3rll:A (ILE672) to (TRP741) CRYSTAL STRUCTURE OF THE T877A ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH (S)-N-(4-CYANO-3-(TRIFLUOROMETHYL)PHENYL)-3-(4- CYANONAPHTHALEN-1-YLOXY)-2-HYDROXY-2-METHYLPROPANAMIDE | STEROID RECEPTOR, DHT, TESTOSTERONE, TRANSCRIPTION
1a28:B (PRO686) to (SER754) HORMONE-BOUND HUMAN PROGESTERONE RECEPTOR LIGAND-BINDING DOMAIN | PROGESTERONE RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION
2oax:A (PRO738) to (SER805) CRYSTAL STRUCTURE OF THE S810L MUTANT MINERALOCORTICOID RECEPTOR ASSOCIATED WITH SC9420 | ALDOSTERONE; STEROID RECEPTOR; NUCLEAR RECEPTOR; TRANSCRIPTION FACTOR; ACTIVATING MUTATION, HYPERTENSION; ANTAGONIST; SPIRONOLACTONE
2oax:B (VAL739) to (SER805) CRYSTAL STRUCTURE OF THE S810L MUTANT MINERALOCORTICOID RECEPTOR ASSOCIATED WITH SC9420 | ALDOSTERONE; STEROID RECEPTOR; NUCLEAR RECEPTOR; TRANSCRIPTION FACTOR; ACTIVATING MUTATION, HYPERTENSION; ANTAGONIST; SPIRONOLACTONE
2oax:C (PRO738) to (SER805) CRYSTAL STRUCTURE OF THE S810L MUTANT MINERALOCORTICOID RECEPTOR ASSOCIATED WITH SC9420 | ALDOSTERONE; STEROID RECEPTOR; NUCLEAR RECEPTOR; TRANSCRIPTION FACTOR; ACTIVATING MUTATION, HYPERTENSION; ANTAGONIST; SPIRONOLACTONE
2oax:D (VAL739) to (SER805) CRYSTAL STRUCTURE OF THE S810L MUTANT MINERALOCORTICOID RECEPTOR ASSOCIATED WITH SC9420 | ALDOSTERONE; STEROID RECEPTOR; NUCLEAR RECEPTOR; TRANSCRIPTION FACTOR; ACTIVATING MUTATION, HYPERTENSION; ANTAGONIST; SPIRONOLACTONE
2oax:E (PRO738) to (SER805) CRYSTAL STRUCTURE OF THE S810L MUTANT MINERALOCORTICOID RECEPTOR ASSOCIATED WITH SC9420 | ALDOSTERONE; STEROID RECEPTOR; NUCLEAR RECEPTOR; TRANSCRIPTION FACTOR; ACTIVATING MUTATION, HYPERTENSION; ANTAGONIST; SPIRONOLACTONE
2oax:F (VAL739) to (SER805) CRYSTAL STRUCTURE OF THE S810L MUTANT MINERALOCORTICOID RECEPTOR ASSOCIATED WITH SC9420 | ALDOSTERONE; STEROID RECEPTOR; NUCLEAR RECEPTOR; TRANSCRIPTION FACTOR; ACTIVATING MUTATION, HYPERTENSION; ANTAGONIST; SPIRONOLACTONE
1nhz:A (LEU532) to (SER599) CRYSTAL STRUCTURE OF THE ANTAGONIST FORM OF GLUCOCORTICOID RECEPTOR | PROTIEN-LIGAND COMPLEX, ANTI PARALLEL ALPHA HELIX SANDWICH, HORMONE RECEPTOR
2ax7:A (ILE672) to (TRP741) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN T877A MUTANT IN COMPLEX WITH S-1 | TRANSCRIPTION
3ru0:A (GLU86) to (SER182) COCRYSTAL STRUCTURE OF HUMAN SMYD3 WITH INHIBITOR SINEFUNGIN BOUND | METHYLTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2b1z:A (THR311) to (LEU379) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH 17METHYL-17ALPHA-DIHYDROEQUILENIN AND A GLUCOC INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
3ry9:A (THR0) to (SER68) CRYSTAL STRUCTURE OF THE RESURRECTED ANCESTRAL GLUCOCORTICOID RECEPTOR 1 IN COMPLEX WITH DOC | RESURRECTED PROTEIN, STEROID RECEPTOR, NUCLEAR RECEPTOR, COMMON ANCESTOR, EVOLUTION, STEROID BINDING PROTEIN
3ry9:B (MET1) to (GLN66) CRYSTAL STRUCTURE OF THE RESURRECTED ANCESTRAL GLUCOCORTICOID RECEPTOR 1 IN COMPLEX WITH DOC | RESURRECTED PROTEIN, STEROID RECEPTOR, NUCLEAR RECEPTOR, COMMON ANCESTOR, EVOLUTION, STEROID BINDING PROTEIN
2p15:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER ALPHA LIGAND BINDING DOMAIN WITH THE AGONIST ORTHO-TRIFLUOROMETHYLPHENYLVINYL ESTRADIOL | NULEAR RECEPTOR, LIGAND BINDING DOMAIN, HELIX 12, HORMONE RECEPTOR
4wuy:A (ASP82) to (CYS181) CRYSTAL STRUCTURE OF PROTEIN LYSINE METHYLTRANSFERASE SMYD2 IN COMPLEX WITH LLY-507, A CELL-ACTIVE, POTENT AND SELECTIVE INHIBITOR | SMYD2 - LLY-507, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3erd:B (THR311) to (TRP383) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DIETHYLSTILBESTROL AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ESTROGEN, AGONIST, COACTIVATOR
3erm:E (ALA25) to (SER81) THE CRYSTAL STRUCTURE OF A CONSERVED PROTEIN WITH UNKNOWN FUNCTION FROM PSEUDOMONAS SYRINGAE PV. TOMATO STR. DC3000 | APC85034, PPSPTO1197, SEUDOMONAS SYRINGAE PV. TOMATO STR. DC3000, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, UNKNOWN FUNCTION
3etl:A (PRO13) to (ASP61) RADA RECOMBINASE FROM METHANOCOCCUS MARIPALUDIS IN COMPLEX WITH AMPPNP | RADA, STRAND EXCHANGE PROTEIN, ATPASE, RECOMBINASE, ATP ANALOGUE, ATP-BINDING, DNA DAMAGE, DNA RECOMBINATION, DNA- BINDING, NUCLEOTIDE-BINDING, DNA BINDING PROTEIN, RECOMBINATION
2bj4:B (THR311) to (ALA382) ESTROGEN RECEPTOR ALPHA LBD IN COMPLEX WITH A PHAGE-DISPLAY DERIVED PEPTIDE ANTAGONIST | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, PEPTIDE ANTAGONIST, LIGAND-BINDING DOMAIN (LBD), DNA-BINDING, NUCLEAR PROTEIN STEROID-BINDING
4hlw:A (PRO671) to (SER740) TARGETING THE BINDING FUNCTION 3 (BF3) SITE OF THE HUMAN ANDROGEN RECEPTOR THROUGH VIRTUAL SCREENING. 2. DEVELOPMENT OF 2-((2- PHENOXYETHYL) THIO)-1H-BENZOIMIDAZOLE DERIVATIVES. | NUCLEAR HORMONE RECEPTOR, ANDROGEN BINDING DOMAIN, TRANSCRIPTIONAL FACTOR, TRANSCRIPTION
3s63:A (SER27) to (ARG79) SAPOSIN-LIKE PROTEIN NA-SLP-1 | SAPOSIN, LIPID-BINDING, LIPID BINDING PROTEIN
3s63:B (SER27) to (ARG79) SAPOSIN-LIKE PROTEIN NA-SLP-1 | SAPOSIN, LIPID-BINDING, LIPID BINDING PROTEIN
3s6a:A (GLY114) to (LEU165) FIC PROTEIN FROM NEISSERIA MENINGITIDIS IN COMPLEX WITH AMPPNP | AMPYLATION, ADENYLYLATION, TRANSFERASE
2piq:A (ILE672) to (TYR739) ANDROGEN RECEPTOR LBD WITH SMALL MOLECULE | ANDROGEN RECEPTOR, INHIBITORS COACTIVATOR BINDING AF-2, HORMONE RECEPTOR
1c3u:A (THR367) to (LEU411) T. MARITIMA ADENYLOSUCCINATE LYASE | PURINE BIOSYNTHESIS, LYASE
1c3u:B (THR367) to (LEU411) T. MARITIMA ADENYLOSUCCINATE LYASE | PURINE BIOSYNTHESIS, LYASE
2pnu:A (PRO671) to (SER740) CRYSTAL STRUCTURE OF HUMAN ANDROGEN RECEPTOR LIGAND-BINDING DOMAIN IN COMPLEX WITH EM-5744 | HAR, DHT, ANDROGEN RECEPTOR, LIGAND BINDING DOMAIN, LBD, ANDROGEN, HORMONE/GENE REGULATION COMPLEX
2pog:B (THR311) to (SER395) BENZOPYRANS AS SELECTIVE ESTROGEN RECEPTOR B AGONISTS (SERBAS). PART 2: STRUCTURE ACTIVITY RELATIONSHIP STUDIES ON THE BENZOPYRAN SCAFFOLD. | NUCLEAR RECEPTOR, LIGAND-BINDING, LIPID BINDING PROTEIN
4xi3:A (THR311) to (SER395) ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN IN COMPLEX WITH BAZEDOXIFENE | ESTROGEN RECEPTOR, SERM, BAZEDOXIFENE, BREAST CANCER, NUCLEAR HORMONE RECEPTOR, SIGNALING PROTEIN
1ovl:E (SER363) to (ALA442) CRYSTAL STRUCTURE OF NURR1 LBD | NUUR1, LBD, TRANSCRIPTION
2qa6:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR ALPHA MUTANT 537S COMPLEXED WITH 4-(6-HYDROXY-1H-INDAZOL-3-YL)BENZENE-1,3-DIOL | PROTEIN-LIGAND COMPLEX, TRANSCRIPTION
3g8o:A (PRO686) to (TRP755) PROGESTERONE RECEPTOR WITH BOUND PYRROLIDINE 1 | PROGESTERONE RECEPTOR, STEROID HORMONE RECEPTOR, NUCLEAR RECEPTOR, PR, PROGESTERONE, ALPHA HELICAL SANDWICH, DNA-BINDING, LIPID- BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, STEROID- BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3g8o:B (PRO686) to (TRP755) PROGESTERONE RECEPTOR WITH BOUND PYRROLIDINE 1 | PROGESTERONE RECEPTOR, STEROID HORMONE RECEPTOR, NUCLEAR RECEPTOR, PR, PROGESTERONE, ALPHA HELICAL SANDWICH, DNA-BINDING, LIPID- BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, STEROID- BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
2qr9:A (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED WITH AN OXABICYCLIC DERIVATIVE COMPOUND | PROTEIN-LIGAND COMPLEX, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
4iv2:B (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DYNAMIC WAY-DERIVATIVE, 5A | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4iv4:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH CONSTRAINED WAY-DERIVATIVE, 5B | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4ivn:B (ASN6) to (GLN49) THE VIBRIO VULNIFICUS NANR PROTEIN COMPLEXED WITH MANNAC-6P | ISOMERASE FOLD, NAN OPERON REGULATOR FOR SIALIC ACID CATABOLISM, TRANSCRIPTION REGULATOR
4ivw:B (ALA312) to (SER395) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH CONSTRAINED WAY-DERIVATIVE, 6B | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4ivy:A (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DYNAMIC WAY-DERIVATIVE, 7A | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4ivy:B (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DYNAMIC WAY-DERIVATIVE, 7A | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
2qse:B (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED WITH BURNED MEAT COMPOUND 4-OH-PHIP | PROTEIN-LIGAND COMPLEX, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
4iw6:B (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH CONSTRAINED WAY-DERIVATIVE, 7B | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4iw8:A (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DYNAMIC WAY-DERIVATIVE, 9A | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
4iwc:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DYNAMIC THIOPHENE-DERIVATIVE | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
1e3k:B (PRO686) to (SER754) HUMAN PROGESTERON RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH THE LIGAND METRIBOLONE (R1881) | HUMAN PROGESTERONE RECEPTOR, LIGAND BINDING DOMAIN
1pzn:A (GLY44) to (ALA91) RAD51 (RADA) | HEPTAMERIC RING; HEPTAMER; RING; OLIGOMER; RAD51 POLYMERIZATION MOTIF; HELIX-HAIRPIN-HELIX; DNA REPAIR; DNA RECOMBINATION; ATPASE; HOMOLOGOUS RECOMBINATION, RECOMBINATION
2r6w:A (THR311) to (SER395) ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN COMPLEXED TO A SERM | ESTROGEN RECEPTOR, LIGAND-BINDING DOMAIN, ALTERNATIVE SPLICING, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, POLYMORPHISM, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
2r6w:B (THR311) to (SER395) ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN COMPLEXED TO A SERM | ESTROGEN RECEPTOR, LIGAND-BINDING DOMAIN, ALTERNATIVE SPLICING, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, POLYMORPHISM, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
2r6y:B (THR311) to (SER395) ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A SERM | ESTROGEN RECEPTOR, LIGAND-BINDING DOMAIN, ALTERNATIVE SPLICING, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, POLYMORPHISM, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
4yao:A (THR383) to (TYR434) REDUCED CYPOR MUTANT - G143DEL | CYTOCHROME P450 REDUCTASE, FMN BINDING, SEMIQUINONE, OXIDOREDUCTASE
4yao:B (THR383) to (TYR434) REDUCED CYPOR MUTANT - G143DEL | CYTOCHROME P450 REDUCTASE, FMN BINDING, SEMIQUINONE, OXIDOREDUCTASE
2ecp:B (ASP388) to (VAL447) THE CRYSTAL STRUCTURE OF THE E. COLI MALTODEXTRIN PHOSPHORYLASE COMPLEX | ACARBOSE, DIABETES, PHOSPHORYLASE, MALP, GLYCOSYLTRANSFERASE
1fez:B (THR41) to (ILE97) THE CRYSTAL STRUCTURE OF BACILLUS CEREUS PHOSPHONOACETALDEHYDE HYDROLASE COMPLEXED WITH TUNGSTATE, A PRODUCT ANALOG | HAD-FAMILY ALPHA/BETA CORE DOMAIN, MG(II) BINDING SITE, 5- HELIX BUNDLE, HYDROLASE
1fez:D (THR41) to (ILE97) THE CRYSTAL STRUCTURE OF BACILLUS CEREUS PHOSPHONOACETALDEHYDE HYDROLASE COMPLEXED WITH TUNGSTATE, A PRODUCT ANALOG | HAD-FAMILY ALPHA/BETA CORE DOMAIN, MG(II) BINDING SITE, 5- HELIX BUNDLE, HYDROLASE
1r5k:A (THR311) to (SER395) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH GW5638 | ALPHA HELIX, HELICAL SANDWICH, DNA BINDING PROTEIN
1r5k:B (THR311) to (SER395) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH GW5638 | ALPHA HELIX, HELICAL SANDWICH, DNA BINDING PROTEIN
1r5k:C (THR311) to (SER395) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH GW5638 | ALPHA HELIX, HELICAL SANDWICH, DNA BINDING PROTEIN
1r6q:B (GLN4) to (THR65) CLPNS WITH FRAGMENTS | CLPA, AAA+, N-TERMINAL DOMAIN, CLPS, CRYSTAL, BINDING MECHANISM, CHAPERONE-PROTEIN BINDING COMPLEX
3hlv:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE AND 16-ALPHA-HYDROXY-ESTRONE ((8S,9R,13S,14R, 16R)-3,16-DIHYDROXY-13-METHYL-7,8,9,11,12,14,15, 16-OCTAHYDRO-6H- CYCLOPENTA[A]PHENANTHREN-17-ONE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HYDROXY-ESTRONE, ALTERNATIVE SPLICING, DNA-BINDING, GLYCOPROTEIN, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACTIVATOR, HORMONE, NUCLEAR RECEPTOR
1rdf:A (THR41) to (ALA102) G50P MUTANT OF PHOSPHONOACETALDEHYDE HYDROLASE IN COMPLEX WITH SUBSTRATE ANALOGUE VINYL SULFONATE | HALOACID DEHALOGENASE, SPECIFICITY LOOP, PHOSPHONATASE, SCHIFF-BASE, HYDROLASE
1rdf:D (THR41) to (ILE97) G50P MUTANT OF PHOSPHONOACETALDEHYDE HYDROLASE IN COMPLEX WITH SUBSTRATE ANALOGUE VINYL SULFONATE | HALOACID DEHALOGENASE, SPECIFICITY LOOP, PHOSPHONATASE, SCHIFF-BASE, HYDROLASE
4k7a:A (PRO671) to (TYR739) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH MINOXIDIL | AANDROGEN RECEPTOR, LIGAND BINDING DOMAIN(LBD), STEROID RECEPTOR COACTIVATOR, 5-ALPHA-DIHYDROTESTOSTERONE(DHT), PROSTATE CANCER, TRANSCRIPTION FACTOR, COACTIVATOR BINDING, CYTOSOL, NUCLEAS, TRANSCRIPTION
4ka7:A (THR562) to (ARG642) STRUCTURE OF ORGANELLAR OLIGOPEPTIDASE (E572Q) IN COMPLEX WITH AN ENDOGENOUS SUBSTRATE | PROTEASE, MITOCHONDRIA, CHLOROPLAST, HYDROLASE-HYDROLASE SUBSTRATE COMPLEX
4ka8:A (THR562) to (ARG642) STRUCTURE OF ORGANELLAR OLIGOPEPTIDASE | PROTEASE, MITOCHONDRIA, CHLOROPLAST, HYDROLASE
2vcb:A (ILE778) to (LYS874) FAMILY 89 GLYCOSIDE HYDROLASE FROM CLOSTRIDIUM PERFRINGENS IN COMPLEX WITH PUGNAC | MUCOPOLYSACCHARIDOSIS, ALPHA-N-ACETYLGLUCOSAMINIDASE, FAMILY 89 GLYCOSIDE HYDROLASE, HYDROLASE, GH89, NAGLU, PUGNAC, SANFILIPPO DISEASE
2f77:X (SER6) to (GLU94) SOLUTION STRUCTURE OF THE R55F MUTANT OF M-PMV MATRIX PROTEIN (P10) | 4 ALPHA-HELICES, VIRAL PROTEIN
2vd6:B (SER395) to (THR450) HUMAN ADENYLOSUCCINATE LYASE IN COMPLEX WITH ITS SUBSTRATE N6-(1,2-DICARBOXYETHYL)-AMP, AND ITS PRODUCTS AMP AND FUMARATE. | PURINE BIOSYNTHESIS, LYASE, EPILEPSY, PURINE METABOLISM
1rql:A (THR41) to (ILE97) CRYSTAL STRUCTURE OF PHOSPONOACETALDEHYDE HYDROLASE COMPLEXED WITH MAGNESIUM AND THE INHIBITOR VINYL SULFONATE | SCHIFF-BASE FORMATION; ACID/BASE CATALYSIS; STRUCTURAL ENZYMOLOGY; HAD SUPERFAMILY, HYDROLASE
1rqn:A (THR41) to (ILE97) PHOSPHONOACETALDEHYDE HYDROLASE COMPLEXED WITH MAGNESIUM | SCHIFF-BASE FORMATION; ACID/BASE CATALYSIS; STRUCTURAL ENZYMOLOGY; HAD SUPERFAMILY, HYDROLASE
1rte:A (HIS22) to (THR127) X-RAY STRUCTURE OF CYANIDE DERIVATIVE OF TRUNCATED HEMOGLOBIN N (TRHBN) FROM MYCOBACTERIUM TUBERCULOSIS | TRUNCATED HEMOGLOBIN, OXYGEN STORAGE/TRANSPORT COMPLEX
3hq5:A (PRO686) to (TRP755) PROGESTERONE RECEPTOR BOUND TO AN ALKYLPYRROLIDINE LIGAND. | NUCLEAR RECEPTOR, PROGESTERONE RECEPTOR, PR, ALTERNATIVE SPLICING, CYTOPLASM, DNA-BINDING, ISOPEPTIDE BOND, LIPID- BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, UBL CONJUGATION, ZINC, ZINC- FINGER, HORMONE BINDING PROTEIN
3hq5:B (PRO686) to (SER754) PROGESTERONE RECEPTOR BOUND TO AN ALKYLPYRROLIDINE LIGAND. | NUCLEAR RECEPTOR, PROGESTERONE RECEPTOR, PR, ALTERNATIVE SPLICING, CYTOPLASM, DNA-BINDING, ISOPEPTIDE BOND, LIPID- BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, UBL CONJUGATION, ZINC, ZINC- FINGER, HORMONE BINDING PROTEIN
3uua:A (THR311) to (SER395) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BISPHENOL-AF | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
3uua:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BISPHENOL-AF | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
3uuc:A (THR311) to (ALA382) CRYSTAL STRUCTURE OF HERA-LBD (WT) IN COMPLEX WITH BISPHENOL-C | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
3uuc:C (THR311) to (TRP383) CRYSTAL STRUCTURE OF HERA-LBD (WT) IN COMPLEX WITH BISPHENOL-C | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4za6:A (GLY114) to (GLY182) STRUCTURE OF THE R. ERYTHROPOLIS TRANSCRIPTIONAL REPRESSOR QSDR FROM TETR FAMILY | QUORUM-SENSING, NAHL DEGRADATION, QSDA TRANSCRIPTIONAL REGULATOR, RHODOCOCCUS ERYTHROPOLIS R138, SIGNALING PROTEIN
4za6:B (GLY114) to (GLY182) STRUCTURE OF THE R. ERYTHROPOLIS TRANSCRIPTIONAL REPRESSOR QSDR FROM TETR FAMILY | QUORUM-SENSING, NAHL DEGRADATION, QSDA TRANSCRIPTIONAL REGULATOR, RHODOCOCCUS ERYTHROPOLIS R138, SIGNALING PROTEIN
2fpl:A (PRO13) to (ASP61) RADA RECOMBINASE IN COMPLEX WITH AMP-PNP AND LOW CONCENTRATION OF K+ | ATPASE, PROTEIN-ATP COMPLEX, RADA/ADP COMPLEX, CO-FACTORS, POTASSIUM-DEPENDENCE, RECOMBINATION
1s56:B (HIS22) to (ILE119) CRYSTAL STRUCTURE OF "TRUNCATED" HEMOGLOBIN N (HBN) FROM MYCOBACTERIUM TUBERCULOSIS, SOAKED WITH XE ATOMS | GROUP I TRUNCATED HEMOGLOBIN, OXYGEN STORAGE/TRANSPORT COMPLEX
1s61:B (HIS22) to (THR127) CRYSTAL STRUCTURE OF "TRUNCATED" HEMOGLOBIN N (HBN) FROM MYCOBACTERIUM TUBERCULOSIS, SOAKED WITH BUTYL-ISOCYANIDE | TRUNCATED HEMOGLOBIN, OXYGEN STORAGE/TRANSPORT COMPLEX
1s9p:A (ASN235) to (ALA304) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAIN OF THE ESTROGEN-RELATED RECEPTOR GAMMA IN COMPLEX WITH DIETHYLSTILBESTROL | LIGAND-BINDING DOMAIN, ANTAGONIST COMPLEX, TRANSCRIPTION
2g62:A (GLU72) to (SER142) CRYSTAL STRUCTURE OF HUMAN PTPA | PPP2R4, MGC2184, PP2A, PR53, PTPA, PROTEIN PHOSPHATASE 2A, REGULATORY SUBUNIT B' (PR 53), HYDROLASE ACTIVATOR
1sqn:A (PRO686) to (TRP755) PROGESTERONE RECEPTOR LIGAND BINDING DOMAIN WITH BOUND NORETHINDRONE | PROGESTERONE RECEPTOR; NUCLEAR RECEPTOR; STEROID RECEPTOR; NORETHINDRONE; BIRTH CONTROL, HORMONE/GROWTH FACTOR RECEPTIOR COMPLEX
1sqn:B (PRO686) to (SER754) PROGESTERONE RECEPTOR LIGAND BINDING DOMAIN WITH BOUND NORETHINDRONE | PROGESTERONE RECEPTOR; NUCLEAR RECEPTOR; STEROID RECEPTOR; NORETHINDRONE; BIRTH CONTROL, HORMONE/GROWTH FACTOR RECEPTIOR COMPLEX
1sr7:A (PRO686) to (TRP755) PROGESTERONE RECEPTOR HORMONE BINDING DOMAIN WITH BOUND MOMETASONE FUROATE | PROGESTERONE RECEPTOR, MOMETASONE, PROGESTERONE, NUCLEAR RECEPTOR, HORMONE RECEPTOR, TRANSCRIPTION
1swv:A (THR41) to (ILE97) CRYSTAL STRUCTURE OF THE D12A MUTANT OF PHOSPHONOACETALDEHYDE HYDROLASE COMPLEXED WITH MAGNESIUM | HAD ENZYME SUPERFAMILY, PHOSPHONOTASE, PHOSPHONOACETALDEHYDE, METAL BINDING, HYDROLASE
1sww:A (THR41) to (ILE97) CRYSTAL STRUCTURE OF THE PHOSPHONOACETALDEHYDE HYDROLASE D12A MUTANT COMPLEXED WITH MAGNESIUM AND SUBSTRATE PHOSPHONOACETALDEHYDE | PHOPSHONOACETALDEHYDE HYDROLASE, PHOSPHONATASE, HAD ENZYM SUPERFAMILY, METAL BINDING
3vhu:A (SER737) to (SER805) MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN WITH SPIRONOLACTONE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ACTIVATING MUTATION, HYPERTENSION, ANTAGONIST, SPIRONOLACTONE, TRANSCRIPTION-INHIBITOR COMPLEX
3vhv:A (SER737) to (SER805) MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN WITH NON-STEROIDAL ANTAGONIST | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ACTIVATING MUTATION, HYPERTENSION, NON-STEROIDAL ANTAGONIST, TRANSCRIPTION-INHIBITOR COMPLEX
2gkm:A (HIS22) to (THR127) CRYSTAL STRUCTURE OF MYCOBACTERIUM TUBERCULOSIS TRHBN TYRB10PHE MUTANT | TRUNCATED HEMOGLOBIN; MUTANT, OXYGEN STORAGE/TRANSPORT COMPLEX
4zn9:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH OXABICYCLIC HEPTENE SULFONATE (OBHS) | PROTEIN LIGAND COMPLEX, TRANSCRIPTION
4zns:B (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH A 3-FLUORO-SUBSTITUTED OBHS DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4znt:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH A 3-BROMO-SUBSTITUTED OBHS DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4znv:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH A 2-METHOXY-SUBSTITUTED OBHS DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
3vkg:A (PRO2876) to (PRO2939) X-RAY STRUCTURE OF AN MTBD TRUNCATION MUTANT OF DYNEIN MOTOR DOMAIN | AAA+ PROTEIN, MOLECULAR MOTOR, MICROTUBLES, MOTOR PROTEIN
1hds:B (GLY23) to (ALA134) MACROMOLECULAR STRUCTURE REFINEMENT BY RESTRAINED LEAST- SQUARES AND INTERACTIVE GRAPHICS AS APPLIED TO SICKLING DEER TYPE III HEMOGLOBIN | OXYGEN TRANSPORT
3vkh:A (PRO2876) to (PRO2939) X-RAY STRUCTURE OF A FUNCTIONAL FULL-LENGTH DYNEIN MOTOR DOMAIN | AAA+ PROTEIN, MOLECULAR MOTOR, MICROTUBLES, MOTOR PROTEIN
3vkh:B (PRO2876) to (HIS2937) X-RAY STRUCTURE OF A FUNCTIONAL FULL-LENGTH DYNEIN MOTOR DOMAIN | AAA+ PROTEIN, MOLECULAR MOTOR, MICROTUBLES, MOTOR PROTEIN
3vkh:B (ASP4300) to (LEU4363) X-RAY STRUCTURE OF A FUNCTIONAL FULL-LENGTH DYNEIN MOTOR DOMAIN | AAA+ PROTEIN, MOLECULAR MOTOR, MICROTUBLES, MOTOR PROTEIN
4ltw:A (LEU3) to (SER70) ANCESTRAL KETOSTEROID RECEPTOR-PROGESTERONE-MIFEPRISTONE COMPLEX | NUCLEAR RECEPTOR, STEROID RECEPTOR, HORMONE RECEPTOR
2hv6:A (GLU72) to (SER142) CRYSTAL STRUCTURE OF THE PHOSPHOTYROSYL PHOSPHATASE ACTIVATOR | PHOSPHOTYROSYL PHOSPHATASE ACTIVATOR, PHOSPHATASE, PP2A, PHOSPHATASE SPECIFICITY, UNKNOWN FUNCTION
2hv6:B (GLU75) to (SER142) CRYSTAL STRUCTURE OF THE PHOSPHOTYROSYL PHOSPHATASE ACTIVATOR | PHOSPHOTYROSYL PHOSPHATASE ACTIVATOR, PHOSPHATASE, PP2A, PHOSPHATASE SPECIFICITY, UNKNOWN FUNCTION
2hv7:A (GLU72) to (SER142) CRYSTAL STRUCTURE OF PHOSPHOTYROSYL PHOSPHATASE ACTIVATOR BOUND TO ATPGAMMAS | PHOSPHOTYROSYL PHOSPHATASE ACTIVATOR, PP2A, PHOSPHATASE, PHOSPHATASE SPECIFICITY, UNKNOWN FUNCTION
2hv7:D (GLU72) to (SER142) CRYSTAL STRUCTURE OF PHOSPHOTYROSYL PHOSPHATASE ACTIVATOR BOUND TO ATPGAMMAS | PHOSPHOTYROSYL PHOSPHATASE ACTIVATOR, PP2A, PHOSPHATASE, PHOSPHATASE SPECIFICITY, UNKNOWN FUNCTION
2hv7:F (GLU72) to (SER142) CRYSTAL STRUCTURE OF PHOSPHOTYROSYL PHOSPHATASE ACTIVATOR BOUND TO ATPGAMMAS | PHOSPHOTYROSYL PHOSPHATASE ACTIVATOR, PP2A, PHOSPHATASE, PHOSPHATASE SPECIFICITY, UNKNOWN FUNCTION
2i0j:C (THR311) to (ALA382) BENZOPYRANS ARE SELECTIVE ESTROGEN RECEPTOR BETA AGONISTS (SERBAS) WITH NOVEL ACTIVITY IN MODELS OF BENIGN PROSTATIC HYPERPLASIA | NUCLEAR RECEPTOR LIGAND BINDING DOMAIN, TRANSCRIPTION
2i15:B (SER251) to (PHE323) CRYSTAL STRUCTURE OF MPN423 FROM MYCOPLASMA PNEUMONIAE | STRUCTURAL GENOMICS, MPN423, HYPOTHETICAL PROTIEN, CRYSTAL STRUCTURE, ALL ALPHA STRUCTURE, PSI, PROTEIN STRUCTURE INITIATIVE, BERKELEY STRUCTURAL GENOMICS CENTER, BSGC, UNKNOWN FUNCTION
2i15:C (SER451) to (PHE523) CRYSTAL STRUCTURE OF MPN423 FROM MYCOPLASMA PNEUMONIAE | STRUCTURAL GENOMICS, MPN423, HYPOTHETICAL PROTIEN, CRYSTAL STRUCTURE, ALL ALPHA STRUCTURE, PSI, PROTEIN STRUCTURE INITIATIVE, BERKELEY STRUCTURAL GENOMICS CENTER, BSGC, UNKNOWN FUNCTION
2i2x:A (LYS350) to (GLY410) CRYSTAL STRUCTURE OF METHANOL:COBALAMIN METHYLTRANSFERASE COMPLEX MTABC FROM METHANOSARCINA BARKERI | TIM BARREL AND HELIX BUNDLE (MTAB); ROSSMAN FOLD AND HELIX BUNDLE (MTAC), TRANSFERASE
2i2x:G (LYS350) to (ALA409) CRYSTAL STRUCTURE OF METHANOL:COBALAMIN METHYLTRANSFERASE COMPLEX MTABC FROM METHANOSARCINA BARKERI | TIM BARREL AND HELIX BUNDLE (MTAB); ROSSMAN FOLD AND HELIX BUNDLE (MTAC), TRANSFERASE
2i2x:I (LYS350) to (GLY410) CRYSTAL STRUCTURE OF METHANOL:COBALAMIN METHYLTRANSFERASE COMPLEX MTABC FROM METHANOSARCINA BARKERI | TIM BARREL AND HELIX BUNDLE (MTAB); ROSSMAN FOLD AND HELIX BUNDLE (MTAC), TRANSFERASE
2i2x:K (LYS350) to (ALA409) CRYSTAL STRUCTURE OF METHANOL:COBALAMIN METHYLTRANSFERASE COMPLEX MTABC FROM METHANOSARCINA BARKERI | TIM BARREL AND HELIX BUNDLE (MTAB); ROSSMAN FOLD AND HELIX BUNDLE (MTAC), TRANSFERASE
2i2x:M (LYS350) to (GLY410) CRYSTAL STRUCTURE OF METHANOL:COBALAMIN METHYLTRANSFERASE COMPLEX MTABC FROM METHANOSARCINA BARKERI | TIM BARREL AND HELIX BUNDLE (MTAB); ROSSMAN FOLD AND HELIX BUNDLE (MTAC), TRANSFERASE
2i2x:O (LYS350) to (ALA409) CRYSTAL STRUCTURE OF METHANOL:COBALAMIN METHYLTRANSFERASE COMPLEX MTABC FROM METHANOSARCINA BARKERI | TIM BARREL AND HELIX BUNDLE (MTAB); ROSSMAN FOLD AND HELIX BUNDLE (MTAC), TRANSFERASE
2i3o:B (GLN185) to (TYR231) CRYSTAL STRUCTURE OF GAMMA-GLUTAMYL TRANSFERASE RELATED PROTEIN FROM THERMOPLASMA ACIDOPHILUM | CRYSTAL STRUCTURE, GAMMA-GLUTAMYL TRANSFERASE RELATED PROTEIN, THERMOPLASMA ACIDOPHILUM, 6324D, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
2i3o:D (GLN185) to (TYR231) CRYSTAL STRUCTURE OF GAMMA-GLUTAMYL TRANSFERASE RELATED PROTEIN FROM THERMOPLASMA ACIDOPHILUM | CRYSTAL STRUCTURE, GAMMA-GLUTAMYL TRANSFERASE RELATED PROTEIN, THERMOPLASMA ACIDOPHILUM, 6324D, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
3j04:F (GLN7) to (GLY52) EM STRUCTURE OF THE HEAVY MEROMYOSIN SUBFRAGMENT OF CHICK SMOOTH MUSCLE MYOSIN WITH REGULATORY LIGHT CHAIN IN PHOSPHORYLATED STATE | PHOSPHORYLATION, 2D CRYSTALLINE ARRAYS, MYOSIN REGULATION, MYOSIN LIGHT CHAINS, STRUCTURAL PROTEIN
1ijx:F (GLU41) to (LEU107) CRYSTAL STRUCTURE OF THE CYSTEINE-RICH DOMAIN OF SECRETED FRIZZLED- RELATED PROTEIN 3 (SFRP-3;FZB) | WNT RECEPTOR, FRIZZLED PROTEIN STRUCTURE, CYSTEINE-RICH, SIGNALING PROTEIN
5a9j:A (ALA804) to (GLN888) CRYSTAL STRUCTURE OF THE HELICASE DOMAIN OF HUMAN DNA POLYMERASE THETA, APO-FORM | HYDROLASE, POLYMERASE, HELICASE, POLQ, DNA REPAIR
5a9j:B (ALA804) to (GLU893) CRYSTAL STRUCTURE OF THE HELICASE DOMAIN OF HUMAN DNA POLYMERASE THETA, APO-FORM | HYDROLASE, POLYMERASE, HELICASE, POLQ, DNA REPAIR
5a9j:D (ALA804) to (GLU893) CRYSTAL STRUCTURE OF THE HELICASE DOMAIN OF HUMAN DNA POLYMERASE THETA, APO-FORM | HYDROLASE, POLYMERASE, HELICASE, POLQ, DNA REPAIR
4m6w:A (SER1983) to (ILE2026) CRYSTAL STRUCTURE OF THE C-TERMINAL SEGMENT OF FANCM IN COMPLEX WITH FAAP24 | FANCM, FAAP24, XPF/MUS81, FANCONI ANEMIA, DNA REPAIR, DNA BINDING PROTEIN
3wdd:A (THR81) to (GLU147) MUTANT N-TERMINAL DOMAIN OF MYCOBACTERIUM TUBERCULOSIS CLPC1, F2Y, BOUND TO CYCLOMARIN A | CHAPERONE, CHAPERONE-ANTIMICROBIAL PROTEIN COMPLEX
4mes:B (SER77) to (LYS172) CRYSTAL STRUCTURE OF THIT COMPLEXED WITH LMG116 | S-COMPONENT, ECF TRANSPORTER, ABC TRANSPORTER, THIAMINE BINDING PROTEIN
3wfg:A (SER737) to (SER805) MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN WITH COMPUOND 2E | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, TRANSCRIPTION, HYPERTENSION, NON-STEROIDAL ANTAGONIST, ACTIVATING MUTATION, TRANSCRIPTION- INHIBITOR COMPLEX
5aga:A (ALA804) to (ASP890) CRYSTAL STRUCTURE OF THE HELICASE DOMAIN OF HUMAN DNA POLYMERASE THETA IN COMPLEX WITH AMPPNP | TRANSFERASE, POLQ, DNA REPAIR
4mg5:B (THR311) to (ALA382) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH CHLORDECONE | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mg6:A (THR311) to (SER395) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BENZYLBUTYLPHTALATE | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mg6:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BENZYLBUTYLPHTALATE | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mg7:A (THR311) to (SER395) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH FERUTININE | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mg8:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH ALPHA-ZEARALANOL | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mg9:A (THR311) to (SER395) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BUTYLPARABEN | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mg9:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BUTYLPARABEN | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mgb:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH TCBPA | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mgb:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH TCBPA | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
2iof:A (THR41) to (ILE97) CRYSTAL STRUCTURE OF PHOSPHONOACETALDEHYDE HYDROLASE WITH SODIUM BOROHYDRIDE-REDUCED SUBSTRATE INTERMEDIATE | PHOSPHONOACETALDEHYDE HYDROLASE, HALOACID DEHALOGENASE SUPERFAMILY
2iof:K (THR41) to (ILE97) CRYSTAL STRUCTURE OF PHOSPHONOACETALDEHYDE HYDROLASE WITH SODIUM BOROHYDRIDE-REDUCED SUBSTRATE INTERMEDIATE | PHOSPHONOACETALDEHYDE HYDROLASE, HALOACID DEHALOGENASE SUPERFAMILY
4mgc:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BENZOPHENONE-2 | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mgc:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH BENZOPHENONE-2 | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mgd:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH HPTE | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
4mgd:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH HPTE | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
2iok:A (THR311) to (ALA382) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH COMPOUND 1D | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ER-ALPHA, ANTAGONIST
4mhw:A (SER77) to (LYS172) CRYSTAL STRUCTURE OF THIT WITH SMALL MOLECULE BAT-25 | S-COMPONENT, ECF TRANSPORTER, ABC TRANSPORTER, SUBSTRATE BINDING DOMAIN FOR THIAMIN, TRANSPORT PROTEIN, THIAMINE BINDING PROTEIN
1vjb:A (LYS236) to (ALA304) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAIN OF THE ESTROGEN-RELATED RECEPTOR GAMMA IN COMPLEX WITH 4- HYDROXYTAMOXIFEN | LIGAND-BINDING DOMAIN, ANTAGONIST COMPLEX, TRANSCRIPTION
4muu:B (SER87) to (LYS182) STRUCTURE OF THIT WITH PYRITHIAMINE BOUND | S-COMPONENT, ECF TRANSPORTER, ABC TRANSPORTER, THIAMINE BINDING PROTEIN
2xok:A (ALA414) to (SER476) REFINED STRUCTURE OF YEAST F1C10 ATPASE COMPLEX TO 3 A RESOLUTION | HYDROLASE, ATP-BINDING, F(O), F(1), ATP SYNTHASE, MITOCHONDRIA, INNER MEMBRANE, TRANSMEMBRANE
4n4d:A (SER77) to (LYS172) STRUCTURE OF THIT WITH AV-38 BOUND | S-COMPONENT, ECF TRANSPORTER, ABC TRANSPORTER, TRANSPORT PROTEIN, THIAMINE BINDING PROTEIN-INHIBITOR COMPLEX
2kob:A (SER63) to (THR119) SOLUTION NMR STRUCTURE OF CLOLEP_01837 (FRAGMENT 61-160) FROM CLOSTRIDIUM LEPTUM. NORTHEAST STRUCTURAL GENOMICS CONSORTIUM TARGET QLR8A | ALPHA BETA, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, NESG, UNKNOWN FUNCTION
2l95:A (ASP7) to (ARG72) SOLUTION STRUCTURE OF CYTOTOXIC T-LYMPHOCYTE ANTIGENT-2(CTLA PROTEIN), CRAMMER AT PH 6.0 | CRAMMER, CYSTEINE PROTEINASE INHIBITOR, INTRINSIC DISORDER P CTLA-2- LIKE PROTEIN, HYDROLASE
3zqt:A (PRO671) to (TYR739) TARGETING THE BINDING FUNCTION 3 SITE OF THE ANDROGEN RECEPTOR THROUGH IN SILICO MOLECULAR MODELING | TRANSCRIPTION, SMALL MOLECULE INHIBITOR
2yat:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF ESTRADIOL DERIVED METAL CHELATE AND ESTROGEN RECEPTOR-LIGAND BINDING DOMAIN COMPLEX | TRANSCRIPTION
4noo:C (LEU949) to (GLY1011) MOLECULAR MECHANISM FOR SELF-PROTECTION AGAINST TYPE VI SECRETION SYSTEM IN VIBRIO CHOLERAE | SELF-PROTECTION, CHITOSANASE-FOLD, THREE-HELICAL BUNDLE, GLYCOSIDE HYDROLASE EFFECTOR, IMMUNITY PROTEIN, IMMUNE SYSTEM
2m9n:A (SER158) to (VAL198) SOLUTION STRUCTURE OF (HHH)2 DOMAIN OF HUMAN FAAP24 | FANCONI ANEMIA, FAAP24, (HHH)2 DOMAIN, DNA BINDING PROTEIN
2yg9:A (PRO61) to (GLY108) STRUCTURE OF AN UNUSUAL 3-METHYLADENINE DNA GLYCOSYLASE II ( ALKA) FROM DEINOCOCCUS RADIODURANS | HYDROLASE, DNA REPAIR
2yg9:B (ASP60) to (GLY108) STRUCTURE OF AN UNUSUAL 3-METHYLADENINE DNA GLYCOSYLASE II ( ALKA) FROM DEINOCOCCUS RADIODURANS | HYDROLASE, DNA REPAIR
4ny3:B (GLU72) to (SER142) HUMAN PTPA IN COMPLEX WITH PEPTIDE | PTPA, PPP2R4, REGULATORY SUBUNIT B' (PR 53), HYDROLASE ACTIVATOR, PROTEIN PHOSPHATASE 2A (PP2A)
1l2i:B (THR311) to (TRP383) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH (R,R)-5,11-CIS-DIETHYL-5,6,11,12- TETRAHYDROCHRYSENE-2,8-DIOL AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ESTROGEN, AGONIST, COACTIVATOR, TRANSCRIPTION RECEPTOR/COACTIVATOR COMPLEX
5ccm:A (HIS83) to (SER182) CRYSTAL STRUCTURE OF SMYD3 WITH SAM AND EPZ030456 | PROTEIN-INHIBITOR COMPLEX, METHYLTRANSFERASE, EPIGENETICS, DRUG DISCOVERY, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4o6f:A (TRP83) to (GLY183) STRUCTURAL BASIS OF ESTROGEN RECEPTOR ALPHA METHYLATION MEDIATED BY HISTONE METHYLTRANSFERASE SMYD2 | HISTONE METHYLTRANSFERASE, SMYD2, ESTROGEN RECEPTOR ER ALPHA, METHYLATION, ESTROGEN SIGNALING, TRANSFERASE
4a2j:A (PRO686) to (TYR753) PR X-RAY STRUCTURES IN AGONIST CONFORMATIONS REVEAL TWO DIFFERENT MECHANISMS FOR PARTIAL AGONISM IN 11BETA- SUBSTITUTED STEROIDS | TRANSCRIPTION, PARTIAL AGONIST
4a2j:B (PRO686) to (SER754) PR X-RAY STRUCTURES IN AGONIST CONFORMATIONS REVEAL TWO DIFFERENT MECHANISMS FOR PARTIAL AGONISM IN 11BETA- SUBSTITUTED STEROIDS | TRANSCRIPTION, PARTIAL AGONIST
4oar:A (PRO686) to (SER754) PROGESTERONE RECEPTOR WITH BOUND ULIPRISTAL ACETATE AND A PEPTIDE FROM THE CO-REPRESSOR SMRT | PROGESTERONE RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, WOMEN HEALTH, CONTRACEPTION, TRANSCRIPTION- PEPTIDE COMPLEX
3k23:B (THR531) to (SER599) GLUCOCORTICOID RECEPTOR WITH BOUND D-PROLINAMIDE 11 | GLUCOCORTICOID RECEPTOR, STEROID HORMONE RECEPTOR, NUCLEAR RECEPTOR, GR, GLUCOCORTICOIDS, ALPHA HELICAL SANDWICH, META-CHANNEL, ALTERNATIVE INITIATION, CHROMATIN REGULATOR, DISEASE MUTATION, DNA- BINDING, METAL-BINDING, NUCLEUS, PSEUDOHERMAPHRODITISM, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC- FINGER, ACTIVATOR
4oed:A (PHE673) to (SER740) CRYSTAL STRUCTURE OF AR-LBD BOUND WITH CO-REGULATOR PEPTIDE | ALPHA-HELIX, HORMONE/GROWTH FACTOR RECEPTOR, PHOSPHORYLATION, HORMONE RECEPTOR-PEPTIDE COMPLEX
4ogh:A (PRO671) to (TRP741) CRYSTAL STRUCTURE OF T877A-AR-LBD | ALPHA HELIX, SIGNAL TRANSDUCTION, CO-REGULATOR, PHOSPHORYLATION, HORMONE RECEPTOR
4oha:A (ILE672) to (TRP741) CRYSTAL STRUCTURE OF T877A-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE | ALPHA-HELIX, HORMONE/GROWTH FACTOR RECEPTOR, PHOSPHORYLATION, HORMONE RECEPTOR-PEPTIDE COMPLEX, SIGNAL TRANSDUCTION
2z46:F (ASN34) to (GLN111) CRYSTAL STRUCTURE OF NATIVE-ORF134 | CHAPERONE, HELIX BUNDLE
2z4j:A (PRO671) to (TYR739) CRYSTAL STRUCTURE OF AR LBD WITH SHP PEPTIDE NR BOX 2 | ANDROGEN RECEPTOR, LIGAND BINDING DOMAIN, SHP, CO-REPRESSOR, TRANSCRIPTION
2o3e:A (ASP467) to (ARG544) CRYSTAL STRUCTURE OF ENGINEERED NEUROLYSIN WITH THIMET OLIGOPEPTIDASE SPECIFICITY FOR NEUROTENSIN CLEAVAGE SITE. | THERMOLYSIN-LIKE DOMAIN, SUBSTRATE-BINDING CHANNEL, HYDROLASE
4oiu:A (PHE673) to (SER740) CRYSTAL STRUCTURE OF T877A-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE | ALPHA-HELIX, HORMONE/GROWTH FACTOR RECEPTOR, PHOSPHORYLATION, HORMONE RECEPTOR-PEPTIDE COMPLEX, SIGNAL TRANSDUCTION
4ojb:A (PRO671) to (LEU741) CRYSTAL STRUCTURE OF W741L-AR-LBD | ALPHA-HELIX, HORMONE/GROWTH FACTOR RECEPTOR, PHOSPHORYLATION, SIGNAL TRANSDUCTION, HORMONE RECEPTOR
4okb:A (PRO671) to (LEU741) CRYSTAL STRUCTURE OF W741L-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE | ALPHA-HELIX, HORMONE/GROWTH FACTOR RECEPTOR, PHOSPHORYLATION, HORMONE RECEPTOR-PEPTIDE COMPLEX, SIGNAL TRANSDUCTION
1xnn:A (ILE672) to (SER740) CRYSTAL STRUCTURE OF THE RAT ANDROGEN RECEPTOR LIGAND BINDING DOMAIN T877A MUTANT COMPLEX WITH (3A-ALPHA-,4- ALPHA 7-ALPHA-,7A-ALPHA-)-3A,4,7,7A-TETRAHYDRO-2-(4-NITRO- 1-NAPHTHALENYL)-4,7-ETHANO-1H-ISOINDOLE-1,3(2H)-DIONE. | ANDROGEN RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, LIGAND-BINDING DOMAIN, HORMONE/GROWTH FACTOR COMPLEX
4okw:A (ILE672) to (LEU741) CRYSTAL STRUCTURE OF W741L-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE | ALPHA-HELIX, HORMONE/GROWTH FACTOR RECEPTOR, PHOSPHORYLATION, HORMONE RECEPTOR-PEPTIDE COMPLEX, SIGNAL TRANSDUCTION
4okx:A (ILE672) to (LEU741) CRYSTAL STRUCTURE OF W741L-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE | ALPHA-HELIX, HORMONE/GROWTH FACTOR RECEPTOR, PHOSPHORYLATION, HORMONE RECEPTOR-PEPTIDE COMPLEX, SIGNAL TRANSDUCTION
4olm:A (PRO671) to (LEU741) CRYSTAL STRUCTURE OF W741L-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE | ALPHA-HELIX, HORMONE/GROWTH FACTOR RECEPTOR, PHOSPHORYLATION, HORMONE RECEPTOR-PEPTIDE COMPLEX
1xpc:A (THR311) to (ALA382) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH COMPOUND 19 | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ER-ALPHA, ANTAGONIST, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
3kba:A (PRO686) to (TRP755) PROGESTERONE RECEPTOR BOUND TO SULFONAMIDE PYRROLIDINE PARTIAL AGONIST | NUCLEAR RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION
3kba:B (PRO686) to (SER754) PROGESTERONE RECEPTOR BOUND TO SULFONAMIDE PYRROLIDINE PARTIAL AGONIST | NUCLEAR RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION
1xq3:A (ILE672) to (TRP741) CRYSTAL STRUCTURE OF THE HUMAN ANDROGEN RECEPTOR LIGAND BINDING DOMAIN BOUND WITH R1881 | CRYSTAL STRUCTURE; HUMAN ANDROGEN RECEPTOR LIGAND BINDING DOMAIN; R1881, TRANSCRIPTION
1xqc:A (THR311) to (ALA382) X-RAY STRUCTURE OF ERALPHA LBD BOUND TO A TETRAHYDROISOQUINOLINE SERM LIGAND AT 2.05A RESOLUTION | ALPHA-HELICAL SANDWICH, NUCLEAR HORMONE RECEPTOR, LIGAND BINDING DOMAIN
1xqc:B (THR311) to (ALA382) X-RAY STRUCTURE OF ERALPHA LBD BOUND TO A TETRAHYDROISOQUINOLINE SERM LIGAND AT 2.05A RESOLUTION | ALPHA-HELICAL SANDWICH, NUCLEAR HORMONE RECEPTOR, LIGAND BINDING DOMAIN
1m7w:A (SER142) to (ALA213) HNF4A LIGAND BINDING DOMAIN WITH BOUND FATTY ACID | TRANSCRIPTION FACTOR
1m7w:B (ILE143) to (HIS214) HNF4A LIGAND BINDING DOMAIN WITH BOUND FATTY ACID | TRANSCRIPTION FACTOR
1m7w:D (SER142) to (HIS214) HNF4A LIGAND BINDING DOMAIN WITH BOUND FATTY ACID | TRANSCRIPTION FACTOR
1mbu:B (GLN4) to (THR65) CRYSTAL STRUCTURE ANALYSIS OF CLPSN HETERODIMER | PROTEIN BINDING
4p19:C (ALA265) to (GLY330) CLOSED, APO INWARD-FACING STATE OF THE GLUTAMATE TRANSPORTER HOMOLOGUE GLTPH | MEMBRANE PROTEIN, SODIUM-COUPLED ASPARTATE TRANSPORTER, INWARD-FACING STATE, APO FORM, TRANSPORT PROTEIN
1y8b:A (THR652) to (HIS723) SOLUTION NMR-DERIVED GLOBAL FOLD OF MALATE SYNTHASE G FROM E.COLI | NMR GLOBAL FOLD, APO-MALATE SYNTHASE G, 82 KDA ENZYME, TRANSFERASE
4p6x:A (THR531) to (SER599) CRYSTAL STRUCTURE OF CORTISOL-BOUND GLUCOCORTICOID RECEPTOR LIGAND BINDING DOMAIN | CORTISOL, GLUCOCORTICOID RECEPTOR, POTENCY, HORMONE-HORMONE RECEPTOR COMPLEX
4p6x:E (VAL533) to (SER599) CRYSTAL STRUCTURE OF CORTISOL-BOUND GLUCOCORTICOID RECEPTOR LIGAND BINDING DOMAIN | CORTISOL, GLUCOCORTICOID RECEPTOR, POTENCY, HORMONE-HORMONE RECEPTOR COMPLEX
4p6x:K (LEU532) to (SER599) CRYSTAL STRUCTURE OF CORTISOL-BOUND GLUCOCORTICOID RECEPTOR LIGAND BINDING DOMAIN | CORTISOL, GLUCOCORTICOID RECEPTOR, POTENCY, HORMONE-HORMONE RECEPTOR COMPLEX
1y9r:A (PRO738) to (SER805) CRYSTAL STRUCTURE OF THE HUMAN MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN BOUND TO DEOXYCORTICOSTERONE AND HARBORING THE S810L MUTATION RESPONSIBLE FOR A SEVERE FORM OF HYPERTENSION | MINERALOCORTICOID RECEPTOR; STEROID RECEPTOR; NUCLEAR RECEPT; TRANSCRIPTION REGULATION; ACTIVATING MUTATION; HYPERTENSION, TRANSCRIPTION, LIGAND BINDING PROTEIN
1y9r:B (VAL739) to (SER805) CRYSTAL STRUCTURE OF THE HUMAN MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN BOUND TO DEOXYCORTICOSTERONE AND HARBORING THE S810L MUTATION RESPONSIBLE FOR A SEVERE FORM OF HYPERTENSION | MINERALOCORTICOID RECEPTOR; STEROID RECEPTOR; NUCLEAR RECEPT; TRANSCRIPTION REGULATION; ACTIVATING MUTATION; HYPERTENSION, TRANSCRIPTION, LIGAND BINDING PROTEIN
1ya3:B (VAL739) to (SER805) CRYSTAL STRUCTURE OF THE HUMAN MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN BOUND TO PROGESTERONE AND HARBORING THE S810L MUTATION RESPONSIBLE FOR A SEVERE FORM OF HYPERTENSION | MINERALOCORTICOID RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR TRANSCRIPTION REGULATION, ACTIVATING MUTATION, HYPERTENSION
1ya3:C (SER737) to (SER805) CRYSTAL STRUCTURE OF THE HUMAN MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN BOUND TO PROGESTERONE AND HARBORING THE S810L MUTATION RESPONSIBLE FOR A SEVERE FORM OF HYPERTENSION | MINERALOCORTICOID RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR TRANSCRIPTION REGULATION, ACTIVATING MUTATION, HYPERTENSION
1yim:A (THR311) to (ALA382) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH COMPOUND 4 | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ER-ALPHA, ANTAGONIST, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
4pf3:A (SER737) to (SER805) MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN WITH COMPUOND 37A | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, HYPERTENSION, NON-STEROIDAL ANTAGONIST, ACTIVATING MUTATION
4akg:B (ARG2620) to (TYR2680) DYNEIN MOTOR DOMAIN - ATP COMPLEX | MOTOR PROTEIN, AAA+ PROTEIN, ASCE PROTEIN, P-LOOP NTPASE, CYTOSKELETAL MOTOR, ATPASE
3l03:B (THR311) to (SER395) CRYSTAL STRUCTURE OF HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE AND ESTETROL (ESTRA-1,3,5(10)-TRIENE-3,15 ALPHA, 16ALPHA,17BETA-TETROL) | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, ESTETROL, DNA-BINDING, GLYCOPROTEIN, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER, ACTIVATOR
3l3z:A (ILE672) to (TYR739) CRYSTAL STRUCTURE OF DHT-BOUND ANDROGEN RECEPTOR IN COMPLEX WITH THE THIRD MOTIF OF STEROID RECEPTOR COACTIVATOR 3 | ANDROGEN RECEPTOR, LIGAND BINDING DOMAIN, STEROID RECEPTOR COACTIVATOR 3, 5-ALPHA-DIHYDROTESTOSTERONE (DHT), PROSTATE CANCER, PROTEIN BINDING
5did:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DIFLUORO-SUBSTITUTED A-CD RING ESTROGEN DERIVATIVE (1S,3AR,5S, 7AS)-5-(2,3-DIFLUORO-4-HYDROXYPHENYL)-7A-METHYLOCTAHYDRO-1H-INDEN-1- OL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5die:B (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A TRIFLUORO-SUBSTITUTED A-CD RING ESTROGEN DERIVATIVE (1S,3AR, 5S,7AS)-7A-METHYL-5-(2,3,5-TRIFLUORO-4-HYDROXYPHENYL)OCTAHYDRO-1H- INDEN-1-OL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dig:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A TRIFLUOROMETHYL-SUBSTITUTED A-CD RING ESTROGEN DERIVATIVE (1S, 3AR,5S,7AS)-5-[4-HYDROXY-2-(TRIFLUOROMETHYL)PHENYL]-7A- METHYLOCTAHYDRO-1H-INDEN-1-OL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4akh:A (PRO2619) to (LYS2679) DYNEIN MOTOR DOMAIN - AMPPNP COMPLEX | MOTOR PROTEIN, MOTOR PROTEIN-TRANSFERASE COMPLEX, AAA+ PROTEIN, ASCE PROTEIN, MOTOR PROTEIN P-LOOP NTPASE, CYTOSKELETAL MOTOR
4akh:B (PRO2619) to (TYR2680) DYNEIN MOTOR DOMAIN - AMPPNP COMPLEX | MOTOR PROTEIN, MOTOR PROTEIN-TRANSFERASE COMPLEX, AAA+ PROTEIN, ASCE PROTEIN, MOTOR PROTEIN P-LOOP NTPASE, CYTOSKELETAL MOTOR
5dke:B (ALA312) to (ALA382) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 3-NAPHTHYL-SUBSTITUTED, METHYL, CIS-DIARYL-ETHYLENE COMPOUND 4,4'-[2-(NAPHTHALEN-2-YL)PROP-1-ENE-1,1-DIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dl4:A (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A PHENYLAMINO-SUBSTITUTED, METHYL, TRIARYL-ETHYLENE DERIVATIVE 4,4'-{2-[3-(PHENYLAMINO)PHENYL]PROP-1-ENE-1,1-DIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dlr:B (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A TRIARYL-ETHYLENE COMPOUND 4,4'-(2-PHENYLETHENE-1,1-DIYL) DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4aki:B (PRO2619) to (LYS2679) DYNEIN MOTOR DOMAIN - LUAC DERIVATIVE | MOTOR PROTEIN, DYNEIN, DYNEIN HEAVY CHAIN, DYNEIN MOTOR DOMAIN, MOTOR PROTEIN AAA+ PROTEIN, ASCE PROTEIN, P-LOOP NTPASE, CYTOSKELETAL MOTOR
4pop:A (SER77) to (LYS172) THIT WITH LMG139 BOUND | S-COMPONENT, THIAMINE-BINDING PROTEIN, ECF MODULE, MEMBRANE, PROTEIN BINDING
4pov:B (SER77) to (LYS172) THIT WITH LMG135 BOUND | S-COMPONENT, THIAMINE-BINDING PROTEIN, ECF MODULE, MEMBRANE, PROTEIN BINDING
4pp6:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH RESVERATROL | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, NUCLEUS, PROTEIN BINDING
5dp0:A (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 4-FLUOROPHENYLAMINO-SUBSTITUTED TRIARYL-ETHYLENE DERIVATIVE 4, 4'-(2-{3-[(4-FLUOROPHENYL)AMINO]PHENYL}ETHENE-1,1-DIYL)DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5drm:A (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DICHLORO-SUBSTITUTED, 2,5-DIARYLTHIOPHENE-CORE LIGAND 4,4'- THIENE-2,5-DIYLBIS(3-CHLOROPHENOL) | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5drm:B (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DICHLORO-SUBSTITUTED, 2,5-DIARYLTHIOPHENE-CORE LIGAND 4,4'- THIENE-2,5-DIYLBIS(3-CHLOROPHENOL) | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4apu:B (PRO686) to (TRP755) PR X-RAY STRUCTURES IN AGONIST CONFORMATIONS REVEAL TWO DIFFERENT MECHANISMS FOR PARTIAL AGONISM IN 11BETA-SUBSTITUTED STEROID | TRANSCRIPTION, ASOPRISNIL, PARTIAL AGONIST
5dtv:B (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DIMETHYL-SUBSTITUTED, 3,4-DIARYLTHIOPHENE DIOXIDE CORE LIGAND | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5due:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A PARA-HYDROXYL-SUBSTITUTED, SULFOXIDE-BRIDGED OXABICYCLIC HEPTENE SULFONATE (SOBHS)-2 ANALOG 4-HYDROXYPHENYL (1S,2S,4S,5S,6R, 7S)-5,6-BIS(4-HYDROXY-2-METHYLPHENYL)-7-THIABICYCLO[2.2.1]HEPTANE-2- SULFONATE 7-OXIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5due:B (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A PARA-HYDROXYL-SUBSTITUTED, SULFOXIDE-BRIDGED OXABICYCLIC HEPTENE SULFONATE (SOBHS)-2 ANALOG 4-HYDROXYPHENYL (1S,2S,4S,5S,6R, 7S)-5,6-BIS(4-HYDROXY-2-METHYLPHENYL)-7-THIABICYCLO[2.2.1]HEPTANE-2- SULFONATE 7-OXIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5duh:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A SULFOXIDE-BRIDGED OXABICYCLIC HEPTENE SULFONATE (SOBHS)-3 ANALOG PHENYL (1S,2S,4S,7S)-5,6-BIS(4-HYDROXY-3-METHYLPHENYL)-7- THIABICYCLO[2.2.1]HEPT-5-ENE-2-SULFONATE 7-OXIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dwe:A (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 2-CHLORO-SUBSTITUTED TRIARYL-IMINE ANALOG 4,4'-[(2- CHLOROPHENYL)CARBONIMIDOYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dxg:B (THR311) to (GLU380) ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN Y537S MUTANT IN COMPLEX WITH STAPLED PEPTIDE SRC2-P5 | ESTROGEN RECEPTOR, HORMONE, STAPLED PEPTIDE, PEPTIDE MIMETIC, BREAST CANCER, HORMONE RECEPTOR-PEPTIDE COMPLEX
1zky:A (THR311) to (LEU379) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH OBCP-3M AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
5dxk:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(9S)-BICYCLO[3.3.1]NON-9- YLMETHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dxp:A (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4-[(E)-(1S,5S)-BICYCLO[3.3.1]NON-9- YLIDENE(PHENYL)METHYL]PHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dxp:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4-[(E)-(1S,5S)-BICYCLO[3.3.1]NON-9- YLIDENE(PHENYL)METHYL]PHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dz0:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(4-METHYLCYCLOHEXYLIDENE) METHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dz1:A (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(4-ETHYLCYCLOHEXYLIDENE) METHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5dzi:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-{[(3S)-3-(2-HYDROXYETHYL) CYCLOHEXYLIDENE]METHANEDIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4q50:A (THR311) to (ALA382) THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN D538G MUTANT IN COMPLEX WITH 4-HYDROXYTAMOXIFEN | ACQUIRED SERM-RESISTANCE, BREAST CANCER, ACTIVATING MUTATION, SERM-ER STRUCTURE, ALPHA HELIX, NUCLEAR HORMONE RECEPTOR, HORMONE BINDING PROTEIN
4q50:B (THR311) to (ALA382) THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN D538G MUTANT IN COMPLEX WITH 4-HYDROXYTAMOXIFEN | ACQUIRED SERM-RESISTANCE, BREAST CANCER, ACTIVATING MUTATION, SERM-ER STRUCTURE, ALPHA HELIX, NUCLEAR HORMONE RECEPTOR, HORMONE BINDING PROTEIN
4q50:D (THR311) to (ALA382) THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN D538G MUTANT IN COMPLEX WITH 4-HYDROXYTAMOXIFEN | ACQUIRED SERM-RESISTANCE, BREAST CANCER, ACTIVATING MUTATION, SERM-ER STRUCTURE, ALPHA HELIX, NUCLEAR HORMONE RECEPTOR, HORMONE BINDING PROTEIN
4q50:E (THR311) to (ALA382) THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN D538G MUTANT IN COMPLEX WITH 4-HYDROXYTAMOXIFEN | ACQUIRED SERM-RESISTANCE, BREAST CANCER, ACTIVATING MUTATION, SERM-ER STRUCTURE, ALPHA HELIX, NUCLEAR HORMONE RECEPTOR, HORMONE BINDING PROTEIN
4q50:F (THR311) to (ALA382) THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN D538G MUTANT IN COMPLEX WITH 4-HYDROXYTAMOXIFEN | ACQUIRED SERM-RESISTANCE, BREAST CANCER, ACTIVATING MUTATION, SERM-ER STRUCTURE, ALPHA HELIX, NUCLEAR HORMONE RECEPTOR, HORMONE BINDING PROTEIN
1zuc:B (PRO686) to (TRP755) PROGESTERONE RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH THE NONSTEROIDAL AGONIST TANAPROGET | PROGESTERONE RECEPTOR, NONSTEROIDAL AGONIST, TANAPROGET, PROGESTERONE, HORMONE, HORMONE/GROWTH FACTOR COMPLEX
1zuc:A (PRO686) to (SER754) PROGESTERONE RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH THE NONSTEROIDAL AGONIST TANAPROGET | PROGESTERONE RECEPTOR, NONSTEROIDAL AGONIST, TANAPROGET, PROGESTERONE, HORMONE, HORMONE/GROWTH FACTOR COMPLEX
2a3i:A (PRO738) to (SER805) STRUCTURAL AND BIOCHEMICAL MECHANISMS FOR THE SPECIFICITY OF HORMONE BINDING AND COACTIVATOR ASSEMBLY BY MINERALOCORTICOID RECEPTOR | TRANSCRIPTION FACTOR, TRANSFERASE
2aa2:A (SER737) to (SER805) MINERALOCORTICOID RECEPTOR WITH BOUND ALDOSTERONE | MINERALOCORTICOID, MR, NUCLEAR RECEPTOR, STEROID RECEPTOR, ALDOSTERONE, TRANSCRIPTION
5ehj:A (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(4AR,8AR)-OCTAHYDRONAPHTHALEN- 2(1H)-YLIDENEMETHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5ehj:B (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-[(4AR,8AR)-OCTAHYDRONAPHTHALEN- 2(1H)-YLIDENEMETHANEDIYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
2aa5:A (SER737) to (SER805) MINERALOCORTICOID RECEPTOR WITH BOUND PROGESTERONE | MINERALOCORTICOID RECEPTOR, MR, NUCLEAR RECEPTOR, STEROID RECEPTOR, PROGESTERONE, TRANSCRIPTION
2aa5:B (SER737) to (SER805) MINERALOCORTICOID RECEPTOR WITH BOUND PROGESTERONE | MINERALOCORTICOID RECEPTOR, MR, NUCLEAR RECEPTOR, STEROID RECEPTOR, PROGESTERONE, TRANSCRIPTION
2aa6:A (SER737) to (SER805) MINERALOCORTICOID RECEPTOR S810L MUTANT WITH BOUND PROGESTERONE | MINERALOCORTICOID RECEPTOR, MR, NUCLEAR RECEPTOR, STEROID RECEPTOR, PROGESTERONE, HYPERTENSION, TRANSCRIPTION
2aa7:A (SER737) to (SER805) MINERALOCORTICOID RECEPTOR WITH BOUND DEOXYCORTICOSTERONE | MINERALOCORTICOID RECEPTOR, MR, NUCLEAR RECEPTOR, STEROID RECEPTOR, DEOXYCORTICOSTERONE, HYPERTENSION, TRANSCRIPTION
2aax:A (SER737) to (GLN803) MINERALOCORTICOID RECEPTOR DOUBLE MUTANT WITH BOUND CORTISONE | MINERALOCORTICOID RECEPTOR, MR, NUCLEAR RECEPTOR, STEROID RECEPTOR, CORTISONE, HYPERTENSION, TRANSCRIPTION
2aax:B (SER737) to (GLN803) MINERALOCORTICOID RECEPTOR DOUBLE MUTANT WITH BOUND CORTISONE | MINERALOCORTICOID RECEPTOR, MR, NUCLEAR RECEPTOR, STEROID RECEPTOR, CORTISONE, HYPERTENSION, TRANSCRIPTION
2ab2:A (SER737) to (SER805) MINERALOCORTICOID RECEPTOR DOUBLE MUTANT WITH BOUND SPIRONOLACTONE | MINERALOCORTICOID RECEPTOR, MR, NUCLEAR RECEPTOR, STEROID RECEPTOR, SPIRONOLACTONE, HYPERTENSION, TRANSCRIPTION
2ab2:B (SER737) to (GLN803) MINERALOCORTICOID RECEPTOR DOUBLE MUTANT WITH BOUND SPIRONOLACTONE | MINERALOCORTICOID RECEPTOR, MR, NUCLEAR RECEPTOR, STEROID RECEPTOR, SPIRONOLACTONE, HYPERTENSION, TRANSCRIPTION
2abi:A (PRO738) to (SER805) CRYSTAL STRUCTURE OF THE HUMAN MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN BOUND TO DEOXYCORTICOSTERONE | MINERALOCORTICOID RECEPTOR, STEROID RECEPTO, NUCLEAR RECEPT, TRANSCRIPTION REGULATION, ACTIVATING MUTATION, HYPERTENSION, TRANSCRIPTION REGULATOR
2abi:B (PRO738) to (SER805) CRYSTAL STRUCTURE OF THE HUMAN MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN BOUND TO DEOXYCORTICOSTERONE | MINERALOCORTICOID RECEPTOR, STEROID RECEPTO, NUCLEAR RECEPT, TRANSCRIPTION REGULATION, ACTIVATING MUTATION, HYPERTENSION, TRANSCRIPTION REGULATOR
2abi:C (SER737) to (SER805) CRYSTAL STRUCTURE OF THE HUMAN MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN BOUND TO DEOXYCORTICOSTERONE | MINERALOCORTICOID RECEPTOR, STEROID RECEPTO, NUCLEAR RECEPT, TRANSCRIPTION REGULATION, ACTIVATING MUTATION, HYPERTENSION, TRANSCRIPTION REGULATOR
3b65:A (PRO671) to (TRP741) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH SARM S-24 | ANDROGEN RECEPTOR, SARM, DISEASE MUTATION, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRIPLET REPEAT EXPANSION, UBL CONJUGATION, ZINC, ZINC-FINGER
3b68:A (PRO671) to (SER740) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH SARM S-4 | ANDROGEN RECEPTOR, SARM, DISEASE MUTATION, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRIPLET REPEAT EXPANSION, UBL CONJUGATION, ZINC, ZINC-FINGER
3mek:A (GLU86) to (SER182) CRYSTAL STRUCTURE OF HUMAN HISTONE-LYSINE N- METHYLTRANSFERASE SMYD3 IN COMPLEX WITH S-ADENOSYL-L- METHIONINE | HISTONE METHYLTRANSFERASE, SET AND MYND DOMAIN-CONTAINING PROTEIN 3, ZINC FINGER MYND DOMAIN-CONTAINING PROTEIN 1, HISTONE H3, DI-METHYLATION, TRI-METHYLATION, TRANSCRIPTIONAL ACTIVATION, DNA-BINDING, MYND-TYPE ZINC FINGER, SET DOMAIN, CHROMATIN MODIFICATION, ALTERNATIVE SPLICING, CHROMATIN REGULATOR, CYTOPLASM, METAL-BINDING, METHYLTRANSFERASE, NUCLEUS, S-ADENOSYL-L-METHIONINE, TRANSFERASE, ZINC, ZINC-FINGER, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
5ex0:A (GLU86) to (CYS180) CRYSTAL STRUCTURE OF HUMAN SMYD3 IN COMPLEX WITH A MAP3K2 PEPTIDE | SET DOMAIN, METHYLATION, CHROMATIN, CANCER, TRANSFERASE
3bqd:A (THR531) to (SER599) DOUBLING THE SIZE OF THE GLUCOCORTICOID RECEPTOR LIGAND BINDING POCKET BY DEACYLCORTIVAZOL | GLUCOCORTICOID RECEPTOR, DEACYLCORTIVAZOL, SRC1, NUCLEAR RECEPTOR COACTIVATOR 1 ISOFORM 1, DIMER INTERFACE, HORMONE BINDING POCKET, CHARGE CLAMP, COACTIVATOR, ALTERNATIVE INITIATION, ALTERNATIVE SPLICING, CHROMATIN REGULATOR, CYTOPLASM, DISEASE MUTATION, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, PSEUDOHERMAPHRODITISM, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, UBL CONJUGATION, ZINC, ZINC- FINGER, ACYLTRANSFERASE, CHROMOSOMAL REARRANGEMENT, PROTO- ONCOGENE, TRANSFERASE, PROTEIN BINDING
3bs5:B (ILE136) to (GLY184) CRYSTAL STRUCTURE OF HCNK2-SAM/DHYP-SAM COMPLEX | STERILE ALPHA MOTIF, SAM DOMAIN, SAM DOMAIN DIMER, SAM DOMAIN COMPLEX, CYTOPLASM, MEMBRANE, SENSORY TRANSDUCTION, VISION, ALTERNATIVE SPLICING, COILED COIL, PHOSPHOPROTEIN, POLYMORPHISM, SIGNALING PROTEIN/MEMBRANE PROTEIN COMPLEX
3c07:B (GLU136) to (ALA209) CRYSTAL STRUCTURE OF A TETR FAMILY TRANSCRIPTIONAL REGULATOR FROM STREPTOMYCES COELICOLOR A3(2) | APC6322, TETR, STREPTOMYCES COELICOLOR A3(2), STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, DNA-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSCRIPTION REGULATOR
3n71:A (CYS90) to (CYS179) CRYSTAL STRUCTURE OF CARDIAC SPECIFIC HISTONE METHYLTRANSFERASE SMYD1 | HISTONE LYSINE METHYLTRANSFERASE, SMYD1, HEART DEVELOPMENT, MYND, TRANSCRIPTION
4c2q:A (ASN374) to (ALA456) CRYSTAL STRUCTURE OF HUMAN TESTIS ANGIOTENSIN-I CONVERTING ENZYME MUTANT R522K | HYDROLASE, CHLORIDE ACTIVATION, HYPERTENSION
4rh7:A (ASN3587) to (ASN3654) CRYSTAL STRUCTURE OF HUMAN CYTOPLASMIC DYNEIN 2 MOTOR DOMAIN IN COMPLEX WITH ADP.VI | AAA+ PROTEIN, MOTOR PROTEIN, DYNEIN MOTOR DOMAIN
5fqr:A (THR311) to (ALA382) SELECTIVE ESTROGEN RECEPTOR DOWNREGULATOR ANTAGONISTS: TETRAHYDROISOQUINOLINE PHENOLS 2. | SIGNALING PROTEIN, BREAST CANCER, ESTROGEN RECEPTOR DOWNREGULATOR, FULVESTRANT, THIQ, NUCLEAR HORMONE RECEPTOR
5fqs:A (THR311) to (ALA382) SELECTIVE ESTROGEN RECEPTOR DOWNREGULATOR ANTAGONISTS: TETRAHYDROISOQUINOLINE PHENOLS 3. | SIGNALING PROTEIN, BREAST CANCER, ESTROGEN RECEPTOR DOWNREGULATOR, FULVESTRANT, THIQ, NUCLEAR HORMONE RECEPTOR
5fqt:A (THR311) to (SER395) SELECTIVE ESTROGEN RECEPTOR DOWNREGULATOR ANTAGONISTS: TETRAHYDROISOQUINOLINE PHENOLS 4. | SIGNALING PROTEIN, BREAST CANCER, ESTROGEN RECEPTOR DOWNREGULATOR, FULVESTRANT, THIQ, NUCLEAR HORMONE RECEPTOR
4cgz:A (VAL1077) to (LYS1153) CRYSTAL STRUCTURE OF THE BLOOM'S SYNDROME HELICASE BLM IN COMPLEX WITH DNA | HYDROLASE-DNA COMPLEX
4cid:A (ALA290) to (ASP367) STRUCTURAL INSIGHTS INTO THE N-TERMINUS OF THE EHD2 ATPASE | HYDROLASE, MECHANOCHEMICAL ATPASE, DYNAMIN SUPERFAMILY
4cnk:A (SER261) to (PHE293) L-AMINOACETONE OXIDASE FROM STREPTOCOCCUS OLIGOFERMENTANS BELONGS TO A NEW 3-DOMAIN FAMILY OF BACTERIAL FLAVOPROTEINS | OXIDOREDUCTASE, FLAVOPROTEINS
3d24:C (LEU197) to (LEU278) CRYSTAL STRUCTURE OF LIGAND-BINDING DOMAIN OF ESTROGEN- RELATED RECEPTOR ALPHA (ERRALPHA) IN COMPLEX WITH THE PEROXISOME PROLIFERATORS-ACTIVATED RECEPTOR COACTIVATOR- 1ALPHA BOX3 PEPTIDE (PGC-1ALPHA) | NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, COACTIVATOR, DNA- BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, POLYMORPHISM, RNA-BINDING, STRUCTURAL GENOMICS, STRUCTURAL PROTEOMICS IN EUROPE, SPINE
3d90:A (PRO686) to (SER754) CRYSTAL STRUCTURE OF THE HUMAN PROGESTERONE RECEPTOR LIGAND- BINDING DOMAIN BOUND TO LEVONORGESTREL | PROGESTERONE RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, WOMEN HEALTH, CONTRACEPTION, ALTERNATIVE SPLICING, DNA-BINDING, LIPID-BINDING, METAL- BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
3d90:B (PRO686) to (SER754) CRYSTAL STRUCTURE OF THE HUMAN PROGESTERONE RECEPTOR LIGAND- BINDING DOMAIN BOUND TO LEVONORGESTREL | PROGESTERONE RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, WOMEN HEALTH, CONTRACEPTION, ALTERNATIVE SPLICING, DNA-BINDING, LIPID-BINDING, METAL- BINDING, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
3ofn:K (ASP413) to (ASN479) STRUCTURE OF FOUR MUTANT FORMS OF YEAST F1 ATPASE: ALPHA-N67I | ATP SYNTHASE, ATP PHOSPHATASE, F1F0 ATPASE, ATP SYNTHESIS, HYDROLASE, ADP, PO4, MITOCHONDRIA
4tuz:B (THR311) to (TRP383) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH ALPHA-ZEARALENOL | NUCLEAR HORMONE RECEPTOR LIGAND BINDING DOMAIN ENDOCRINE DISRUPTOR ENVIRONMENTAL COMPOUND, NUCLEAR PROTEIN
4tv1:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF HERA-LBD (Y537S) IN COMPLEX WITH PROPYLPARABEN | NUCLEAR HORMONE RECEPTOR, LIGAND BINDING DOMAIN, ENDOCRINE DISRUPTOR, ENVIRONMENTAL COMPOUND, HORMONE RECEPTOR
4txy:A (THR26) to (MET95) CRYSTAL STRUCTURE OF VIBRIO CHOLERAE DNCV CYCLIC AMP-GMP SYNTHASE, A PROKARYOTIC CGAS HOMOLOG | NUCLEOTIDYL TRANSFERASE, CYCLIC NUCLEOTIDE SYNTHASE, CGAS
4txy:B (THR26) to (TYR93) CRYSTAL STRUCTURE OF VIBRIO CHOLERAE DNCV CYCLIC AMP-GMP SYNTHASE, A PROKARYOTIC CGAS HOMOLOG | NUCLEOTIDYL TRANSFERASE, CYCLIC NUCLEOTIDE SYNTHASE, CGAS
4txz:B (GLU28) to (TYR93) CRYSTAL STRUCTURE OF VIBRIO CHOLERAE DNCV CYCLIC AMP-GMP SYNTHASE IN COMPLEX WITH NONHYDROLYZABLE GTP | NUCLEOTIDYL TRANSFERASE, CYCLIC NUCLEOTIDE SYNTHASE, CGAS
4ty0:A (THR26) to (MET95) CRYSTAL STRUCTURE OF VIBRIO CHOLERAE DNCV CYCLIC AMP-GMP SYNTHASE IN COMPLEX WITH LINEAR INTERMEDIATE 5' PPPA(3',5')PG | NUCLEOTIDYL TRANSFERASE, CYCLIC NUCLEOTIDE SYNTHASE, CGAS, TRANSFERASE
4ty0:B (THR26) to (ILE92) CRYSTAL STRUCTURE OF VIBRIO CHOLERAE DNCV CYCLIC AMP-GMP SYNTHASE IN COMPLEX WITH LINEAR INTERMEDIATE 5' PPPA(3',5')PG | NUCLEOTIDYL TRANSFERASE, CYCLIC NUCLEOTIDE SYNTHASE, CGAS, TRANSFERASE
4u0l:A (THR25) to (TYR92) STRUCTURE OF THE VIBRIO CHOLERAE DI-NUCLEOTIDE CYCLASE (DNCV) MUTANT D131A-D133A | REGULATION, MUTATION, TRANSFERASE
4u0m:A (THR25) to (TYR92) STRUCTURE OF THE VIBRIO CHOLERAE DI-NUCLEOTIDE CYCLASE (DNCV) MUTANT D193N IN COMPLEX WITH ATP, GTP AND 5MTHFGLU2 | REGULATION, MUTATION, TRANSFERASE
4u0m:B (THR25) to (TYR92) STRUCTURE OF THE VIBRIO CHOLERAE DI-NUCLEOTIDE CYCLASE (DNCV) MUTANT D193N IN COMPLEX WITH ATP, GTP AND 5MTHFGLU2 | REGULATION, MUTATION, TRANSFERASE
4u0z:A (LEU258) to (ARG308) EUKARYOTIC FIC DOMAIN CONTAINING PROTEIN WITH BOUND APCPP | TPR, FIC, APCPP, ADENYLATION, TRANSFERASE
4u0z:B (LEU258) to (ARG308) EUKARYOTIC FIC DOMAIN CONTAINING PROTEIN WITH BOUND APCPP | TPR, FIC, APCPP, ADENYLATION, TRANSFERASE
4u0z:C (LEU258) to (ARG308) EUKARYOTIC FIC DOMAIN CONTAINING PROTEIN WITH BOUND APCPP | TPR, FIC, APCPP, ADENYLATION, TRANSFERASE
4u0z:D (LEU258) to (ARG308) EUKARYOTIC FIC DOMAIN CONTAINING PROTEIN WITH BOUND APCPP | TPR, FIC, APCPP, ADENYLATION, TRANSFERASE
4u0z:E (LEU258) to (ARG308) EUKARYOTIC FIC DOMAIN CONTAINING PROTEIN WITH BOUND APCPP | TPR, FIC, APCPP, ADENYLATION, TRANSFERASE
4u0z:F (LEU258) to (ARG308) EUKARYOTIC FIC DOMAIN CONTAINING PROTEIN WITH BOUND APCPP | TPR, FIC, APCPP, ADENYLATION, TRANSFERASE
4u0z:G (LEU258) to (ARG308) EUKARYOTIC FIC DOMAIN CONTAINING PROTEIN WITH BOUND APCPP | TPR, FIC, APCPP, ADENYLATION, TRANSFERASE
4u0z:H (LEU258) to (ARG308) EUKARYOTIC FIC DOMAIN CONTAINING PROTEIN WITH BOUND APCPP | TPR, FIC, APCPP, ADENYLATION, TRANSFERASE
3dt3:A (THR311) to (ALA382) HUMAN ESTROGEN RECEPTOR ALPHA LBD WITH GW368 | ESTROGEN RECEPTOR, NUCLEAR RECEPTOR, SERM, TRANSCRIPTION FACTOR, ALPHA-HELICAL SANDWICH, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3os8:C (THR311) to (TRP383) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3os8:D (THR311) to (TRP383) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3os9:A (THR311) to (SER395) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3os9:B (THR311) to (SER395) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3os9:C (THR311) to (SER395) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3os9:D (THR311) to (SER395) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3osa:A (THR311) to (SER395) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3osa:B (THR311) to (SER395) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3osa:C (THR311) to (TRP383) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3osa:D (THR311) to (TRP383) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3oxg:A (GLU86) to (SER182) HUMAN LYSINE METHYLTRANSFERASE SMYD3 IN COMPLEX WITH ADOHCY (FORM III) | SMYD PROTEINS, MYND, SET DOMAIN, HISTONE LYSINE METHYLTRANSFERASE, HISTONE METHYLATION, H3K4, TRANSFERASE
3oxl:A (GLU86) to (SER182) HUMAN LYSINE METHYLTRANSFERASE SMYD3 IN COMPLEX WITH ADOHCY (FORM II) | SMYD PROTEINS, MYND, SET DOMAIN, HISTONE LYSINE METHYLTRANSFERASE, HISTONE METHYLATION, H3K4, TRANSFERASE
5hi7:A (HIS83) to (SER182) CO-CRYSTAL STRUCTURE OF HUMAN SMYD3 WITH AN AZA-SAH COMPOUND | SMYD3, METHYLTRANSFERASE, ONCOLOGY, INHIBITOR, TRANSFERASE-INHIBITOR COMPLEX
3p47:A (THR57) to (CYS145) CRYSTAL STRUCTURE OF ENTAMOEBA HISTOLYTICA SERINE ACETYLTRANSFERASE 1 IN COMPLEX WITH L-CYSTEINE | SERINE ACETYLTRANSFERASE, CYSTEINE SYNTHASE, ACETYLTRANSFERASE, TRANSFERASE
5hq8:A (GLU86) to (SER182) CO-CRYSTAL STRUCTURE OF HUMAN SMYD3 WITH A MEKK2 PEPTIDE AT 2.13A | SMYD3, METHYLTRANSFERASE, ONCOLOGY, TRANSFERASE
5hq8:B (GLU86) to (SER182) CO-CRYSTAL STRUCTURE OF HUMAN SMYD3 WITH A MEKK2 PEPTIDE AT 2.13A | SMYD3, METHYLTRANSFERASE, ONCOLOGY, TRANSFERASE
4u9l:A (ARG353) to (ALA449) STRUCTURE OF A MEMBRANE PROTEIN | CHANNEL, MAGNESIUM, METAL TRANSPORT
4uda:A (PRO738) to (SER805) MR IN COMPLEX WITH DEXAMETHASONE | SIGNALING PROTEIN, NUCLEAR HORMONE RECEPTOR, LIGAND COMPLEX, PEPTIDE COMPLEX
4udb:A (VAL739) to (SER805) MR IN COMPLEX WITH DESISOBUTYRYLCICLESONIDE | SIGNALING PROTEIN, NUCLEAR HORMONE RECEPTOR, LIGAND COMPLEX, PEPTIDE COMPLEX
4udc:A (VAL533) to (SER599) GR IN COMPLEX WITH DEXAMETHASONE | SIGNALING PROTEIN, NUCLEAR HORMONE RECEPTOR, LIGAND COMPLEX, PEPTIDE COMPLEX
3pdn:A (HIS83) to (SER182) CRYSTAL STRUCTURE OF SMYD3 IN COMPLEX WITH METHYLTRANSFERASE INHIBITOR SINEFUNGIN | ROSSMANN FOLD, ZINC FINGER, METHYLTRANSFERASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4uur:B (GLY30) to (ILE142) COLD-ADAPTED TRUNCATED HEMOGLOBIN FROM THE ANTARCTIC MARINE BACTERIUM PSEUDOALTEROMONAS HALOPLANKTIS TAC125 | OXIDOREDUCTASE
4ezj:A (GLN550) to (ALA612) POTENT AND SELECTIVE INHIBITORS OF PI3K-DELTA: OBTAINING ISOFORM SELECTIVITY FROM THE AFFINITY POCKET AND TRYPTOPHAN SHELF | KINASE P110, P110-GAMMA, LIPID KINASE, CYTOPLASMIC, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3qwp:A (LYS84) to (SER182) CRYSTAL STRUCTURE OF SET AND MYND DOMAIN CONTAINING 3; ZINC FINGER MYND DOMAIN-CONTAINING PROTEIN 1 | SMYD3,SET AND MYND DOMAIN, ZINC FINGER MYND DOMAIN-CONTAINING PROTEIN 1, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSFERASE
4fhn:X (LEU7) to (GLU56) NUP37-NUP120 FULL-LENGTH COMPLEX FROM SCHIZOSACCHAROMYCES POMBE | PROTEIN COMPLEX,STRUCTURAL PROTEIN,NUCLEAR PORE COMPLEX,MRNA TRANSPORT,PROTEIN TRANSPORT, WD REPEAT, HELICAL DOMAIN, TRANSLOCATION, TRANSPORT, ROSSMANN FOLD, DEHYDROGENASE, NADP BINDING DOMAIN, STRUCTURAL PROTEIN-OXIDOREDUCTASE COMPLEX
4w8f:A (PRO2619) to (TYR2680) CRYSTAL STRUCTURE OF THE DYNEIN MOTOR DOMAIN IN THE AMPPNP-BOUND STATE | CYTOPLASMIC DYNEIN, MICROTUBULE, ATPASE, AAA+, AMPPNP
4fn9:A (SER2) to (TYR69) X-RAY CRYSTAL STRUCTURE OF THE ANCESTRAL 3-KETO STEROID RECEPTOR - PROGESTERONE COMPLEX | HORMONE, ANCESTRAL, STEROID RECEPTOR, NUCLEAR RECEPTOR, PROGESTERONE RECEPTOR, CYTOSOLIC, NUCLEAR, STEROID-BINDING PROTEIN
4fn9:B (ILE4) to (GLN68) X-RAY CRYSTAL STRUCTURE OF THE ANCESTRAL 3-KETO STEROID RECEPTOR - PROGESTERONE COMPLEX | HORMONE, ANCESTRAL, STEROID RECEPTOR, NUCLEAR RECEPTOR, PROGESTERONE RECEPTOR, CYTOSOLIC, NUCLEAR, STEROID-BINDING PROTEIN
5kce:B (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-METHYL, 2-CHLOROBENZYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, SIGNALING PROTEIN, TRANSCRIPTION
5kcf:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-ETHYL, 4-METHOXYBENZYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5kct:B (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-ETHYL, 4-CHLOROBENZYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5kcu:A (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-ETHYL, ALPHA-NAPHTHYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5kd9:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-TRIFLUOROETHYL 4-CHLOROBENZYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
3rlj:A (PRO671) to (TRP741) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH SARM S-22 | STEROID RECEPTOR, DHT, TESTOSTERONE, TRANSCRIPTION
2axa:A (ILE672) to (SER740) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH S-1 | TRANSCRIPTION
1bg3:A (SER746) to (LEU807) RAT BRAIN HEXOKINASE TYPE I COMPLEX WITH GLUCOSE AND INHIBITOR GLUCOSE-6-PHOSPHATE | HEXOKINASE, PHOSPHOTRANSFERASE
2pix:A (PRO671) to (TYR739) AR LBD WITH SMALL MOLECULE | AR LBD IHNIBITORS COACTIVATOR BINDING, HORMONE RECEPTOR
2q70:B (THR311) to (SER395) ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN COMPLXED TO A BENZOPYRAN LIGAND | TRANSCRIPTION FACTOR, ESTROGEN RECEPTOR
3g3b:B (THR89) to (THR118) STRUCTURE OF A LAMPREY VARIABLE LYMPHOCYTE RECEPTOR MUTANT IN COMPLEX WITH A PROTEIN ANTIGEN | VLR, ANTIBODY, X-RAY, CRYSTALLOGRAPHY, ALLERGEN, ANTIMICROBIAL, BACTERIOLYTIC ENZYME, GLYCOSIDASE, HYDROLASE, HYDROLASE/IMMUNE SYSTEM COMPLEX
3gn8:A (THR0) to (SER68) X-RAY CRYSTAL STRUCTURE OF ANCGR2 IN COMPLEX WITH DEXAMETHASONE | NUCLEAR RECEPTOR, GR2, EVOLUTION, GLUCOCORTICOID RECEPTOR, DEXAMETHASONE, CORTISOL, ACTIVATOR, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, TRANSCRIPTION, TRANSCRIPTION REGULATION, HORMONE/HORMONE ACTIVATOR COMPLEX
3tg4:A (TRP83) to (CYS181) STRUCTURE OF SMYD2 IN COMPLEX WITH SAM | SET DOMAIN, METHYLTRANSFERASE, CO FACTOR BINDING, TRANSFERASE
1err:A (THR311) to (LEU379) HUMAN ESTROGEN RECEPTOR LIGAND-BINDING DOMAIN IN COMPLEX WITH RALOXIFENE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, STEROID, ANTAGONIST
1err:B (THR311) to (LEU379) HUMAN ESTROGEN RECEPTOR LIGAND-BINDING DOMAIN IN COMPLEX WITH RALOXIFENE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, STEROID, ANTAGONIST
2gln:A (HIS22) to (THR127) CRYSTAL STRUCTURE OF MYCOBACTERIUM TUBERCULOSIS TRHBN, GLNE11ALA MUTANT | TRUNCATED HEMOGLOBIN; MUTANT, OXYGEN STORAGE/TRANSPORT COMPLEX
2gln:B (HIS22) to (THR127) CRYSTAL STRUCTURE OF MYCOBACTERIUM TUBERCULOSIS TRHBN, GLNE11ALA MUTANT | TRUNCATED HEMOGLOBIN; MUTANT, OXYGEN STORAGE/TRANSPORT COMPLEX
4zn7:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH DIETHYLSTILBESTROL | NUCLEAR RECEPTOR TRANSCRIPTION FACTOR NUCLEUS PROTEIN-LIGAND COMPLEX, TRANSCRIPTION
4znu:A (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH A 2-METHYL-SUBSTITUTED OBHS DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
2w8y:A (PRO686) to (SER754) RU486 BOUND TO THE PROGESTERONE RECEPTOR IN A DESTABILIZED AGONISTIC CONFORMATION | RECEPTOR, PROGESTERONE RECEPTOR, RU-486, MIFEPRISTONE
2w8y:B (PRO686) to (TRP755) RU486 BOUND TO THE PROGESTERONE RECEPTOR IN A DESTABILIZED AGONISTIC CONFORMATION | RECEPTOR, PROGESTERONE RECEPTOR, RU-486, MIFEPRISTONE
5aav:B (THR311) to (TRP383) OPTIMIZATION OF A NOVEL BINDING MOTIF TO TO (E)-3-(3,5- DIFLUORO-4-((1R,3R)-2-(2-FLUORO-2-METHYLPROPYL)-3-METHYL-2, 3,4,9-TETRAHYDRO-1H-PYRIDO(3,4-B)INDOL-1-YL)PHENYL)ACRYLIC ACID (AZD9496), A POTENT AND ORALLY BIOAVAILABLE SELECTIVE ESTROGEN RECEPTOR DOWNREGULATOR AND ANTAGONIST | SIGNALING PROTEIN, BREAST CANCER, ESTROGEN RECEPTOR DOWNREGULATOR, FULVESTRANT, AZD9496, NUCLEAR HORMONE RECEPTOR
5acc:A (THR311) to (ALA382) A NOVEL ORAL SELECTIVE ESTROGEN RECEPTOR DOWN-REGULATOR, AZD9496, DRIVES TUMOUR GROWTH INHIBITION IN ESTROGEN RECEPTOR POSITIVE AND ESR1 MUTANT MODELS | SIGNALING PROTEIN, SERD, METASTATIC BREAST CANCER, ER MUTATION, ESR1 MUTATION, COMBINATION THERAPY
3wff:A (PRO738) to (SER805) MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN WITH COMPUOND 2B | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, TRANSCRIPTION, HYPERTENSION, NON-STEROIDAL ANTAGONIST, ACTIVATING MUTATION, TRANSCRIPTION- INHIBITOR COMPLEX
5ak2:A (THR311) to (SER395) OXYPHENYLPROPENOIC ACIDS AS ORAL SELECTIVE ESTROGEN RECEPTOR DOWN-REGULATORS. | SIGNALING PROTEIN
5ak2:B (THR311) to (TRP383) OXYPHENYLPROPENOIC ACIDS AS ORAL SELECTIVE ESTROGEN RECEPTOR DOWN-REGULATORS. | SIGNALING PROTEIN
3j9t:Q (THR64) to (ASP155) YEAST V-ATPASE STATE 1 | V-ATPASE, V-TYPE ATPASE, VACUOLAR-TYPE ATPASE, PROTON PUMP, HYDROLASE
2jfa:B (THR311) to (SER395) ESTROGEN RECEPTOR ALPHA LBD IN COMPLEX WITH AN AFFINITY- SELECTED COREPRESSOR PEPTIDE | TRANSCRIPTION, TRANSCRIPTION FACTOR, PHAGE DISPLAY, METAL-BINDING, COREPRESSOR, LIPID-BINDING, TRANSCRIPTION REGULATION, LIGAND-BINDING DOMAIN (LBD), NUCLEAR PROTEIN, PHOSPHORYLATION, STEROID- BINDING, RECEPTOR, ZINC-FINGER, DNA-BINDING, NUCLEAR RECEPTOR, PEPTIDE ANTAGONIST
3zrb:B (PRO686) to (TRP755) STRUCTURAL BASIS FOR AGONISM AND ANTAGONISM FOR A SET OF CHEMICALLY RELATED PROGESTERONE RECEPTOR MODULATORS | RECEPTOR, AGONIST, ANTAGONIST
2yg8:B (PRO61) to (GLY108) STRUCTURE OF AN UNUSUAL 3-METHYLADENINE DNA GLYCOSYLASE II ( ALKA) FROM DEINOCOCCUS RADIODURANS | HYDROLASE, DNA REPAIR
5ccl:A (GLU86) to (SER182) CRYSTAL STRUCTURE OF SMYD3 WITH SAM AND OXINDOLE COMPOUND | PROTEIN-INHIBITOR COMPLEX, METHYLTRANSFERASE, EPIGENETICS, DRUG DISCOVERY, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5cj6:A (ILE672) to (SER740) CRYSTAL STRUCTURE OF A SELECTIVE ANDROGEN RECEPTOR MODULATOR BOUND TO THE LIGAND BINDING DOMAIN OF THE HUMAN ANDROGEN RECEPTOR | ANDROGEN RECEPTOR, NUCLEAR HORMONE RECEPTOR, SIGNALING PROTEIN
3l3n:A (ASN374) to (GLY474) TESTIS ACE CO-CRYSTAL STRUCTURE WITH NOVEL INHIBITOR LISW | ENZYME-INHIBITOR COMPLEX, ANGIOTENSIN-CONVERTING ENZYME (ACE) INHIBITORS, TESTIS, CARBOXYPEPTIDASE, HYDROLASE
4ppp:B (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH FLUORO-RESVERATROL | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, PROTEIN BINDING
4pps:B (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH AN A-CD RING ESTROGEN DERIVATIVE | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, PROTEIN BINDING
5dyb:A (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-(3,4-DIHYDRONAPHTHALEN-2(1H)- YLIDENEMETHANEDIYL)DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
3b5r:A (PRO671) to (TRP741) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH SARM C-31 | ANDROGEN RECEPTOR, NONSTEROIDAL, SARM, DISEASE MUTATION, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRIPLET REPEAT EXPANSION, UBL CONJUGATION, ZINC, ZINC-FINGER
4qox:A (ILE348) to (ILE435) CRYSTAL STRUCTURE OF CDPK4 FROM PLASMODIUM FALCIPARUM, PF3D7_0717500 | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, CDPK, PLASMODIUM, MALARIA, TRANSFERASE
5ex3:A (HIS83) to (SER182) CRYSTAL STRUCTURE OF HUMAN SMYD3 IN COMPLEX WITH A VEGFR1 PEPTIDE | SET DOMAIN, METHYLATION, CHROMATIN, CANCER, TRANSFERASE
3bkl:A (LEU375) to (GLY474) TESTIS ACE CO-CRYSTAL STRUCTURE WITH KETONE ACE INHIBITOR KAW | ENZYME-INHIBITOR COMPLEX, GEM-DIOL, DOMAIN-SELECTIVE, CARBOXYPEPTIDASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, METAL-BINDING, METALLOPROTEASE, PHOSPHOPROTEIN, PROTEASE, SECRETED, TRANSMEMBRANE
4bla:D (CYS544) to (THR601) CRYSTAL STRUCTURE OF FULL-LENGTH HUMAN SUPPRESSOR OF FUSED (SUFU) MUTANT LACKING A REGULATORY SUBDOMAIN (CRYSTAL FORM II) | SIGNALING PROTEIN, SUGAR BINDING PROTEIN-SIGNALING PROTEIN COMPLEX, HEDGEHOG GENE REGULATION, SIGNAL TRANSDUCTION, GLI, TRANSCRIPTION FACTOR
5eyv:A (ASN391) to (ASP441) CRYSTAL STRUCTURE OF ADENYLOSUCCINATE LYASE FROM SCHISTOSOMA MANSONI IN APO FORM. | LYASE
5fqv:A (THR311) to (ALA382) SELECTIVE ESTROGEN RECEPTOR DOWNREGULATOR ANTAGONISTS: TETRAHYDROISOQUINOLINE PHENOLS 5. | SIGNALING PROTEIN, BREAST CANCER, ESTROGEN RECEPTOR DOWNREGULATOR, FULVESTRANT, THIQ, NUCLEAR HORMONE RECEPTOR
4cts:B (HIS123) to (LYS181) CRYSTAL STRUCTURE ANALYSIS AND MOLECULAR MODEL OF A COMPLEX OF CITRATE SYNTHASE WITH OXALOACETATE AND S-ACETONYL- COENZYME A | OXO-ACID-LYASE
4u03:A (THR25) to (TYR92) STRUCTURE OF THE VIBRIO CHOLERAE DI-NUCLEOTIDE CYCLASE (DNCV) IN COMPLEX WITH GTP AND 5MTHFGLU2 | REGULATION, TRANSFERASE
4u03:B (THR25) to (TYR92) STRUCTURE OF THE VIBRIO CHOLERAE DI-NUCLEOTIDE CYCLASE (DNCV) IN COMPLEX WITH GTP AND 5MTHFGLU2 | REGULATION, TRANSFERASE
5hcv:A (VAL739) to (SER805) IDENTIFICATION OF SPIROOXINDOLE AND DIBENZOXAZEPINE MOTIFS AS POTENT MINERALOCORTICOID RECEPTOR ANTAGONISTS | MINERALOCORTICOID RECEPTOR, LIGAND-BINDING DOMAIN, MR-LBD, ANTAGONISTS, CO-CRYSTAL, SIGNALING PROTEIN
5hcv:B (VAL739) to (SER805) IDENTIFICATION OF SPIROOXINDOLE AND DIBENZOXAZEPINE MOTIFS AS POTENT MINERALOCORTICOID RECEPTOR ANTAGONISTS | MINERALOCORTICOID RECEPTOR, LIGAND-BINDING DOMAIN, MR-LBD, ANTAGONISTS, CO-CRYSTAL, SIGNALING PROTEIN
5hcv:C (PRO738) to (SER805) IDENTIFICATION OF SPIROOXINDOLE AND DIBENZOXAZEPINE MOTIFS AS POTENT MINERALOCORTICOID RECEPTOR ANTAGONISTS | MINERALOCORTICOID RECEPTOR, LIGAND-BINDING DOMAIN, MR-LBD, ANTAGONISTS, CO-CRYSTAL, SIGNALING PROTEIN
3oxf:A (HIS83) to (SER182) HUMAN LYSINE METHYLTRANSFERASE SMYD3 IN COMPLEX WITH ADOHCY (FORM I) | SMYD PROTEINS, MYND, SET DOMAIN, HISTONE LYSINE METHYLTRANSFERASE, HISTONE METHYLATION, H3K4, TRANSFERASE
3oxf:B (GLU86) to (SER182) HUMAN LYSINE METHYLTRANSFERASE SMYD3 IN COMPLEX WITH ADOHCY (FORM I) | SMYD PROTEINS, MYND, SET DOMAIN, HISTONE LYSINE METHYLTRANSFERASE, HISTONE METHYLATION, H3K4, TRANSFERASE
3r2a:D (VAL232) to (GLY304) CRYSTAL STRUCTURE OF RXRALPHA LIGAND-BINDING DOMAIN COMPLEXED WITH COREPRESSOR SMRT2 AND ANTAGONIST RHEIN | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING DOMAIN, TRANSCRIPTION
5kcd:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-METHYL SUBSTITUTED OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
5kcd:B (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-METHYL SUBSTITUTED OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION