3rqe:D (ILE117) to (THR207) CEREBRAL CAVERNOUS MALFORMATION 3 (CCM3) IN COMPLEX WITH PAXILLIN LD1 | PROTEIN-PEPTIDE COMPLEX, PROTEIN BINDING, FAT DOMAIN, DIMERIZATION, CEREBRAL CAVERNOUS MALFORMATION
2oo1:A (SER309) to (MET415) CRYSTAL STRUCTURE OF THE BROMO DOMAIN 2 OF HUMAN BROMODOMAIN CONTAINING PROTEIN 3 (BRD3) | BRD3, BROMODOMAIN CONTAINING PROTEIN 3, ORFX, RING3 LIKE GENE, RING3L, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, SIGNALING PROTEIN
2oo1:C (LYS307) to (MET415) CRYSTAL STRUCTURE OF THE BROMO DOMAIN 2 OF HUMAN BROMODOMAIN CONTAINING PROTEIN 3 (BRD3) | BRD3, BROMODOMAIN CONTAINING PROTEIN 3, ORFX, RING3 LIKE GENE, RING3L, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, SIGNALING PROTEIN
2b8i:A (TYR4) to (GLU76) CRYSTAL STRUCTURE AND FUNCTIONAL STUDIES REVEAL THAT PAS FACTOR FROM VIBRIO VULNIFICUS IS A NOVEL MEMBER OF THE SAPOSIN-FOLD FAMILY | FOUR HELIX BUNDLE, LIPID BINDING PROTEIN
4x2i:A (THR60) to (LYS160) DISCOVERY OF BENZOTRIAZOLO DIAZEPINES AS ORALLY-ACTIVE INHIBITORS OF BET BROMODOMAINS: CRYSTAL STRUCTURE OF BRD4 WITH CPI-13 | BET, CPI-13, SIGNALING PROTEIN
3s91:A (THR36) to (MET140) CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD3 IN COMPLEX WITH THE INHIBITOR JQ1 | BRD3, BROMODOMAIN CONTAINING PROTEIN 3, ORFX, RING3 LIKE GENE, RING3L, JQ1, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, UNKNOWN FUNCTION
3s92:A (SER309) to (MET415) CRYSTAL STRUCTURE OF THE SECOND BROMODOMAIN OF HUMAN BRD3 IN COMPLEX WITH THE INHIBITOR JQ1 | BRD3, BROMODOMAIN CONTAINING PROTEIN 3, ORFX, RING3 LIKE GENE, RING3L, JQ1, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, UNKNOWN FUNCTION
4hxl:A (THR60) to (LYS160) BRD4 BROMODOMAIN 1 COMPLEX WITH 3-CYCLOHEXYL-N-{3-(2-OXO-2,3-DIHYDRO- 1,3-THIAZOL-4-YL)-5-[(THIOPHEN-2-YLSULFONYL)AMINO]PHENYL}PROPANAMIDE INHIBITOR | BRD4, BROMODOMAIN, FOUR ALPHA HELICES, PROTEIN BINDING-INHIBITOR COMPLEX
4hxm:A (THR60) to (LYS160) BRD4 BROMODOMAIN 1 COMPLEX WITH N-{3-(2-OXO-2,3-DIHYDRO-1,3-THIAZOL-4- YL)-5-[(THIOPHEN-2-YLSULFONYL)AMINO]PHENYL}BUTANAMIDE INHIBITOR | BRD4, BROMODOMAIN, FOUR ALPHA HELICES, PROTEIN BINDING-INHIBITOR COMPLEX
4hxn:A (THR60) to (LYS160) BRD4 BROMODOMAIN 1 COMPLEX WITH 4-(2-FLUOROPHENYL)-1,3-THIAZOL-2(3H)- ONE INHIBITOR | BRD4, BROMODOMAIN, FOUR ALPHA HELICES, PROTEIN BINDING-INHIBITOR COMPLEX
4hxo:A (THR60) to (LYS160) BRD4 BROMODOMAIN 1 COMPLEX WITH 3-{[(3-METHYL-1,2-OXAZOL-5-YL) METHYL]SULFANYL}[1,2,4]TRIAZOLO[4,3-A]PYRIDINE INHIBITOR | BRD4, BROMODOMAIN, FOUR ALPHA HELICES, PROTEIN BINDING-INHIBITOR COMPLEX
4hxp:A (THR60) to (LYS160) BRD4 BROMODOMAIN 1 COMPLEX WITH 4-(2-OXO-1,3-OXAZOLIDIN-3-YL)BENZAMIDE INHIBITOR | BRD4, BROMODOMAIN, FOUR ALPHA HELICES, PROTEIN BINDING-INHIBITOR COMPLEX
4hxs:A (THR60) to (LYS160) BRD4 BROMODOMAIN 1 COMPLEX WITH N-[3-(2-OXO-2,3-DIHYDRO-1,3-THIAZOL-4- YL)PHENYL]-1-PHENYLMETHANESULFONAMIDE INHIBITOR | BRD4, BROMODOMAIN, FOUR ALPHA HELICES, PROTEIN BINDING-INHIBITOR COMPLEX
3fkm:X (LYS334) to (GLY438) PLASMODIUM FALCIPARUM BROMODOMAIN-CONTAINING PROTEIN PF10_0328 | BROMODOMAIN, MALARIA, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, SIGNALING PROTEIN
3svf:A (THR60) to (LEU164) CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH A DIHYDRO-QUINAZOLIN LIGAND | BROMODOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, UNKNOWN FUNCTION
3g0l:A (LYS1868) to (THR1968) CRYSTAL STRUCTURE OF HUMAN BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN 2B (BAZ2B) | BAZB2, BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN, 2B, KIAA1476, WALP4, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
4ir3:A (ASP1869) to (VAL1971) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BAZ2B IN COMPLEX WITH 1- [7-AMINO-1-(PYRIMIDIN-2-YL)INDOLIZIN-3-YL]ETHANONE (GSK2833282A) | SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSCRIPTION, BROMODOMAIN, ACETYLATED LYSINE BINDING PROTEIN, KIAA1476, WALP4
4ir5:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BAZ2B IN COMPLEX WITH 1- {1-[2-(HYDROXYMETHYL)PHENYL]-7-PHENOXYINDOLIZIN-3-YL}ETHANONE (GSK2847449A) | SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSCRIPTION, BROMODOMAIN, ACETYLATED LYSINE BINDING PROTEIN, KIAA1476, WALP4
4ir6:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BAZ2B IN COMPLEX WITH 1- {1-[2-(METHYLSULFONYL)PHENYL]-7-PHENOXYINDOLIZIN-3-YL}ETHANONE (GSK2838097A) | SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSCRIPTION, BROMODOMAIN, ACETYLATED LYSINE BINDING PROTEIN, KIAA1476, WALP4
4xua:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BAZ2B IN COMPLEX WITH E11919 BAZ2-ICR ANALOGUE | TRANSCRIPTION, BROMODOMAIN, ACETYLATED LYSINE BINDING PROTEIN, KIAA1476, WALP4, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
4xub:A (LYS1868) to (VAL1971) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BAZ2B IN COMPLEX WITH BAZ2-ICR CHEMICAL PROBE | TRANSCRIPTION, BROMODOMAIN, ACETYLATED LYSINE BINDING PROTEIN, KIAA1476, WALP4, SGC, STRUCTURAL GENOMICS CONSORTIUM
3gg3:B (ASP726) to (GLU826) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN PCAF | PCAF, K(LYSINE) ACETYLTRANSFERASE 2B, KAT2B, GCN5, GCN5L, P, P/CAF, CREBBP-ASSOCIATED FACTOR, P300/CBP-ASSOCIATED FACTOR, SGC, STRUCTURAL GENOMICS CONSORTIUM, ACYLTRANSFERASE, BROMODOMAIN, CELL CYCLE, HOST-VIRUS INTERACTION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE
4y03:B (THR624) to (GLU732) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN PB1 IN COMPLEX WITH SALICYLIC ACID | COMPLEX, SMALL MOLECULE, STRUCTURAL GENOMICS CONSORTIUM, SGC, CELL CYCLE
4j1p:A (GLY344) to (MET453) X-RAY CRYSTAL STRUCTURE OF BROMODOMAIN 2 OF HUMAN BRD2 IN COMPLEX WITH RVX208 TO 1.08 A RESOLUTION | BRD2, BROMODOMAIN, SIGNALING PROTEIN-INHIBITOR COMPLEX
4yad:A (THR901) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMODOMAIN COMPLEXED WITH 2,4- DIMETHOXY-N-(1-METHYL-2-OXO-1,2,3,4-TETRAHYDROQUINOLIN-6-YL)BENZENE- 1-SULFONAMIDE (3B) | CENTER FOR BIOMOLECULAR STRUCTURE AND FUNCTION, BROMODOMAIN, TRIM24, INHIBITOR, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
4yad:B (THR901) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMODOMAIN COMPLEXED WITH 2,4- DIMETHOXY-N-(1-METHYL-2-OXO-1,2,3,4-TETRAHYDROQUINOLIN-6-YL)BENZENE- 1-SULFONAMIDE (3B) | CENTER FOR BIOMOLECULAR STRUCTURE AND FUNCTION, BROMODOMAIN, TRIM24, INHIBITOR, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
4yat:A (THR901) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMODOMAIN COMPLEXED WITH N-(1,3- DIMETHYL-2-OXO-2,3-DIHYDRO-1H-1,3-BENZODIAZOL-5-YL)-4-METHOXYBENZENE- 1-SULFONAMIDE (5B) | CENTER FOR BIOMOLECULAR STRUCTURE AND FUNCTION, BROMODOMAIN, TRIM24, INHIBITOR, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
4yat:B (THR901) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMODOMAIN COMPLEXED WITH N-(1,3- DIMETHYL-2-OXO-2,3-DIHYDRO-1H-1,3-BENZODIAZOL-5-YL)-4-METHOXYBENZENE- 1-SULFONAMIDE (5B) | CENTER FOR BIOMOLECULAR STRUCTURE AND FUNCTION, BROMODOMAIN, TRIM24, INHIBITOR, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
4ybm:A (PRO902) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMODOMAIN COMPLEXED WITH N-{6-[3- (BENZYLOXY)PHENOXY]-1,3-DIMETHYL-2-OXO-2,3-DIHYDRO-1H-1,3- BENZODIAZOL-5-YL}-3,4-DIMETHOXYBENZENE-1-SULFONAMIDE (7B) | CENTER FOR BIOMOLECULAR STRUCTURE AND FUNCTION, BROMODOMAIN, TRIM24, INHIBITOR, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
4ybm:B (PRO902) to (LEU1004) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMODOMAIN COMPLEXED WITH N-{6-[3- (BENZYLOXY)PHENOXY]-1,3-DIMETHYL-2-OXO-2,3-DIHYDRO-1H-1,3- BENZODIAZOL-5-YL}-3,4-DIMETHOXYBENZENE-1-SULFONAMIDE (7B) | CENTER FOR BIOMOLECULAR STRUCTURE AND FUNCTION, BROMODOMAIN, TRIM24, INHIBITOR, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
4ybs:A (THR901) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMODOMAIN COMPLEXED WITH N-{1,3- DIMETHYL-6-[3-(2-METHYLPROPOXY)PHENOXY]-2-OXO-2,3-DIHYDRO-1H-1,3- BENZODIAZOL-5-YL}-1,2-DIMETHYL-1H-IMIDAZOLE-4-SULFONAMIDE (7G) | CENTER FOR BIOMOLECULAR STRUCTURE AND FUNCTION, BROMODOMAIN, TRIM24, INHIBITOR, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
4ybt:A (PRO902) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMODOMAIN COMPLEXED WITH N-{1,3- DIMETHYL-2-OXO-6-[3-(OXOLAN-3-YLMETHOXY)PHENOXY]-2,3-DIHYDRO-1H-1,3- BENZODIAZOL-5-YL}-1-METHYL-1H-IMIDAZOLE-4-SULFONAMIDE (7L) | CENTER FOR BIOMOLECULAR STRUCTURE AND FUNCTION, BROMODOMAIN, TRIM24, INHIBITOR, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
4yc9:A (PRO902) to (LEU1004) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMODOMAIN COMPLEXED WITH N-(6-{3-[4- (DIMETHYLAMINO)BUTOXY]-5-PROPOXYPHENOXY}-1,3-DIMETHYL-2-OXO-2,3- DIHYDRO-1H-1,3-BENZODIAZOL-5-YL)-3,4-DIMETHOXYBENZENE-1-SULFONAMIDE (8I) | CENTER FOR BIOMOLECULAR STRUCTURE AND FUNCTION, BROMODOMAIN, TRIM24, INHIBITOR, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
1eqf:A (ASP1380) to (LYS1484) CRYSTAL STRUCTURE OF THE DOUBLE BROMODOMAIN MODULE FROM HUMAN TAFII250 | FOUR-HELIX BUNDLE, ACETYLATED HISTONE-TAIL BINDING PROTEIN, TRANSCRIPTION
1eqf:A (ASP1502) to (TYR1607) CRYSTAL STRUCTURE OF THE DOUBLE BROMODOMAIN MODULE FROM HUMAN TAFII250 | FOUR-HELIX BUNDLE, ACETYLATED HISTONE-TAIL BINDING PROTEIN, TRANSCRIPTION
3tvi:L (ILE50) to (ARG114) CRYSTAL STRUCTURE OF CLOSTRIDIUM ACETOBUTYLICUM ASPARTATE KINASE (CAAK): AN IMPORTANT ALLOSTERIC ENZYME FOR INDUSTRIAL AMINO ACIDS PRODUCTION | STRUCTURAL GENOMICS, ACT DOMAINS, REGULATORY DOMAINS, KINASE, TRANSFERASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
2e3k:C (LEU350) to (MET453) CRYSTAL STRUCTURE OF THE HUMAN BRD2 SECOND BROMODOMAIN IN COMPLEXED WITH THE ACETYLATED HISTONE H4 PEPTIDE | BROMODOMAIN, BINDS TO ACETYLATED HISTONE TAILS, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, TRANSCRIPTION
2e3k:D (GLN349) to (MET453) CRYSTAL STRUCTURE OF THE HUMAN BRD2 SECOND BROMODOMAIN IN COMPLEXED WITH THE ACETYLATED HISTONE H4 PEPTIDE | BROMODOMAIN, BINDS TO ACETYLATED HISTONE TAILS, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, TRANSCRIPTION
4yk0:A (MET1095) to (GLU1188) CRYSTAL STRUCTURE OF THE CBP BROMODOMAIN IN COMPLEX WITH CPI098 | CBP, CPI098, TRANSFERASE
4yk0:B (MET1095) to (GLU1188) CRYSTAL STRUCTURE OF THE CBP BROMODOMAIN IN COMPLEX WITH CPI098 | CBP, CPI098, TRANSFERASE
4yk0:D (MET1095) to (GLN1187) CRYSTAL STRUCTURE OF THE CBP BROMODOMAIN IN COMPLEX WITH CPI098 | CBP, CPI098, TRANSFERASE
3u5m:A (SER959) to (SER1082) CRYSTAL STRUCTURE OF TRIM33 PHD-BROMO IN THE FREE STATE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, TRANSCRIPTION
3u5m:B (SER959) to (SER1082) CRYSTAL STRUCTURE OF TRIM33 PHD-BROMO IN THE FREE STATE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, TRANSCRIPTION
3u5m:C (SER959) to (TYR1081) CRYSTAL STRUCTURE OF TRIM33 PHD-BROMO IN THE FREE STATE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, TRANSCRIPTION
3u5m:D (SER959) to (TYR1081) CRYSTAL STRUCTURE OF TRIM33 PHD-BROMO IN THE FREE STATE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, TRANSCRIPTION
3u5m:E (SER959) to (TYR1081) CRYSTAL STRUCTURE OF TRIM33 PHD-BROMO IN THE FREE STATE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, TRANSCRIPTION
3u5m:F (SER959) to (SER1082) CRYSTAL STRUCTURE OF TRIM33 PHD-BROMO IN THE FREE STATE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, TRANSCRIPTION
3u5m:G (SER959) to (TYR1081) CRYSTAL STRUCTURE OF TRIM33 PHD-BROMO IN THE FREE STATE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, TRANSCRIPTION
3u5m:H (PRO960) to (TYR1081) CRYSTAL STRUCTURE OF TRIM33 PHD-BROMO IN THE FREE STATE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, TRANSCRIPTION
3u5m:I (SER959) to (SER1082) CRYSTAL STRUCTURE OF TRIM33 PHD-BROMO IN THE FREE STATE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, TRANSCRIPTION
3u5m:J (SER959) to (SER1082) CRYSTAL STRUCTURE OF TRIM33 PHD-BROMO IN THE FREE STATE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, TRANSCRIPTION
3u5m:K (SER959) to (SER1082) CRYSTAL STRUCTURE OF TRIM33 PHD-BROMO IN THE FREE STATE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, TRANSCRIPTION
3u5m:L (SER959) to (TYR1081) CRYSTAL STRUCTURE OF TRIM33 PHD-BROMO IN THE FREE STATE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, TRANSCRIPTION
3u5n:A (SER959) to (SER1082) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-20) K9ME3K14AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, TRANSCRIPTION
3u5n:B (SER959) to (SER1082) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-20) K9ME3K14AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, TRANSCRIPTION
3u5o:A (PRO960) to (ILE1080) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-22) K9ME3K14ACK18AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, TRANSCRIPTION
3u5o:B (PRO960) to (ILE1080) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-22) K9ME3K14ACK18AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, TRANSCRIPTION
3u5o:C (PRO960) to (ILE1080) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-22) K9ME3K14ACK18AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, TRANSCRIPTION
3u5o:D (SER959) to (ILE1080) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-22) K9ME3K14ACK18AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, TRANSCRIPTION
3u5o:E (SER959) to (ILE1080) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-22) K9ME3K14ACK18AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, TRANSCRIPTION
3u5o:F (PRO960) to (ILE1080) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-22) K9ME3K14ACK18AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, TRANSCRIPTION
3u5o:G (PRO960) to (TYR1081) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-22) K9ME3K14ACK18AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, TRANSCRIPTION
3u5o:H (PRO960) to (SER1082) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-22) K9ME3K14ACK18AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, TRANSCRIPTION
3u5p:A (SER959) to (TYR1081) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-28) K9ME3K14ACK18ACK23AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, K23AC, TRANSCRIPTION
3u5p:B (SER959) to (ILE1080) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-28) K9ME3K14ACK18ACK23AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, K23AC, TRANSCRIPTION
3u5p:C (SER959) to (ILE1080) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-28) K9ME3K14ACK18ACK23AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, K23AC, TRANSCRIPTION
3u5p:D (SER959) to (GLU1079) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-28) K9ME3K14ACK18ACK23AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, K23AC, TRANSCRIPTION
3u5p:E (SER959) to (SER1082) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-28) K9ME3K14ACK18ACK23AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, K23AC, TRANSCRIPTION
3u5p:F (SER959) to (ILE1080) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-28) K9ME3K14ACK18ACK23AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, K23AC, TRANSCRIPTION
3u5p:G (SER959) to (ILE1080) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-28) K9ME3K14ACK18ACK23AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, K23AC, TRANSCRIPTION
3u5p:H (SER959) to (TYR1081) CRYSTAL STRUCTURE OF THE COMPLEX OF TRIM33 PHD-BROMO AND H3(1-28) K9ME3K14ACK18ACK23AC HISTONE PEPTIDE | TRIM33, PHD, BROMODOMAIN, TGF-BETA, EPIGENETICS, HISTONE, METHYLATION, K9ME3, K14AC, K18AC, K23AC, TRANSCRIPTION
3hme:B (PRO24) to (MET121) CRYSTAL STRUCTURE OF HUMAN BROMODOMAIN CONTAINING 9 ISOFORM 1 (BRD9) | BRD9, BROMODOMAIN CONTAINING 9 ISOFORM 1, LAVS3040, PRO9856, RHABDOMYOSARCOMA ANTIGEN MU-RMS-40.8, SARCOMA ANTIGEN NY-SAR-29, BROMODOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, SIGNALING PROTEIN
4yy4:A (GLN26) to (SER122) CRYSTAL STRUCTURE OF BRD9 BROMODOMAIN BOUND TO DMSO | COMPLEX, PROTEIN BINDING
4yy6:A (THR23) to (LYS123) CRYSTAL STRUCTURE OF BRD9 BROMODOMAIN BOUND TO A BUTYRYLLYSINE PEPTIDE | BROMODOMAIN-BUTYRYLLYSINE COMPLEX, PROTEIN BINDING
4yyd:A (ILE25) to (MET121) CRYSTAL STRUCTURE OF BRD9 BROMODOMAIN BOUND TO A CROTONYLLYSINE PEPTIDE | BROMODOMAIN-CROTONYLLYSINE COMPLEX, PROTEIN BINDING
4yyg:A (GLN26) to (MET121) CRYSTAL STRUCTURE OF BRD9 BROMODOMAIN BOUND TO A BUTYRYLLYSINE PEPTIDE | BROMODOMAIN-BUTYRYLLYSINE COMPLEX, PROTEIN BINDING
4yyh:A (THR23) to (LYS123) CRYSTAL STRUCTURE OF BRD9 BROMODOMAIN BOUND TO A CROTONYLLYSINE PEPTIDE | BROMODOMAIN-CROTONYLLYSINE COMPLEX, PROTEIN BINDING
4yyh:B (THR23) to (SER122) CRYSTAL STRUCTURE OF BRD9 BROMODOMAIN BOUND TO A CROTONYLLYSINE PEPTIDE | BROMODOMAIN-CROTONYLLYSINE COMPLEX, PROTEIN BINDING
4yym:A (ASP1501) to (TYR1607) CRYSTAL STRUCTURE OF TAF1 BD2 BROMODOMAIN BOUND TO A BUTYRYLLYSINE PEPTIDE | BROMODOMAIN-BUTYRYLLYSINE COMPLEX, PROTEIN BINDING
4yym:B (ASP1502) to (TYR1607) CRYSTAL STRUCTURE OF TAF1 BD2 BROMODOMAIN BOUND TO A BUTYRYLLYSINE PEPTIDE | BROMODOMAIN-BUTYRYLLYSINE COMPLEX, PROTEIN BINDING
2f6j:A (THR70) to (LYS170) CRYSTAL STRUCTURE OF PHD FINGER-LINKER-BROMODOMAIN FRAGMENT OF HUMAN BPTF IN THE H3(1-15)K4ME3 BOUND STATE | PHD FINGER; BROMO DOMAIN; HISTONE TAIL BINDING; METHYLATION, TRANSCRIPTION
2f6j:B (THR70) to (LYS170) CRYSTAL STRUCTURE OF PHD FINGER-LINKER-BROMODOMAIN FRAGMENT OF HUMAN BPTF IN THE H3(1-15)K4ME3 BOUND STATE | PHD FINGER; BROMO DOMAIN; HISTONE TAIL BINDING; METHYLATION, TRANSCRIPTION
2f6j:C (THR70) to (LYS170) CRYSTAL STRUCTURE OF PHD FINGER-LINKER-BROMODOMAIN FRAGMENT OF HUMAN BPTF IN THE H3(1-15)K4ME3 BOUND STATE | PHD FINGER; BROMO DOMAIN; HISTONE TAIL BINDING; METHYLATION, TRANSCRIPTION
2f6n:A (THR70) to (LEU169) CRYSTAL STRUCTURE OF PHD FINGER-LINKER-BROMODOMAIN FRAGMENT OF HUMAN BPTF IN THE FREE FORM | PHD FINGER; BROMO DOMAIN; HISTONE TAIL BINDING; METHYLATION, TRANSCRIPTION
4z1q:A (THR60) to (LEU164) CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 BOUND TO BENZOTRIAZOLO-DIAZEPINE SCAFFOLD | BROMODOMAIN, TRANSCRIPTION
4z1q:B (THR60) to (LEU164) CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 BOUND TO BENZOTRIAZOLO-DIAZEPINE SCAFFOLD | BROMODOMAIN, TRANSCRIPTION
4z1s:A (VAL69) to (LEU164) CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 WITH BENZOTRIAZOLO-DIAZEPINE SCAFFOLD | BROMODOMAIN, SIGNALING PROTEIN
4z1s:B (VAL69) to (ASN162) CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 WITH BENZOTRIAZOLO-DIAZEPINE SCAFFOLD | BROMODOMAIN, SIGNALING PROTEIN
4z6h:A (THR23) to (MET121) CRYSTAL STRUCTURE OF BRD9 BROMODOMAIN IN COMPLEX WITH A VALEROLACTAM QUINOLONE LIGAND | LYSINE-ACETYLATED HISTONE BINDING, CHROMATIN REGULATOR, TRANSCRIPTION, BROMODOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
4z6i:A (THR23) to (MET121) CRYSTAL STRUCTURE OF BRD9 BROMODOMAIN IN COMPLEX WITH A SUBSTITUTED VALEROLACTAM QUINOLONE LIGAND | LYSINE-ACETYLATED HISTONE BINDING, CHROMATIN REGULATOR, TRANSCRIPTION, BROMODOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
4z6i:B (THR23) to (MET121) CRYSTAL STRUCTURE OF BRD9 BROMODOMAIN IN COMPLEX WITH A SUBSTITUTED VALEROLACTAM QUINOLONE LIGAND | LYSINE-ACETYLATED HISTONE BINDING, CHROMATIN REGULATOR, TRANSCRIPTION, BROMODOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
3uv2:A (THR2803) to (HIS2911) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN NUCLEOSOME-REMODELING FACTOR SUBUNIT BPTF | BROMODOMAIN, BPTF, FALZ, FAC1, BROMODOMAIN AND PHD FINGER-CONTAINING TRANSCRIPTION FACTOR, FETAL ALZ-50 CLONE 1 PROTEIN, FETAL ALZHEIMER ANTIGEN, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
4kly:B (THR28) to (LEU113) CRYSTAL STRUCTURE OF A BLUE-LIGHT ABSORBING PROTEORHODOPSIN MUTANT D97N FROM HOT75 | ION TRANSPORT, PROTON PUMP, RETINYLIDENE SCHIFF BASE, MEMBRANE, PROTON TRANSPORT
3uv4:A (ASP1523) to (ASP1629) CRYSTAL STRUCTURE OF THE SECOND BROMODOMAIN OF HUMAN TRANSCRIPTION INITIATION FACTOR TFIID SUBUNIT 1 (TAF1) | STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
3uv4:B (ASP1523) to (ASP1629) CRYSTAL STRUCTURE OF THE SECOND BROMODOMAIN OF HUMAN TRANSCRIPTION INITIATION FACTOR TFIID SUBUNIT 1 (TAF1) | STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
2fsa:A (THR70) to (LYS170) CRYSTAL STRUCTURE OF PHD FINGER-LINKER-BROMODOMAIN FRAGMENT OF HUMAN BPTF IN THE H3(1-15)K4ME2 BOUND STATE | PHD FINGER, BROMODOMAIN, PEPTIDE COMPLEX, TRANSCRIPTION
2fsa:B (THR70) to (LYS170) CRYSTAL STRUCTURE OF PHD FINGER-LINKER-BROMODOMAIN FRAGMENT OF HUMAN BPTF IN THE H3(1-15)K4ME2 BOUND STATE | PHD FINGER, BROMODOMAIN, PEPTIDE COMPLEX, TRANSCRIPTION
2fsa:C (THR70) to (LYS170) CRYSTAL STRUCTURE OF PHD FINGER-LINKER-BROMODOMAIN FRAGMENT OF HUMAN BPTF IN THE H3(1-15)K4ME2 BOUND STATE | PHD FINGER, BROMODOMAIN, PEPTIDE COMPLEX, TRANSCRIPTION
3i3j:A (MET1059) to (GLU1152) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN EP300 | STRUCTURAL GENOMICS BROMODOMAIN, P300, CONSORTIUM, SGC, STRUCTURAL GENOMICS CONSORTIUM, BROMODOMAIN, CELL CYCLE, CITRULLINATION, DISEASE MUTATION, HOST-VIRUS INTERACTION, METAL-BINDING, METHYLATION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, ZINC-FINGER
3i3j:B (MET1059) to (GLU1152) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN EP300 | STRUCTURAL GENOMICS BROMODOMAIN, P300, CONSORTIUM, SGC, STRUCTURAL GENOMICS CONSORTIUM, BROMODOMAIN, CELL CYCLE, CITRULLINATION, DISEASE MUTATION, HOST-VIRUS INTERACTION, METAL-BINDING, METHYLATION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, ZINC-FINGER
3i3j:C (MET1059) to (GLU1152) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN EP300 | STRUCTURAL GENOMICS BROMODOMAIN, P300, CONSORTIUM, SGC, STRUCTURAL GENOMICS CONSORTIUM, BROMODOMAIN, CELL CYCLE, CITRULLINATION, DISEASE MUTATION, HOST-VIRUS INTERACTION, METAL-BINDING, METHYLATION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, ZINC-FINGER
3i3j:D (MET1059) to (GLU1152) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN EP300 | STRUCTURAL GENOMICS BROMODOMAIN, P300, CONSORTIUM, SGC, STRUCTURAL GENOMICS CONSORTIUM, BROMODOMAIN, CELL CYCLE, CITRULLINATION, DISEASE MUTATION, HOST-VIRUS INTERACTION, METAL-BINDING, METHYLATION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, ZINC-FINGER
3i3j:E (MET1059) to (GLU1152) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN EP300 | STRUCTURAL GENOMICS BROMODOMAIN, P300, CONSORTIUM, SGC, STRUCTURAL GENOMICS CONSORTIUM, BROMODOMAIN, CELL CYCLE, CITRULLINATION, DISEASE MUTATION, HOST-VIRUS INTERACTION, METAL-BINDING, METHYLATION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, ZINC-FINGER
3i3j:F (LYS1050) to (GLU1152) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN EP300 | STRUCTURAL GENOMICS BROMODOMAIN, P300, CONSORTIUM, SGC, STRUCTURAL GENOMICS CONSORTIUM, BROMODOMAIN, CELL CYCLE, CITRULLINATION, DISEASE MUTATION, HOST-VIRUS INTERACTION, METAL-BINDING, METHYLATION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, ZINC-FINGER
3i3j:G (MET1059) to (GLU1152) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN EP300 | STRUCTURAL GENOMICS BROMODOMAIN, P300, CONSORTIUM, SGC, STRUCTURAL GENOMICS CONSORTIUM, BROMODOMAIN, CELL CYCLE, CITRULLINATION, DISEASE MUTATION, HOST-VIRUS INTERACTION, METAL-BINDING, METHYLATION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, ZINC-FINGER
3i3j:H (LYS1050) to (GLU1152) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN EP300 | STRUCTURAL GENOMICS BROMODOMAIN, P300, CONSORTIUM, SGC, STRUCTURAL GENOMICS CONSORTIUM, BROMODOMAIN, CELL CYCLE, CITRULLINATION, DISEASE MUTATION, HOST-VIRUS INTERACTION, METAL-BINDING, METHYLATION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, ZINC-FINGER
3i3j:I (MET1059) to (GLU1152) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN EP300 | STRUCTURAL GENOMICS BROMODOMAIN, P300, CONSORTIUM, SGC, STRUCTURAL GENOMICS CONSORTIUM, BROMODOMAIN, CELL CYCLE, CITRULLINATION, DISEASE MUTATION, HOST-VIRUS INTERACTION, METAL-BINDING, METHYLATION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, ZINC-FINGER
3i3j:J (MET1059) to (GLU1152) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN EP300 | STRUCTURAL GENOMICS BROMODOMAIN, P300, CONSORTIUM, SGC, STRUCTURAL GENOMICS CONSORTIUM, BROMODOMAIN, CELL CYCLE, CITRULLINATION, DISEASE MUTATION, HOST-VIRUS INTERACTION, METAL-BINDING, METHYLATION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, ZINC-FINGER
3i3j:K (LYS1050) to (GLU1152) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN EP300 | STRUCTURAL GENOMICS BROMODOMAIN, P300, CONSORTIUM, SGC, STRUCTURAL GENOMICS CONSORTIUM, BROMODOMAIN, CELL CYCLE, CITRULLINATION, DISEASE MUTATION, HOST-VIRUS INTERACTION, METAL-BINDING, METHYLATION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, ZINC-FINGER
3i3j:L (MET1059) to (GLU1152) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN EP300 | STRUCTURAL GENOMICS BROMODOMAIN, P300, CONSORTIUM, SGC, STRUCTURAL GENOMICS CONSORTIUM, BROMODOMAIN, CELL CYCLE, CITRULLINATION, DISEASE MUTATION, HOST-VIRUS INTERACTION, METAL-BINDING, METHYLATION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, ZINC-FINGER
2gf5:A (ASP111) to (GLN169) STRUCTURE OF INTACT FADD (MORT1) | DEATH DOMAIN, DEATH EFFECTOR DOMAIN, APOPTOSIS, DEATH- INDUCING SIGNALING COMPLEX
2grc:A (PRO1456) to (ASP1569) 1.5 A STRUCTURE OF BROMODOMAIN FROM HUMAN BRG1 PROTEIN, A CENTRAL ATPASE OF SWI/SNF REMODELING COMPLEX | BROMODOMAIN, BRG1, CHROMATIN REMODELLING, ACELY-LYSINE BINDING, PROTEIN-PROTEIN INTERACTIONS, HYDROLASE
4zql:A (THR901) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 WITH 3,4-DIMETHOXY-N-(6-(4- METHOXYPHENOXY)-1,3-DIMETHYL-2-OXO-2,3-DIHYDRO-1H-BENZO[D]IMIDAZOL-5- YL)BENZENESULFONAMIDE INHIBITOR | TRANSCRIPTIONAL COACTIVATOR, HISTONE H3 MODIFICATIONS, E3 PROTEIN- UBIQUITIN LIGASE ACTIVITY, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, LIGASE
4zql:B (THR901) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 WITH 3,4-DIMETHOXY-N-(6-(4- METHOXYPHENOXY)-1,3-DIMETHYL-2-OXO-2,3-DIHYDRO-1H-BENZO[D]IMIDAZOL-5- YL)BENZENESULFONAMIDE INHIBITOR | TRANSCRIPTIONAL COACTIVATOR, HISTONE H3 MODIFICATIONS, E3 PROTEIN- UBIQUITIN LIGASE ACTIVITY, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, LIGASE
2wp2:B (VAL38) to (MET132) STRUCTURE OF BRDT BROMODOMAIN BD1 BOUND TO A DIACETYLATED HISTONE H4 PEPTIDE. | TRANSCRIPTION-PEPTIDE COMPLEX, TRANSCRIPTION REGULATION, BRDT, ACETYLLYSINE, NUCLEUS, COILED COIL, CHROMOSOMAL PROTEIN, NUCLEOSOME
4lys:A (THR60) to (ASN162) CRYSTAL STRUCTURE OF BRD4(1) BOUND TO COLCHICEINE | BROMODOMAIN, BRD4 INHIBITOR, EPIGENETIC READER PROTEIN, ACETYLATED LYSINE, HISTONE TAIL, NUCLEUS, PROTEIN BINDING-INHIBITOR COMPLEX
5a5n:A (SER979) to (GLU1091) CRYSTAL STRUCTURE OF HUMAN ATAD2 BROMODOMAIN IN COMPLEX WITH (2S)-2,6-DIACETAMIDO-N-METHYLHEXANAMIDE | HYDROLASE, INHIBITOR, EPIGENETICS, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2
5a5o:A (MET980) to (GLU1091) CRYSTAL STRUCTURE OF HUMAN ATAD2 BROMODOMAIN IN COMPLEX WITH 3-METHYL-1,2-DIHYDROQUINOLIN-2-ONE | HYDROLASE, INHIBITOR, ATAD2, BROMODOMAIN, EPIGENETICS
5a5q:A (SER979) to (LEU1093) CRYSTAL STRUCTURE OF HUMAN ATAD2 BROMODOMAIN IN COMPLEX WITH 3-METHYL-8-PIPERIDIN-4-YLAMINO-1,2-DIHYDRO-1,7- NAPHTHYRIDIN-2-ONE HYDROCHLORIDE | HYDROLASE, INHIBITOR, ATAD2 , BROMODOMAIN, EPIGENETICS, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2
5a5r:A (SER979) to (GLU1091) CRYSTAL STRUCTURE OF HUMAN ATAD2 BROMODOMAIN IN COMPLEX WITH 5-5-METHOXYPYRIDIN-3-YL-3-METHYL-8-PIPERIDIN-4- YLAMINO-1,2-DIHYDRO-1,7-NAPHTHYRIDIN-2-ONE | HYDROLASE, INHIBITOR, ATAD2 , BROMODOMAIN, EPIGENETICS, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2
5a81:A (SER979) to (GLU1091) CRYSTAL STRUCTURE OF HUMAN ATAD2 BROMODOMAIN IN COMPLEX WITH 8-(3R,4R)-3-(CYCLOHEXYLMETHOXY)PIPERIDIN-4-YL-AMINO-3- METHYL-1,2-DIHYDRO-1,7-NAPHTHYRIDIN-2-ONE | HYDROLASE, INHIBITOR, ATAD2, BROMODOMAIN, EPIGENETICS, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2
5a82:A (SER979) to (GLU1091) CRYSTAL STRUCTURE OF HUMAN ATAD2 BROMODOMAIN IN COMPLEX WITH 4-(3R,4R)-4-(3-METHYL-2-OXO-1,2-DIHYDRO-1,7- NAPHTHYRIDIN-8-YL)AMINOPIPERIDIN-3-YLOXYMETHYL)-1-THIANE-1, 1-DIONE | INHIBITOR, ATAD2 , BROMODOMAIN, EPIGENETICS, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2
5a83:A (SER979) to (GLU1091) CRYSTAL STRUCTURE OF HUMAN ATAD2 BROMODOMAIN IN COMPLEX WITH 4-((3R,4R)-4-3-METHYL-5-(5-METHYLPYRIDIN-3-YL)-2-OXO- 1,2-DIHYDROQUINOLIN-8-YL-AMINOPIPERIDIN-3-YLOXYMETHYL)-1- THIANE-1,1-DIONE | HYDROLASE, INHIBITOR, ATAD2, BROMODOMAIN, EPIGENETICS, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2
5ad2:B (THR60) to (LEU164) BIVALENT BINDING TO BET BROMODOMAINS | TRANSCRIPTION
5ad3:B (THR60) to (LEU164) BIVALENT BINDING TO BET BROMODOMAINS | TRANSCRIPTION
4n3w:A (PRO1087) to (GLU1188) CRYSTAL STRUCTURE OF THE BROMODOMAIN-PHD FINGER MODULE OF HUMAN TRANSCRIPTIONAL CO-ACTIVATOR CBP IN COMPLEX WITH ACETYLATED HISTONE 4 PEPTIDE (H4K20AC). | HISTONE BINDING, TRANSFERASE-NUCLEAR PROTEIN COMPLEX
4n4f:A (PRO1087) to (GLU1188) CRYSTAL STRUCTURE OF THE BROMODOMAIN-PHD FINGER MODULE OF HUMAN TRANSCRIPTIONAL CO-ACTIVATOR CBP IN COMPLEX WITH DI-ACETYLATED HISTONE 4 PEPTIDE (H412ACK16AC). | TRANSCRIPTIONAL CO-ACTIVATOR, HISTONE, TRANSCRIPTION-PROTEIN BINDING COMPLEX
4n4g:A (ASN154) to (CYS258) CRYSTAL STRUCTURE OF THE BROMO-PWWP OF THE MOUSE ZINC FINGER MYND-TYPE CONTAINING 11 ISOFORM ALPHA | TANDEM BROMODOMAIN-ZINC FINGER-PWWP MOTIF, HISTONE H3.3-SPECIFIC, TRANSCRIPTION
4n4h:A (GLN156) to (CYS258) CRYSTAL STRUCTURE OF THE BROMO-PWWP OF THE MOUSE ZINC FINGER MYND-TYPE CONTAINING 11 ISOFORM ALPHA IN COMPLEX WITH HISTONE H3.1K36ME3 | TANDEM BROMODOMAIN-ZINC FINGER-PWWP MOTIF, HISTONE H3.3-SPECIFIC, TRANSCRIPTION
2xry:A (GLY233) to (TYR314) X-RAY STRUCTURE OF ARCHAEAL CLASS II CPD PHOTOLYASE FROM METHANOSARCINA MAZEI | DNA DAMAGE, DNA REPAIR, LYASE
2xrz:A (GLY233) to (ILE302) X-RAY STRUCTURE OF ARCHAEAL CLASS II CPD PHOTOLYASE FROM METHANOSARCINA MAZEI IN COMPLEX WITH INTACT CPD-LESION | LYASE-DNA COMPLEX, PHOTOLYASE, DNA DAMAGE, DNA REPAIR, CLASS II, INTACT CPD-LESION, PROTEIN-DNA COMPLEX, WATER CLUSTER
5bt3:A (LYS1050) to (GLU1152) CRYSTAL STRUCTURE OF EP300 BROMODOMAIN IN COMPLEX WITH SGC-CBP30 CHEMICAL PROBE | P300, TRANSCRIPTION REGULATION, HISTONE ACETYLTRANSFERASE, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
4nqk:A (THR121) to (ARG179) STRUCTURE OF AN UBIQUITIN COMPLEX | CARD DOMAIN, HYDROLASE-APOPTOSIS COMPLEX
4nqn:A (THR23) to (MET133) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BRD9 IN COMPLEX WITH A TRIAZOLO-PHTHALAZINE LIGAND | STRUCTURAL GENOMICS CONSORTIUM, SGC, BROMODOMAIN, INHIBITION, TRANSCRIPTION, SMALL MOLECULE INHIBITOR, TRANSCRIPTION-INHIBITOR COMPLEX
4nr4:A (MET1095) to (GLU1188) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CREBBP IN COMPLEX WITH AN ISOXAZOLYL-BENZIMIDAZOLE LIGAND | STRUCTURAL GENOMICS CONSORTIUM, SGC, CHEMICAL TOOL, SMALL MOLECULE INHIBITOR, TRANSCRIPTION, TRANSCRIPTION-INHIBITOR COMPLEX
4nr9:A (ASP1869) to (VAL1971) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BAZ2B IN COMPLEX WITH ACETYLATED LYSINE | SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSCRIPTION, BROMODOMAIN, ACETYLATED LYSINE BINDING PROTEIN, KIAA1476, WALP4
4nra:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BAZ2B IN COMPLEX WITH COMPOUND-6 E11322 | SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSCRIPTION, BROMODOMAIN, ACETYLATED LYSINE BINDING PROTEIN, KIAA1476, WALP4
4nrb:A (ASP1869) to (PHE1969) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BAZ2B IN COMPLEX WITH COMPOUND-1 N01197 | SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSCRIPTION, BROMODOMAIN, ACETYLATED LYSINE BINDING PROTEIN, KIAA1476, WALP4
4nrc:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BAZ2B IN COMPLEX WITH COMPOUND-3 N01186 | SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSCRIPTION, BROMODOMAIN, ACETYLATED LYSINE BINDING PROTEIN, KIAA1476, WALP4
4ns5:A (GLU157) to (CYS258) CRYSTAL STRUCTURE OF HUMAN BS69 BROMO-ZINC FINGER-PWWP | ZINC FINGER, CHROMATIN BINDING, HISTONE, NUCLEUS, TRANSCRIPTION REGULATOR
2yem:A (VAL350) to (MET457) CRYSTAL STRUCTURE OF THE SECOND BROMODOMAIN OF HUMAN BRD4 WITH THE INHIBITOR GW841819X | SIGNALING PROTEIN, HISTONE, EPIGENETIC READER
4nyx:A (LYS1086) to (GLU1188) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CREBBP IN COMPLEX WITH A DIHYDROQUINOXALINONE LIGAND | CREBBP, CREB BINDING, KAT3A, RSTS, RST, BROMODOMAIN, TRANSCRIPTION, STRUCTURAL GENOMICS CONSORTIUM, SGC
5c8g:B (PRO20) to (LEU124) CRYSTAL STRUCTURE ANALYSIS OF PP-BRD20 FROM TB427TMP COMPLEXED WITH BI-2536 | STRUCTURAL GENOMICS CONSORTIUM, SGC, BROMODOMAIN, PP-BRD20, TB427TMP, GENE REGULATION
3zyu:B (THR60) to (LEU164) CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH I-BET151(GSK1210151A) | SIGNALING PROTEIN, BROMODOMAIN, I-151, INHIBITOR, HISTONE, EPIGENETIC READER
4o76:B (THR60) to (LEU164) CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH TG101209 | BROMODOMAIN, CAP, HUNK1, MCAP, PROTEIN BINDING-INHIBITOR COMPLEX, MITOTIC CHROMOSOME ASSOCIATED PROTEIN, CELL CYCLE, INHIBITOR, TRANSCRIPTION-INHIBITOR COMPLEX
4a2w:B (ASP117) to (GLY177) STRUCTURE OF FULL-LENGTH DUCK RIG-I | HYDROLASE, SUPERFAMILY 2 RNA HELICASE, ATP AND DSRNA BINDING, CARD, ANTIVIRAL SIGNALLING PATHWAY
2yw5:A (THR36) to (ALA128) SOLUTION STRUCTURE OF THE BROMODOMAIN FROM HUMAN BROMODOMAIN CONTAINING PROTEIN 3 | BROMODOMAIN, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, SIGNALING PROTEIN
4ogj:B (THR60) to (LEU164) CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH THE INHIBITOR TG-101348 | BROMODOMAIN, BROMODOMAIN CONTAINING PROTEIN 4, JAK2 KINASE INHIBITOR, FLT3 KINASE INHIBITOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION-INHIBITOR COMPLEX
5coi:A (VAL70) to (LEU164) CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH BENZO[CD]INDOL-2(1H)-ONE LIGAND | BRD4, BROMODOMAIN, FOUR ALPHA HELICES, TRANSCRIPTION-TRANSCR, SIGNALING PROTEIN-INHIBITOR COMPLEX
5cq3:A (ASP1866) to (THR1968) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN PROTEIN 2B (BAZ2B) IN COMPLEX WITH 6-HYDROXYPICOLINIC ACID (SGC - DIAMOND I04-1 FRAGMENT SCREENING) | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
5cq6:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN PROTEIN 2B (BAZ2B) IN COMPLEX WITH 2,6- PYRIDINEDICARBOXYLIC ACID (SGC - DIAMOND I04-1 FRAGMENT SCREENING) | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
5cq7:A (ASP1869) to (PHE1969) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN PROTEIN 2B (BAZ2B) IN COMPLEX WITH N,N- DIMETHYLQUINOXALINE-6-CARBOXAMIDE (SGC - DIAMOND I04-1 FRAGMENT SCREENING) | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
5cq8:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN PROTEIN 2B (BAZ2B) IN COMPLEX WITH 4'- HYDROXYACETOPHENONE (SGC - DIAMOND I04-1 FRAGMENT SCREENING) | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
5csl:A (LEU838) to (GLU905) CRYSTAL STRUCTURE OF THE 500 KD YEAST ACETYL-COA CARBOXYLASE HOLOENZYME DIMER | ACETYL-COA CARBOXYLASE, LIGASE
5cu8:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN PROTEIN 2B (BAZ2B) IN COMPLEX WITH 2-AMINO-6- CHLOROBENZOTHIAZOLE (SGC - DIAMOND I04-1 FRAGMENT SCREENING) | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
5cua:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN PROTEIN 2B (BAZ2B) IN COMPLEX WITH 1-ACETYL-4-(4- HYDROXYPHENYL)PIPERAZINE (SGC - DIAMOND I04-1 FRAGMENT SCREENING) | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
5cuc:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN PROTEIN 2B (BAZ2B) IN COMPLEX WITH N-ACETYL-2- PHENYLETHYLAMINE (SGC - DIAMOND I04-1 FRAGMENT SCREENING) | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
5d0c:A (VAL70) to (LEU164) CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH BENZO[CD]INDOL-2(1H)-ONE LIGAND | BRD4, BROMODOMAIN, FOUR ALPHA HELICES, BROMODOMAIN BINDING INHIBITOR, SIGNALING PROTEIN-INHIBITOR COMPLEX
5d7x:A (THR631) to (GLU737) CRYSTAL STRUCTURE OF THE HUMAN BRPF1 BROMODOMAIN IN COMPLEX WITH XZ08 | BROMODOMAIN AND PHD FINGER-CONTAINING PROTEIN 1(BRPF1), MONOCYTIC LEUKEMIA ZINC-FINGER (MOZ), INHIBITOR, DNA BINDING PROTEIN
3aad:A (ASP1503) to (TYR1607) STRUCTURE OF THE HISTONE CHAPERONE CIA/ASF1-DOUBLE BROMODOMAIN COMPLEX LINKING HISTONE MODIFICATIONS AND SITE-SPECIFIC HISTONE EVICTION | PROTEIN-PROTEIN COMPLEX, BROMODOMAIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, CHAPERONE, CHROMATIN REGULATOR, TRANSCRIPTION-CHAPERONE COMPLEX
4pkl:A (ASN13) to (THR102) BROMODOMAIN OF TRYPANOSOMA BRUCEI BDF2 WITH IBET-151 | SIGNALING PROTEIN, INHIBITOR, HISTONE, EPIGENETIC READER, SIGNALING PROTEIN-INHIBITOR COMPLEX
4pkl:B (ASN13) to (THR102) BROMODOMAIN OF TRYPANOSOMA BRUCEI BDF2 WITH IBET-151 | SIGNALING PROTEIN, INHIBITOR, HISTONE, EPIGENETIC READER, SIGNALING PROTEIN-INHIBITOR COMPLEX
5dkc:A (PRO1381) to (LYS1490) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BRM (SMARCA2) IN COMPLEX WITH PFI-3 CHEMICAL PROBE | SWI-SNF COMPLEX, CHROMATIN REMODELING, BRG ASSOCIATED FACTORS (BAF), TRANSCRIPTION, HYDROLASE
5dkd:A (ASN1457) to (LYS1566) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BRG1 (SMARCA4) IN COMPLEX WITH PFI-3 CHEMICAL PROBE | SWI-SNF COMPLEX, CHROMATIN REMODELING, BRG ASSOCIATED FACTORS (BAF), TRANSCRIPTION, HYDROLASE
5dkd:B (LEU1458) to (LYS1566) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BRG1 (SMARCA4) IN COMPLEX WITH PFI-3 CHEMICAL PROBE | SWI-SNF COMPLEX, CHROMATIN REMODELING, BRG ASSOCIATED FACTORS (BAF), TRANSCRIPTION, HYDROLASE
5dkh:A (LYS1382) to (GLU1491) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BRM (SMARCA2) IN COMPLEX WITH A HYDROXYPHENYL PROPENONE INHIBITOR 17 | SWI-SNF COMPLEX, CHROMATIN REMODELING, BRG ASSOCIATED FACTORS (BAF), TRANSCRIPTION
5dkh:B (PRO1381) to (LYS1490) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BRM (SMARCA2) IN COMPLEX WITH A HYDROXYPHENYL PROPENONE INHIBITOR 17 | SWI-SNF COMPLEX, CHROMATIN REMODELING, BRG ASSOCIATED FACTORS (BAF), TRANSCRIPTION
4q0n:A (THR624) to (GLU732) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN POLY-BROMODOMAIN CONTAINING PROTEIN 1 (PB1) IN COMPLEX WITH A HYDROXYPHENYL-PROPENONE LIGAND | PB1, POLYBROMO 1 ISOFORM 1, BAF180, POLYBROMO-1D, PBRM1, BRG1- ASSOCIATED FACTOR 180, BROMODOMAIN, CHROMATIN REGULATOR, DNA- BINDING, NUCLEUS, TRANSCRIPTION, TRANSCRIPTION REGULATION, STRUCTURAL GENOMICS CONSORTIUM, SGC
4q0n:C (THR624) to (ASP730) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN POLY-BROMODOMAIN CONTAINING PROTEIN 1 (PB1) IN COMPLEX WITH A HYDROXYPHENYL-PROPENONE LIGAND | PB1, POLYBROMO 1 ISOFORM 1, BAF180, POLYBROMO-1D, PBRM1, BRG1- ASSOCIATED FACTOR 180, BROMODOMAIN, CHROMATIN REGULATOR, DNA- BINDING, NUCLEUS, TRANSCRIPTION, TRANSCRIPTION REGULATION, STRUCTURAL GENOMICS CONSORTIUM, SGC
4q0n:D (PRO625) to (GLU732) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN POLY-BROMODOMAIN CONTAINING PROTEIN 1 (PB1) IN COMPLEX WITH A HYDROXYPHENYL-PROPENONE LIGAND | PB1, POLYBROMO 1 ISOFORM 1, BAF180, POLYBROMO-1D, PBRM1, BRG1- ASSOCIATED FACTOR 180, BROMODOMAIN, CHROMATIN REGULATOR, DNA- BINDING, NUCLEUS, TRANSCRIPTION, TRANSCRIPTION REGULATION, STRUCTURAL GENOMICS CONSORTIUM, SGC
4q0n:E (PRO625) to (GLU732) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN POLY-BROMODOMAIN CONTAINING PROTEIN 1 (PB1) IN COMPLEX WITH A HYDROXYPHENYL-PROPENONE LIGAND | PB1, POLYBROMO 1 ISOFORM 1, BAF180, POLYBROMO-1D, PBRM1, BRG1- ASSOCIATED FACTOR 180, BROMODOMAIN, CHROMATIN REGULATOR, DNA- BINDING, NUCLEUS, TRANSCRIPTION, TRANSCRIPTION REGULATION, STRUCTURAL GENOMICS CONSORTIUM, SGC
4q0n:G (THR624) to (GLU732) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN POLY-BROMODOMAIN CONTAINING PROTEIN 1 (PB1) IN COMPLEX WITH A HYDROXYPHENYL-PROPENONE LIGAND | PB1, POLYBROMO 1 ISOFORM 1, BAF180, POLYBROMO-1D, PBRM1, BRG1- ASSOCIATED FACTOR 180, BROMODOMAIN, CHROMATIN REGULATOR, DNA- BINDING, NUCLEUS, TRANSCRIPTION, TRANSCRIPTION REGULATION, STRUCTURAL GENOMICS CONSORTIUM, SGC
4q0n:H (THR624) to (LEU731) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN POLY-BROMODOMAIN CONTAINING PROTEIN 1 (PB1) IN COMPLEX WITH A HYDROXYPHENYL-PROPENONE LIGAND | PB1, POLYBROMO 1 ISOFORM 1, BAF180, POLYBROMO-1D, PBRM1, BRG1- ASSOCIATED FACTOR 180, BROMODOMAIN, CHROMATIN REGULATOR, DNA- BINDING, NUCLEUS, TRANSCRIPTION, TRANSCRIPTION REGULATION, STRUCTURAL GENOMICS CONSORTIUM, SGC
5dyu:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF BAZ2B BROMODOMAIN IN COMPLEX WITH FRAGMENT F39 | FOUR HELICAL BUNDLE, TRANSCRIPTION
5dyx:A (ASP1866) to (THR1968) CRYSTAL STRUCTURE OF BAZ2B BROMODOMAIN IN COMPLEX WITH FRAGMENT F59 | FOUR HELICAL BUNDLE, TRANSCRIPTION
3lqj:A (GLU1631) to (VAL1765) CRYSTAL STRUCTURE OF MLL1 PHD3-BROMO COMPLEXED WITH H3(1-9)K4ME3 PEPTIDE | PHD FINGER, BROMODOMAIN, MLL1, LEUKEMIA, H3(1-9)K4ME3, CHROMOSOMAL PROTEIN, DNA-BINDING, NUCLEOSOME CORE, NUCLEUS, TRANSFERASE
3lqj:B (TRP1632) to (PRO1767) CRYSTAL STRUCTURE OF MLL1 PHD3-BROMO COMPLEXED WITH H3(1-9)K4ME3 PEPTIDE | PHD FINGER, BROMODOMAIN, MLL1, LEUKEMIA, H3(1-9)K4ME3, CHROMOSOMAL PROTEIN, DNA-BINDING, NUCLEOSOME CORE, NUCLEUS, TRANSFERASE
3aqb:A (ASP40) to (TYR127) M. LUTEUS B-P 26 HETERODIMERIC HEXAPRENYL DIPHOSPHATE SYNTHASE IN COMPLEX WITH MAGNESIUM | PRENYLTRANSFERASE, TRANSFERASE
3aqc:A (ASP40) to (TYR127) M. LUTEUS B-P 26 HETERODIMERIC HEXAPRENYL DIPHOSPHATE SYNTHASE IN COMPLEX WITH MAGNESIUM AND FPP ANALOGUE | PRENYLTRANSFERASE, TRANSFERASE
5e73:A (ASP1866) to (THR1968) CRYSTAL STRUCTURE OF BAZ2B BROMODOMAIN IN COMPLEX WITH ACETYLINDOLE COMPOUND UZH47 | FOUR HELICAL BUNDLE, TRANSCRIPTION
5e74:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF BAZ2B BROMODOMAIN IN COMPLEX WITH ACETYLINDOLE COMPOUND UZH50 | FOUR HELICAL BUNDLE, TRANSCRIPTION
5e7d:A (THR624) to (LEU731) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN PB1 IN COMPLEX WITH A HYDROXYPHENYL LIGAND | BROMODOMAIN, CHEMICAL PROBE, LIGAND, INHIBITOR, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
5e7d:B (THR624) to (LEU731) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN PB1 IN COMPLEX WITH A HYDROXYPHENYL LIGAND | BROMODOMAIN, CHEMICAL PROBE, LIGAND, INHIBITOR, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
5e7d:C (THR624) to (ASP730) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN PB1 IN COMPLEX WITH A HYDROXYPHENYL LIGAND | BROMODOMAIN, CHEMICAL PROBE, LIGAND, INHIBITOR, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
5e7d:D (THR624) to (ASP730) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN PB1 IN COMPLEX WITH A HYDROXYPHENYL LIGAND | BROMODOMAIN, CHEMICAL PROBE, LIGAND, INHIBITOR, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
3lxj:A (MET952) to (LEU1067) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN AAA DOMAIN CONTAINING 2B (ATAD2B) | ATPASE FAMILY, AAA DOMAIN CONTAINING 2B, ATAD2B, BROMODOMAIN, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, HYDROLASE
3lxj:B (SER951) to (LEU1067) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN AAA DOMAIN CONTAINING 2B (ATAD2B) | ATPASE FAMILY, AAA DOMAIN CONTAINING 2B, ATAD2B, BROMODOMAIN, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, HYDROLASE
3lxj:C (GLU953) to (LEU1067) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN AAA DOMAIN CONTAINING 2B (ATAD2B) | ATPASE FAMILY, AAA DOMAIN CONTAINING 2B, ATAD2B, BROMODOMAIN, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, HYDROLASE
3lxj:D (SER951) to (LEU1067) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN AAA DOMAIN CONTAINING 2B (ATAD2B) | ATPASE FAMILY, AAA DOMAIN CONTAINING 2B, ATAD2B, BROMODOMAIN, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, NUCLEOTIDE- BINDING, PHOSPHOPROTEIN, HYDROLASE
5e9l:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF BAZ2B BROMODOMAIN IN COMPLEX WITH FRAGMENT F103 | FOUR HELICAL BUNDLE, TRANSCRIPTION
5e9m:A (LYS1868) to (THR1968) CRYSTAL STRUCTURE OF BAZ2B BROMODOMAIN IN COMPLEX WITH N- METHYLTRIMETHYLACETAMIDE | FOUR HELICAL BUNDLE, TRANSCRIPTION
5e9v:A (THR139) to (MET236) CRYSTAL STRUCTURE OF BRD9 BROMODOMAIN IN COMPLEX WITH AN INDOLIZINE LIGAND | BROMODOMAIN, TRANSCRIPTION, CHROMATIN REGULATION
5e9v:B (THR139) to (MET236) CRYSTAL STRUCTURE OF BRD9 BROMODOMAIN IN COMPLEX WITH AN INDOLIZINE LIGAND | BROMODOMAIN, TRANSCRIPTION, CHROMATIN REGULATION
5e9y:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF BAZ2B BROMODOMAIN IN COMPLEX WITH MPD | FOUR HELICAL BUNDLE, TRANSCRIPTION
5ea1:A (ASN1457) to (GLU1565) CRYSTAL STRUCTURE OF SMARCA4 BROMODOMAIN IN COMPLEX WITH MPD | FOUR HELICAL BUNDLE, TRANSCRIPTION
5ea1:B (PRO1456) to (SER1559) CRYSTAL STRUCTURE OF SMARCA4 BROMODOMAIN IN COMPLEX WITH MPD | FOUR HELICAL BUNDLE, TRANSCRIPTION
4qc1:A (ASP2062) to (PHE2165) CRYSTAL STRUCTURE OF HUMAN BAZ2B BROMODOMAIN IN COMPLEX WITH AN ACETYLATED HISTONE 3 PEPTIDE (H3K14AC) | BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN PROTEIN 2B, HWALP4, KIAA1476, TRANSCRIPTIONAL REGULATION, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
4qc1:B (SER2063) to (PHE2165) CRYSTAL STRUCTURE OF HUMAN BAZ2B BROMODOMAIN IN COMPLEX WITH AN ACETYLATED HISTONE 3 PEPTIDE (H3K14AC) | BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN PROTEIN 2B, HWALP4, KIAA1476, TRANSCRIPTIONAL REGULATION, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
4qc3:B (SER2063) to (THR2164) CRYSTAL STRUCTURE OF HUMAN BAZ2B BROMODOMAIN IN COMPLEX WITH A DIACETYLATED HISTONE 4 PEPTIDE (H4K8ACK12AC) | BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN PROTEIN 2B, HWALP4, KIAA1476, TRANSCRIPTIONAL REGULATION, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
5eic:B (LYS1086) to (GLU1188) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CREBBP IN COMPLEX WITH AYC | TRANSFERASE, TRANSFERASE-INHIBITOR COMPLEX
4qns:B (HIS1356) to (ILE1460) CRYSTAL STRUCTURE OF BROMODOMAIN FROM PLASMODIUM FACIPARUM GCN5, PF3D7_0823300 | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, BROMODOMAIN, HISTONE, MALARIA, TRANSFERASE
4qns:C (GLN1360) to (ALA1459) CRYSTAL STRUCTURE OF BROMODOMAIN FROM PLASMODIUM FACIPARUM GCN5, PF3D7_0823300 | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, BROMODOMAIN, HISTONE, MALARIA, TRANSFERASE
4qns:D (GLN1360) to (ALA1459) CRYSTAL STRUCTURE OF BROMODOMAIN FROM PLASMODIUM FACIPARUM GCN5, PF3D7_0823300 | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, BROMODOMAIN, HISTONE, MALARIA, TRANSFERASE
5epb:A (SER979) to (LEU1093) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN ATAD2 IN COMPLEX WITH COMPOUND 49 | HYDROLASE INHIBITOR COMPLEX, TRANSFERASE
4qr3:A (THR60) to (LYS160) BRD4 BROMODOMAIN 1 COMPLEX WITH ITS NOVEL INHIBITORS | BRD4, BROMODOMAIN, FOUR ALPHA HELICES, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
4qr4:A (THR60) to (LYS160) BRD4 BROMODOMAIN 1 COMPLEX WITH ITS NOVEL INHIBITORS | BRD4, BROMODOMAIN, FOUR ALPHA HELICES, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
4qr5:A (THR60) to (LYS160) BRD4 BROMODOMAIN 1 COMPLEX WITH ITS NOVEL INHIBITORS | BRD4, BROMODOMAIN, FOUR ALPHA HELICES, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
4bhw:A (LYS1050) to (GLU1152) STRUCTURAL BASIS FOR AUTOINHIBITION OF THE ACETYLTRANSFERASE ACTIVITY OF P300 | TRANSFERASE, BROMODOMAIN, PHD DOMAIN, RING DOMAIN, HAT DOMAIN, ENHANCEOSOME
4qsq:A (MET980) to (GLU1091) STRUCTURE OF THE BROMODOMAIN OF HUMAN ATPASE FAMILY AAA DOMAIN- CONTAINING PROTEIN 2 (ATAD2) WITH BOUND DMSO | STRUCTURAL GENOMICS CONSORTIUM (SGC), SIGNALING PROTEIN, BROMODOMAIN, ACTYL-LYSINE BINDING, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2, EPIGENETICS
4qsr:A (MET980) to (LEU1093) STRUCTURE OF THE BROMODOMAIN OF HUMAN ATPASE FAMILY AAA DOMAIN- CONTAINING PROTEIN 2 (ATAD2) WITH BOUND MPD | STRUCTURAL GENOMICS CONSORTIUM (SGC), SIGNALING PROTEIN, BROMODOMAIN, ACTYL-LYSINE BINDING, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2, EPIGENETICS
4qss:A (MET980) to (LEU1093) STRUCTURE OF THE BROMODOMAIN OF HUMAN ATPASE FAMILY AAA DOMAIN- CONTAINING PROTEIN 2 (ATAD2) IN COMPLEX WITH N-METHYL-2-PYRROLIDONE (NMP) | STRUCTURAL GENOMICS CONSORTIUM (SGC), SIGNALING PROTEIN, BROMODOMAIN, ACTYL-LYSINE BINDING, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2, EPIGENETICS
4qst:A (SER979) to (GLU1091) STRUCTURE OF THE BROMODOMAIN OF HUMAN ATPASE FAMILY AAA DOMAIN- CONTAINING PROTEIN 2 (ATAD2) IN COMPLEX WITH 1-METHYLQUINOLIN 2-ONE | STRUCTURAL GENOMICS CONSORTIUM (SGC), SIGNALING PROTEIN, BROMODOMAIN, ACTYL-LYSINE BINDING, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2, EPIGENETICS
4qsu:A (MET980) to (GLU1091) STRUCTURE OF THE BROMODOMAIN OF HUMAN ATPASE FAMILY AAA DOMAIN- CONTAINING PROTEIN 2 (ATAD2) IN COMPLEX WITH THYMINE | STRUCTURAL GENOMICS CONSORTIUM (SGC), SIGNALING PROTEIN, BROMODOMAIN, ACTYL-LYSINE BINDING, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2, EPIGENETICS
4qsw:A (SER979) to (GLU1091) STRUCTURE OF THE BROMODOMAIN OF HUMAN ATPASE FAMILY AAA DOMAIN- CONTAINING PROTEIN 2 (ATAD2) IN COMPLEX WITH 5-METHYL URIDINE | STRUCTURAL GENOMICS CONSORTIUM (SGC), SIGNALING PROTEIN, BROMODOMAIN, ACTYL-LYSINE BINDING, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2, EPIGENETICS
4qsx:A (SER979) to (GLU1091) STRUCTURE OF THE BROMODOMAIN OF HUMAN ATPASE FAMILY AAA DOMAIN- CONTAINING PROTEIN 2 (ATAD2) IN COMPLEX WITH 3'-DEOXY THYMIDINE | STRUCTURAL GENOMICS CONSORTIUM (SGC), SIGNALING PROTEIN, BROMODOMAIN, ACTYL-LYSINE BINDING, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2, EPIGENETICS
5etb:A (THR631) to (LYS738) CRYSTAL STRUCTURE OF THE HUMAN BRPF1 BROMODOMAIN IN COMPLEX WITH SEED13 | BROMODOMAIN AND PHD FINGER-CONTAINING PROTEIN 1(BRPF1), MONOCYTIC LEUKEMIA ZINC-FINGER (MOZ), INHIBITOR, TRANSCRIPTION, DNA BINDING PROTEIN
5eu1:A (THR23) to (MET121) CRYSTAL STRUCTURE OF BRD9 IN COMPLEX WITH BI-7273 | BROMODOMAIN, INHIBITOR, TRANSCRIPTION
5eu1:B (PRO24) to (MET121) CRYSTAL STRUCTURE OF BRD9 IN COMPLEX WITH BI-7273 | BROMODOMAIN, INHIBITOR, TRANSCRIPTION
4qut:A (MET980) to (GLU1091) STRUCTURE OF THE BROMODOMAIN OF HUMAN ATPASE FAMILY AAA DOMAIN- CONTAINING PROTEIN 2 (ATAD2) COMPLEXED WITH HISTONE H4-K(AC)12 | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, SIGNALING PROTEIN, BROMODOMAIN, ACTYL-LYSINE BINDING, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2, EPIGENETICS, HISTONE, BROMODOMAIN- HISTONE, STRUCTURAL GENOMICS CONSORTIUM (SGC)
5eva:A (THR631) to (LYS738) CRYSTAL STRUCTURE OF THE HUMAN BRPF1 BROMODOMAIN IN COMPLEX WITH SEED16 | BROMODOMAIN AND PHD FINGER-CONTAINING PROTEIN 1(BRPF1), MONOCYTIC LEUKEMIA ZINC-FINGER (MOZ), INHIBITOR, TRANSCRIPTION, DNA BINDING PROTEIN
5f1h:A (THR23) to (MET133) CRYSTAL STRUCTURE OF THE BRD9 BROMODAMIAN IN COMPLEX WITH BI-9564. | BROMODOMAIN, INHIBITOR, TRANSCRIPTION
5f1h:B (THR23) to (MET121) CRYSTAL STRUCTURE OF THE BRD9 BROMODAMIAN IN COMPLEX WITH BI-9564. | BROMODOMAIN, INHIBITOR, TRANSCRIPTION
5f1l:A (THR23) to (MET121) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF BRD9 IN COMPLEX WITH COMPOUND 9. | BROMODOMAIN, INHIBITOR, TRANSCRIPTION
5f25:A (THR23) to (SER134) CRYSTAL STRUCTURE OF THE BRD9 BROMODOMAIN IN COMPLEX WITH COMPOUND 4. | BROMODOMAIN, INHIBITOR, TRANSCRIPTION
5f25:B (THR23) to (MET121) CRYSTAL STRUCTURE OF THE BRD9 BROMODOMAIN IN COMPLEX WITH COMPOUND 4. | BROMODOMAIN, INHIBITOR, TRANSCRIPTION
5f2p:A (THR23) to (SER134) CRYSTAL STRUCTURE OF THE BRD9 BROMODOMAIN IN COMPLEX WITH COMPOUND 3. | BROMODOMAIN, INHIBITOR, REGULATORY PROTEINS, TRANSCRIPTION
5f2p:B (PRO24) to (SER134) CRYSTAL STRUCTURE OF THE BRD9 BROMODOMAIN IN COMPLEX WITH COMPOUND 3. | BROMODOMAIN, INHIBITOR, REGULATORY PROTEINS, TRANSCRIPTION
4qy4:C (LEU1383) to (LYS1487) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN SMARCA2 | SMARCA2 BAF190B BRM SNF2A SNF2L2, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, UNKNOWN FUNCTION
4qyl:A (THR6) to (GLN99) CRYSTAL STRUCTURE OF THE HUMAN BRPF1 BROMODOMAIN IN COMPLEX WITH A HISTONE H2AK5AC PEPTIDE | BROMODOMAIN-PHD FINGER PROTEIN 1 (BRPF1), HISTONE ACETYLTRANSFERASE (HAT), MONOCYTIC LEUKEMIA ZINC-FINGER (MOZ), EPIGENETICS, CHROMATIN READER, BROMODOMAIN, HISTONE POST-TRANSCRIPTIONAL MODIFICATION (PTM) READER DOMAIN, ACETYLLYSINE, NUCLEUS, PROTEIN BINDING
4qyl:B (THR6) to (GLN99) CRYSTAL STRUCTURE OF THE HUMAN BRPF1 BROMODOMAIN IN COMPLEX WITH A HISTONE H2AK5AC PEPTIDE | BROMODOMAIN-PHD FINGER PROTEIN 1 (BRPF1), HISTONE ACETYLTRANSFERASE (HAT), MONOCYTIC LEUKEMIA ZINC-FINGER (MOZ), EPIGENETICS, CHROMATIN READER, BROMODOMAIN, HISTONE POST-TRANSCRIPTIONAL MODIFICATION (PTM) READER DOMAIN, ACETYLLYSINE, NUCLEUS, PROTEIN BINDING
4qyl:C (THR6) to (GLN99) CRYSTAL STRUCTURE OF THE HUMAN BRPF1 BROMODOMAIN IN COMPLEX WITH A HISTONE H2AK5AC PEPTIDE | BROMODOMAIN-PHD FINGER PROTEIN 1 (BRPF1), HISTONE ACETYLTRANSFERASE (HAT), MONOCYTIC LEUKEMIA ZINC-FINGER (MOZ), EPIGENETICS, CHROMATIN READER, BROMODOMAIN, HISTONE POST-TRANSCRIPTIONAL MODIFICATION (PTM) READER DOMAIN, ACETYLLYSINE, NUCLEUS, PROTEIN BINDING
4qyl:D (THR6) to (GLN99) CRYSTAL STRUCTURE OF THE HUMAN BRPF1 BROMODOMAIN IN COMPLEX WITH A HISTONE H2AK5AC PEPTIDE | BROMODOMAIN-PHD FINGER PROTEIN 1 (BRPF1), HISTONE ACETYLTRANSFERASE (HAT), MONOCYTIC LEUKEMIA ZINC-FINGER (MOZ), EPIGENETICS, CHROMATIN READER, BROMODOMAIN, HISTONE POST-TRANSCRIPTIONAL MODIFICATION (PTM) READER DOMAIN, ACETYLLYSINE, NUCLEUS, PROTEIN BINDING
3c1m:A (VAL45) to (LEU126) CYRSTAL STRUCTURE OF THREONINE-SENSITIVE ASPARTOKINASE FROM METHANOCOCCUS JANNASCHII WITH MGAMP-PNP AND L-ASPARTATE | KINASE, ALLOSTERIC INHIBITION, THREONINE-SENSITIVE, ACT DOMAIN, AMINO-ACID BIOSYNTHESIS, THREONINE BIOSYNTHESIS, TRANSFERASE
3c1m:C (VAL45) to (ILE125) CYRSTAL STRUCTURE OF THREONINE-SENSITIVE ASPARTOKINASE FROM METHANOCOCCUS JANNASCHII WITH MGAMP-PNP AND L-ASPARTATE | KINASE, ALLOSTERIC INHIBITION, THREONINE-SENSITIVE, ACT DOMAIN, AMINO-ACID BIOSYNTHESIS, THREONINE BIOSYNTHESIS, TRANSFERASE
3c1m:D (GLU44) to (LEU126) CYRSTAL STRUCTURE OF THREONINE-SENSITIVE ASPARTOKINASE FROM METHANOCOCCUS JANNASCHII WITH MGAMP-PNP AND L-ASPARTATE | KINASE, ALLOSTERIC INHIBITION, THREONINE-SENSITIVE, ACT DOMAIN, AMINO-ACID BIOSYNTHESIS, THREONINE BIOSYNTHESIS, TRANSFERASE
5fb0:A (GLU774) to (PHE872) CRYSTAL STRUCTURE OF A PHD FINGER BOUND TO HISTONE H3 T3PH PEPTIDE | ZINC FINGER PROTEIN, BROMODOMAIN, TRANSCRIPTION-STRUCTURAL PROTEIN COMPLEX
5fb0:C (GLU774) to (PHE872) CRYSTAL STRUCTURE OF A PHD FINGER BOUND TO HISTONE H3 T3PH PEPTIDE | ZINC FINGER PROTEIN, BROMODOMAIN, TRANSCRIPTION-STRUCTURAL PROTEIN COMPLEX
5fb1:A (PRO773) to (ALA873) CRYSTAL STRUCTURE OF A PHD FINGER BOUND TO HISTONE H3 K9ME3 PEPTIDE | ZINC FINGER PROTEIN, BROMODOMAIN, TRANSCRIPTION-STRUCTURAL PROTEIN COMPLEX
3c20:B (GLU44) to (ILE125) CRYSTAL STRUCTURE OF THREONINE-SENSITIVE ASPARTOKINASE FROM METHANOCOCCUS JANNASCHII WITH L-ASPARTATE | KINASE, ALLOSETRIC INHIBITION, THERONINE-SENSITIVE, ACT DOMAIN, AMINO-ACID BIOSYNTHESIS, THREONINE BIOSYNTHESIS, TRANSFERASE
5fe0:A (ASP724) to (GLY828) CRYSTAL STRUCTURE OF HUMAN PCAF BROMODOMAIN IN COMPLEX WITH ACETYLLYSINE | SIGNALING PROTEIN, BROMODOMAIN, HISTONE ACETYLTRANSFERASE KAT2B, HISTONE, ACETYLATION, ACETYLLYSINE, EPIGENETICS, STRUCTURAL GENOMICS CONSORTIUM (SGC)
5fe0:B (ASP724) to (GLY828) CRYSTAL STRUCTURE OF HUMAN PCAF BROMODOMAIN IN COMPLEX WITH ACETYLLYSINE | SIGNALING PROTEIN, BROMODOMAIN, HISTONE ACETYLTRANSFERASE KAT2B, HISTONE, ACETYLATION, ACETYLLYSINE, EPIGENETICS, STRUCTURAL GENOMICS CONSORTIUM (SGC)
5fe1:A (ASP724) to (GLY828) CRYSTAL STRUCTURE OF HUMAN PCAF BROMODOMAIN IN COMPLEX WITH FRAGMENT BR004 (FRAGMENT 1) | SIGNALING PROTEIN, BROMODOMAIN, HISTONE ACETYLTRANSFERASE KAT2B, HISTONE, ACETYLATION, ACETYLLYSINE, EPIGENETICS, STRUCTURAL GENOMICS CONSORTIUM (SGC)
5fe1:B (ARG723) to (GLY828) CRYSTAL STRUCTURE OF HUMAN PCAF BROMODOMAIN IN COMPLEX WITH FRAGMENT BR004 (FRAGMENT 1) | SIGNALING PROTEIN, BROMODOMAIN, HISTONE ACETYLTRANSFERASE KAT2B, HISTONE, ACETYLATION, ACETYLLYSINE, EPIGENETICS, STRUCTURAL GENOMICS CONSORTIUM (SGC)
5fe5:B (ASP724) to (GLY828) CRYSTAL STRUCTURE OF HUMAN PCAF BROMODOMAIN IN COMPLEX WITH FRAGMENT MB093 (FRAGMENT 7) | SIGNALING PROTEIN, BROMODOMAIN, HISTONE ACETYLTRANSFERASE KAT2B, HISTONE, ACETYLATION, ACETYLLYSINE, EPIGENETICS, STRUCTURAL GENOMICS CONSORTIUM (SGC)
5fe7:B (ARG723) to (GLY828) CRYSTAL STRUCTURE OF HUMAN PCAF BROMODOMAIN IN COMPLEX WITH FRAGMENT ZB2216 (FRAGMENT 11) | SIGNALING PROTEIN, BROMODOMAIN, HISTONE ACETYLTRANSFERASE KAT2B, HISTONE, ACETYLATION, ACETYLLYSINE, EPIGENETICS, STRUCTURAL GENOMICS CONSORTIUM (SGC)
5fe8:A (ASP724) to (GLY828) CRYSTAL STRUCTURE OF HUMAN PCAF BROMODOMAIN IN COMPLEX WITH COMPOUND SL1126 (COMPOUND 12) | SIGNALING PROTEIN, BROMODOMAIN, HISTONE ACETYLTRANSFERASE KAT2B, HISTONE, ACETYLATION, ACETYLLYSINE, EPIGENETICS, STRUCTURAL GENOMICS CONSORTIUM (SGC)
5fe9:B (ARG723) to (GLY828) CRYSTAL STRUCTURE OF HUMAN PCAF BROMODOMAIN IN COMPLEX WITH COMPOUND SL1122 (COMPOUND 13) | SIGNALING PROTEIN, BROMODOMAIN, HISTONE ACETYLTRANSFERASE KAT2B, HISTONE, ACETYLATION, ACETYLLYSINE, EPIGENETICS, STRUCTURAL GENOMICS CONSORTIUM (SGC)
5ffw:A (THR631) to (GLN724) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BRPF1 IN COMPLEX WITH H4K5ACK8AC HISTONE PEPTIDE | PEREGRIN, MOZ-MORF COMPLEX, TRANSCRIPTION
5fh6:C (THR656) to (LEU763) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN PB1 IN COMPLEX WITH COMPOUND 10 | PBRM1, BRG1-ASSOCIATED FACTOR 180, TRANSCRIPTION, CHROMATIN REMODELING
3crd:A (VAL26) to (LEU76) NMR STRUCTURE OF THE RAIDD CARD DOMAIN, 15 STRUCTURES | CASPASE RECRUITMENT DOMAIN, APOPTOSIS, HOMOPHILIC INTERACTION
3nxb:A (ASP439) to (LYS537) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CECR2 | STRUCTURAL GENOMICS CONSORTIUM, SGC, CECR2, CAT EYE SYNDROME CHROMOSOME REGION CANDIDATE 2, BROMODOMAIN, STRUCTURAL GENOMICS, TRANSCRIPTION
3nxb:B (ASP438) to (LYS537) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CECR2 | STRUCTURAL GENOMICS CONSORTIUM, SGC, CECR2, CAT EYE SYNDROME CHROMOSOME REGION CANDIDATE 2, BROMODOMAIN, STRUCTURAL GENOMICS, TRANSCRIPTION
3o33:B (PRO902) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMO IN THE FREE STATE | PHD FINGER, BROMODOMAIN, TRIM24, BREAST CANCER, TRANSCRIPTION
3o33:C (PRO902) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMO IN THE FREE STATE | PHD FINGER, BROMODOMAIN, TRIM24, BREAST CANCER, TRANSCRIPTION
3o35:A (PRO902) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMO COMPLEXED WITH H3(23-31)K27AC PEPTIDE | TRIM24, PHD FINGER, BROMODOMAIN, H3K27 ACETYLATION, BREAST CANCER, TRANSCRIPTION-PROTEIN BINDING COMPLEX
3o35:B (PRO902) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMO COMPLEXED WITH H3(23-31)K27AC PEPTIDE | TRIM24, PHD FINGER, BROMODOMAIN, H3K27 ACETYLATION, BREAST CANCER, TRANSCRIPTION-PROTEIN BINDING COMPLEX
3o36:A (PRO902) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMO COMPLEXED WITH H4(14-19)K16AC PEPTIDE | TRIM24, PHD FINGER, BROMODOMAIN, H4K16 ACETYLATION, BREAST CANCER, TRANSCRIPTION-PROTEIN BINDING COMPLEX
3o36:B (PRO902) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMO COMPLEXED WITH H4(14-19)K16AC PEPTIDE | TRIM24, PHD FINGER, BROMODOMAIN, H4K16 ACETYLATION, BREAST CANCER, TRANSCRIPTION-PROTEIN BINDING COMPLEX
3o37:A (PRO902) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMO COMPLEXED WITH H3(1-10)K4 PEPTIDE | TRIM24, PHD FINGER, BROMODOMAIN, UNMODIFIED H3K4, BREAST CANCER, TRANSCRIPTION, TRANSCRIPTION-PROTEIN BINDING COMPLEX
3o37:B (PRO902) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMO COMPLEXED WITH H3(1-10)K4 PEPTIDE | TRIM24, PHD FINGER, BROMODOMAIN, UNMODIFIED H3K4, BREAST CANCER, TRANSCRIPTION, TRANSCRIPTION-PROTEIN BINDING COMPLEX
3o37:C (PRO902) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMO COMPLEXED WITH H3(1-10)K4 PEPTIDE | TRIM24, PHD FINGER, BROMODOMAIN, UNMODIFIED H3K4, BREAST CANCER, TRANSCRIPTION, TRANSCRIPTION-PROTEIN BINDING COMPLEX
3o37:D (THR901) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMO COMPLEXED WITH H3(1-10)K4 PEPTIDE | TRIM24, PHD FINGER, BROMODOMAIN, UNMODIFIED H3K4, BREAST CANCER, TRANSCRIPTION, TRANSCRIPTION-PROTEIN BINDING COMPLEX
4cos:A (THR150) to (CYS255) CRYSTAL STRUCTURE OF THE PHD-BROMO-PWWP CASSETTE OF HUMAN PRKCBP1 | TRANSCRIPTION, PHD DOMAIN, BROMO DOMAIN, PWWP DOMAIN
5g4r:A (LEU630) to (GLN724) BROMODOMAIN OF HUMAN BRPF1 WITH N-1,3-DIMETHYL-6-2R-2- METHYLPIPERAZIN-1-YL-2-OXO-2,3-DIHYDRO-1H-1,3-BENZODIAZOL- 5-YL-2-METHOXYBENZAMIDE | TRANSCRIPTION
5g4s:A (THR631) to (GLY726) BROMODOMAIN OF HUMAN BRPF1 WITH N-1,3-DIMETHYL-6-2R-2- METHYLPIPERAZIN-1-YL-2-OXO-2,3-DIHYDRO-1H-1,3-BENZODIAZOL- 5-YL-N-ETHYL-2-METHOXYBENZAMIDE | TRANSCRIPTION
4cup:A (LYS1868) to (THR1968) CRYSTAL STRUCTURE OF HUMAN BAZ2B IN COMPLEX WITH FRAGMENT-1 N09421 | TRANSCRIPTION
4cur:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF HUMAN BAZ2B IN COMPLEX WITH FRAGMENT-3 N09555 | TRANSCRIPTION
4cus:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF HUMAN BAZ2B IN COMPLEX WITH FRAGMENT-4 N09496 | TRANSCRIPTION
4cuu:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF HUMAN BAZ2B IN COMPLEX WITH FRAGMENT-6 N09645 | TRANSCRIPTION
3dai:A (SER979) to (LEU1093) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF THE HUMAN ATAD2 | ATPASE FAMILY, AAA DOMAIN CONTAINING 2, ANCCA, AAA+ NUCLEAR COREGULATOR CANCER-ASSOCIATED PRO2000 PROTEIN, TWO AAA DOMAIN CONTAINING PROTEIN, SGC, STRUCTURAL GENOMICS CONSORTIUM, ATP- BINDING, BROMODOMAIN, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SIGNALING PROTEIN
4ts8:A (MET1095) to (GLU1188) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CREBBP IN COMPLEX WITH XZ08 | TRANSCRIPTION, INHIBITOR, TRANSFERASE
4tt2:A (GLN981) to (LEU1093) CRYSTAL STRUCTURE OF ATAD2A BROMODOMAIN COMPLEXED WITH H4(1-20)K5AC PEPTIDE | BROMODOMAIN-ACETYLATED HISTONE COMPLEX, GENE REGULATION
4tt4:A (SER979) to (GLU1091) CRYSTAL STRUCTURE OF ATAD2A BROMODOMAIN COMPLEXED WITH H3(1-21)K14AC PEPTIDE | BROMODOMAIN-ACETYLATED HISTONE COMPLEX, GENE REGULATION
4tt4:B (SER979) to (GLU1091) CRYSTAL STRUCTURE OF ATAD2A BROMODOMAIN COMPLEXED WITH H3(1-21)K14AC PEPTIDE | BROMODOMAIN-ACETYLATED HISTONE COMPLEX, GENE REGULATION
4tt6:A (SER979) to (LEU1093) CRYSTAL STRUCTURE OF ATAD2A BROMODOMAIN DOUBLE MUTANT N1063A-Y1064A IN APO FORM | ACETYLLYSINE READER DEFICIENT BROMODOMAIN, GENE REGULATION
4tte:A (SER979) to (GLU1091) CRYSTAL STRUCTURE OF ATAD2A BROMODOMAIN COMPLEXED WITH METHYL 3-AMINO- 5-(3,5-DIMETHYL-1,2-OXAZOL-4-YL)BENZOATE | ATAD2 BROMODOMAIN INHIBITOR COMPLEX, GENE REGULATION
4tu4:A (SER979) to (GLU1091) CRYSTAL STRUCTURE OF ATAD2A BROMODOMAIN COMPLEXED WITH 3-(3,5- DIMETHYL-1,2-OXAZOL-4-YL)-5-[(PHENYLSULFONYL)AMINO]BENZOICACID | ATAD2A - BROMODOMAIN- INHIBITOR COMPLEX, GENE REGULATION
3oni:A (LEU346) to (MET453) CRYSTAL STRUCTURE OF THE SECOND BROMODOMAIN OF HUMAN BRD2 IN COMPLEX WITH THE INHIBITOR JQ1 | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, BROMODOMAIN, INHIBITION, PROBE, CELL CYCLE
4tyl:A (SER979) to (GLU1091) FRAGMENT-BASED SCREENING OF THE BROMODOMAIN OF ATAD2 | BROMODOMAIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4tz8:A (SER979) to (LEU1093) STRUCTURE OF HUMAN ATAD2 BROMODOMAIN BOUND TO FRAGMENT INHIBITOR | ATAD2, BROMODOMAIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3dwy:A (MET1095) to (GLU1188) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CREBBP | BROMODOMAIN, CREB BINDING PROTEIN, STRUCTURAL GENOMICS CONSORTIUM, SGC, ACTIVATOR, DISEASE MUTATION, HOST-VIRUS INTERACTION, METAL- BINDING, METHYLATION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, ZINC-FINGER
3dwy:B (MET1095) to (GLU1188) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CREBBP | BROMODOMAIN, CREB BINDING PROTEIN, STRUCTURAL GENOMICS CONSORTIUM, SGC, ACTIVATOR, DISEASE MUTATION, HOST-VIRUS INTERACTION, METAL- BINDING, METHYLATION, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, ZINC-FINGER
3p1c:B (MET1095) to (GLU1188) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CREBBP IN COMPLEX WITH ACETYLATED LYSINE | STRUCTURAL GENOMICS CONSORTIUM, CBP, CREBBP, CREB BINDING PROTEIN ISOFORM A, KAT3A, RSTS, RST, BROMODOMAIN, SGC, TRANSCRIPTION
3p41:A (ASN66) to (SER196) CRYSTAL STRUCTURE OF POLYPRENYL SYNTHETASE FROM PSEUDOMONAS FLUORESCENS PF-5 COMPLEXED WITH MAGNESIUM AND ISOPRENYL PYROPHOSPHATE | STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, NEW YORK STRUCTURAL GENOMIX RESEARCH CONSORTIUM, NYSGXRC, ISOPRENE BIOSYNTHESIS, TRANSFERASE, PSI-2, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS
5i1q:A (ASP1503) to (GLU1606) SECOND BROMODOMAIN OF TAF1 BOUND TO A PYRROLOPYRIDONE COMPOUND | TAF1(2) SECOND BROMODOMAIN OF TAF1 SMALL-MOLECULE LIGAND BOUND, PROTEIN BINDING-INHIBITOR COMPLEX
5i29:A (ASP1501) to (GLU1606) TAF1(2) BOUND TO A PYRROLOPYRIDONE COMPOUND | TAF1(2), SECOND BROMODOMAIN OF TAF1, INHIBITOR-BOUND, PROTEIN BINDING-INHIBITOR COMPLEX
5i40:A (THR23) to (LYS123) BRD9 IN COMPLEX WITH CPD1 (6-METHYL-1,6-DIHYDRO-7H-PYRROLO[2,3- C]PYRIDIN-7-ONE) | BROMODOMAIN INHIBITOR EPIGENETICS STRUCTURE-BASED DRUG DESIGN, RNA BINDING PROTEIN
4uit:A (THR23) to (SER122) BROMODOMAIN OF HUMAN BRD9 WITH 7-(3,4-DIMETHOXYPHENYL)-2-(4- METHANESULFONYLPIPERAZINE-1-CARBONYL)-5-METHYL-4H,5H- THIENO-3,2-C-PYRIDIN-4-ONE | TRANSCRIPTION, BRD9, INHIBITOR, HISTONE, EPIGENETIC READER, BROMODOMAIN
4uiu:A (THR23) to (SER122) BROMODOMAIN OF HUMAN BRD9 WITH 7-(3,4-DIMETHOXYPHENYL)-N-(1, 1-DIOXO-1-THIAN-4-YL)-5-METHYL-4-OXO-4H,5H-THIENO-3,2-C- PYRIDINE-2-CARBOXAMIDE | TRANSCRIPTION, BRD9, INHIBITOR, HISTONE, EPIGENETIC READER, BROMODOMAIN
4uiv:A (THR23) to (SER122) BROMODOMAIN OF HUMAN BRD9 WITH N-(1,1-DIOXO-1-THIAN-4-YL)-5- METHYL-4-OXO-7-3-(TRIFLUOROMETHYL)PHENYL-4H,5H-THIENO-3,2- C-PYRIDINE-2-CARBOXIMIDAMIDE | TRANSCRIPTION, INHIBITOR, HISTONE, EPIGENETIC READER
4uiw:A (THR23) to (SER122) BROMODOMAIN OF HUMAN BRD9 WITH N-(1,1-DIOXO-1-THIAN-4-YL)-5- ETHYL-4-OXO-7-3-(TRIFLUOROMETHYL)PHENYL-4H,5H-THIENO-3,2-C- PYRIDINE-2-CARBOXIMIDAMIDE | TRANSCRIPTION, INHIBITOR, HISTONE, EPIGENETIC READER
4uix:C (THR60) to (LYS160) N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH 7-(3,4- DIMETHOXYPHENYL)-N-(1,1-DIOXO-1-THIAN-4-YL)-5-METHYL-4-OXO- 4H,5H-THIENO-3,2-C-PYRIDINE-2-CARBOXAMIDE | TRANSCRIPTION, INHIBITOR, HISTONE, EPIGENETIC READER, BROMODOMAIN, BRD4, BROMODOMAIN CONTAINING PROTEIN 4, ANTAGONIST
5i6e:A (LYS837) to (GLU905) CRYSTAL STRUCTURE OF THE CENTRAL DOMAIN OF YEAST ACETYL-COA CARBOXYLASE | CARBOXYLASE, FATTY ACID METABOLISM, MULTIENZYME, CARRIER PROTEIN- DEPENDENT ENZYME, LIGASE
5i7x:A (THR23) to (SER122) BRD9 IN COMPLEX WITH CPD2 (N,N-DIMETHYL-3-(6-METHYL-7-OXO-6,7-DIHYDRO- 1H-PYRROLO[2,3-C]PYRIDIN-4-YL)BENZAMIDE) | BROMODOMAIN INHIBITOR EPIGENETICS STRUCTURE-BASED DRUG DESIGN, RNA BINDING PROTEIN
5i7y:A (THR23) to (SER122) BRD9 IN COMPLEX WITH CPD4 ((E)-3-(6-(BUT-2-EN-1-YL)-7-OXO-6,7-DIHYDRO- 1H-PYRROLO[2,3-C]PYRIDIN-4-YL)-N,N-DIMETHYLBENZAMIDE) | BRD9, BROMODOMAIN, EPIGENETICS, STRUCTURE-BASED DESIGN, TRANSCRIPTION
5i86:A (LYS1086) to (LEU1196) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CREBBP BOUND TO THE BENZODIAZEPINONE G02778174 | BROMODOMAIN INHIBITOR, PROTEIN BINDING-INHIBITOR COMPLEX
5i86:B (LYS1086) to (LEU1196) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CREBBP BOUND TO THE BENZODIAZEPINONE G02778174 | BROMODOMAIN INHIBITOR, PROTEIN BINDING-INHIBITOR COMPLEX
5i89:A (PRO1087) to (ILE1189) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CREBBP BOUND TO THE BENZODIAZEPINONE G02857790 | BROMODOMAIN INHIBITOR, PROTEIN BINDING-INHIBITOR COMPLEX
5i8g:A (LYS1086) to (GLU1188) CBP IN COMPLEX WITH CPD637 ((R)-4-METHYL-6-(1-METHYL-3-(1-METHYL-1H- PYRAZOL-4-YL)-1H-INDAZOL-5-YL)-1,3,4,5-TETRAHYDRO-2H-BENZO[B][1, 4]DIAZEPIN-2-ONE) | CREBBP, BROMODOMAIN, EPIGENETICS, STRUCTURE-BASED DRUG DESIGN, TRANSCRIPTION-PROTEIN BINDING COMPLEX
5ig6:A (ASP346) to (MET453) ULTRA-HIGH RESOLUTION CRYSTAL STRUCTURE OF SECOND BROMODOMAIN OF BRD2 IN COMPLEX WITH INHIBITOR 6B3 | BET-FAMILY, INHIBITOR, TRANSCRIPTION
5igl:A (GLY1513) to (LEU1650) CRYSTAL STRUCTURE OF THE SECOND BROMODOMAIN OF HUMAN TAF1L IN COMPLEX WITH BROMOSPORINE (BSP) | TRANSCRIPTION, TAF1/TAFII250, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
5igm:A (THR139) to (MET236) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BRD9 IN COMPLEX WITH BROMOSPORINE (BSP) | CHROMATIN REMODELING, TRANSCRIPTION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
5igm:B (PRO140) to (MET237) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BRD9 IN COMPLEX WITH BROMOSPORINE (BSP) | CHROMATIN REMODELING, TRANSCRIPTION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
5ign:A (THR23) to (MET120) CRYSTAL STRUCTURE OF HUMAN BRD9 BROMODOMAIN IN COMPLEX WITH LP99 CHEMICAL PROBE | LYSINE-ACETYLATED HISTONE BINDING, CHROMATIN REGULATOR, TRANSCRIPTION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
5ign:B (PRO24) to (MET121) CRYSTAL STRUCTURE OF HUMAN BRD9 BROMODOMAIN IN COMPLEX WITH LP99 CHEMICAL PROBE | LYSINE-ACETYLATED HISTONE BINDING, CHROMATIN REGULATOR, TRANSCRIPTION, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
5ii2:A (THR656) to (GLU764) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN POLYBROMO (PB1) IN COMPLEX WITH 2-(3,4-DIHYDROXYPHENYL)-5,7-DIHYDROXY-4H-CHROMEN-4-ONE | BROMODOMAIN, COMPLEX, SMALL MOLECULE, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
3q2f:A (LYS1868) to (LYS1970) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BAZ2B IN COMPLEX WITH A TRIAZOLO LIGAND | BAZB2, BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN, 2B, KIAA1476, WALP4, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
4uyg:D (LEU350) to (MET453) C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH I-BET726 (GSK1324726A) | TRANSCRIPTION, INHIBITOR, HISTONE, EPIGENETIC READER, BET, BRD2
3qzs:A (THR70) to (ALA174) CRYSTAL STRUCTURE OF BPTF BROMO IN COMPLEX WITH HISTONE H4K16AC - FORM I | PROTEIN-PEPTIDE COMPLEX, TRANSCRIPTION-NUCLEAR PROTEIN COMPLEX
3qzs:B (THR70) to (ALA174) CRYSTAL STRUCTURE OF BPTF BROMO IN COMPLEX WITH HISTONE H4K16AC - FORM I | PROTEIN-PEPTIDE COMPLEX, TRANSCRIPTION-NUCLEAR PROTEIN COMPLEX
3qzt:A (THR70) to (LYS173) CRYSTAL STRUCTURE OF BPTF BROMO IN COMPLEX WITH HISTONE H4K16AC - FORM II | PROTEIN-PEPTIDE COMPLEX, ALL ALPHA HELIX, TRANSCRIPTION, HISTONE H4, NUCLEAR, TRANSCRIPTION-NUCLEAR PROTEIN COMPLEX
4flp:A (VAL39) to (MET133) CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRDT IN COMPLEX WITH THE INHIBITOR JQ1 | BRDT, BROMODOMAIN CONTAINING PROTEIN TESTIS SPECIFIC, NUCLEUS, TRANSCRIPTION, TRANSCRIPTION REGULATION, STRUCTURAL GENOMICS CONSORTIUM, SGC, BROMODOMAIN, TRANSCRIPTION REGULATOR-INHIBITOR COMPLEX
4flp:B (THR29) to (MET133) CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRDT IN COMPLEX WITH THE INHIBITOR JQ1 | BRDT, BROMODOMAIN CONTAINING PROTEIN TESTIS SPECIFIC, NUCLEUS, TRANSCRIPTION, TRANSCRIPTION REGULATION, STRUCTURAL GENOMICS CONSORTIUM, SGC, BROMODOMAIN, TRANSCRIPTION REGULATOR-INHIBITOR COMPLEX
3rcw:C (PRO566) to (LEU675) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BRD1 | TRANSCRIPTION, BROMODOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
3rcw:F (PRO566) to (GLU676) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BRD1 | TRANSCRIPTION, BROMODOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
3rh2:A (ASP107) to (SER210) CRYSTAL STRUCTURE OF A TETR-LIKE TRANSCRIPTIONAL REGULATOR (SAMA_0099) FROM SHEWANELLA AMAZONENSIS SB2B AT 2.42 A RESOLUTION | DNA/RNA-BINDING 3-HELICAL BUNDLE, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI- BIOLOGY, DNA BINDING PROTEIN
5khm:A (THR60) to (LEU164) THE FIRST BET BROMODOMAIN OF BRD4 BOUND TO COMPOUND 13 IN A BIVALENT MANNER | BROMODOMAIN, TRANSCRIPTION FACTOR
5ktw:A (LYS1086) to (GLU1188) CREBBP BROMODOMAIN IN COMPLEX WITH CPD 44 (3-((5-ACETYL-1- (CYCLOPROPYLMETHYL)-4,5,6,7-TETRAHYDRO-1H-PYRAZOLO[4,3-C]PYRIDIN-3- YL)AMINO)-N-ISOPROPYLBENZAMIDE) | CREBBP BROMODOMAIN, TRANSFERASE
5ktw:C (LYS1086) to (GLU1188) CREBBP BROMODOMAIN IN COMPLEX WITH CPD 44 (3-((5-ACETYL-1- (CYCLOPROPYLMETHYL)-4,5,6,7-TETRAHYDRO-1H-PYRAZOLO[4,3-C]PYRIDIN-3- YL)AMINO)-N-ISOPROPYLBENZAMIDE) | CREBBP BROMODOMAIN, TRANSFERASE
5l8t:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF BAZ2B BROMODOMAIN IN COMPLEX WITH 3-AMINO-2- METHYLPYRIDINE DERIVATIVE 2 | FOUR HELICAL BUNDLE, TRANSCRIPTION
5l97:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF BAZ2B BROMODOMAIN IN COMPLEX WITH 3-AMINO-2- METHYLPYRIDINE DERIVATIVE 3 | FOUR HELICAL BUNDLE, TRANSCRIPTION
5l99:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF BAZ2B BROMODOMAIN IN COMPLEX WITH 3-AMINO-2- METHYLPYRIDINE DERIVATIVE 6 | FOUR HELICAL BUNDLE, TRANSCRIPTION
5lj0:A (SER979) to (GLU1091) CRYSTAL STRUCTURE OF HUMAN ATAD2 BROMODOMAIN IN COMPLEX WITH 8-(((3R, 4R,5S)-3-((4,4-DIFLUOROCYCLOHEXYL)METHOXY)-5-METHOXYPIPERIDIN-4-YL) AMINO)-3-METHYL-5-(5-METHYLPYRIDIN-3-YL)-1,7-NAPHTHYRIDIN-2(1H)-ONE | INHIBITOR, ATAD2, BROMODOMAIN, EPIGENETICS, ATPASE FAMILY AAA DOMAIN- CONTAINING PROTEIN 2, TRANSCRIPTION
5lvq:A (GLN727) to (GLY828) CRYSTAL STRUCTURE OF HUMAN PCAF BROMODOMAIN IN COMPLEX WITH COMPOUND-D (CPD-D), N-METHYL-2-(TETRAHYDRO-2H-PYRAN-4-YLOXY)BENZAMIDE | SIGNALING PROTEIN, BROMODOMAIN, HISTONE ACETYLTRANSFERASE KAT2B, HISTONE, ACETYLATION, ACETYLLYSINE, EPIGENETICS, STRUCTURAL GENOMICS CONSORTIUM (SGC), TRANSFERASE
5lvq:B (ASP726) to (GLY828) CRYSTAL STRUCTURE OF HUMAN PCAF BROMODOMAIN IN COMPLEX WITH COMPOUND-D (CPD-D), N-METHYL-2-(TETRAHYDRO-2H-PYRAN-4-YLOXY)BENZAMIDE | SIGNALING PROTEIN, BROMODOMAIN, HISTONE ACETYLTRANSFERASE KAT2B, HISTONE, ACETYLATION, ACETYLLYSINE, EPIGENETICS, STRUCTURAL GENOMICS CONSORTIUM (SGC), TRANSFERASE
1n72:A (ASP724) to (GLY828) STRUCTURE AND LIGAND OF A HISTONE ACETYLTRANSFERASE BROMODOMAIN | HISTONE ACETYLTRANSFERASE BROMODOMAIN, 4-HELICAL BUNDLE
4hxk:A (THR60) to (LYS160) BRD4 BROMODOMAIN 1 COMPLEX WITH 6,7-DIHYDROTHIENO[3,2-C]PYRIDIN-5(4H)- YL(1H-IMIDAZOL-1-YL)METHANONE INHIBITOR | BRD4, BROMODOMAIN, FOUR ALPHA HELICES, PROTEIN BINDING-INHIBITOR COMPLEX
4hxr:A (THR60) to (LYS160) BRD4 BROMODOMAIN 1 COMPLEX WITH N-[3-(2-OXO-2,3-DIHYDRO-1,3-THIAZOL-4- YL)PHENYL]THIOPHENE-2-SULFONAMIDE INHIBITOR | BRD4, BROMODOMAIN, FOUR ALPHA HELICES, PROTEIN BINDING-INHIBITOR COMPLEX
4xy8:A (PRO24) to (MET120) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF BRD9 IN COMPLEX WITH A 2- AMINE-9H-PURINE LIGAND | BROMODOMAIN, LIGAND, COMPLEX, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
4yab:A (THR901) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMODOMAIN COMPLEXED WITH 1-METHYL-5- (2-METHYL-1 3-THIAZOL-4-YL)-2 3-DIHYDRO-1H-INDOL-2-ONE (1) | CENTER FOR BIOMOLECULAR STRUCTURE AND FUNCTION, BROMODOMAIN, TRIM24, INHIBITOR, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
4yab:B (THR901) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMODOMAIN COMPLEXED WITH 1-METHYL-5- (2-METHYL-1 3-THIAZOL-4-YL)-2 3-DIHYDRO-1H-INDOL-2-ONE (1) | CENTER FOR BIOMOLECULAR STRUCTURE AND FUNCTION, BROMODOMAIN, TRIM24, INHIBITOR, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
4yax:A (PRO902) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMODOMAIN COMPLEXED WITH N-[6-(4- METHOXYPHENOXY)-1,3-DIMETHYL-2-OXO-2,3-DIHYDRO-1H-1,3-BENZODIAZOL-5- YL]BENZENESULFONAMIDE (5G) | CENTER FOR BIOMOLECULAR STRUCTURE AND FUNCTION, BROMODOMAIN, TRIM24, INHIBITOR, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
4yax:B (PRO902) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMODOMAIN COMPLEXED WITH N-[6-(4- METHOXYPHENOXY)-1,3-DIMETHYL-2-OXO-2,3-DIHYDRO-1H-1,3-BENZODIAZOL-5- YL]BENZENESULFONAMIDE (5G) | CENTER FOR BIOMOLECULAR STRUCTURE AND FUNCTION, BROMODOMAIN, TRIM24, INHIBITOR, TRANSCRIPTION-TRANSCRIPTION INHIBITOR COMPLEX
3tu3:B (SER587) to (ASN683) 1.92 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE FULL-LENGTH SPCU IN COMPLEX WITH FULL-LENGTH EXOU FROM THE TYPE III SECRETION SYSTEM OF PSEUDOMONAS AERUGINOSA | TYPE III SECRETION SYSTEM, PSEUDOMONAS AERUGINOSA, EXOU, SPCU, INFECTIOUS DISEASES, STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, SPCU- CHAPERONE, EXOU - PHOSPHOLIPASE A2, TOXIN-TOXIN CHAPERONE COMPLEX
4yyn:A (ASP1502) to (TYR1607) CRYSTAL STRUCTURE OF TAF1 BD2 BROMODOMAIN BOUND TO A CROTONYLLYSINE PEPTIDE | BROMODOMAIN-CROTONYLLYSINE COMPLEX, PROTEIN BINDING
4yyn:B (ASP1502) to (TYR1607) CRYSTAL STRUCTURE OF TAF1 BD2 BROMODOMAIN BOUND TO A CROTONYLLYSINE PEPTIDE | BROMODOMAIN-CROTONYLLYSINE COMPLEX, PROTEIN BINDING
4kcx:B (ASN30) to (MET133) BRDT IN COMPLEX WITH DINACICLIB | BRDT, BROMODOMAIN CONTAINING PROTEIN TESTIS SPECIFIC, CELL CYCLE- INHIBITOR COMPLEX
3uv5:A (ASP1523) to (TYR1628) CRYSTAL STRUCTURE OF THE TANDEM BROMODOMAINS OF HUMAN TRANSCRIPTION INITIATION FACTOR TFIID SUBUNIT 1 (TAF1) | TANDEM BROMODOMAIN, TAF1, CELL CYCLE GENE 1 PROTEIN, TBP-ASSOCIATED FACTOR 250 KDA, TRANSCRIPTION INITIATION FACTOR TFIID 250 KDA SUBUNIT, TFII-250, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
4ldf:A (SER12) to (ILE112) CRYSTAL STRUCTURE OF CPBRD2 FROM CRYPTOSPORIDIUM, CGD3_3190 | STRUCTURAL GENOMICS CONSORTIUM, SGC, BROMODOMAIN, TRANSFERASE
5a5p:A (SER979) to (GLU1091) CRYSTAL STRUCTURE OF HUMAN ATAD2 BROMODOMAIN IN COMPLEX WITH 8-2-(DIMETHYLAMINO)ETHYLAMINO-3-METHYL-1,2- DIHYDROQUINOLIN-2-ONE | HYDROLASE, INHIBITOR, ATAD2 , BROMODOMAIN, EPIGENETICS, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2
5a7c:D (SER309) to (MET415) CRYSTAL STRUCTURE OF THE SECOND BROMODOMAIN OF HUMAN BRD3 IN COMPLEX WITH COMPOUND | DNA BINDING PROTEIN, BRD3, BROMODOMAIN CONTAINING PROTEIN 3, RING3-LIKE PROTEIN, BRD3 DOMAIN 2
2jbw:A (LYS8) to (TRP86) CRYSTAL STRUCTURE OF THE 2,6-DIHYDROXY-PSEUDO-OXYNICOTINE HYDROLASE. | HYDROLASE, ALPHA/BETA HYDROLASE, META-CLEAVAGE PATHWAY, RETRO- FRIEDEL- CRAFTS ACYLATION, NICOTINE DEGRADATION, HYPOTHETICAL PROTEIN, PLASMID, CATALYTIC TRIAD, C-C BOND CLEAVAGE
2jbw:B (LYS8) to (GLN83) CRYSTAL STRUCTURE OF THE 2,6-DIHYDROXY-PSEUDO-OXYNICOTINE HYDROLASE. | HYDROLASE, ALPHA/BETA HYDROLASE, META-CLEAVAGE PATHWAY, RETRO- FRIEDEL- CRAFTS ACYLATION, NICOTINE DEGRADATION, HYPOTHETICAL PROTEIN, PLASMID, CATALYTIC TRIAD, C-C BOND CLEAVAGE
4n4i:A (GLN156) to (CYS258) CRYSTAL STRUCTURE OF THE BROMO-PWWP OF THE MOUSE ZINC FINGER MYND-TYPE CONTAINING 11 ISOFORM ALPHA IN COMPLEX WITH HISTONE H3.3K36ME3 | TANDEM BROMODOMAIN-ZINC FINGER-PWWP MOTIF, HISTONE H3.3-SPECIFIC, TRANSCRIPTION
5c4q:A (GLU14) to (ARG103) CRYSTAL STRUCTURE ANALYSIS OF BROMODOMAIN FROM LEISHMANIA DONOVANI COMPLEXED WITH BROMOSPORINE | STRUCTURAL GENOMICS CONSORTIUM, SGC, BROMODOMAIN, BROMOSPORINE, LEISHMANIA DONOVANI, TRANSCRIPTION
5c4q:B (LYS13) to (ARG103) CRYSTAL STRUCTURE ANALYSIS OF BROMODOMAIN FROM LEISHMANIA DONOVANI COMPLEXED WITH BROMOSPORINE | STRUCTURAL GENOMICS CONSORTIUM, SGC, BROMODOMAIN, BROMOSPORINE, LEISHMANIA DONOVANI, TRANSCRIPTION
4nyv:A (LYS1086) to (GLU1188) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CREBBP IN COMPLEX WITH A QUINAZOLIN-ONE LIGAND | CREBBP, CREB BINDING, KAT3A, RSTS, RST, BROMODOMAIN, TRANSCRIPTION, STRUCTURAL GENOMICS CONSORTIUM, SGC
4nyv:C (LYS1086) to (GLU1188) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CREBBP IN COMPLEX WITH A QUINAZOLIN-ONE LIGAND | CREBBP, CREB BINDING, KAT3A, RSTS, RST, BROMODOMAIN, TRANSCRIPTION, STRUCTURAL GENOMICS CONSORTIUM, SGC
2yyn:A (THR18) to (LEU121) CRYSTAL STURCTURE OF HUMAN BROMODOMAIN PROTEIN | BROMO DOMAIN, TRANSCRIPTION, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
2yyn:D (THR18) to (LEU121) CRYSTAL STURCTURE OF HUMAN BROMODOMAIN PROTEIN | BROMO DOMAIN, TRANSCRIPTION, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
5cq5:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN PROTEIN 2B (BAZ2B) IN COMPLEX WITH 2,3- ETHYLENEDIOXYBENZOIC ACID (SGC - DIAMOND I04-1 FRAGMENT SCREENING) | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
5cqa:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF BROMODOMAIN ADJACENT TO ZINC FINGER DOMAIN PROTEIN 2B (BAZ2B) IN COMPLEX WITH N-METHYL-2,3- DIHYDROTHIENO[3,4-B][1,4]DIOXINE-5-CARBOXAMIDE (SGC - DIAMOND I04-1 FRAGMENT SCREENING) | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
5dw1:D (SER347) to (MET453) X-RAY CRYSTAL STRUCTURE OF HUMAN BRD2(BD2) IN COMPLEX WITH RVX297 TO 1.55 A RESOLUTION | BROMODOMAIN, PROTEIN BINDING-INHIBITOR COMPLEX
5egu:A (THR60) to (LEU164) FIRST DOMAIN OF HUMAN BROMODOMAIN BRD4 IN COMPLEX WITH INHIBITOR 3- BUTYL-8-(6-BUTYL-5,7-DIMETHYL-[1,2,4]TRIAZOLO[1,5-A]PYRIMIDIN-2- YLSULFANYLMETHYL)-7-ETHYL-3,7-DIHYDROPURINE-2,6-DIONE | INHIBITOR, HISTONE, EPIGENETIC READER, BROMODOMAIN, BRD4, BRD4_BD1, BRD4_BD1 06-NOV, TRANSCRIPTION
5egu:C (THR60) to (LEU164) FIRST DOMAIN OF HUMAN BROMODOMAIN BRD4 IN COMPLEX WITH INHIBITOR 3- BUTYL-8-(6-BUTYL-5,7-DIMETHYL-[1,2,4]TRIAZOLO[1,5-A]PYRIMIDIN-2- YLSULFANYLMETHYL)-7-ETHYL-3,7-DIHYDROPURINE-2,6-DIONE | INHIBITOR, HISTONE, EPIGENETIC READER, BROMODOMAIN, BRD4, BRD4_BD1, BRD4_BD1 06-NOV, TRANSCRIPTION
3mb4:A (THR624) to (GLU732) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN POLY-BROMODOMAIN CONTAINING PROTEIN 1 (PB1) WITH NMP | PB1, POLYBROMO 1 ISOFORM 1, BAF180, POLYBROMO-1D, PBRM1, BRG1- ASSOCIATED FACTOR 180, STRUCTURAL GENOMICS CONSORTIUM, SGC, BROMODOMAIN, CHROMATIN REGULATOR, DNA-BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION
4qsv:A (SER979) to (LEU1093) STRUCTURE OF THE BROMODOMAIN OF HUMAN ATPASE FAMILY AAA DOMAIN- CONTAINING PROTEIN 2 (ATAD2) IN COMPLEX WITH THYMIDINE | STRUCTURAL GENOMICS CONSORTIUM (SGC), SIGNALING PROTEIN, BROMODOMAIN, ACTYL-LYSINE BINDING, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2, EPIGENETICS
3mqm:A (GLU2433) to (SER2546) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN ASH1L | ASH1L, ASH1, KIAA1420, ABSENT SMALL AND HOMEOTIC DISKS PROTEIN 1 HOMOLOG, LYSINE N-METHYLTRANSFERASE 2H, KMT2H, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
3mqm:B (GLU2433) to (SER2546) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN ASH1L | ASH1L, ASH1, KIAA1420, ABSENT SMALL AND HOMEOTIC DISKS PROTEIN 1 HOMOLOG, LYSINE N-METHYLTRANSFERASE 2H, KMT2H, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
5fg4:A (PHE633) to (GLN724) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BRPF1 IN COMPLEX WITH OF-1 CHEMICAL PROBE | PEREGRIN, MOZ-MORF COMPLEX, TRANSCRIPTION
5fh7:B (THR656) to (GLU764) CRYSTAL STRUCTURE OF THE FIFTH BROMODOMAIN OF HUMAN PB1 IN COMPLEX WITH COMPOUND 18 | PBRM1, BRG1-ASSOCIATED FACTOR 180, TRANSCRIPTION, CHROMATIN REMODELING
4cdn:A (GLU234) to (TYR315) CRYSTAL STRUCTURE OF M. MAZEI PHOTOLYASE WITH ITS IN VIVO RECONSTITUTED 8-HDF ANTENNA CHROMOPHORE | LYASE, PHOTOLYASE, DNA REPAIR, METHANOSARCINA MAZEI, ANTENNA CHROMOPHORE, 8-HDF, FAD
4cdn:B (GLU234) to (TYR315) CRYSTAL STRUCTURE OF M. MAZEI PHOTOLYASE WITH ITS IN VIVO RECONSTITUTED 8-HDF ANTENNA CHROMOPHORE | LYASE, PHOTOLYASE, DNA REPAIR, METHANOSARCINA MAZEI, ANTENNA CHROMOPHORE, 8-HDF, FAD
4rvr:A (ASP1869) to (THR1968) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN BAZ2B IN COMPLEX WITH GSK2801 | SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSCRIPTION, ACETYLATED LYSINE BINDING PROTEIN, KIAA1476, WALP4, CHEMICAL PROBE
3o34:A (THR901) to (PRO1006) CRYSTAL STRUCTURE OF TRIM24 PHD-BROMO COMPLEXED WITH H3(13-32)K23AC PEPTIDE | TRIM24, PHD FINGER, BROMODOMAIN, H3K23AC, BREAST CANCER, TRANSCRIPTION-PROTEIN BINDING COMPLEX
4tqn:A (MET1095) to (GLU1188) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CREBBP IN COMPLEX WITH UL04 | TRANSCRIPTION/INHIBITOR, TRANSFERASE
4tu6:A (MET980) to (GLU1092) CRYSTAL STRUCTURE OF APO ATAD2A BROMODOMAIN WITH N1064 ALTERNATE CONFORMATION | BROMODOMAIN- CONSERVED ASPARAGINE CONFORMATIONS, GENE REGULATION
4tu6:C (GLU983) to (GLU1091) CRYSTAL STRUCTURE OF APO ATAD2A BROMODOMAIN WITH N1064 ALTERNATE CONFORMATION | BROMODOMAIN- CONSERVED ASPARAGINE CONFORMATIONS, GENE REGULATION
5hfr:A (LYS307) to (MET415) CRYSTAL STRUCTURE OF THE SECOND BROMODOMAIN H395R MUTANT OF HUMAN BRD3 | TRANSCRIPTION REGULATION, POST TRANSLATIONAL MODIFICATIONS RECOGNITION, TRANSCRIPTION
5hfr:B (SER309) to (MET415) CRYSTAL STRUCTURE OF THE SECOND BROMODOMAIN H395R MUTANT OF HUMAN BRD3 | TRANSCRIPTION REGULATION, POST TRANSLATIONAL MODIFICATIONS RECOGNITION, TRANSCRIPTION
3p1f:A (LYS1086) to (GLU1188) CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN CREBBP IN COMPLEX WITH A HYDROQUINAZOLIN LIGAND | STRUCTURAL GENOMICS CONSORTIUM, SGC, CBP, CREBBP, CREB BINDING PROTEIN ISOFORM A, KAT3A, RSTS, RST, BROMODOMAIN, TRANSCRIPTION
5i8b:A (LYS1086) to (GLU1188) CBP IN COMPLEX WITH CPD23 ((R)-6-(3-(BENZYLOXY)PHENYL)-4-METHYL-1,3,4, 5-TETRAHYDRO-2H-BENZO[B][1,4]DIAZEPIN-2-ONE) | CREBBP, BROMODOMAIN, EPIGENETICS, STRUCTURE-BASED DRUG DESIGN, TRANSCRIPTION-PROTEIN BINDING COMPLEX
3qzv:A (THR70) to (LYS170) CRYSTAL STRUCTURE OF BPTF PHD-LINKER-BROMO IN COMPLEX WITH HISTONE H4K12AC PEPTIDE | PROTEIN-PEPTIDE COMPLEX, ZINC FINGER, ALPHA HELIX BUNDLE, TRANSCRIPTION, HISTONE H4, NUCLEAR, TRANSCRIPTION-NUCLEAR PROTEIN COMPLEX