1n71:D (THR106) to (THR174) CRYSTAL STRUCTURE OF AMINOGLYCOSIDE 6'-ACETYLTRANSFERASE TYPE II IN COMPLEX WITH COENZYME A | AMINOGLYCOSIDE 6'-N-ACETYLTRANSFERASE, ANTIBIOTIC RESISTANCE, COENZYME A
2ajr:A (GLY60) to (ASP100) CRYSTAL STRUCTURE OF POSSIBLE 1-PHOSPHOFRUCTOKINASE (EC 2.7.1.56) (TM0828) FROM THERMOTOGA MARITIMA AT 2.46 A RESOLUTION | TM0828, POSSIBLE 1-PHOSPHOFRUCTOKINASE (EC 2.7.1.56), STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI, TRANSFERASE
1a79:B (ARG18) to (SER46) CRYSTAL STRUCTURE OF THE TRNA SPLICING ENDONUCLEASE FROM METHANOCOCCUS JANNASCHII | ENDONUCLEASE, TRNA ENDONUCLEASE
2oh1:C (ARG140) to (LYS173) CRYSTAL STRUCTURE OF ACETYLTRANSFERASE GNAT FAMILY (YP_013287.1) FROM LISTERIA MONOCYTOGENES 4B F2365 AT 1.46 A RESOLUTION | YP_013287.1, ACETYLTRANSFERASE GNAT FAMILY, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, TRANSFERASE
2asy:A (LEU5) to (GLY51) SOLUTION STRUCTURE OF YDHR PROTEIN FROM ESCHERICHIA COLI | DIMERIC APHA+BETA BARREL, HOMODIMER, STRUCTURAL GENOMICS, ONTARIO CENTRE FOR STRUCTURAL PROTEOMICS, OCSP, UNKNOWN FUNCTION
4wjw:B (PRO44) to (TYR95) CRYSTAL STRUCTURE OF THE CHS5-CHS6 EXOMER CARGO ADAPTOR COMPLEX BOUND TO PORTION OF CHS3 | ADAPTOR PROTEIN, CARGO BINDING, VESICULAR TRAFFICKING, CHITIN SYNTHASE, BIOSYNTHETIC PROTEIN, TRANSPORT PROTEIN-TRANSFERASE COMPLEX
1nj1:A (LEU76) to (LEU114) CRYSTAL STRUCTURE OF PROLYL-TRNA SYNTHETASE FROM METHANOTHERMOBACTER THERMAUTOTROPHICUS BOUND TO CYSTEINE SULFAMOYL ADENYLATE | PROTEIN-AMINOACYLADENYLATE COMPLEX CLASS-II TRNA SYNTHETASE, LIGASE
1nj5:A (LEU76) to (LEU114) CRYSTAL STRUCTURE OF PROLYL-TRNA SYNTHETASE FROM METHANOTHERMOBACTER THERMAUTOTROPHICUS BOUND TO PROLINE SULFAMOYL ADENYLATE | PROTEIN-AMINOACYLADENYLATE COMPLEX CLASS-II TRNA SYNTHETASE, LIGASE
2ayp:A (VAL35) to (PHE83) CRYSTAL STRUCTURE OF CHK1 WITH AN INDOL INHIBITOR | PROTEIN-INHIBITOR COMPLEX, TRANSFERASE
4wnp:D (VAL43) to (GLU93) STRUCTURE OF ULK1 BOUND TO A POTENT INHIBITOR | KINASE, AUTOPHAGY, INHIBITOR
4h1m:A (GLU450) to (PRO506) CRYSTAL STRUCTURE OF PYK2 WITH THE INDOLE 10C | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4wov:A (VAL639) to (MET685) CRYSTAL STRUCTURE OF TYROSINE KINASE 2 JH2 (PSEUDO KINASE DOMAIN) COMPLEXED WITH BMS-066 AKA 2-METHOXY-N-({6-[3-METHYL-7-(METHYLAMINO)- 3,5,8,10-TETRAAZATRICYCLO[7.3.0.0, 6]DODECA-1(9),2(6),4,7,11-PENTAEN- 11-YL]PYRIDIN-2-YL}METHY L)ACETAMIDE | KINASE, TYK2, PSEUDOKINASE, TRANSFERASE-INHIBITOR COMPLEX
4wov:B (VAL639) to (MET685) CRYSTAL STRUCTURE OF TYROSINE KINASE 2 JH2 (PSEUDO KINASE DOMAIN) COMPLEXED WITH BMS-066 AKA 2-METHOXY-N-({6-[3-METHYL-7-(METHYLAMINO)- 3,5,8,10-TETRAAZATRICYCLO[7.3.0.0, 6]DODECA-1(9),2(6),4,7,11-PENTAEN- 11-YL]PYRIDIN-2-YL}METHY L)ACETAMIDE | KINASE, TYK2, PSEUDOKINASE, TRANSFERASE-INHIBITOR COMPLEX
2ow3:B (GLU80) to (ASP133) GLYCOGEN SYNTHASE KINASE-3 BETA IN COMPLEX WITH BIS- (INDOLE)MALEIMIDE PYRIDINOPHANE INHIBITOR | KINASE-INHIBITOR COMPLEX, TRANSFERASE
3f3t:A (VAL292) to (GLU339) KINASE DOMAIN OF CSRC IN COMPLEX WITH INHIBITOR RL38 (TYPE III) | ALLOSTERIC, TYPE III, DFG-OUT, ALTERNATIVE SPLICING, ATP- BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
1o6x:A (GLY9) to (ARG53) NMR SOLUTION STRUCTURE OF THE ACTIVATION DOMAIN OF HUMAN PROCARBOXYPEPTIDASE A2 | ACTIVATION DOMAIN, HYDROLASE, CARBOXYPEPTIDASE, METALLOPROTE
2br1:A (GLU33) to (PHE83) STRUCTURE-BASED DESIGN OF NOVEL CHK1 INHIBITORS: INSIGHTS INTO HYDROGEN BONDING AND PROTEIN-LIGAND AFFINITY | TRANSFERASE, DRUG DESIGN, FURANOPYRIMIDINE, MOLECULAR RECOGNITION, ONCOLOGY, PYRROLOPYRIMIDINE, X-RAY CRYSTALLOGRAPHY, KINASE
3f6x:C (VAL292) to (GLU339) C-SRC KINASE DOMAIN IN COMPLEX WITH SMALL MOLECULE INHIBITOR | KINASE, ATP-BINDING, ALTERNATIVE SPLICING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE- PROTEIN KINASE
3f88:A (VAL82) to (VAL131) GLYCOGEN SYNTHASE KINASE 3BETA INHIBITOR COMPLEX | ENZYME, PROTEIN KINASE, INHIBITOR, ALTERNATIVE SPLICING, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, WNT SIGNALING PATHWAY
4hwt:A (ASN409) to (LEU441) CRYSTAL STRUCTURE OF HUMAN THREONYL-TRNA SYNTHETASE BOUND TO A NOVEL INHIBITOR | AMINOACYL-TRNA SYNTHETASE, PROTEIN-INHIBITOR COMPLEX, LIGASE-LIGASE INHIBITOR COMPLEX
3sg8:B (PHE43) to (THR96) CRYSTAL STRUCTURE OF AMINOGLYCOSIDE-2''-PHOSPHOTRANSFERASE TYPE IVA TOBRAMYCIN COMPLEX | ANTIBIOTIC RESISTANCE ENZYME, TRANSFERASE, AMINOGLYCOSIDE, PHOSPHORYLATION, TRANSFERASE-ANTIBIOTIC COMPLEX
3sg9:B (PHE43) to (THR96) CRYSTAL STRUCTURE OF AMINOGLYCOSIDE-2''-PHOSPHOTRANSFERASE TYPE IVA KANAMYCIN A COMPLEX | ANTIBIOTIC RESISTANCE ENZYME, TRANSFERASE, AMINOGLYCOSIDE, PHOSPHOTRANSFERASE, TRANSFERASE-ANTIBIOTIC COMPLEX
3sgc:A (PHE43) to (THR96) CRYSTAL STRUCTURE OF APO AMINOGLYCOSIDE-2''-PHOSPHOTRANSFERASE TYPE IVA | TRANSFERASE, AMINOGLYCOSIDE, PHOSPHORYLATION, ANTIBIOTIC RESISTANCE ENZYME
2pul:B (ALA57) to (MET114) STRUCTURES OF 5-METHYLTHIORIBOSE KINASE REVEAL SUBSTRATE SPECIFICITY AND UNUSUAL MODE OF NUCLEOTIDE BINDING | 5-METHYLTHIORIBOSE KINASE, METHIONINE RECYCLING PATHWAY, TRANSFERASE
4i5p:A (LYS106) to (GLU160) SELECTIVE & BRAIN-PERMEABLE POLO-LIKE KINASE-2 (PLK-2) INHIBITORS THAT REDUCE -SYNUCLEIN PHOSPHORYLATION IN RAT BRAIN | POLO-LIKE KINASE-2 (PLK-2), SYNUCLEIN, PARKINSON'S DISEASE, KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4i6b:A (LYS106) to (GLU160) SELECTIVE & BRAIN-PERMEABLE POLO-LIKE KINASE-2 (PLK-2) INHIBITORS THAT REDUCE -SYNUCLEIN PHOSPHORYLATION IN RAT BRAIN | POLO-LIKE KINASE-2 (PLK-2), SYNUCLEIN, PARKINSONS DISEASE, KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3soc:B (VAL216) to (ALA268) CRYSTAL STRUCTURE OF ACTIVIN RECEPTOR TYPE-IIA (ACVR2A) KINASE DOMAIN IN COMPLEX WITH A QUINAZOLIN | STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE, PROTEIN KINASE
1cm0:B (LEU603) to (GLU649) CRYSTAL STRUCTURE OF THE PCAF/COENZYME-A COMPLEX | P300/CBP ASSOCIATED FACTOR, COENZYME A, ACETYLTRANSFERASE, COACTIVATOR, SIGNALING PROTEIN
4ibm:A (VAL1027) to (GLU1077) CRYSTAL STRUCTURE OF INSULIN RECEPTOR KINASE DOMAIN IN COMPLEX WITH AN INHIBITOR IRFIN-1 | IRK, KINASE, ATP BINDING, PHOSPHORYLATION, MEMBRANE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3fw7:A (VAL245) to (THR293) STRUCTURE OF BERBERINE BRIDGE ENZYME, H104A VARIANT | BI-COVALENT FLAVINYLATION, N-GLYCOSYLATION, ALAKLOID BIOSYNTHESIS, OXIDOREDUCTASE, ALKALOID METABOLISM, CYTOPLASMIC VESICLE, FAD, FLAVOPROTEIN, GLYCOPROTEIN
3fw9:A (VAL245) to (THR293) STRUCTURE OF BERBERINE BRIDGE ENZYME IN COMPLEX WITH (S)-SCOULERINE | BI-COVALENT FLAVINYLATION, N-GLYCOSYLATION, ALAKLOID BIOSYNTHESIS, OXIDOREDUCTASE, ALKALOID METABOLISM, CYTOPLASMIC VESICLE, FAD, FLAVOPROTEIN, GLYCOPROTEIN
3fxz:A (GLY293) to (VAL343) CRYSTAL STRUCTURE OF PAK1 KINASE DOMAIN WITH RUTHENIUM COMPLEX LAMBDA-FL172 | TRANSFERASE, KINASE, ATP-BINDING, PHOSPHORYLATION, ALLOSTERIC ENZYME, ALTERNATIVE SPLICING, APOPTOSIS, CELL JUNCTION, CYTOPLASM, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE
3svv:A (VAL292) to (GLU339) CRYSTAL STRUCTURE OF T338C C-SRC COVALENTLY BOUND TO VINYLSULFONAMIDE- PYRAZOLOPYRIMIDINE 9 | COVALENTLY BOUND LIGAND, CYSTEINE GATEKEEPER, SRC, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3g0e:A (ALA616) to (GLU671) KIT KINASE DOMAIN IN COMPLEX WITH SUNITINIB | KIT KINASE DOMAIN, SUTENT BINDING, DRUG RESISTANCE, ATP- BINDING, DISEASE MUTATION, GLYCOPROTEIN, IMMUNOGLOBULIN DOMAIN, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, RECEPTOR, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, TRANSFERASE
3g2e:C (LEU1) to (ASP55) STRUCTURE OF PUTATIVE OORC SUBUNIT OF 2-OXOGLUTARATE:ACCEPTOR OXIDOREDUCTASE FROM CAMPYLOBACTER JEJUNI | STRUCTURAL GENOMICS, OORC SUBUNIT OF 2-OXOGLUTARATE:ACCEPTOR OXIDOREDUCTASE, OORC, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, OXIDOREDUCTASE
3g5d:B (VAL292) to (GLU339) KINASE DOMAIN OF CSRC IN COMPLEX WITH DASATINIB | TYPE II, DFG-OUT, TYROSINE-PROTEIN KINASE, DASATINIB, ATP-BINDING, KINASE, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
1pca:A (GLY9) to (ARG55) THREE DIMENSIONAL STRUCTURE OF PORCINE PANCREATIC PROCARBOXYPEPTIDASE A. A COMPARISON OF THE A AND B ZYMOGENS AND THEIR DETERMINANTS FOR INHIBITION AND ACTIVATION | HYDROLASE(C-TERMINAL PEPTIDASE)
1pcp:A (GLU1) to (TYR106) SOLUTION STRUCTURE OF A TREFOIL-MOTIF-CONTAINING CELL GROWTH FACTOR, PORCINE SPASMOLYTIC PROTEIN | GROWTH FACTOR
2cmw:A (GLU68) to (GLU119) STRUCTURE OF HUMAN CASEIN KINASE 1 GAMMA-1 IN COMPLEX WITH 2-(2-HYDROXYETHYLAMINO)-6-(3-CHLOROANILINO)-9- ISOPROPYLPURINE (CASP TARGET) | WNT SIGNALING PATHWAY, SERINE/THREONINE-PROTEIN KINASE, KINASE, TRANSFERASE, ATP-BINDING, PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE PROTEIN KINASE
2qml:A (ILE142) to (GLU181) CRYSTAL STRUCTURE OF AN UNCHARACTERIZED PROTEIN (BH2621) FROM BACILLUS HALODURANS AT 1.55 A RESOLUTION | STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, UNKNOWN FUNCTION
2qq7:A (VAL292) to (GLU339) CRYSTAL STRUCTURE OF DRUG RESISTANT SRC KINASE DOMAIN WITH IRREVERSIBLE INHIBITOR | SRC KINASE DOMAIN, DRUG RESISTANCE, IRREVERSIBLE INHIBITOR, ALTERNATIVE SPLICING, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
4ix4:A (VAL197) to (ALA262) CRYSTAL STRUCTURE OF A STT7 HOMOLOG FROM MICROMONAS ALGAE IN COMPLEX WITH ADP | PROTEIN KINASE, CANONICAL PROTEIN KINASE FOLD, ATP BINDING, TRANSFERASE
4ix5:A (VAL197) to (ALA262) CRYSTAL STRUCTURE OF A STT7 HOMOLOG FROM MICROMONAS ALGAE IN COMPLEX WITH AMP-PNP | PROTEIN KINASE, CANONICAL PROTEIN KINASE FOLD, ATP BINDING, TRANSFERASE
4ix6:A (VAL197) to (ALA262) CRYSTAL STRUCTURE OF A STT7 HOMOLOG FROM MICROMONAS ALGAE SOAKED WITH ATP | PROTEIN KINASE, CANONICAL PROTEIN KINASE FOLD, ATP BINDING, TRANSFERASE
4ix6:B (VAL197) to (ALA262) CRYSTAL STRUCTURE OF A STT7 HOMOLOG FROM MICROMONAS ALGAE SOAKED WITH ATP | PROTEIN KINASE, CANONICAL PROTEIN KINASE FOLD, ATP BINDING, TRANSFERASE
1pyt:A (GLY9) to (ARG55) TERNARY COMPLEX OF PROCARBOXYPEPTIDASE A, PROPROTEINASE E, AND CHYMOTRYPSINOGEN C | TERNARY COMPLEX (ZYMOGEN), SERINE PROTEINASE, C-TERMINAL PEPTIDASE
3gsy:A (VAL245) to (THR293) STRUCTURE OF BERBERINE BRIDGE ENZYME IN COMPLEX WITH DEHYDROSCOULERINE | COMPLEX WITH DEHYDROSCOULERINE, BICOVALENT FLAVINYLATION, N- GLYCOSYLATION, P-CRESOL METHYL HYDROXYLASE SUPERFAMILY, ALKALOID METABOLISM, CYTOPLASMIC VESICLE, FAD, FLAVOPROTEIN, GLYCOPROTEIN, OXIDOREDUCTASE
4j71:B (GLY79) to (ASP133) CRYSTAL STRUCTURE OF GSK3B IN COMPLEX WITH INHIBITOR 1R | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, KINASE, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4j7b:A (LYS62) to (GLU117) CRYSTAL STRUCTURE OF POLO-LIKE KINASE 1 | FIRST COMPLEX STRUCTURE OF KD AND PBD DOMAIN, REGULATOR OF MITOSIS, PHOSPHORYLATED TARGET PROTEIN, TRANSFERASE
4j7b:D (LYS62) to (VAL115) CRYSTAL STRUCTURE OF POLO-LIKE KINASE 1 | FIRST COMPLEX STRUCTURE OF KD AND PBD DOMAIN, REGULATOR OF MITOSIS, PHOSPHORYLATED TARGET PROTEIN, TRANSFERASE
4j95:A (VAL514) to (GLU565) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC K659N MUTATION RESPONSIBLE FOR AN UNCLASSIFIED CRANIOSYNOSTOSIS SYNDROME IN SPACE GROUP C2. | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, RECEPTOR TYROSINE KINASE, ATP BINDING, TRANSFERASE
4j95:D (VAL514) to (GLU565) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC K659N MUTATION RESPONSIBLE FOR AN UNCLASSIFIED CRANIOSYNOSTOSIS SYNDROME IN SPACE GROUP C2. | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, RECEPTOR TYROSINE KINASE, ATP BINDING, TRANSFERASE
4j97:B (VAL514) to (LYS569) CRYSTAL STRUCURE OF FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN HARBORING THE PATHOGENIC GAIN-OF-FUNCTION K659E MUTATION IDENTIFIED IN ENDOMETRIAL CANCER. | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, RECEPTOR TYROSINE KINASE, ATP BINDING, TRANSFERASE
3thb:A (LYS76) to (ARG135) STRUCTURE OF PLK1 KINASE DOMAIN IN COMPLEX WITH A BENZOLACTAM-DERIVED INHIBITOR | KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1q4l:A (GLU80) to (LEU130) GSK-3 BETA COMPLEXED WITH INHIBITOR I-5 | KINASE, INSULIN PATHWAY, TRANSFERASE
1q5k:B (GLU80) to (ASP133) CRYSTAL STRUCTURE OF GLYCOGEN SYNTHASE KINASE 3 IN COMPLEXED WITH INHIBITOR | KINASE-INHIBITOR COMPLEX, TRANSFERASE
1q5y:A (GLY52) to (ILE98) NICKEL-BOUND C-TERMINAL REGULATORY DOMAIN OF NIKR | NICKEL BINDING, REGULATORY DOMAIN, BETA SANDWICH, METAL BINDING PROTEIN
3tpd:A (ILE179) to (GLU234) STRUCTURE OF PHIPA, MONOCLINIC FORM | HIPA, PERSISTENCE, MULTIDRUG TOLERANCE, HIPB, TRANSFERASE
3tpt:A (ILE179) to (GLU234) STRUCTURE OF HIPA(D309Q) BOUND TO ADP | PERSISTENCE, MULTIDRUG TOLERANCE, HIPA, HIPB, TRANSFERASE
3tr5:A (GLU392) to (VAL437) STRUCTURE OF A PEPTIDE CHAIN RELEASE FACTOR 3 (PRFC) FROM COXIELLA BURNETII | PROTEIN SYNTHESIS, TRANSLATION
2dyl:A (GLY159) to (GLU213) CRYSTAL STRUCTURE OF HUMAN MITOGEN-ACTIVATED PROTEIN KINASE KINASE 7 ACTIVATED MUTANT (S287D, T291D) | MKK7, KINASE, ACTIVATED MUTANT, ATP-BINDING, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, TRANSFERASE
1qkh:A (ARG29) to (TYR61) SOLUTION STRUCTURE OF THE RIBOSOMAL PROTEIN S19 FROM THERMUS THERMOPHILUS | RIBOSOME, RIBOSOMAL PROTEIN, THERMUS THERMOPHILUS, S19
1f8i:D (THR235) to (LYS262) CRYSTAL STRUCTURE OF ISOCITRATE LYASE:NITROPROPIONATE:GLYOXYLATE COMPLEX FROM MYCOBACTERIUM TUBERCULOSIS | ALPHA-BETA BARREL, SWAPPED HELICES, CLOSED CONFORMATION, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, LYASE
3u81:A (THR164) to (GLY214) CRYSTAL STRUCTURE OF A SAH-BOUND SEMI-HOLO FORM OF RAT CATECHOL-O- METHYLTRANSFERASE | METHYLTRANSFERASE, NEUROTRANSMITTER DEGRADATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3ucq:A (HIS203) to (TRP245) CRYSTAL STRUCTURE OF AMYLOSUCRASE FROM DEINOCOCCUS GEOTHERMALIS | THERMOSTABILITY, AMYLOSE SYNTHESIS, SUCROSE ISOMERIZATION, BETA/ALPHA-BARREL, CARBOHYDRATE BINDING, TRANSFERASE, GLYCOSIDE HYDROLASE, GLUCOSYLTRANSFERASE
3ueq:A (TYR209) to (TRP247) CRYSTAL STRUCTURE OF AMYLOSUCRASE FROM NEISSERIA POLYSACCHAREA IN COMPLEX WITH TURANOSE | BETA/ALPHA-BARREL, GLYCOSIDE HYDROLASE, AMYLOSE SYNTHESIS, SUCROSE ISOMERIZATION, GLUCOSYLTRANSFERASE, CARBOHYDRATE, TRANSFERASE
3uer:A (HIS203) to (TRP245) CRYSTAL STRUCTURE OF AMYLOSUCRASE FROM DEINOCOCCUS GEOTHERMALIS IN COMPLEX WITH TURANOSE | ALPHA/BETA-BARREL, CARBOHYDRATE, TRANSFERASE, GLUCOSYLTRANSFERASE, GLYCOSIDE HYDROLASE, THERMOSTABILITY, AMYLOSE SYNTHESIS, SUCROSE ISOMERIZATION
3hko:A (ARG33) to (VAL88) CRYSTAL STRUCTURE OF A CDPK KINASE DOMAIN FROM CRYPTOSPORIDIUM PARVUM, CGD7_40 | STRUCTURAL GENOMICS, PROTIST PARASITE, CRYPTOSPORIDIUM PARVUM, CDPK, ZINC FINGER, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3uh0:A (LEU93) to (LYS129) CRYSTAL STRUCTURE OF THE YEAST MITOCHONDRIAL THREONYL-TRNA SYNTHETASE (MST1) IN COMPLEX WITH THREONYL SULFAMOYL ADENYLATE | THREONYL-TRNA SYNTHETASE, TRNA, THREONINE TRNA, THREONYL ADENYLATE, THREONYL SULFAMOYL ADENYLATE, AMINOACYL-TRNA SYNTHETASE CLASS II, LIGASE
2f2h:C (PRO348) to (TYR387) STRUCTURE OF THE YICI THIOSUGAR MICHAELIS COMPLEX | BETA8ALPHA8 BARREL, HYDROLASE
4yye:B (LEU93) to (LEU128) CRYSTAL STRUCTURE OF THE YEAST MITOCHONDRIAL THREONYL-TRNA SYNTHETASE (MST1) IN COMPLEX WITH THE CANONICAL TRNATHR AND THREONYL SULFAMOYL ADENYLATE | AMINOACYL-TRNA SYNTHETASE, THRRS, MST1, TRNA, RIBONUCLEOPROTEIN COMPLEX, LIGASE-RNA COMPLEX
1g3n:A (ARG38) to (ASP102) STRUCTURE OF A P18(INK4C)-CDK6-K-CYCLIN TERNARY COMPLEX | CYCLIN-DEPENDENT KINASE, INK4 INHIBITOR, VIRAL CYCLIN, CELL CYCLE, SIGNALING PROTEIN
1g3n:E (ARG38) to (ASP102) STRUCTURE OF A P18(INK4C)-CDK6-K-CYCLIN TERNARY COMPLEX | CYCLIN-DEPENDENT KINASE, INK4 INHIBITOR, VIRAL CYCLIN, CELL CYCLE, SIGNALING PROTEIN
3uqg:B (VAL292) to (GLU339) C-SRC KINASE DOMAIN IN COMPLEX WITH BUMPLESS BKI ANALOG UW1243 | TYROSINE PROTEIN KINASE, ATP-BINDING, KINASE DOMAIN, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
2fia:A (ARG110) to (GLU155) THE CRYSTAL STRUCTURE OF THE ACETYLTRANSFERASE FROM ENTEROCOCCUS FAECALIS | ACETYLTRANSFERASE, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSFERASE
2fia:B (ARG110) to (GLU157) THE CRYSTAL STRUCTURE OF THE ACETYLTRANSFERASE FROM ENTEROCOCCUS FAECALIS | ACETYLTRANSFERASE, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSFERASE
4zgz:D (VAL172) to (GLU219) STRUCTURE OF HUMAN ANTIZYME INHIBITOR IN COMPLEX WITH A C-TERMINAL FRAGMENT OF ANTIZYME | TIM BARREL DOMAIN, BETA-SHEET DOMAIN, INHIBITION, ANTIZYME, PLASMA, PROTEIN BINDING
4kr3:A (MET128) to (LEU242) GLYCYL-TRNA SYNTHETASE MUTANT E71G IN COMPLEX WITH TRNA-GLY | ROSSMANN FOLD, AMINOACYLATION, TRNA-GLY, LIGASE-RNA COMPLEX
3v8h:B (ARG111) to (ALA154) CRYSTAL STRUCTURE OF THYMIDYLATE SYNTHASE FROM BURKHOLDERIA THAILANDENSIS | SSGCID, THYMIDYLATE SYNTHASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, TRANSFERASE
3i4e:A (ASP236) to (LYS263) CRYSTAL STRUCTURE OF ISOCITRATE LYASE FROM BURKHOLDERIA PSEUDOMALLEI | ISOCITRATE LYASE, STRUCTURAL GENOMICS, LYASE, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, SSGCID
3i4e:C (ASP236) to (LYS263) CRYSTAL STRUCTURE OF ISOCITRATE LYASE FROM BURKHOLDERIA PSEUDOMALLEI | ISOCITRATE LYASE, STRUCTURAL GENOMICS, LYASE, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, SSGCID
2vya:A (PRO231) to (ARG285) CRYSTAL STRUCTURE OF FATTY ACID AMIDE HYDROLASE CONJUGATED WITH THE DRUG-LIKE INHIBITOR PF-750 | HYDROLASE, FATTY ACID AMIDE HYDROLYSE, GOLGI APPARATUS, ENDOPLASMIC RETICULUM, INHIBITOR, DRUG- LIKE, TRANSMEMBRANE, FAAH, CHIMERA, MEMBRANE, COVALENT, HUMANIZED
1t0g:A (HIS8) to (VAL40) HYPOTHETICAL PROTEIN AT2G24940.1 FROM ARABIDOPSIS THALIANA HAS A CYTOCHROME B5 LIKE FOLD | STRUCTURAL GENOMICS, HYPOTHETICAL PROTEIN, AT2G24940.1, PSI, PROTEIN STRUCTURE INITIATIVE, CENTER FOR EUKARYOTIC STRUCTURAL GENOMICS, CESG, UNKNOWN FUNCTION
2gqc:A (VAL6) to (VAL42) SOLUTION STRUCTURE OF THE N-TERMINAL DOMAIN OF RHOMBOID INTRAMEMBRANE PROTEASE FROM P. AERUGINOSA | ALPHA-BETA DOMAIN, HYDROLASE
4lgg:A (VAL292) to (GLU339) STRUCTURE OF 3MB-PP1 BOUND TO ANALOG-SENSITIVE SRC KINASE | KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2hak:D (GLY76) to (GLY134) CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1 | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE
2hak:E (ARG77) to (GLY134) CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK1/PAR-1 | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE
2hw0:A (TRP17) to (ASN63) NMR SOLUTION STRUCTURE OF THE NUCLEASE DOMAIN FROM THE REPLICATOR INITIATOR PROTEIN FROM PORCINE CIRCOVIRUS PCV2 | ALPHA+BETA, HYDROLASE, REPLICATION
3w3t:A (ASP637) to (HIS668) CRYSTAL STRUCTURE OF KAP121P | HEAT REPEAT, NUCLEAR IMPORT, PROTEIN TRANSPORT
3w3u:A (ASP637) to (HIS668) CRYSTAL STRUCTURE OF KAP121P MUTANT R349A/Q350A/D353A/E396A/N430K/D438A/N477A | HEAT REPEAT, NUCLEAR IMPORT, PROTEIN TRANSPORT
3w3w:A (ASP637) to (HIS668) CRYSTAL STRUCTURE OF KAP121P BOUND TO STE12P | HEAT REPEAT, NUCLEAR IMPORT, PROTEIN TRANSPORT-DNA BINDING PROTEIN COMPLEX
2hz4:C (VAL268) to (GLU316) ABL KINASE DOMAIN UNLIGATED AND IN COMPLEX WITH TETRAHYDROSTAUROSPORINE | TYROSINE KINASE, TRANSFERASE
3w3x:A (ASP637) to (HIS668) CRYSTAL STRUCTURE OF KAP121P BOUND TO PHO4P | HEAT REPEAT, NUCLEAR IMPORT, PROTEIN TRANSPORT-TRANSCRIPTION COMPLEX
3w3y:A (ASP637) to (HIS668) CRYSTAL STRUCTURE OF KAP121P BOUND TO NUP53P | HEAT REPEAT, NUCLEAR IMPORT, PROTEIN TRANSPORT-DNA BINDING PROTEIN COMPLEX
2hzi:B (VAL268) to (GLU316) ABL KINASE DOMAIN IN COMPLEX WITH PD180970 | TYROSINE KINASE, TRANSFERASE
2i0x:A (MET1) to (GLY35) HYPOTHETICAL PROTEIN PF1117 FROM PYROCOCCUS FURIOSUS | PF1117, HYPOTHETICAL PROTEIN, PYROCOCCUS FURIOSUS, PSI, STRUCTURAL GENOMICS, SOUTHEAST COLLABORATORY FOR STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, SECSG, UNKNOWN FUNCTION
1igw:A (ASP239) to (HIS266) CRYSTAL STRUCTURE OF THE ISOCITRATE LYASE FROM THE A219C MUTANT OF ESCHERICHIA COLI | BETA BARREL, LYASE
2i4n:A (THR73) to (TYR106) RHODOPSEUDOMONAS PALUSTRIS PROLYL-TRNA SYNTHETASE IN COMPLEX WITH CYSAMS | ALPHA BETA, LIGASE
2i4n:B (THR73) to (TYR106) RHODOPSEUDOMONAS PALUSTRIS PROLYL-TRNA SYNTHETASE IN COMPLEX WITH CYSAMS | ALPHA BETA, LIGASE
2i4o:B (THR73) to (TYR106) RHODOPSEUDOMONAS PALUSTRIS PROLYL-TRNA SYNTHETASE IN COMPLEX WITH ATP | ALPHA BETA, LIGASE
2i8e:A (ALA2) to (GLY39) STRUCTURE OF SSO1404, A PREDICTED DNA REPAIR-ASSOCIATED PROTEIN FROM SULFOLOBUS SOLFATARICUS P2 | DNA REPAIR, UNKNOWN FUNCTION, STRUCTURAL GENOMICS, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, PSI, PROTEIN STRUCTURE INITIATIVE
5a9w:A (THR306) to (ARG361) STRUCTURE OF GDPCP BIPA | RIBOSOMAL PROTEIN, RIBOSOME, TRANSLATIONAL GTPASE FACTORS
5a9y:A (VAL487) to (ARG529) STRUCTURE OF PPGPP BIPA | RIBOSOMAL PROTEIN, BIPA, RIBOSOME, TRANSLATIONAL GTPASE FACTORS
2idl:A (ALA23) to (GLU71) CRYSTAL STRUCTURE OF CONSERVED PROTEIN OF UNKNOWN FUNCTION FROM STREPTOCOCCUS PNEUMONIAE | CONSERVED HYPOTHETICAL, MCSG, PSI2, MAD, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, UNKNOWN FUNCTION
2iew:A (LEU27) to (GLU118) CRYSTAL STRUCTURE OF INOSITOL PHOSPHATE MULTIKINASE IPK2 FROM S. CEREVISIAE | ATP-GRASP FOLD RELATED, TRANSFERASE
2if8:A (LEU27) to (GLU118) CRYSTAL STRUCTURE OF INOSITOL PHOSPHATE MULTIKINASE IPK2 IN COMPLEX WITH ADP AND MN2+ FROM S. CEREVISIAE | ATP-GRASP FOLD RELATED, TRANSFERASE
4mkc:A (PRO1144) to (GLU1197) CRYSTAL STRUCTURE OF ANAPLASTIC LYMPHOMA KINASE COMPLEXED WITH LDK378 | KINASE DOMAIN, PHOSPHOTRANSFERASE, ATP BINDING, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3j3s:3 (LEU127) to (ASN169) STRUCTURAL DYNAMICS OF THE MECA-CLPC COMPLEX REVEALED BY CRYO-EM | CLPC, MECA, AAA+ ATPASE, PROTEIN UNFOLDING, CHAPERONE
1je5:A (ARG35) to (TYR111) CRYSTAL STRUCTURE OF GP2.5, A SINGLE-STRANDED DNA BINDING PROTEIN ENCODED BY BACTERIOPHAGE T7 | OB-FOLD, BETA BARREL, DNA BINDING PROTEIN
1je5:B (ARG35) to (TYR111) CRYSTAL STRUCTURE OF GP2.5, A SINGLE-STRANDED DNA BINDING PROTEIN ENCODED BY BACTERIOPHAGE T7 | OB-FOLD, BETA BARREL, DNA BINDING PROTEIN
2xix:A (ALA65) to (PRO125) PROTEIN KINASE PIM-1 IN COMPLEX WITH FRAGMENT-1 FROM CRYSTALLOGRAPHIC FRAGMENT SCREEN | ATP-BINDING, PHOSPHORYLATION, TRANSFERASE
1w2c:B (GLY205) to (GLN249) HUMAN INOSITOL (1,4,5) TRISPHOSPHATE 3-KINASE COMPLEXED WITH MN2+/AMPPNP/INS(1,4,5)P3 | INOSITOL PHOSPHATE KINASE, AMPPNP, IP3, TRANSFERASE
4n70:A (ALA65) to (GLU121) PIM1 COMPLEXED WITH A PYRIDYLCARBOXAMIDE | KINASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1w7p:C (GLN147) to (ILE199) THE CRYSTAL STRUCTURE OF ENDOSOMAL COMPLEX ESCRT-II (VPS22/VPS25/VPS36) | ESCRT-II COMPLEX, ENDOSOMAL PROTEIN SORTING, PROTEIN TRANSPORT
2jnj:A (GLY10) to (ILE49) SOLUTION STRUCTURE OF THE P8 TFIIH SUBUNIT | PROTEIN, TRANSCRIPTION
2jnj:B (GLY10) to (ILE49) SOLUTION STRUCTURE OF THE P8 TFIIH SUBUNIT | PROTEIN, TRANSCRIPTION
3zj0:A (PRO165) to (ARG202) THE HUMAN O-GLCNACASE C-TERMINAL DOMAIN IS A PSEUDO HISTONE ACETYLTRANSFERASE | TRANSFERASE, O-GLCNAC HAT, HISTONE ACETYLTRANSFERASE, OGA HAT DOMAIN
4ni2:B (ILE562) to (SER605) CRYSTAL STRUCTURE OF THE HETERODIMERIC CATALYTIC DOMAIN OF WILD-TYPE HUMAN SOLUBLE GUANYLATE CYCLASE | HETERODIMERIC, LYASE, CGMP BIOSYNTHESIS, NITRIC OXIDE, CYCLASE, GTP- BINDING, METAL-BINDING, NUCLEOTIDE BINDING, CYTOSOL
2kdo:A (MET174) to (CYS212) STRUCTURE OF THE HUMAN SHWACHMAN-BODIAN-DIAMOND SYNDROME PROTEIN, SBDS | SBDS PROTEIN, NMR PROTEIN STRUCTURE, RNA-INTERACTING PROTEIN, DISEASE MUTATION, PHOSPHOPROTEIN, RIBOSOME BIOGENESIS, RNA BINDING PROTEIN
5c01:A (VAL639) to (GLU691) CRYSTAL STRUCTURE OF KINASE | PSEUDOKINASE DOMAIN, TRANSFERASE
5c01:B (VAL639) to (HIS692) CRYSTAL STRUCTURE OF KINASE | PSEUDOKINASE DOMAIN, TRANSFERASE
5c03:A (VAL639) to (HIS692) CRYSTAL STRUCTURE OF KINASE | PSEUDOKINASE DOMAIN, TRANSFERASE
5c03:B (VAL639) to (HIS692) CRYSTAL STRUCTURE OF KINASE | PSEUDOKINASE DOMAIN, TRANSFERASE
3znj:2 (MET1) to (VAL58) CRYSTAL STRUCTURE OF UNLIGANDED CLCF FROM R.OPACUS 1CP IN CRYSTAL FORM 1. | LYASE, FERREDOXIN FOLD, DEHALOGENATION, 3-CHLOROCATECHOL PATHWAY
3znj:Z (MET1) to (VAL58) CRYSTAL STRUCTURE OF UNLIGANDED CLCF FROM R.OPACUS 1CP IN CRYSTAL FORM 1. | LYASE, FERREDOXIN FOLD, DEHALOGENATION, 3-CHLOROCATECHOL PATHWAY
3znj:c (MET1) to (VAL58) CRYSTAL STRUCTURE OF UNLIGANDED CLCF FROM R.OPACUS 1CP IN CRYSTAL FORM 1. | LYASE, FERREDOXIN FOLD, DEHALOGENATION, 3-CHLOROCATECHOL PATHWAY
3zon:A (VAL639) to (HIS692) HUMAN TYK2 PSEUDOKINASE DOMAIN BOUND TO A KINASE INHIBITOR | TRANSFERASE, JAK
2yaa:A (GLY36) to (GLY98) CRYSTAL STRUCTURE OF THE AUTOINHIBITED FORM OF MOUSE DAPK2 IN COMPLEX WITH ATP | TRANSFERASE, APOPTOSIS
2yac:A (LYS76) to (ARG135) CRYSTAL STRUCTURE OF POLO-LIKE KINASE 1 IN COMPLEX WITH NMS-P937 | TRANSFERASE, ATP-BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, NUCLEUS
3zrl:A (GLY79) to (ASP133) IDENTIFICATION OF 2-(4-PYRIDYL)THIENOPYRIDINONES AS GSK-3BETA INHIBITORS | TRANSFERASE-PEPTIDE COMPLEX, KINASE
3zsh:A (VAL50) to (THR106) X-RAY STRUCTURE OF P38ALPHA BOUND TO SCIO-469 | TRANSFERASE
5c4l:B (PHE43) to (THR96) CONFORMATIONAL ALTERNATE OF SISOMICIN IN COMPLEX WITH APH(2")-IVA | AMINOGLYCOSIDE PHOSPHOTRANSFERASE, ANTIBIOTIC RESISTANCE, TRANSFERASE
3zut:A (ASN44) to (GLY99) THE STRUCTURE OF OST1 (D160A) KINASE | TRANSFERASE, KINASE REGULATION, PLANT ABIOTIC STRESS, SIGNALING
1kwm:B (GLY9) to (LYS57) HUMAN PROCARBOXYPEPTIDASE B: THREE-DIMENSIONAL STRUCTURE AND IMPLICATIONS FOR THROMBIN-ACTIVATABLE FIBRINOLYSIS INHIBITOR (TAFI) | HYDROLASE, PROCARBOXYPEPTIDASE B
4nzr:M (GLY80) to (GLY143) CRYSTAL STRUCTURE OF THE ANTIBODY-BINDING REGION OF PROTEIN M (PROTEIN M TD) IN COMPLEX WITH ANTI-HIV ANTIBODY PGT135 FAB | LEUCINE-RICH REPEAT, BROAD ANTIBODY-BINDING, BLOCK ANTIBODY-ANTIGEN UNION, VARIABLE REGION, IMMUNE SYSTEM-PROTEIN BINDING COMPLEX
1l1l:A (GLN573) to (GLU607) CRYSTAL STRUCTURE OF B-12 DEPENDENT (CLASS II) RIBONUCLEOTIDE REDUCTASE | 10-STRANDED ALPHA-BETA BARREL, CENTRAL FINGER LOOP, OXIDOREDUCTASE
1l1l:B (GLN573) to (LYS611) CRYSTAL STRUCTURE OF B-12 DEPENDENT (CLASS II) RIBONUCLEOTIDE REDUCTASE | 10-STRANDED ALPHA-BETA BARREL, CENTRAL FINGER LOOP, OXIDOREDUCTASE
1l1l:D (GLN573) to (LYS611) CRYSTAL STRUCTURE OF B-12 DEPENDENT (CLASS II) RIBONUCLEOTIDE REDUCTASE | 10-STRANDED ALPHA-BETA BARREL, CENTRAL FINGER LOOP, OXIDOREDUCTASE
4o4c:A (GLN34) to (GLU86) CRYSTAL STRUCTURE OF AN INOSITOL HEXAKISPHOSPHATE KINASE APO-EHIP6KA | PDKG KINASE, INOSITOL PHOSPHATE, TRANSFERASE
4o4c:B (GLN34) to (GLU86) CRYSTAL STRUCTURE OF AN INOSITOL HEXAKISPHOSPHATE KINASE APO-EHIP6KA | PDKG KINASE, INOSITOL PHOSPHATE, TRANSFERASE
2ym8:A (VAL35) to (PHE83) CRYSTAL STRUCTURE OF CHECKPOINT KINASE 1 (CHK1) IN COMPLEX WITH INHIBITORS | TRANSFERASE, DNA REPAIR, SERINE/THREONINE KINASE
3k5h:C (PRO310) to (PRO362) CRYSTAL STRUCTURE OF CARBOXYAMINOIMIDAZOLE RIBONUCLEOTIDE SYNTHASE FROM ASPERIGILLUS CLAVATUS COMPLEXED WITH ATP | PURINE BIOSYNTHESIS, ATP-GRASP, LYASE
3k83:B (PRO231) to (ARG285) CRYSTAL STRUCTURE ANALYSIS OF A BIPHENYL/OXAZOLE/CARBOXYPYRIDINE ALPHA-KETOHETEROCYCLE INHIBITOR BOUND TO A HUMANIZED VARIANT OF FATTY ACID AMIDE HYDROLASE | FAAH, OXAZOLE, CONJUGATE, COVALENT MODIFICATION, HYDROLASE, MEMBRANE, TRANSMEMBRANE, MONOTOPIC, FATTY ACID, SERINE HYDROLASE, ENDOCANNABINOID, REVERSIBLE INHIBITOR.
1m0v:A (ALA64) to (VAL101) NMR STRUCTURE OF THE TYPE III SECRETORY DOMAIN OF YERSINIA YOPH COMPLEXED WITH THE SKAP-HOM PHOSPHO-PEPTIDE N-ACETYL- DEPYDDPF-NH2 | HIGH RESOLUTION STRUCTURE, HYDROLASE
2zit:A (VAL488) to (THR533) STRUCTURE OF THE EEF2-EXOA-NAD+ COMPLEX | ELONGATION FACTOR, TOXIN, ADP-RIBOSYLATION, TOXIN-SUBSTRATE COMPLEX, CYTOPLASM, GTP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTEIN BIOSYNTHESIS, RNA-BINDING, RRNA- BINDING, GLYCOSYLTRANSFERASE, NAD, TRANSFERASE, BIOSYNTHETIC PROTEIN/TRANSFERASE COMPLEX
1m52:A (VAL268) to (GLU316) CRYSTAL STRUCTURE OF THE C-ABL KINASE DOMAIN IN COMPLEX WITH PD173955 | KINASE, KINASE INHIBITOR, PD173955, ACTIVATION LOOP, TRANSFERASE
1xsi:A (PRO348) to (TYR387) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
1xsj:E (PRO348) to (TYR387) STRUCTURE OF A FAMILY 31 ALPHA GLYCOSIDASE | BETA(8)ALPHA(8) BARREL AND BETA SANDWICH DOMAINS, HYDROLASE
4acc:B (GLU80) to (LEU130) GSK3B IN COMPLEX WITH INHIBITOR | TRANSFERASE
1mbb:A (ASN233) to (ALA264) OXIDOREDUCTASE | FLAVOENZYME, OXIDOREDUCTASE
4ach:A (GLY79) to (ASP133) GSK3B IN COMPLEX WITH INHIBITOR | TRANSFERASE
1y10:A (GLY331) to (ARG376) MYCOBACTERIAL ADENYLYL CYCLASE RV1264, HOLOENZYME, INHIBITED STATE | ADENYLYL CYCLASE FOLD, LYASE
1y10:D (GLY331) to (ARG376) MYCOBACTERIAL ADENYLYL CYCLASE RV1264, HOLOENZYME, INHIBITED STATE | ADENYLYL CYCLASE FOLD, LYASE
3kk9:A (LEU37) to (ASP90) CAMKII SUBSTRATE COMPLEX B | CAMKII, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE
5d11:B (VAL292) to (GLU339) KINASE DOMAIN OF CSRC IN COMPLEX WITH RL235 | KINASE INHIBITOR, DRUG RESISTANCE, TRANSFERASE
4p2f:A (GLY384) to (TYR420) MONOMERIC FORM OF A SINGLE MUTANT (F363R) OF MYCOBACTERIAL ADENYLYL CYCLASE RV1625C | ADENYLYL CYCLASE, SINGLE MUTANT, ALPHA/BETA FOLD, SIGNAL TRANSDUCTION
4p3n:B (ASN376) to (LEU408) STRUCTURAL BASIS FOR FULL-SPECTRUM INHIBITION OF THREONYL-TRNA SYNTHETASE BY BORRELIDIN 1 | SYNTHETASE, INHIBITOR, LIGASE-LIGASE INHIBITOR COMPLEX
4p3n:C (ASN376) to (LEU408) STRUCTURAL BASIS FOR FULL-SPECTRUM INHIBITION OF THREONYL-TRNA SYNTHETASE BY BORRELIDIN 1 | SYNTHETASE, INHIBITOR, LIGASE-LIGASE INHIBITOR COMPLEX
3kmw:A (ILE217) to (HIS270) CRYSTAL STRUCTURE OF THE ILK/ALPHA-PARVIN CORE COMPLEX (MGATP) | CELL ADHESION, ANK REPEAT, ATP-BINDING, CELL JUNCTION, CELL MEMBRANE, INTEGRIN-BINDING PROTEIN, MEMBRANE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, PSEUDOKINASE, ACTIN-BINDING, ALTERNATIVE SPLICING, CYTOPLASM, CYTOSKELETON
3a17:C (ILE214) to (ALA284) CRYSTAL STRUCTURE OF ALDOXIME DEHYDRATASE (OXDRE) IN COMPLEX WITH BUTYRALDOXIME (CO-CRYSTAL) | BETA BARREL, HEME PROTEIN, LYASE
3a17:G (ILE214) to (ALA284) CRYSTAL STRUCTURE OF ALDOXIME DEHYDRATASE (OXDRE) IN COMPLEX WITH BUTYRALDOXIME (CO-CRYSTAL) | BETA BARREL, HEME PROTEIN, LYASE
4p7k:A (VAL208) to (ILE254) RAT COMT IN COMPLEX WITH SINEFUNGIN | METHYLTRANSFERASE, NEUROTRANSMITTER DEGRADATION, TRANSFERASE, ALTERNATIVE INITIATION, CATECHOLAMINE METABOLISM, CELL MEMBRANE, METAL-BINDING, PHOSPHOPROTEIN, S-ADENOSYL-L-METHIONINE, SIGNAL- ANCHOR, TRANSMEMBRANE ANCHOR, ENZYME MECHANISM, CONFORMATIONAL CHANGE
1msv:B (GLY278) to (LYS327) THE S68A S-ADENOSYLMETHIONINE DECARBOXYLASE PROENZYME PROCESSING MUTANT. | SPERMIDINE BIOSYNTHESIS, LYASE, DECARBOXYLASE, PYRUVATE, S- ADENOSYLMETHIONINE, SANDWICH, ALLOSTERIC ENZYME, PYRUVOYL
1ybu:A (SER414) to (ASP456) MYCOBACTERIUM TUBERCULOSIS ADENYLYL CYCLASE RV1900C CHD, IN COMPLEX WITH A SUBSTRATE ANALOG. | CYCLASE HOMOLOGY DOMAIN, CHD, RV1900C, HYDROLASE
1ybu:B (SER414) to (ASP456) MYCOBACTERIUM TUBERCULOSIS ADENYLYL CYCLASE RV1900C CHD, IN COMPLEX WITH A SUBSTRATE ANALOG. | CYCLASE HOMOLOGY DOMAIN, CHD, RV1900C, HYDROLASE
1ybu:C (SER414) to (ASP456) MYCOBACTERIUM TUBERCULOSIS ADENYLYL CYCLASE RV1900C CHD, IN COMPLEX WITH A SUBSTRATE ANALOG. | CYCLASE HOMOLOGY DOMAIN, CHD, RV1900C, HYDROLASE
1ybu:D (SER414) to (ASP456) MYCOBACTERIUM TUBERCULOSIS ADENYLYL CYCLASE RV1900C CHD, IN COMPLEX WITH A SUBSTRATE ANALOG. | CYCLASE HOMOLOGY DOMAIN, CHD, RV1900C, HYDROLASE
1mt5:G (PRO231) to (ARG285) CRYSTAL STRUCTURE OF FATTY ACID AMIDE HYDROLASE | AMIDASE SIGNATURE, HYDROLASE
1mt5:M (PRO231) to (ARG285) CRYSTAL STRUCTURE OF FATTY ACID AMIDE HYDROLASE | AMIDASE SIGNATURE, HYDROLASE
1mt5:N (GLY233) to (ARG285) CRYSTAL STRUCTURE OF FATTY ACID AMIDE HYDROLASE | AMIDASE SIGNATURE, HYDROLASE
5d79:A (SER251) to (ILE307) STRUCTURE OF BBE-LIKE #28 FROM ARABIDOPSIS THALIANA | COVALENT FAD BINDING, BERBERINE BRIDGE ENZYME LIKE, PLANT ENZYME, OXIDOREDUCTASE
3krj:A (VAL613) to (GLU664) CFMS TYROSINE KINASE IN COMPLEX WITH 4-CYANO-1H-IMIDAZOLE-2-CARBOXYLIC ACID (2-CYCLOHEX-1-ENYL-4-PIPERIDIN-4-YL-PHENYL)-AMIDE | KINASE, INHIBITOR, CHIMERA, ATP-BINDING, DISULFIDE BOND, GLYCOPROTEIN, IMMUNOGLOBULIN DOMAIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1mw0:A (TYR209) to (TRP247) AMYLOSUCRASE MUTANT E328Q CO-CRYSTALLIZED WITH MALTOHEPTAOSE THEN SOAKED WITH MALTOHEPTAOSE. | (BETA-ALPHA)8 BARREL, PROTEIN-SUGAR COMPLEX, TRANSFERASE
1mw1:A (TYR209) to (TRP247) AMYLOSUCRASE SOAKED WITH 14MM SUCROSE. | (BETA-ALPHA)8 BARREL, PROTEIN-SUGAR COMPLEX, TRANSFERASE
1mw2:A (TYR209) to (TRP247) AMYLOSUCRASE SOAKED WITH 100MM SUCROSE | (BETA-ALPHA)8 BARREL, PROTEIN-SUGAR COMPLEX, TRANSFERASE
1yhw:A (GLY293) to (GLU345) CRYSTAL STRUCTURE OF PAK1 KINASE DOMAIN WITH ONE POINT MUTATIONS (K299R) | KINASE; ACTIVE CONFORMATION; ACTIVATION LOOP; ATP BINDING SITE, SIGNALING PROTEIN, TRANSFERASE
1yi6:B (VAL292) to (GLU339) C-TERM TAIL SEGMENT OF HUMAN TYROSINE KINASE (258-533) | SRC, TYROSINE KINASE, PHOSPHORYLATION, REGULATION, SH2, SH3, TRANSFERASE
1yk3:A (ILE165) to (GLU204) CRYSTAL STRUCTURE OF RV1347C FROM MYCOBACTERIUM TUBERCULOSIS | ACYLTRANSFERASE, GCN5-RELATED FOLD, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
1yk3:C (ILE165) to (GLU204) CRYSTAL STRUCTURE OF RV1347C FROM MYCOBACTERIUM TUBERCULOSIS | ACYLTRANSFERASE, GCN5-RELATED FOLD, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
1yk3:H (ILE165) to (GLU204) CRYSTAL STRUCTURE OF RV1347C FROM MYCOBACTERIUM TUBERCULOSIS | ACYLTRANSFERASE, GCN5-RELATED FOLD, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
1n0v:D (VAL488) to (THR533) CRYSTAL STRUCTURE OF ELONGATION FACTOR 2 | G-PROTEIN CIS-PROLINE, TRANSLATION
5de2:A (VAL58) to (ALA116) STRUCTURAL MECHANISM OF NEK7 ACTIVATION BY NEK9-INDUCED DIMERISATION | PROTEIN KINASE, MITOSIS, PROTEIN-PROTEIN INTERACTION, TRANSFERASE
3ac2:A (HIS267) to (GLU317) CRYSTAL STRUCTURE OF PYRAZOLO PYRIMIDINE DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3ac3:A (VAL270) to (GLU317) CRYSTAL STRUCTURE OF PYRAZOLO PYRIMIDINE DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3ac5:A (VAL270) to (GLU317) CRYSTAL STRUCTURE OF TRIAZOLO PYRIMIDINE DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3ac8:A (HIS267) to (GLU317) CRYSTAL STRUCTURE OF PYRAZOLO PYRIMIDINE DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, ALTERNATIVE SPLICING, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3ad4:A (HIS267) to (GLU317) CRYSTAL STRUCTURE OF METHOXY BENZOFURAN DERIVATIVE BOUND TO THE KINASE DOMAIN OF HUMAN LCK, (AUTO-PHOSPHORYLATED ON TYR394) | TYROSINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, SIGNAL TRANSDUCTION, KINASE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
1yue:A (THR270) to (ILE331) BACTERIOPHAGE T4 CAPSID VERTEX PROTEIN GP24 | GP24, BACTERIOPHAGE T4, CAPSID PROTEIN, VERTEX, BACTERIOPHAGE, VIRUS, HK97, MAD, VIRAL PROTEIN
1yxu:B (ALA65) to (GLU121) CRYSTAL STRUCTURE OF KINASE PIM1 IN COMPLEX WITH AMP | SER/THR PROTEIN KINASE, TRANSFERASE
1z7m:A (SER46) to (LEU81) ATP PHOSPHORIBOSYL TRANSFERASE (HISZG ATP-PRTASE) FROM LACTOCOCCUS LACTIS | ATP-PRT, HISTIDINE BIOSYNTHESIS, TRANSFERASE, HISZG, ALLOSTERIC, EVOLUTION
1z7m:C (SER46) to (LEU81) ATP PHOSPHORIBOSYL TRANSFERASE (HISZG ATP-PRTASE) FROM LACTOCOCCUS LACTIS | ATP-PRT, HISTIDINE BIOSYNTHESIS, TRANSFERASE, HISZG, ALLOSTERIC, EVOLUTION
3akj:A (GLU32) to (LYS88) CRYSTAL STRUCTURE OF A HELICOBACTER PYLORI PROINFLAMMATORY KINASE CTKA | PROTEIN KINASE, TRANSFERASE
3akk:A (GLU32) to (LYS88) CRYSTAL STRUCTURE OF A HELICOBACTER PYLORI PROINFLAMMATORY KINASE CTKA | PROTEIN KINASE, TRANSFERASE
5dql:C (THR235) to (LYS262) CRYSTAL STRUCTURE OF 2-VINYL GLYOXYLATE MODIFIED ISOCITRATE LYASE FROM MYCOBACTERIUM TUBERCULOSIS | LYASE-LYASE INHIBITOR COMPLEX
5dql:D (THR235) to (LYS262) CRYSTAL STRUCTURE OF 2-VINYL GLYOXYLATE MODIFIED ISOCITRATE LYASE FROM MYCOBACTERIUM TUBERCULOSIS | LYASE-LYASE INHIBITOR COMPLEX
3lj6:B (PRO231) to (ARG285) 3D-CRYSTAL STRUCTURE OF HUMANIZED-RAT FATTY ACID AMIDE HYDROLASE (FAAH) CONJUGATED WITH THE DRUG-LIKE UREA INHIBITOR PF-3845 AT 2.42A RESOLUTION | PROTEIN-INHIBITOR COMPLEX, FAAH, FATTY ACID AMIDE HYDROLASE, UREA, INHIBITOR, COVALENT, ENDOPLASMIC RETICULUM, GOLGI APPARATUS, MEMBRANE, TRANSMEMBRANE, HYDROLASE
3lj7:A (PRO231) to (ALA284) 3D-CRYSTAL STRUCTURE OF HUMANIZED-RAT FATTY ACID AMIDE HYDROLASE (FAAH) CONJUGATED WITH CARBAMATE INHIBITOR URB597 | PROTEIN-INHIBITOR COMPLEX, FAAH, FATTY ACID AMIDE HYDROLASE, CARBAMATE, INHIBITOR, COVALENT, ENDOPLASMIC RETICULUM, GOLGI APPARATUS, MEMBRANE, TRANSMEMBRANE, HYDROLASE
4pyn:A (VAL208) to (ILE254) HUMANIZED RAT COMT IN COMPLEX WITH SAH | METHYLTRANSFERASE, NEUROTRANSMITTER DEGRADATION, ALTERNATIVE INITIATION, CATECHOLAMINE METABOLISM, CELL MEMBRANE, MAGNESIUM, MEMBRANE, METAL-BINDING, PHOSPHOPROTEIN, SIGNAL-ANCHOR, TRANSMEMBRANE ANCHOR, ENZYME MECHANISM, CONFORMATIONAL CHANGE, TRANSFERASE
5dwr:A (ALA65) to (GLU121) IDENTIFICATION OF N-(4-((1R,3S,5S)-3-AMINO-5-METHYLCYCLOHEXYL)PYRIDIN- 3-YL)-6-(2,6-DIFLUOROPHENYL)-5-FLUOROPICOLINAMIDE (PIM447), A POTENT AND SELECTIVE PROVIRAL INSERTION SITE OF MOLONEY MURINE LEUKEMIA (PIM) 1,2 AND 3 KINASE INHIBITOR IN CLINICAL TRIALS FOR HEMATOLOGICAL MALIGNANCIES | PIM1, MOLONEY MURINE LEUKEMIA, PIM447, KINASE INHIBITOR, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4q15:A (LEU318) to (ILE356) CRYSTAL STRUCTURE OF PROLYL-TRNA SYNTHETASE (PRORS, PROLINE--TRNA LIGASE) FROM PLASMODIUM FALCIPARUM IN COMPLEX WITH HALOFUGINONE AND AMPPNP IN SPACE GROUP P212121 AT 2.35 A | STRUCTURAL GENOMICS, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, SSGCID, PROLYL-TRNA SYNTHETASE, LIGASE
1zm2:A (VAL488) to (THR533) STRUCTURE OF ADP-RIBOSYLATED EEF2 IN COMPLEX WITH CATALYTIC FRAGMENT OF ETA | ELONGATION FACTOR, TOXIN, ADP-RIBOSYLATION, BIOSYNTHETIC PROTEIN/TRANSFERASE COMPLEX
1zm3:A (VAL488) to (THR533) STRUCTURE OF THE APO EEF2-ETA COMPLEX | ELONGATION FACTOR, TOXIN, ADP-RIBOSYLATION, BIOSYNTHETIC PROTEIN/TRANSFERASE COMPLEX
4at4:A (ILE583) to (GLU634) CRYSTAL STRUCTURE OF TRKB KINASE DOMAIN IN COMPLEX WITH EX429 | TRANSFERASE
1zm9:A (VAL488) to (THR533) STRUCTURE OF EEF2-ETA IN COMPLEX WITH PJ34 | ELONGATION FACTOR, TOXIN, ADP-RIBOSYLATION, BIOSYNTHETIC PROTEIN/TRANSFERASE COMPLEX
1zmv:B (LYS77) to (GLY134) CATALYTIC AND UBIQUTIN-ASSOCIATED DOMAINS OF MARK2/PAR-1: K82R MUTANT | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN,TRANSFERASE
5e1s:A (ALA1023) to (GLU1077) THE CRYSTAL STRUCTURE OF INSR TYROSINE KINASE IN COMPLEX WITH THE INHIBITOR BI 885578 | KINASE, INSR, IGF-1R, INHIBITOR, TRANSFERASE
1zxe:C (ARG623) to (GLU792) CRYSTAL STRUCTURE OF EIF2ALPHA PROTEIN KINASE GCN2: D835N INACTIVATING MUTANT IN APO FORM | TRANSLATION REGULATOR, PROTEIN KINASE, SIGNAL TRANSDUCTION, AMINO- ACID STARVATION, STARVATION STRESS RESPONSE, EIF2ALPHA KINASE, TRANSFERASE
1zy4:B (SER622) to (ASN793) CRYSTAL STRUCTURE OF EIF2ALPHA PROTEIN KINASE GCN2: R794G HYPERACTIVATING MUTANT IN APO FORM. | TRANSLATION REGULATOR, PROTEIN KINASE, SIGNAL TRANSDUCTION, AMINO- ACID STARVATION, STARVATION STRESS RESPONSE, EIF2ALPHA KINASE, TRANSFERASE
4ays:A (PHE198) to (THR239) THE STRUCTURE OF AMYLOSUCRASE FROM D. RADIODURANS | TRANSFERASE, GLUCAN SYNTHESIS, GH-13
4azw:A (TYR249) to (PRO312) CRYSTAL STRUCTURE OF MONOMERIC WBDD. | TRANSFERASE, METHYLTRANSFERASE
4qiw:D (THR157) to (THR192) CRYSTAL STRUCTURE OF EURYARCHAEAL RNA POLYMERASE FROM THERMOCOCCUS KODAKARENSIS | TRANSCRIPTION, DNA-DIRECTED RNA POLYMERASE
4qiw:O (THR157) to (THR192) CRYSTAL STRUCTURE OF EURYARCHAEAL RNA POLYMERASE FROM THERMOCOCCUS KODAKARENSIS | TRANSCRIPTION, DNA-DIRECTED RNA POLYMERASE
4qjv:A (THR157) to (THR192) THE X-RAY CRYSTAL STRUCTURE OF RPO3/RPO11 HETERODIMER OF EURYARCHAEAL RNA POLYMERASE FROM THERMOCOCCUS KODAKARENSIS | TRANSCRIPTION, RNA POLYMERASE, TRANSFERASE
3mcu:D (LYS122) to (ALA169) CRYSTAL STRUCTURE OF THE DIPICOLINATE SYNTHASE CHAIN B FROM BACILLUS CEREUS. NORTHEAST STRUCTURAL GENOMICS CONSORTIUM TARGET BCR215. | NESG, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, OXIDOREDUCTASE
3b78:A (VAL488) to (THR533) STRUCTURE OF THE EEF2-EXOA(R551H)-NAD+ COMPLEX | ELONGATION FACTOR, TOXIN, ADP-RIBOSYLATION, TOXIN-SUBSTRATE COMPLEX, CYTOPLASM, GTP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTEIN BIOSYNTHESIS, RNA-BINDING, RRNA- BINDING, GLYCOSYLTRANSFERASE, NAD, TRANSFERASE, BIOSYNTHETIC PROTEIN/TRANSFERASE COMPLEX
4qmu:A (LYS48) to (GLU100) MST3 IN COMPLEX WITH JNJ-7706621, 4-({5-AMINO-1-[(2,6-DIFLUOROPHENYL) CARBONYL]-1H-1,2,4-TRIAZOL-3-YL}AMINO)BENZENESULFONAMIDE | PROTEIN KINASE, MST3, STK24, STERILE 20-LIKE KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qmy:A (LYS48) to (GLY104) MST3 IN COMPLEX WITH STAUROSPORINE | PROTEIN KINASE, MST3, STK24, STERILE 20-LIKE KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qq5:A (VAL505) to (GLU556) CRYSTAL STRUCTURE OF FGF RECEPTOR (FGFR) 4 KINASE HARBORING THE V550L GATE-KEEPER MUTATION IN COMPLEX WITH FIIN-2, AN IRREVERSIBLE TYROSINE KINASE INHIBITOR CAPABLE OF OVERCOMING FGFR KINASE GATE-KEEPER MUTATIONS | KINASE DOMAIN FOLD, CELL SIGNALING, PHOSPHOTRANSFERASE, PLASMAMEMBRANE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ms9:A (VAL268) to (GLU316) ABL KINASE IN COMPLEX WITH IMATINIB AND A FRAGMENT (FRAG1) IN THE MYRISTATE POCKET | KINASE, FRAGMENT-BASED SCREENING, FBS, TRANSFERASE, TRANSFERASE- TRANSFERASE REGULATOR COMPLEX
3bkt:A (GLY52) to (ILE98) COPPER-BOUND C-TERMINAL DOMAIN OF NIKR | NIKR, NICKEL REGULATORY PROTEIN, TRANSCRIPTION FACTOR, BETA SANDWICH, DNA-BINDING, METAL-BINDING, REPRESSOR, TRANSCRIPTION REGULATION, METAL BINDING PROTEIN
3my0:K (VAL226) to (HIS278) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3my0:S (VAL226) to (HIS278) CRYSTAL STRUCTURE OF THE ACVRL1 (ALK1) KINASE DOMAIN BOUND TO LDN- 193189 | PROTEIN KINASE, SERINE/THREONINE-PROTEIN KINASE RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
5f9z:A (ILE259) to (ILE297) CRYSTAL STRUCTURE OF PROLYL-TRNA SYNTHETASE FROM CRYPTOSPORIDIUM PARVUM COMPLEXED WITH HALOFUGINONE AND AMPPNP | SSGCID, PROLYL-TRNA LIGASE, CRYPTOSPORIDIUM PARVUM, ATP BINDING, AMINOACYLATION, HALOFUGINONE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, PRORS, LIGASE
3c14:B (ASP1037) to (THR1077) COMPLEX OF GS-ALPHA WITH THE CATALYTIC DOMAINS OF MAMMALIAN ADENYLYL CYCLASE: COMPLEX WITH PYROPHOSPHATE AND CA | ADENYLYL CYCLASE, GSALPHA, PYROPHOSPHATE, CAMP BIOSYNTHESIS, GLYCOPROTEIN, LYASE, MAGNESIUM, MEMBRANE, METAL-BINDING, PHOSPHOPROTEIN, TRANSMEMBRANE, GTP-BINDING, LIPOPROTEIN, NUCLEOTIDE- BINDING, PALMITATE, TRANSDUCER, LYASE-LYASE INHIBITOR COMPLEX
3c15:B (ASP1037) to (THR1077) COMPLEX OF GS-ALPHA WITH THE CATALYTIC DOMAINS OF MAMMALIAN ADENYLYL CYCLASE: COMPLEX WITH PYROPHOSPHATE AND MG | ADENYLYL CYCLASE, GSALPHA, PYROPHOSPHATE, MAGNESIUM, ALTERNATIVE SPLICING, CAMP BIOSYNTHESIS, GLYCOPROTEIN, LYASE, MEMBRANE, METAL-BINDING, PHOSPHOPROTEIN, TRANSMEMBRANE, GTP-BINDING, LIPOPROTEIN, NUCLEOTIDE-BINDING, PALMITATE, TRANSDUCER, LYASE/LYASE INHIBITOR COMPLEX
4r2n:A (ASN297) to (THR332) CRYSTAL STRUCTURE OF RV3772 IN COMPLEX WITH ITS SUBSTRATE | AMINOTRANSFERASE, TRANSFERASE
4r2n:C (ASN297) to (THR332) CRYSTAL STRUCTURE OF RV3772 IN COMPLEX WITH ITS SUBSTRATE | AMINOTRANSFERASE, TRANSFERASE
4r2n:D (ASN297) to (THR332) CRYSTAL STRUCTURE OF RV3772 IN COMPLEX WITH ITS SUBSTRATE | AMINOTRANSFERASE, TRANSFERASE
4r5z:A (ASN297) to (THR332) CRYSTAL STRUCTURE OF RV3772 ENCODED AMINOTRANSFERASE | AMINOTRANSFERASE, TRANSFERASE
4r5z:B (ASN297) to (THR332) CRYSTAL STRUCTURE OF RV3772 ENCODED AMINOTRANSFERASE | AMINOTRANSFERASE, TRANSFERASE
4r5z:C (ASN297) to (THR332) CRYSTAL STRUCTURE OF RV3772 ENCODED AMINOTRANSFERASE | AMINOTRANSFERASE, TRANSFERASE
4r6v:A (VAL500) to (GLU551) CRYSTAL STRUCTURE OF FGF RECEPTOR (FGFR) 4 KINASE HARBORING THE V550L GATE-KEEPER MUTATION IN COMPLEX WITH FIIN-3, AN IRREVERSIBLE TYROSINE KINASE INHIBITOR CAPABLE OF OVERCOMING FGFR KINASE GATE-KEEPER MUTATIONS | KINASE DOMAIN FOLD, CELL SIGNALING, PHOSPHOTRANSFERASE, PLASMAMEMBRANE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4r77:B (LYS40) to (SER93) CRYSTAL STRUCTURE OF CHOLINE KINASE LICA FROM STREPTOCOCCUS PNEUMONIAE | A PROTEIN KINASE-LIKE FOLD, CHOLINE/ETHANOLAMINE KINASE, ATP/CHOLINE BINDING, TRANSFERASE
5fir:I (THR704) to (ASP785) CRYSTAL STRUCTURE OF C. ELEGANS XRN2 IN COMPLEX WITH THE XRN2-BINDING DOMAIN OF PAXT-1 | HYDROLASE, 5'-3' EXORIBONUCLEASE, MIRNA TURNOVER
3cb4:A (GLN294) to (GLY341) THE CRYSTAL STRUCTURE OF LEPA | GTPASE, OB-FOLD, GTP-BINDING, MEMBRANE, NUCLEOTIDE-BINDING, TRANSLATION
3cb4:C (GLN294) to (GLY341) THE CRYSTAL STRUCTURE OF LEPA | GTPASE, OB-FOLD, GTP-BINDING, MEMBRANE, NUCLEOTIDE-BINDING, TRANSLATION
3cb4:F (GLN294) to (GLY341) THE CRYSTAL STRUCTURE OF LEPA | GTPASE, OB-FOLD, GTP-BINDING, MEMBRANE, NUCLEOTIDE-BINDING, TRANSLATION
5foq:B (ARG424) to (ARG522) ACETYLCHOLINESTERASE IN COMPLEX WITH C7653 | HYDROLASE, SIGNALING PROTEIN, QUANTUM CHEMISTRY, DENSITY FUNCTIONAL THEORY, DRUG DESIGN
4cm0:A (VAL425) to (TYR462) CRYSTAL STRUCTURE OF HUMAN SOLUBLE ADENYLYL CYCLASE WITH ALPHA,BETA-METHYLENEADENOSINE-5'-TRIPHOSPHATE SOAKED WITH BICARBONATE | LYASE, BICARBONATE, ACTIVATOR
3cze:A (HIS203) to (THR243) CRYSTAL STRUCTURE ANALYSIS OF SUCROSE HYDROLASE (SUH)- TRIS COMPLEX | (ALPHA/BETA)8-BARREL, HYDROLASE
3czk:A (HIS203) to (THR243) CRYSTAL STRUCTURE ANALYSIS OF SUCROSE HYDROLASE(SUH) E322Q- SUCROSE COMPLEX | (ALPHA/BETA)8-BARREL, HYDROLASE
3czl:A (HIS203) to (THR243) CRYSTAL STRUCTURE ANALYSIS OF SUCROSE HYDROLASE(SUH) E322Q- GLUCOSE COMPLEX | (ALPHA/BETA)8-BARREL, HYDROLASE
3d2j:A (VAL245) to (THR293) STRUCTURE OF BERBERINE BRIDGE ENZYME FROM ESCHSCHOLZIA CALIFORNICA, TETRAGONAL CRYSTAL FORM | BI-COVALENT FLAVINYLATION, N-GLYCOSYLATION, ALAKLOID BIOSYNTHESIS, P- CRESOL METHYLHYDROXYLASE SUPERFAMILY, OXIDOREDUCTASE
3d2s:A (ASP180) to (CYS221) CRYSTAL STRUCTURE OF MBNL1 TANDEM ZINC FINGER 3 AND 4 DOMAIN IN COMPLEX WITH CGCUGU RNA | TANDEM ZINC FINGER DOMAIN, RNA, METAL-BINDING, NUCLEUS, RNA-BINDING, ZINC-FINGER, METAL BINDING PROTEIN-RNA COMPLEX
3d2s:C (ASP180) to (CYS221) CRYSTAL STRUCTURE OF MBNL1 TANDEM ZINC FINGER 3 AND 4 DOMAIN IN COMPLEX WITH CGCUGU RNA | TANDEM ZINC FINGER DOMAIN, RNA, METAL-BINDING, NUCLEUS, RNA-BINDING, ZINC-FINGER, METAL BINDING PROTEIN-RNA COMPLEX
4ct2:A (LYS111) to (SER160) HUMAN PDK1-PKCZETA KINASE CHIMERA | TRANSFERASE, ALLOSTERIC REGULATION, ALLOSTERIC SITE, PHOSPHORYLATION, AGC PROTEIN KINASE, CHIMERIC PROTEIN
3d5v:A (LYS62) to (GLU117) CRYSTAL STRUCTURE OF AN ACTIVATED (THR->ASP) POLO-LIKE KINASE 1 (PLK1) CATALYTIC DOMAIN. | POLO-LIKE KINASE 1, PLK1, CATALYTIC DOMAIN, SMALL-MOLECULE INHIBITOR, KINASE, TRANSFERASE
3d5w:A (LYS62) to (GLU117) CRYSTAL STRUCTURE OF A PHOSPHORYLATED POLO-LIKE KINASE 1 (PLK1) CATALYTIC DOMAIN IN COMPLEX WITH ADP. | POLO-LIKE KINASE 1, PLK1, CATALYTIC DOMAIN, SMALL-MOLECULE INHIBITOR, KINASE, TRANSFERASE
3d5x:A (LYS62) to (GLU117) CRYSTAL STRUCTURE OF AN ACTIVATED (THR->ASP) POLO-LIKE KINASE 1 (PLK1) CATALYTIC DOMAIN IN COMPLEX WITH WORTMANNIN. | POLO-LIKE KINASE 1, PLK1, CATALYTIC DOMAIN, SMALL-MOLECULE INHIBITOR, KINASE, TRANSFERASE
3d66:A (SER3) to (ASN51) CRYSTAL STRUCTURE OF THROMBIN-ACTIVATABLE FIBRINOLYSIS INHIBITOR (TAFI) | ALPHA/BETA HYDROLASE FOLD, CARBOXYPEPTIDASE, GLYCOPROTEIN, METAL- BINDING, METALLOPROTEASE, PROTEASE, SECRETED, ZYMOGEN, HYDROLASE
5gep:A (ASP354) to (ALA401) SULFITE REDUCTASE HEMOPROTEIN CARBON MONOXIDE COMPLEX REDUCED WITH CRII EDTA | OXIDOREDUCTASE, SIROHEME FEII, [4FE-4S] +1, CARBON MONOXIDE COMPLEX, INHIBITOR
3dgv:A (ARG3) to (ASN51) CRYSTAL STRUCTURE OF THROMBIN ACTIVATABLE FIBRINOLYSIS INHIBITOR (TAFI) | BLOOD COAGULATION, FIBRINOLYSIS, CARBOXYPEPTIDASE, PROTEIN STABILITY, GLYCOPROTEIN, HYDROLASE, METAL-BINDING, METALLOPROTEASE, PROTEASE, SECRETED, ZYMOGEN
3dgv:B (ARG3) to (ASN51) CRYSTAL STRUCTURE OF THROMBIN ACTIVATABLE FIBRINOLYSIS INHIBITOR (TAFI) | BLOOD COAGULATION, FIBRINOLYSIS, CARBOXYPEPTIDASE, PROTEIN STABILITY, GLYCOPROTEIN, HYDROLASE, METAL-BINDING, METALLOPROTEASE, PROTEASE, SECRETED, ZYMOGEN
4ttv:A (ASN376) to (LEU408) CRYSTAL STRUCTURE OF HUMAN THRRS COMPLEXING WITH A BIOENGINEERED MACROLIDE BC194 | TRNA, SYNTHETASE, INHIBITOR, MACROLIDE, LIGASE-ANTIBIOTIC COMPLEX
4ttv:C (ASN376) to (LEU408) CRYSTAL STRUCTURE OF HUMAN THRRS COMPLEXING WITH A BIOENGINEERED MACROLIDE BC194 | TRNA, SYNTHETASE, INHIBITOR, MACROLIDE, LIGASE-ANTIBIOTIC COMPLEX
4d2w:D (GLY34) to (GLU87) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN
4twp:A (VAL268) to (GLU316) THE CRYSTAL STRUCTURE OF HUMAN ABL1 T315I GATEKEEPER MUTANT KINASE DOMAIN IN COMPLEX WITH AXITINIB | GATEKEEPER MUTANT KINASE DOMAIN DFGIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3dnv:A (ILE179) to (GLU234) MDT PROTEIN | PERSISTENCE, MDT, DNA-BINDING, REPRESSOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSCRIPTION/DNA COMPLEX
3dnt:A (HIS178) to (GLU234) STRUCTURES OF MDT PROTEINS | MDT, PERSISTENCE, MULTIDRUG RESISTANCE, TOLERANCE, TRANSFERASE
3ooi:A (GLU123) to (ALA158) CRYSTAL STRUCTURE OF HUMAN HISTONE-LYSINE N-METHYLTRANSFERASE NSD1 SET DOMAIN IN COMPLEX WITH S-ADENOSYL-L-METHIONINE | SET DOMAIN, HISTONE-LYSINE N-METHYLTRANSFERASE, S-ADENOSYL-L- METHIONINE, TRANSFERASE
5h37:B (GLU62) to (LYS123) CRYO-EM STRUCTURE OF ZIKA VIRUS COMPLEXED WITH FAB C10 AT PH 8.0 | IGG NAG, VIRUS-IMMUNE SYSTEM COMPLEX
3dqw:B (VAL292) to (GLU339) C-SRC KINASE DOMAIN THR338ILE MUTANT IN COMPLEX WITH ATPGS | SRC, KINASE, ACTIVE, GATEKEEPER, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3dqw:D (VAL292) to (GLU339) C-SRC KINASE DOMAIN THR338ILE MUTANT IN COMPLEX WITH ATPGS | SRC, KINASE, ACTIVE, GATEKEEPER, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3dqx:A (VAL292) to (GLU339) CHICKEN C-SRC KINASE DOMAIN IN COMPLEX WITH ATPGS | SRC, KINASE, ACTIVE, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
3dul:B (ASN167) to (LYS222) CRYSTAL STRUCTURE ANALYSIS OF THE O-METHYLTRANSFERASE FROM BACILLUS CEREUS | ALTERNATING OF ALPHA AND BETA, METHYLTRANSFERASE, TRANSFERASE
4dfu:A (PHE43) to (THR96) INHIBITION OF AN ANTIBIOTIC RESISTANCE ENZYME: CRYSTAL STRUCTURE OF AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(2")-ID/APH(2")-IVA IN COMPLEX WITH KANAMYCIN INHIBITED WITH QUERCETIN | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, EUKARYOTIC PROTEIN KINASE-LIKE FOLD, TRANSFERASE- ANTIBIOTIC-INHIBITOR COMPLEX, AMINOGLYCOSIDE PHOSPHOTRANSFERASE, KINASE, TRANSFERASE, AMINOGLYCOSIDES, KANAMYCIN, FLAVANOIDS, QUERCETIN, INTRACELLULAR, ANTIBOTIC, TRANSFERASE-ANTIBOTIC-INHIBITOR COMPLEX
5hlp:A (GLY79) to (LEU130) X-RAY CRYSTAL STRUCTURE OF GSK3B IN COMPLEX WITH BRD3937 | PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4do3:A (PRO231) to (ARG285) STRUCTURE OF FAAH WITH A NON-STEROIDAL ANTI-INFLAMMATORY DRUG | AMIDASE, HYDROLASE, ANANDAMIDE, NSAID, DRUG, COX, INHIBITOR, INFLAMMATION, PAIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4do3:B (GLY233) to (ARG285) STRUCTURE OF FAAH WITH A NON-STEROIDAL ANTI-INFLAMMATORY DRUG | AMIDASE, HYDROLASE, ANANDAMIDE, NSAID, DRUG, COX, INHIBITOR, INFLAMMATION, PAIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5ht0:A (GLY57) to (GLY122) CRYSTAL STRUCTURE OF AN ANTIBIOTIC_NAT FAMILY AMINOGLYCOSIDE ACETYLTRANSFERASE HMB0038 FROM AN UNCULTURED SOIL METAGENOMIC SAMPLE IN COMPLEX WITH COENZYME A | ANTIBIOTIC_NAT FAMILY, ACETYLTRANSFERASE, AMINOGLYCOSIDE, ANTIBIOTIC RESISTANCE, METAGENOME, SOIL, COENZYME A, CSGID, TRANSFERASE, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES
5ht0:C (ALA56) to (GLY122) CRYSTAL STRUCTURE OF AN ANTIBIOTIC_NAT FAMILY AMINOGLYCOSIDE ACETYLTRANSFERASE HMB0038 FROM AN UNCULTURED SOIL METAGENOMIC SAMPLE IN COMPLEX WITH COENZYME A | ANTIBIOTIC_NAT FAMILY, ACETYLTRANSFERASE, AMINOGLYCOSIDE, ANTIBIOTIC RESISTANCE, METAGENOME, SOIL, COENZYME A, CSGID, TRANSFERASE, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES
5ht0:D (ALA56) to (GLY122) CRYSTAL STRUCTURE OF AN ANTIBIOTIC_NAT FAMILY AMINOGLYCOSIDE ACETYLTRANSFERASE HMB0038 FROM AN UNCULTURED SOIL METAGENOMIC SAMPLE IN COMPLEX WITH COENZYME A | ANTIBIOTIC_NAT FAMILY, ACETYLTRANSFERASE, AMINOGLYCOSIDE, ANTIBIOTIC RESISTANCE, METAGENOME, SOIL, COENZYME A, CSGID, TRANSFERASE, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES
5ht0:E (ALA56) to (GLY122) CRYSTAL STRUCTURE OF AN ANTIBIOTIC_NAT FAMILY AMINOGLYCOSIDE ACETYLTRANSFERASE HMB0038 FROM AN UNCULTURED SOIL METAGENOMIC SAMPLE IN COMPLEX WITH COENZYME A | ANTIBIOTIC_NAT FAMILY, ACETYLTRANSFERASE, AMINOGLYCOSIDE, ANTIBIOTIC RESISTANCE, METAGENOME, SOIL, COENZYME A, CSGID, TRANSFERASE, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES
5hvf:A (SER3) to (PHE49) CRYSTAL STRUCTURE OF THROMBIN-ACTIVATABLE FIBRINOLYSIS INHIBITOR IN COMPLEX WITH AN INHIBITORY NANOBODY (VHH-I83) | PROCARBOXYPEPTIDASE U, THROMBIN-ACTIVATABLE FIBRINOLYSIS INHIBITOR, TAFI, PROCARBOXYPEPTIDASE R, PLASMA PROCARBOXYPEPTIDASE B, NANOBODY, ANTIBODY FRAGMENT, PROTEIN COMPLEX, HYDROLASE/HYDROLASE INHIBITOR, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5hvh:A (SER3) to (PHE49) CRYSTAL STRUCTURE OF THROMBIN-ACTIVATABLE FIBRINOLYSIS INHIBITOR IN COMPLEX WITH TWO INHIBITORY NANOBODIES | PROCARBOXYPEPTIDASE U, THROMBIN-ACTIVATABLE FIBRINOLYSIS INHIBITOR, TAFI, PROCARBOXYPEPTIDASE R, PLASMA PROCARBOXYPEPTIDASE B, NANOBODY, ANTIBODY FRAGMENT, PROTEIN COMPLEX, HYDROLASE/HYDROLASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5hvk:A (MET365) to (GLU414) CRYSTAL STRUCTURE OF LIMK1 MUTANT D460N IN COMPLEX WITH FULL-LENGTH COFILIN-1 | KINASE SUBSTRATE ACTIN-REMODELING, TRANSFERASE
5hvk:C (MET365) to (GLU414) CRYSTAL STRUCTURE OF LIMK1 MUTANT D460N IN COMPLEX WITH FULL-LENGTH COFILIN-1 | KINASE SUBSTRATE ACTIN-REMODELING, TRANSFERASE
5hyn:F (SER639) to (ALA677) STRUCTURE OF HUMAN POLYCOMB REPRESSIVE COMPLEX 2 (PRC2) WITH ONCOGENIC HISTONE H3K27M PEPTIDE | CHROMATIN MODIFICATION COMPLEX, TRANSFERASE
4uf4:A (GLY22) to (ARG66) CRYSTAL STRUCTURE OF THE HUMAN CARBOXYPEPTIDASE A1 IN COMPLEX WITH A THIIRANE MECHANISM-BASED INHIBITOR | HYDROLASE
4uf4:B (GLY22) to (ARG66) CRYSTAL STRUCTURE OF THE HUMAN CARBOXYPEPTIDASE A1 IN COMPLEX WITH A THIIRANE MECHANISM-BASED INHIBITOR | HYDROLASE
3peh:A (HIS279) to (VAL323) CRYSTAL STRUCTURE OF THE N-TERMINAL DOMAIN OF AN HSP90 FROM PLASMODIUM FALCIPARUM, PFL1070C IN THE PRESENCE OF A THIENOPYRIMIDINE DERIVATIVE | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, HEAT SHOCK PROTEIN, CHAPERONE, ATP BINDING
4ump:A (GLU35) to (GLU87) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE
4ump:C (GLU35) to (VAL85) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE
4ump:D (GLU35) to (GLU87) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE
3pr0:B (PRO231) to (ARG285) CRYSTAL STRUCTURE OF A COVALENTLY BOUND ALPHA-KETOHETEROCYCLE INHIBITOR (PHENHEXYL/OXADIAZOLE/PYRIDINE) TO A HUMANIZED VARIANT OF FATTY ACID AMIDE HYDROLASE | PROTEIN-INHIBITOR COMPLEX, FAAH, OXADIAZOLE, ALPHA-KETOHETEROCYCLE, ENDOCANNABINOID DEGRADATION, MEMBRANE PROTEIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5ih8:A (GLU35) to (GLU87) MELK IN COMPLEX WITH NVS-MELK1 | KINASE UBA DOMAIN INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ih9:A (GLU35) to (GLU87) MELK IN COMPLEX WITH NVS-MELK8A | KINASE UBA DOMAIN INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ecc:A (PRO3) to (GLY74) CHIMERIC GST CONTAINING INSERTS OF KININOGEN PEPTIDES | GST, DOMAIN 5 OF HUMAN HIGH MOLECULAR WEIGHT KININOGEN, BIOSYNTHETIC PROTEIN, TRANSFERASE, PROTEIN BINDING
4eo4:A (LEU93) to (LEU128) CRYSTAL STRUCTURE OF THE YEAST MITOCHONDRIAL THREONYL-TRNA SYNTHETASE (MST1) IN COMPLEX WITH SERYL SULFAMOYL ADENYLATE | AMINOACYL-TRNA SYNTHETASE CLASS II, THREONYL-TRNA SYNTHETASE, THREONINE TRNA, MITOCHONDRIA, LIGASE
3q4t:B (VAL216) to (ALA268) CRYSTAL STRUCTURE OF ACTIVIN RECEPTOR TYPE-IIA (ACVR2A) KINASE DOMAIN IN COMPLEX WITH DORSOMORPHIN | STRUCTURAL GENOMICS CONSORTIUM, SGC, PROTEIN KINASE, TRANSFERASE
3q52:A (GLY293) to (GLU345) STRUCTURE OF PHOSPHORYLATED PAK1 KINASE DOMAIN | KINASE DOMAIN, SIGNALLING PATHWAY, TRANSFERASE
3q60:A (LEU257) to (MET337) CRYSTAL STRUCTURE OF VIRULENT ALLELE ROP5B PSEUDOKINASE DOMAIN BOUND TO ATP | PSEUDOKINASE, TOXOPLASMA, TRANSFERASE, 551.M00238, ROP5
4f0f:A (VAL1052) to (GLU1106) CRYSTAL STRUCTURE OF THE ROCO4 KINASE DOMAIN BOUND TO APPCP FROM D. DISCOIDEUM | PROTEIN KINASE, LRRK2, ROCO, KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, SIGNALING PROTEIN
5j0a:B (TYR78) to (TYR117) CRYSTAL STRUCTURE OF PDZ-BINDING KINASE | PROTEIN KINASE, TRANSFERASE
4f78:A (LEU111) to (TYR170) CRYSTAL STRUCTURE OF VANCOMYCIN RESISTANCE D,D-DIPEPTIDASE VANXYG | CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, NIAID, ALPHA+BETA PROTEIN, METALLOPEPTIDASE, HEDGEHOG/DD-PEPTIDASE FOLD, MEROPS M15B SUBFAMILY, ZN2+-DEPENDENT D,D-DIPEPTIDASE, VANCOMYCIN RESISTANCE, D-ALANINE-D-ALANINE, HYDROLASE
3qk5:B (PRO231) to (ARG285) CRYSTAL STRUCTURE OF FATTY ACID AMIDE HYDROLASE WITH SMALL MOLECULE INHIBITOR | PROTEIN-INHIBITOR COMPLEX, FAAH, FATTY-ACID AMIDE HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3qkv:A (PRO231) to (ALA284) CRYSTAL STRUCTURE OF FATTY ACID AMIDE HYDROLASE WITH SMALL MOLECULE COMPOUND | PROTEIN-INHIBITOR COMPLEX, FAAH, FATTY-ACID AMIDE HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3qkv:B (PRO231) to (ARG285) CRYSTAL STRUCTURE OF FATTY ACID AMIDE HYDROLASE WITH SMALL MOLECULE COMPOUND | PROTEIN-INHIBITOR COMPLEX, FAAH, FATTY-ACID AMIDE HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4fif:B (LYS345) to (MET395) CATALYTIC DOMAIN OF HUMAN PAK4 WITH RPKPLVDP PEPTIDE | SERINE/THREONINE-PROTEIN KINASE PAK4, KINASE DOMAIN, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE-PEPTIDE COMPLEX
3r5g:B (GLY370) to (ASP410) CRYSTAL STRUCTURE OF THE ADENYLYL CYCLASE CYAB FROM P. AERUGINOSA | ADENYLYL CYCLASE, LYASE
4flo:A (TYR209) to (TRP247) CRYSTAL STRUCTURE OF AMYLOSUCRASE DOUBLE MUTANT A289P-F290C FROM NEISSERIA POLYSACCHAREA | BETA/ALPHA-BARREL, GLYCOSIDE HYDROLASE, AMYLOSE SYNTHESIS, SUCROSE ISOMERIZATION, GLUCOSYLTRANSFERASE, CARBOHYDRATE, TRANSFERASE
4fls:A (TYR210) to (TRP247) CRYSTAL STRUCTURE OF AMYLOSUCRASE INACTIVE DOUBLE MUTANT F290K-E328Q FROM NEISSERIA POLYSACCHAREA IN COMPLEX WITH SUCROSE. | BETA/ALPHA-BARREL, GLYCOSIDE HYDROLASE, AMYLOSE SYNTHESIS, SUCROSE ISOMERIZATION, GLUCOSYLTRANSFERASE CARBOHYDRATE, TRANSFERASE
5jga:A (VAL60) to (GLY109) CRYSTAL STRUCTURE OF HUMAN TAK1/TAB1 FUSION PROTEIN IN COMPLEX WITH LIGAND 11C | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, TAK1-TAB1 KINASE
4fpi:D (MET1) to (VAL58) CRYSTAL STRUCTURE OF 5-CHLOROMUCONOLACTONE ISOMERASE FROM RHODOCOCCUS OPACUS 1CP | ISOMERASE, INTRAMOLECULAR OXIDOREDUCTASE
4ftr:A (VAL35) to (PHE83) CRYSTAL STRUCTURE OF THE CHK1 | TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gh2:A (VAL35) to (PHE83) CRYSTAL STRUCTURE OF THE CHK1 | TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5kta:A (GLU126) to (LYS164) APO FDHC- A NUCLEOTIDE-LINKED SUGAR GNAT | GNAT, SUGAR, O-ANTIGEN, TRANSFERASE
5lsu:A (GLU1095) to (ALA1130) STRUCTURE OF THE EPIGENETIC ONCOGENE MMSET AND INHIBITION BY N-ALKYL SINEFUNGIN DERIVATIVES | LYSINE METHYLTRANSFERASE MMSET SET DOMAIN, TRANSFERASE
5lsu:B (GLU1095) to (ALA1130) STRUCTURE OF THE EPIGENETIC ONCOGENE MMSET AND INHIBITION BY N-ALKYL SINEFUNGIN DERIVATIVES | LYSINE METHYLTRANSFERASE MMSET SET DOMAIN, TRANSFERASE
5lsz:A (THR1574) to (ALA1617) STRUCTURE OF THE EPIGENETIC ONCOGENE MMSET AND INHIBITION BY N-ALKYL SINEFUNGIN DERIVATIVES | LYSINE METHYLTRANSFERASE SETD2 SET DOMAIN, SETD2#1, TRANSFERASE
5lt6:B (LEU1577) to (ALA1617) STRUCTURE OF THE EPIGENETIC ONCOGENE MMSET AND INHIBITION BY N-ALKYL SINEFUNGIN DERIVATIVES | LYSINE METHYLTRANSFERASE SETD2 SET DOMAIN, SETD2#1, TRANSFERASE
5te0:A (GLY68) to (LEU125) CRYSTAL STRUCTURE OF ADAPTOR PROTEIN 2 ASSOCIATED KINASE (AAK1) IN COMPLEX WITH BIBF 1120 | TRANSFERASE, PROTEIN KINASE DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2ofu:A (VAL270) to (GLU317) X-RAY CRYSTAL STRUCTURE OF 2-AMINOPYRIMIDINE CARBAMATE 43 BOUND TO LCK | LCK, KINASE DOMAIN, TRANSFERASE
2aop:A (ASP354) to (ALA401) SULFITE REDUCTASE: REDUCED WITH CRII EDTA, SIROHEME FEII, [4FE-4S] +1, PHOSPHATE BOUND | OXIDOREDUCTASE, SIROHEME FEII, [4FE-4S] +1, PHOSPHATE COMPLEX, REDUCED, CRII EDTA
1ady:A (ILE43) to (LEU78) HISTIDYL-TRNA SYNTHETASE IN COMPLEX WITH HISTIDYL-ADENYLATE | HISTIDYL-ADENYLATE, AMINO ACID, TRNA SYNTHETASE
1ady:B (ILE43) to (LEU78) HISTIDYL-TRNA SYNTHETASE IN COMPLEX WITH HISTIDYL-ADENYLATE | HISTIDYL-ADENYLATE, AMINO ACID, TRNA SYNTHETASE
1ady:C (ILE43) to (LEU78) HISTIDYL-TRNA SYNTHETASE IN COMPLEX WITH HISTIDYL-ADENYLATE | HISTIDYL-ADENYLATE, AMINO ACID, TRNA SYNTHETASE
1ady:D (ILE43) to (LEU78) HISTIDYL-TRNA SYNTHETASE IN COMPLEX WITH HISTIDYL-ADENYLATE | HISTIDYL-ADENYLATE, AMINO ACID, TRNA SYNTHETASE
1nj8:A (MET60) to (LEU98) CRYSTAL STRUCTURE OF PROLYL-TRNA SYNTHETASE FROM METHANOCALDOCOCCUS JANASCHII | CLASS-II TRNA SYNTHETASE, LIGASE
1nj8:C (MET60) to (LEU98) CRYSTAL STRUCTURE OF PROLYL-TRNA SYNTHETASE FROM METHANOCALDOCOCCUS JANASCHII | CLASS-II TRNA SYNTHETASE, LIGASE
2p8i:B (TRP12) to (THR64) CRYSTAL STRUCTURE OF PUTATIVE DIOXYGENASE (YP_555069.1) FROM BURKHOLDERIA XENOVORANS LB400 AT 1.40 A RESOLUTION | YP_555069.1, PUTATIVE DIOXYGENASE, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, OXIDOREDUCTASE
2p8i:D (TRP12) to (THR64) CRYSTAL STRUCTURE OF PUTATIVE DIOXYGENASE (YP_555069.1) FROM BURKHOLDERIA XENOVORANS LB400 AT 1.40 A RESOLUTION | YP_555069.1, PUTATIVE DIOXYGENASE, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, OXIDOREDUCTASE
2c3l:A (GLU33) to (GLY89) IDENTIFICATION OF A BURIED POCKET FOR POTENT AND SELECTIVE INHIBITION OF CHK1: PREDICTION AND VERIFICATION | DRUG DESIGN, MOLECULAR MODELING, MOLECULAR RECOGNITION, ONCOLOGY, ATP-BINDING, CELL CYCLE, DNA DAMAGE, DNA REPAIR, KINASE, NUCLEAR PROTEIN, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, UBL CONJUGATION
2pvf:A (VAL514) to (LYS569) CRYSTAL STRUCTURE OF TYROSINE PHOSPHORYLATED ACTIVATED FGF RECEPTOR 2 (FGFR2) KINASE DOMAIN IN COMPLEX WITH ATP ANALOG AND SUBSTRATE PEPTIDE | KINASE DOMAIN FOLD CONSISTING OF N- AND C-LOBES, TRANSFERASE
3fw8:A (VAL245) to (THR293) STRUCTURE OF BERBERINE BRIDGE ENZYME, C166A VARIANT | BI-COVALENT FLAVINYLATION, N-GLYCOSYLATION, ALAKLOID BIOSYNTHESIS, OXIDOREDUCTASE, ALKALOID METABOLISM, CYTOPLASMIC VESICLE, FAD, FLAVOPROTEIN, GLYCOPROTEIN
2r0i:A (GLY76) to (GLY134) CRYSTAL STRUCTURE OF A KINASE MARK2/PAR-1 MUTANT | SERINE/THREONINE PROTEIN KINASE; MARK; PAR-1; KIN1; UBA DOMAIN, SIGNALING PROTEIN, TRANSFERASE
2e1r:A (VAL489) to (THR533) STRUCTURE OF EEF2 IN COMPLEX WITH A SORDARIN DERIVATIVE | PROTEIN-LIGAND COMPLEX, G-PROTEIN, TRANSLATION
4yg8:B (PRO44) to (GLY100) CRYSTAL STRUCTURE OF THE CHS5-CHS6 EXOMER CARGO ADAPTOR COMPLEX | FN3, BRCT, TETRATRICOPEPTIDE REPEAT, CARGO ADAPTOR, TRANSPORT PROTEIN
3udb:D (GLU45) to (GLY99) CRYSTAL STRUCTURE OF SNRK2.6 | SNRK2.6, KINASE, ABA SIGNALING PATHWAY, ABI1, TRANSFERASE
3udb:F (GLU45) to (GLY99) CRYSTAL STRUCTURE OF SNRK2.6 | SNRK2.6, KINASE, ABA SIGNALING PATHWAY, ABI1, TRANSFERASE
2v5q:B (LYS76) to (GLU131) CRYSTAL STRUCTURE OF WILD-TYPE PLK-1 KINASE DOMAIN IN COMPLEX WITH A SELECTIVE DARPIN | DESIGN ANKYRIN REPEAT PROTEIN, TRANSFERASE COMPLEX, PHOSPHORYLATION, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, KINASE, NUCLEUS, TRANSFERASE, ATP-BINDING, SERINE/THREONINE PROTEIN KINASE
2v7a:A (VAL268) to (GLU316) CRYSTAL STRUCTURE OF THE T315I ABL MUTANT IN COMPLEX WITH THE INHIBITOR PHA-739358 | KINASE, NUCLEUS, MYRISTATE, CYTOPLASM, MANGANESE, CELL ADHESION, METAL-BINDING, PROTO-ONCOGENE, TYROSINE-PROTEIN KINASE, CHROMOSOMAL REARRANGEMENT, TRANSFERASE, LIPOPROTEIN, POLYMORPHISM, CYTOSKELETON, MAGNESIUM, SH2 DOMAIN, SH3 DOMAIN, ATP-BINDING, NUCLEOTIDE-BINDING, ALTERNATIVE SPLICING, PHOSPHORYLATION, KINASE INHIBITOR, T315I ABL MUTANT
1s3a:A (GLU18) to (ARG68) NMR SOLUTION STRUCTURE OF SUBUNIT B8 FROM HUMAN NADH- UBIQUINONE OXIDOREDUCTASE COMPLEX I (CI-B8) | CI-B8, NDUFA2, COMPLEX I, NMR, OXIDOREDUCTASE
1sou:A (LYS43) to (HIS86) NMR STRUCTURE OF AQUIFEX AEOLICUS 5,10- METHENYLTETRAHYDROFOLATE SYNTHETASE: NORTHEAST STRUCTURAL GENOMICS CONSORTIUM TARGET QR46 | STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, NESG, LIGASE
2wap:A (PRO231) to (ALA284) 3D-CRYSTAL STRUCTURE OF HUMANIZED-RAT FATTY ACID AMIDE HYDROLASE (FAAH) CONJUGATED WITH THE DRUG-LIKE UREA INHIBITOR PF-3845 | FATTY ACID AMIDE HYDROLASE, UREA INHIBITOR, GOLGI APPARATUS, ENDOPLASMIC RETICULUM, ACYL- ENZYME, TRANSMEMBRANE, PHOSPHOPROTEIN, FAAH, DRUG, MEMBRANE, HYDROLASE, INHIBITOR
2wap:B (PRO231) to (ALA284) 3D-CRYSTAL STRUCTURE OF HUMANIZED-RAT FATTY ACID AMIDE HYDROLASE (FAAH) CONJUGATED WITH THE DRUG-LIKE UREA INHIBITOR PF-3845 | FATTY ACID AMIDE HYDROLASE, UREA INHIBITOR, GOLGI APPARATUS, ENDOPLASMIC RETICULUM, ACYL- ENZYME, TRANSMEMBRANE, PHOSPHOPROTEIN, FAAH, DRUG, MEMBRANE, HYDROLASE, INHIBITOR
3w0m:A (ARG44) to (GLY97) CRYSTAL STRUCTURE OF A THERMOSTABLE MUTANT OF AMINOGLYCOSIDE PHOSPHOTRANSFERASE APH(4)-IA, APO FORM | PHOSPHOTRANSFERASE, TRANSFERASE
2wpg:A (HIS204) to (THR244) SUCROSE HYDROLASE | HYDROLASE, ENZYME, SUCROSE HYDROLYSIS, GLYCOSYL HYDROLASE FAMILY 13
2i4l:B (THR73) to (TYR106) RHODOPSEUDOMONAS PALUSTRIS PROLYL-TRNA SYNTHETASE | ALPHA BETA, LIGASE
2i4l:C (THR73) to (TYR106) RHODOPSEUDOMONAS PALUSTRIS PROLYL-TRNA SYNTHETASE | ALPHA BETA, LIGASE
2i69:A (LEU62) to (THR123) CRYSTAL STRUCTURE OF THE WEST NILE VIRUS ENVELOPE GLYCOPROTEIN | VIRAL MEMBRANE FUSION PROTEIN, RECEPTOR BINDING, ANTIBODY EPITOPE, IGC, BETA SANDWICH, GLYCOPROTEIN, VIRAL PROTEIN
2x7o:A (GLU227) to (VAL279) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH AN INDOLINONE INHIBITOR | KINASE, TRANSFERASE, GLYCOPROTEIN
2x7o:B (GLU227) to (VAL279) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH AN INDOLINONE INHIBITOR | KINASE, TRANSFERASE, GLYCOPROTEIN
2x7o:C (GLU227) to (VAL279) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH AN INDOLINONE INHIBITOR | KINASE, TRANSFERASE, GLYCOPROTEIN
2x7o:D (GLU227) to (VAL279) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH AN INDOLINONE INHIBITOR | KINASE, TRANSFERASE, GLYCOPROTEIN
2x7o:E (GLU227) to (VAL279) CRYSTAL STRUCTURE OF TGFBRI COMPLEXED WITH AN INDOLINONE INHIBITOR | KINASE, TRANSFERASE, GLYCOPROTEIN
2ivy:A (LEU4) to (GLY39) CRYSTAL STRUCTURE OF HYPOTHETICAL PROTEIN SSO1404 FROM SULFOLOBUS SOLFATARICUS P2 | STRUCTURAL GENOMICS, UNKNOWN FUNCTION, CAS, RNAI, CRISPR
2y3y:A (GLU62) to (THR110) HOLO-NI(II) HPNIKR IS A SYMMETRIC TETRAMER CONTAINING FOUR CANONIC SQUARE-PLANAR NI(II) IONS AT PHYSIOLOGICAL PH | TRANSCRIPTION, METAL BINDING
2m9m:A (GLY17) to (SER53) SOLUTION STRUCTURE OF ERCC4 DOMAIN OF HUMAN FAAP24 | FANCONI ANEMIA, FAAP24, ERCC4 DOMAIN, DNA BINDING PROTEIN
2ywh:A (MET296) to (GLY343) CRYSTAL STRUCTURE OF GDP-BOUND LEPA FROM AQUIFEX AEOLICUS | G DOMAIN, BETA-BARREL, FERREDOXIN-LIKE DOMAIN, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, TRANSLATION
4a4l:A (LYS76) to (ARG135) CRYSTAL STRUCTURE OF POLO-LIKE KINASE 1 IN COMPLEX WITH A 5-(2-AMINO-PYRIMIDIN-4-YL)-1H-PYRROLE INHIBITOR | TRANSFERASE
1y11:A (GLY331) to (ARG376) MYCOBACTERIAL ADENYLYL CYCLASE RV1264, HOLOENZYME, ACTIVE STATE | ADENYLYL CYCLASE FOLD, LYASE
1ybt:A (SER414) to (ARG455) MYCOBACTERIUM TUBERCULOSIS ADENYLYL CYCLASE, RV1900C CHD | CYCLASE HOMOLOGY DOMAIN, CHD, RV1900C, HYDROLASE
1ybt:D (SER414) to (VAL452) MYCOBACTERIUM TUBERCULOSIS ADENYLYL CYCLASE, RV1900C CHD | CYCLASE HOMOLOGY DOMAIN, CHD, RV1900C, HYDROLASE
1ydl:A (GLY7) to (PHE44) CRYSTAL STRUCTURE OF THE HUMAN TFIIH, NORTHEAST STRUCTURAL GENOMICS TARGET HR2045. | ALPHA-BETA PROTEIN, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, NESG, TRANSCRIPTION
3a8x:B (ASP268) to (GLY328) CRYSTAL STRUCTURE OF PKCIOTA KINASE DOMAIN | PROTEIN KINASE C IOTA, TRANSFERASE
1yol:A (VAL294) to (GLU341) CRYSTAL STRUCTURE OF SRC KINASE DOMAIN IN COMPLEX WITH CGP77675 | PROTEIN TYROSINE KINASE, TRANSFERASE
1z7n:A (SER46) to (LEU81) ATP PHOSPHORIBOSYL TRANSFERASE (HISZG ATP-PRTASE) FROM LACTOCOCCUS LACTIS WITH BOUND PRPP SUBSTRATE | ATP-PRT, PRPP, HISTIDINE BIOSYNTHESIS, TRANSFERASE, HISZG, ALLOSTERIC
3lo3:C (ALA3) to (PRO59) THE CRYSTAL STRUCTURE OF A CONSERVED FUNCTIONALLY UNKNOWN PROTEIN FROM COLWELLIA PSYCHRERYTHRAEA 34H. | STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, STRUCTURE GENOMICS, UNKNOWN FUNCTION
3lo3:E (ALA3) to (GLU57) THE CRYSTAL STRUCTURE OF A CONSERVED FUNCTIONALLY UNKNOWN PROTEIN FROM COLWELLIA PSYCHRERYTHRAEA 34H. | STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, STRUCTURE GENOMICS, UNKNOWN FUNCTION
3lo3:H (ALA3) to (PRO59) THE CRYSTAL STRUCTURE OF A CONSERVED FUNCTIONALLY UNKNOWN PROTEIN FROM COLWELLIA PSYCHRERYTHRAEA 34H. | STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, STRUCTURE GENOMICS, UNKNOWN FUNCTION
3lo3:I (ALA3) to (GLU57) THE CRYSTAL STRUCTURE OF A CONSERVED FUNCTIONALLY UNKNOWN PROTEIN FROM COLWELLIA PSYCHRERYTHRAEA 34H. | STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, STRUCTURE GENOMICS, UNKNOWN FUNCTION
1zm4:A (VAL488) to (THR533) STRUCTURE OF THE EEF2-ETA-BTAD COMPLEX | ELONGATION FACTOR, TOXIN, ADP-RIBOSYLATION, BIOSYNTHETIC PROTEIN/TRANSFERASE COMPLEX
1zm4:E (VAL488) to (THR533) STRUCTURE OF THE EEF2-ETA-BTAD COMPLEX | ELONGATION FACTOR, TOXIN, ADP-RIBOSYLATION, BIOSYNTHETIC PROTEIN/TRANSFERASE COMPLEX
3lvp:D (VAL1030) to (GLU1080) CRYSTAL STRUCTURE OF BISPHOSPHORYLATED IGF1-R KINASE DOMAIN (2P) IN COMPLEX WITH A BIS-AZAINDOLE INHIBITOR | PROTEIN KINASE, TYROSINE KINASE, TYROSINE PHOSPHORYLATION, PROTEIN- SUBSTRATE COMPLEX, TRANSFERASE
5es1:A (ARG80) to (ALA137) CRYSTAL STRUCTURE OF MICROTUBULE AFFINITY-REGULATING KINASE 4 CATALYTIC DOMAIN IN COMPLEX WITH A PYRAZOLOPYRIMIDINE INHIBITOR | MARK4 PAR-1 SERINE/THREONINE PROTEIN KINASE11, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3bgp:A (ALA65) to (GLU121) HUMAN PIM-1 COMPLEXED WITH A BENZOISOXAZOLE INHIBITOR VX1 | KINASE INHIBITOR PHOSPHORYLATION, ALTERNATIVE INITIATION, ATP-BINDING, CYTOPLASM, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3mr7:A (GLY127) to (PRO169) CRYSTAL STRUCTURE OF ADENYLATE/GUANYLATE CYCLASE/HYDROLASE FROM SILICIBACTER POMEROYI | ALPHA-BETA FOLD, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, HYDROLASE
5fxs:A (VAL1030) to (GLU1080) IGFR-1R COMPLEX WITH A PYRIMIDINE INHIBITOR. | TRANSFERASE
3czg:A (HIS203) to (THR243) CRYSTAL STRUCTURE ANALYSIS OF SUCROSE HYDROLASE (SUH)- GLUCOSE COMPLEX | (ALPHA/BETA)8-BARREL, HYDROLASE
3dk7:A (VAL268) to (GLU316) CRYSTAL STRUCTURE OF MUTANT ABL KINASE DOMAIN IN COMPLEX WITH SMALL MOLECULE FRAGMENT | DRUG DISCOVERY, ABL KINASE, FRAGMENT BASED, ALTERNATIVE SPLICING, ATP-BINDING, CELL ADHESION, CHROMOSOMAL REARRANGEMENT, CYTOPLASM, CYTOSKELETON, KINASE, LIPOPROTEIN, MAGNESIUM, MANGANESE, METAL-BINDING, MYRISTATE, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE
3p1z:D (SER18) to (SER57) CRYSTAL STRUCTURE OF THE APEROPYRUM PERNIX RNA SPLICING ENDONUCLEASE | MIXED ANTIPARALLEL AND PARALLEL BETA-SHEET, HETEROTETRAMER, RNA SPLICING, RNA, SPLICING ENDONUCLEASE, HYDROLASE
3q3b:A (GLU80) to (ASP133) 6-AMINO-4-(PYRIMIDIN-4-YL)PYRIDONES: NOVEL GLYCOGEN SYNTHASE KINASE-3 INHIBITORS | KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5jlb:A (THR1574) to (ALA1617) CRYSTAL STRUCTURE OF SETD2 BOUND TO HISTONE H3.3 K36I PEPTIDE | SET DOMAIN, TRANSFERASE
5lt8:A (LEU1577) to (ALA1617) STRUCTURE OF THE EPIGENETIC ONCOGENE MMSET AND INHIBITION BY N-ALKYL SINEFUNGIN DERIVATIVES | LYSINE METHYLTRANSFERASE SETD2 SET DOMAIN, TRANSFERASE