3e63:A (SER936) to (ILE992) FRAGMENT BASED DISCOVERY OF JAK-2 INHIBITORS | DRUG DISCOVERY, JAK2, FRAGMENT BASED, ATP-BINDING, DISEASE MUTATION, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, SH2 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
2oid:C (SER269) to (SER328) CRYSTAL STRUCTURE OF IRAK4 KINASE DOMAIN COMPLEXED WITH AMPPNP | KINASE, TRANSFERASE
3efw:A (THR217) to (ASP274) STRUCTURE OF AURORAA WITH PYRIDYL-PYRIMIDINE UREA INHIBITOR | AURORAA, STK6_HUMAN, ATP-BINDING, CELL CYCLE, KINASE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE-INHIBITOR COMPLEX
3efw:B (THR217) to (ASP274) STRUCTURE OF AURORAA WITH PYRIDYL-PYRIMIDINE UREA INHIBITOR | AURORAA, STK6_HUMAN, ATP-BINDING, CELL CYCLE, KINASE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE-INHIBITOR COMPLEX
4h3b:A (LEU153) to (ASP207) CRYSTAL STRUCTURE OF JNK3 IN COMPLEX WITH SAB PEPTIDE | SH3BP-5, MAPK, KINASE, TRANSFERASE
2b4f:A (THR77) to (ASP138) STRUCTURE OF A COLD-ADAPTED FAMILY 8 XYLANASE IN COMPLEX WITH SUBSTRATE | HYDROLASE, XYLAN DEGRADATION, PSYCHROPHILIC, COLD ADAPTATION, TEMPERATURE, GLYCOSYL HYDROLASE, FAMILY 8
3en7:B (SER345) to (VAL402) TARGETED POLYPHARMACOLOGY: CRYSTAL STRUCTURE OF THE C-SRC KINASE DOMAIN IN COMPLEX WITH S1, A MULTITARGETED KINASE INHIBITOR | SRC, TYROSINE, KINASE, POLYPHARMACOLOGY, INHIBITOR, MULTITARGET, PHOSPHOINOSITIDE, TRANSFERASE, SIGNALING, PYRAZOLOPYRIMIDINE, KINASE-INHIBITOR COMPLEX, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TYROSINE-PROTEIN KINASE
3eqb:A (SER150) to (LEU206) X-RAY STRUCTURE OF THE HUMAN MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1 (MEK1) IN A COMPLEX WITH LIGAND AND MGATP | PROTEIN KINASE STRUCTURE, MITOGEN ACTIVATED PROTEIN KINASE KINASE, SIGNAL TRANSDUCTION, LIGAND CO-COMPLEX, TERNARY CO- COMPLEX WITH KINASE, LIGAND AND MGATP, NON-COMPETITIVE PROTEIN KINASE INHIBITOR, TRANSFERASE, ACETYLATION, ATP- BINDING, DISEASE MUTATION, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TYROSINE- PROTEIN KINASE
3eqd:A (SER150) to (LEU206) X-RAY STRUCTURE OF THE HUMAN MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1 (MEK1) IN A BINARY COMPLEX WITH ATP-GS AND MG2P | MEK1 KINASE, ATP-BINDING, DISEASE MUTATION, KINASE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE
3eqg:A (SER150) to (LYS205) X-RAY STRUCTURE OF THE HUMAN MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1 (MEK1) IN A TERNARY COMPLEX WITH PD, ADP AND MG2P | MEK1 KINASE, ATP-BINDING, DISEASE MUTATION, KINASE, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE
1nyr:A (ASP144) to (LEU180) STRUCTURE OF STAPHYLOCOCCUS AUREUS THREONYL-TRNA SYNTHETASE COMPLEXED WITH ATP | THREONYL-TRNA SYNTHETASE, ATP, THREONINE, LIGASE
1b38:A (LEU87) to (LEU143) HUMAN CYCLIN-DEPENDENT KINASE 2 | PROTEIN KINASE, TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, ATP-BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, PHOSPHORYLATION
2p55:A (SER150) to (LEU206) X-RAY STRUCTURE OF THE HUMAN MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1 (MEK1) IN A COMPLEX WITH LIGAND AND MGATP | PROTEIN KINASE STRUCTURE; MITOGEN ACTIVATED PROTEIN KINASE KINASE; SIGNAL TRANSDUCTION; LIGAND CO-COMPLEX, TERNARY CO- COMPLEX WITH KINASE, LIGAND AND MGATP; NON-COMPETITIVE PROTEIN KINASE INHIBITOR, TRANSFERASE
2bhh:A (LEU87) to (LEU143) HUMAN CYCLIN DEPENDENT PROTEIN KINASE 2 IN COMPLEX WITH THE INHIBITOR 4-HYDROXYPIPERINDINESULFONYL-INDIRUBINE | 3D-STRUCTURE, ARYLAMINE N-ACETYLTRANSFERASE, ATP-BINDING, CELL CYCLE, CELL DIVISION, DRUG METABOLISM, ISONIAZID, MITOSIS, MYCOBACTERIA, NAT, PHOSPHORYLATION, POLYMORPHISM, SERINE-THREONINE-PROTEIN KINASE, TRANSFERASE
4x21:B (LEU153) to (ASP207) THE MAP KINASE JNK3 AS TARGET FOR HALOGEN BONDING | MAPK, HALOGEN BOND COMPLEX, TRANSFERASE
1bi7:A (ASP104) to (LEU161) MECHANISM OF G1 CYCLIN DEPENDENT KINASE INHIBITION FROM THE STRUCTURE OF THE CDK6-P16INK4A TUMOR SUPPRESSOR COMPLEX | CYCLIN DEPENDENT KINASE, CYCLIN DEPENDENT KINASE INHIBITORY PROTEIN, CDK, INK4, CELL CYCLE, MULTIPLE TUMOR SUPPRESSOR, MTS1, COMPLEX (KINASE/ANTI-ONCOGENE)
3ezv:A (LEU87) to (LEU143) CDK-2 WITH INDAZOLE INHIBITOR 9 BOUND AT ITS ACTIVE SITE | KINASE, PKC, PROTEIN KINASE, INHIBITOR, ATP-BINDING, CELL CYCLE, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4x7h:A (LEU896) to (GLY954) CO-CRYSTAL STRUCTURE OF PERK BOUND TO N-{5-[(6,7-DIMETHOXYQUINOLIN-4- YL)OXY]PYRIDIN-2-YL}-1-METHYL-3-OXO-2-PHENYL-5-(PYRIDIN-4-YL)-2,3- DIHYDRO-1H-PYRAZOLE-4-CARBOXAMIDE INHIBITOR | CATALYTIC DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR, COMPLEX
4x7o:A (LEU896) to (VAL953) CO-CRYSTAL STRUCTURE OF PERK BOUND TO 1-[5-(4-AMINO-2,7-DIMETHYL-7H- PYRROLO[2,3-D]PYRIMIDIN-5-YL)-2,3-DIHYDRO-1H-INDOL-1-YL]-2-[3-FLUORO- 5-(TRIFLUOROMETHYL)PHENYL]ETHANONE INHIBITOR | CATALYTIC DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR, COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3s8r:B (GLY317) to (VAL364) CRYSTAL STRUCTURES OF GLUTARYL 7-AMINOCEPHALOSPORANIC ACID ACYLASE: INSIGHT INTO AUTOPROTEOLYTIC ACTIVATION | MOTIF, ACYLASE, HYDROLASE
4i4f:A (LEU507) to (LEU562) STRUCTURE OF FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH AN ALLOSTERIC BINDING PYRAZOLOBENZOTHIAZINE COMPOUND. | PHOSPHORYLATED ON TYROSINES, LOCALIZED TO FOCAL ADHESIONS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3skx:A (PRO472) to (ASP513) CRYSTAL STRUCTURE OF THE ATP BINDING DOMAIN OF ARCHAEOGLOBUS FULGIDUS COPB | P1B-ATPASE, ATP BINDING DOMAIN, COPPER(II) TRANSPORTER, MEMBRANE PROTEIN, HYDROLASE
2c43:A (PRO52) to (LEU104) STRUCTURE OF AMINOADIPATE-SEMIALDEHYDE DEHYDROGENASE- PHOSPHOPANTETHEINYL TRANSFERASE IN COMPLEX WITH COENZYME A | TRANSFERASE, FATTY ACID BIOSYNTHESIS, COENZYME A
2c6l:A (LYS88) to (LEU143) CRYSTAL STRUCTURE OF THE HUMAN CDK2 COMPLEXED WITH THE TRIAZOLOPYRIMIDINE INHIBITOR | TRANSFERASE, SERINE/THREONINE PROTEIN KINASE, CDK2, ATP-BINDING, CELL CYCLE, MITOSIS, PHOSPHORYLATION, TRIAZOLOPYRIMIDINE INHIBITOR, CELL DIVISION, KINASE, POLYMORPHISM, NUCLEOTIDE-BINDING
4ic7:D (LEU144) to (ILE198) CRYSTAL STRUCTURE OF THE ERK5 KINASE DOMAIN IN COMPLEX WITH AN MKK5 BINDING FRAGMENT | KINASE DOMAIN, SIGNALING PROTEIN COMPLEX, TRANSFERASE
3fz1:A (LYS88) to (LEU143) CRYSTAL STRUCTURE OF A BENZTHIOPHENE INHIBITOR BOUND TO HUMAN CYCLIN-DEPENDENT KINASE-2 (CDK-2) | CDK-2, MK-2, MK2, MAPKAP KINASE-2, SER/THR KINASE, CELL DIVISON KINASE-2, CYCLIN, BENZOTHIOPHENE, ATP-BINDING, CELL CYCLE, CELL DIVISION, KINASE, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
1p2a:A (LEU87) to (LEU143) THE STRUCTURE OF CYCLIN DEPENDENT KINASE 2 (CKD2) WITH A TRISUBSTITUTED NAPHTHOSTYRIL INHIBITOR | CYCLIN DEPENDENT KINASE, NAPHTHOSTYRIL OXINDOLE, TRANSFERASE
4xr7:I (SER383) to (HIS445) STRUCTURE OF THE SACCHAROMYCES CEREVISIAE PAN2-PAN3 CORE COMPLEX | RNA DEGRADATION, DEADENYLATION, HYDROLASE, PSEUDOKINASE
2clx:A (LYS88) to (LEU143) 4-ARYLAZO-3,5-DIAMINO-1H-PYRAZOLE CDK INHIBITORS: SAR STUDY, CRYSTAL STRUCTURE IN COMPLEX WITH CDK2, SELECTIVITY, AND CELLULAR EFFECTS | TRANSFERASE, SERINE/THREONINE- PROTEIN KINASE, PHOSPHORYLATION, NUCLEOTIDE-BINDING, CDK2, KINASE, MITOSIS, CELL CYCLE, ATP-BINDING, POLYMORPHISM, CELL DIVISION, SERINE-THREONINE-PROTEIN KINASE
1dik:A (PRO290) to (ASN338) PYRUVATE PHOSPHATE DIKINASE | TRANSFERASE, KINASE, PHOSPHOTRANSFERASE
1dl2:A (ASN129) to (LYS195) CRYSTAL STRUCTURE OF CLASS I ALPHA-1,2-MANNOSIDASE FROM SACCHAROMYCES CEREVISIAE AT 1.54 ANGSTROM RESOLUTION | ALPHA-ALPHA HELIX BARREL, HYDROLASE
3gc0:A (LEU98) to (ASP159) STRUCTURE OF THE CMGC CDK KINASE FROM GIARDIA LAMBLIA IN COMPLEX WITH AMP | SSGCID, KINASE, CMGC CDK, AMP, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE
2qq7:B (CYS345) to (PHE405) CRYSTAL STRUCTURE OF DRUG RESISTANT SRC KINASE DOMAIN WITH IRREVERSIBLE INHIBITOR | SRC KINASE DOMAIN, DRUG RESISTANCE, IRREVERSIBLE INHIBITOR, ALTERNATIVE SPLICING, ATP-BINDING, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE, TYROSINE-PROTEIN KINASE
4itj:A (ASN99) to (ASP156) CRYSTAL STRUCTURE OF RIP1 KINASE IN COMPLEX WITH NECROSTATIN-4 | ALPHA/BETA, RIP1 KINASE, NECROPTOSIS, NECROSTATINS, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3gfw:A (LEU609) to (ASP664) CRYSTAL STRUCTURE OF HUMAN DUAL SPECIFICITY PROTEIN KINASE (TTK) IN COMPLEX WITH A PYROLO-PYRIDIN LIGAND | TTK, HMPS1, PYT, ESK, KINASE, DUAL SPECIFICITY, PHOSPHOTYROSINE PICKED THREONINE KINASE, SGC, STRUCTURAL GENOMICS CONSORTIUM, ATP- BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE
1pxi:A (LEU87) to (LEU143) HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR 4-(2,5-DICHLORO-THIOPHEN-3-YL)-PYRIMIDIN-2- YLAMINE | PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, 3D-STRUCTURE.
1pxn:A (LEU87) to (LEU143) HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR 4-[4-(4-METHYL-2-METHYLAMINO-THIAZOL-5-YL)- PYRIMIDIN-2-YLAMINO]-PHENOL | PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, 3D-STRUCTURE.
2r3g:A (LYS88) to (LEU143) CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH INHIBITOR | SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE, INHIBITION, CYCLIN-DEPENDENT KINASE, CANCER, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE
2r3q:A (LEU87) to (LEU143) CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH INHIBITOR | SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE, INHIBITION, CYCLIN-DEPENDENT KINASE, CANCER, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE
2r3r:A (LEU87) to (LEU143) CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH INHIBITOR | SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE, INHIBITION, CYCLIN-DEPENDENT KINASE, CANCER, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE
3tcp:B (LEU679) to (VAL739) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF THE PROTO-ONCOGENE TYROSINE-PROTEIN KINASE MER IN COMPLEX WITH INHIBITOR UNC569 | TYROSINE KINASE, ACUTE LYMPHOBLASTIC LEUKEMIA, RATIONAL STRUCTURE- BASED DRUG DESIGN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2r82:A (PRO290) to (GLN335) PYRUVATE PHOSPHATE DIKINASE (PPDK) TRIPLE MUTANT R219E/E271R/S262D ADAPTS A SECOND CONFORMATIONAL STATE | PHOSPHOTRANSFERASE, CONFORMATIONAL TRANSITION, SWIVELING DOMAIN, REMOTE ACTIVE SITES, ATP-BINDING, KINASE, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, TRANSFERASE
2rfe:B (LEU774) to (ILE829) CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN THE EGFR KINASE DOMAIN AND A MIG6 PEPTIDE | KINASE DOMAIN, INHIBITION, DIMER, PEPTIDE, ALTERNATIVE SPLICING, ANTI-ONCOGENE, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, UBL CONJUGATION, CYTOPLASM
2rfs:A (LEU1165) to (VAL1220) X-RAY STRUCTURE OF SU11274 BOUND TO C-MET | C-MET, RECEPTOR TYROSINE KINASE, SU11274, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, PROTO-ONCOGENE, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE
4yf9:F (THR161) to (ALA205) STRUCTURE OF N-ACYLHOMOSERINE LACTONE ACYLASE MACQ | ACYLASE, NTN-HYDROLASE FOLD, HYDROLASE
4yf9:I (THR161) to (ALA205) STRUCTURE OF N-ACYLHOMOSERINE LACTONE ACYLASE MACQ | ACYLASE, NTN-HYDROLASE FOLD, HYDROLASE
4yfa:F (THR161) to (ALA205) STRUCTURE OF N-ACYLHOMOSERINE LACTONE ACYLASE MACQ IN COMPLEX WITH DECANOIC ACID | ACYLASE, PRODUCT COMPLEX, NTN-HYDROLASE FOLD, HYDROLASE
4yfa:I (THR161) to (ALA205) STRUCTURE OF N-ACYLHOMOSERINE LACTONE ACYLASE MACQ IN COMPLEX WITH DECANOIC ACID | ACYLASE, PRODUCT COMPLEX, NTN-HYDROLASE FOLD, HYDROLASE
4yfb:C (THR161) to (ALA205) STRUCTURE OF N-ACYLHOMOSERINE LACTONE ACYLASE MACQ IN COMPLEX WITH PHENYLACETIC ACID | ACYLASE, PRODUCT COMPLEX, NTN-HYDROLASE FOLD, HYDROLASE
4yfb:F (THR161) to (ALA205) STRUCTURE OF N-ACYLHOMOSERINE LACTONE ACYLASE MACQ IN COMPLEX WITH PHENYLACETIC ACID | ACYLASE, PRODUCT COMPLEX, NTN-HYDROLASE FOLD, HYDROLASE
4yfb:L (THR161) to (ALA205) STRUCTURE OF N-ACYLHOMOSERINE LACTONE ACYLASE MACQ IN COMPLEX WITH PHENYLACETIC ACID | ACYLASE, PRODUCT COMPLEX, NTN-HYDROLASE FOLD, HYDROLASE
3h10:A (VAL218) to (ILE272) AURORA A INHIBITOR COMPLEX | PROTEIN:INHIBITOR COMPLEX AURORA-A, CELL CYCLE, SERINE/THREONINE, PROTEIN KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4jqe:A (ASP159) to (LEU212) CRYSTAL STRUCTURE OF SCCK2 ALPHA IN COMPLEX WITH AMPPN | PROTEIN KINASE, PROTEIN PHOSPHORYLATION, TRANSFERASE
3h4j:B (LEU118) to (ASP174) CRYSTAL STRUCTURE OF POMBE AMPK KDAID FRAGMENT | AMPK, KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4jx3:A (ASP128) to (LEU184) CRYSTAL STRUCTURE OF PIM1 KINASE | HUMAN PROTEIN KINASES, SERINE/THREONINE-PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
3uc3:A (LEU103) to (ASP161) THE CRYSTAL STRUCTURE OF SNF1-RELATED KINASE 2.3 | SNRK2, KINASE, ABA SIGNALING, TRANSFERASE
4yr8:C (LEU115) to (ASP169) CRYSTAL STRUCTURE OF JNK IN COMPLEX WITH A REGULATOR PROTEIN | KINASE DOMAIN, CATALYTIC DOMAIN, TRANSFERASE-HYDROLASE COMPLEX
1fmi:A (ASN327) to (PRO386) CRYSTAL STRUCTURE OF HUMAN CLASS I ALPHA1,2-MANNOSIDASE | ALPHA-ALPHA7 BARREL, HYDROLASE
1fmi:A (ASP523) to (LYS588) CRYSTAL STRUCTURE OF HUMAN CLASS I ALPHA1,2-MANNOSIDASE | ALPHA-ALPHA7 BARREL, HYDROLASE
3uib:A (LEU119) to (ILE174) MAP KINASE LMAMPK10 FROM LEISHMANIA MAJOR IN COMPLEX WITH SB203580 | EUKARIOTIC PROTEIN KINASE FOLD, TRANSFERASE
4k9y:A (LEU507) to (LEU562) FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH 1-[4-(6-AMINO- PURIN-9-YL)-PHENYL]-3-(5-TERT-BUTYL-2-P-TOLYL-2H-PYRAZOL-3-YL)-UREA | TYROSINE PROTEIN KINASE, TRANSFERASE, ATP BINDING, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3hmj:A (THR1792) to (LEU1851) SACCHAROMYCES CEREVISIAE FAS TYPE I | FAS, PPT, PHOSPHOPANTETHEINE TRANSFERASE, FATTY ACID, MULTIENYZME, FATTY ACID BIOSYNTHESIS, LIPID SYNTHESIS, MULTIFUNCTIONAL ENZYME, NAD, NADP, OXIDOREDUCTASE, PHOSPHOPROTEIN, HYDROLASE, LYASE
3hmj:B (THR1792) to (LEU1851) SACCHAROMYCES CEREVISIAE FAS TYPE I | FAS, PPT, PHOSPHOPANTETHEINE TRANSFERASE, FATTY ACID, MULTIENYZME, FATTY ACID BIOSYNTHESIS, LIPID SYNTHESIS, MULTIFUNCTIONAL ENZYME, NAD, NADP, OXIDOREDUCTASE, PHOSPHOPROTEIN, HYDROLASE, LYASE
3hmj:C (THR1792) to (LEU1851) SACCHAROMYCES CEREVISIAE FAS TYPE I | FAS, PPT, PHOSPHOPANTETHEINE TRANSFERASE, FATTY ACID, MULTIENYZME, FATTY ACID BIOSYNTHESIS, LIPID SYNTHESIS, MULTIFUNCTIONAL ENZYME, NAD, NADP, OXIDOREDUCTASE, PHOSPHOPROTEIN, HYDROLASE, LYASE
4kd1:A (LYS88) to (LEU143) CDK2 IN COMPLEX WITH DINACICLIB | PROTEIN KINASE, DINACICLIB, TRANSFERASE-TRANSFERASE, CELL CYCLE- INHIBITOR COMPLEX
1g3n:A (LEU105) to (LEU161) STRUCTURE OF A P18(INK4C)-CDK6-K-CYCLIN TERNARY COMPLEX | CYCLIN-DEPENDENT KINASE, INK4 INHIBITOR, VIRAL CYCLIN, CELL CYCLE, SIGNALING PROTEIN
1g3n:E (LEU105) to (LEU161) STRUCTURE OF A P18(INK4C)-CDK6-K-CYCLIN TERNARY COMPLEX | CYCLIN-DEPENDENT KINASE, INK4 INHIBITOR, VIRAL CYCLIN, CELL CYCLE, SIGNALING PROTEIN
3uok:A (VAL218) to (ASP274) AURORA A IN COMPLEX WITH YL5-81-1 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uok:B (VAL218) to (ASP274) AURORA A IN COMPLEX WITH YL5-81-1 | PROTEIN KINASE, AURORA A, INHIBITOR, DFG-OUT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4kke:A (LEU153) to (ASP207) THE CRYSTAL STRUCTURE OF AMP-BOUND JNK3 | KINASE DOMAIN, KINASE, C-JUN, TRANSFERASE
4kkh:A (LEU153) to (ASP207) THE CRYSTAL STRUCTURE OF INHIBITOR-BOUND JNK3 | KINASE DOMAIN, KINASE, C-JUN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3v01:A (LEU151) to (LEU206) DISCOVERY OF NOVEL ALLOSTERIC MEK INHIBITORS POSSESSING CLASSICAL AND NON-CLASSICAL BIDENTATE SER212 INTERACTIONS. | KINASE, TRANSFERASE-INHIBITOR COMPLEX
4knb:A (LEU1165) to (ALA1221) C-MET IN COMPLEX WITH OSI LIGAND | PROTEIN KINASE, TRANSFERASE
1gk1:B (GLY148) to (VAL195) STRUCTURE-BASED PREDICTION OF MODIFICATIONS IN GLUTARYLAMIDASE TO ALLOW SINGLE-STEP ENZYMATIC PRODUCTION OF 7-AMINOCEPHALOSPORANIC ACID FROM CEPHALOSPORIN C | HYDROLASE, CEPHALOSPORIN ACYLASE, GLUTARYL ACYLASE, CEPHALOSPORIN C, CATALYTIC TRIAD, NTN-HYDROLASE, X-RAZ STRUCTURE
4zeg:A (LEU609) to (ASP664) CRYSTAL STRUCTURE OF TTK KINASE DOMAIN IN COMPLEX WITH A PYRAZOLOPYRIMIDINE INHIBITOR | KINASE, TTK, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2g01:A (LEU115) to (ILE167) PYRAZOLOQUINOLONES AS NOVEL, SELECTIVE JNK1 INHIBITORS | JNK1, C-JUN N-TERMINAL KINASE, PROTEIN KINASE JNK1 INHIBITORS, TRANSFERASE
2vta:A (LEU87) to (LEU143) IDENTIFICATION OF N-(4-PIPERIDINYL)-4-(2,6- DICHLOROBENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXAMIDE (AT7519), A NOVEL CYCLIN DEPENDENT KINASE INHIBITOR USING FRAGMENT- BASED X-RAY CRYSTALLOGRAPHY AND STRUCTURE BASED DRUG DESIGN. | TRANSFERASE, MITOSIS, CELL CYCLE, CELL DIVISION, SERINE/THREONINE PROTEIN KINASE, PHOSPHORYLATION
2vth:A (LYS88) to (LEU143) IDENTIFICATION OF N-(4-PIPERIDINYL)-4-(2,6- DICHLOROBENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXAMIDE (AT7519), A NOVEL CYCLIN DEPENDENT KINASE INHIBITOR USING FRAGMENT- BASED X-RAY CRYSTALLOGRAPHY AND STRUCTURE BASED DRUG DESIGN | TRANSFERASE, MITOSIS, CELL CYCLE, SERINE/THREONINE PROTEIN KINASE
2vtr:A (LEU87) to (LEU143) IDENTIFICATION OF N-(4-PIPERIDINYL)-4-(2,6- DICHLOROBENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXAMIDE (AT7519), A NOVEL CYCLIN DEPENDENT KINASE INHIBITOR USING FRAGMENT- BASED X-RAY CRYSTALLOGRAPHY AND STRUCTURE BASED DRUG DESIGN. | TRANSFERASE, MITOSIS, CELL CYCLE, SERINE/THREONINE PROTEIN KINASE
4zji:D (SER351) to (LEU405) PAK1 IN COMPLEX WITH 2-CHLORO-5-ETHYL-8-FLUORO-11-(4-METHYLPIPERAZIN- 1-YL)-DIBENZODIAZEPINE | INHIBITOR, KINASE, PAK1, ALLOSTERIC, TRANSFERASE
4zjj:C (SER351) to (LEU405) PAK1 IN COMPLEX WITH (S)-N-(TERT-BUTYL)-3-((2-CHLORO-5-ETHYL-8-FLUORO- DIBENZODIAZEPIN-11-YL)AMINO)PYRROLIDINE-1-CARBOXAMIDE | PAK1, INHIBITOR, KINASE, ALLOSTERIC, TRANSFERASE
4zjj:D (SER351) to (LEU405) PAK1 IN COMPLEX WITH (S)-N-(TERT-BUTYL)-3-((2-CHLORO-5-ETHYL-8-FLUORO- DIBENZODIAZEPIN-11-YL)AMINO)PYRROLIDINE-1-CARBOXAMIDE | PAK1, INHIBITOR, KINASE, ALLOSTERIC, TRANSFERASE
1gz8:A (LYS88) to (LEU143) HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR 2-AMINO-6-(3'-METHYL-2'-OXO)BUTOXYPURINE | KINASE, PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, CELL DIVISION, MITOSIS, INHIBITION, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, 3D-STRUCTURE.
4l01:B (LEU675) to (ASP739) CRYSTAL STRUCTURE OF THE V658F APO JAK1 PSEUDOKINASE DOMAIN | KINASE DOMAIN FOLD, REGULATORY, TRANSFERASE
4zp5:B (SER112) to (LEU169) MAP4K4 IN COMPLEX WITH INHIBITOR | KINASE, INHIBITOR, TRANSFERASE-INHIBITOR COMPLEX
4zse:B (LEU798) to (ILE853) CRYSTAL STRUCTURE OF EGFR 696-1022 T790M/V948R, CRYSTAL FORM II | EGFR, T790M, V948R, TRANSFERASE
2w5a:A (LEU94) to (LEU157) HUMAN NEK2 KINASE ADP-BOUND | SER/THR PROTEIN KINASE, KINASE, NUCLEUS, MEIOSIS, MITOSIS, CYTOPLASM, SERINE/THREONINE-PROTEIN KINASE, METAL-BINDING, PHOSPHOPROTEIN, NUCLEOTIDE-BINDING, MAGNESIUM, CELL CYCLE, ATP-BINDING, TRANSFERASE, CENTROSOME SPLITTING, ALTERNATIVE SPLICING, COILED COIL, POLYMORPHISM, CELL DIVISION
4zts:A (VAL218) to (ASP274) HUMAN AURORA A CATALYTIC DOMAIN BOUND TO FK1142 | AURORA, KINASE, INHIBITOR, TRANSFERASE
4lfi:A (ASP159) to (LEU212) CRYSTAL STRUCTURE OF SCCK2 ALPHA IN COMPLEX WITH GMPPNP | PROTEIN KINASE, PROTEIN PHOSPHORYLATION, TRANSFERASE
4lfi:B (ASP159) to (LEU212) CRYSTAL STRUCTURE OF SCCK2 ALPHA IN COMPLEX WITH GMPPNP | PROTEIN KINASE, PROTEIN PHOSPHORYLATION, TRANSFERASE
4lgd:A (SER106) to (LEU162) STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5 | HIPPO, MST AUTOACTIVATION, RASSF, SARAH DOMAIN, DIMERIZATION, SIGNALING PROTEIN
4lgd:D (SER106) to (ASP164) STRUCTURAL BASIS FOR AUTOACTIVATION OF HUMAN MST2 KINASE AND ITS REGULATION BY RASSF5 | HIPPO, MST AUTOACTIVATION, RASSF, SARAH DOMAIN, DIMERIZATION, SIGNALING PROTEIN
2h34:B (ASP100) to (LEU155) APOENZYME CRYSTAL STRUCTURE OF THE TUBERCULOSIS SERINE/THREONINE KINASE, PKNE | APOENZYME, SERINE/THREONINE PROTEIN KINASE, TRANSFERASE
2w96:B (LEU100) to (ASP158) CRYSTAL STRUCTURE OF CDK4 IN COMPLEX WITH A D-TYPE CYCLIN | SERINE/THREONINE-PROTEIN KINASE, CHROMOSOMAL REARRANGEMENT, ATP-BINDING, TRANSFERASE, POLYMORPHISM, CELL DIVISION, PROTO-ONCOGENE, PHOSPHOPROTEIN, DISEASE MUTATION, NUCLEOTIDE-BINDING, CYCLIN DEPENDENT KINASE, KINASE, CYCLIN, ONCOLOGY, CELL CYCLE, DRUG DESGN
2w99:B (ASP99) to (LEU156) CRYSTAL STRUCTURE OF CDK4 IN COMPLEX WITH A D-TYPE CYCLIN | SERINE/THREONINE-PROTEIN KINASE, CHROMOSOMAL REARRANGEMENT, ATP-BINDING, TRANSFERASE, POLYMORPHISM, CELL DIVISION, PROTO-ONCOGENE, PHOSPHOPROTEIN, DISEASE MUTATION, NUCLEOTIDE-BINDING, CYCLIN DEPENDENT KINASE, KINASE, CYCLIN, ONCOLOGY, CELL CYCLE, DRUG DESGN
2w9f:B (LEU100) to (ASP158) CRYSTAL STRUCTURE OF CDK4 IN COMPLEX WITH A D-TYPE CYCLIN | SERINE/THREONINE-PROTEIN KINASE, CHROMOSOMAL REARRANGEMENT, ATP-BINDING, TRANSFERASE, POLYMORPHISM, CELL DIVISION, PROTO-ONCOGENE, PHOSPHOPROTEIN, DISEASE MUTATION, NUCLEOTIDE-BINDING, CYCLIN DEPENDENT KINASE, KINASE, CYCLIN, ONCOLOGY, CELL CYCLE, DRUG DESGN
2w9z:B (ASP99) to (ASP158) CRYSTAL STRUCTURE OF CDK4 IN COMPLEX WITH A D-TYPE CYCLIN | TRANSFERASE, CYCLIN DEPENDENT KINASE, TRANSFERASE ONCOLOGY, CELL CYCLE, DRUG DESIGN
2was:A (THR1792) to (GLY1853) STRUCTURE OF THE FUNGAL TYPE I FAS PPT DOMAIN | COA, FAS, PPT, NAD, NADP, TRANSFERASE, PHOSPHOPROTEIN, OXIDOREDUCTASE, LIPID SYNTHESIS, PHOSPHOPANTETHEINE TRANSFERASE, PHOSPHOPANTETHEINE, MULTIFUNCTIONAL ENZYME, FATTY ACID BIOSYNTHESIS, PHOSPHOPANTETHEINYLATION
2was:B (THR1792) to (LEU1851) STRUCTURE OF THE FUNGAL TYPE I FAS PPT DOMAIN | COA, FAS, PPT, NAD, NADP, TRANSFERASE, PHOSPHOPROTEIN, OXIDOREDUCTASE, LIPID SYNTHESIS, PHOSPHOPANTETHEINE TRANSFERASE, PHOSPHOPANTETHEINE, MULTIFUNCTIONAL ENZYME, FATTY ACID BIOSYNTHESIS, PHOSPHOPANTETHEINYLATION
2was:C (THR1792) to (LEU1851) STRUCTURE OF THE FUNGAL TYPE I FAS PPT DOMAIN | COA, FAS, PPT, NAD, NADP, TRANSFERASE, PHOSPHOPROTEIN, OXIDOREDUCTASE, LIPID SYNTHESIS, PHOSPHOPANTETHEINE TRANSFERASE, PHOSPHOPANTETHEINE, MULTIFUNCTIONAL ENZYME, FATTY ACID BIOSYNTHESIS, PHOSPHOPANTETHEINYLATION
2was:E (THR1792) to (GLY1853) STRUCTURE OF THE FUNGAL TYPE I FAS PPT DOMAIN | COA, FAS, PPT, NAD, NADP, TRANSFERASE, PHOSPHOPROTEIN, OXIDOREDUCTASE, LIPID SYNTHESIS, PHOSPHOPANTETHEINE TRANSFERASE, PHOSPHOPANTETHEINE, MULTIFUNCTIONAL ENZYME, FATTY ACID BIOSYNTHESIS, PHOSPHOPANTETHEINYLATION
2was:F (THR1792) to (LEU1851) STRUCTURE OF THE FUNGAL TYPE I FAS PPT DOMAIN | COA, FAS, PPT, NAD, NADP, TRANSFERASE, PHOSPHOPROTEIN, OXIDOREDUCTASE, LIPID SYNTHESIS, PHOSPHOPANTETHEINE TRANSFERASE, PHOSPHOPANTETHEINE, MULTIFUNCTIONAL ENZYME, FATTY ACID BIOSYNTHESIS, PHOSPHOPANTETHEINYLATION
2wat:A (THR1792) to (LEU1851) STRUCTURE OF THE FUNGAL TYPE I FAS PPT DOMAIN IN COMPLEX WITH COA | COA, FAS, PPT, NAD, NADP, TRANSFERASE, PHOSPHOPROTEIN, OXIDOREDUCTASE, LIPID SYNTHESIS, PHOSPHOPANTETHEINE TRANSFERASE, PHOSPHOPANTETHEINE, MULTIFUNCTIONAL ENZYME, FATTY ACID BIOSYNTHESIS, PHOSPHOPANTETHEINYLATION
2wat:B (THR1792) to (GLY1853) STRUCTURE OF THE FUNGAL TYPE I FAS PPT DOMAIN IN COMPLEX WITH COA | COA, FAS, PPT, NAD, NADP, TRANSFERASE, PHOSPHOPROTEIN, OXIDOREDUCTASE, LIPID SYNTHESIS, PHOSPHOPANTETHEINE TRANSFERASE, PHOSPHOPANTETHEINE, MULTIFUNCTIONAL ENZYME, FATTY ACID BIOSYNTHESIS, PHOSPHOPANTETHEINYLATION
2wat:C (THR1792) to (GLY1853) STRUCTURE OF THE FUNGAL TYPE I FAS PPT DOMAIN IN COMPLEX WITH COA | COA, FAS, PPT, NAD, NADP, TRANSFERASE, PHOSPHOPROTEIN, OXIDOREDUCTASE, LIPID SYNTHESIS, PHOSPHOPANTETHEINE TRANSFERASE, PHOSPHOPANTETHEINE, MULTIFUNCTIONAL ENZYME, FATTY ACID BIOSYNTHESIS, PHOSPHOPANTETHEINYLATION
2wat:D (THR1792) to (GLY1853) STRUCTURE OF THE FUNGAL TYPE I FAS PPT DOMAIN IN COMPLEX WITH COA | COA, FAS, PPT, NAD, NADP, TRANSFERASE, PHOSPHOPROTEIN, OXIDOREDUCTASE, LIPID SYNTHESIS, PHOSPHOPANTETHEINE TRANSFERASE, PHOSPHOPANTETHEINE, MULTIFUNCTIONAL ENZYME, FATTY ACID BIOSYNTHESIS, PHOSPHOPANTETHEINYLATION
2wat:E (THR1792) to (LEU1851) STRUCTURE OF THE FUNGAL TYPE I FAS PPT DOMAIN IN COMPLEX WITH COA | COA, FAS, PPT, NAD, NADP, TRANSFERASE, PHOSPHOPROTEIN, OXIDOREDUCTASE, LIPID SYNTHESIS, PHOSPHOPANTETHEINE TRANSFERASE, PHOSPHOPANTETHEINE, MULTIFUNCTIONAL ENZYME, FATTY ACID BIOSYNTHESIS, PHOSPHOPANTETHEINYLATION
2wat:F (THR1792) to (GLY1853) STRUCTURE OF THE FUNGAL TYPE I FAS PPT DOMAIN IN COMPLEX WITH COA | COA, FAS, PPT, NAD, NADP, TRANSFERASE, PHOSPHOPROTEIN, OXIDOREDUCTASE, LIPID SYNTHESIS, PHOSPHOPANTETHEINE TRANSFERASE, PHOSPHOPANTETHEINE, MULTIFUNCTIONAL ENZYME, FATTY ACID BIOSYNTHESIS, PHOSPHOPANTETHEINYLATION
4lmn:A (SER150) to (LEU206) CRYSTAL STRUCTURE OF MEK1 KINASE BOUND TO GDC0973 | KINASE, PHOSPHORYLATION, BRAF, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2wkm:A (LEU1165) to (VAL1220) X-RAY STRUCTURE OF PHA-00665752 BOUND TO THE KINASE DOMAIN OF C-MET | HEPATOCYTE GROWTH FACTOR RECEPTOR, C-MET, KINASE, INHIBITOR, TRANSFERASE
3vvh:B (SER150) to (LEU206) X-RAY STRUCTURE OF THE HUMAN MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1 (MEK1) IN COMPLEX WITH AN INHIBITOR AND MGATP | KINASE DOMAIN, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3vvh:C (SER150) to (LEU206) X-RAY STRUCTURE OF THE HUMAN MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1 (MEK1) IN COMPLEX WITH AN INHIBITOR AND MGATP | KINASE DOMAIN, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3w32:A (CYS797) to (ILE853) EGFR KINASE DOMAIN COMPLEXED WITH COMPOUND 20A | ANTI-ONCOGENE, CELL CYCLE, DISEASE MUTATION, KINASE DOMAIN, RECEPTOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2hwo:A (CYS345) to (VAL402) CRYSTAL STRUCTURE OF SRC KINASE DOMAIN IN COMPLEX WITH COVALENT INHIBITOR | KINASE, COVALENT, QUINAZOLINE, MODIFICATION, TRANSFERASE
4m67:A (THR290) to (ALA348) CRYSTAL STRUCTURE OF THE HUMAN MLKL KINASE-LIKE DOMAIN | KINASE-LIKE, A SUBSTRATE OF RIP3, RIP3, SIGNALING PROTEIN
4m68:A (THR279) to (ALA335) CRYSTAL STRUCTURE OF THE MOUSE MLKL KINASE-LIKE DOMAIN | KINASE-LIKE, SUBSTRATE OF RIP3, RIP3, SIGNALING PROTEIN
4m69:B (THR279) to (GLY336) CRYSTAL STRUCTURE OF THE MOUSE RIP3-MLKL COMPLEX | KINASE, PHOSPHORYLATION, TRANSFERASE-SIGNALING PROTEIN COMPLEX
2x0s:A (MET321) to (ASN365) 3.0 A RESOLUTION CRYSTAL STRUCTURE OF GLYCOSOMAL PYRUVATE PHOSPHATE DIKINASE FROM TRYPANOSOMA BRUCEI | KINASE, TRANSFERASE, TROPICAL PARASITE
4mf1:B (CYS442) to (VAL498) ITK KINASE DOMAIN IN COMPLEX WITH BENZOTHIAZOLE INHIBITOR 12B (1S,2S)- 2-{4-[(DIMETHYLAMINO)METHYL]PHENYL}-N-[6-(1H-PYRAZOL-4-YL)-1,3- BENZOTHIAZOL-2-YL]CYCLOPROPANECARBOXAMIDE | PROTEIN KINASE, PHOSPHOTRANSFER CATALYST, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3wig:A (SER151) to (LEU207) HUMAN MEK1 KINASE IN COMPLEX WITH CH5126766 AND MGAMP-PNP | KINASE, KINASE INHIBITOR, ALLOSTERIC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1v0p:B (LEU86) to (ASP143) STRUCTURE OF P. FALCIPARUM PFPK5-PURVALANOL B LIGAND COMPLEX | TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PHOSPHORYLATION, CDK
2x6d:A (THR217) to (ALA273) AURORA-A BOUND TO AN INHIBITOR | TRANSFERASE, MITOSIS
2x6e:A (THR217) to (ALA273) AURORA-A BOUND TO AN INHIBITOR | TRANSFERASE, MITOSIS, CELL CYCLE
4mne:A (SER150) to (LEU206) CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4mne:D (SER150) to (LEU206) CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4mne:H (SER150) to (LEU206) CRYSTAL STRUCTURE OF THE BRAF:MEK1 COMPLEX | RAF, MAPK, KINASE DOMAIN, ATP-BINDING, ERK, RAS, PAK, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5ane:A (LEU87) to (LEU143) CRYSTAL STRUCTURE OF CDK2 IN COMPLEX WITH 6-METHOXY-7H- PURINE PROCESSED WITH THE CRYSTALDIRECT AUTOMATED MOUNTING AND CRYO-COOLING TECHNOLOGY | TRANSFERASE, PROTEIN KINASE, INHIBITOR, AUTOMATED CRYSTAL HARVESTING, AUTOMATED CRYO-COOLING, CRYSTALDIRECT
3j3u:E (THR744) to (ALA807) STRUCTURAL DYNAMICS OF THE MECA-CLPC COMPLEX REVEALED BY CRYO-EM | CLPC, MECA, AAA+ ATPASE, PROTEIN UNFOLDING, CHAPERONE
3j3u:F (THR744) to (ALA807) STRUCTURAL DYNAMICS OF THE MECA-CLPC COMPLEX REVEALED BY CRYO-EM | CLPC, MECA, AAA+ ATPASE, PROTEIN UNFOLDING, CHAPERONE
5ani:A (LEU87) to (LEU143) CRYSTAL STRUCTURE OF CDK2 IN COMPLEX WITH 6-CHLORO-7H- PURINE PROCESSED WITH THE CRYSTALDIRECT AUTOMATED MOUNTING AND CRYO-COOLING TECHNOLOGY | TRANSFERASE, PROTEIN KINASE, INHIBITOR, AUTOMATED CRYSTAL HARVESTING, AUTOMATED CRYO-COOLING, CRYSTALDIRECT
5anj:A (LEU87) to (LEU143) CRYSTAL STRUCTURE OF CDK2 IN COMPLEX WITH N-(9H-PURIN-6-YL) THIOPHENE-2-CARBOXAMIDE PROCESSED WITH THE CRYSTALDIRECT AUTOMATED MOUNTING AND CRYO-COOLING TECHNOLOGY | TRANSFERASE, PROTEIN KINASE, INHIBITOR, AUTOMATED CRYSTAL HARVESTING, AUTOMATED CRYO-COOLING, CRYSTALDIRECT
5ap7:A (LEU609) to (ASP664) NATURALLY OCCURRING MUTATIONS IN THE MPS1 GENE PREDISPOSE CELLS TO KINASE INHIBITOR DRUG RESISTANCE. | TRANSFERASE, MPS1, MITOSIS
2j4z:B (VAL218) to (ASP274) STRUCTURE OF AURORA-2 IN COMPLEX WITH PHA-680626 | TRANSFERASE, PHOSPHORYLATION, NUCLEOTIDE-BINDING, KINASE, CELL CYCLE, ATP-BINDING, NUCLEOTIDE- BINDING, SERINE/THREONINE-PROTEIN KINASE, SERINE-THREONINE-PROTEIN KINASE
1jow:B (ASP104) to (LEU161) CRYSTAL STRUCTURE OF A COMPLEX OF HUMAN CDK6 AND A VIRAL CYCLIN | CDK-CYCLIN COMPLEX, CYCLIN FOLD, CELL CYCLE/TRANSFERASE COMPLEX
1vyz:A (LEU87) to (LEU143) STRUCTURE OF CDK2 COMPLEXED WITH PNU-181227 | PROTEIN KINASE, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, PHOSPHORYLATION, CELL DIVISION, CYCLIN
2jav:A (LEU94) to (LEU157) HUMAN KINASE WITH PYRROLE-INDOLINONE LIGAND | TRANSFERASE, PHOSPHORYLATION, NUCLEOTIDE-BINDING, ATP-BINDING, CELL DIVISION, METAL-BINDING, NUCLEAR PROTEIN, SERINE/THREONINE-PROTEIN KINASE, SERINE/THREONINE PROTEIN KINASE, KINASE, MEIOSIS, MITOSIS, MAGNESIUM, CELL CYCLE
2jc6:C (LEU106) to (ILE163) CRYSTAL STRUCTURE OF HUMAN CALMODULIN-DEPENDENT PROTEIN KINASE 1D | TRANSFERASE, ATP-BINDING, NUCLEAR PROTEIN, PHOSPHORYLATION
5bnj:A (LEU104) to (ASP173) CDK8/CYCC IN COMPLEX WITH 8-{3-CHLORO-5-[4-(1-METHYL-1H-PYRAZOL-4-YL)- PHENYL]-PYRIDIN- 4-YL}-2,8-DIAZA-SPIRO[4.5]DECAN-1-ONE | CDK8 KINASE / CYCLIN C, TRANSFERASE
3zhp:C (SER106) to (LEU160) HUMAN MST3 (STK24) IN COMPLEX WITH MO25BETA | CELL CYCLE, MO25,
3zhp:D (SER106) to (LEU160) HUMAN MST3 (STK24) IN COMPLEX WITH MO25BETA | CELL CYCLE, MO25,
4neu:A (LEU100) to (ILE154) X-RAY STRUCTURE OF RECEPTOR INTERACTING PROTEIN 1 (RIP1)KINASE DOMAIN WITH A 1-AMINOISOQUINOLINE INHIBITOR | KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
5bx0:A (SER150) to (LYS205) AN AUTOMATED MICROSCALE THERMOPHORESIS SCREENING APPROACH FOR FRAGMENT-BASED LEAD DISCOVERY | FRAGMENT SCREENING, MICROSCALE THERMOPHORESIS, TRANSFERASE
3zls:A (SER150) to (LEU206) CRYSTAL STRUCTURE OF MEK1 IN COMPLEX WITH FRAGMENT 6 | TRANSFERASE
3zlw:A (SER150) to (LEU206) CRYSTAL STRUCTURE OF MEK1 IN COMPLEX WITH FRAGMENT 3 | TRANSFERASE
3zly:A (SER150) to (LYS205) CRYSTAL STRUCTURE OF MEK1 IN COMPLEX WITH FRAGMENT 8 | TRANSFERASE
5c01:A (LEU695) to (LEU757) CRYSTAL STRUCTURE OF KINASE | PSEUDOKINASE DOMAIN, TRANSFERASE
5c01:B (LEU695) to (LEU757) CRYSTAL STRUCTURE OF KINASE | PSEUDOKINASE DOMAIN, TRANSFERASE
5c03:A (ASP696) to (LEU757) CRYSTAL STRUCTURE OF KINASE | PSEUDOKINASE DOMAIN, TRANSFERASE
5c03:B (LEU695) to (LEU757) CRYSTAL STRUCTURE OF KINASE | PSEUDOKINASE DOMAIN, TRANSFERASE
3zon:A (ASP696) to (ASP759) HUMAN TYK2 PSEUDOKINASE DOMAIN BOUND TO A KINASE INHIBITOR | TRANSFERASE, JAK
1kre:B (HIS329) to (SER401) STRUCTURE OF P. CITRINUM ALPHA 1,2-MANNOSIDASE REVEALS THE BASIS FOR DIFFERENCES IN SPECIFICITY OF THE ER AND GOLGI CLASS I ENZYMES | (ALPHA/ALPHA)7-BARREL, HYDROLASE
2no3:B (LEU115) to (ILE167) NOVEL 4-ANILINOPYRIMIDINES AS POTENT JNK1 INHIBITORS | JNK1, C-JUN N-TERMINAL KINASE, JNK1 INHIBITORS, ANILINOPYRIMIDINES JNK1 INHIBITORS, SIGNALING PROTEIN/INHIBITOR COMPLEX
4o0s:A (VAL218) to (ALA273) CRYSTAL STRUCTURES OF HUMAN KINASE AURORA A | PROTEIN KINASE, TRANSFERASE
4o0u:A (VAL218) to (ILE272) CRYSTAL STRUCTURES OF HUMAN KINASE AURORA A | PROTEIN KINASE AURORA A, PROTEIN KINASE, TRANSFERASE
3zzw:B (LEU561) to (ILE631) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF ROR2 | TRANSFERASE, NEUROTROPHIC TYROSINE KINASE, RECEPTOR-RELATED 2, ROR2, NTRKR2, KINASE, STRUCTURAL GENOMICS CONSORTIUM, SGC
5cen:A (GLN197) to (SER253) CRYSTAL STRUCTURE OF DLK (KINASE DOMAIN) | KINASE, TRANSFERASE
5ceo:A (GLN197) to (ASP254) DLK IN COMPLEX WITH INHIBITOR 2-((6-(3,3-DIFLUOROPYRROLIDIN-1-YL)-4- (1-(OXETAN-3-YL)PIPERIDIN-4-YL)PYRIDIN-2-YL)AMINO)ISONICOTINONITRILE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ceq:A (LEU198) to (SER253) DLK IN COMPLEX WITH INHIBITOR 2-((1-CYCLOPENTYL-5-(1-(OXETAN-3-YL) PIPERIDIN-4-YL)-1H-PYRAZOL-3-YL)AMINO)ISONICOTINONITRILE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3jxw:A (ASP128) to (LEU184) DISCOVERY OF 3H-BENZO[4,5]THIENO[3,2-D]PYRIMIDIN-4-ONES AS POTENT, HIGHLY SELECTIVE AND ORALLY BIOAVAILABLE PIM KINASES INHIBITORS | PIM-1, ALTERNATIVE INITIATION, ATP-BINDING, CELL MEMBRANE, CYTOPLASM, KINASE, MANGANESE, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
4obp:B (SER112) to (LEU169) MAP4K4 IN COMPLEX WITH INHIBITOR (COMPOUND 29), 6-(2-FLUOROPYRIDIN-4- YL)PYRIDO[3,2-D]PYRIMIDIN-4-AMINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4obq:A (SER112) to (ASP171) MAP4K4 IN COMPLEX WITH INHIBITOR (COMPOUND 31), N-[3-(4- AMINOQUINAZOLIN-6-YL)-5-FLUOROPHENYL]-2-(PYRROLIDIN-1-YL)ACETAMIDE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4obq:B (SER112) to (LEU169) MAP4K4 IN COMPLEX WITH INHIBITOR (COMPOUND 31), N-[3-(4- AMINOQUINAZOLIN-6-YL)-5-FLUOROPHENYL]-2-(PYRROLIDIN-1-YL)ACETAMIDE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2z7r:A (LEU149) to (ASP205) CRYSTAL STRUCTURE OF THE N-TERMINAL KINASE DOMAIN OF HUMAN RSK1 BOUND TO STAUROSPORINE | PROTEIN KINASE, CANCER, KINASE INHIBITOR, ATP-BINDING, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2z7s:A (LEU149) to (ASP205) CRYSTAL STRUCTURE OF THE N-TERMINAL KINASE DOMAIN OF HUMAN RSK1 BOUND TO PURVALNOL A | PROTEIN KINASE, CANCER, KINASE INHIBITOR, TRANSFERASE
1xwq:A (THR77) to (ASP138) STRUCTURE OF A COLD-ADAPTED FAMILY 8 XYLANASE | HYDROLASE, XYLAN DEGRADATION, PSYCHROPHILIC, COLD ADAPTATION, TEMPERATURE, GLYCOSYL HYDROLASE, FAMILY 8
4p69:A (PRO421) to (PHE473) ACEK (D477A) ICDH COMPLEX | TRANSFERASE, HYDROLASE-OXIDOREDUCTASE COMPLEX
4p69:B (LEU422) to (ASP475) ACEK (D477A) ICDH COMPLEX | TRANSFERASE, HYDROLASE-OXIDOREDUCTASE COMPLEX
1y91:A (LYS88) to (LEU143) CRYSTAL STRUCTURE OF HUMAN CDK2 COMPLEXED WITH A PYRAZOLO[1, 5-A]PYRIMIDINE INHIBITOR | SERINE/THREONINE PROTEIN KINASE, CDK2, ATP-BINDING, CELL CYCLE, MITOSIS, PHOSPHORYLATION, PYRAZOLOPYRIMIDINE INHIBITOR, TRANSFERASE
5d7v:A (SER271) to (VAL328) CRYSTAL STRUCTURE OF PTK6 KINASE DOMAIN | TRANSFERASE, KINASE, BRK, APO
5d7v:C (SER271) to (VAL328) CRYSTAL STRUCTURE OF PTK6 KINASE DOMAIN | TRANSFERASE, KINASE, BRK, APO
5d7v:D (LEU272) to (VAL328) CRYSTAL STRUCTURE OF PTK6 KINASE DOMAIN | TRANSFERASE, KINASE, BRK, APO
5d9h:A (MET158) to (ILE220) CRYSTAL STRUCTURE OF SPAK (STK39) DIMER IN THE BASAL ACTIVITY STATE | KINASE, STE20, HYPERTENSION, STK39, TRANSFERASE
3ktb:B (GLN53) to (GLN86) CRYSTAL STRUCTURE OF ARSENICAL RESISTANCE OPERON TRANS-ACTING REPRESSOR FROM BACTEROIDES VULGATUS ATCC 8482 | ALPHA-BETA-ALPHA SANDWICH, HELIX-TURN-HELIX, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSCRIPTION REGULATOR
3ktb:D (GLN53) to (GLN86) CRYSTAL STRUCTURE OF ARSENICAL RESISTANCE OPERON TRANS-ACTING REPRESSOR FROM BACTEROIDES VULGATUS ATCC 8482 | ALPHA-BETA-ALPHA SANDWICH, HELIX-TURN-HELIX, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSCRIPTION REGULATOR
1ykr:A (LEU87) to (LEU143) CRYSTAL STRUCTURE OF CDK2 WITH AN AMINOIMIDAZO PYRIDINE INHIBITOR | CELL CYCLE DIVISION PROTEIN KINASE 2, CDK2, TRANSFERASE
5de2:A (LEU119) to (GLY178) STRUCTURAL MECHANISM OF NEK7 ACTIVATION BY NEK9-INDUCED DIMERISATION | PROTEIN KINASE, MITOSIS, PROTEIN-PROTEIN INTERACTION, TRANSFERASE
5de2:B (LEU119) to (GLY178) STRUCTURAL MECHANISM OF NEK7 ACTIVATION BY NEK9-INDUCED DIMERISATION | PROTEIN KINASE, MITOSIS, PROTEIN-PROTEIN INTERACTION, TRANSFERASE
5di1:A (SER112) to (ASP171) MAP4K4 IN COMPLEX WITH AN INHIBITOR | KINASE, INHIBITOR, COMPLEX, MEDICINAL CHEMISTRY, TRANSFERASE- INHIBITOR COMPLEX
3le6:A (LEU87) to (LEU143) THE STRUCTURE OF CYCLIN DEPENDENT KINASE 2 (CKD2) WITH A PYRAZOLOBENZODIAZEPINE INHIBITOR | CYCLIN-DEPENDENT KINASE 2 DRUG DESIGN, ATP-BINDING, CELL CYCLE, CELL DIVISION, KINASE, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5dqo:D (PRO286) to (HIS351) CRYSTAL STRUCTURE OF Y347F MUTANT OF HUMAN PRIMASE P58 IRON-SULFUR CLUSTER DOMAIN | IRON-SULFUR CLUSTER, DNA PRIMING, REPLICATION
4aoi:A (LEU1165) to (VAL1220) CRYSTAL STRUCTURE OF C-MET KINASE DOMAIN IN COMPLEX WITH 4-( 3-((1H- PYRROLO(2,3-B)PYRIDIN-3-YL)METHYL)-(1,2,4)TRIAZOLO( 4,3-B)(1,2,4) TRIAZIN-6-YL)BENZONITRILE | TRANSFERASE, KINASE INHIBITOR
4q2a:A (THR308) to (ASP368) WNK1: A CHLORIDE SENSOR VIA AUTOPHOSPHORYLATION | PROTEIN SERINE/THREONINE KINASE, KINASE, ATP-BINDING, UNPHOSPHORYLATED, TRANSFERASE
1zy4:B (THR795) to (GLY852) CRYSTAL STRUCTURE OF EIF2ALPHA PROTEIN KINASE GCN2: R794G HYPERACTIVATING MUTANT IN APO FORM. | TRANSLATION REGULATOR, PROTEIN KINASE, SIGNAL TRANSDUCTION, AMINO- ACID STARVATION, STARVATION STRESS RESPONSE, EIF2ALPHA KINASE, TRANSFERASE
4azv:A (LEU316) to (ASP369) CO-CRYSTAL STRUCTURE OF WBDD AND KINASE INHIBITOR GW435821X. | TRANSFERASE, METHYLTRANSFERASE
4b0g:A (THR217) to (ASP274) COMPLEX OF AURORA-A BOUND TO AN IMIDAZOPYRIDINE-BASED INHIBITOR | TRANSFERASE, MITOSIS
3lzb:A (LEU774) to (ASP831) EGFR KINASE DOMAIN COMPLEXED WITH AN IMIDAZO[2,1-B]THIAZOLE INHIBITOR | EPIDERMAL GROWTH FACTOR KINASE DOMAIN, MULTITARGETED SMALL MOLECULE KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3lzb:B (LEU774) to (ILE829) EGFR KINASE DOMAIN COMPLEXED WITH AN IMIDAZO[2,1-B]THIAZOLE INHIBITOR | EPIDERMAL GROWTH FACTOR KINASE DOMAIN, MULTITARGETED SMALL MOLECULE KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3lzb:C (LEU774) to (ILE829) EGFR KINASE DOMAIN COMPLEXED WITH AN IMIDAZO[2,1-B]THIAZOLE INHIBITOR | EPIDERMAL GROWTH FACTOR KINASE DOMAIN, MULTITARGETED SMALL MOLECULE KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3lzb:D (LEU774) to (ASP831) EGFR KINASE DOMAIN COMPLEXED WITH AN IMIDAZO[2,1-B]THIAZOLE INHIBITOR | EPIDERMAL GROWTH FACTOR KINASE DOMAIN, MULTITARGETED SMALL MOLECULE KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3mbl:A (SER150) to (LEU206) CRYSTAL STRUCTURE OF THE HUMAN MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1 (MEK 1) IN COMPLEX WITH LIGAND AND MGADP | KINASE INHIBITOR, TRANSFERASE
4bbm:B (ILE87) to (ASP144) CRYSTAL STRUCTURE OF THE HUMAN CDKL2 KINASE DOMAIN WITH BOUND TCS 2312 | TRANSFERASE, PHOSPHO-MIMETIC
3bbw:A (LEU779) to (ILE834) CRYSTAL STRUCTURE OF THE ERBB4 KINASE IN ITS INACTIVE CONFORMATION | INACTIVE KINASE CONFORMATION, ALTERNATIVE SPLICING, ATP- BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
3bel:A (LEU798) to (ILE853) X-RAY STRUCTURE OF EGFR IN COMPLEX WITH OXIME INHIBITOR | KINASE DOMAIN, ALTERNATIVE SPLICING, ANTI-ONCOGENE, ATP- BINDING, CELL CYCLE, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE, UBL CONJUGATION
4qu3:A (THR195) to (ILE241) GES-2 ERTAPENEM ACYL-ENZYME COMPLEX | ANTIBIOTIC RESISTANCE, BETA-LACTAMASE, HYDROLASE, ERTAPENEM, HYDROLASE-ANTIBIOTIC COMPLEX
4qu3:B (THR195) to (ILE241) GES-2 ERTAPENEM ACYL-ENZYME COMPLEX | ANTIBIOTIC RESISTANCE, BETA-LACTAMASE, HYDROLASE, ERTAPENEM, HYDROLASE-ANTIBIOTIC COMPLEX
5ew9:A (VAL218) to (ASP274) CRYSTAL STRUCTURE OF AURORA A KINASE DOMAIN BOUND TO MK-5108 | TRANSFERASE, PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4bn1:A (VAL218) to (ILE272) CRYSTAL STRUCTURE OF V174M MUTANT OF AURORA-A KINASE | TRANSFERASE, PROTEIN KINASE, MITOSIS
3ccn:A (LEU1165) to (VAL1220) X-RAY STRUCTURE OF C-MET WITH TRIAZOLOPYRIDAZINE INHIBITOR. | C-MET KINASE TRIAZOLOPYRIDAZINE, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO- ONCOGENE, RECEPTOR, TRANSFERASE, TRANSMEMBRANE, TYROSINE- PROTEIN KINASE
3nfd:A (SER36) to (GLY117) CHRONOBACTERIUM AMMONIAGENES ACPS-COA COMPLEX | ACYL CARRIER PROTEIN SYNTHASE, MYCOBACTERIUM TUBERCULOSIS, ACYL CARRIER PROTEIN, FATTY ACID SYNTHASE, TRANSFERASE
3nfd:B (SER36) to (GLY117) CHRONOBACTERIUM AMMONIAGENES ACPS-COA COMPLEX | ACYL CARRIER PROTEIN SYNTHASE, MYCOBACTERIUM TUBERCULOSIS, ACYL CARRIER PROTEIN, FATTY ACID SYNTHASE, TRANSFERASE
3nfd:C (SER36) to (GLY117) CHRONOBACTERIUM AMMONIAGENES ACPS-COA COMPLEX | ACYL CARRIER PROTEIN SYNTHASE, MYCOBACTERIUM TUBERCULOSIS, ACYL CARRIER PROTEIN, FATTY ACID SYNTHASE, TRANSFERASE
3nfd:D (SER36) to (GLY117) CHRONOBACTERIUM AMMONIAGENES ACPS-COA COMPLEX | ACYL CARRIER PROTEIN SYNTHASE, MYCOBACTERIUM TUBERCULOSIS, ACYL CARRIER PROTEIN, FATTY ACID SYNTHASE, TRANSFERASE
3nfd:E (SER36) to (GLY117) CHRONOBACTERIUM AMMONIAGENES ACPS-COA COMPLEX | ACYL CARRIER PROTEIN SYNTHASE, MYCOBACTERIUM TUBERCULOSIS, ACYL CARRIER PROTEIN, FATTY ACID SYNTHASE, TRANSFERASE
3nfd:F (SER36) to (GLY117) CHRONOBACTERIUM AMMONIAGENES ACPS-COA COMPLEX | ACYL CARRIER PROTEIN SYNTHASE, MYCOBACTERIUM TUBERCULOSIS, ACYL CARRIER PROTEIN, FATTY ACID SYNTHASE, TRANSFERASE
4c3r:A (VAL218) to (ASP274) STRUCTURE OF DEPHOSPHORYLATED AURORA A (122-403) BOUND TO AMPPCP | TRANSFERASE, AURORA A, ACTIVATION, CELL CYCLE, CANCER
3cth:A (ASP1164) to (ALA1221) CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF THE HEPATOCYTE GROWTH FACTOR RECEPTOR C-MET IN COMPLEX WITH A AMINOPYRIDINE BASED INHIBITOR | RECEPTOR TYROSINE KINASE, SIGNAL TRANSDUCTION, GRB2, SHC, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
5fwk:K (ASP99) to (ALA157) ATOMIC CRYOEM STRUCTURE OF HSP90-CDC37-CDK4 COMPLEX | SIGNALING PROTEIN, HSP90, CDC37, CDK4, CHAPERONE, KINASE, UNFOLDING
5fwl:K (ASP99) to (LEU156) ATOMIC CRYOEM STRUCTURE OF HSP90-CDC37-CDK4 COMPLEX | HSP90, CDC37, CDK4, CHAPERONE, KINASE, UNFOLDING
5fwm:K (ASP99) to (ALA157) ATOMIC CRYOEM STRUCTURE OF HSP90-CDC37-CDK4 COMPLEX | HSP90, CDC37, CDK4, CHAPERONE, KINASE, UNFOLDING
5fwp:K (ASP99) to (LEU156) ATOMIC CRYOEM STRUCTURE OF HSP90-CDC37-CDK4 COMPLEX | HSP90, CDC37, CDK4, CHAPERONE, KINASE, UNFOLDING
3o17:A (ASN114) to (ILE167) CRYSTAL STRUCTURE OF JNK1-ALPHA1 ISOFORM | KINASE, SERINE THREONINE PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
3o17:B (LEU115) to (GLY171) CRYSTAL STRUCTURE OF JNK1-ALPHA1 ISOFORM | KINASE, SERINE THREONINE PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
3o50:B (TYR219) to (ASP274) CRYSTAL STRUCTURE OF BENZAMIDE 9 BOUND TO AURORAA | AURORAA, KINASE DOMAIN, TRANSFERASE
3dae:A (GLU138) to (ASP195) CRYSTAL STRUCTURE OF PHOSPHORYLATED SNF1 KINASE DOMAIN | KINASE, AMPK, SNF1, ATP-BINDING, CARBOHYDRATE METABOLISM, MEMBRANE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3dae:B (GLU138) to (ASP195) CRYSTAL STRUCTURE OF PHOSPHORYLATED SNF1 KINASE DOMAIN | KINASE, AMPK, SNF1, ATP-BINDING, CARBOHYDRATE METABOLISM, MEMBRANE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
3daj:A (VAL218) to (ASP274) CRYSTAL STRUCTURE OF AURORA A COMPLEXED WITH AN INHIBITOR DISCOVERED THROUGH SITE-DIRECTED DYNAMIC TETHERING | PROTEIN-SMALL MOLECULE INHIBITOR COMPLEX, KINASE, TRANSFERASE
5gop:A (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 COMPLEXED WITH SUCROSE | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
5gop:B (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 COMPLEXED WITH SUCROSE | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
5gop:C (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 COMPLEXED WITH SUCROSE | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
5goq:A (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 COMPLEXED WITH GLUCOSE | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
5goq:B (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 COMPLEXED WITH GLUCOSE | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
5goq:C (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 COMPLEXED WITH GLUCOSE | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
5gor:A (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
5gor:B (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
5gor:C (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
5gor:D (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
5gor:E (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
5gor:F (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
3orn:A (LEU151) to (LEU206) MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1 (MEK1) IN COMPLEX WITH CH4987655 AND MGAMP-PNP | KINASE, KINASE INHIBITOR, ALLOSTERIC, MITOGEN-ACTIVATED PROTEIN KINASE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5hbh:A (ASP103) to (ASP173) CDK8-CYCC IN COMPLEX WITH 5-{5-CHLORO-4-[1-(2-METHOXY-ETHYL)-1,8- DIAZA-SPIRO[4.5]DEC-8-YL]-PYRIDIN-3-YL}-1-METHYL-1,3-DIHYDRO- BENZO[C]ISOTHIAZOLE 2,2-DIOXIDE | CDK8 KINASE / CYCLIN C, TRANSFERASE
4u3y:B (SER112) to (LEU169) APO MITOGEN-ACTIVATED PROTEIN KINASE KINASE KINASE KINASE 4 (MAP4K4) | KINASE, TRANSFERASE
4u3z:B (SER112) to (LEU169) APO MAP4K4 T181E PHOSPHOMIMETIC MUTANT | KINASE, TRANSFERASE
4u40:B (ILE113) to (LEU169) MITOGEN-ACTIVATED PROTEIN KINASE KINASE KINASE KINASE 4 (MAP4K4) BOUND TO AMPPNP | KINASE, TRANSFERASE
4u41:B (SER112) to (LEU169) MAP4K4 BOUND TO INHIBITOR COMPOUND 1 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4u43:B (SER112) to (LEU169) MAP4K4 IN COMPLEX WITH INHIBITOR (COMPOUND 6) | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4u44:B (SER112) to (LEU169) MAP4K4 IN COMPLEX WITH INHIBITOR (COMPOUND 16) | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4u45:B (ILE113) to (LEU169) MAP4K4 IN COMPLEX WITH INHIBITOR (COMPOUND 25) | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3dy7:A (LEU151) to (LEU206) X-RAY STRUCTURE OF THE HUMAN MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1 (MEK1) IN A COMPLEX WITH LIGAND AND MGATP | DUAL SPECIFICITY PROTEIN KINASE, NON-ATP-COMPETITIVE KINASE INHIBITOR, INHIBITOR-BOUND PROTEIN KINASE, ATP-BOUND PROTEIN KINASE, ACETYLATION, ATP-BINDING, DISEASE MUTATION, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE- PROTEIN KINASE, TRANSFERASE, TYROSINE-PROTEIN KINASE
4u81:A (LEU151) to (LEU206) MEK1 KINASE BOUND TO SMALL MOLECULE INHIBITOR G659 | KINASE, COMPLEX, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4u80:A (SER150) to (LEU206) MEK 1 KINASE BOUND TO G799 | KINASE, INHIBITOR, COMPLEX
5hlw:A (ASP1164) to (VAL1220) CRYSTAL STRUCTURE OF C-MET MUTANT Y1230H IN COMPLEX WITH COMPOUND 14 | TRANSFERASE, TRANSFERASE INHIBITOR
5ho6:A (LEU1165) to (ALA1221) CRYSTAL STRUCTURE OF CMET IN COMPLEX WITH CMPD. | TRANSFERASE
5hoa:A (ASP1164) to (VAL1220) CRYSTAL STRUCTURE OF C-MET L1195V IN COMPLEX WITH SAR125844 | TRANSFERASE, INHIBITOR
5hvy:A (HIS106) to (ILE171) CDK8/CYCC IN COMPLEX WITH COMPOUND 20 | TRANSFERASE-TRANSCRIPTION COMPLEX
3pgq:A (ALA1632) to (THR1692) CRYSTAL STRUCTURE OF THE CARBOXYLTRANSFERASE DOMAIN OF S. CEREVISIAE ACETYL COA CARBOXYLASE IN COMPLEX WITH PINOXADEN | TRANSFERASE, CARBOXYLTRANSFERASE, LIGASE
3phf:A (GLU522) to (SER555) CRYSTAL STRUCTURE OF THE EPSTEIN-BARR VIRUS GH AND GL COMPLEX | VIRUS ENTRY, MEMBRANE FUSION, GLYCOPROTEIN, VIRAL PROTEIN
3phf:C (ASP523) to (SER555) CRYSTAL STRUCTURE OF THE EPSTEIN-BARR VIRUS GH AND GL COMPLEX | VIRUS ENTRY, MEMBRANE FUSION, GLYCOPROTEIN, VIRAL PROTEIN
3phf:G (ASP523) to (SER555) CRYSTAL STRUCTURE OF THE EPSTEIN-BARR VIRUS GH AND GL COMPLEX | VIRUS ENTRY, MEMBRANE FUSION, GLYCOPROTEIN, VIRAL PROTEIN
3phf:I (GLU522) to (SER555) CRYSTAL STRUCTURE OF THE EPSTEIN-BARR VIRUS GH AND GL COMPLEX | VIRUS ENTRY, MEMBRANE FUSION, GLYCOPROTEIN, VIRAL PROTEIN
3phf:K (ASP523) to (SER555) CRYSTAL STRUCTURE OF THE EPSTEIN-BARR VIRUS GH AND GL COMPLEX | VIRUS ENTRY, MEMBRANE FUSION, GLYCOPROTEIN, VIRAL PROTEIN
3phf:Q (ASP523) to (SER555) CRYSTAL STRUCTURE OF THE EPSTEIN-BARR VIRUS GH AND GL COMPLEX | VIRUS ENTRY, MEMBRANE FUSION, GLYCOPROTEIN, VIRAL PROTEIN
3phf:S (GLU522) to (SER555) CRYSTAL STRUCTURE OF THE EPSTEIN-BARR VIRUS GH AND GL COMPLEX | VIRUS ENTRY, MEMBRANE FUSION, GLYCOPROTEIN, VIRAL PROTEIN
3phf:W (GLU522) to (SER555) CRYSTAL STRUCTURE OF THE EPSTEIN-BARR VIRUS GH AND GL COMPLEX | VIRUS ENTRY, MEMBRANE FUSION, GLYCOPROTEIN, VIRAL PROTEIN
3phf:Y (GLU522) to (SER555) CRYSTAL STRUCTURE OF THE EPSTEIN-BARR VIRUS GH AND GL COMPLEX | VIRUS ENTRY, MEMBRANE FUSION, GLYCOPROTEIN, VIRAL PROTEIN
3phf:1 (ASP523) to (SER555) CRYSTAL STRUCTURE OF THE EPSTEIN-BARR VIRUS GH AND GL COMPLEX | VIRUS ENTRY, MEMBRANE FUSION, GLYCOPROTEIN, VIRAL PROTEIN
3phf:3 (GLU522) to (SER555) CRYSTAL STRUCTURE OF THE EPSTEIN-BARR VIRUS GH AND GL COMPLEX | VIRUS ENTRY, MEMBRANE FUSION, GLYCOPROTEIN, VIRAL PROTEIN
4dxe:B (THR31) to (TYR92) 2.52 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE ACYL-CARRIER-PROTEIN SYNTHASE (ACPS)-ACYL CARRIER PROTEIN (ACP) PROTEIN-PROTEIN COMPLEX FROM STAPHYLOCOCCUS AUREUS SUBSP. AUREUS COL | ACYL-CARRIER-PROTEIN SYNTHASE, ACYL CARRIER PROTEIN, TYPE II FATTY ACID SYNTHESIS PATHWAY, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES (CSGID), TRANSFERASE
4e57:B (GLY313) to (VAL360) CRYSTAL STRUCTURE OF SPACER 6AA-SHORTENED CEPHALOSPORIN ACYLASE MUTANT | CEPHALOSPORIN ACYLASE, SPACER, AUTOCLEAVAGE, HYDROLASE, GLUTARYL-7- AMINOCEPHALOSPORANIC-ACID ACYLASE, N-TERMINAL NUCLEOPHILE (NTN) HYDROLASE SUPERFAMILY
3pxi:A (THR744) to (ALA807) STRUCTURE OF MECA108:CLPC | CLPB, PROTEOLYSIS, CLPC, CLPX, HSP100/CLP, AAA+ PROTEINS, PROTEIN BINDING
3pxi:B (THR744) to (ALA807) STRUCTURE OF MECA108:CLPC | CLPB, PROTEOLYSIS, CLPC, CLPX, HSP100/CLP, AAA+ PROTEINS, PROTEIN BINDING
3pxi:C (THR744) to (ALA807) STRUCTURE OF MECA108:CLPC | CLPB, PROTEOLYSIS, CLPC, CLPX, HSP100/CLP, AAA+ PROTEINS, PROTEIN BINDING
4ek4:A (LYS88) to (LEU143) CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH AMINOPYRAZOLE INHIBITOR | ALPHA AND BETA PROTEIN (A+B), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ez5:A (LEU105) to (ASP163) CDK6 (MONOMERIC) IN COMPLEX WITH INHIBITOR | PROTEIN KINASE, ATP BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4f70:A (LEU104) to (ASP173) CRYSTAL STRUCTURE OF HUMAN CDK8/CYCC IN COMPLEX WITH COMPOUND 4 (1-[3- TERT-BUTYL-1-(4-METHYLPHENYL)-1H-PYRAZOL-5-YL]-3-[2-(MORPHOLIN-4-YL) ETHYL]UREA) | PROTEIN KINASE COMPLEX, PROTEROS, TRANSFERASE-TRANSCRIPTION-INHIBITOR COMPLEX
4f7j:A (LEU104) to (ALA172) CRYSTAL STRUCTURE OF HUMAN CDK8/CYCC IN COMPLEX WITH COMPOUND 3 (1-[3- TERT-BUTYL-1-(4-METHYLPHENYL)-1H-PYRAZOL-5-YL]-3-(2-HYDROXYETHYL) UREA) | PROTEIN KINASE COMPLEX, PROTEROS, TRANSFERASE-TRANSCRIPTION-INHIBITOR COMPLEX
3qmn:A (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:B (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:C (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:D (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:E (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:F (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:G (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:H (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:I (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:J (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:K (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:L (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:M (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:N (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:O (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:P (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:Q (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:R (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:S (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:T (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:U (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:V (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:W (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
3qmn:X (THR32) to (LEU90) CRYSTAL STRUCTURE OF 4'-PHOSPHOPANTETHEINYL TRANSFERASE ACPS FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA SANDWICH, TRANSFERASE, ACYL CARRIER PROTEIN, CYTOSOL
4ux9:A (LEU115) to (ILE167) CRYSTAL STRUCTURE OF JNK1 BOUND TO A MKK7 DOCKING MOTIF | TRANSFERASE, JNK1, INTRINSICALLY DISORDERED DOMAINS, MKK7
4ux9:B (LEU115) to (GLY171) CRYSTAL STRUCTURE OF JNK1 BOUND TO A MKK7 DOCKING MOTIF | TRANSFERASE, JNK1, INTRINSICALLY DISORDERED DOMAINS, MKK7
4ux9:D (LEU115) to (ILE167) CRYSTAL STRUCTURE OF JNK1 BOUND TO A MKK7 DOCKING MOTIF | TRANSFERASE, JNK1, INTRINSICALLY DISORDERED DOMAINS, MKK7
4v1a:c (GLU219) to (VAL260) STRUCTURE OF THE LARGE SUBUNIT OF THE MAMMALIAN MITOCHONDRIAL RIBOSOME, PART 2 OF 2 | RIBOSOME, TRANSLATION, LARGE RIBOSOMAL SUBUNIT, MITORIBOSOME, MAMMALIAN MITOCHONDRIAL RIBOSOME, CRYO-EM
3qql:A (LEU87) to (LEU143) CDK2 IN COMPLEX WITH INHIBITOR L3 | PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qrt:A (LEU87) to (LEU143) CDK2 IN COMPLEX WITH INHIBITOR NSK-MC2-55 | PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ff8:A (LEU601) to (VAL661) INHIBITOR BOUND STRUCTURE OF THE KINASE DOMAIN OF THE MURINE RECEPTOR TYROSINE KINASE TYRO3 (SKY) | RECEPTOR PROTEIN TYROSINE KINASE, PHOSPHOTRANSFERASE, GAS6 (LIGAND), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fkp:A (LEU87) to (LEU143) CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH OXINDOLE INHIBITOR | ALPHA AND BETA PROTEIN (A+B), TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fkv:A (LEU87) to (LEU143) CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH OXINDOLE INHIBITOR | ALPHA AND BETA PROTEIN (A+B), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5j9q:I (ASP240) to (GLY288) CRYSTAL STRUCTURE OF THE NUA4 CORE COMPLEX | NUA4, NUCLEOSOME, HISTONE, ACETYLATION, TRANSFERASE
3r7u:A (LEU87) to (LEU143) CDK2 IN COMPLEX WITH INHIBITOR KVR-1-75 | PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r9n:A (LEU87) to (LEU143) CDK2 IN COMPLEX WITH INHIBITOR RC-2-21 | PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3rcd:C (LEU806) to (GLY865) HER2 KINASE DOMAIN COMPLEXED WITH TAK-285 | KINASE DOMAIN, RECEPTOR, TRANSFERASE, TYROSINE-PROTEIN KINASE, TYROSINE KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, ANTI-ONCOGENE, CELL CYCLE, DISEASE, MUTATION, ATP-BINDING, NUCLEOTIDE-BINDING, GLYCOPROTEIN, PHOSPHOPROTEIN, MEMBRANE, SECRETED
3rhk:A (ASP1164) to (VAL1220) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF C-MET KINASE IN COMPLEX WITH ARQ 197 | KINASE, RECEPTOR TYROSINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5l8j:A (VAL218) to (ILE272) AURORA-A KINASE DOMAIN IN COMPLEX WITH VNAR-D01 S93R | KINASE, VNAR, INHIBITOR, TRANSFERASE
5l8k:A (VAL218) to (ASP274) AURORA-A KINASE DOMAIN IN COMPLEX WITH VNAR-D01 (CRYSTAL FORM 2) | KINASE, VNAR, INHIBITOR, TRANSFERASE
5m51:A (LEU94) to (GLY158) NEK2 BOUND TO ARYLAMINOPURINE COMPOUND 8 | PROTEIN KINASE, INHIBITOR, CENTROSOME SEPARATION, TRANSFERASE- INHIBITOR COMPLEX
1bi8:A (LEU105) to (LEU161) MECHANISM OF G1 CYCLIN DEPENDENT KINASE INHIBITION FROM THE STRUCTURES CDK6-P19INK4D INHIBITOR COMPLEX | CYCLIN DEPENDENT KINASE, CYCLIN DEPENDENT KINASE INHIBITORY PROTEIN, CDK, INK4, CELL CYCLE, COMPLEX (KINASE/INHIBITOR)
1bi8:C (LEU105) to (LEU161) MECHANISM OF G1 CYCLIN DEPENDENT KINASE INHIBITION FROM THE STRUCTURES CDK6-P19INK4D INHIBITOR COMPLEX | CYCLIN DEPENDENT KINASE, CYCLIN DEPENDENT KINASE INHIBITORY PROTEIN, CDK, INK4, CELL CYCLE, COMPLEX (KINASE/INHIBITOR)
3sqv:A (GLU489) to (CYS548) CRYSTAL STRUCTURE OF E. COLI O157:H7 E3 UBIQUITIN LIGASE, NLEL, WITH A HUMAN E2, UBCH7 | EFFECTOR PROTEIN, PENTAPEPTIDE, HECT DOMAIN, HECT E3 UBIQUITIN LIGASE, E2 UBIQUITIN CONJUGATING ENZYME, PROTEIN-PROTEIN COMPLEX, UBIQUITIN TRANSFER, UBIQUITIN, UBIQUITINATION, LIGASE-SIGNALING PROTEIN COMPLEX
3g33:A (LEU105) to (ASP163) CRYSTAL STRUCTURE OF CDK4/CYCLIN D3 | SER/THR PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, ATP-BINDING, CELL DIVISION, DISEASE MUTATION, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, CYCLIN
3g33:C (LEU105) to (ASP163) CRYSTAL STRUCTURE OF CDK4/CYCLIN D3 | SER/THR PROTEIN KINASE, CELL CYCLE, PHOSPHORYLATION, ATP-BINDING, CELL DIVISION, DISEASE MUTATION, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, CYCLIN
3gbz:A (LEU98) to (ASP159) STRUCTURE OF THE CMGC CDK KINASE FROM GIARDIA LAMBLIA | SSGCID, KINASE, CMGC CDK, ATP-BINDING, NUCLEOTIDE-BINDING, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE
2r3f:A (LYS88) to (LEU143) CRYSTAL STRUCTURE OF CYCLIN-DEPENDENT KINASE 2 WITH INHIBITOR | SERINE/THREONINE-PROTEIN KINASE, CELL CYCLE, INHIBITION, CYCLIN-DEPENDENT KINASE, CANCER, ATP-BINDING, CELL DIVISION, MITOSIS, NUCLEOTIDE-BINDING, PHOSPHORYLATION, POLYMORPHISM, TRANSFERASE
1fo3:A (ASN327) to (PRO386) CRYSTAL STRUCTURE OF HUMAN CLASS I ALPHA1,2-MANNOSIDASE IN COMPLEX WITH KIFUNENSINE | ALPHA-ALPHA7 BARREL, HYDROLASE
1g6i:A (ASN129) to (LYS195) CRYSTAL STRUCTURE OF THE YEAST ALPHA-1,2-MANNOSIDASE WITH BOUND 1- DEOXYMANNOJIRIMYCIN AT 1.59 A RESOLUTION | ALPHA-ALPHA7 BARREL, HYDROLASE
4kkg:A (LEU153) to (ASP207) CRYSTAL STRUCTURE OF APO AND AMP-BOUND JNK3 | KINASE DOMAIN, KINASE, C-JUN, TRANSFERASE
3v04:A (LEU151) to (LEU206) DISCOVERY OF NOVEL ALLOSTERIC MEK INHIBITORS POSSESSING CLASSICAL AND NON-CLASSICAL BIDENTATE SER212 INTERACTIONS. | KINASE, TRANSFERASE-INHIBITOR COMPLEX
3v5q:B (LEU625) to (ILE695) DISCOVERY OF A SELECTIVE TRK INHIBITOR WITH EFFICACY IN RODENT CANCER TUMOR MODELS | KINASE DOMAIN, KINASE, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1h14:A (THR77) to (ASP138) STRUCTURE OF A COLD-ADAPTED FAMILY 8 XYLANASE | HYDROLASE, XYLAN DEGRADATION, PSYCHROPHILIC, COLD ADAPTATION, TEMPERATURE, GLYCOSYL HYDROLASE, FAMILY 8
2kdn:A (TYR18) to (SER61) SOLUTION STRUCTURE OF PFE0790C, A PUTATIVE BOLA-LIKE PROTEIN FROM THE PROTOZOAN PARASITE PLASMODIUM FALCIPARUM. | NMR SOLUTION STRUCTURE, SSGCID, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, STRUCTURAL GENOMICS, MALARIA, UNKNOWN FUNCTION
3zlx:A (SER150) to (LEU206) CRYSTAL STRUCTURE OF MEK1 IN COMPLEX WITH FRAGMENT 18 | TRANSFERASE
5cep:A (LEU198) to (SER253) DLK IN COMPLEX WITH INHIBITOR N-(1-ISOPROPYL-5-(PIPERIDIN-4-YL)-1H- PYRAZOL-3-YL)-4-(TRIFLUOROMETHYL)PYRIDIN-2-AMINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5clr:A (ASP152) to (ASP213) CRYSTAL STRUCTURE OF LEGK4_APO KINASE | LEGIONELLA, BACTERIAL EFFECTORS, SERINE/THREONINE KINASE, TYPE IV SECRETION SYSTEM, TRANSFERASE
4otw:A (SER775) to (VAL831) HER3 PSEUDOKINASE DOMAIN BOUND TO BOSUTINIB | RECEPTOR TYROSINE KINASE, PSEUDOKINASE, BOSUTINIB, MEMBRANE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5d7a:A (VAL113) to (ASP171) CRYSTAL STRUCTURE OF THE KINASE DOMAIN OF TRAF2 AND NCK-INTERACTING PROTEIN KINASE WITH NCB-0846 | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4pds:A (LEU281) to (ILE337) CRYSTAL STRUCTURE OF RAD53 KINASE DOMAIN AND SCD2 IN COMPLEX WITH AMPPNP | KINASE DOMAIN, ANP, C-LOBE, ACTIVATION SEGMENT EXCHANGE, TRANSFERASE
4aua:A (LEU105) to (ASP163) LIGANDED X-RAY CRYSTAL STRUCTURE OF CYCLIN DEPENDENT KINASE 6 (CDK6) | TRANSFERASE
2a8z:A (THR77) to (ASP138) STRUCTURE OF A COLD-ADAPTED FAMILY 8 XYLANASE | HYDROLASE, XYLAN DEGRADATION, PSYCHROPHILIC, COLD ADAPTATION, TEMPERATURE, GLYCOSYL HYDROLASE, FAMILY 8
2ae3:B (GLY148) to (VAL195) GLUTARYL 7-AMINOCEPHALOSPORANIC ACID ACYLASE: MUTATIONAL STUDY OF ACTIVATION MECHANISM | AUTOPROTEOLYSIS, PRECURSOR ACTIVATION, INTERMEDIATE STRUCTURE, CEPHALOSPORIN ACYLASE, HYDROLASE
4bg2:A (GLY206) to (SER249) X-RAY CRYSTAL STRUCTURE OF PATF FROM PROCHLORON DIDEMNI | TRANSFERASE, PATELLAMIDE, CYANOBACTINS, NATURAL PRODUCTS, PRENYL TRANSFERASES
4bg2:B (GLY206) to (SER249) X-RAY CRYSTAL STRUCTURE OF PATF FROM PROCHLORON DIDEMNI | TRANSFERASE, PATELLAMIDE, CYANOBACTINS, NATURAL PRODUCTS, PRENYL TRANSFERASES
5eyc:A (LEU1165) to (VAL1220) CRYSTAL STRUCTURE OF C-MET IN COMPLEX WITH NAPHTHYRIDINONE INHIBITOR 5 | PHOSPHOTRANSFERASE, INHIBITOR, CANCER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5eym:A (SER150) to (LEU206) MEK1 IN COMPLEX WITH BI 847325 | KINASE, INHIBITOR, TRANSFERASE
5eym:B (SER150) to (LEU206) MEK1 IN COMPLEX WITH BI 847325 | KINASE, INHIBITOR, TRANSFERASE
3ne9:A (SER36) to (GLY117) CHRONOBACTERIUM AMMOINIAGENES APO-ACPS STRUCUTRE | ACYL CARRIER PROTEIN SYNTHASE, ACYL CARRIER PROTEIN, FATTY ACID SYNTHASE, ACPS, MYCOBACTERIUM TUBERCULOSIS STRUCTURAL PROTEOMICS PROJECT, TRANSFERASE, XMTB, STRUCTURAL GENOMICS
3nux:A (LEU105) to (ALA162) CDK6 (MONOMERIC) IN COMPLEX WITH INHIBITOR | KINASE, PROTEIN KINASE, ATP BINDING, PHOSPHORYLATION, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4rru:A (GLY180) to (SER218) MYC3 N-TERMINAL JAZ-BINDING DOMAIN[5-242] FROM ARABIDOPSIS | HELIX-SHEET-HELIX FOLD, TRANSCRIPTION FACTOR, JAZ REPRESSORS, NUCLEAR, TRANSCRIPTION REGULATOR
4rvt:B (SER112) to (VAL170) MAP4K4 IN COMPLEX WITH A PYRIDIN-2(1H)-ONE DERIVATIVE | PYRIDIN-2(1H)-ONE LIGAND, TYPE I, DFG-IN, SERINE/THREONINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4czy:B (THR359) to (LEU423) COMPLEX OF NEUROSPORA CRASSA PAN2 (WD40-CS1) WITH PAN3 (PSEUDOKINASE AND C-TERM) | GENE REGULATION, WD40 DOMAIN, PSEUDOKINASE, C-TERMINAL KNOB DOMAIN, DEADENYLATION, MRNA DECAY, PAN2-PAN3 COMPLEX
4d1x:A (LEU87) to (LEU143) CDK2 IN COMPLEX WITH LUCIFERIN | TRANSFERASE, KINASE
5goo:A (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 COMPLEXED WITH FRUCTOSE | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
5goo:B (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 COMPLEXED WITH FRUCTOSE | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
5goo:C (PHE51) to (GLY118) CRYSTAL STRUCTURE OF ALKALINE INVERTASE INVA FROM ANABAENA SP. PCC 7120 COMPLEXED WITH FRUCTOSE | ALKALINE INVERTASES, CYANOBACTERIA, GLYCOSIDE HYDROLASE FAMILY 100, SUCROSE HYDROLYSIS, HYDROLASE
4u79:A (LEU153) to (ASP207) CRYSTAL STRUCTURE OF HUMAN JNK3 IN COMPLEX WITH A BENZENESULFONAMIDE INHIBITOR. | TRANSFERASE
4umq:A (LEU94) to (ILE149) STRUCTURE OF MELK IN COMPLEX WITH INHIBITORS | TRANSFERASE, FRAGMENT BASED DRUG DESIGN
5iev:A (LEU87) to (LEU143) CRYSTAL STRUCTURE OF BAY 1000394 (RONICICLIB) BOUND TO CDK2 | ANTINEOPLASTIC AGENTS, CYCLIN-DEPENDENT KINASES, DOSE-RESPONSE RELATIONSHIP, DRUG, DRUG DISCOVERY, HELA CELLS, NEOPLASMS, PROTEIN KINASE INHIBITORS, PYRIMIDINES, STRUCTURE-ACTIVITY RELATIONSHIP, STRUCTURE-KINETICS RELATIONSHIP, SULFOXIDES, BIOPHYSICAL ASSAYS, TUMOR, TRANSFERASE
4ek5:A (LYS88) to (LEU143) CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH AMINOPYRAZOLE INHIBITOR | ALPHA AND BETA PROTEIN (A+B), TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qa8:A (LEU104) to (ILE164) CRYSTAL STRUCTURE OF INHIBITOR OF KAPPA B KINASE BETA | KINASE UBIQUITIN-LIKE DOMAIN, PHOSPHORYLATION, KINASE DOMAIN, UBIQUITIN-LIKE DOMAIN, KINASE, SUBSTRATE BINDING, IMMUNE SYSTEM, SIGNALING PROTEIN
3qa8:C (LEU104) to (ILE164) CRYSTAL STRUCTURE OF INHIBITOR OF KAPPA B KINASE BETA | KINASE UBIQUITIN-LIKE DOMAIN, PHOSPHORYLATION, KINASE DOMAIN, UBIQUITIN-LIKE DOMAIN, KINASE, SUBSTRATE BINDING, IMMUNE SYSTEM, SIGNALING PROTEIN
3qlf:A (SER345) to (VAL402) CRYSTAL STRUCTURE OF THE L317I MUTANT OF THE C-SRC TYROSINE KINASE DOMAIN COMPLEXED WITH PYRAZOLOPYRIMIDINE 5 | C-SRC L317I MUTANT, TYROSINE KINASE, TRANSFERASE, PYRAZOLOPYRIMIDINE 5
4uyn:A (VAL218) to (ASP274) SAR156497 AN EXQUISITELY SELECTIVE INHIBITOR OF AURORA KINASES | TRANSFERASE
4uzd:A (VAL218) to (ASP274) SAR156497 AN EXQUISITELY SELECTIVE INHIBITOR OF AURORA KINASES | TRANSFERASE
4uzd:B (VAL218) to (ASP274) SAR156497 AN EXQUISITELY SELECTIVE INHIBITOR OF AURORA KINASES | TRANSFERASE
4fkr:A (LEU87) to (LEU143) CRYSTAL STRUCTURE OF THE CDK2 IN COMPLEX WITH OXINDOLE INHIBITOR | ALPHA AND BETA PROTEIN (A+B), TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r7v:A (LYS88) to (LEU143) CDK2 IN COMPLEX WITH INHIBITOR KVR-1-9 | PROTEIN KINASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5l2t:A (LEU105) to (LEU161) THE X-RAY CO-CRYSTAL STRUCTURE OF HUMAN CDK6 AND RIBOCICLIB. | CYCLIN-DEPENDENT KINASE, KINASE INHIBITOR, KINASE SELECTIVITY, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX