTURE OF 5,8-DI-AMINO-1,4-DI-HYDROXY- ANTHRAQUINONE/CK2 KINASE COMPLEX | KINASE, INHIBITOR-ENZYME COMPLEX, TRANSFERASE
2zh9:A (ASP88) to (LYS142) COMPLEX STRUCTURE OF AFCCA WITH TRNAMINIDU | TRANSFERASE/RNA, ATP-BINDING, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEOTIDYLTRANSFERASE, RNA REPAIR, RNA- BINDING, TRNA PROCESSING
5csp:A (GLY46) to (LEU88) CRYSTAL STRUCTURE OF CK2ALPHA WITH COMPOUND 5 BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
1xsi:A (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsi:B (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsi:C (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsi:D (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsi:E (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsi:F (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsj:A (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsj:B (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsj:C (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsj:D (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsj:E (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsj:F (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
4a9v:A (LYS271) to (GLY322) PSEUDOMONAS FLUORESCENS PHOX | HYDROLASE, BETA-PROPELLER
3ke6:B (GLY300) to (GLY355) THE CRYSTAL STRUCTURE OF THE RSBU AND RSBW DOMAINS OF RV1364C FROM MYCOBACTERIUM TUBERCULOSIS | ANTI-SIGMA FACTOR, ANTI-SIGMA FACTOR ANTAGONIST, PHOSPHATASE, PP2C, SERINE KINASE, ATPASE, UNKNOWN FUNCTION
1xsk:A (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE GLYCOSYL-ENZYME INTERMEDIATE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsk:B (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE GLYCOSYL-ENZYME INTERMEDIATE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsk:C (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE GLYCOSYL-ENZYME INTERMEDIATE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsk:D (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE GLYCOSYL-ENZYME INTERMEDIATE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsk:E (GLN214) to (PHE257) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE GLYCOSYL-ENZYME INTERMEDIATE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsk:F (GLN214) to (THR258) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE GLYCOSYL-ENZYME INTERMEDIATE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
2zlf:A (LYS423) to (ILE485) THE STRUCTURAL BASIS FOR PEPTIDOMIMETIC INHIBITION OF EUKARYOTIC RIBONUCLEOTIDE REDUCTASE | PEPTIDOMIMETIC INHIBITION EUKARYOTIC RIBONUCLEOTIDE REDUCTASE, ALLOSTERIC ENZYME, ATP-BINDING, CYTOPLASM, DNA REPLICATION, NUCLEOTIDE-BINDING, OXIDOREDUCTASE, PHOSPHOPROTEIN
4orm:A (CYS209) to (LEU240) CRYSTAL STRUCTURE OF PLASMODIUM FALCIPARUM DIHYDROOROTATE DEHYDROGENASE BOUND WITH INHIBITOR DSM338 (N-[3,5-DIFLUORO-4- (TRIFLUOROMETHYL)PHENYL]-5-METHYL-2-(TRIFLUOROMETHYL)[1,2, 4]TRIAZOLO[1,5-A]PYRIMIDIN-7-AMINE) | ALPHA/BETA BARREL, OXIDOREDUCTASE, FMN, MITOCHONDRIAL MEMBRANE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
5cxz:A (LEU377) to (LEU427) SYK CATALYTIC DOMAIN COMPLEXED WITH NAPHTHYRIDINE INHIBITOR | TRANSFERASE/TRANSFERASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5cz3:A (VAL78) to (TYR113) CRYSTAL STRUCTURE OF MYXOMA VIRUS M64 | HOST-RANGE, POXVIRUS, MYXOMA, BETA-SANDWICH, VIRAL PROTEIN
5cz3:B (VAL78) to (TYR113) CRYSTAL STRUCTURE OF MYXOMA VIRUS M64 | HOST-RANGE, POXVIRUS, MYXOMA, BETA-SANDWICH, VIRAL PROTEIN
4otp:A (THR180) to (GLU261) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF THE HUMAN RIOK1 ATYPICAL PROTEIN KINASE IN COMPLEX WITH ADP/MG2+ | ATYPICAL KINASE DOMAIN, RIO DOMAIN, RIBOSOME BIOGENESIS, PRE-40S, PRERIBOSOME, PHOSPHORYLATION, TRANSFERASE
1m93:B (ASN172) to (LEU214) 1.65 A STRUCTURE OF CLEAVED VIRAL SERPIN CRMA | SERPIN, CRMA, APOPTOSIS, ICE INHIBITOR, VIRAL PROTEIN
4ouc:A (ILE490) to (GLU548) STRUCTURE OF HUMAN HASPIN IN COMPLEX WITH HISTONE H3 SUBSTRATE | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE, HISTONE, KINASE SUBSTRATE COMPLEX, CHROMATIN REGULATOR
1y1q:B (LEU2044) to (GLY2085) CRYSTAL STRUCTURE OF THE URIDINE PHOSPHORYLASE FROM SALMONELLA TYPHIMURIUM IN COMPLEX WITH URIDINE-5P-MONOPHOSPHATE AND SULFATE ION AT 2.35A RESOLUTION | NUCLEOSIDE PHOSPHORYLASE, TRANSFERASE
1mdw:B (SER236) to (VAL307) CRYSTAL STRUCTURE OF CALCIUM-BOUND PROTEASE CORE OF CALPAIN II REVEALS THE BASIS FOR INTRINSIC INACTIVATION | CALPAIN CYSTEINE PROTEASE FOLD, TWO COOPERATIVE CALCIUM SITES, HELIX INSTABILITY, TRYPTOPHAN-BASED ACTIVE SITE BLOCKAGE, HYDROLASE
1mhs:A (LEU446) to (VAL484) MODEL OF NEUROSPORA CRASSA PROTON ATPASE | ION TRANSPORT, PROTON PUMP, MEMBRANE PROTEIN, P-TYPE ATPASE, ACTIVE TRANSPORT, CRYO-ELECTRON MICROSCOPY, PROTON TRANSPORT
1mhs:B (LEU446) to (VAL484) MODEL OF NEUROSPORA CRASSA PROTON ATPASE | ION TRANSPORT, PROTON PUMP, MEMBRANE PROTEIN, P-TYPE ATPASE, ACTIVE TRANSPORT, CRYO-ELECTRON MICROSCOPY, PROTON TRANSPORT
4p0f:A (PHE207) to (THR253) CLEAVED SERPIN 42DA (C 2 2 21) | SERPIN 42DA, SERPIN 4, SERINE PROTEASE INHIBITOR, NEUROSERPIN, DROSOPHILA
4afj:A (ILE62) to (LEU104) 5-ARYL-4-CARBOXAMIDE-1,3-OXAZOLES: POTENT AND SELECTIVE GSK-3 INHIBITORS | TRANSFERASE-PEPTIDE COMPLEX, KINASE
3kls:A (SER940) to (LEU992) STRUCTURE OF COMPLEMENT C5 IN COMPLEX WITH SSL7 | OB-FOLD, B-GRASP DOMAIN, FN3 DOMAIN, CLEAVAGE ON PAIR OF BASIC RESIDUES, COMPLEMENT ALTERNATE PATHWAY, COMPLEMENT PATHWAY, CYTOLYSIS, DISULFIDE BOND, GLYCOPROTEIN, IMMUNE RESPONSE, INFLAMMATORY RESPONSE, INNATE IMMUNITY, MEMBRANE ATTACK COMPLEX, SECRETED, IMMUNE SYSTEM
3kls:B (SER940) to (LEU992) STRUCTURE OF COMPLEMENT C5 IN COMPLEX WITH SSL7 | OB-FOLD, B-GRASP DOMAIN, FN3 DOMAIN, CLEAVAGE ON PAIR OF BASIC RESIDUES, COMPLEMENT ALTERNATE PATHWAY, COMPLEMENT PATHWAY, CYTOLYSIS, DISULFIDE BOND, GLYCOPROTEIN, IMMUNE RESPONSE, INFLAMMATORY RESPONSE, INNATE IMMUNITY, MEMBRANE ATTACK COMPLEX, SECRETED, IMMUNE SYSTEM
3km9:A (VAL934) to (LEU992) STRUCTURE OF COMPLEMENT C5 IN COMPLEX WITH THE C-TERMINAL BETA-GRASP DOMAIN OF SSL7 | OB-FOLD, BETA-GRASP DOMAIN, FN3 DOMAIN, CLEAVAGE ON PAIR OF BASIC RESIDUES, COMPLEMENT ALTERNATE PATHWAY, COMPLEMENT PATHWAY, CYTOLYSIS, DISULFIDE BOND, GLYCOPROTEIN, IMMUNE RESPONSE, INFLAMMATORY RESPONSE, INNATE IMMUNITY, MEMBRANE ATTACK COMPLEX, SECRETED, IMMUNE SYSTEM
3km9:B (VAL934) to (LEU992) STRUCTURE OF COMPLEMENT C5 IN COMPLEX WITH THE C-TERMINAL BETA-GRASP DOMAIN OF SSL7 | OB-FOLD, BETA-GRASP DOMAIN, FN3 DOMAIN, CLEAVAGE ON PAIR OF BASIC RESIDUES, COMPLEMENT ALTERNATE PATHWAY, COMPLEMENT PATHWAY, CYTOLYSIS, DISULFIDE BOND, GLYCOPROTEIN, IMMUNE RESPONSE, INFLAMMATORY RESPONSE, INNATE IMMUNITY, MEMBRANE ATTACK COMPLEX, SECRETED, IMMUNE SYSTEM
2zyz:D (GLY104) to (SER154) PYROBACULUM AEROPHILUM SPLICING ENDONUCLEASE | SPLICING ENDONUCLEASE, CRENARCHAEA, HETEROTETRAMER, RNA PROCESSING, ENDONUCLEASE, HYDROLASE, NUCLEASE, TRNA PROCESSING, SPLICING
4p9s:B (LEU650) to (GLY695) CRYSTAL STRUCTURE OF THE MATURE FORM OF RAT DMGDH | DIMETHYLGLYCINE DEHYDROGENASE, RAT, OXIDOREDUCTASE
4pa0:B (ILE801) to (PHE851) OMECAMTIV MERCARBIL BINDING SITE ON THE HUMAN BETA-CARDIAC MYOSIN MOTOR DOMAIN | CARDIAC, MYOSIN, MOTOR, OMECAMTIV MERCARBIL, MOTOR-FLUORESCENT PROTEIN COMPLEX
1yhs:A (GLN37) to (VAL96) CRYSTAL STRUCTURE OF PIM-1 BOUND TO STAUROSPORINE | PROTEIN KINASE, PROTO-ONCOGENE, TRANSFERASE
1mxo:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH AN M.CARBOXYPHENYLGLYCYLBORONIC ACID BEARING THE CEPHALOTHIN R1 SIDE CHAIN | AMPC, BETA-LACTAMASE, CEPHALOSPORINASE, SERINE HYDROLASE
1mxo:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH AN M.CARBOXYPHENYLGLYCYLBORONIC ACID BEARING THE CEPHALOTHIN R1 SIDE CHAIN | AMPC, BETA-LACTAMASE, CEPHALOSPORINASE, SERINE HYDROLASE
3a7i:A (LEU23) to (CYS77) HUMAN MST3 KINASE IN COMPLEX WITH ADENINE | TWO-LOBE PROTEIN KINASE FOLD, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, TRANSFERASE
1my8:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH AN M.CARBOXYPHENYLGLYCYLBORONIC ACID BEARING THE CEPHALOTHIN R1 SIDE CHAIN | AMPC, BETA-LACTAMASE, CEPHALOSPORINASE, SERINE HYDROLASE
1my8:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH AN M.CARBOXYPHENYLGLYCYLBORONIC ACID BEARING THE CEPHALOTHIN R1 SIDE CHAIN | AMPC, BETA-LACTAMASE, CEPHALOSPORINASE, SERINE HYDROLASE
3a8j:A (GLY80) to (GLY132) CRYSTAL STRUCTURE OF ET-EHRED COMPLEX | GLYCINE CLEAVAGE SYSTEM, AMINOTRANSFERASE, TRANSFERASE, LIPOYL, TRANSFERASE-TRANSPORT PROTEIN COMPLEX
3a8j:B (GLY80) to (GLY132) CRYSTAL STRUCTURE OF ET-EHRED COMPLEX | GLYCINE CLEAVAGE SYSTEM, AMINOTRANSFERASE, TRANSFERASE, LIPOYL, TRANSFERASE-TRANSPORT PROTEIN COMPLEX
3a8j:D (GLY80) to (GLY132) CRYSTAL STRUCTURE OF ET-EHRED COMPLEX | GLYCINE CLEAVAGE SYSTEM, AMINOTRANSFERASE, TRANSFERASE, LIPOYL, TRANSFERASE-TRANSPORT PROTEIN COMPLEX
3a8k:A (GLY80) to (GLY132) CRYSTAL STRUCTURE OF ETD97N-EHRED COMPLEX | GLYCINE CLEAVAGE SYSTEM, AMINOTRANSFERASE, TRANSFERASE, LIPOYL, TRANSFERASE-TRANSPORT PROTEIN COMPLEX
3a8k:C (GLY80) to (GLY132) CRYSTAL STRUCTURE OF ETD97N-EHRED COMPLEX | GLYCINE CLEAVAGE SYSTEM, AMINOTRANSFERASE, TRANSFERASE, LIPOYL, TRANSFERASE-TRANSPORT PROTEIN COMPLEX
3a8k:D (GLY80) to (GLY132) CRYSTAL STRUCTURE OF ETD97N-EHRED COMPLEX | GLYCINE CLEAVAGE SYSTEM, AMINOTRANSFERASE, TRANSFERASE, LIPOYL, TRANSFERASE-TRANSPORT PROTEIN COMPLEX
1yk3:C (TYR90) to (GLY142) CRYSTAL STRUCTURE OF RV1347C FROM MYCOBACTERIUM TUBERCULOSIS | ACYLTRANSFERASE, GCN5-RELATED FOLD, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
1yk3:G (TYR90) to (GLY142) CRYSTAL STRUCTURE OF RV1347C FROM MYCOBACTERIUM TUBERCULOSIS | ACYLTRANSFERASE, GCN5-RELATED FOLD, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
1yk3:H (TYR90) to (GLY142) CRYSTAL STRUCTURE OF RV1347C FROM MYCOBACTERIUM TUBERCULOSIS | ACYLTRANSFERASE, GCN5-RELATED FOLD, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
3a8w:A (ILE251) to (ALA300) CRYSTAL STRUCTURE OF PKCIOTA KINASE DOMAIN | PROTEIN KINASE C IOTA, KINASE DOMAIN, ATP COMPLEX, TRANSFERASE
3a8w:B (ILE251) to (SER301) CRYSTAL STRUCTURE OF PKCIOTA KINASE DOMAIN | PROTEIN KINASE C IOTA, KINASE DOMAIN, ATP COMPLEX, TRANSFERASE
5dcp:A (GLU1775) to (LEU1812) CRYSTAL STRUCTURE OF THE HUMAN FILAMIN B IG-LIKE DOMAINS 16-17 | CYTOSKELETON, ADHESION, IMMUNOGLOBULIN-LIKE, ACTIN BINDING PROTEIN, STRUCTURAL PROTEIN
3acs:A (ASP237) to (ARG297) CRYSTAL STRUCTURE OF CELLVIBRIO GILVUS CELLOBIOSE PHOSPHORYLASE W488F MUTANT | BETA-SANDWICH, (ALPHA/ALPHA)6 BARREL, PHOSPHORYLASE, GLYCOSIDE HYDROLASE FAMILY 94, TRANSFERASE
3ad7:A (MET756) to (GLY802) HETEROTETRAMERIC SARCOSINE OXIDASE FROM CORYNEBACTERIUM SP. U-96 IN COMPLEX WITH METHYLTHIO ACETATE | SARCOSINE OXIDASE, LIGAND COMPLEX, OXIDOREDUCTASE
3ad8:A (MET756) to (GLY802) HETEROTETRAMERIC SARCOSINE OXIDASE FROM CORYNEBACTERIUM SP. U-96 IN COMPLEX WITH PYRROLE 2-CARBOXYLATE | SARCOSINE OXIDASE, LIGAND COMPLEX, OXIDOREDUCTASE
3ada:A (MET756) to (GLY802) HETEROTETRAMERIC SARCOSINE OXIDASE FROM CORYNEBACTERIUM SP. U-96 IN COMPLEX WITH SULFITE | SARCOSINE OXIDASE, LIGAND COMPLEX, OXIDOREDUCTASE
3ada:C (ASN149) to (ALA196) HETEROTETRAMERIC SARCOSINE OXIDASE FROM CORYNEBACTERIUM SP. U-96 IN COMPLEX WITH SULFITE | SARCOSINE OXIDASE, LIGAND COMPLEX, OXIDOREDUCTASE
1yr3:A (ASN45) to (THR98) ESCHERICHIA COLI PURINE NUCLEOSIDE PHOSPHORYLASE II, THE PRODUCT OF THE XAPA GENE | PURINE NUCLEOSIDE PHOSPHORYLASE GUANINE XANTHINE, TRANSFERASE
1yr3:B (ASN45) to (THR98) ESCHERICHIA COLI PURINE NUCLEOSIDE PHOSPHORYLASE II, THE PRODUCT OF THE XAPA GENE | PURINE NUCLEOSIDE PHOSPHORYLASE GUANINE XANTHINE, TRANSFERASE
1yr3:F (ASN45) to (THR98) ESCHERICHIA COLI PURINE NUCLEOSIDE PHOSPHORYLASE II, THE PRODUCT OF THE XAPA GENE | PURINE NUCLEOSIDE PHOSPHORYLASE GUANINE XANTHINE, TRANSFERASE
3l4t:A (ALA240) to (ILE281) CRYSTAL COMPLEX OF N-TERMINAL HUMAN MALTASE-GLUCOAMYLASE WITH BJ2661 | GLYCOSIDE HYDROLASE FAMILY 31, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, GLYCOSIDASE, HYDROLASE, MEMBRANE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, SIGNAL-ANCHOR, SULFATION, TRANSMEMBRANE
3l4v:A (ALA240) to (ILE281) CRYSTAL COMPLEX OF N-TERMINAL HUMAN MALTASE-GLUCOAMYLASE WITH KOTALANOL | GLYCOSIDE HYDROLASE FAMILY 31, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, GLYCOSIDASE, HYDROLASE, MEMBRANE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, SIGNAL-ANCHOR, SULFATION, TRANSMEMBRANE
3l4z:A (ALA240) to (ILE281) CRYSTAL COMPLEX OF N-TERMINAL HUMAN MALTASE-GLUCOAMYLASE WITH SALACINOL | GLYCOSIDE HYDROLASE FAMILY 31, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, GLYCOSIDASE, HYDROLASE, MEMBRANE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, SIGNAL-ANCHOR, SULFATION, TRANSMEMBRANE
1ywv:A (ASP108) to (GLY137) CRYSTAL STRUCTURES OF PROTO-ONCOGENE KINASE PIM1: A TARGET OF ABERRANT SOMATIC HYPERMUTATIONS IN DIFFUSE LARGE CELL LYMPHOMA | SER/THR PROTEIN KINASE, TRANSFERASE
5dls:A (VAL12) to (LEU62) IDENTIFICATION OF NOVEL, IN VIVO ACTIVE CHK1 INHIBITORS UTILIZING STRUCTURE GUIDED DRUG DESIGN | CHK1, V158411, FRAGMENT, KINASE, TRANSFERASE
4ppj:C (GLU85) to (LYS134) CRYSTAL STRUCTURE OF PHANTA, A WEAKLY FLUORESCENT PHOTOCHROMIC GFP- LIKE PROTEIN. ON STATE | GFP, FLUORESCENT PROTEIN, CHROMOPHORE, CHROMOPROTEIN, PHOTOSWITCHING
4ppk:A (GLU85) to (LYS134) CRYSTAL STRUCTURE OF ECGP123 T69V VARIANT AT PH 7.5 | GFP, FLUORESCENT PROTEIN, CHROMOPHORE, PHOTOSWITCHING
4ppl:B (TYR87) to (LYS134) CRYSTAL STRUCTURE OF ECGP123 H193Q VARIANT AT PH 7.5 | GFP, FLUORESCENT PROTEIN, CHROMOPHORE, CHROMOPROTEIN, PHOTOSWITCHING
1zb9:A (LEU8) to (ALA60) CRYSTAL STRUCTURE OF XYLELLA FASTIDIOSA ORGANIC PEROXIDE RESISTANCE PROTEIN | OXIDOREDUCTASE
1zc2:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF PLASMID-ENCODED CLASS C BETA-LACTAMASE CMY-2 COMPLEXED WITH CITRATE MOLECULE | BETA-LACTAMASE CEPHALOSPORINASE, AMPC-TYPE, SERINE HYDROLASE, CITRATE
4px6:A (LEU377) to (LEU427) SYK CATALYTIC DOMAIN IN COMPLEX WITH A POTENT PYRIDOPYRIMIDINONE INHIBITOR | KINASE DOMAIN, PHOSPHOTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4aq0:A (THR227) to (VAL268) STRUCTURE OF THE GH92 FAMILY GLYCOSYL HYDROLASE CCMAN5 IN COMPLEX WITH DEOXYMANNOJIRIMYCIN | HYDROLASE, MANNOSIDASE
4aq0:B (THR227) to (VAL268) STRUCTURE OF THE GH92 FAMILY GLYCOSYL HYDROLASE CCMAN5 IN COMPLEX WITH DEOXYMANNOJIRIMYCIN | HYDROLASE, MANNOSIDASE
5du3:B (PRO309) to (LEU352) ACTIVE FORM OF HUMAN C1-INHIBITOR | SERINE PROTEASE INHIBITOR, HYDROLASE INHIBITOR
1zgp:A (GLY90) to (LYS138) CRYSTAL STRUCTURE OF THE DISCOSOMA RED FLUORESCENT PROTEIN (DSRED) VARIANT K70M | RFP, RED, FLUORESCENT PROTEIN, DSRED, DRFP583, CHROMOPHORE, GFP, CORAL, BETA BARREL, BETA CAN, LUMINESCENT PROTEIN
3lmi:A (PHE586) to (LEU659) CRYSTAL STRUCTURE OF THE INACTIVE ALPHA-KINASE DOMAIN OF MYOSIN HEAVY CHAIN KINASE A (D766A) COMPLEX WITH ATP | PROTEIN KINASE LIKE FOLD, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, ALPHA-KINASE, COILED COIL, WD REPEAT, TRANSFERASE
4as0:A (ASP108) to (GLU135) CYCLOMETALATED PHTHALIMIDES AS PROTEIN KINASE INHIBITORS | TRANSFERASE, PIM1, OCTASPORINE, RUTHENIUM, KINASE INHIBITOR
3lpo:A (ALA268) to (VAL309) CRYSTAL STRUCTURE OF THE N-TERMINAL DOMAIN OF SUCRASE-ISOMALTASE | GLYCOSIDE HYDROLASE FAMILY 31, ISOMALTASE, ALPHA-GLUCOSIDASE, CELL MEMBRANE, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, GLYCOSIDASE, HYDROLASE, MEMBRANE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, SIGNAL-ANCHOR, SULFATION, TRANSMEMBRANE
3lpo:B (ALA268) to (VAL309) CRYSTAL STRUCTURE OF THE N-TERMINAL DOMAIN OF SUCRASE-ISOMALTASE | GLYCOSIDE HYDROLASE FAMILY 31, ISOMALTASE, ALPHA-GLUCOSIDASE, CELL MEMBRANE, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, GLYCOSIDASE, HYDROLASE, MEMBRANE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, SIGNAL-ANCHOR, SULFATION, TRANSMEMBRANE
3lpo:C (ALA268) to (VAL309) CRYSTAL STRUCTURE OF THE N-TERMINAL DOMAIN OF SUCRASE-ISOMALTASE | GLYCOSIDE HYDROLASE FAMILY 31, ISOMALTASE, ALPHA-GLUCOSIDASE, CELL MEMBRANE, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, GLYCOSIDASE, HYDROLASE, MEMBRANE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, SIGNAL-ANCHOR, SULFATION, TRANSMEMBRANE
3lpo:D (ALA268) to (VAL309) CRYSTAL STRUCTURE OF THE N-TERMINAL DOMAIN OF SUCRASE-ISOMALTASE | GLYCOSIDE HYDROLASE FAMILY 31, ISOMALTASE, ALPHA-GLUCOSIDASE, CELL MEMBRANE, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, GLYCOSIDASE, HYDROLASE, MEMBRANE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, SIGNAL-ANCHOR, SULFATION, TRANSMEMBRANE
3lpp:A (ALA268) to (VAL309) CRYSTAL COMPLEX OF N-TERMINAL SUCRASE-ISOMALTASE WITH KOTALANOL | GLYCOSIDE HYDROLASE FAMILY 31, ISOMALTASE, ALPHA-GLUCOSIDASE, CELL MEMBRANE, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, GLYCOSIDASE, HYDROLASE, MEMBRANE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, SIGNAL-ANCHOR, SULFATION, TRANSMEMBRANE
3lpp:B (ALA268) to (VAL309) CRYSTAL COMPLEX OF N-TERMINAL SUCRASE-ISOMALTASE WITH KOTALANOL | GLYCOSIDE HYDROLASE FAMILY 31, ISOMALTASE, ALPHA-GLUCOSIDASE, CELL MEMBRANE, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, GLYCOSIDASE, HYDROLASE, MEMBRANE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, SIGNAL-ANCHOR, SULFATION, TRANSMEMBRANE
3lpp:C (ALA268) to (VAL309) CRYSTAL COMPLEX OF N-TERMINAL SUCRASE-ISOMALTASE WITH KOTALANOL | GLYCOSIDE HYDROLASE FAMILY 31, ISOMALTASE, ALPHA-GLUCOSIDASE, CELL MEMBRANE, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, GLYCOSIDASE, HYDROLASE, MEMBRANE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, SIGNAL-ANCHOR, SULFATION, TRANSMEMBRANE
3lpp:D (ALA268) to (VAL309) CRYSTAL COMPLEX OF N-TERMINAL SUCRASE-ISOMALTASE WITH KOTALANOL | GLYCOSIDE HYDROLASE FAMILY 31, ISOMALTASE, ALPHA-GLUCOSIDASE, CELL MEMBRANE, DISEASE MUTATION, DISULFIDE BOND, GLYCOPROTEIN, GLYCOSIDASE, HYDROLASE, MEMBRANE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, SIGNAL-ANCHOR, SULFATION, TRANSMEMBRANE
1zp9:D (GLY53) to (GLY131) CRYSTAL STRUCTURE OF FULL-LEGNTH A.FULGIDUS RIO1 SERINE KINASE BOUND TO ATP AND MN2+ IONS. | RIO1, RIOK1, SERINE KINASE, PROTEIN KINASE, MANGANESE, RIBOSOME BIOGENESIS, TRANSFERASE
3lsk:B (GLU432) to (GLY530) PYRANOSE 2-OXIDASE T169S ACETATE COMPLEX | OXIDOREDUCTASE, GMC OXIDOREDUCTASE, T169S MUTANT, ACETATE COMPLEX, CLOSED STATE, ROSSMANN FOLD, PHBH FOLD, HOMOTETRAMER, COVALENTLY BOUND FAD
1zxe:B (LEU605) to (ALA648) CRYSTAL STRUCTURE OF EIF2ALPHA PROTEIN KINASE GCN2: D835N INACTIVATING MUTANT IN APO FORM | TRANSLATION REGULATOR, PROTEIN KINASE, SIGNAL TRANSDUCTION, AMINO- ACID STARVATION, STARVATION STRESS RESPONSE, EIF2ALPHA KINASE, TRANSFERASE
5e68:B (LEU4) to (LEU59) HIGH RESOLUTION CRYSTAL STRUCTURE OF LUXS - QUORUM SENSOR MOLECULAR COMPLEX FROM SALMONELLA TYPHI AT 1.58 ANGSTROMS | QUROUM SENSING PROTEIN, LUXS, SALMONELLA TYPHI, S-RIBOSYLHOMOCYSTEINE LYASE, LYASE
4q7j:G (PRO391) to (TRP431) COMPLEX STRUCTURE OF VIRAL RNA POLYMERASE | RNA POLYMERASE, RNA BINDING MOTIF, RNA DEPENDENT RNA POLYMERIZATION, TRANSLATION-TRANSFERASE COMPLEX
4b0t:A (ASN52) to (ASP108) STRUCTURE OF THE PUP LIGASE PAFA OF THE PROKARYOTIC UBIQUITIN-LIKE MODIFICATION PATHWAY IN COMPLEX WITH ADP | LIGASE, PUPYLATION, DEPUPYLATION, PROKARYOTIC UBIQUITIN-LIKE PROTEIN, PROTEASOME
4b0t:B (ASN52) to (ASP108) STRUCTURE OF THE PUP LIGASE PAFA OF THE PROKARYOTIC UBIQUITIN-LIKE MODIFICATION PATHWAY IN COMPLEX WITH ADP | LIGASE, PUPYLATION, DEPUPYLATION, PROKARYOTIC UBIQUITIN-LIKE PROTEIN, PROTEASOME
5e8u:A (GLY212) to (THR251) TGF-BETA RECEPTOR TYPE 1 KINASE DOMAIN (T204D,I211V,Y249F,S280T, Y282F,S287N,A350C,L352F) | ALK5, KINASE DOMAIN, TRANSFERASE
3avv:A (PHE1087) to (TRP1126) STRUCTURE OF VIRAL RNA POLYMERASE COMPLEX 3 | RNA POLYMERASE, TRANSLATION, TRANSFERASE-RNA COMPLEX
3b2w:A (LEU251) to (GLN294) CRYSTAL STRUCTURE OF PYRIMIDINE AMIDE 11 BOUND TO LCK | LCK, KINASE DOMAIN, ALTERNATIVE SPLICING, ATP-BINDING, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, DISEASE MUTATION, HOST-VIRUS INTERACTION, LIPOPROTEIN, MEMBRANE, MYRISTATE, NUCLEOTIDE-BINDING, PALMITATE, PHOSPHORYLATION, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE
3ma3:A (GLN37) to (VAL96) CRYSTAL STRUCTURE OF HUMAN PROTO-ONCOGENE SERINE THREONINE KINASE (PIM1) IN COMPLEX WITH A CONSENSUS PEPTIDE AND A NAPHTHO-DIFURAN LIGAND | ONCOGENE, KINASE, SERINE-THREONINE, PIM1, STRUCTURAL GENOMICS CONSORTIUM, SGC, ALTERNATIVE INITIATION, ATP-BINDING, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, HOST-VIRUS INTERACTION, VIRAL IMMUNOEVASION, VIRION, VIRULENCE, CELL CYCLE, CELL MEMBRANE
5ei0:A (GLN248) to (GLY286) STRUCTURE OF RCL-CLEAVED VASPIN (SERPINA12) | SERPIN, CLEAVED, ADIPOKINE, HYDROLASE INHIBITOR
5ei0:E (GLN248) to (GLY286) STRUCTURE OF RCL-CLEAVED VASPIN (SERPINA12) | SERPIN, CLEAVED, ADIPOKINE, HYDROLASE INHIBITOR
3mej:A (PHE74) to (ASP153) CRYSTAL STRUCTURE OF PUTATIVE TRANSCRIPTIONAL REGULATOR YWTF FROM BACILLUS SUBTILIS, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM TARGET SR736 | STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, NESG, TRANSCRIPTIONAL REGULATOR
4qmp:A (GLY31) to (CYS77) MST3 IN COMPLEX WITH CDK1/2 INHIBITOR III, 5-AMINO-3-{[4- (AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4- TRIAZOLE-1-CARBOTHIOAMIDE | PROTEIN KINASE, MST3, STK24, STERILE 20-LIKE KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4be7:D (ARG131) to (ILE180) MUTANT (K220R) OF THE HSDR SUBUNIT OF THE ECOR124I RESTRICTION ENZYME IN COMPLEX WITH ATP | HYDROLASE, DNA RESTRICTION, DNA MODIFICATION
4beb:A (ASN132) to (GLN179) MUTANT (K220E) OF THE HSDR SUBUNIT OF THE ECOR124I RESTRICTION ENZYME IN COMPLEX WITH ATP | HYDROLASE, DNA MODIFICATION
4beb:B (ASN132) to (GLN179) MUTANT (K220E) OF THE HSDR SUBUNIT OF THE ECOR124I RESTRICTION ENZYME IN COMPLEX WITH ATP | HYDROLASE, DNA MODIFICATION
4beb:C (ASN132) to (ILE180) MUTANT (K220E) OF THE HSDR SUBUNIT OF THE ECOR124I RESTRICTION ENZYME IN COMPLEX WITH ATP | HYDROLASE, DNA MODIFICATION
4beb:D (ASN132) to (GLN179) MUTANT (K220E) OF THE HSDR SUBUNIT OF THE ECOR124I RESTRICTION ENZYME IN COMPLEX WITH ATP | HYDROLASE, DNA MODIFICATION
4bec:A (ASN132) to (GLN179) MUTANT (K220A) OF THE HSDR SUBUNIT OF THE ECOR124I RESTRICTION ENZYME IN COMPLEX WITH ATP | HYDROLASE, DNA MODIFICATION
4bec:B (ASN132) to (GLN179) MUTANT (K220A) OF THE HSDR SUBUNIT OF THE ECOR124I RESTRICTION ENZYME IN COMPLEX WITH ATP | HYDROLASE, DNA MODIFICATION
5er0:D (GLU352) to (GLU409) WATER-FORMING NADH OXIDASE FROM LACTOBACILLUS BREVIS (LBNOX) | NADH OXIDASE, FAD, MOLECULAR OXYGEN, OXIDOREDUCTASE
4bfr:A (CYS770) to (GLY825) DISCOVERY AND OPTIMIZATION OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS FOR THE TREATMENT OF PHOSPHATASE AND TENSIN HOMOLOGUE (PTEN)-DEFICIENT CANCERS | TRANSFERASE, INHIBITOR
4bfr:A (TYR833) to (ASN860) DISCOVERY AND OPTIMIZATION OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS FOR THE TREATMENT OF PHOSPHATASE AND TENSIN HOMOLOGUE (PTEN)-DEFICIENT CANCERS | TRANSFERASE, INHIBITOR
4bfr:B (CYS770) to (GLY825) DISCOVERY AND OPTIMIZATION OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS FOR THE TREATMENT OF PHOSPHATASE AND TENSIN HOMOLOGUE (PTEN)-DEFICIENT CANCERS | TRANSFERASE, INHIBITOR
4bfr:B (TYR833) to (ASN860) DISCOVERY AND OPTIMIZATION OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS FOR THE TREATMENT OF PHOSPHATASE AND TENSIN HOMOLOGUE (PTEN)-DEFICIENT CANCERS | TRANSFERASE, INHIBITOR
3bgz:A (GLN37) to (LYS95) HUMAN PIM-1 KINASE IN COMPLEX WITH DIPHENYL INDOLE INHIBITOR VX3 | KINASE INHIBITOR PHOSPHORYLATION, ALTERNATIVE INITIATION, ATP-BINDING, CYTOPLASM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3bgz:A (ASP108) to (GLY137) HUMAN PIM-1 KINASE IN COMPLEX WITH DIPHENYL INDOLE INHIBITOR VX3 | KINASE INHIBITOR PHOSPHORYLATION, ALTERNATIVE INITIATION, ATP-BINDING, CYTOPLASM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
5eti:A (ASN26) to (LYS76) STRUCTURE OF DEAD KINASE MAPK14 | MAPK14, DEAD KINASE, P38, INACTIVE KINASE, TRANSFERASE
4qtc:A (ILE490) to (GLU548) STRUCTURE OF HUMAN HASPIN (GSG2) IN COMPLEX WITH SCH772984 REVEALING THE FIRST TYPE-I BINDING MODE | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE, KINASE, INHIBITOR, ALLOSTERIC, STRUCTURAL GENOMICS CONSORTIUM (SGC), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5evi:A (TYR258) to (ASN286) CRYSTAL STRUCTURE OF BETA-LACTAMASE/D-ALANINE CARBOXYPEPTIDASE FROM PSEUDOMONAS SYRINGAE | ALPHA-BETA-FOLD, STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, HYDROLASE
5evi:B (TYR258) to (ASN286) CRYSTAL STRUCTURE OF BETA-LACTAMASE/D-ALANINE CARBOXYPEPTIDASE FROM PSEUDOMONAS SYRINGAE | ALPHA-BETA-FOLD, STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, HYDROLASE
3bkb:A (GLY568) to (PHE604) CRYSTAL STRUCTURE OF HUMAN FELINE SARCOMA VIRAL ONCOGENE HOMOLOGUE (V- FES) | FES, V-FES, FUJINAMI, AVIAN SARCOMA, VIRAL, ONCOGENE, FELINE SARCOMA VIRUS, SGC, STRUCTURAL GENOMICS CONSORTIUM, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3bls:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE FROM ESCHERICHIA COLI | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE
3bls:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE FROM ESCHERICHIA COLI | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE
3bm6:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH A P.CARBOXYPHENYLBORONIC ACID | AMPC, BETA-LACTAMASES, CEPHALOSPORINASE, SERINE HYDROLASE, COVALENT INHIBITION, ANTIBIOTIC RESISTANCE, PERIPLASM, HYDROLASE
3bm6:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH A P.CARBOXYPHENYLBORONIC ACID | AMPC, BETA-LACTAMASES, CEPHALOSPORINASE, SERINE HYDROLASE, COVALENT INHIBITION, ANTIBIOTIC RESISTANCE, PERIPLASM, HYDROLASE
3my0:C (VAL208) to (VAL249) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:I (VAL208) to (VAL249) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:N (VAL208) to (VAL249) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
5f7c:A (SER260) to (THR302) CRYSTAL STRUCTURE OF FAMILY 31 ALPHA-GLUCOSIDASE (BT_0339) FROM BACTEROIDES THETAIOTAOMICRON | FAMILY GLYCOSIDE HYDROLASE, HYDROLASE
5f7c:B (SER260) to (THR302) CRYSTAL STRUCTURE OF FAMILY 31 ALPHA-GLUCOSIDASE (BT_0339) FROM BACTEROIDES THETAIOTAOMICRON | FAMILY GLYCOSIDE HYDROLASE, HYDROLASE
5f7c:C (SER260) to (THR302) CRYSTAL STRUCTURE OF FAMILY 31 ALPHA-GLUCOSIDASE (BT_0339) FROM BACTEROIDES THETAIOTAOMICRON | FAMILY GLYCOSIDE HYDROLASE, HYDROLASE
5f7c:D (SER260) to (THR302) CRYSTAL STRUCTURE OF FAMILY 31 ALPHA-GLUCOSIDASE (BT_0339) FROM BACTEROIDES THETAIOTAOMICRON | FAMILY GLYCOSIDE HYDROLASE, HYDROLASE
5f7u:A (SER335) to (THR382) CYCLOALTERNAN-FORMING ENZYME FROM LISTERIA MONOCYTOGENES IN COMPLEX WITH PENTASACCHARIDE SUBSTRATE | COMPLEX, STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, SUGAR BINDING PROTEIN
4r3z:C (LYS586) to (PRO623) CRYSTAL STRUCTURE OF HUMAN ARGRS-GLNRS-AIMP1 COMPLEX | AMINO-ACYL TRNA SYNTHETASE COMPLEX, MULTI-SYNTHETASE COMPLEX, LIGATION AMINO ACID TO TRNA, PROTEIN BINDING-LIGASE COMPLEX
4r5o:D (GLY351) to (ALA383) CRYSTAL STRUCTURE OF A QUINONPROTEIN ALCOHOL DEHYDROGENASE-LIKE PROTEIN (BT1487) FROM BACTEROIDES THETAIOTAOMICRON VPI-5482 AT 2.64 A RESOLUTION | TWO DOMAIN PROTEIN, IMMUNOGLOBULIN-LIKE BETA-SANDWICH FOLD, PF16407 FAMILY, DUF5015, 7-BLADED BETA-PROPELLER, YVTN REPEAT FAMILY, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, UNKNOWN FUNCTION
3c4c:B (GLN461) to (THR508) B-RAF KINASE IN COMPLEX WITH PLX4720 | B-RAF, BRAF, RAF, PROTO-ONCOGENE, SERINE/THREONINE KINASE, ATP-BINDING, CARDIOMYOPATHY, CYTOPLASM, DISEASE MUTATION, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ZINC, ZINC-FINGER
4r71:D (PRO392) to (TRP432) STRUCTURE OF THE QBETA HOLOENZYME COMPLEX IN THE P1211 CRYSTAL FORM | OB FOLD, TRANSLATION, VIRAL PROTEIN-RIBOSOMAL PROTEIN COMPLEX
3n89:A (ILE367) to (LEU420) KH DOMAINS | KH DOMAINS, RNA BINDING, GERMLINE DEVELOPMENT, CELL CYCLE
4r84:B (LYS24) to (ALA72) CRYSTAL STRUCTURE OF SIALYLTRANSFERASE FROM PHOTOBACTERIUM DAMSELA WITH CMP-3F(A)NEU5AC BOUND | ROSSMANN FOLD, GLYCOSYLTRANSFERASE GT-B STRUCTURAL GROUP, TRANSFERASE
4r84:D (GLU25) to (ALA72) CRYSTAL STRUCTURE OF SIALYLTRANSFERASE FROM PHOTOBACTERIUM DAMSELA WITH CMP-3F(A)NEU5AC BOUND | ROSSMANN FOLD, GLYCOSYLTRANSFERASE GT-B STRUCTURAL GROUP, TRANSFERASE
3cd3:A (ILE567) to (TYR614) CRYSTAL STRUCTURE OF PHOSPHORYLATED HUMAN FELINE SARCOMA VIRAL ONCOGENE HOMOLOGUE (V-FES) IN COMPLEX WITH STAUROSPORINE AND A CONSENSUS PEPTIDE | FES, V-FES, FUJINAMI, AVIAN SARCOMA, VIRAL, ONCOGENE, FELINE SARCOMA VIRUS, ACTIVE, SGC, STRUCTURAL GENOMICS CONSORTIUM, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
4rbl:A (GLN37) to (VAL96) CRYSTAL STRUCTURE OF SER/THR KINASE PIM1 IN COMPLEX WITH MITOXANTRONE DERIVATIVES | KINASE, PHOSPHORYLATION, SIGNALING PROTEIN
4rbl:A (ASP108) to (GLU135) CRYSTAL STRUCTURE OF SER/THR KINASE PIM1 IN COMPLEX WITH MITOXANTRONE DERIVATIVES | KINASE, PHOSPHORYLATION, SIGNALING PROTEIN
3cd8:A (GLY1085) to (ASP1133) X-RAY STRUCTURE OF C-MET WITH TRIAZOLOPYRIDAZINE INHIBITOR. | C-MET, KINASE, TRIAZOLOPYRIDAZINE, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
4rc2:A (ASP108) to (GLY137) CRYSTAL STRUCTURE OF SER/THR KINASE PIM1 IN COMPLEX WITH MITOXANTRONE DERIVATIVES | KINASE, PHOSPHORYLATION, SIGNALING PROTEIN
4rc4:A (ASP108) to (GLY137) CRYSTAL STRUCTURE OF SER/THR KINASE PIM1 IN COMPLEX WITH MITOXANTRONE DERIVATIVES | KINASE, PHOSPHORYLATION, SIGNALING PROTEIN
5fk0:B (SER453) to (MET496) YEAST DELTA-COP-I MU-HOMOLOGY DOMAIN | STRUCTURAL PROTEIN, COP-I, VESICLE COAT PROTEIN
3cff:H (PHE88) to (ASN135) PHOTOSWITCHABLE RED FLUORESCENT PROTEIN PSRFP, ON-STATE | BETA BARREL, BETA CAN, CHROMOPHORE, PHOTOACTIVATION, FLUORESCENT PROTEIN
3cfu:B (GLY158) to (ILE206) CRYSTAL STRUCTURE OF THE YJHA PROTEIN FROM BACILLUS SUBTILIS. NORTHEAST STRUCTURAL GENOMICS CONSORTIUM TARGET SR562 | YJHA_BACSU, YJHA, LIPOPROTEIN, SR562, NESG, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, MEMBRANE, PALMITATE
3cgl:F (SER96) to (LYS138) CRYSTAL STRUCTURE AND RAMAN STUDIES OF DSFP483, A CYAN FLUORESCENT PROTEIN FROM DISCOSOMA STRIATA | BETA BARREL, CHROMOPHORE, LUMINESCENCE, PHOTOPROTEIN, FLUORESCENT PROTEIN
4c49:A (ILE218) to (LEU258) REACTIVE LOOP CLEAVED HUMAN CBG IN COMPLEX WITH CORTISOL | TRANSPORT PROTEIN, CORTICOSTEROID BINDING GLOBULIN, SERPIN, HORMONE CARRIER
4c61:B (LEU852) to (LEU905) INHIBITORS OF JAK2 KINASE DOMAIN | KINASE, TRANSFERASE
4c62:B (HIS848) to (LEU905) INHIBITORS OF JAK2 KINASE DOMAIN | TRANSFERASE
4c9c:A (HIS80) to (HIS155) CRYSTAL STRUCTURE OF THE STRAWBERRY PATHOGENESIS-RELATED 10 (PR-10) FRA A 1E PROTEIN (FORM A) | START, PYR/PYL/RCAR, ALLERGEN, BET V 1
4caa:A (PRO228) to (LEU267) CLEAVED ANTICHYMOTRYPSIN T345R | SERPIN, SERINE PROTEASE INHIBITOR, ANTICHYMOTRYPSIN
5fri:A (GLY212) to (THR251) ALK5 IN COMPLEX WITHA AN N-(4-ANILINO-2-PYRIDYL)ACETAMIDE INHIBITOR. | TRANSFERASE
3nqn:A (LEU81) to (LEU154) CRYSTAL STRUCTURE OF A PROTEIN WITH UNKNOWN FUNCTION. (DR_2006) FROM DEINOCOCCUS RADIODURANS AT 1.88 A RESOLUTION | PROTEIN WITH UNKNOWN FUNCTION, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, UNKNOWN FUNCTION
4rob:A (PHE234) to (ILE276) 2.8A RESOLUTION STRUCTURE OF SRPN2 (K198C) FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE INHIBITOR, INSECT IMMUNITY, HYDROLASE INHIBITOR
4rob:B (PHE234) to (ILE276) 2.8A RESOLUTION STRUCTURE OF SRPN2 (K198C) FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE INHIBITOR, INSECT IMMUNITY, HYDROLASE INHIBITOR
4rob:C (PHE234) to (ILE276) 2.8A RESOLUTION STRUCTURE OF SRPN2 (K198C) FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE INHIBITOR, INSECT IMMUNITY, HYDROLASE INHIBITOR
4ro9:B (PHE234) to (ILE276) 2.0A RESOLUTION STRUCTURE OF SRPN2 (S358E) FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE INHIBITOR, INSECT IMMUNITY, HYDROLASE INHIBITOR
4ro9:C (PHE234) to (ILE276) 2.0A RESOLUTION STRUCTURE OF SRPN2 (S358E) FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE INHIBITOR, INSECT IMMUNITY, HYDROLASE INHIBITOR
4rsq:A (PHE234) to (ILE276) 2.9A RESOLUTION STRUCTURE OF SRPN2 (K198C/E359C) FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE, INSECT IMMUNITY, HYDROLASE INHIBITOR
4rsq:B (PHE234) to (ILE276) 2.9A RESOLUTION STRUCTURE OF SRPN2 (K198C/E359C) FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE, INSECT IMMUNITY, HYDROLASE INHIBITOR
4rsq:C (PHE234) to (ILE276) 2.9A RESOLUTION STRUCTURE OF SRPN2 (K198C/E359C) FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE, INSECT IMMUNITY, HYDROLASE INHIBITOR
4rsq:E (PHE234) to (ILE276) 2.9A RESOLUTION STRUCTURE OF SRPN2 (K198C/E359C) FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE, INSECT IMMUNITY, HYDROLASE INHIBITOR
4rsq:F (PHE234) to (ILE276) 2.9A RESOLUTION STRUCTURE OF SRPN2 (K198C/E359C) FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE, INSECT IMMUNITY, HYDROLASE INHIBITOR
4rsq:G (PHE234) to (ILE276) 2.9A RESOLUTION STRUCTURE OF SRPN2 (K198C/E359C) FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE, INSECT IMMUNITY, HYDROLASE INHIBITOR
4rsq:H (PHE234) to (ILE276) 2.9A RESOLUTION STRUCTURE OF SRPN2 (K198C/E359C) FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE, INSECT IMMUNITY, HYDROLASE INHIBITOR
4rsq:L (PHE234) to (ILE276) 2.9A RESOLUTION STRUCTURE OF SRPN2 (K198C/E359C) FROM ANOPHELES GAMBIAE | SERPIN, SERINE PROTEASE, INSECT IMMUNITY, HYDROLASE INHIBITOR
3ctt:A (ALA240) to (ILE281) CRYSTAL COMPLEX OF N-TERMINAL HUMAN MALTASE-GLUCOAMYLASE WITH CASUARINE | GLYCOSYL HYDROLASE FAMILY 31, ALPHA-GLUCOSIDASE, GLYCOPROTEIN, GLYCOSIDASE, MEMBRANE, MULTIFUNCTIONAL ENZYME, SIGNAL-ANCHOR, SULFATION, TRANSMEMBRANE, HYDROLASE
3cu7:A (VAL934) to (VAL991) HUMAN COMPLEMENT COMPONENT 5 | MG DOMAIN, COMPLEMENT, INFLAMMATION, ANAPHYLATOXIN, CLEAVAGE ON PAIR OF BASIC RESIDUES, COMPLEMENT ALTERNATE PATHWAY, COMPLEMENT PATHWAY, CYTOLYSIS, GLYCOPROTEIN, IMMUNE RESPONSE, INFLAMMATORY RESPONSE, INNATE IMMUNITY, MEMBRANE ATTACK COMPLEX, SECRETED, IMMUNE SYSTEM
3cu7:B (VAL934) to (VAL991) HUMAN COMPLEMENT COMPONENT 5 | MG DOMAIN, COMPLEMENT, INFLAMMATION, ANAPHYLATOXIN, CLEAVAGE ON PAIR OF BASIC RESIDUES, COMPLEMENT ALTERNATE PATHWAY, COMPLEMENT PATHWAY, CYTOLYSIS, GLYCOPROTEIN, IMMUNE RESPONSE, INFLAMMATORY RESPONSE, INNATE IMMUNITY, MEMBRANE ATTACK COMPLEX, SECRETED, IMMUNE SYSTEM
3o0v:A (TYR306) to (LYS351) CRYSTAL STRUCTURE OF THE CALRETICULIN LECTIN DOMAIN | JELLY ROLL FOLD, CHAPERONE, CARBOHYDRATE BINDING; CALCIUM BINDING
4rx7:A (LEU377) to (LEU427) SYK CATALYTIC DOMAIN COMPLEXED WITH A POTENT TRIAZINE INHIBITOR | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5fyk:H (ASP56) to (ILE89) CRYSTAL STRUCTURE AT 3.7 A RESOLUTION OF FULLY GLYCOSYLATED HIV-1 CLADE JR-FL SOSIP.664 PREFUSION ENV TRIMER IN COMPLEX WITH BROADLY NEUTRALIZING ANTIBODIES PGT122, 35O22 AND VRC01 | VIRAL PROTEIN, HIV, ENVELOPE, GLYCAN, TRIMER
3o86:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A SULFONAMIDE BORONIC ACID INHIBITOR | CONTAINS ALPHA HELICES AND A BETA SANDWICH / BETA-LACTAMASE-LIKE FOLD / AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE
3o87:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A SULFONAMIDE BORONIC ACID INHIBITOR | CONTAINS ALPHA HELICES AND A BETA SANDWICH / BETA-LACTAMASE-LIKE FOLD / AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE
3o88:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A SULFONAMIDE BORONIC ACID INHIBITOR | CONTAINS ALPHA HELICES AND A BETA SANDWICH / BETA-LACTAMASE-LIKE FOLD / AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE
3o88:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A SULFONAMIDE BORONIC ACID INHIBITOR | CONTAINS ALPHA HELICES AND A BETA SANDWICH / BETA-LACTAMASE-LIKE FOLD / AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE
4crl:A (VAL27) to (GLU72) CRYSTAL STRUCTURE OF HUMAN CDK8-CYCLIN C IN COMPLEX WITH CORTISTATIN A | TRANSFERASE, CYCLIN-DEPENDENT KINASE 8, CDK8, CYCLIN C, CCNC, CORTISTATIN A, MEDIATOR KINASE, MEDIATOR COMPLEX, SUPER-ENHANCER, TRANSCRIPTION
5g5h:B (HIS226) to (GLN274) ESCHERICHIA COLI PERIPLAMIC ALDEHYDE OXIDASE R440H MUTANT | OXIDOREDUCTASE, PAOABC, XANTHINE OXIDASE FAMILY, HETEROTRIMER, E.COLI DETOXIFICATION,
4tn6:A (ILE15) to (GLN60) CK1D IN COMPLEX WITH INHIBITOR | SER/THR KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ocs:A (LEU405) to (GLU445) CRYSTAL STRUCTURE OF BRUTON'S TYROSINE KINASE IN COMPLEX WITH INHIBITOR CGI1746 | TYROSINE KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4toz:A (ALA211) to (GLY260) MPPA PERIPLASMIC MUREIN TRIPEPTIDE BINDING PROTEIN, UNLIGANDED OPEN FORM | PERIPLASMIC LIGAND BINDING PROTEIN, MUREIN TRIPEPTIDE BINDING PROTEIN, PEPTIDE BINDING PROTEIN
4toz:B (ALA211) to (GLY260) MPPA PERIPLASMIC MUREIN TRIPEPTIDE BINDING PROTEIN, UNLIGANDED OPEN FORM | PERIPLASMIC LIGAND BINDING PROTEIN, MUREIN TRIPEPTIDE BINDING PROTEIN, PEPTIDE BINDING PROTEIN
4trl:A (GLY620) to (GLN669) STRUCTURE OF EPHRIN TYPE-A RECEPTOR 2 | ACTIVE STATE, PHOSPHORYLATED
5ghv:A (LEU377) to (LEU427) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5ghv:B (LEU377) to (LEU427) CRYSTAL STRUCTURE OF AN INHIBITOR-BOUND SYK | SYK KINASE, INHIBITOR, SPLEEN TYROSINE KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4tvy:B (ASP122) to (GLY212) APO RESORUFIN LIGASE | E. COLI LPLA, COMPUTATIONAL ENZYME DESIGN, TRANSFERASE
3dlz:A (ILE490) to (LEU545) CRYSTAL STRUCTURE OF HUMAN HASPIN IN COMPLEX WITH AMP | HASPIN, GERM CELL ASSOCIATED 2, HAPLOID GERM CELL SPECIFIC NUCLEAR PROTEIN KINASE, SGC, STRUCTURAL GENOMICS CONSORTIUM, ATP-BINDING, CELL CYCLE, CHROMATIN REGULATOR, MAGNESIUM, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4d4q:A (VAL180) to (HIS221) CRYSTAL STRUCTURE OF KTI13/ATS1 | TRANSLATION, TRNA MODIFICATION, DIPHTHAMIDE MODIFICATION
4d4q:B (VAL180) to (HIS221) CRYSTAL STRUCTURE OF KTI13/ATS1 | TRANSLATION, TRNA MODIFICATION, DIPHTHAMIDE MODIFICATION
3dmr:A (GLY6) to (SER51) STRUCTURE OF DMSO REDUCTASE FROM RHODOBACTER CAPSULATUS AT PH 7.0 | OXIDOREDUCTASE, DMSO, MOLYBDOPTERIN, PH 7
3du8:A (ILE62) to (LEU104) CRYSTAL STRUCTURE OF GSK-3 BETA IN COMPLEX WITH NMS-869553A | PROTEIN KINASE, ALTERNATIVE SPLICING, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
3du8:B (ASP58) to (LEU104) CRYSTAL STRUCTURE OF GSK-3 BETA IN COMPLEX WITH NMS-869553A | PROTEIN KINASE, ALTERNATIVE SPLICING, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
5hbh:A (VAL27) to (GLU72) CDK8-CYCC IN COMPLEX WITH 5-{5-CHLORO-4-[1-(2-METHOXY-ETHYL)-1,8- DIAZA-SPIRO[4.5]DEC-8-YL]-PYRIDIN-3-YL}-1-METHYL-1,3-DIHYDRO- BENZO[C]ISOTHIAZOLE 2,2-DIOXIDE | CDK8 KINASE / CYCLIN C, TRANSFERASE
4u45:B (ILE24) to (LEU73) MAP4K4 IN COMPLEX WITH INHIBITOR (COMPOUND 25) | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3dxk:F (PRO50) to (ALA98) STRUCTURE OF BOS TAURUS ARP2/3 COMPLEX WITH BOUND INHIBITOR CK0944636 | BETA-PROPELLER, ACETYLATION, ACTIN-BINDING, ATP-BINDING, CELL PROJECTION, CYTOPLASM, CYTOSKELETON, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, WD REPEAT, STRUCTURAL PROTEIN
3dxm:F (PRO50) to (ALA98) STRUCTURE OF BOS TAURUS ARP2/3 COMPLEX WITH BOUND INHIBITOR CK0993548 | BETA-PROPELLER, STRUCTURAL PROTEIN
3p02:A (LYS115) to (ASN160) CRYSTAL STRUCTURE OF A PROTEIN OF UNKNOWN FUNCTION (BACOVA_00267) FROM BACTEROIDES OVATUS AT 1.55 A RESOLUTION | STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, UNKNOWN FUNCTION
4dit:A (ASP58) to (LEU104) CRYSTAL STRUCTURE OF GSK3BETA IN COMPLEX WITH A IMIDAZOPYRIDINE INHIBITOR | KINASE, Y216 PHOSPHORYLATION, PHOSPHOTRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4djj:A (GLY37) to (PHE83) CRYSTAL STRUCTURE OF THE COMPLEX OF PEPTIDYL-TRNA HYDROLASE FROM PSEUDOMONAS AERUGINOSA WITH PIMELIC ACID AT 2.9 ANGSTROM RESOLUTION | ESTERASE, HYDROLASE
5hln:A (ASP58) to (LEU104) X-RAY CRYSTAL STRUCTURE OF GSK3B IN COMPLEX WITH CHIR99021 | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hln:B (ASP58) to (LEU104) X-RAY CRYSTAL STRUCTURE OF GSK3B IN COMPLEX WITH CHIR99021 | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4dmr:A (GLY6) to (SER48) REDUCED DMSO REDUCTASE FROM RHODOBACTER CAPSULATUS WITH BOUND DMSO SUBSTRATE | OXIDOREDUCTASE, DMSO, MOLYBDOPTERIN, SUBSTRATE BOUND
4dnv:A (MET228) to (SER276) CRYSTAL STRUCTURE OF THE W285F MUTANT OF UVB-RESISTANCE PROTEIN UVR8 | WD40 REPEATS, UV-B PERCEPTION, COP1, GENE REGULATION
5htb:A (ILE490) to (GLU548) CRYSTAL STRUCTURE OF HASPIN (GSG2) IN COMPLEX WITH BISUBSTRATE INHIBITOR ARC-3353 | TRANSFERASE, KINASE, INHIBITOR, ALLOSTERIC, STRUCTURAL GENOMICS CONSORTIUM (SGC), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, BISUBSTRATE INHIBITOR
4dta:B (GLY29) to (ILE67) CRYSTAL STRUCTURE OF F95M AMINOGLYCOSIDE-2''-PHOSPHOTRANSFERASE TYPE IVA IN COMPLEX WITH ADENOSINE | AMINOGLYCOSIDE KINASE, TRANSFERASE
4dtk:A (LEU44) to (VAL96) NOVEL AND SELECTIVE PAN-PIM KINASE INHIBITOR | PIM1, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4dtk:A (ASP108) to (GLY137) NOVEL AND SELECTIVE PAN-PIM KINASE INHIBITOR | PIM1, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5i5k:B (VAL934) to (SER993) STRUCTURE OF COMPLEMENT C5 IN COMPLEX WITH ECULIZUMAB | COMPLEMENT, FAB, IMMUNE SYSTEM
5i5k:A (VAL934) to (GLU995) STRUCTURE OF COMPLEMENT C5 IN COMPLEX WITH ECULIZUMAB | COMPLEMENT, FAB, IMMUNE SYSTEM
4uni:C (ASP570) to (SER616) BETA-(1,6)-GALACTOSIDASE FROM BIFIDOBACTERIUM ANIMALIS SUBSP. LACTIS BL-04 IN COMPLEX WITH GALACTOSE | HYDROLASE, GH42
4unt:D (ASN54) to (ASP87) INDUCED MONOMER OF THE MCG VARIABLE DOMAIN | IMMUNE SYSTEM, BENCE-JONES, LIGHT CHAINS, IMMUNOGLOBULIN, AMYLOID
4unt:G (ASN54) to (ASP87) INDUCED MONOMER OF THE MCG VARIABLE DOMAIN | IMMUNE SYSTEM, BENCE-JONES, LIGHT CHAINS, IMMUNOGLOBULIN, AMYLOID
4e0b:D (GLU246) to (VAL309) 2.17 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF MALATE DEHYDROGENASE FROM VIBRIO VULNIFICUS CMCP6 | MALATE DEHYDROGENASE, OXIDOREDUCTASE, TYPE III SECRETION SYSTEM, VIRULENCE, PATHOGENESIS, TOXIN, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID
4e3c:B (GLU16) to (ARG67) X-RAY CRYSTAL STRUCTURE OF HUMAN IKK2 IN AN ACTIVE CONFORMATION | KANASE, AUTO-PHOSPHORYLATION, NEMO BINDING, TRANSFERASE
4e3i:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A DESIGNED 3- CARBOXYL BENZYL SULFONAMIDE BORONIC ACID INHIBITOR | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4e3i:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A DESIGNED 3- CARBOXYL BENZYL SULFONAMIDE BORONIC ACID INHIBITOR | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4e3j:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A DESIGNED 4- TETRAZOLYL BENZENE SULFONAMIDE BORONIC ACID INHIBITOR | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4e3k:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A DESIGNED 4- TETRAZOLYL PYRIDINE SULFONAMIDE BORONIC ACID INHIBITOR | AMPC BETA-LACTAMASE, CLASS C, CEPHALOSPORINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4e3k:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A DESIGNED 4- TETRAZOLYL PYRIDINE SULFONAMIDE BORONIC ACID INHIBITOR | AMPC BETA-LACTAMASE, CLASS C, CEPHALOSPORINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4e3l:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A 3-CHLORO-4- TETRAZOLYL BENZENE SULFONAMIDE BORONIC ACID INHIBITOR | AMPC BETA-LACTAMASE, CLASS C, CEPHALOSPORINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4e3m:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A 2-CHLORO-4- TETRAZOLYL BENZENE SULFONAMIDE BORONIC ACID INHIBITOR | AMPC BETA-LACTAMASE, CLASS C, CEPHALOSPORINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4e3m:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A 2-CHLORO-4- TETRAZOLYL BENZENE SULFONAMIDE BORONIC ACID INHIBITOR | AMPC BETA-LACTAMASE, CLASS C, CEPHALOSPORINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4e3n:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A 2- TRIFLUOROMETHYL-4-TETRAZOLYL BENZENE SULFONAMIDE BORONIC ACID INHIBITOR | AMPC BETA-LACTAMASE, CLASS C, CEPHALOSPORINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4e3n:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A 2- TRIFLUOROMETHYL-4-TETRAZOLYL BENZENE SULFONAMIDE BORONIC ACID INHIBITOR | AMPC BETA-LACTAMASE, CLASS C, CEPHALOSPORINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4e3o:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A SMALL CHLOROMETHYL SULFONAMIDE BORONIC ACID INHIBITOR | AMPC BETA-LACTAMASE, CLASS C, CEPHALOSPORINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4e3o:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH A SMALL CHLOROMETHYL SULFONAMIDE BORONIC ACID INHIBITOR | AMPC BETA-LACTAMASE, CLASS C, CEPHALOSPORINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4uq8:Q (UNK32) to (UNK98) ELECTRON CRYO-MICROSCOPY OF BOVINE COMPLEX I | NADH DEHYDROGENASE, RESPIRATORY COMPLEX, OXIDOREDUCTASE
3pre:A (CYS801) to (THR857) QUINAZOLINES WITH INTRA-MOLECULAR HYDROGEN BONDING SCAFFOLD (IMHBS) AS PI3K/MTOR DUAL INHIBITORS. | PHOSPHOINOSITIDE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3prz:A (GLY868) to (SER894) QUINAZOLINES WITH INTRA-MOLECULAR HYDROGEN BONDING SCAFFOLD (IMHBS) AS PI3K/MTOR DUAL INHIBITORS. | PHOSPHOINOSITIDE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4eb1:I (PHE266) to (GLU306) HYPERSTABLE IN-FRAME INSERTION VARIANT OF ANTITHROMBIN | SERPIN, HYDROLASE INHIBITOR, BLOOD CLOTTING
3pvm:A (SER940) to (LEU992) STRUCTURE OF COMPLEMENT C5 IN COMPLEX WITH CVF | IMMUNE SYSTEM, COMPLEMENT
3pvm:C (SER940) to (LEU992) STRUCTURE OF COMPLEMENT C5 IN COMPLEX WITH CVF | IMMUNE SYSTEM, COMPLEMENT
5ime:B (ILE276) to (ASN322) CRYSTAL STRUCTURE OF P21-ACTIVATED KINASE 1 (PAK1) IN COMPLEX WITH COMPOUND 9 | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4eny:A (GLN37) to (VAL96) CRYSTAL STRUCTURE OF PIM-1 KINASE IN COMPLEX WITH (2E,5Z)-2-(2- CHLOROPHENYLIMINO)-5-(4-HYDROXY-3-METHOXYBENZYLIDENE)THIAZOLIDIN-4- ONE | PIM-1 KINASE, TRANSFERASE-INHIBITOR COMPLEX
4eny:A (ASP108) to (GLY137) CRYSTAL STRUCTURE OF PIM-1 KINASE IN COMPLEX WITH (2E,5Z)-2-(2- CHLOROPHENYLIMINO)-5-(4-HYDROXY-3-METHOXYBENZYLIDENE)THIAZOLIDIN-4- ONE | PIM-1 KINASE, TRANSFERASE-INHIBITOR COMPLEX
4eqv:G (SER85) to (ALA143) STRUCTURE OF SACCHAROMYCES CEREVISIAE INVERTASE | GLYCOSIDASE GH32, BETA-PROPELLER, HYDROLASE, CARBOHYDRATE/SUGAR BINDING
4erm:A (ARG434) to (TYR495) CRYSTAL STRUCTURE OF THE DATP INHIBITED E. COLI CLASS IA RIBONUCLEOTIDE REDUCTASE COMPLEX AT 4 ANGSTROMS RESOLUTION | PROTEIN-PROTEIN COMPLEX, ALPHA/BETA BARREL, ATP CONE, DI-IRON CENTER, OXIDOREDUCTASE, RNR ALPHA, RNR BETA, THIOREDOXIN, RIBONUCLEOTIDE REDUCTION, CYTOSOL
4erm:B (ARG434) to (TYR495) CRYSTAL STRUCTURE OF THE DATP INHIBITED E. COLI CLASS IA RIBONUCLEOTIDE REDUCTASE COMPLEX AT 4 ANGSTROMS RESOLUTION | PROTEIN-PROTEIN COMPLEX, ALPHA/BETA BARREL, ATP CONE, DI-IRON CENTER, OXIDOREDUCTASE, RNR ALPHA, RNR BETA, THIOREDOXIN, RIBONUCLEOTIDE REDUCTION, CYTOSOL
4erm:C (ARG434) to (GLN496) CRYSTAL STRUCTURE OF THE DATP INHIBITED E. COLI CLASS IA RIBONUCLEOTIDE REDUCTASE COMPLEX AT 4 ANGSTROMS RESOLUTION | PROTEIN-PROTEIN COMPLEX, ALPHA/BETA BARREL, ATP CONE, DI-IRON CENTER, OXIDOREDUCTASE, RNR ALPHA, RNR BETA, THIOREDOXIN, RIBONUCLEOTIDE REDUCTION, CYTOSOL
4erm:D (ARG434) to (GLN496) CRYSTAL STRUCTURE OF THE DATP INHIBITED E. COLI CLASS IA RIBONUCLEOTIDE REDUCTASE COMPLEX AT 4 ANGSTROMS RESOLUTION | PROTEIN-PROTEIN COMPLEX, ALPHA/BETA BARREL, ATP CONE, DI-IRON CENTER, OXIDOREDUCTASE, RNR ALPHA, RNR BETA, THIOREDOXIN, RIBONUCLEOTIDE REDUCTION, CYTOSOL
3qde:A (ASN232) to (ASN292) THE STRUCTURE OF CELLOBIOSE PHOSPHORYLASE FROM CLOSTRIDIUM THERMOCELLUM IN COMPLEX WITH PHOSPHATE | CELLULASE, CELLOBIOSE, PHOSPHATE, PHOSPHORYLASE, TRANSFERASE
3qde:B (ASN232) to (GLN290) THE STRUCTURE OF CELLOBIOSE PHOSPHORYLASE FROM CLOSTRIDIUM THERMOCELLUM IN COMPLEX WITH PHOSPHATE | CELLULASE, CELLOBIOSE, PHOSPHATE, PHOSPHORYLASE, TRANSFERASE
3qf9:A (ASP108) to (GLU135) CRYSTAL STRUCTURE OF HUMAN PROTO-ONCOGENE SERINE THREONINE KINASE (PIM1) IN COMPLEX WITH A CONSENSUS PEPTIDE AND A FURAN- THIAZOLIDINEDIONE LIGAND | TRANSFERASE/PEPTIDE, COMPLEX TRANSFERASE-PEPTIDE, PIM1,KINASE, CANCER, LEUKEMIA, ATP-BINDING, NUCLEAR PROTEIN, NUCLEOTIDE-BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3qg0:B (ASP237) to (ALA299) CRYSTAL STRUCTURE OF CELLVIBRIO GILVUS CELLOBIOSE PHOSPHORYLASE COMPLEXED WITH PHOSPHATE AND 1-DEOXYNOJIRIMYCIN | ALPHA(6)/ALPHA(6) BARREL, PHOSPHORYLASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4f6u:A (VAL27) to (LEU73) CRYSTAL STRUCTURE OF HUMAN CDK8/CYCC IN COMPLEX WITH COMPOUND 5 (1-[3- TERT-BUTYL-1-(4-METHYLPHENYL)-1H-PYRAZOL-5-YL]-3-[3-(MORPHOLIN-4-YL) PROPYL]UREA) | PROTEIN KINASE COMPLEX, PROTEROS, TRANSFERASE-TRANSCRIPTION-INHIBITOR COMPLEX
4f70:A (VAL27) to (LEU73) CRYSTAL STRUCTURE OF HUMAN CDK8/CYCC IN COMPLEX WITH COMPOUND 4 (1-[3- TERT-BUTYL-1-(4-METHYLPHENYL)-1H-PYRAZOL-5-YL]-3-[2-(MORPHOLIN-4-YL) ETHYL]UREA) | PROTEIN KINASE COMPLEX, PROTEROS, TRANSFERASE-TRANSCRIPTION-INHIBITOR COMPLEX
4f7n:A (VAL27) to (LEU73) CRYSTAL STRUCTURE OF HUMAN CDK8/CYCC IN COMPLEX WITH COMPOUND 11 (1- [3-TERT-BUTYL-1-(4-METHYLPHENYL)-1H-PYRAZOL-5-YL]-3-(5- HYDROXYPENTYL)UREA) | PROTEIN KINASE COMPLEX, PROTEROS, TRANSFERASE-TRANSCRIPTION-INHIBITOR COMPLEX
4f8c:A (LYS160) to (GLN212) STRUCTURE OF THE CIF:NEDD8 COMPLEX - YERSINIA PSEUDOTUBERCULOSIS CYCLE INHIBITING FACTOR IN COMPLEX WITH HUMAN NEDD8 | EFFECTOR-HOST TARGET COMPLEX, GLUTAMINE DEAMIDASE, DEAMIDATION, BACTERIAL EFFECTOR, CELL CYCLE-PROTEIN BINDING COMPLEX
4f8c:C (LYS160) to (LYS213) STRUCTURE OF THE CIF:NEDD8 COMPLEX - YERSINIA PSEUDOTUBERCULOSIS CYCLE INHIBITING FACTOR IN COMPLEX WITH HUMAN NEDD8 | EFFECTOR-HOST TARGET COMPLEX, GLUTAMINE DEAMIDASE, DEAMIDATION, BACTERIAL EFFECTOR, CELL CYCLE-PROTEIN BINDING COMPLEX
4ux2:A (VAL486) to (CYS527) CRYO-EM STRUCTURE OF ANTAGONIST-BOUND E2P GASTRIC H,K-ATPASE (SCH.E2.MGF) | TRANSPORT PROTEIN, HYDROLASE, POTASSIUM-TRANSPORTING ATPASE
4ux3:A (ARG5) to (LEU49) COHESIN SMC3-HD:SCC1-N COMPLEX FROM YEAST | PROTEIN BINDING, COHESIN, MITOSIS, CHROMOSOME SEGREGATION, KLEISIN, SMC
4f9v:B (GLN76) to (SER132) STRUCTURE OF C113A/C136A MUTANT VARIANT OF GLYCOSYLATED GLUTAMINYL CYCLASE FROM DROSOPHILA MELANOGASTER | ALPHA/BETA HYDROLASE, PGLU FORMATION, PE, ALZHEIMER'S DISEASE, PYROGLUTAMATE, PGLU-AMYLOID, GLYCOSYLATION, TRANSFERASE, HYDROLASE
4v0g:B (ILE825) to (LEU878) JAK3 IN COMPLEX WITH A COVALENT EGFR INHIBITOR | TRANSFERASE, EGFR MUTANT, T790M
4v0i:A (CYS749) to (GLN803) WATER NETWORK DETERMINES SELECTIVITY FOR A SERIES OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS OVER PI3K-DELTA | TRANSFERASE, PI3K, KINASE SELECTIVITY
4v0i:A (TYR813) to (LEU839) WATER NETWORK DETERMINES SELECTIVITY FOR A SERIES OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS OVER PI3K-DELTA | TRANSFERASE, PI3K, KINASE SELECTIVITY
4v0i:B (CYS749) to (GLN803) WATER NETWORK DETERMINES SELECTIVITY FOR A SERIES OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS OVER PI3K-DELTA | TRANSFERASE, PI3K, KINASE SELECTIVITY
4v0i:B (TYR813) to (LEU839) WATER NETWORK DETERMINES SELECTIVITY FOR A SERIES OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS OVER PI3K-DELTA | TRANSFERASE, PI3K, KINASE SELECTIVITY
4feu:F (ARG27) to (TRP74) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR ANTHRAPYRAZOLONE SP600125 | ANTHRAPYRAZOLONE, SP600125, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fex:B (ARG27) to (TRP74) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR TYRPHOSTIN AG1478 | TYRPHOSTIN, 4-ANILINOQUINAZOLINE, TYRPHOSTIN AG1478, AG1478, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fex:C (ARG27) to (TRP74) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR TYRPHOSTIN AG1478 | TYRPHOSTIN, 4-ANILINOQUINAZOLINE, TYRPHOSTIN AG1478, AG1478, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3que:A (ASN26) to (MET78) HUMAN P38 MAP KINASE IN COMPLEX WITH SKEPINONE-L | KINASE DOMAIN, PHOSPHATE TRANSFERASE, DIBENZOSUBERONE DERIVATIVE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fic:A (VAL271) to (ALA311) KINASE DOMAIN OF CSRC IN COMPLEX WITH A HINGE REGION-BINDING FRAGMENT | HINGE BINDING FRAGMENT, TYPE I, DFG-IN, TYROSINE-PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4w6r:A (VAL93) to (GLY134) CRYSTAL STRUCTURE OF FULL-LENGTH SPLIT GFP MUTANT D102C DISULFIDE DIMER, P 1 SPACE GROUP | FLUORESCENT PROTEIN, DIMER, DISULFIDE
3r00:A (LEU44) to (VAL96) THE DISCOVERY OF NOVEL BENZOFURAN-2-CARBOXYLIC ACIDS AS POTENT PIM-1 INHIBITORS | KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r00:A (ASP108) to (GLU135) THE DISCOVERY OF NOVEL BENZOFURAN-2-CARBOXYLIC ACIDS AS POTENT PIM-1 INHIBITORS | KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r02:A (LEU44) to (VAL96) THE DISCOVERY OF NOVEL BENZOFURAN-2-CARBOXYLIC ACIDS AS POTENT PIM-1 INHIBITORS | KINASE, PIM1, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r02:A (ASP108) to (GLU135) THE DISCOVERY OF NOVEL BENZOFURAN-2-CARBOXYLIC ACIDS AS POTENT PIM-1 INHIBITORS | KINASE, PIM1, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r1m:A (ARG203) to (ALA256) STRUCURE OF BIFUNCTIONAL FRUCTOSE 1,6-BISPHOSPHATE ALDOLASE/PHOSPHATASE (ALDOLASE FORM) | SULFOLOBUS FRUCTOSE-1,6-BISPHOSPHATASE-LIKE FOLD, HYDROLASE/ALDOLASE, MG BINDING, METAL BINDING PROTEIN
4fn0:A (GLY85) to (ASN128) CRYSTAL STRUCTURE OF MOUSE NECTIN-2 EXTRACELLULAR FRAGMENT D1-D2, 2ND CRYSTAL FORM | IMMUNOGLOBULIN-LIKE DOMAIN, IG DOMAIN, VIRAL ENTRY RECEPTOR, CELL ADHESION
3r9r:A (ALA12) to (LEU63) STRUCTURE OF A PHOSPHORIBOSYLAMINOIMIDAZOLE-SUCCINOCARBOXAMIDE SYNTHASE FROM MYCOBACTERIUM ABSCESSUS ATCC 19977 / DSM 44196 | SSGCID, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, PHOSPHORIBOSYLAMINOIMIDAZOLE-SUCCINOCARBOXAMIDE SYNTHASE, LIGASE
4g22:A (ILE388) to (ASP433) STRUCTURE OF A LYS-HCT MUTANT FROM COFFEA CANEPHORA (CRYSTAL FORM 1) | BAHD SUPERFAMILY, HYDROXYCINNAMOYLTRANSFERASE, TRANSFERASE
5k6l:A (ALA527) to (GLY568) STRUCTURE OF A GH3 B-GLUCOSIDASE FROM COW RUMEN METAGENOME | GLYCOSIDE HYDROLASE, METAGENOME, B-GLICOSIDASE, FUNCTIONAL FOOD, PREBIOTICS, MICROBIOTA, HYDROLASE
4gka:B (GLN44) to (LEU106) CRYSTAL STRUCTURE OF PURINE NUCLEOSIDE PHOSPHORYLASE (W16Y, W94Y, W178Y, H257W) MUTANT FROM HUMAN COMPLEXED WITH PHOSPHATE | PURINE NUCLEOSIDE PHOSPHORYLASE, NUCLEOSIDE BINDING, PURINE BASE BINDING, PURINE-NUCLEOSIDE PHOSPHORYLASE ACTIVITY, DRUG BINDING, TRANSFERASE ACTIVITY, TRANSFERRING GLYCOSYL GROUPS, PHOSPHATE ION BINDING, INTRACELLULAR, CYTOSOL, TRANSFERASE
4gkh:K (ALA29) to (TRP74) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR 1-NA-PP1 | PYRAZOLOPYRIMIDINE, 1-NA-PP1, BUMPED KINASE INHIBITOR, BKI, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR
4gki:A (ARG27) to (TRP74) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR 1-NM-PP1 | PYRAZOLOPYRIMIDINE, 1-NM-PP1, BUMPED KINASE INHIBITOR, BKI, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR
4gki:K (ARG27) to (TRP74) CRYSTAL STRUCTURE OF THE AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(3')-IA, WITH SUBSTRATE KANAMYCIN AND SMALL MOLECULE INHIBITOR 1-NM-PP1 | PYRAZOLOPYRIMIDINE, 1-NM-PP1, BUMPED KINASE INHIBITOR, BKI, PROTEIN KINASE INHIBITOR, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, ALPHA/BETA PROTEIN, TRANSFERASE, PHOSPHOTRANSFERASE, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, AMINOGLYCOSIDES, KANAMYCIN, GTP, INTRACELLULAR
5kjs:A (ILE387) to (LEU430) CRYSTAL STRUCTURE OF ARABIDOPSIS THALIANA HCT | PHENYLPROPANOID METABOLISM, BAHD, ACYLTRANSFERASE, TRANSFERASE
5kjt:A (ILE387) to (LEU430) CRYSTAL STRUCTURE OF ARABIDOPSIS THALIANA HCT IN COMPLEX WITH P- COUMAROYL-COA | PHENYLPROPANOID METABOLISM, HCT, BAHD, ACYLTRANSFERASE, TRANSFERASE
5kjv:A (ILE381) to (GLN426) CRYSTAL STRUCTURE OF COLEUS BLUMEI HCT | PHENYLPROPANOID METABOLISM, BAHD, HCT, ACYLTRANSFERASE, TRANSFERASE
5kjv:B (ILE381) to (GLN426) CRYSTAL STRUCTURE OF COLEUS BLUMEI HCT | PHENYLPROPANOID METABOLISM, BAHD, HCT, ACYLTRANSFERASE, TRANSFERASE
5l46:A (LEU657) to (GLY702) CRYSTAL STRUCTURE OF HUMAN DIMETHYLGLYCINE-DEHYDROGENASE | ELECTRON TRANSFER, COVALENT FLAVINYLATION, OXIDOREDUCTASE, ONE-CARBON METABOLISM
5li9:A (ILE260) to (SER310) STRUCTURE OF A NUCLEOTIDE-BOUND FORM OF PKCIOTA CORE KINASE DOMAIN | APKC, POLARITY, COMPLEX, TRANSFERASE
5lov:C (GLY43) to (GLY81) DZ-2384 TUBULIN COMPLEX | CELL CYCLE, TUBULIN FOLD, CYTOSKELETON, MICROTUBULE
5luf:Q (UNK32) to (UNK98) CRYO-EM OF BOVINE RESPIRASOME | MITOCHONDRIA, SUPERCOMPLEX, RESPIRATORY CHAIN, OXIDOREDUCTASE
5t68:A (LEU377) to (LEU427) CRYSTAL STRUCTURE OF SYK CATALYTIC DOMAIN IN COMPLEX WITH A FURO[3,2- D]PYRIMIDINE | SPLEEN TYROSINE KINASE SYK CATALYTIC DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5tbo:A (CYS209) to (LEU240) CRYSTAL STRUCTURE OF PLASMODIUM FALCIPARUM DIHYDROOROTATE DEHYDROGENASE BOUND WITH INHIBITOR DSM421 | OXIDOREDUCTASE, ALPHA/BETA BARREL, FMN, MITOCHONDRIAL MEMBRANE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
5tqy:A (PRO14) to (LYS67) CRYOEM RECONSTRUCTION OF HUMAN IKK1, CLOSED CONFORMATION 3 | KINASE, CONSERVED HELIX-LOOP-HELIX, TRANSCRIPTION, ONCOGENE, TRANSFERASE
5tqy:B (PRO14) to (LYS67) CRYOEM RECONSTRUCTION OF HUMAN IKK1, CLOSED CONFORMATION 3 | KINASE, CONSERVED HELIX-LOOP-HELIX, TRANSCRIPTION, ONCOGENE, TRANSFERASE
5tr6:A (LEU377) to (LEU427) DISCOVERY OF TAK-659, AN ORALLY AVAILABLE INVESTIGATIONAL INHIBITOR OF SPLEEN TYROSINE KINASE (SYK) | INHIBITOR, KINASE, LEUKEMIA, LYMPHOMA, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
7api:A (PHE227) to (GLU266) THE S VARIANT OF HUMAN ALPHA1-ANTITRYPSIN, STRUCTURE AND IMPLICATIONS FOR FUNCTION AND METABOLISM | PROTEINASE INHIBITOR
8api:A (PHE227) to (GLU266) THE S VARIANT OF HUMAN ALPHA1-ANTITRYPSIN, STRUCTURE AND IMPLICATIONS FOR FUNCTION AND METABOLISM | PROTEINASE INHIBITOR
3rse:F (PRO50) to (ALA98) STRUCTURAL AND BIOCHEMICAL CHARACTERIZATION OF TWO BINDING SITES FOR NUCLEATION PROMOTING FACTOR WASP-VCA ON ARP2/3 COMPLEX | HETEROHEPTAMER, HEPTAMERIC HETEROCOMPLEX, F-ACTIN BRANCH INITIATION, ACTIN, CYTOSOL, STRUCTURAL PROTEIN
4wnm:A (LEU377) to (LEU427) SYK CATALYTIC DOMAIN IN COMPLEX WITH A POTENT TRIAZOLOPYRIDINE INHIBITOR | SYK CATALYTIC DOMAIN IN COMPLEX WITH A POTENT TRIAZOLOPYRIDINE BASED INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4wt6:A (GLN37) to (VAL96) CRYSTAL STRUCTURE OF HUMAN PIM-1 KINASE IN COMPLEX WITH A THIADIAZOLAMINE-INDOLE INHIBITOR. | TRANSFERASE, SERINE/THREONINE PROTEIN KINASE
3er8:C (MET333) to (ASN374) CRYSTAL STRUCTURE OF THE HETERODIMERIC VACCINIA VIRUS MRNA POLYADENYLATE POLYMERASE COMPLEX WITH TWO FRAGMENTS OF RNA | POLYADENYLATE POLYMERASE, TRANSLOCATION, SINGLE TRANDED RNA POLY(A) POLYMERASE, RNA PROTEIN COMPLEX, PROCESSIVITY, HETERODIMER, NUCLEOTIDYLTRANSFERASE, POXVIRUS; METHYLTRANSFERASE, MRNA CAPPING, MRNA PROCESSING, S-ADENOSYL-L-METHIONINE, TRANSCRIPTION, TRANSFERASE, TRANSFERASE/DNA, RNA COMPLEX, TRANSFERASE-DNA
3er8:D (MET333) to (ASN374) CRYSTAL STRUCTURE OF THE HETERODIMERIC VACCINIA VIRUS MRNA POLYADENYLATE POLYMERASE COMPLEX WITH TWO FRAGMENTS OF RNA | POLYADENYLATE POLYMERASE, TRANSLOCATION, SINGLE TRANDED RNA POLY(A) POLYMERASE, RNA PROTEIN COMPLEX, PROCESSIVITY, HETERODIMER, NUCLEOTIDYLTRANSFERASE, POXVIRUS; METHYLTRANSFERASE, MRNA CAPPING, MRNA PROCESSING, S-ADENOSYL-L-METHIONINE, TRANSCRIPTION, TRANSFERASE, TRANSFERASE/DNA, RNA COMPLEX, TRANSFERASE-DNA
2beh:L (PHE258) to (LEU299) CRYSTAL STRUCTURE OF ANTITHROMBIN VARIANT S137A/V317C/T401C WITH PLASMA LATENT ANTITHROMBIN | ANTITHROMBIN DIMER, BLOOD CLOTTING
2p9p:F (PRO50) to (ALA98) CRYSTAL STRUCTURE OF BOVINE ARP2/3 COMPLEX CO-CRYSTALLIZED WITH ADP | ACTIN, WD REPEAT,COMPLEX, STRUCTURAL PROTEIN
2bkk:A (ARG18) to (LEU67) CRYSTAL STRUCTURE OF AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH (3')-IIIA IN COMPLEX WITH THE INHIBITOR AR_3A | TRANSFERASE/PEPTIDE, TRANSFERASE/DESIGNED PROTEIN COMPLEX, ANKYRIN REPEAT, CO-CRYSTALLIZATION, INHIBITOR DESIGN, DRUG DESIGN, ENZYME INHIBITION, KINASE INHIBITION, DESIGNED REPEAT PROTEIN, ANTIBIOTIC RESISTANCE, ATP-BINDING, KINASE, PLASMID, TRANSFERASE
4x3v:A (LYS424) to (ILE483) CRYSTAL STRUCTURE OF HUMAN RIBONUCLEOTIDE REDUCTASE 1 BOUND TO INHIBITOR | COMPLEX, REDUCATSE, INHIBITOR, ENZYME, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
3f2n:A (ILE490) to (LEU545) CRYSTAL STRUCTURE OF HUMAN HASPIN WITH AN IMIDAZO-PYRIDAZINE LIGAND | HASPIN, GERM CELL ASSOCIATED 2, HAPLOID GERM CELL SPECIFIC NUCLEAR PROTEIN KINASE, ATP-BINDING, CELL CYCLE, CHROMATIN REGULATOR, KINASE, MAGNESIUM, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
2bro:A (GLY16) to (LEU62) STRUCTURE-BASED DESIGN OF NOVEL CHK1 INHIBITORS: INSIGHTS INTO HYDROGEN BONDING AND PROTEIN-LIGAND AFFINITY | DRUG DESIGN, FURANOPYRIMIDINE, MOLECULAR RECOGNITION, ONCOLOGY, PYRROLOPYRIMIDINE, ATP-BINDING, CELL CYCLE, DNA DAMAGE, KINASE, NUCLEAR PROTEIN, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2bwx:A (LEU352) to (VAL423) HIS354ALA ESCHERICHIA COLI AMINOPEPTIDASE P | AMINOPEPTIDASE P, METALLOENZYME, 'PITA-BREAD' ENZYME, PROLINE-SPECIFIC ENZYME, MANGANESE ENZYME, HYDROLASE
2pu2:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE WITH BOUND PHTHALAMIDE INHIBITOR | AMPC BETA-LACAMASE PHTHALAMIDE, HYDROLASE
2pu2:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE WITH BOUND PHTHALAMIDE INHIBITOR | AMPC BETA-LACAMASE PHTHALAMIDE, HYDROLASE
2pvr:A (GLY46) to (LEU88) CRYSTAL STRUCTURE OF THE CATALYTIC SUBUNIT OF PROTEIN KINASE CK2 (C- TERMINAL DELETION MUTANT 1-335) IN COMPLEX WITH TWO SULFATE IONS | EUKARYOTIC PROTEIN KINASE FOLD, CMGC KINASES, SIGNALING PROTEIN, TRANSFERASE
2c61:A (ASP125) to (ARG165) CRYSTAL STRUCTURE OF THE NON-CATALYTIC B SUBUNIT OF A-TYPE ATPASE FROM M. MAZEI GO1 | HYDROLASE, A-TYPE ATP SYNTHASE, H+ ATPASE, A1AO, NON-CATALYTIC, ATP SYNTHESIS, HYDROGEN ION TRANSPORT, ION TRANSPORT, TRANSPORT
3spl:B (ILE52) to (VAL84) CRYSTAL STRUCTURE OF APRATAXIN ORTHOLOG HNT3 IN COMPLEX WITH DNA AND AMP | HIT DOMAIN, ZINC FINGER, DNA DEADENYLASE, DNA BINDING, AMP BINDING, HYDROLASE-DNA COMPLEX
3spl:C (ILE52) to (VAL84) CRYSTAL STRUCTURE OF APRATAXIN ORTHOLOG HNT3 IN COMPLEX WITH DNA AND AMP | HIT DOMAIN, ZINC FINGER, DNA DEADENYLASE, DNA BINDING, AMP BINDING, HYDROLASE-DNA COMPLEX
1oyh:L (PHE258) to (LEU299) CRYSTAL STRUCTURE OF P13 ALANINE VARIANT OF ANTITHROMBIN | THROMBIN; INHIBITION; HEPARIN ANALOGUE; SERINE PROTEASE INHIBITOR, BLOOD CLOTTING
3svs:B (PHE88) to (LYS135) CRYSTAL STRUCTURE OF MKATE MUTANT S158A/S143C AT PH 4.0 | FLUORENSCENT PROTEIN, PH SENSOR, FLUORESCENT PROTEIN
3t1p:A (PHE227) to (GLU266) CRYSTAL STRUCTURE OF AN ALPHA-1-ANTITRYPSIN TRIMER | SERPIN, PROTEASE INHIBITOR, PLASMA, HYDROLASE INHIBITOR
1ds5:A (VAL45) to (LEU88) DIMERIC CRYSTAL STRUCTURE OF THE ALPHA SUBUNIT IN COMPLEX WITH TWO BETA PEPTIDES MIMICKING THE ARCHITECTURE OF THE TETRAMERIC PROTEIN KINASE CK2 HOLOENZYME. | PROTEIN-COMPLEX, TETRAMER, TRANSFERASE
4ivc:B (LEU881) to (LEU932) JAK1 KINASE (JH1 DOMAIN) IN COMPLEX WITH THE INHIBITOR (TRANS-4-{2- [(1R)-1-HYDROXYETHYL]IMIDAZO[4,5-D]PYRROLO[2,3-B]PYRIDIN-1(6H)- YL}CYCLOHEXYL)ACETONITRILE | PROTEIN KINASE, PHOSPHO TRANSFER, PHOSPHO TYROSINE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3t9i:A (ASP108) to (GLY137) PIM1 COMPLEXED WITH A NOVEL 3,6-DISUBSTITUTED INDOLE AT 2.6 ANG RESOLUTION | KINASE, PHOSPHOTRANSFERASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4y3u:A (GLU482) to (CYS525) THE STRUCTURE OF PHOSPHOLAMBAN BOUND TO THE CALCIUM PUMP SERCA1A | CA-ATPASE, SERCA1A, MEMBRANE PROTEIN
2d7p:A (ALA53) to (PHE95) SOLUTION STRUCTURE OF THE 22TH FILAMIN DOMAIN FROM HUMAN FILAMIN C | BETA-SANDWICH, IMMUNOGLOBULIN-LIKE FOLD, FILAMIN DOMAIN, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, STRUCTURAL PROTEIN
3gsg:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT-BASED INHIBITOR | HYDROLASE, ANTIBIOTIC RESISTANCE, PERIPLASM, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
3gv9:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT-BASED INHIBITOR | HYDROLASE, ANTIBIOTIC RESISTANCE, PERIPLASM, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
3gv9:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT-BASED INHIBITOR | HYDROLASE, ANTIBIOTIC RESISTANCE, PERIPLASM, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1eml:A (TYR92) to (GLY134) GREEN FLUORESCENT PROTEIN FROM AEQUOREA VICTORIA, MUTANT | FLUORESCENT PROTEIN, BETA-BARREL, BIOLUMINESCENCE, LUMINESCENCE
4jsp:B (ILE2222) to (LYS2258) STRUCTURE OF MTORDELTAN-MLST8-ATPGAMMAS-MG COMPLEX | KINASE, TRANSFERASE
4jsp:A (ILE2222) to (LYS2258) STRUCTURE OF MTORDELTAN-MLST8-ATPGAMMAS-MG COMPLEX | KINASE, TRANSFERASE
4jsx:B (ILE2222) to (LYS2258) STRUCTURE OF MTORDELTAN-MLST8-TORIN2 COMPLEX | KINASE, TRANSFERASE
4jsx:A (ILE2222) to (LYS2258) STRUCTURE OF MTORDELTAN-MLST8-TORIN2 COMPLEX | KINASE, TRANSFERASE
3ham:B (SER25) to (LEU63) STRUCTURE OF THE GENTAMICIN-APH(2")-IIA COMPLEX | AMINOGLYCOSIDE, GENTAMICIN, ANTIBIOTIC RESISTANCE, TRANSFERASE
2eay:A (ASN95) to (GLU170) CRYSTAL STRUCTURE OF BIOTIN PROTEIN LIGASE FROM AQUIFEX AEOLICUS | BIOTIN BIOSYNTHESIS, DIMER, X-RAY DIFFRACTION, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, LIGASE
4ysa:A (PRO72) to (ILE111) COMPLETELY OXIDIZED STRUCTURE OF COPPER NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS | NITRITE, COPPER, REDUCTASE, OXIDOREDUCTASE
4ysq:A (PRO72) to (ILE111) STRUCTURE OF COPPER NITRITE REDUCTASE FROM GEOBACILLUS THERMODENITRIFICANS - 8.38 MGY | NITRITE, COPPER, REDUCTASE, OXIDOREDUCTASE
3uus:A (ILE430) to (TYR495) CRYSTAL STRUCTURE OF THE DATP INHIBITED E. COLI CLASS IA RIBONUCLEOTIDE REDUCTASE COMPLEX | 10 STRANDED ALPHA/BETA BARREL, DATP BOUND, DI-IRON, OXIDOREDUCTASE
3uus:B (ILE430) to (TYR495) CRYSTAL STRUCTURE OF THE DATP INHIBITED E. COLI CLASS IA RIBONUCLEOTIDE REDUCTASE COMPLEX | 10 STRANDED ALPHA/BETA BARREL, DATP BOUND, DI-IRON, OXIDOREDUCTASE
3uwc:A (ILE160) to (HIS212) STRUCTURE OF AN AMINOTRANSFERASE (DEGT-DNRJ-ERYC1-STRS FAMILY) FROM COXIELLA BURNETII IN COMPLEX WITH PMP | LIPOPOLYSACCHARIDE BIOSYNTHESIS, TRANSFERASE
2ftx:A (GLN146) to (GLY182) CRYSTAL STRUCTURE OF THE YEAST KINETOCHORE SPC24/SPC25 GLOBULAR DOMAIN | ALPHA-BETA, COMPLEX, COILED-COIL, STRUCTURAL PROTEIN, PROTEIN BINDING
4kns:A (PRO59) to (GLU99) REDUCED CRYSTAL STRUCTURE OF THE NITROSOMONAS EUROPAEA COPPER NITRITE REDUCTASE AT PH 6.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
4kns:B (PRO59) to (GLU99) REDUCED CRYSTAL STRUCTURE OF THE NITROSOMONAS EUROPAEA COPPER NITRITE REDUCTASE AT PH 6.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
4kns:C (PRO59) to (GLU99) REDUCED CRYSTAL STRUCTURE OF THE NITROSOMONAS EUROPAEA COPPER NITRITE REDUCTASE AT PH 6.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
4kns:D (PRO59) to (GLU99) REDUCED CRYSTAL STRUCTURE OF THE NITROSOMONAS EUROPAEA COPPER NITRITE REDUCTASE AT PH 6.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
4kns:E (PRO59) to (GLU99) REDUCED CRYSTAL STRUCTURE OF THE NITROSOMONAS EUROPAEA COPPER NITRITE REDUCTASE AT PH 6.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
4kns:F (PRO59) to (GLU99) REDUCED CRYSTAL STRUCTURE OF THE NITROSOMONAS EUROPAEA COPPER NITRITE REDUCTASE AT PH 6.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
4knt:A (PRO59) to (GLU99) COPPER NITRITE REDUCTASE FROM NITROSOMONAS EUROPAEA PH 8.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
4knt:B (PRO59) to (GLU99) COPPER NITRITE REDUCTASE FROM NITROSOMONAS EUROPAEA PH 8.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
4knt:C (PRO59) to (GLU99) COPPER NITRITE REDUCTASE FROM NITROSOMONAS EUROPAEA PH 8.5 | NITRITE REDUCTASE, OXIDOREDUCTASE
1sm2:A (ILE369) to (LYS412) CRYSTAL STRUCTURE OF THE PHOSPHORYLATED INTERLEUKIN-2 TYROSINE KINASE CATALYTIC DOMAIN | PROTEIN KINASE, IMMUNOLOGY, TRANSFERASE
2vx3:B (ILE165) to (HIS213) CRYSTAL STRUCTURE OF THE HUMAN DUAL SPECIFICITY TYROSINE- PHOSPHORYLATION-REGULATED KINASE 1A | SERINE/THREONINE-PROTEIN KINASE, MINIBRAIN HOMOLOG, NUCLEOTIDE-BINDING, TRANSFERASE, PHOSPHOPROTEIN, TYROSINE-PROTEIN KINASE, CASP8, KINASE
4kz3:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 44 (5-CHLORO-3-SULFAMOYLTHIOPHENE-2-CARBOXYLIC ACID) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4kz3:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 44 (5-CHLORO-3-SULFAMOYLTHIOPHENE-2-CARBOXYLIC ACID) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4kz6:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 13 ((2R,6R)-6-METHYL-1-(3-SULFANYLPROPANOYL)PIPERIDINE-2-CARBOXYLIC ACID) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4kz6:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 13 ((2R,6R)-6-METHYL-1-(3-SULFANYLPROPANOYL)PIPERIDINE-2-CARBOXYLIC ACID) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4kzb:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 50 (N-(METHYLSULFONYL)-N-PHENYL-ALANINE) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4kzb:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE IN COMPLEX WITH FRAGMENT 50 (N-(METHYLSULFONYL)-N-PHENYL-ALANINE) | AMPC BETA-LACTAMASE, CLASS C, HYDROLASE, CEPHALOSPORINASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4zle:A (CYS242) to (LYS287) CELLOBIONIC ACID PHOSPHORYLASE - LIGAND FREE STRUCTURE | (ALPHA/ALPHA)6 BARREL, GLYCOSIDE HYDROLASE FAMILY 94, OXIDATIVE CELLULOSE DEGRADATION SYSTEM, INTRACELLULAR ENZYME, TRANSFERASE
4zlg:A (CYS242) to (LYS287) CELLOBIONIC ACID PHOSPHORYLASE - GLUCONIC ACID COMPLEX | (ALPHA/ALPHA)6 BARREL, GLYCOSIDE HYDROLASE FAMILY 94, OXIDATIVE CELLULOSE DEGRADATION SYSTEM, INTRACELLULAR ENZYME, TRANSFERASE
1h5n:A (GLY6) to (SER48) DMSO REDUCTASE MODIFIED BY THE PRESENCE OF DMS AND AIR | OXIDOREDUCTASE, REDUCTASE, DMSO, DMS, MOLYBDOPTERIN
1h8f:A (ASP58) to (LEU104) GLYCOGEN SYNTHASE KINASE 3 BETA. | KINASE, INSULIN PATHWAY
1h8f:B (ASP58) to (LEU104) GLYCOGEN SYNTHASE KINASE 3 BETA. | KINASE, INSULIN PATHWAY
1tk1:A (PHE111) to (ASP182) YEAST OXYGEN-DEPENDENT COPROPORPHYRINOGEN OXIDASE | COPROPORPHYRINOGEN OXIDASE, HEME BIOSYNTHESIS, ENZYME, OXIDOREDUCTASE
2wb8:A (ILE490) to (GLU548) CRYSTAL STRUCTURE OF HASPIN KINASE | HISTONE MODIFICATION, PHOSPHOPROTEIN, ATYPICAL KINASE, SERINE/THREONINE-PROTEIN KINASE, NUCLEOTIDE-BINDING, CHROMATIN REGULATOR, CELL CYCLE, HISTONE H3, ATP-BINDING, TRANSFERASE, GSG2, KINASE, HASPIN, NUCLEUS, MITOSIS
2hds:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH 4-METHANESULFONYLAMINO BENZOIC ACID | AMPC BETA-LACTAMASE FRAGMENT-BASED DRUG DESIGN, HYDROLASE
3w55:A (ILE31) to (ARG77) THE STRUCTURE OF ERK2 IN COMPLEX WITH FR148083 | PROTEIN KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1iem:A (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH A BORONIC ACID INHIBITOR (1, CEFB4) | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE
1iem:B (TYR259) to (ASP288) CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH A BORONIC ACID INHIBITOR (1, CEFB4) | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE
2i72:A (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH 5-DIFORMYLAMINOMETHYL- BENZO[B]THIOPHEN-2-BORONIC ACID | AMPC, BETA-LACTAMASE, CEPHALOSPORINASE, SERINE HYDROLASE
2wy0:C (PHE286) to (ILE327) CRYSTAL STRUCTURE OF MOUSE ANGIOTENSINOGEN IN THE OXIDISED FORM WITH SPACE GROUP P6122 | GLYCOPROTEIN, HYPERTENSION, VASOCONSTRICTOR, RENIN, SERPINS, VASOACTIVE, ANGIOTENSIN, HORMONE
5aed:A (TYR202) to (LEU243) A BACTERIAL PROTEIN STRUCTURE IN GLYCOSIDE HYDROLASE FAMILY 31 | HYDROLASE, GH31, ALPHA-SULFOQUINOVOSIDASE
5aed:B (TYR202) to (LEU243) A BACTERIAL PROTEIN STRUCTURE IN GLYCOSIDE HYDROLASE FAMILY 31 | HYDROLASE, GH31, ALPHA-SULFOQUINOVOSIDASE
5aee:A (TYR202) to (LEU243) A BACTERIAL PROTEIN STRUCTURE IN GLYCOSIDE HYDROLASE FAMILY 31 | HYDROLASE, GH31, ALPHA-SULFOQUINOVOSIDASE
5aee:B (TYR202) to (LEU243) A BACTERIAL PROTEIN STRUCTURE IN GLYCOSIDE HYDROLASE FAMILY 31 | HYDROLASE, GH31, ALPHA-SULFOQUINOVOSIDASE
4mvf:A (ASP75) to (LEU124) CRYSTAL STRUCTURE OF PLASMODIUM FALCIPARUM CDPK2 COMPLEXED WITH INHIBITOR STAUROSPORINE | EF-HANDS, PROTEIN S/T KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, CALCIUM DEPENDENT PROTEIN KINASE, CALCIUM BINDING DOMAIN
2xj2:A (ASP108) to (GLU135) PROTEIN KINASE PIM-1 IN COMPLEX WITH SMALL MOLECULE INHIBITOR | TRANSFERASE, PHOSPHORYLATION, PROTEIN KINASE FOLD
4mxy:B (LEU273) to (LEU308) SRC M314L T338M DOUBLE MUTANT BOUND TO KINASE INHIBITOR BOSUTINIB | KINASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3x1n:A (PRO72) to (ILE111) NITRITE-BOUND THERMOSTABLE COPPER NITRITE REDUCTASE AT 320 K | GREEK KEY BETA BARREL, NITRITE REDUCTASE, CYTOCHROME C551, OXIDOREDUCTASE
4n6y:A (ASP108) to (GLY137) PIM1 COMPLEXED WITH A PHENYLCARBOXAMIDE | KINASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4nbm:A (MET228) to (SER276) CRYSTAL STRUCTURE OF UVB PHOTORECEPTOR UVR8 AND LIGHT-INDUCED STRUCTURAL CHANGES AT 180K | 7-BLADE BETA-PROPELLER, GENE REGULATION
4nbm:B (MET228) to (SER276) CRYSTAL STRUCTURE OF UVB PHOTORECEPTOR UVR8 AND LIGHT-INDUCED STRUCTURAL CHANGES AT 180K | 7-BLADE BETA-PROPELLER, GENE REGULATION
4nbm:D (MET228) to (SER276) CRYSTAL STRUCTURE OF UVB PHOTORECEPTOR UVR8 AND LIGHT-INDUCED STRUCTURAL CHANGES AT 180K | 7-BLADE BETA-PROPELLER, GENE REGULATION
1wbq:B (LEU352) to (VAL423) ZN MG SUBSTITUTED AMINOPEPTIDASE P FROM E. COLI | HYDROLASE, PROLINE-SPECIFIC PEPTIDASE, METALLOENZYME, PITA-BREAD FOLD, DINUCLEAR HYDROLASE, METAL BINDING PROTEIN
1wbq:C (LEU352) to (VAL423) ZN MG SUBSTITUTED AMINOPEPTIDASE P FROM E. COLI | HYDROLASE, PROLINE-SPECIFIC PEPTIDASE, METALLOENZYME, PITA-BREAD FOLD, DINUCLEAR HYDROLASE, METAL BINDING PROTEIN
1wbq:D (LEU352) to (VAL423) ZN MG SUBSTITUTED AMINOPEPTIDASE P FROM E. COLI | HYDROLASE, PROLINE-SPECIFIC PEPTIDASE, METALLOENZYME, PITA-BREAD FOLD, DINUCLEAR HYDROLASE, METAL BINDING PROTEIN
2xzb:A (VAL486) to (CYS527) PIG GASTRIC H,K-ATPASE WITH BOUND BEF AND SCH28080 | HYDROLASE, ION PUMP, H/K-ATPASE, P-TYPE ATPASE, MEMBRANE PROTEIN, BERYLLIUM FLUORIDE, ATP-BINDING, ACID SUPPRESSANT
1ke0:A (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH THE INHIBITOR 4-(CARBOXYVIN-2-YL) PHENYLBORONIC ACID | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, PHENYLBORONIC ACID
1ke0:B (TYR259) to (ASP288) X-RAY CRYSTAL STRUCTURE OF AMPC BETA-LACTAMASE FROM E. COLI IN COMPLEX WITH THE INHIBITOR 4-(CARBOXYVIN-2-YL) PHENYLBORONIC ACID | CEPHALOSPORINASE, BETA-LACTAMASE, SERINE HYDROLASE, PHENYLBORONIC ACID
1woo:A (TYR169) to (ILE217) CRYSTAL STRUCTURE OF T-PROTEIN OF THE GLYCINE CLEAVAGE SYSTEM | GLYCINE CLEAVAGE SYSTEM, TETRAHYDROFOLATE, T-PROTEIN, TRANSFERASE
3jpv:A (LEU44) to (VAL96) CRYSTAL STRUCTURE OF HUMAN PROTO-ONCOGENE SERINE THREONINE KINASE (PIM1) IN COMPLEX WITH A CONSENSUS PEPTIDE AND A PYRROLO[2,3- A]CARBAZOLE LIGAND | ONCOGENE, KINASE, SERINE-THREONINE, PIM1, PYRROLO[2,3-A]CARBAZOLE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ALTERNATIVE INITIATION, ATP- BINDING, CELL MEMBRANE, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSFERASE - TRANSFERASE INHIBITOR COMPLEX
3jpv:A (ASP108) to (GLY137) CRYSTAL STRUCTURE OF HUMAN PROTO-ONCOGENE SERINE THREONINE KINASE (PIM1) IN COMPLEX WITH A CONSENSUS PEPTIDE AND A PYRROLO[2,3- A]CARBAZOLE LIGAND | ONCOGENE, KINASE, SERINE-THREONINE, PIM1, PYRROLO[2,3-A]CARBAZOLE, STRUCTURAL GENOMICS CONSORTIUM, SGC, ALTERNATIVE INITIATION, ATP- BINDING, CELL MEMBRANE, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TRANSFERASE - TRANSFERASE INHIBITOR COMPLEX
4a0a:A (ALA956) to (HIS991) STRUCTURE OF HSDDB1-DRDDB2 BOUND TO A 16 BP CPD-DUPLEX ( PYRIMIDINE AT D-1 POSITION) AT 3.6 A RESOLUTION (CPD 3) | DNA BINDING PROTEIN-DNA COMPLEX, DNA DAMAGE REPAIR
1xgj:B (TYR259) to (ASP288) AMPC BETA-LACTAMASE IN COMPLEX WITH 3-(4-CARBOXY-2-HYDROXY- PHENYLSULFAMOYL)-THIOPHENE-2-CARBOXYLIC ACID | AMPC,BETA-LACTAMASE, CEPHALOSPORINASE, SERINE HYDROLASE
3jy0:A (ASP108) to (GLY137) DISCOVERY OF 3H-BENZO[4,5]THIENO[3,2-D]PYRIMIDIN-4-ONES AS POTENT, HIGHLY SELECTIVE AND ORALLY BIOAVAILABLE PIM KINASES INHIBITORS | PIM-1, ALTERNATIVE INITIATION, ATP-BINDING, CELL MEMBRANE, CYTOPLASM, KINASE, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
1xws:A (LEU44) to (VAL96) CRYSTAL STRUCTURE OF THE HUMAN PIM1 KINASE DOMAIN | PIM1, KINASE, CANCER, LEUKEMIA, TRANSFERASE
5d1y:A (LYS424) to (ILE481) LOW RESOLUTION CRYSTAL STRUCTURE OF HUMAN RIBONUCLEOTIDE REDUCTASE ALPHA6 HEXAMER IN COMPLEX WITH DATP | DEOXYRIBONUCLEOTIDE, OLIGOMERIZATION, ATP CONE, OXIDOREDUCTASE
5d1y:B (LYS424) to (ILE481) LOW RESOLUTION CRYSTAL STRUCTURE OF HUMAN RIBONUCLEOTIDE REDUCTASE ALPHA6 HEXAMER IN COMPLEX WITH DATP | DEOXYRIBONUCLEOTIDE, OLIGOMERIZATION, ATP CONE, OXIDOREDUCTASE
4pab:A (LEU650) to (GLY695) CRYSTAL STRUCTURE OF THE PRECURSOR FORM OF RAT DMGDH COMPLEXED WITH TETRAHYDROFOLATE | DIMETHYLGLYCINE DEHYDROGENASE, RAT, TETRAHYDROFOLATE, OXIDOREDUCTASE
4pab:B (LEU650) to (GLY695) CRYSTAL STRUCTURE OF THE PRECURSOR FORM OF RAT DMGDH COMPLEXED WITH TETRAHYDROFOLATE | DIMETHYLGLYCINE DEHYDROGENASE, RAT, TETRAHYDROFOLATE, OXIDOREDUCTASE
3ad9:A (MET756) to (GLY802) HETEROTETRAMERIC SARCOSINE OXIDASE FROM CORYNEBACTERIUM SP. U-96 SARCOSINE-REDUCED FORM | SARCOSINE OXIDASE, OXIDOREDUCTASE
3ad9:C (ASN149) to (ALA196) HETEROTETRAMERIC SARCOSINE OXIDASE FROM CORYNEBACTERIUM SP. U-96 SARCOSINE-REDUCED FORM | SARCOSINE OXIDASE, OXIDOREDUCTASE
4pj1:S (GLY3) to (VAL41) CRYSTAL STRUCTURE OF THE HUMAN MITOCHONDRIAL CHAPERONIN SYMMETRICAL 'FOOTBALL' COMPLEX | HUMAN, MITOCHONDRIAL, CHAPERONIN, COMPLEX, SYMMETRIC, CHAPERONE
3l4u:A (ALA240) to (ILE281) CRYSTAL COMPLEX OF N-TERMINAL HUMAN MALTASE-GLUCOAMYLASE WITH DE-O-SULFONATED KOTALANOL | GLYCOSIDE HYDROLASE FAMILY 31, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, GLYCOSIDASE, HYDROLASE, MEMBRANE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, SIGNAL-ANCHOR, SULFATION, TRANSMEMBRANE
5djw:A (GLU127) to (THR165) CRYSTAL STRUCTURE OF FAMILY 31 ALPHA-GLUCOSIDASE (BT_3299) FROM BACTEROIDES THETAIOTAOMICRON | FAMILY GLYCOSIDE HYDROLASE 31, ALPHA-GLUCOSIDASE, CARBOHYDRATE BINDING PROTEIN
1yxa:A (THR249) to (LEU289) SERPINA3N, A MURINE ORTHOLOGUE OF HUMAN ANTICHYMOTRYPSIN | SERPIN, ANTICHYMOTRYPSIN, PROTEASE INHIBITOR, REACTIVE CENTRE LOOP, PLASMA, HYDROLASE INHIBITOR
3at2:A (VAL42) to (ARG89) CRYSTAL STRUCTURE OF CK2ALPHA | CK2, KINASE, TRANSFERASE
5e8t:A (GLY212) to (THR251) TGF-BETA RECEPTOR TYPE 1 KINASE DOMAIN (T204D) | ALK5, SB431542, KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, TRANSFERASE
3c13:A (GLY46) to (LEU88) LOW PH-VALUE CRYSTAL STRUCTURE OF EMODIN IN COMPLEX WITH THE CATALYTIC SUBUNIT OF PROTEIN KINASE CK2 | PROTEIN KINASE CK2, CASEIN KINASE 2, EUKARYOTIC PROTEIN KINASES, EMODIN, ATP-COMPETITIVE INHIBITOR, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
3n5i:A (GLY183) to (ARG279) CRYSTAL STRUCTURE OF THE PRECURSOR (S250A MUTANT) OF THE N-TERMINAL BETA-AMINOPEPTIDASE BAPA | NTN HYDROLASE, ALPHA-BETA-BETA-ALPHA SANDWICH, BETA-AMINOPEPTIDASE, BETA-PEPTIDE, HYDROLASE
3n5i:C (GLY183) to (ARG279) CRYSTAL STRUCTURE OF THE PRECURSOR (S250A MUTANT) OF THE N-TERMINAL BETA-AMINOPEPTIDASE BAPA | NTN HYDROLASE, ALPHA-BETA-BETA-ALPHA SANDWICH, BETA-AMINOPEPTIDASE, BETA-PEPTIDE, HYDROLASE
5fjx:A (ASP454) to (MSE496) YEAST DELTA-COP-I MU-HOMOLOGY DOMAIN COMPLEXED WITH GCS1 WXXF PEPTIDE | PROTEIN TRANSPORT, COP-I, VESICLE COAT PROTEIN
4rg0:A (LEU405) to (GLU445) CRYSTAL STRUCTURE OF BTK KINASE DOMAIN COMPLEXED WITH 2-[8-FLUORO-2- [2-(HYDROXYMETHYL)-3-[1-METHYL-5-[[5-(4-METHYLPIPERAZIN-1-YL)-2- PYRIDYL]AMINO]-6-OXO-3-PYRIDYL]PHENYL]-1-OXO-3,4-DIHYDROISOQUINOLIN- 6-YL]-2-METHYL-PROPANENITRILE | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3om8:A (ASN3) to (TRP41) THE CRYSTAL STRUCTURE OF A HYDROLASE FROM PSEUDOMONAS AERUGINOSA PA01 | STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, HYDROLASE
3om8:B (ASN3) to (TRP41) THE CRYSTAL STRUCTURE OF A HYDROLASE FROM PSEUDOMONAS AERUGINOSA PA01 | STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, HYDROLASE
4d9s:A (MET228) to (SER276) CRYSTAL STRUCTURE OF ARABIDOPSIS THALIANA UVR8 (UV RESISTANCE LOCUS 8) | UV RESISTANCE, UV-B PHOTORECEPTOR, TRYPTOPHAN CHROMOPHORES, HOMODIMER, COP1, CHROMATIN-BINDING PROTEIN
3dwl:F (PRO50) to (ALA98) CRYSTAL STRUCTURE OF FISSION YEAST ARP2/3 COMPLEX LACKING THE ARP2 SUBUNIT | PROPELLOR, ACTIN-BINDING, ATP-BINDING, CYTOSKELETON, NUCLEOTIDE- BINDING, WD REPEAT, STRUCTURAL PROTEIN
3dwl:K (PRO50) to (ALA98) CRYSTAL STRUCTURE OF FISSION YEAST ARP2/3 COMPLEX LACKING THE ARP2 SUBUNIT | PROPELLOR, ACTIN-BINDING, ATP-BINDING, CYTOSKELETON, NUCLEOTIDE- BINDING, WD REPEAT, STRUCTURAL PROTEIN
3owk:A (VAL42) to (LEU88) HUMAN CK2 CATALYTIC DOMAIN IN COMPLEX WITH A BENZOPYRIDOINDOLE DERIVATIVE INHIBITOR | SERINE/THREONINE-PROTEIN KINASE, CK2, INHIBITOR, BENZOPYRIDOINDOLE, ELLIPTICINE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3p1y:D (LYS79) to (ALA111) CRYSTAL STRUCTURE OF THE CHIMERIC ARCHAEOGLOBUS FULGIDUS RNA SPLICING ENDONUCLEASE WITH THE BROADEST SUBSTRATE SPECIFICITY | PROTEIN HOMODIMER, RNA SPLICING ENDONUCLEASE, BROAD SUBSTRATE SPECIFICITY, HYDROLASE
3p1z:L (GLY109) to (SER159) CRYSTAL STRUCTURE OF THE APEROPYRUM PERNIX RNA SPLICING ENDONUCLEASE | MIXED ANTIPARALLEL AND PARALLEL BETA-SHEET, HETEROTETRAMER, RNA SPLICING, RNA, SPLICING ENDONUCLEASE, HYDROLASE
4dtb:A (GLY29) to (ILE67) CRYSTAL STRUCTURE OF F95Y AMINOGLYCOSIDE-2''-PHOSPHOTRANSFERASE TYPE IVA IN COMPLEX WITH GUANOSINE | AMINOGLYCOSIDE KINASE, TRANSFERASE
4umq:A (ILE17) to (LEU64) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN
4uu0:A (GLU482) to (CYS525) CRYSTAL STRUCTURE OF (SR) CALCIUM-ATPASE E2(TG) IN THE PRESENCE OF 14:1 PC | HYDROLASE, CA2+-ATPASE, P-TYPE ATPASE, CATION PUMP, MEMBRANE PROTEIN, LIPID BINDING, LIPID BINDING SITES, DMPC
4eb8:A (GLN44) to (LEU106) CRYSTAL STRUCTURE OF PURINE NUCLEOSIDE PHOSPHORYLASE (W16Y, W94Y, W178Y, H257W) MUTANT FROM HUMAN COMPLEXED WITH DADME-IMMG AND PHOSPHATE | PNP,IMMUCILLIN, PURINE NUCLEOSIDE PHOSPHORYLASE, NUCLEOSIDE BINDING, PURINE BASE BINDING, PURINE-NUCLEOSIDE PHOSPHORYLASE ACTIVITY, DRUG BINDING, TRANSFERASE ACTIVITY, TRANSFERRING GLYCOSYL GROUPS, PHOSPHATE ION BINDING, INTRACELLULAR, CYTOSOL, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4eb8:B (GLN44) to (LEU106) CRYSTAL STRUCTURE OF PURINE NUCLEOSIDE PHOSPHORYLASE (W16Y, W94Y, W178Y, H257W) MUTANT FROM HUMAN COMPLEXED WITH DADME-IMMG AND PHOSPHATE | PNP,IMMUCILLIN, PURINE NUCLEOSIDE PHOSPHORYLASE, NUCLEOSIDE BINDING, PURINE BASE BINDING, PURINE-NUCLEOSIDE PHOSPHORYLASE ACTIVITY, DRUG BINDING, TRANSFERASE ACTIVITY, TRANSFERRING GLYCOSYL GROUPS, PHOSPHATE ION BINDING, INTRACELLULAR, CYTOSOL, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3pzu:B (GLN41) to (ASN75) P212121 CRYSTAL FORM OF THE ENDO-1,4-BETA-GLUCANASE FROM BACILLUS SUBTILIS 168 | ALPHA/BETA BARREL, GLYCOSYL HYDROLASE, CELLULOSE BINDING, HYDROLASE
3q04:A (GLY46) to (LEU88) CRYSTAL STRUCTURE OF THE APO-FORM OF HUMAN CK2 ALPHA AT PH 8.5 | PROTEIN KINASE, APO-FORM, TRANSFERASE
3q3b:B (ILE62) to (LEU104) 6-AMINO-4-(PYRIMIDIN-4-YL)PYRIDONES: NOVEL GLYCOGEN SYNTHASE KINASE-3 INHIBITORS | KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qa8:A (LYS18) to (LYS67) CRYSTAL STRUCTURE OF INHIBITOR OF KAPPA B KINASE BETA | KINASE UBIQUITIN-LIKE DOMAIN, PHOSPHORYLATION, KINASE DOMAIN, UBIQUITIN-LIKE DOMAIN, KINASE, SUBSTRATE BINDING, IMMUNE SYSTEM, SIGNALING PROTEIN
3qa8:B (LYS18) to (LYS67) CRYSTAL STRUCTURE OF INHIBITOR OF KAPPA B KINASE BETA | KINASE UBIQUITIN-LIKE DOMAIN, PHOSPHORYLATION, KINASE DOMAIN, UBIQUITIN-LIKE DOMAIN, KINASE, SUBSTRATE BINDING, IMMUNE SYSTEM, SIGNALING PROTEIN
3qa8:C (LYS18) to (LYS67) CRYSTAL STRUCTURE OF INHIBITOR OF KAPPA B KINASE BETA | KINASE UBIQUITIN-LIKE DOMAIN, PHOSPHORYLATION, KINASE DOMAIN, UBIQUITIN-LIKE DOMAIN, KINASE, SUBSTRATE BINDING, IMMUNE SYSTEM, SIGNALING PROTEIN
3qa8:D (LYS18) to (LYS67) CRYSTAL STRUCTURE OF INHIBITOR OF KAPPA B KINASE BETA | KINASE UBIQUITIN-LIKE DOMAIN, PHOSPHORYLATION, KINASE DOMAIN, UBIQUITIN-LIKE DOMAIN, KINASE, SUBSTRATE BINDING, IMMUNE SYSTEM, SIGNALING PROTEIN
3qa8:E (LYS18) to (LYS67) CRYSTAL STRUCTURE OF INHIBITOR OF KAPPA B KINASE BETA | KINASE UBIQUITIN-LIKE DOMAIN, PHOSPHORYLATION, KINASE DOMAIN, UBIQUITIN-LIKE DOMAIN, KINASE, SUBSTRATE BINDING, IMMUNE SYSTEM, SIGNALING PROTEIN
3qa8:F (LYS18) to (LYS67) CRYSTAL STRUCTURE OF INHIBITOR OF KAPPA B KINASE BETA | KINASE UBIQUITIN-LIKE DOMAIN, PHOSPHORYLATION, KINASE DOMAIN, UBIQUITIN-LIKE DOMAIN, KINASE, SUBSTRATE BINDING, IMMUNE SYSTEM, SIGNALING PROTEIN
3qa8:G (LYS18) to (LYS67) CRYSTAL STRUCTURE OF INHIBITOR OF KAPPA B KINASE BETA | KINASE UBIQUITIN-LIKE DOMAIN, PHOSPHORYLATION, KINASE DOMAIN, UBIQUITIN-LIKE DOMAIN, KINASE, SUBSTRATE BINDING, IMMUNE SYSTEM, SIGNALING PROTEIN
3qa8:H (LYS18) to (LYS67) CRYSTAL STRUCTURE OF INHIBITOR OF KAPPA B KINASE BETA | KINASE UBIQUITIN-LIKE DOMAIN, PHOSPHORYLATION, KINASE DOMAIN, UBIQUITIN-LIKE DOMAIN, KINASE, SUBSTRATE BINDING, IMMUNE SYSTEM, SIGNALING PROTEIN
4f0p:B (ARG318) to (ARG376) MSPJI RESTRICTION ENDONUCLEASE - P31 FORM | ENDONUCLEASE, DNA METHYLATION DEPENDENT, SRA DOMAIN, EPIGENETICS TOOL, CYTOSINE METHYLATION-DEPENDENT ENDONUCLEASE, HYDROLASE
4g0b:B (ILE388) to (ASP433) STRUCTURE OF NATIVE HCT FROM COFFEA CANEPHORA | BAHD SUPERFAMILY, HYDROXYCINNAMOYL TRANSFERASE, TRANSFERASE
4gfg:A (LEU377) to (LEU427) CRYSTAL STRUCTURE OF SPLEEN TYROSINE KINASE COMPLEXED WITH R9021 | SYK, SPLEEN TYPROSINE KINASE, PYRIMIDINE-5-CARBOXAMIDE, ATP-BINDING, HOST-VIRUS INTERACTION, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SH2 DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5knd:F (GLU126) to (ARG166) CRYSTAL STRUCTURE OF THE PI-BOUND V1 COMPLEX | P-LOOP, HYDROLASE, NA(+)-ATPASE, ATP BINDING
5kyy:B (LYS726) to (CYS781) CRYSTAL STRUCTURE OF SEC23 AND TANGO1 PEPTIDE4 COMPLEX | COPII COAT, COLLAGEN SECRETION, CARGO ADAPTER, VESICLE, PROTEIN TRANSPORT
5lxd:A (ILE155) to (ASP204) CRYSTAL STRUCTURE OF DYRK2 IN COMPLEX WITH EHT 1610 (COMPOUND 2) | TRANSFERASE, KINASE, INHIBITOR, UNUSUAL BINDING MODE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
5lxd:B (ILE155) to (ASP204) CRYSTAL STRUCTURE OF DYRK2 IN COMPLEX WITH EHT 1610 (COMPOUND 2) | TRANSFERASE, KINASE, INHIBITOR, UNUSUAL BINDING MODE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC