4gs8:A (ASP655) to (SER721) STRUCTURE ANALYSIS OF CYSTEINE FREE INSULIN DEGRADING ENZYME (IDE) WITH COMPOUND BDM43079 [{[(S)-2-(1H-IMIDAZOL-4-YL)-1-METHYLCARBAMOYL- ETHYLCARBAMOYL]-METHYL}-(3-PHENYL-PROPYL)-AMINO]-ACETIC ACID | INSULIN DEGRADING ENZYME, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4gs8:B (ASP655) to (SER721) STRUCTURE ANALYSIS OF CYSTEINE FREE INSULIN DEGRADING ENZYME (IDE) WITH COMPOUND BDM43079 [{[(S)-2-(1H-IMIDAZOL-4-YL)-1-METHYLCARBAMOYL- ETHYLCARBAMOYL]-METHYL}-(3-PHENYL-PROPYL)-AMINO]-ACETIC ACID | INSULIN DEGRADING ENZYME, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4waf:A (ARG975) to (HIS1048) CRYSTAL STRUCTURE OF A NOVEL TETRAHYDROPYRAZOLO[1,5-A]PYRAZINE IN AN ENGINEERED PI3K ALPHA | PI3K, CHIMERA, LIPID KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gsc:B (ASP655) to (SER721) STRUCTURE ANALYSIS OF INSULIN DEGRADING ENZYME WITH COMPOUND BDM41559 ((S)-2-[2-(CARBOXYMETHYL-PHENETHYL-AMINO)-ACETYLAMINO]-3-(1H- IMIDAZOL-4-YL)-PROPIONIC ACID METHYL ESTER) | INSULIN DEGRADING ENZYME, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4wbe:A (ARG133) to (GLY220) CRYSTAL STRUCTURE OF THE HR-1 DOMAIN OF HUMAN CAPRIN-1 IN THE C121 SPACE GROUP | ALL ALPHA HELICAL, RNA BINDING PROTEIN
4wbe:B (ARG133) to (GLY220) CRYSTAL STRUCTURE OF THE HR-1 DOMAIN OF HUMAN CAPRIN-1 IN THE C121 SPACE GROUP | ALL ALPHA HELICAL, RNA BINDING PROTEIN
4wbe:C (ARG133) to (GLY220) CRYSTAL STRUCTURE OF THE HR-1 DOMAIN OF HUMAN CAPRIN-1 IN THE C121 SPACE GROUP | ALL ALPHA HELICAL, RNA BINDING PROTEIN
4gsf:A (GLU656) to (SER721) THE STRUCTURE ANALYSIS OF CYSTEINE FREE INSULIN DEGRADING ENZYME (IDE) WITH (S)-2-{2-[CARBOXYMETHYL-(3-PHENYL-PROPIONYL)-AMINO]- ACETYLAMINO}-3-(3H-IMIDAZOL-4-YL)-PROPIONIC ACID METHYL ESTER | INSULIN DEGRADING ENZYME, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4gsf:B (ASP655) to (SER721) THE STRUCTURE ANALYSIS OF CYSTEINE FREE INSULIN DEGRADING ENZYME (IDE) WITH (S)-2-{2-[CARBOXYMETHYL-(3-PHENYL-PROPIONYL)-AMINO]- ACETYLAMINO}-3-(3H-IMIDAZOL-4-YL)-PROPIONIC ACID METHYL ESTER | INSULIN DEGRADING ENZYME, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4wbp:A (GLU134) to (GLY220) CRYSTAL STRUCTURE OF THE HR-1 DOMAIN OF HUMAN CAPRIN-1 IN THE P3121 SPACE GROUP | ALL ALPHA HELICAL, RNA BINDING PROTEIN
4wbp:B (ARG133) to (GLY220) CRYSTAL STRUCTURE OF THE HR-1 DOMAIN OF HUMAN CAPRIN-1 IN THE P3121 SPACE GROUP | ALL ALPHA HELICAL, RNA BINDING PROTEIN
4gtn:A (SER290) to (GLU365) STRUCTURE OF ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE FROM ACINETOBACTER BAYLYI | TRANSFERASE, PHOSPHORIBOSE BINDING
1n93:X (MET235) to (ARG287) CRYSTAL STRUCTURE OF THE BORNA DISEASE VIRUS NUCLEOPROTEIN | RNA VIRUS NUCLEOPROTEIN TETRAMER, VIRAL PROTEIN
3rn9:A (SER289) to (TRP338) STRUCTURE OF THE TOLUENE/O-XYLENE MONOOXYGENASE HYDROXYLASE T201S/L272E DOUBLE MUTANT | TOLUENE, HYDROXYLASE, FOUR-HELIX BUNDLE, DIIRON, OXYGEN PATHWAY, OXIDOREDUCTASE
3rp6:A (ASP331) to (GLY384) CRYSTAL STRUCTURE OF KLEBSIELLA PNEUMONIAE HPXO COMPLEXED WITH FAD | FAD-BINDING PROTEIN, MONOOXYGENASE, OXIDOREDUCTASE
3rp8:A (ASP331) to (GLY384) CRYSTAL STRUCTURE OF KLEBSIELLA PNEUMONIAE R204Q HPXO COMPLEXED WITH FAD | FAD-BINDING PROTEIN, MONOOXYGENASE, OXIDOREDUCTASE
4gxn:A (GLU110) to (TYR172) DIETHYLPHOSPHONATE INHIBITED STRUCTURE OF THE PROTEUS MIRABILIS LIPASE | LIPASE, HYDROLASE, A/B HYDROLASE FOLD, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2awi:A (ILE4) to (ALA65) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, REGULATORY DOMAIN, TRANSCRIPTION
2awi:B (ILE4) to (ALA65) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, REGULATORY DOMAIN, TRANSCRIPTION
2awi:D (LYS3) to (GLY66) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, REGULATORY DOMAIN, TRANSCRIPTION
2awi:E (ILE4) to (ALA65) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, REGULATORY DOMAIN, TRANSCRIPTION
2awi:F (ILE4) to (GLY66) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, REGULATORY DOMAIN, TRANSCRIPTION
2awi:G (ILE4) to (GLY66) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, REGULATORY DOMAIN, TRANSCRIPTION
2awi:H (GLY5) to (GLY66) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, REGULATORY DOMAIN, TRANSCRIPTION
2awi:I (ILE4) to (GLY66) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, REGULATORY DOMAIN, TRANSCRIPTION
2awi:J (SER6) to (GLY66) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, REGULATORY DOMAIN, TRANSCRIPTION
2awi:K (GLY5) to (ALA65) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, REGULATORY DOMAIN, TRANSCRIPTION
2awi:L (GLY5) to (ALA65) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, REGULATORY DOMAIN, TRANSCRIPTION
2axu:B (ILE4) to (ALA65) STRUCTURE OF PRGX | REPRESSOR, PHEROMONE, DNA BINDING, DOMAIN, TRANSCRIPTION
2axu:C (ILE4) to (GLY66) STRUCTURE OF PRGX | REPRESSOR, PHEROMONE, DNA BINDING, DOMAIN, TRANSCRIPTION
2axu:E (GLY5) to (ALA65) STRUCTURE OF PRGX | REPRESSOR, PHEROMONE, DNA BINDING, DOMAIN, TRANSCRIPTION
2axu:F (ILE4) to (GLY66) STRUCTURE OF PRGX | REPRESSOR, PHEROMONE, DNA BINDING, DOMAIN, TRANSCRIPTION
2axu:G (ILE4) to (GLY66) STRUCTURE OF PRGX | REPRESSOR, PHEROMONE, DNA BINDING, DOMAIN, TRANSCRIPTION
2axu:H (SER6) to (GLY66) STRUCTURE OF PRGX | REPRESSOR, PHEROMONE, DNA BINDING, DOMAIN, TRANSCRIPTION
2axu:I (SER6) to (ALA65) STRUCTURE OF PRGX | REPRESSOR, PHEROMONE, DNA BINDING, DOMAIN, TRANSCRIPTION
2axu:K (ILE4) to (ALA65) STRUCTURE OF PRGX | REPRESSOR, PHEROMONE, DNA BINDING, DOMAIN, TRANSCRIPTION
2axu:L (GLY5) to (ALA65) STRUCTURE OF PRGX | REPRESSOR, PHEROMONE, DNA BINDING, DOMAIN, TRANSCRIPTION
2axv:A (ILE4) to (ALA65) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, DOMAIN, TRANSCRIPTION
2axv:B (ILE4) to (ALA65) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, DOMAIN, TRANSCRIPTION
2axv:C (ILE4) to (ALA65) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, DOMAIN, TRANSCRIPTION
2axv:D (ILE4) to (ALA65) STRUCTURE OF PRGX Y153C MUTANT | REPRESSOR, PHEROMONE, DNA BINDING, DOMAIN, TRANSCRIPTION
1nom:A (LEU122) to (GLU147) DNA POLYMERASE BETA (POL B) (E.C.2.7.7.7), 31-KD DOMAIN; SOAKED IN THE PRESENCE OF MNCL2 (5 MILLIMOLAR) | DNA-DIRECTED DNA POLYMERASE, DNA REPLICATION, DNA REPAIR, NUCLEOTIDYLTRANSFERASE
3rxy:A (GLY68) to (GLU126) CRYSTAL STRUCTURE OF NIF3 SUPERFAMILY PROTEIN FROM SPHAEROBACTER THERMOPHILUS | STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, NIF3 SUPERFAMILY, UNKNOWN FUNCTION
4h80:H (LEU22) to (ALA82) CRYSTAL STRUCTURE OF HUMAN ALDH3A1 WITH ITS ISOZYME SELECTIVE INHIBITOR - N-[4-(4-METHYLSULFONYL-2-NITROANILINO)PHENYL]ACETAMIDE | CATALYZES BENZALDEHYDE, ROSSMANN FOLD, DEHYDROGENASE, NADP+ BINDING, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
1b3b:F (PRO336) to (GLY412) THERMOTOGA MARITIMA GLUTAMATE DEHYDROGENASE MUTANT N97D, G376K | METABOLIC ROLE, GLUTAMATE, DEHYDROGENASE, MUTANT, OXIDOREDUCTASE
4wwn:A (SER1003) to (LYS1078) CRYSTAL STRUCTURE OF HUMAN PI3K-GAMMA IN COMPLEX WITH (S)-N-(1-(7- FLUORO-2-(PYRIDIN-2-YL)QUINOLIN-3-YL)ETHYL)-9H-PURIN-6-AMINE AMG319 INHIBITOR | KINASE, PHOSPHOTRANSFER, PIP2
4wwo:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF HUMAN PI3K-GAMMA IN COMPLEX WITH PHENYLQUINOLINE INHIBITOR N-{(1S)-1-[8-CHLORO-2-(3-FLUOROPHENYL)QUINOLIN-3-YL]ETHYL}- 9H-PURIN-6-AMINE | KINASE, PHOSPHOTRANSFER, PIP2
4wwp:A (SER1003) to (LYS1078) CRYSTAL STRUCTURE OF HUMAN PI3K-GAMMA IN COMPLEX WITH PYRIDINYLQUINOLINE INHIBITOR N-{(1S)-1-[8-CHLORO-2-(2-METHYLPYRIDIN- 3-YL)QUINOLIN-3-YL]ETHYL}-9H-PURIN-6-AMINE | KINASE, PHOSPHOTRANSFER, PIP2
3ert:A (SER341) to (MET396) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH 4- HYDROXYTAMOXIFEN | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ESTROGEN, ANTAGONIST
1o17:A (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYL-TRANSFERASE (TRPD) | NUCLEOSIDE-PHOSPHORYLASES, TRANSFERASE
1o17:B (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYL-TRANSFERASE (TRPD) | NUCLEOSIDE-PHOSPHORYLASES, TRANSFERASE
1o17:C (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYL-TRANSFERASE (TRPD) | NUCLEOSIDE-PHOSPHORYLASES, TRANSFERASE
1o17:D (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYL-TRANSFERASE (TRPD) | NUCLEOSIDE-PHOSPHORYLASES, TRANSFERASE
3s2a:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF PI3K-GAMMA IN COMPLEX WITH A QUINOLINE INHIBITOR | P110-GAMMA, KINASE, PHOSPHOTRANSFER, P101, P84, LEUKOCYTES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4x1e:B (TYR108) to (GLY185) CRYSTAL STRUCTURE OF UNLIGANDED E. COLI TRANSCRIPTIONAL REGULATOR RUTR, W167A MUTANT | TRANSCRIPTIONAL REGULATOR, TETR FAMILY MEMBER, ARGININE AND PYRIMIDINE BIOSYNTHESIS, DNA BINDING, TRANSCRIPTION
1bgf:A (GLN3) to (GLN41) STAT-4 N-DOMAIN | TRANSCRIPTION FACTOR, REGULATION, DNA-BINDING
4hkm:A (GLU274) to (ALA343) CRYSTAL STRUCTURE OF AN ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TARGET ID NYSGRC-016600) FROM XANTHOMONAS CAMPESTRIS | STRUCTURAL GENOMICS, NYSGRC, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, TRANSFERASE
4hkm:B (ASP271) to (THR342) CRYSTAL STRUCTURE OF AN ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TARGET ID NYSGRC-016600) FROM XANTHOMONAS CAMPESTRIS | STRUCTURAL GENOMICS, NYSGRC, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, TRANSFERASE
2bma:A (SER369) to (GLY446) THE CRYSTAL STRUCTURE OF PLASMODIUM FALCIPARUM GLUTAMATE DEHYDROGENASE, A PUTATIVE TARGET FOR NOVEL ANTIMALARIAL DRUGS | PLASMODIUM FALCIPARUM, MALARIA, GLUTAMATE DEHYDROGENASE, DRUG DESIGN, CRYSTAL STRUCTURE ANALYSIS, OLIGOMER ORGANIZATION, NADP, OXIDOREDUCTASE
2bma:B (SER369) to (GLY446) THE CRYSTAL STRUCTURE OF PLASMODIUM FALCIPARUM GLUTAMATE DEHYDROGENASE, A PUTATIVE TARGET FOR NOVEL ANTIMALARIAL DRUGS | PLASMODIUM FALCIPARUM, MALARIA, GLUTAMATE DEHYDROGENASE, DRUG DESIGN, CRYSTAL STRUCTURE ANALYSIS, OLIGOMER ORGANIZATION, NADP, OXIDOREDUCTASE
2bma:C (SER369) to (GLY446) THE CRYSTAL STRUCTURE OF PLASMODIUM FALCIPARUM GLUTAMATE DEHYDROGENASE, A PUTATIVE TARGET FOR NOVEL ANTIMALARIAL DRUGS | PLASMODIUM FALCIPARUM, MALARIA, GLUTAMATE DEHYDROGENASE, DRUG DESIGN, CRYSTAL STRUCTURE ANALYSIS, OLIGOMER ORGANIZATION, NADP, OXIDOREDUCTASE
2bma:D (SER369) to (GLY446) THE CRYSTAL STRUCTURE OF PLASMODIUM FALCIPARUM GLUTAMATE DEHYDROGENASE, A PUTATIVE TARGET FOR NOVEL ANTIMALARIAL DRUGS | PLASMODIUM FALCIPARUM, MALARIA, GLUTAMATE DEHYDROGENASE, DRUG DESIGN, CRYSTAL STRUCTURE ANALYSIS, OLIGOMER ORGANIZATION, NADP, OXIDOREDUCTASE
2bma:E (SER369) to (GLY446) THE CRYSTAL STRUCTURE OF PLASMODIUM FALCIPARUM GLUTAMATE DEHYDROGENASE, A PUTATIVE TARGET FOR NOVEL ANTIMALARIAL DRUGS | PLASMODIUM FALCIPARUM, MALARIA, GLUTAMATE DEHYDROGENASE, DRUG DESIGN, CRYSTAL STRUCTURE ANALYSIS, OLIGOMER ORGANIZATION, NADP, OXIDOREDUCTASE
2bma:F (SER369) to (GLY446) THE CRYSTAL STRUCTURE OF PLASMODIUM FALCIPARUM GLUTAMATE DEHYDROGENASE, A PUTATIVE TARGET FOR NOVEL ANTIMALARIAL DRUGS | PLASMODIUM FALCIPARUM, MALARIA, GLUTAMATE DEHYDROGENASE, DRUG DESIGN, CRYSTAL STRUCTURE ANALYSIS, OLIGOMER ORGANIZATION, NADP, OXIDOREDUCTASE
4x58:A (ASP293) to (ILE370) ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE VARIANT N138A FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH PRPP AND MG | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MYCOBACTERIUM TUBERCULOSIS, MAGNESIUM, TRYPTOPHAN, MUTATION, TRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE
4x58:B (GLN295) to (ILE370) ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE VARIANT N138A FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH PRPP AND MG | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MYCOBACTERIUM TUBERCULOSIS, MAGNESIUM, TRYPTOPHAN, MUTATION, TRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE
4x59:A (ALA294) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE VARIANT P180A FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH PRPP AND MG | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MYCOBACTERIUM TUBERCULOSIS, MAGNESIUM, TRYPTOPHAN, MUTATION, TRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE
4x59:B (ASP293) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE VARIANT P180A FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH PRPP AND MG | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MYCOBACTERIUM TUBERCULOSIS, MAGNESIUM, TRYPTOPHAN, MUTATION, TRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE
4x5b:A (ASP293) to (GLN369) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE VARIANT R193L FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH PRPP AND MG | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MYCOBACTERIUM TUBERCULOSIS, MAGNESIUM, TRYPTOPHAN, MUTATION, TRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE
4x5a:A (ASP293) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE VARIANT R193A FROM MYCOBACTERIUM TUBERCULOSIS REMAINS LIGAND-FREE WHEN CO-CRYSTALLISED WITH PRPP AND MG | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MYCOBACTERIUM TUBERCULOSIS, MAGNESIUM, TRYPTOPHAN, MUTATION, TRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE
4x5a:B (ALA294) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE VARIANT R193A FROM MYCOBACTERIUM TUBERCULOSIS REMAINS LIGAND-FREE WHEN CO-CRYSTALLISED WITH PRPP AND MG | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MYCOBACTERIUM TUBERCULOSIS, MAGNESIUM, TRYPTOPHAN, MUTATION, TRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE
4x5c:B (ALA294) to (GLN369) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE VARIANT R193L FROM MYCOBACTERIUM TUBERCULOSIS WITH PYROPHOSPHATE/PRPP AND MG2+ BOUND | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MYCOBACTERIUM TUBERCULOSIS, MAGNESIUM, TRYPTOPHAN, MUTATION, TRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE
4x5e:A (ALA294) to (GLN369) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE VARIANT R194A FROM MYCOBACTERIUM TUBERCULOSIS WITH PYROPHOSPHATE, MG2+ AND ANTHRANILATE BOUND | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MYCOBACTERIUM TUBERCULOSIS, MAGNESIUM, TRYPTOPHAN, MUTATION, TRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE
4x5e:B (ASP293) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE VARIANT R194A FROM MYCOBACTERIUM TUBERCULOSIS WITH PYROPHOSPHATE, MG2+ AND ANTHRANILATE BOUND | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MYCOBACTERIUM TUBERCULOSIS, MAGNESIUM, TRYPTOPHAN, MUTATION, TRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE
1bpd:A (THR121) to (LYS148) CRYSTAL STRUCTURE OF RAT DNA POLYMERASE BETA: EVIDENCE FOR A COMMON POLYMERASE MECHANISM | NUCLEOTIDYLTRANSFERASE
2bpc:A (THR121) to (LYS148) CRYSTAL STRUCTURE OF RAT DNA POLYMERASE BETA: EVIDENCE FOR A COMMON POLYMERASE MECHANISM | NUCLEOTIDYLTRANSFERASE
2bpq:A (ASP293) to (ARG368) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (APO STRUCTURE) | TRANSFERASE, TRYPTOPHAN BIOSYNTHESIS, ANTHRANILATE, TRANSFERASE PHOSPHORIBOSYLTRANSFERASE, AMINO-ACID BIOSYNTHESIS, AROMATIC AMINO ACID BIOSYNTHESIS, GLYCOSYLTRANSFERASE, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, STRUCTURAL GENOMICS
2bpq:B (ASP293) to (GLN369) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (APO STRUCTURE) | TRANSFERASE, TRYPTOPHAN BIOSYNTHESIS, ANTHRANILATE, TRANSFERASE PHOSPHORIBOSYLTRANSFERASE, AMINO-ACID BIOSYNTHESIS, AROMATIC AMINO ACID BIOSYNTHESIS, GLYCOSYLTRANSFERASE, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, STRUCTURAL GENOMICS
1bvu:B (PRO338) to (GLY414) GLUTAMATE DEHYDROGENASE FROM THERMOCOCCUS LITORALIS | OXIDOREDUCTASE, THERMAL STABILITY
1bvu:E (PRO338) to (GLY414) GLUTAMATE DEHYDROGENASE FROM THERMOCOCCUS LITORALIS | OXIDOREDUCTASE, THERMAL STABILITY
4hs9:A (ILE111) to (PRO173) METHANOL TOLERANT MUTANT OF THE PROTEUS MIRABILIS LIPASE | LIPASE, HYDROLASE, ALPHA/BETA HYDROLASE
1c1h:A (LYS18) to (GLU73) CRYSTAL STRUCTURE OF BACILLUS SUBTILIS FERROCHELATASE IN COMPLEX WITH N-METHYL MESOPORPHYRIN | ROSSMANN FOLD, ALPHA/BETA FOLD, FERROCHELATASE, HEME SYNTHESIS, PORPHYRIN METALLATION, PI-HELIX, LYASE
3sd5:A (SER1003) to (LYS1078) CRYSTAL STRUCTURE OF PI3K GAMMA WITH 5-(2,4-DIMORPHOLINOPYRIMIDIN-6- YL)-4-(TRIFLUOROMETHYL)PYRIDIN-2-AMINE | LIPID KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3sks:A (ALA68) to (SER147) CRYSTAL STRUCTURE OF A PUTATIVE OLIGOENDOPEPTIDASE F FROM BACILLUS ANTHRACIS STR. AMES | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, OLIGOENDOPEPTIDASE, PROTEASE, HYDROLASE
4ifh:A (ASP655) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN DEGRADING ENZYME (IDE) IN COMPLEX WITH COMPOUND BDM44619 | INSULIN DEGRADING ENZYME, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4ifh:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN DEGRADING ENZYME (IDE) IN COMPLEX WITH COMPOUND BDM44619 | INSULIN DEGRADING ENZYME, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2chx:A (SER1003) to (GLY1079) A PHARMACOLOGICAL MAP OF THE PI3-K FAMILY DEFINES A ROLE FOR P110ALPHA IN SIGNALING: THE STRUCTURE OF COMPLEX OF PHOSPHOINOSITIDE 3-KINASE GAMMA WITH INHIBITOR PIK-90 | PHOSPHOINOSITIDE, KINASE, LIPID, INHIBITOR, 3-KINASE, SIGNALING, QUINAZOLINONE, TRANSFERASE
2chz:A (PRO1004) to (ASP1077) A PHARMACOLOGICAL MAP OF THE PI3-K FAMILY DEFINES A ROLE FOR P110ALPHA IN SIGNALING: THE STRUCTURE OF COMPLEX OF PHOSPHOINOSITIDE 3-KINASE GAMMA WITH INHIBITOR PIK-93 | PHOSPHOINOSITIDE, KINASE, LIPID, INHIBITOR, 3-KINASE, SIGNALING, PHENYLTHIAZOLE, QUINAZOLINONE, TRANSFERASE
3gag:C (ASP84) to (GLU127) CRYSTAL STRUCTURE OF A NITROREDUCTASE-LIKE PROTEIN (SMU.346) FROM STREPTOCOCCUS MUTANS AT 1.70 A RESOLUTION | FMN-DEPENDENT NITROREDUCTASE-LIKE FOLD, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, OXIDOREDUCTASE
3gbr:A (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYL-TRANSFERASE (TRPD) DOUBLE MUTANT D83G F149S FROM S. SOLFATARICUS | TRANSFERASE, AMINO-ACID BIOSYNTHESIS, AROMATIC AMINO ACID BIOSYNTHESIS, GLYCOSYLTRANSFERASE, TRYPTOPHAN BIOSYNTHESIS
3gbr:B (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYL-TRANSFERASE (TRPD) DOUBLE MUTANT D83G F149S FROM S. SOLFATARICUS | TRANSFERASE, AMINO-ACID BIOSYNTHESIS, AROMATIC AMINO ACID BIOSYNTHESIS, GLYCOSYLTRANSFERASE, TRYPTOPHAN BIOSYNTHESIS
4iuw:A (ASP144) to (ASP207) CRYSTAL STRUCTURE OF PEPO FROM LACTOBACILLUS RHAMNOSIS HN001 (DR20) | NEUTRAL PEPTIDASE, ZN METALLOPEPTIDASE, ENDOPEPTIDASE, HYDROLASE
1pp1:X (MSE235) to (ARG287) CRYSTAL STRUCTURE OF THE BORNA DISEASE VIRUS NUCLEOPROTEIN | RNA VIRUS NUCLEOPROTEIN TETRAMER, VIRAL PROTEIN
1ppv:A (LEU144) to (THR179) ISOPENTENYLPYROPHOSPHATE-DIMETHYLALLYLPYROPHOSPHATE ISOMERASE IN COMPLEX WITH THE BROMOHYDRINE OF IPP | COMPLEX, ISOMERASE
1ppw:A (ALA145) to (THR179) ISOPENTENYLPYROPHOSPHATE-DIMETHYLALLYLPYROPHOSPHATE ISOMERASE IN COMPLEX WITH THE BROMOHYDRINE OF IPP | COMPLEX, ISOMERASE
3t8m:A (SER1003) to (GLY1079) RATIONAL DESIGN OF PI3K-ALPHA INHIBITORS THAT EXHIBIT SELECTIVITY OVER THE PI3K-BETA ISOFORM | KINASE P110, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4iym:B (PRO60) to (LYS118) CRYSTAL STRUCTURE OF PUTATIVE METHYLMALONATE-SEMIALDEHYDE DEHYDROGENASE FROM SINORHIZOBIUM MELILOTI 1021 COMPLEXED WITH NAD, TARGET 011934 | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, OXIDOREDUCTASE
4iym:J (PRO60) to (LYS118) CRYSTAL STRUCTURE OF PUTATIVE METHYLMALONATE-SEMIALDEHYDE DEHYDROGENASE FROM SINORHIZOBIUM MELILOTI 1021 COMPLEXED WITH NAD, TARGET 011934 | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, OXIDOREDUCTASE
4iym:O (PRO60) to (LYS118) CRYSTAL STRUCTURE OF PUTATIVE METHYLMALONATE-SEMIALDEHYDE DEHYDROGENASE FROM SINORHIZOBIUM MELILOTI 1021 COMPLEXED WITH NAD, TARGET 011934 | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, OXIDOREDUCTASE
4y06:A (LEU281) to (GLY366) CRYSTAL STRUCTURE OF THE DAP BII (G675R) DIPEPTIDE COMPLEX | HYDROLASE
4y06:B (LEU281) to (GLN365) CRYSTAL STRUCTURE OF THE DAP BII (G675R) DIPEPTIDE COMPLEX | HYDROLASE
1pvf:B (LEU144) to (THR179) E.COLI IPP ISOMERASE IN COMPLEX WITH DIPHOSPHATE | IPP ISOMERASE
4j6i:A (SER1003) to (LYS1078) DISCOVERY OF THIAZOLOBENZOXEPIN PI3-KINASE INHIBITORS THAT SPARE THE PI3-KINASE BETA ISOFORM | BETA-SPARING, SBDD, CATALYTIC SUBUNIT GAMMA, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1e7v:A (SER1003) to (GLY1079) STRUCTURE DETERMINANTS OF PHOSPHOINOSITIDE 3-KINASE INHIBITION BY WORTMANNIN, LY294002, QUERCETIN, MYRICETIN AND STAUROSPORINE | TRANSFERASE, SECONDARY MESSENGER GENERATION PI3K, PI 3K, LY294002
1e8w:A (SER1003) to (GLY1079) STRUCTURE DETERMINANTS OF PHOSPHOINOSITIDE 3-KINASE INHIBITION BY WORTMANNIN, LY294002, QUERCETIN, MYRICETIN AND STAUROSPORINE | PHOSPHOINOSITIDE 3-KINASE GAMMA, SECONDARY MESSENGER GENERATION, PI3K, PI 3K, QUERCETIN
1e8x:A (HIS1005) to (GLY1079) STRUCTURAL INSIGHTS INTO PHOSHOINOSITIDE 3-KINASE ENZYMATIC MECHANISM AND SIGNALLING | PHOSPHOINOSITIDE 3-KINASE GAMMA, SECONDARY MESSENGER GENERATION, PI3K, PI 3K
1e8y:A (SER1003) to (GLY1079) STRUCTURE DETERMINANTS OF PHOSPHOINOSITIDE 3-KINASE INHIBITION BY WORTMANNIN, LY294002, QUERCETIN, MYRICETIN AND STAUROSPORINE | PHOSPHOINOSITIDE 3-KINASE GAMMA, SECONDARY MESSENGER GENERATION, PI3K, PI 3K
4y86:A (PHE254) to (LEU294) CRYSTAL STRUCTURE OF PDE9 IN COMPLEX WITH RACEMIC INHIBITOR C33 | PHOSPHODIESTERASE 9A, INHIBITOR SELECTIVITY POCKET, PHARMACOKINETICS, ENANTIOMERIC DIFFERENTIATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4y86:B (PHE254) to (LEU294) CRYSTAL STRUCTURE OF PDE9 IN COMPLEX WITH RACEMIC INHIBITOR C33 | PHOSPHODIESTERASE 9A, INHIBITOR SELECTIVITY POCKET, PHARMACOKINETICS, ENANTIOMERIC DIFFERENTIATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4y8c:A (PHE254) to (LEU294) CRYSTAL STRUCTURE OF PHOSPHODIESTERASE 9 IN COMPLEX WITH (S)-C33 | PHOSPHODIESTERASE 9A, INHIBITOR SELECTIVITY POCKET, PHARMACOKINETICS, ENANTIOMERIC DIFFERENTIATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2dq0:B (ASP3) to (LEU106) CRYSTAL STRUCTURE OF SERYL-TRNA SYNTHETASE FROM PYROCOCCUS HORIKOSHII COMPLEXED WITH A SERYL-ADENYLATE ANALOG | COILED-COIL, HOMODIMER, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, LIGASE
1q80:A (SER1) to (PRO86) SOLUTION STRUCTURE AND DYNAMICS OF NEREIS SARCOPLASMIC CALCIUM BINDING PROTEIN | ALL-ALPHA, METAL BINDING PROTEIN
2r9s:A (ALA231) to (VAL298) C-JUN N-TERMINAL KINASE 3 WITH 3,5-DISUBSTITUTED QUINOLINE INHIBITOR | JNK3, SIGNALING PROTEIN, TRANSFERASE
2rd0:A (THR974) to (ALA1046) STRUCTURE OF A HUMAN P110ALPHA/P85ALPHA COMPLEX | DISEASE MUTATION, KINASE, ONCOGENE, TRANSFERASE, HOST-VIRUS INTERACTION, PHOSPHORYLATION, SH2 DOMAIN, SH3 DOMAIN, TRANSFERASE- ONCOPROTEIN COMPLEX
3tuv:A (LYS656) to (SER721) CRYSTAL STRUCTURE OF INSULYSIN WITH BOUND ATP | THERMOLYSIN-LIKE FOLD ACTIVE SITE REGION, HYDROLYASE, PEPTIDASE, HYDROLASE
4jps:A (ARG975) to (HIS1048) CO-CRYSTAL STRUCTURES OF THE LIPID KINASE PI3K ALPHA WITH PAN AND ISOFORM SELECTIVE INHIBITORS | CLASS I PHOSPHATIDYLINOSITOL 3-KINASES, P85 ALPHA, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3h44:B (ASP655) to (SER721) CRYSTAL STRUCTURE OF INSULIN DEGRADING ENZYME IN COMPLEX WITH MACROPHAGE INFLAMMATORY PROTEIN 1 ALPHA | IDE, MIP1ALPHA, CYTOPLASM, HYDROLASE, METAL-BINDING, METALLOPROTEASE, POLYMORPHISM, PROTEASE, ZINC, CHEMOTAXIS, CYTOKINE, DISULFIDE BOND, INFLAMMATORY RESPONSE, SECRETED, HYDROLASE-CYTOKINE COMPLEX
3twp:A (ASP293) to (ILE370) CRYSTAL STRUCTURE OF M. TUBERCULOSIS TRPD IN COMPLEX WITH AN INHIBITOR | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, TRANSFERASE, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3twp:B (ASP293) to (ILE370) CRYSTAL STRUCTURE OF M. TUBERCULOSIS TRPD IN COMPLEX WITH AN INHIBITOR | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, TRANSFERASE, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3twp:C (ASP293) to (ILE370) CRYSTAL STRUCTURE OF M. TUBERCULOSIS TRPD IN COMPLEX WITH AN INHIBITOR | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, TRANSFERASE, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3twp:D (ASP293) to (ILE370) CRYSTAL STRUCTURE OF M. TUBERCULOSIS TRPD IN COMPLEX WITH AN INHIBITOR | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, TRANSFERASE, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ykn:A (ARG1975) to (HIS2047) PI3K ALPHA LIPID KINASE WITH ACTIVE SITE INHIBITOR | "LIPID KINASE", INHIBITOR, COMPLEX, PI3K, PI3K ALPHA, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4jt6:B (ARG2397) to (THR2533) STRUCTURE OF MTORDELTAN-MLST8-PI-103 COMPLEX | KINASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3hgz:B (ASP655) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME IN COMPLEX WITH AMYLIN | INSULIN DEGRADING ENZYME, IDE, AMYLIN, CYSTEIN FREE, CYTOPLASM, HYDROLASE, METAL-BINDING, METALLOPROTEASE, POLYMORPHISM, PROTEASE, ZINC, AMIDATION, AMYLOID, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISULFIDE BOND, HORMONE, SECRETED
2elc:A (GLY259) to (ALA329) CRYSTAL STRUCTURE OF TTHA1842 FROM THERMUS THERMOPHILUS HB8 | TRANSFERASE, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
2elc:D (GLY259) to (ARG328) CRYSTAL STRUCTURE OF TTHA1842 FROM THERMUS THERMOPHILUS HB8 | TRANSFERASE, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
3hiz:A (THR974) to (MET1043) CRYSTAL STRUCTURE OF P110ALPHA H1047R MUTANT IN COMPLEX WITH NISH2 OF P85ALPHA | P110, P85, PI3KCA, PI3K, PIK3R1, PHOSPHATIDILYNOSITOL 3,4,5- TRIPHOSPHATE, H1047R, ATP-BINDING, DISEASE MUTATION, KINASE, NUCLEOTIDE-BINDING, ONCOGENE, POLYMORPHISM, TRANSFERASE, ALTERNATIVE SPLICING, HOST-VIRUS INTERACTION, PHOSPHOPROTEIN, SH2 DOMAIN, SH3 DOMAIN, UBL CONJUGATION, TRANSFERASE/ONCOPROTEIN COMPLEX
2v4l:A (SER1003) to (LYS1078) COMPLEX OF HUMAN PHOSPHOINOSITIDE 3-KINASE CATALYTIC SUBUNIT GAMMA (P110 GAMMA) WITH PIK-284 | TRANSFERASE, LIPID KINASE, PHOSPHOINOSITIDE, PYRAZOLOPYRIMIDINE, S1, KINASE, PIK-284, 3-KINASE, INHIBITOR, SIGNALING
2van:A (THR121) to (LYS148) NUCLEOTIDYL TRANSFER MECHANISM OF MISMATCHED DNTP INCORPORATION BY DNA POLYMERASE B BY STRUCTURAL AND KINETIC ANALYSES | NUCLEOTIDYLTRANSFERASE, DNA-DIRECTED DNA POLYMERASE, LYASE, NUCLEUS, DNA DAMAGE, DNA SYNTHESIS, DNA REPLICATION, DNA REPAIR, TRANSFERASE, DNA-BINDING, METAL-BINDING
4z3n:A (LEU105) to (GLY179) CRYSTAL STRUCTURE OF THE MATE TRANSPORTER CLBM | TRANSPORTER, TRANSPORT PROTEIN
1g73:D (LYS322) to (GLU357) CRYSTAL STRUCTURE OF SMAC BOUND TO XIAP-BIR3 DOMAIN | HELIX BUNDLE, ZINC-BINDING DOMAIN, APOPTOSIS/APOPTOSIS INHIBITOR COMPLEX
4z3p:A (VAL326) to (GLY400) MATE TRANSPORTER CLBM IN COMPLEX WITH RB+ | TRANSPORTER, TRANSPORT PROTEIN
1ryu:A (GLY64) to (GLU109) SOLUTION STRUCTURE OF THE SWI1 ARID | ARID, SWI1, NMR, STRUCTURAL GENOMICS, PROTEIN-DNA INTERACTION, DNA BINDING PROTEIN
3ut2:A (GLY158) to (GLY210) CRYSTAL STRUCTURE OF FUNGAL MAGKATG2 | CATALASE-PEROXIDASE, KATG, FUNGAL, HEME ENZYME, OXIDOREDUCTASE
3uu1:A (ASP293) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS142) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uu1:B (ASP293) to (GLN369) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS142) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uu1:C (ASP293) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS142) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3uu1:D (ASP293) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS142) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4klt:A (THR121) to (LYS148) DNA POLYMERASE BETA MISMATCHED PRODUCT COMPLEX WITH MN2+, 30 MIN | DNA POLYMERASE, TRANSFERASE, LYASE-DNA COMPLEX
1gfz:A (ILE735) to (PRO794) FLAVOPIRIDOL INHIBITS GLYCOGEN PHOSPHORYLASE BY BINDING AT THE INHIBITOR SITE | GLYCOGEN PHOSPHORYLASE, GLYCOGEN METABOLISM, DIABETES, FLAVOPIRIDOL, INHIBITOR SITE, TRANSFERASE
3uxn:A (THR121) to (LYS148) CRYSTAL STRUCTURE OF RAT DNA POLYMERASE BETA, WILD TYPE APOENZYME | DNA POLYMERASE, BASE EXCISION REPAIR, TRANSFERASE
3uxo:A (THR121) to (GLU147) CRYSTAL STRUCTURE OF RAT DNA POLYMERASE BETA MUTATOR I260Q APOENZYME | DNA POLYMERASE BETA, BER, TRANSFERASE, LYASE
3uxp:A (THR121) to (ARG149) CO-CRYSTAL STRUCTURE OF RAT DNA POLYMERASE BETA MUTATOR I260Q: ENZYME- DNA-DDTTP | POL BETA, REPAIR POLYMERASE, BER, TRANSFERASE, LYASE-DNA COMPLEX
2fon:A (GLY547) to (ALA606) X-RAY CRYSTAL STRUCTURE OF LEACX1, AN ACYL-COA OXIDASE FROM LYCOPERSICON ESCULENTUM (TOMATO) | OXIDOREDUCTASE, PEROXISOMAL BETA-OXIDATION, FAD COFACTOR
2fon:B (GLY547) to (ALA606) X-RAY CRYSTAL STRUCTURE OF LEACX1, AN ACYL-COA OXIDASE FROM LYCOPERSICON ESCULENTUM (TOMATO) | OXIDOREDUCTASE, PEROXISOMAL BETA-OXIDATION, FAD COFACTOR
1gk1:C (SER98) to (VAL151) STRUCTURE-BASED PREDICTION OF MODIFICATIONS IN GLUTARYLAMIDASE TO ALLOW SINGLE-STEP ENZYMATIC PRODUCTION OF 7-AMINOCEPHALOSPORANIC ACID FROM CEPHALOSPORIN C | HYDROLASE, CEPHALOSPORIN ACYLASE, GLUTARYL ACYLASE, CEPHALOSPORIN C, CATALYTIC TRIAD, NTN-HYDROLASE, X-RAZ STRUCTURE
3hyq:A (PHE144) to (ASN177) CRYSTAL STRUCTURE OF ISOPENTENYL-DIPHOSPHATE DELTA-ISOMERASE FROM SALMONELLA ENTERICASE | ALPHA-BETA STRUCTURE, ISOMERASE, ISOPRENE BIOSYNTHESIS, MAGNESIUM, MANGANESE, METAL-BINDING, STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID
1set:B (ASP3) to (VAL101) CRYSTAL STRUCTURES AT 2.5 ANGSTROMS RESOLUTION OF SERYL-TRNA SYNTHETASE COMPLEXED WITH TWO DIFFERENT ANALOGUES OF SERYL-ADENYLATE | LIGASE, SYNTHETASE
3v72:A (THR121) to (LYS148) CRYSTAL STRUCTURE OF RAT DNA POLYMERASE BETA MUTATOR E295K: ENZYME- DSDNA | DNA REPAIR POLYMERASE, E295K, MUTATOR, DNA BINDING PROTEIN-DNA COMPLEX
3v7j:A (THR121) to (LYS148) CO-CRYSTAL STRUCTURE OF WILD TYPE RAT POLYMERASE BETA: ENZYME-DNA BINARY COMPLEX | PROTEIN-DNA COMPLEX, REPAIR POLYMERASE, TRANSFERASE-DNA COMPLEX
3v7k:A (THR121) to (LYS148) CO-CRYSTAL STRUCTURE OF K72E VARIANT OF RAT POLYMERASE BETA: ENZYME- DNA BINARY COMPLEX | PROTEIN-DNA COMPLEX, REPAIR POLYMERASE, TRANSFERASE-DNA COMPLEX
3i1y:A (GLY391) to (MET469) CRYSTAL STRUCTURE OF SOLUBLE EPOXIDE HYDROLASE | HYDROLASE, AROMATIC HYDROCARBONS CATABOLISM, CYTOPLASM, DETOXIFICATION, MAGNESIUM, METAL-BINDING, PEROXISOME, POLYMORPHISM
3v94:H (ALA370) to (VAL411) TCRPDEC1 CATALYTIC DOMAIN IN COMPLEX WITH INHIBITOR WYQ16 | TRYPANOSOMA PDE PARASITE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2g48:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME IN COMPLEX WITH AMYLIN | PROTEIN-PEPTIDE COMPLEX, HYDROLASE
2g49:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME IN COMPLEX WITH GLUCAGON | PROTEIN-PEPTIDE COMPLEX, HYDROLASE
2g54:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF ZN-BOUND HUMAN INSULIN-DEGRADING ENZYME IN COMPLEX WITH INSULIN B CHAIN | PROTEIN-PEPTIDE COMPLEX, HYDROLASE
2g56:A (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME IN COMPLEX WITH INSULIN B CHAIN | PROTEIN-PEPTIDE COMPLEX, HYDROLASE
2g56:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME IN COMPLEX WITH INSULIN B CHAIN | PROTEIN-PEPTIDE COMPLEX, HYDROLASE
2g73:B (LEU144) to (THR179) Y104F MUTANT TYPE 1 IPP ISOMERASE COMPLEX WITH EIPP | COMPLEX, ISOMERASE
1sry:A (ASP3) to (VAL101) REFINED CRYSTAL STRUCTURE OF THE SERYL-TRNA SYNTHETASE FROM THERMUS THERMOPHILUS AT 2.5 ANGSTROMS RESOLUTION | LIGASE(SYNTHETASE)
1sry:B (ASP3) to (VAL101) REFINED CRYSTAL STRUCTURE OF THE SERYL-TRNA SYNTHETASE FROM THERMUS THERMOPHILUS AT 2.5 ANGSTROMS RESOLUTION | LIGASE(SYNTHETASE)
4kz0:A (HIS1005) to (LYS1078) STRUCTURE OF PI3K GAMMA WITH IMIDAZOPYRIDINE INHIBITORS | LIPID KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4kzc:A (SER1003) to (GLY1079) STRUCTURE OF PI3K GAMMA WITH IMIDAZOPYRIDINE INHIBITORS | LIPID KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4l23:A (THR974) to (HIS1047) CRYSTAL STRUCTURE OF P110ALPHA COMPLEXED WITH NISH2 OF P85ALPHA AND PI-103 | ATP BINDING, PI-103, SIGNALING PROTEIN-TRANSFERASE-INHIBITOR COMPLEX
4l2o:A (LEU22) to (ALA82) CRYSTAL STRUCTURE OF HUMAN ALDH3A1 WITH ITS SELECTIVE INHIBITOR 1-(4- FLUOROPHENYL)SULFONYL-2-METHYLBENZIMIDAZOLE | CATALYZES BENZALDEHYDE, ROSSMANN FOLD, DEHYDROGENASE, NADP+ BINDING, OXIDOREDUCTASE-INHIBITOR COMPLEX
4l2o:B (LEU22) to (ALA82) CRYSTAL STRUCTURE OF HUMAN ALDH3A1 WITH ITS SELECTIVE INHIBITOR 1-(4- FLUOROPHENYL)SULFONYL-2-METHYLBENZIMIDAZOLE | CATALYZES BENZALDEHYDE, ROSSMANN FOLD, DEHYDROGENASE, NADP+ BINDING, OXIDOREDUCTASE-INHIBITOR COMPLEX
4l2o:E (LEU22) to (ALA82) CRYSTAL STRUCTURE OF HUMAN ALDH3A1 WITH ITS SELECTIVE INHIBITOR 1-(4- FLUOROPHENYL)SULFONYL-2-METHYLBENZIMIDAZOLE | CATALYZES BENZALDEHYDE, ROSSMANN FOLD, DEHYDROGENASE, NADP+ BINDING, OXIDOREDUCTASE-INHIBITOR COMPLEX
4l2o:G (LEU22) to (ALA82) CRYSTAL STRUCTURE OF HUMAN ALDH3A1 WITH ITS SELECTIVE INHIBITOR 1-(4- FLUOROPHENYL)SULFONYL-2-METHYLBENZIMIDAZOLE | CATALYZES BENZALDEHYDE, ROSSMANN FOLD, DEHYDROGENASE, NADP+ BINDING, OXIDOREDUCTASE-INHIBITOR COMPLEX
1t33:B (VAL116) to (THR190) STRUCTURAL GENOMICS, THE CRYSTAL STRUCTURE OF A PUTATIVE TRANSCRIPTIONAL REPRESSOR (TETR/ACRR FAMILY) FROM SALMONELLA TYPHIMURIM LT2 | STRUCTURAL GENOMICS, TRANSCRIPTIONAL REPRESSOR, TETR/CCRR FAMILY, HELIX TURN HELIX DNA BINDING DOMAIN, PSI, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSCRIPTION
4l2y:A (THR974) to (HIS1048) CRYSTAL STRUCTURE OF P110ALPHA COMPLEXED WITH NISH2 OF P85ALPHA AND COMPOUND 9D | ATP BINDING, SIGNALING PROTEIN-TRANSFERASE-INHIBITOR COMPLEX
3ibe:A (SER1003) to (LYS1078) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR BOUND TO PI3 KINASE GAMMA | PI3KINASE INHIBITOR, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, TRANSFERASE
4zof:A (ASP293) to (GLN369) LOBENZARIT-LIKE INHIBITOR BOUND IN THE ACTIVE SITE OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | INHIBITOR, COMPLEX, LOBENZARIT-LIKE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYLPYROPHOSPHATE, PRPP, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4zof:B (ASP293) to (GLN369) LOBENZARIT-LIKE INHIBITOR BOUND IN THE ACTIVE SITE OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | INHIBITOR, COMPLEX, LOBENZARIT-LIKE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYLPYROPHOSPHATE, PRPP, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4zoj:A (ALA294) to (GLN369) METHYLSULFANYL-CONTAINING INHIBITOR BOUND IN THE ACTIVE SITE OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | INHIBITOR, COMPLEX, LOBENZARIT-LIKE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYLPYROPHOSPHATE, PRPP, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4zoj:B (ASP293) to (GLN369) METHYLSULFANYL-CONTAINING INHIBITOR BOUND IN THE ACTIVE SITE OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | INHIBITOR, COMPLEX, LOBENZARIT-LIKE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYLPYROPHOSPHATE, PRPP, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4zok:A (ALA294) to (GLN369) METHYLSULFONYL-CONTAINING INHIBITOR BOUND IN THE SUBSTRATE CAPTURE SITE OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | INHIBITOR, COMPLEX, LOBENZARIT-LIKE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYLPYROPHOSPHATE, PRPP, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ih7:A (SER183) to (SER231) CRYSTAL STRUCTURE OF CATALYTICALLY ACTIVE HUMAN 8-OXOGUANINE GLYCOSYLASE DISTALLY CROSSLINKED TO GUANINE-CONTAINING DNA | DISULFIDE CROSSLINK, DNA GLYCOSYLASE, UNDAMAGED DNA, (HYDROLASE, LYASE)-DNA COMPLEX, DNA DAMAGE, DNA REPAIR, GLYCOSIDASE, HYDROLASE, LYASE, MITOCHONDRION, MULTIFUNCTIONAL ENZYME, NUCLEUS
4zop:A (ARG975) to (HIS1048) CO-CRYSTAL STRUCTURE OF LIPID KINASE PI3K ALPHA WITH A SELECTIVE PHOSPHATIDYLINOSITOL-3 KINASE ALPHA INHIBITOR | LIPID KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1h8b:A (ASP5) to (GLY69) EF-HANDS 3,4 FROM ALPHA-ACTININ / Z-REPEAT 7 FROM TITIN | STRUCTURAL PROTEIN, Z-DISK STRUCTURAL COMPLEX
1tah:A (SER117) to (ASN178) THE CRYSTAL STRUCTURE OF TRIACYLGLYCEROL LIPASE FROM PSEUDOMONAS GLUMAE REVEALS A PARTIALLY REDUNDANT CATALYTIC ASPARTATE | HYDROLASE(CARBOXYLIC ESTERASE)
4ztv:A (GLN295) to (ILE370) NON-ANTHRANILATE-LIKE INHIBITOR (TAMU-A7) COMPLEXED WITH ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS IN ABSENCE OF PRPP | NON-ANTHRANILATE-LIKE INHIBITOR, TRPD, ANPRT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
4ztv:B (ALA294) to (GLN369) NON-ANTHRANILATE-LIKE INHIBITOR (TAMU-A7) COMPLEXED WITH ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS IN ABSENCE OF PRPP | NON-ANTHRANILATE-LIKE INHIBITOR, TRPD, ANPRT, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
1he8:A (SER1003) to (GLY1079) RAS G12V - PI 3-KINASE GAMMA COMPLEX | KINASE/HYDROLASE, COMPLEX (PHOSPHOINOSITIDE KINASE/RAS), PHOSPHOINOSITIDE 3-KINASE GAMMA - H-RAS G12V COMPLEX, PHOSPHATIDYLINOSITOL 3-KINASE, PI3K, PI 3-K, PI 3-KINASE, SECOND MESSENGER GENERATION, RAS EFFECTOR, H-RAS G12V, ONCOGENE PROTEIN, GMPPNP, GTP, RAS-BINDING DOMAIN, HEAT DOMAIN
2h1j:A (GLU81) to (SER147) 3.1 A X-RAY STRUCTURE OF PUTATIVE OLIGOENDOPEPTIDASE F: CRYSTALS GROWN BY MICROFLUIDIC SEEDING | STRUCTURAL GENOMICS, MICROFLUIDIC SEEDING, PSI-2, PROTEIN STRUCTURE INITIATIVE, ACCELERATED TECHNOLOGIES CENTER FOR GENE TO 3D STRUCTURE, ATCG3D, HYDROLASE
2h1n:A (ASP67) to (SER147) 3.0 A X-RAY STRUCTURE OF PUTATIVE OLIGOENDOPEPTIDASE F: CRYSTALS GROWN BY VAPOR DIFFUSION TECHNIQUE | STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, PSI, HYDROLASE
3ir6:C (PRO82) to (GLY153) CRYSTAL STRUCTURE OF NARGHI MUTANT NARG-H49S | OXIDOREDUCTASE, NITRATE REDUCTASE, ELECTRON TRANSFER, MEMBRANE PROTEIN, 4FE-4S, CELL MEMBRANE, ELECTRON TRANSPORT, IRON, IRON-SULFUR, MEMBRANE, METAL-BINDING, MOLYBDENUM, NITRATE ASSIMILATION, TRANSPORT, 3FE-4S, CELL INNER MEMBRANE, FORMYLATION, HEME, TRANSMEMBRANE
3isd:A (THR121) to (LYS148) TERNARY COMPLEX OF HUMAN DNA POLYMERASE BETA WITH AN ABASIC SITE (THF): DAPCPP MISMATCH | NUCLEOTIDYL TRANSFERASE, DNA POLYMERASE BETA, ABASIC SITE, TETRAHYDROFURAN, TERNARY COMPLEX, GAPPED DNA, 'A-RULE', DNA DAMAGE, DNA REPAIR, DNA REPLICATION, DNA SYNTHESIS, DNA- BINDING, DNA-DIRECTED DNA POLYMERASE, LYASE, MAGNESIUM, METAL-BINDING, METHYLATION, NUCLEOTIDYLTRANSFERASE, NUCLEUS, POLYMORPHISM, SODIUM, TRANSFERASE, TRANSFERASE/DNA COMPLEX
2wby:B (ASP655) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME IN COMPLEX WITH INSULIN | HYDROLASE/HORMONE, GLUCOSE METABOLISM, CARBOHYDRATE METABOLISM, DISEASE MUTATION, DIABETES MELLITUS, ZINC, DIOXANE, INSULIN, HORMONE, SECRETED, PROTEASE, DISULFIDE BOND, PHARMACEUTICAL, METALLOPROTEASE, HUMAN INSULIN-DEGRADNG ENZYME, HYDROLASE, CYTOPLASM, POLYMORPHISM, METAL-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES
2wc0:B (ASP655) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN DEGRADING ENZYME IN COMPLEX WITH IODINATED INSULIN | HYDROLASE/HORMONE, ZINC, DIOXANE, INSULIN, HORMONE, PROTEASE, SECRETED, HUMAN INSULIN-DEGRADING ENZYME, DISULFIDE BOND, METALLOPROTEASE, GLUCOSE METABOLISM, CARBOHYDRATE METABOLISM, HYDROLASE, CYTOPLASM, POLYMORPHISM, METAL-BINDING, CLEAVAGE ON PAIR OF BASIC RESIDUES
2hne:B (LEU132) to (GLY184) CRYSTAL STRUCTURE OF L-FUCONATE DEHYDRATASE FROM XANTHOMONAS CAMPESTRIS PV. CAMPESTRIS STR. ATCC 33913 | STRUCTURAL GENOMICS, L-FUCONATE DEHYDRATASE, ENOLASE SUPERFAMILY, NYSGXRC TARGET T2188, PSI, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, UNKNOWN FUNCTION
2wk3:A (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME IN COMPLEX WITH AMYLOID-BETA (1-42) | POLYMORPHISM, METAL-BINDING, METALLOPROTEASE, IDE, ZINC, PROTEASE, HYDROLASE, CYTOPLASM, AMYLOID-BETA (1-42)
2wk3:B (ASP655) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME IN COMPLEX WITH AMYLOID-BETA (1-42) | POLYMORPHISM, METAL-BINDING, METALLOPROTEASE, IDE, ZINC, PROTEASE, HYDROLASE, CYTOPLASM, AMYLOID-BETA (1-42)
3vvr:A (LYS315) to (GLY390) CRYSTAL STRUCTURE OF MATE IN COMPLEX WITH MAD5 | MATE, MULTIDRUG TRANSPORTER, MACROCYCLIC PEPTIDE, TRANSPORT PROTEIN, TRANSPORT PROTEIN-INHIBITOR COMPLEX
4lrz:A (ARG5) to (ASP60) CRYSTAL STRUCTURE OF THE E.COLI DHAR(N)-DHAL COMPLEX | COILED-COIL, HELIX ROTATION, GAF, PAS, TRANSCRIPTIONAL REGULATION COMPLEX, TRANSFERASE-TRANSCRIPTION REGULATOR COMPLEX
4lrz:C (THR6) to (ASP60) CRYSTAL STRUCTURE OF THE E.COLI DHAR(N)-DHAL COMPLEX | COILED-COIL, HELIX ROTATION, GAF, PAS, TRANSCRIPTIONAL REGULATION COMPLEX, TRANSFERASE-TRANSCRIPTION REGULATOR COMPLEX
3vz0:B (SER45) to (ALA105) STRUCTURAL INSIGHTS INTO COFACTOR AND SUBSTRATE SELECTION BY GOX0499 | GOX0499, SUBSTRATE SELECTION, COFACTOR PREFERENCE, OXIDOREDUCTASE
4lte:A (GLU656) to (SER721) STRUCTURE OF CYSTEINE-FREE HUMAN INSULIN DEGRADING ENZYME IN COMPLEX WITH MACROCYCLIC INHIBITOR | HYDROLASE, METAL-BINDING, METALLOPROTEASE, PROTEASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4lte:B (GLU656) to (SER721) STRUCTURE OF CYSTEINE-FREE HUMAN INSULIN DEGRADING ENZYME IN COMPLEX WITH MACROCYCLIC INHIBITOR | HYDROLASE, METAL-BINDING, METALLOPROTEASE, PROTEASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1i9a:A (LEU144) to (PHE178) STRUCTURAL STUDIES OF CHOLESTEROL BIOSYNTHESIS: MEVALONATE 5-DIPHOSPHATE DECARBOXYLASE AND ISOPENTENYL DIPHOSPHATE ISOMERASE | ALPHA/BETA PROTEIN, ISOMERASE, MN2+, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
4m0r:B (ALA294) to (GLN369) TRIANTHRANILATE-LIKE ANALOGUE BOUND TO ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD). | MAGNESIUM BINDING, PHOSPHORIBOSYLPYROPHOSPHATE, PRPP, INHIBITOR COMPLEX, TRI-ANTHRANILATE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2wxf:A (ASN949) to (SER1026) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH PIK-39. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
2wxi:A (GLU951) to (SER1026) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH SW30. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
2wxm:A (GLU951) to (SER1026) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH DL06. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
2wxn:A (GLU951) to (ARG1024) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH DL07. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
2wxp:A (GLU951) to (SER1026) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH GDC-0941. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
3w9u:A (ILE111) to (TYR172) CRYSTAL STRUCTURE OF LIPK107 | LIPASE, HYDROLASE
2wxq:A (GLU951) to (GLU1025) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH AS15. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
2wxr:A (GLU951) to (SER1026) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
1is2:A (LYS549) to (ALA609) CRYSTAL STRUCTURE OF PEROXISOMAL ACYL-COA OXIDASE-II FROM RAT LIVER | OXIDOREDUCTASE, FAD
4m9h:A (THR121) to (LYS148) DNA POLYMERASE BETA E295K SOAKED WITH DTTP | DNA POLYMERASE, LYASE, DNA COMPLEX, TRANSFERASE-DNA COMPLEX
4m9j:A (THR121) to (LYS148) DNA POLYMERASE BETA E295K SOAKED WITH DUMPNPP | DNA POLYMERASE, LYASE, DNA COMPLEX, TRANSFERASE-DNA COMPLEX
4m9l:A (THR121) to (LYS148) DNA POLYMERASE BETA E295K SOAKED WITH DCTP | DNA POLYMERASE, LYASE, DNA COMPLEX, TRANSFERASE-DNA COMPLEX
4m9n:A (THR121) to (LYS148) DNA POLYMERASE BETA E295K SOAKED WITH DATP | DNA POLYMERASE, LYASE, DNA COMPLEX, TRANSFERASE-DNA COMPLEX
5ac2:A (SER83) to (GLN141) HUMAN ALDEHYDE DEHYDROGENASE 1A1 WITH DUOCARMYCIN ANALOG | OXIDOREDUCTASE, OXIDATION-REDUCTION PROCESS, ALDEHYDE DEHYDROGENASE ACTIVITY
4mdz:A (ASP321) to (ARG357) METALLO-ENZYME FROM P. MARINA | STRUCTURAL GENOMICS, OXFORD PROTEIN PRODUCTION FACILITY, OPPF, PHOSPHOHYDROLASE, HYDROLASE
4mdz:B (MET322) to (ARG360) METALLO-ENZYME FROM P. MARINA | STRUCTURAL GENOMICS, OXFORD PROTEIN PRODUCTION FACILITY, OPPF, PHOSPHOHYDROLASE, HYDROLASE
5ae8:A (ASN949) to (ASN1032) CRYSTAL STRUCTURE OF MOUSE PI3 KINASE DELTA IN COMPLEX WITH GSK2269557 | TRANSFERASE, PI3 KINASE DELTA
1uxp:A (GLY76) to (LYS131) STRUCTURAL BASIS FOR ALLOSTERIC REGULATION AND SUBSTRATE SPECIFICITY OF THE NON-PHOSPHORYLATING GLYCERALDEHYDE-3-PHOSPHATE DEHYDROGENASE (GAPN) FROM THERMOPROTEUS TENAX | OXIDOREDUCTASE, GAPN, ALDH, ADP, GLYCOLYSIS, REGULATION, CATALYSIS OXIDOREDUCTASE
1uxr:A (GLY76) to (LYS132) STRUCTURAL BASIS FOR ALLOSTERIC REGULATION AND SUBSTRATE SPECIFICITY OF THE NON-PHOSPHORYLATING GLYCERALDEHYDE-3-PHOSPHATE DEHYDROGENASE (GAPN) FROM THERMOPROTEUS TENAX | GAPN, ALDH, FRUCTOSE 6-PHOSPHATE, GLYCOLYSIS, REGULATION, CATALYSIS, OXIDOREDUCTASE
4mf2:A (THR121) to (LYS148) STRUCTURE OF HUMAN DNA POLYMERASE BETA COMPLEXED WITH O6MG AS THE TEMPLATE BASE IN A 1-NUCLEOTIDE GAPPED DNA | PROTEIN-DNA COMPLEX, POLYMERASE X FAMILY, DNA POLYMERASE, TRANSFERASE-DNA COMPLEX
4mf8:A (LEU122) to (LYS148) STRUCTURE OF HUMAN DNA POLYMERASE BETA COMPLEXED WITH NICKED DNA CONTAINING A MISMATCHED TEMPLATE O6MG AND INCOMING CTP | DNA POLYMERASE X FAMILY, DNA SYNTHESIS, TRANSFERASE-DNA COMPLEX
2x6f:A (SER854) to (MET933) THE CRYSTAL STRUCTURE OF THE DROSOPHILA CLASS III PI3-KINASE VPS34 IN COMPLEX WITH 3-METHYLADENINE | TRANSFERASE
2x6h:A (HIS856) to (MET933) THE CRYSTAL STRUCTURE OF THE DROSOPHILA CLASS III PI3-KINASE VPS34 | TRANSFERASE
2x6j:A (HIS856) to (MET933) THE CRYSTAL STRUCTURE OF THE DROSOPHILA CLASS III PI3-KINASE VPS34 IN COMPLEX WITH PIK-93 | TRANSFERASE
2x6k:A (SER854) to (MET933) THE CRYSTAL STRUCTURE OF THE DROSOPHILA CLASS III PI3-KINASE VPS34 IN COMPLEX WITH PI-103 | PI103, PI-103, AUTOPHAGY, TRANSFERASE, PI3K CLASS III, PHOSPHOINOSITIDE 3-KINASE CLASS III
5akg:A (GLY391) to (MET469) LIGAND COMPLEX STRUCTURE OF SOLUBLE EPOXIDE HYDROLASE | HYDROLASE
5am4:A (GLY391) to (ASN468) LIGAND COMPLEX STRUCTURE OF SOLUBLE EPOXIDE HYDROLASE | HYDROLASE
1jba:A (LYS96) to (ARG175) UNMYRISTOYLATED GCAP-2 WITH THREE CALCIUM IONS BOUND | EF-HAND, CALCIUM-BINDING PROTEIN, GUANYLYL CYCLASE REGULATION, LYASE
1v8g:B (GLY259) to (ARG328) CRYSTAL STRUCTURE OF ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM THERMUS THERMOPHILUS HB8 | TRYPTOPHAN BIOSYNTHESIS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, STRUCTURAL GENOMICS, TRANSFERASE
3woi:A (LEU281) to (GLY364) CRYSTAL STRUCTURE OF THE DAP BII (S657A) | CHYMOTRYPSIN FOLD, S46 PEPTIDASE, HYDROLASE
3wok:B (LEU281) to (GLN365) CRYSTAL STRUCTURE OF THE DAP BII (SPACE) | CHYMOTRYPSIN FOLD, S46 PEPTIDASE, HYDROLASE
5an4:A (SER183) to (SER231) CRYSTAL STRUCTURE OF THE HUMAN 8-OXOGUANINE GLYCOSYLASE (OGG1) PROCESSED WITH THE CRYSTALDIRECT AUTOMATED MOUNTING AND CRYO-COOLING TECHNOLOGY | HYDROLASE, ALLERGEN, PYR/PYL/RCAR, BET V 1, FLAVONOIDS, AUTOMATED CRYSTAL HARVESTING, AUTOMATED CRYO-COOLING, CRYSTALDIRECT
3wop:B (ALA282) to (GLY366) CRYSTAL STRUCTURE OF THE DAP BII HEXAPEPTIDE COMPLEX II | CHYMOTRYPSIN FOLD, S46 PEPTIDASE, HYDROLASE-HORMONE COMPLEX
3woq:B (ALA282) to (GLY366) CRYSTAL STRUCTURE OF THE DAP BII HEXAPEPTIDE COMPLEX III | CHYMOTRYPSIN FOLD, S46 PEPTIDASE, HYDROLASE-HORMONE COMPLEX
2xeq:D (PRO516) to (CYS589) HUMAN PATL1 C-TERMINAL DOMAIN | MRNA DECAPPING, P-BODIES, RNA BINDING PROTEIN
1vj5:A (GLY389) to (ASN467) HUMAN SOLUBLE EPOXIDE HYDROLASE- N-CYCLOHEXYL-N'-(4- IODOPHENYL)UREA COMPLEX | DOMAIN-SWAPPED DIMER, HYDROLASE
2xhi:A (SER183) to (SER231) SEPARATION-OF-FUNCTION MUTANTS UNRAVEL THE DUAL REACTION MODE OF HUMAN 8-OXOGUANINE DNA GLYCOSYLASE | LYASE-DNA COMPLEX, LYASE/DNA COMPLEX, SEPARATION-OF-FUNCTION MUTANT, HELIX-HAIRPIN-HELIX, DNA REPAIR
1vqu:A (ASP290) to (ASN362) CRYSTAL STRUCTURE OF ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE 2 (17130499) FROM NOSTOC SP. AT 1.85 A RESOLUTION | 17130499, ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE 2, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI, TRANSFERASE
1vqu:B (ASP290) to (GLY361) CRYSTAL STRUCTURE OF ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE 2 (17130499) FROM NOSTOC SP. AT 1.85 A RESOLUTION | 17130499, ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE 2, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI, TRANSFERASE
2jbu:A (ASP655) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN DEGRADING ENZYME COMPLEXED WITH CO-PURIFIED PEPTIDES. | METAL-BINDING, METALLOPROTEASE, ZINC, PROTEASE, HYDROLASE, ENZYME ASSAY, INSULIN DEGRADING ENZYME
2jbu:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN DEGRADING ENZYME COMPLEXED WITH CO-PURIFIED PEPTIDES. | METAL-BINDING, METALLOPROTEASE, ZINC, PROTEASE, HYDROLASE, ENZYME ASSAY, INSULIN DEGRADING ENZYME
5b6b:A (ASN143) to (LEU211) COMPLEX OF LATS1 AND PHOSPHOMIMETIC MOB1B | MOB1 LATS1 HIPPO PATHWAY, METAL BINDING PROTEIN-SIGNALING PROTEIN COMPLEX
5b6b:B (MET145) to (LEU211) COMPLEX OF LATS1 AND PHOSPHOMIMETIC MOB1B | MOB1 LATS1 HIPPO PATHWAY, METAL BINDING PROTEIN-SIGNALING PROTEIN COMPLEX
5b6b:D (MET145) to (LEU211) COMPLEX OF LATS1 AND PHOSPHOMIMETIC MOB1B | MOB1 LATS1 HIPPO PATHWAY, METAL BINDING PROTEIN-SIGNALING PROTEIN COMPLEX
5b6b:F (PHE144) to (LEU211) COMPLEX OF LATS1 AND PHOSPHOMIMETIC MOB1B | MOB1 LATS1 HIPPO PATHWAY, METAL BINDING PROTEIN-SIGNALING PROTEIN COMPLEX
5b6b:H (MET145) to (SER213) COMPLEX OF LATS1 AND PHOSPHOMIMETIC MOB1B | MOB1 LATS1 HIPPO PATHWAY, METAL BINDING PROTEIN-SIGNALING PROTEIN COMPLEX
5b6b:K (MET145) to (LEU211) COMPLEX OF LATS1 AND PHOSPHOMIMETIC MOB1B | MOB1 LATS1 HIPPO PATHWAY, METAL BINDING PROTEIN-SIGNALING PROTEIN COMPLEX
5b6b:O (ASN143) to (LEU211) COMPLEX OF LATS1 AND PHOSPHOMIMETIC MOB1B | MOB1 LATS1 HIPPO PATHWAY, METAL BINDING PROTEIN-SIGNALING PROTEIN COMPLEX
4n5v:A (ASP293) to (ILE370) ALTERNATIVE SUBSTRATES OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE
4n5v:B (ALA294) to (GLN369) ALTERNATIVE SUBSTRATES OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE
2jg4:B (GLU656) to (SER721) SUBSTRATE-FREE IDE STRUCTURE IN ITS CLOSED CONFORMATION | HYDROLASE, METAL-BINDING, METALLOPROTEASE, PROTEASE, ZINC, X-RAY CRYSTALLOGRAPHY
5bne:B (ALA294) to (GLN369) BIANTHRANILATE-LIKE INHIBITOR WITH 6 ATOM "LINE" AND PHOSPHONATE "HOOK" FISHING FOR HYDROGEN BOND DONORS IN MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | INHIBITOR, COMPLEX, LOBENZARIT-LIKE ANALOGUE, TRPD, ANPRT, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYLPYROPHOSPHATE, PRPP, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5bne:C (ASP293) to (GLN369) BIANTHRANILATE-LIKE INHIBITOR WITH 6 ATOM "LINE" AND PHOSPHONATE "HOOK" FISHING FOR HYDROGEN BOND DONORS IN MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | INHIBITOR, COMPLEX, LOBENZARIT-LIKE ANALOGUE, TRPD, ANPRT, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYLPYROPHOSPHATE, PRPP, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5bne:D (GLN295) to (GLN369) BIANTHRANILATE-LIKE INHIBITOR WITH 6 ATOM "LINE" AND PHOSPHONATE "HOOK" FISHING FOR HYDROGEN BOND DONORS IN MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | INHIBITOR, COMPLEX, LOBENZARIT-LIKE ANALOGUE, TRPD, ANPRT, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYLPYROPHOSPHATE, PRPP, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5bo2:A (GLN295) to (GLN369) BIANTHRANILATE-LIKE INHIBITOR WITH 4-ATOM "LINE" AND PHOSPHONATE "HOOK" FISHING FOR HYDROGEN BOND DONORS IN MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | LOBENZARIT-LIKE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, MAGNESIUM BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5bo2:B (ALA294) to (GLN369) BIANTHRANILATE-LIKE INHIBITOR WITH 4-ATOM "LINE" AND PHOSPHONATE "HOOK" FISHING FOR HYDROGEN BOND DONORS IN MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | LOBENZARIT-LIKE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, MAGNESIUM BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5bo3:A (ASP293) to (GLN369) BIANTHRANILATE-LIKE INHIBITOR WITH 5 ATOM "LINE" AND PHOSPHONATE "HOOK" FISHING FOR HYDROGEN BOND DONORS IN MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | INHIBITOR, COMPLEX, LOBENZARIT-LIKE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, MAGNESIUM BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5bo3:B (GLN295) to (ILE370) BIANTHRANILATE-LIKE INHIBITOR WITH 5 ATOM "LINE" AND PHOSPHONATE "HOOK" FISHING FOR HYDROGEN BOND DONORS IN MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | INHIBITOR, COMPLEX, LOBENZARIT-LIKE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, MAGNESIUM BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2jhj:A (THR163) to (GLU202) 3-METHYLADENINE DNA-GLYCOSYLASE FROM ARCHAEOGLOBUS FULGIDUS | ALKA, DNA REPAIR, N1-METHYLADENINE, N3-METHYLCYTOSINE, HYPERTHERMOPHILES, ARCHAEOGLOBUS FULGIDUS, HYDROLASE
2jhj:B (THR163) to (GLU202) 3-METHYLADENINE DNA-GLYCOSYLASE FROM ARCHAEOGLOBUS FULGIDUS | ALKA, DNA REPAIR, N1-METHYLADENINE, N3-METHYLCYTOSINE, HYPERTHERMOPHILES, ARCHAEOGLOBUS FULGIDUS, HYDROLASE
2jhn:A (THR163) to (GLU202) 3-METHYLADENINE DNA-GLYCOSYLASE FROM ARCHAEOGLOBUS FULGIDUS | ALKA, DNA REPAIR, N1-METHYLADENINE, N3-METHYLCYTOSINE, HYPERTHERMOPHILES, ARCHAEOGLOBUS FULGIDUS, HYDROLASE
2jhn:B (THR163) to (GLU202) 3-METHYLADENINE DNA-GLYCOSYLASE FROM ARCHAEOGLOBUS FULGIDUS | ALKA, DNA REPAIR, N1-METHYLADENINE, N3-METHYLCYTOSINE, HYPERTHERMOPHILES, ARCHAEOGLOBUS FULGIDUS, HYDROLASE
4n8q:B (GLN295) to (GLN369) ALTERNATIVE SUBSTRATES OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE
5bpc:A (THR121) to (LYS148) DNA POLYMERASE BETA TERNARY COMPLEX WITH A TEMPLATING 5CLC AND INCOMING DATP ANALOG | TRANSFERASE, LYASE/DNA, LIGASE-DNA COMPLEX
4n93:A (ASP293) to (ILE370) ALTERNATIVE SUBSTRATES OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE
4n93:B (GLN295) to (GLN369) ALTERNATIVE SUBSTRATES OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE
5brm:C (PHE144) to (LEU211) STRUCTURAL BASIS FOR MOB1-DEPENDENT ACTIVATION OF THE CORE MST-LATS KINASE CASCADE IN HIPPO SIGNALING | MST2, MOB1, HIPPO, TRANSFERASE-SIGNALING PROTEIN COMPLEX
5brm:E (PHE144) to (LEU211) STRUCTURAL BASIS FOR MOB1-DEPENDENT ACTIVATION OF THE CORE MST-LATS KINASE CASCADE IN HIPPO SIGNALING | MST2, MOB1, HIPPO, TRANSFERASE-SIGNALING PROTEIN COMPLEX
4nd2:A (ALA164) to (LYS244) CRYSTAL STRUCTURE OF THE LACTATE DEHYDROGENASE FROM CRYPTOSPORIDIUM PARVUM COMPLEXED WITH SUBSTRATE (PYRUVIC ACID) AND COFACTOR ANALOG (3-ACETYLPYRIDINE ADENINE DINUCLEOTIDE) | ROSSMANN FOLD, DEHYDROGENASE, NAD BINDING, OXIDOREDUCTASE
3zim:A (THR974) to (ALA1046) DISCOVERY OF A POTENT AND ISOFORM-SELECTIVE TARGETED COVALENT INHIBITOR OF THE LIPID KINASE PI3KALPHA | TRANSFERASE
2jrk:A (GLU20) to (GLU86) NMR STRUCTURE AND EPITOPE MAPPING OF BLO T 5 | BLO T 5, 3 HELICES BUNDLE, DUST MITE ALLERGEN
2y3a:A (LYS972) to (SER1046) CRYSTAL STRUCTURE OF P110BETA IN COMPLEX WITH ICSH2 OF P85BETA AND THE DRUG GDC-0941 | TRANSFERASE, PHOSPHOINOSITIDE 3-KINASE, RTK
5byt:A (GLN295) to (GLN369) PRPP COMPLEXED WITH A SINGLE MG IN THE ACTIVE SITE OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | PRPP, PHOSPHORIBOYSL PYROPHOSPHATE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, MAGNESIUM BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5byt:B (ALA294) to (GLN369) PRPP COMPLEXED WITH A SINGLE MG IN THE ACTIVE SITE OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | PRPP, PHOSPHORIBOYSL PYROPHOSPHATE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, MAGNESIUM BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1khd:A (THR278) to (ALA343) CRYSTAL STRUCTURE ANALYSIS OF THE ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE FROM ERWINIA CAROTOVORA AT 1.9 RESOLUTION (CURRENT NAME, PECTOBACTERIUM CAROTOVORUM) | TYPE 3 PRT FOLD, NUCLEOTIDE BINDING FOLD, TRANSFERASE
5c2l:A (ALA294) to (ILE370) MAGNESIUM SOAKED INTO THE ACTIVE SITE OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | PHOSPHORIBOSYLTRANSFERASE, MAGNESIUM BINDING, TBSGC, TRANSFERASE, TB STRUCTURAL GENOMICS CONSORTIUM
5c2l:B (ALA294) to (GLN369) MAGNESIUM SOAKED INTO THE ACTIVE SITE OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | PHOSPHORIBOSYLTRANSFERASE, MAGNESIUM BINDING, TBSGC, TRANSFERASE, TB STRUCTURAL GENOMICS CONSORTIUM
1ko9:A (SER183) to (SER231) NATIVE STRUCTURE OF THE HUMAN 8-OXOGUANINE DNA GLYCOSYLASE HOGG1 | HELIX-HAIRPIN-HELIX DNA-GLYCOSYLASE, HYDROLASE
2mlf:C (GLU94) to (PHE156) NMR STRUCTURE OF THE DILATED CARDIOMYOPATHY MUTATION G159D IN TROPONIN C BOUND TO THE ANCHORING REGION OF TROPONIN I | TROPONIN C, METAL BINDING PROTEIN, DILATED CARDIOMYOPATHY, G159D, EF- HAND
3zvv:A (SER1003) to (GLY1079) FRAGMENT BOUND TO PI3KINASE GAMMA | TRANSFERASE, PI3 KINASE GAMMA
1x83:B (LEU144) to (THR179) Y104F IPP ISOMERASE REACTED WITH (S)-BROMOHYDRINE OF IPP | ISOMERASE, COMPLEX
1x84:A (LEU144) to (THR179) IPP ISOMERASE (WT) REACTED WITH (S)-BROMOHYDRINE OF IPP | ISOMERASE, COMPLEX
4nvr:A (LEU171) to (ALA236) 2.22 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF A PUTATIVE ACYLTRANSFERASE FROM SALMONELLA ENTERICA | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA/BETA HYDROLASE FAMILY, TRANSFERASE
4nvr:B (LEU171) to (ALA236) 2.22 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF A PUTATIVE ACYLTRANSFERASE FROM SALMONELLA ENTERICA | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA/BETA HYDROLASE FAMILY, TRANSFERASE
4nvr:C (LEU171) to (THR228) 2.22 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF A PUTATIVE ACYLTRANSFERASE FROM SALMONELLA ENTERICA | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA/BETA HYDROLASE FAMILY, TRANSFERASE
4nvr:D (LEU171) to (ALA227) 2.22 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF A PUTATIVE ACYLTRANSFERASE FROM SALMONELLA ENTERICA | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA/BETA HYDROLASE FAMILY, TRANSFERASE
5c6n:A (ARG89) to (GLU163) PROTEIN A | PROTEIN A, TRANSPORT PROTEIN
5c6n:A (TYR312) to (GLY386) PROTEIN A | PROTEIN A, TRANSPORT PROTEIN
5c6o:A (ARG89) to (GLU163) PROTEIN B | PROTEIN BINDING, TRANSPORT PROTEIN
5c6o:A (GLN311) to (GLY386) PROTEIN B | PROTEIN BINDING, TRANSPORT PROTEIN
4nxo:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF INSULIN DEGRADING ENZYME IN COMPLEX WITH BDM44768 | HYDROLASE, INHIBITOR, CYSTEINE FREE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4nxu:B (LEU404) to (GLN462) CRYSTAL STRUCTURE OF THE CYTOSOLIC DOMAIN OF HUMAN MID51 | PROTEIN-NUCLEOTIDE COMPLEX, NUCLEOTIDYLTRANSFERASE, PROTEIN-PROTEIN INTERACTION, ADP, GDP, DRP1, MEMBRANE-ANCHORED, TRANSFERASE
4nxu:C (LEU404) to (GLN462) CRYSTAL STRUCTURE OF THE CYTOSOLIC DOMAIN OF HUMAN MID51 | PROTEIN-NUCLEOTIDE COMPLEX, NUCLEOTIDYLTRANSFERASE, PROTEIN-PROTEIN INTERACTION, ADP, GDP, DRP1, MEMBRANE-ANCHORED, TRANSFERASE
4nxv:A (LEU404) to (GLN462) CRYSTAL STRUCTURE OF THE CYTOSOLIC DOMAIN OF HUMAN MID51 | PROTEIN-NUCLEOTIDE COMPLEX, NUCLEOTIDYLTRANSFERASE, PROTEIN-PROTEIN INTERACTION, ADP, GDP, MEMBRANE-ANCHORED, TRANSFERASE, MITOCHONDRIAL FISSION, MITOCHONDRIA
4nxv:C (LEU404) to (GLN462) CRYSTAL STRUCTURE OF THE CYTOSOLIC DOMAIN OF HUMAN MID51 | PROTEIN-NUCLEOTIDE COMPLEX, NUCLEOTIDYLTRANSFERASE, PROTEIN-PROTEIN INTERACTION, ADP, GDP, MEMBRANE-ANCHORED, TRANSFERASE, MITOCHONDRIAL FISSION, MITOCHONDRIA
4nxv:D (LEU404) to (GLN462) CRYSTAL STRUCTURE OF THE CYTOSOLIC DOMAIN OF HUMAN MID51 | PROTEIN-NUCLEOTIDE COMPLEX, NUCLEOTIDYLTRANSFERASE, PROTEIN-PROTEIN INTERACTION, ADP, GDP, MEMBRANE-ANCHORED, TRANSFERASE, MITOCHONDRIAL FISSION, MITOCHONDRIA
4ny8:A (THR121) to (LYS148) DNA POLYMERASE BETA WITH O6MG IN THE TEMPLATE BASE OPPOSITE TO INCOMING NON-HYDROLYZABLE CTP WITH MANGANESE IN THE ACTIVE SITE | DNA BINDING, DNA POLYMERASE FOLD, NUCLEOTIDYL TRANSFER, NUCLEOLUS, TRANSFERASE, LYASE-DNA COMPLEX
1kw2:A (GLY389) to (ASN472) CRYSTAL STRUCTURE OF UNCOMPLEXED VITAMIN D-BINDING PROTEIN | DBP, VITAMIN D-BINDING PROTEIN, ACTIN SCAVENGER SYSTEM, ACTIN-BINDING PROTEIN, TRANSPORT PROTEIN
1kw2:B (GLY389) to (ASN472) CRYSTAL STRUCTURE OF UNCOMPLEXED VITAMIN D-BINDING PROTEIN | DBP, VITAMIN D-BINDING PROTEIN, ACTIN SCAVENGER SYSTEM, ACTIN-BINDING PROTEIN, TRANSPORT PROTEIN
5c7s:A (ASP293) to (GLN369) PRPP COMPLEXED WITH TWO MN2+ IN THE ACTIVE SITE OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, PHOSPHORIBOSYL PYROPHOSPHATE, MAGNESIUM BINDING, TBSGC, TB STRUCTURAL GENOMICS CONSORTIUM, TRANSFERASE
5c7s:B (GLN295) to (GLN369) PRPP COMPLEXED WITH TWO MN2+ IN THE ACTIVE SITE OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, PHOSPHORIBOSYL PYROPHOSPHATE, MAGNESIUM BINDING, TBSGC, TB STRUCTURAL GENOMICS CONSORTIUM, TRANSFERASE
1kzg:A (GLU624) to (PHE683) DBSCDC42(Y889F) | GUANINE NUCLEOTIDE EXCHANGE FACTOR, SMALL G-PROTEIN, CDC42, DBS, DH/PH, SIGNALING PROTEIN
3jsi:A (PHE254) to (LEU294) HUMAN PHOSPHODIESTERASE 9 IN COMPLEX WITH INHIBITOR | PHOSPHODIESTERASE, INHIBITOR, ALTERNATIVE SPLICING, CGMP, HYDROLASE, MANGANESE, METAL-BINDING, PHOSPHOPROTEIN
3jsi:B (PHE254) to (LEU294) HUMAN PHOSPHODIESTERASE 9 IN COMPLEX WITH INHIBITOR | PHOSPHODIESTERASE, INHIBITOR, ALTERNATIVE SPLICING, CGMP, HYDROLASE, MANGANESE, METAL-BINDING, PHOSPHOPROTEIN
4o5c:A (THR121) to (LYS148) STRUCTURE OF HUMAN DNA POLYMERASE COMPLEXED WITH N7-MG AS THE TEMPLATE BASE IN A 1-NUCLEOTIDE GAPPED DNA | DNA BINDING, POLYMERASE FOLD, NUCLEOTIDYL TRANSFER, DNA, NUCLEUS, TRANSFERASE, LYASE-DNA COMPLEX
4o5e:A (THR121) to (LYS148) STRUCTURE OF HUMAN DNA POLYMERASE COMPLEXED WITH N7MG IN THE TEMPLATE BASE PAIRED WITH INCOMING NON-HYDROLYZABLE TTP | DNA BINDING, POLYMERASE FOLD, NUCLEOTIDYL TRANSFER, DNA, NUCLEUS, TRANSFERASE, LYASE-DNA COMPLEX
2ypu:B (GLU656) to (SER721) HUMAN INSULIN DEGRADING ENZYME E111Q IN COMPLEX WITH INHIBITOR COMPOUND 41367 | HYDROLASE, M16A METALLOPROTEASE
4oai:Z (ALA405) to (GLN462) CRYSTAL STRUCTURE OF THE CYTOSOLIC DOMAIN OF MOUSE MID51 DIMER MUTANT | NUCLEOTIDYL TRANSFERASE FOLD, TRANSFERASE
5ci6:A (ALA231) to (LEU302) CRYSTAL STRUCTURE OF ARABIDOPSIS THALIANA MPK6 | KINASE, APOENZYME, TRANSFERASE
4oht:B (LEU45) to (MET104) CRYSTAL STRUCTURE OF SUCCINIC SEMIALDEHYDE DEHYDROGENASE FROM STREPTOCOCCUS PYOGENES IN COMPLEX WITH NADP+ AS THE COFACTOR | SSADH, GABD, OXIDOREDUCTASE, ROSSMANN FOLD, DEHYDROGENASE, NADP BINDING
4a55:A (THR974) to (ASP1045) CRYSTAL STRUCTURE OF P110ALPHA IN COMPLEX WITH ISH2 OF P85ALPHA AND THE INHIBITOR PIK-108 | TRANSFERASE, ONCOGENE, LIPID KINASE, MEMBRANE BINDING, CANCER MUTATIONS, TUMOURS, GROWTH FACTOR SIGNALLING, PI3-KINASE INHIBITOR, NON-ATP COMPETITIVE LIGAND BINDING SITE, STRUCTURE-ACTIVITY RELATIONSHIP, ENZYME REGULATION
3k75:D (THR121) to (LYS148) X-RAY CRYSTAL STRUCTURE OF REDUCED XRCC1 BOUND TO DNA POL BETA CATALYTIC DOMAIN | ALLOSTERIC DISULFIDE, XRCC1, POL BETA, DNA DAMAGE, DNA REPAIR, NUCLEUS, PHOSPHOPROTEIN, DNA REPLICATION, DNA SYNTHESIS, DNA- BINDING, DNA-DIRECTED DNA POLYMERASE, LYASE, MAGNESIUM, METAL- BINDING, METHYLATION, NUCLEOTIDYLTRANSFERASE, TRANSFERASE, DNA- BINDING PROTEIN
3k75:E (LEU122) to (LYS148) X-RAY CRYSTAL STRUCTURE OF REDUCED XRCC1 BOUND TO DNA POL BETA CATALYTIC DOMAIN | ALLOSTERIC DISULFIDE, XRCC1, POL BETA, DNA DAMAGE, DNA REPAIR, NUCLEUS, PHOSPHOPROTEIN, DNA REPLICATION, DNA SYNTHESIS, DNA- BINDING, DNA-DIRECTED DNA POLYMERASE, LYASE, MAGNESIUM, METAL- BINDING, METHYLATION, NUCLEOTIDYLTRANSFERASE, TRANSFERASE, DNA- BINDING PROTEIN
4ovu:A (ARG975) to (HIS1047) CRYSTAL STRUCTURE OF P110ALPHA IN COMPLEX WITH NISH2 OF P85ALPHA | P110, P85, PI3KCA, PI3K, PIK3R1, PHOSPHATIDILYNOSITOL 3,4,5 TRIPHOSPHATE, PIP2, PHOSPHATIDYLINOSITOL 4,5 BISPHOSPHATE, LIPID KINASE, PHOSPHOINOSITIDE, 3-KINASE, SIGNALING, PHOSPHATIDYLINOSITOL 3-KINASE
4owm:B (GLN295) to (GLN369) ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH 3-FLUOROANTHRANILATE, PRPP AND MAGNESIUM | ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE
4own:B (GLN295) to (GLN369) ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH 5-FLUOROANTHRANILATE, PRPP AND MAGNESIUM | ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE
4owo:A (ASP293) to (GLN369) ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH 6-FLUOROANTHRANILATE, PRPP AND MAGNESIUM | ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE
4owo:B (ASP293) to (GLN369) ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH 6-FLUOROANTHRANILATE, PRPP AND MAGNESIUM | ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE
4owq:A (ASP293) to (ILE370) ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH 3-METHYLANTHRANILATE, PRPP AND MAGNESIUM | ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE
4owq:B (ALA294) to (GLN369) ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH 3-METHYLANTHRANILATE, PRPP AND MAGNESIUM | ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE
4owu:A (ASP293) to (ILE370) ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH 5-METHYLANTHRANILATE, PRPP AND MAGNESIUM | ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE
4owu:B (ALA294) to (GLN369) ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH 5-METHYLANTHRANILATE, PRPP AND MAGNESIUM | ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE
4oys:A (GLU793) to (ALA873) CRYSTAL STRUCTURE OF VPS34 IN COMPLEX WITH SAR405. | LIPID KINASE
3koo:A (GLY391) to (ASN468) CRYSTAL STRUCTURE OF SOLUBLE EPOXIDE HYDROLASE | HYDROLASE
3ksy:A (PHE307) to (LEU343) CRYSTAL STRUCTURE OF THE HISTONE DOMAIN, DH-PH UNIT, AND CATALYTIC UNIT OF THE RAS ACTIVATOR SON OF SEVENLESS (SOS) | RAS, SOS, RAS ACTIVATOR, SON OF SEVENLESS, DISEASE MUTATION, GUANINE-NUCLEOTIDE RELEASING FACTOR, SIGNALING PROTEIN
3ktu:A (SER183) to (SER231) STRUCTURE OF HUMAN 8-OXOGUANINE GLYCOSYLASE 1 BOUND TO FLUORNINATED OXOG-CONTAINING DNA | 8-OXOGUANINE, 2'-FLUORO-8-OXOGUANINE, PROTEIN-DNA COMPLEX, DNA GLYCOSYLASE, BASE EXCSION REPAIR, DNA DAMAGE, DNA REPAIR, HYDROLASE, LYASE-DNA COMPLEX
5db7:A (THR121) to (LYS148) STRUCTURE OF HUMAN DNA POLYMERASE BETA HOST-GUEST COMPLEX WITH THE N7MG BASE PAIRED WITH A DT | HUMAN DNA POLYMERASE, TRANSFERASE-DNA COMPLEX
5db8:A (THR121) to (LYS148) STRUCTURE OF HUMAN DNA POLYMERASE BETA HOST-GUEST COMPLEX WITH THE N7MG BASE PAIRED WITH A DA | HUMAN DNA POLYMERASE, TRANSFERASE-DNA COMPLEX
5dba:A (THR121) to (LYS148) STRUCTURE OF HUMAN DNA POLYMERASE BETA HOST-GUEST COMPLEX WITH THE DG BASE PAIRED WITH A DT | HUMAN DNA POLYMERASE, TRANSFERASE-DNA COMPLEX
5dbc:A (THR121) to (LYS148) STRUCTURE OF HUMAN DNA POLYMERASE BETA HOST-GUEST COMPLEX WITH THE DG BASE PAIRED WITH A DG | HUMAN DNA POLYMERASE, TRANSFERASE-DNA COMPLEX
4pes:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF INSULIN DEGRADING ENZYME COMPLEXED WITH INHIBITOR TERT-BUTYL [(2S)-2-(2,5-DIFLUOROPHENYL)-3-(QUINOLIN-3-YL) PROPYL]CARBAMATE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4pf7:A (ASP655) to (SER721) CRYSTAL STRUCTURE OF INSULIN DEGRADING ENZYME COMPLEXED WITH INHIBITOR | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4pf7:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF INSULIN DEGRADING ENZYME COMPLEXED WITH INHIBITOR | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4pf9:A (GLU656) to (SER721) CRYSTAL STRUCTURE OF INSULIN DEGRADING ENZYME COMPLEXED WITH INHIBITOR | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4pf9:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF INSULIN DEGRADING ENZYME COMPLEXED WITH INHIBITOR | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4pfc:A (GLU656) to (SER721) CRYSTAL STRUCTURE OF INSULIN DEGRADING ENZYME COMPLEXED WITH INHIBITOR | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4pfc:B (ASP655) to (SER721) CRYSTAL STRUCTURE OF INSULIN DEGRADING ENZYME COMPLEXED WITH INHIBITOR | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3l08:A (SER1003) to (GLY1079) STRUCTURE OF PI3K GAMMA WITH A POTENT INHIBITOR: GSK2126458 | PI3K GAMMA, LIPID KINASE, PHOSPHOINOSITIDE, INHIBITOR, GSK2126458, SIGNALING, KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, TRANSFERASE
4pgy:A (THR121) to (LYS148) STRUCTURE OF HUMAN DNA POLYMERASE BETA COMPLEXED WITH A NICKED DNA CONTAINING A GT AT N-1 POSITION AND GC AT N POSITION | HUMAN DNA POLYMERASE BETA, NUCLEOTIDYL TRANSFER
4ph4:B (GLU793) to (PHE871) THE CRYSTAL STRUCTURE OF HUMAN VPS34 IN COMPLEX WITH PIK-III | VPS34, AUTOPHAGY, CLASS III, PHOSPHATIDYLINOSITOL-3-KINASE, PIK3C3
4pha:A (THR121) to (LYS148) STRUCTURE OF HUMAN DNA POLYMERASE BETA COMPLEXED WITH A IN THE TEMPLATE BASE PAIRED WITH INCOMING NON-HYDROLYZABLE CTP | HUMAN DNA POLYMERASE BETA
3l13:A (SER1003) to (GLY1079) CRYSTAL STRUCTURES OF PAN-PI3-KINASE AND DUAL PAN-PI3-KINASE/MTOR INHIBITORS | KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, TRANSFERASE, PI3K-GAMMA P110 GAMMA
3l17:A (SER1003) to (LYS1078) DISCOVERY OF (THIENOPYRIMIDIN-2-YL)AMINOPYRIMIDINES AS POTENT, SELECTIVE, AND ORALLY AVAILABLE PAN-PI3-KINASE AND DUAL PAN-PI3- KINASE/MTOR INHIBITORS FOR THE TREATMENT OF CANCER | KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, TRANSFERASE, PI3K-GAMMA P110 GAMMA
3ahm:A (GLU68) to (SER147) PZ PEPTIDASE A | HYDROLASE
3ahn:A (GLU68) to (SER147) PZ PEPTIDASE A WITH INHIBITOR 1 | HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3aho:A (VAL84) to (SER147) PZ PEPTIDASE A WITH INHIBITOR 2 | HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4ps3:A (SER1003) to (LYS1078) STRUCTURE OF PI3K GAMMA IN COMPLEX WITH 1-[6-(5-METHOXYPYRIDIN-3-YL)- 1,3-BENZOTHIAZOL-2-YL]-3-[2-(1-PROPYL-1H-IMIDAZOL-4-YL)ETHYL]UREA | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ps8:A (SER1003) to (LYS1078) STRUCTURE OF PI3K GAMMA IN COMPLEX WITH N-[6-(5,6-DIMETHOXYPYRIDIN-3- YL)-1,3-BENZOTHIAZOL-2-YL]ACETAMIDE | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1z9u:B (VAL21) to (GLY65) STRUCTURAL GENOMICS, THE CRYSTAL STRUCTURE OF THE ACETYL TRANSFERASE, MODIFIES N-TERMINAL SERINE OF 50S RIBOSOMAL SUBUNIT PROTEIN L7/L12 FROM SALMONELLA TYPHIMURIUM | ACETYL TRANSFERASE, L7/L12, SALMONELLA TYPHIMURIUM, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSFERASE
4anv:A (SER1003) to (GLY1079) COMPLEXES OF PI3KGAMMA WITH ISOFORM SELECTIVE INHIBITORS. | TRANSFERASE
4anw:A (SER1003) to (GLY1079) COMPLEXES OF PI3KGAMMA WITH ISOFORM SELECTIVE INHIBITORS. | TRANSFERASE
4anx:A (SER1003) to (GLY1079) COMPLEXES OF PI3KGAMMA WITH ISOFORM SELECTIVE INHIBITORS. | TRANSFERASE
4aof:A (SER1003) to (GLY1079) SELECTIVE SMALL MOLECULE INHIBITOR DISCOVERED BY CHEMOPROTEOMIC ASSAY PLATFORM REVEALS REGULATION OF TH17 CELL DIFFERENTIATION BY PI3KGAMMA | TRANSFERASE
3amj:C (THR370) to (LEU435) THE CRYSTAL STRUCTURE OF THE HETERODIMER OF M16B PEPTIDASE FROM SPHINGOMONAS SP. A1 | ALPHA/BETA, ZINC PEPTIDASE, ZINC BINDING, HYDROLASE
3lj3:A (SER1003) to (GLY1079) PI3-KINASE-GAMMA WITH A PYRROLOPYRIDINE-BENZOFURAN INHIBITOR | ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, TRANSFERASE
3ans:A (GLY391) to (ASN468) HUMAN SOLUBLE EPOXIDE HYDROLASE IN COMPLEX WITH A SYNTHETIC INHIBITOR | HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5dxh:A (ARG975) to (ALA1046) P110ALPHA/P85ALPHA WITH COMPOUND 5 | LIPID KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5dxh:D (THR974) to (ALA1046) P110ALPHA/P85ALPHA WITH COMPOUND 5 | LIPID KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5dxu:A (ASN949) to (VAL1031) P110DELTA/P85ALPHA WITH GDC-0326 | LIPID KINASE, INHIBITOR, TRANSFERASE-INHIBITOR COMPLEX
3aoe:F (ASP341) to (GLY416) CRYSTAL STRUCTURE OF HETERO-HEXAMERIC GLUTAMATE DEHYDROGENASE FROM THERMUS THERMOPHILUS (LEU BOUND FORM) | ROSSMANN FOLD, GLUTAMATE DEHYDROGENASE, DEHYDROGENASE, NADH, OXIDOREDUCTASE
3aoe:C (ASP341) to (GLY416) CRYSTAL STRUCTURE OF HETERO-HEXAMERIC GLUTAMATE DEHYDROGENASE FROM THERMUS THERMOPHILUS (LEU BOUND FORM) | ROSSMANN FOLD, GLUTAMATE DEHYDROGENASE, DEHYDROGENASE, NADH, OXIDOREDUCTASE
3aoe:D (ASP341) to (GLY416) CRYSTAL STRUCTURE OF HETERO-HEXAMERIC GLUTAMATE DEHYDROGENASE FROM THERMUS THERMOPHILUS (LEU BOUND FORM) | ROSSMANN FOLD, GLUTAMATE DEHYDROGENASE, DEHYDROGENASE, NADH, OXIDOREDUCTASE
3aog:E (ASP346) to (GLY421) CRYSTAL STRUCTURE OF GLUTAMATE DEHYDROGENASE (GDHB) FROM THERMUS THERMOPHILUS (GLU BOUND FORM) | GLUTAMATE DEHYDROGENASE, DEHYDROGENASE, NAD(H), OXIDOREDUCTASE
3aog:I (ASP346) to (GLY421) CRYSTAL STRUCTURE OF GLUTAMATE DEHYDROGENASE (GDHB) FROM THERMUS THERMOPHILUS (GLU BOUND FORM) | GLUTAMATE DEHYDROGENASE, DEHYDROGENASE, NAD(H), OXIDOREDUCTASE
3aog:K (ASP346) to (GLY421) CRYSTAL STRUCTURE OF GLUTAMATE DEHYDROGENASE (GDHB) FROM THERMUS THERMOPHILUS (GLU BOUND FORM) | GLUTAMATE DEHYDROGENASE, DEHYDROGENASE, NAD(H), OXIDOREDUCTASE
1zpq:A (LYS6) to (GLU59) STRUCTURE OF BACTERIOPHAGE LAMBDA CII PROTEIN | HELIX-TURN-HELIX, TRANSCRIPTION ACTIVATION, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSCRIPTION ACTIVATOR
1zqu:A (LEU122) to (GLU147) DNA POLYMERASE BETA (POL B) (E.C.2.7.7.7), 31-KD DOMAIN; SOAKED IN THE PRESENCE OF ARTIFICIAL MOTHER LIQUOR | DNA-DIRECTED DNA POLYMERASE, DNA REPLICATION, DNA REPAIR, NUCLEOTIDYLTRANSFERASE
1zqv:A (THR121) to (LYS148) DNA POLYMERASE BETA (POL B) (E.C.2.7.7.7), 31-KD DOMAIN; SOAKED IN THE PRESENCE OF CACL2 (150 MILLIMOLAR) | DNA-DIRECTED DNA POLYMERASE, DNA REPLICATION, DNA REPAIR, NUCLEOTIDYLTRANSFERASE
1zqy:A (LEU122) to (GLU147) DNA POLYMERASE BETA (POL B) (E.C.2.7.7.7), 31-KD DOMAIN; SOAKED IN THE PRESENCE OF MGCL2 (50 MILLIMOLAR) | DNA-DIRECTED DNA POLYMERASE, DNA REPLICATION, DNA REPAIR, NUCLEOTIDYLTRANSFERASE
1zqz:A (LEU122) to (ARG149) DNA POLYMERASE BETA (POL B) (E.C.2.7.7.7), 31-KD DOMAIN; SOAKED IN THE PRESENCE OF MNCL2 (50 MILLIMOLAR) | DNA-DIRECTED DNA POLYMERASE, DNA REPLICATION, DNA REPAIR, NUCLEOTIDYLTRANSFERASE
3ls8:A (GLU793) to (PHE871) CRYSTAL STRUCTURE OF HUMAN PIK3C3 IN COMPLEX WITH 3-[4-(4- MORPHOLINYL)THIENO[3,2-D]PYRIMIDIN-2-YL]-PHENOL | ALPHA/BETA PROTEIN, PIK3C3, PHOSPHATIDYLINOSITOL 3-KINASE CATALYTIC SUBUNIT TYPE 3, COMPOUND 15E, STRUCTURAL GENOMICS, SGC STOCKHOLM, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, TRANSFERASE, INHIBITOR, PHOSPHATIDYLINOSITOL
3ls8:B (GLU793) to (PHE871) CRYSTAL STRUCTURE OF HUMAN PIK3C3 IN COMPLEX WITH 3-[4-(4- MORPHOLINYL)THIENO[3,2-D]PYRIMIDIN-2-YL]-PHENOL | ALPHA/BETA PROTEIN, PIK3C3, PHOSPHATIDYLINOSITOL 3-KINASE CATALYTIC SUBUNIT TYPE 3, COMPOUND 15E, STRUCTURAL GENOMICS, SGC STOCKHOLM, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, TRANSFERASE, INHIBITOR, PHOSPHATIDYLINOSITOL
3apd:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF HUMAN PI3K-GAMMA IN COMPLEX WITH CH5108134 | PHOSPHOINOSITIDE 3-KINASE GAMMA, KINASE, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3apf:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF HUMAN PI3K-GAMMA IN COMPLEX WITH CH5039699 | PHOSPHOINOSITIDE 3-KINASE GAMMA, KINASE, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3lss:A (ILE5) to (LEU134) TRYPANOSOMA BRUCEI SERYL-TRNA SYNTHETASE IN COMPLEX WITH ATP | AMINOACYL-TRNA SYNTHETASE, TRNA LIGASE, AARS, SERRS, TRANSLATION, ATP-BINDING, NUCLEOTIDE-BINDING, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, LIGASE
1zvw:A (ASP293) to (ILE370) THE CRYSTAL STRUCTURE OF TRPD (RV2192C) FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH PRPP AND MAGNESIUM | ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, MYCOBACTERIUM TUBERCULOSIS STRUCTURAL PROTEOMICS PROJECT, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
1zvw:B (ASP293) to (GLN369) THE CRYSTAL STRUCTURE OF TRPD (RV2192C) FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH PRPP AND MAGNESIUM | ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, MYCOBACTERIUM TUBERCULOSIS STRUCTURAL PROTEOMICS PROJECT, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
1zxy:A (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE FROM SULFOLOBUS SOLFATARICUS IN COMPLEX WITH PRPP AND MAGNESIUM | ANTHRANILATE POSPHORIBOSYLTRANSFERASE, TRPD, PRPP
1zxy:B (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE FROM SULFOLOBUS SOLFATARICUS IN COMPLEX WITH PRPP AND MAGNESIUM | ANTHRANILATE POSPHORIBOSYLTRANSFERASE, TRPD, PRPP
1zxy:C (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE FROM SULFOLOBUS SOLFATARICUS IN COMPLEX WITH PRPP AND MAGNESIUM | ANTHRANILATE POSPHORIBOSYLTRANSFERASE, TRPD, PRPP
1zxy:D (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE FROM SULFOLOBUS SOLFATARICUS IN COMPLEX WITH PRPP AND MAGNESIUM | ANTHRANILATE POSPHORIBOSYLTRANSFERASE, TRPD, PRPP
1zyk:A (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE IN COMPLEX WITH PRPP, ANTHRANILATE AND MAGNESIUM | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, PRPP, ANTHRANILATE, TRPD
1zyk:B (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE IN COMPLEX WITH PRPP, ANTHRANILATE AND MAGNESIUM | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, PRPP, ANTHRANILATE, TRPD
1zyk:C (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE IN COMPLEX WITH PRPP, ANTHRANILATE AND MAGNESIUM | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, PRPP, ANTHRANILATE, TRPD
1zyk:D (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE IN COMPLEX WITH PRPP, ANTHRANILATE AND MAGNESIUM | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, PRPP, ANTHRANILATE, TRPD
4q9i:A (GLU93) to (ILE182) P-GLYCOPROTEIN COCRYSTALLISED WITH QZ-ALA | MEMBRANE PROTEIN, TRANSPORTER, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2a4z:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF HUMAN PI3KGAMMA COMPLEXED WITH AS604850 | PROTEIN-INHIBITOR COMPLEX, PI3KG, TRANSFERASE
4qdl:B (LEU213) to (GLU276) CRYSTAL STRUCTURE OF E.COLI CAS1-CAS2 COMPLEX | CRISPR-CAS, CAS1-CAS2 COMPLEX, CRISPR ADAPTATION, HYDROLASE
4qia:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN DEGRADING ENZYME (IDE) IN COMPLEX WITH INHIBITOR N-BENZYL-N-(CARBOXYMETHYL)GLYCYL-L-HISTIDINE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX, INHIBITOR:41371
3mjw:A (PRO1004) to (LYS1078) PI3 KINASE GAMMA WITH A BENZOFURANONE INHIBITOR | 3D-STRUCTURE,ATP-BINDING,COMPLETE PROTEOME,KINASE,NUCLEOTIDE-BINDING, TRANSFERASE, TRANSFERASE
5ep8:A (ASN249) to (GLY317) X-RAY STRUCTURE OF THE COMPLEX PYRIMIDINE-NUCLEOSIDE PHOSPHORYLASE FROM BACILLUS SUBTILIS WITH SULFATE ION | TRANSFERASE, PYRIMIDINE-NUCLEOSIDE PHOSPHORYLASE, NP-2 SUPERFAMILY
5ep8:B (ASN249) to (GLY317) X-RAY STRUCTURE OF THE COMPLEX PYRIMIDINE-NUCLEOSIDE PHOSPHORYLASE FROM BACILLUS SUBTILIS WITH SULFATE ION | TRANSFERASE, PYRIMIDINE-NUCLEOSIDE PHOSPHORYLASE, NP-2 SUPERFAMILY
4bfr:A (THR970) to (GLU1045) DISCOVERY AND OPTIMIZATION OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS FOR THE TREATMENT OF PHOSPHATASE AND TENSIN HOMOLOGUE (PTEN)-DEFICIENT CANCERS | TRANSFERASE, INHIBITOR
4bfr:B (THR970) to (GLU1045) DISCOVERY AND OPTIMIZATION OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS FOR THE TREATMENT OF PHOSPHATASE AND TENSIN HOMOLOGUE (PTEN)-DEFICIENT CANCERS | TRANSFERASE, INHIBITOR
4bht:C (GLY369) to (GLY445) STRUCTURAL DETERMINANTS OF COFACTOR SPECIFICITY AND DOMAIN FLEXIBILITY IN BACTERIAL GLUTAMATE DEHYDROGENASES | OXIDOREDUCTASE
5exr:B (GLN275) to (ILE316) CRYSTAL STRUCTURE OF HUMAN PRIMOSOME | HUMAN PRIMOSOME, COMPLEX, PRIMASE, DNA POLYMERASE ALPHA, PRIMER, DNA REPLICATION, DNA, RNA, REPLICASE, REPLICATION
5exr:F (GLN275) to (ILE316) CRYSTAL STRUCTURE OF HUMAN PRIMOSOME | HUMAN PRIMOSOME, COMPLEX, PRIMASE, DNA POLYMERASE ALPHA, PRIMER, DNA REPLICATION, DNA, RNA, REPLICASE, REPLICATION
5f4z:D (ARG242) to (ILE307) THE CRYSTAL STRUCTURE OF AN EPOXIDE HYDROLASE FROM STREPTOMYCES CARZINOSTATICUS SUBSP. NEOCARZINOSTATICUS | EPOXIDE HYDROLASE, STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, HYDROLASE
3n3z:B (PHE254) to (LEU294) CRYSTAL STRUCTURE OF PDE9A (E406A) MUTANT IN COMPLEX WITH IBMX | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3n56:A (ASP655) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME (IDE) IN COMPLEX WITH HUMAN B-TYPE NATRIURETIC PEPTIDE (BNP) | INSULYSIN, INSULINASE, A-BETA DEGRADING ENZYME, CRYPTIDASE, HYDROLASE, HORMONE, DISEASE MUTATION, DIABETES MELLITUS, INSULIN, CARDIAC, SECRETED, PROTEASE, DISULFIDE BOND, METALLOPROTEASE, HUMAN INSULIN-DEGRADNG ENZYME, METAL-BINDING, NATRIURETIC PEPTIDE, NATRIURETIC FACTOR, CARDIOVASCULAR REGULATION, HYDROLASE-HORMONE COMPLEX
3n56:B (ASP655) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME (IDE) IN COMPLEX WITH HUMAN B-TYPE NATRIURETIC PEPTIDE (BNP) | INSULYSIN, INSULINASE, A-BETA DEGRADING ENZYME, CRYPTIDASE, HYDROLASE, HORMONE, DISEASE MUTATION, DIABETES MELLITUS, INSULIN, CARDIAC, SECRETED, PROTEASE, DISULFIDE BOND, METALLOPROTEASE, HUMAN INSULIN-DEGRADNG ENZYME, METAL-BINDING, NATRIURETIC PEPTIDE, NATRIURETIC FACTOR, CARDIOVASCULAR REGULATION, HYDROLASE-HORMONE COMPLEX
3n57:A (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME (IDE) IN COMPLEX WITH HUMAN ATRIAL NATRIURETIC PEPTIDE (ANP) | INSULYSIN, INSULINASE, A-BETA DEGRADING ENZYME, CRYPTIDASE, HYDROLASE, HORMONE, DISEASE MUTATION, DIABETES MELLITUS, INSULIN, CARDIAC, SECRETED, PROTEASE, DISULFIDE BOND, METALLOPROTEASE, HUMAN INSULIN-DEGRADNG ENZYME, METAL-BINDING, NATRIURETIC PEPTIDE, NATRIURETIC FACTOR, CARDIOVASCULAR REGULATION, HYDROLASE-HORMONE COMPLEX
3n57:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME (IDE) IN COMPLEX WITH HUMAN ATRIAL NATRIURETIC PEPTIDE (ANP) | INSULYSIN, INSULINASE, A-BETA DEGRADING ENZYME, CRYPTIDASE, HYDROLASE, HORMONE, DISEASE MUTATION, DIABETES MELLITUS, INSULIN, CARDIAC, SECRETED, PROTEASE, DISULFIDE BOND, METALLOPROTEASE, HUMAN INSULIN-DEGRADNG ENZYME, METAL-BINDING, NATRIURETIC PEPTIDE, NATRIURETIC FACTOR, CARDIOVASCULAR REGULATION, HYDROLASE-HORMONE COMPLEX
5fi4:A (ARG975) to (HIS1048) DISCOVERY OF IMIDAZO[1,2-A]-PYRIDINE INHIBITORS OF PAN-PI3 KINASES THAT ARE EFFICACIOUS IN A MOUSE XENOGRAFT MODEL | LIPID KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5fic:C (ASN84) to (GLY160) OPEN FORM OF MURINE ACID SPHINGOMYELINASE IN PRESENCE OF LIPID | SMPD1, ASM, ASMASE, SPHINGOMYELINASE, HYDROLASE
4r8z:B (HIS327) to (ALA365) CRYSTAL STRUCTURE OF PA4781 HD-GYP DOMAIN FROM PSEUDOMONAS AERUGINOSA AT 2.2A RESOLUTION SHOWING A BI-METALLIC NI ION CENTER | BIMETALLIC, C-DI-GMP, PDE, PHOSPHDIESTERASE, CYCLIC-DI-GMP, BIOFILM, HYDROLASE
4ral:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF INSULIN DEGRADING ENZYME IN COMPLEX WITH MACROPHAGE INFLAMMATORY PROTEIN 1 BETA | IDE, MIP1ALPHA, METAL-BINDING, METALLOPROTEASE, CHEMOTAXIS, INFLAMMATORY RESPONSE, HYDROLASE-CYTOKINE COMPLEX
4re9:A (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN DEGRADING ENZYME (IDE) IN COMPLEX WITH COMPOUND 71290 | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4re9:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN DEGRADING ENZYME (IDE) IN COMPLEX WITH COMPOUND 71290 | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4rea:A (TYR374) to (ARG424) A NUCLEASE DNA COMPLEX | HJC, TPR, SAP, STRUCTURAL SPECIFIC NUCLEASE, FANCD2, NUCLEUS, HYDROLASE-DNA COMPLEX
4rea:B (TYR374) to (ARG424) A NUCLEASE DNA COMPLEX | HJC, TPR, SAP, STRUCTURAL SPECIFIC NUCLEASE, FANCD2, NUCLEUS, HYDROLASE-DNA COMPLEX
4rec:A (TYR374) to (ARG424) A NUCLEASE-DNA COMPLEX FORM 3 | HJC, TPR, SAP, STRUCTURE SPECIFIC NUCLEASE, FANCID2, NUCLEUS, HYDROLASE-DNA COMPLEX
4reb:A (TYR374) to (LYS425) STRUCTURAL INSIGHTS INTO 5' FLAP DNA UNWINDING AND INCISION BY THE HUMAN FAN1 DIMER | HJC, TPR, SAP, STRUCTURE SPECIFIC NUCLEASE, FANCID2, NUCLEUS, HYDROLASE-DNA COMPLEX
4ri8:A (TYR374) to (ARG424) FAN1 NUCLEASE BOUND TO 5' PHOSPHORYLATED P(DG)/3'(DT-DT-DT-DT) DOUBLE FLAP DNA | NUCLEASE, HYDROLASE-DNA COMPLEX
4ri8:B (TYR374) to (ARG424) FAN1 NUCLEASE BOUND TO 5' PHOSPHORYLATED P(DG)/3'(DT-DT-DT-DT) DOUBLE FLAP DNA | NUCLEASE, HYDROLASE-DNA COMPLEX
4ri9:A (TYR374) to (ARG424) FAN1 NUCLEASE BOUND TO 5' PHOSPHORYLATED P(DT)/3'(DT-DT-DT-DT-DT-DT- DT-DT) DOUBLE FLAP DNA | NUCLEASE, HYDROLASE-DNA COMPLEX
4ri9:B (TYR374) to (ARG424) FAN1 NUCLEASE BOUND TO 5' PHOSPHORYLATED P(DT)/3'(DT-DT-DT-DT-DT-DT- DT-DT) DOUBLE FLAP DNA | NUCLEASE, HYDROLASE-DNA COMPLEX
4ria:A (PRO373) to (ARG424) FAN1 NUCLEASE BOUND TO 5' PHOSPHORYLATED NICKED DNA | NUCLEASE, HYDROLASE-DNA COMPLEX
4ria:B (TYR374) to (ARG424) FAN1 NUCLEASE BOUND TO 5' PHOSPHORYLATED NICKED DNA | NUCLEASE, HYDROLASE-DNA COMPLEX
4rib:A (TYR374) to (ARG424) FAN1 NUCLEASE BOUND TO 5' PHOSPHORYLATED P(DT) SINGLE FLAP DNA | NUCLEASE, HYDROLASE-DNA COMPLEX
4rib:B (TYR374) to (ARG424) FAN1 NUCLEASE BOUND TO 5' PHOSPHORYLATED P(DT) SINGLE FLAP DNA | NUCLEASE, HYDROLASE-DNA COMPLEX
4ric:A (TYR374) to (ARG424) FAN1 NUCLEASE BOUND TO 5' HYDROXYL (DT-DT) SINGLE FLAP DNA | NUCLEASE, HYDROLASE-DNA COMPLEX
4ric:B (TYR374) to (ARG424) FAN1 NUCLEASE BOUND TO 5' HYDROXYL (DT-DT) SINGLE FLAP DNA | NUCLEASE, HYDROLASE-DNA COMPLEX
4caz:A (MET66) to (ILE123) CRYSTAL STRUCTURE OF BETAINE ALDEHYDE DEHYDROGENASE FROM PSEUDOMONAS AERUGINOSA IN COMPLEX WITH NADH | ALDEHYDE OXIDATION, NADH COMPLEX, OXIDOREDUCTASE
4cbb:C (THR64) to (ILE123) APO FORM OF BETAINE ALDEHYDE DEHYDROGENASE FROM PSEUDOMONAS AERUGINOSA | OXIDOREDUCTASE, ALDEHYDE OXIDATION
4rpy:A (THR121) to (LYS148) HUMAN DNA POLYMERASE BETA WITH GAPPED DNA CONTAINING AN 8-OXO-7,8- DIHYDRO-GUANINE(8-OXOG) AND DCTP SOAKED WITH MGCL2 FOR 30 S | X-FAMILY, POL BETA, TRANSFERASE-DNA COMPLEX
4rpz:A (THR121) to (LYS148) HUMAN DNA POLYMERASE BETA WITH GAPPED DNA CONTAINING AN 8-OXO-7,8- DIHYDRO-GUANINE (8-OXOG)AND DCTP SOAKED WITH MGCL2 FOR 60 S | X-FAMILY, POL BETA, TRANSFERASE-DNA COMPLEX
4rq3:A (THR121) to (LYS148) PRECATALYTIC TERNARY COMPLEX OF HUMAN DNA POLYMERASE BETA WITH GAPPED DNA CONTAINING AN 8-OXO-7,8-DIHYDRO-GUANINE (8-OXOG) AND DATP IN THE PRESENCE OF CACL2 | X-FAMILY, POL BETA, TRANSFERASE-DNA COMPLEX
4rq4:A (THR121) to (LYS148) HUMAN DNA POLYMERASE BETA WITH GAPPED DNA CONTAINING AN 8-OXO-7,8- DIHYDRO-GUANINE(8-OXOG) AND DATP SOAKED WITH MGCL2 FOR 30 S | X-FAMILY, POL BETA, TRANSFERASE-DNA COMPLEX
4rq8:A (THR121) to (GLU147) HUMAN DNA POLYMERASE BETA WITH GAPPED DNA CONTAINING AN 8-OXO-7,8- DIHYDRO-GUANINE(8-OXOG) AND DATP SOAKED WITH MNCL2 FOR 35 S | X-FAMILY, POL BETA, TRANSFERASE-DNA COMPLEX
3csf:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF PI3K P110GAMMA CATALYTICAL DOMAIN IN COMPLEX WITH ORGANORUTHENIUM INHIBITOR DW2 | PHOSPHOINOSITIDE 3-KINASE GAMMA, PI3K, TRANSFERASE
3cst:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF PI3K P110GAMMA CATALYTICAL DOMAIN IN COMPLEX WITH ORGANORUTHENIUM INHIBITOR E5E2 | PHOSPHOINOSITIDE 3-KINASE GAMMA, PI3K, TRANSFERASE
3nzs:A (SER1003) to (LYS1078) STRUCTURE-BASED OPTIMIZATION OF PYRAZOLO -PYRIMIDINE AND -PYRIDINE INHIBITORS OF PI3-KINASE | KINASE P110, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3nzu:A (SER1003) to (GLY1079) STRUCTURE-BASED OPTIMIZATION OF PYRAZOLO -PYRIMIDINE AND -PYRIDINE INHIBITORS OF PI3-KINASE | KINASE P110, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3cww:A (GLU656) to (SER721) CRYSTAL STRUCTURE OF IDE-BRADYKININ COMPLEX | A-BETA DEGRADING ENZYME, CRIPTIDASE, BRADYKININ, KININS, HYDROLASE
3cww:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF IDE-BRADYKININ COMPLEX | A-BETA DEGRADING ENZYME, CRIPTIDASE, BRADYKININ, KININS, HYDROLASE
4co6:A (MSE264) to (LEU313) CRYSTAL STRUCTURE OF THE NIPAH VIRUS RNA FREE NUCLEOPROTEIN-PHOSPHOPROTEIN COMPLEX | CHAPERONE, VIRAL PROTEIN, VIRAL REPLICATION, PARAMYXOVIRUS
5g2n:A (SER1003) to (LYS1078) X-RAY STRUCTURE OF PI3KINASE GAMMA IN COMPLEX WITH COPANLISIB | TRANSFERASE
3dbs:A (SER1003) to (LYS1078) STRUCTURE OF PI3K GAMMA IN COMPLEX WITH GDC0941 | PI3K GAMMA, INHIBITOR, KINASE, TRANSFERASE
3ofi:A (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME IN COMPLEX WITH UBIQUITIN | PROTEIN-PEPTIDE COMPLEX, HYDROLASE, HUMAN INSULIN-DEGRADING ENZYME, UBIQUITIN, EXOSITE
3ofi:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME IN COMPLEX WITH UBIQUITIN | PROTEIN-PEPTIDE COMPLEX, HYDROLASE, HUMAN INSULIN-DEGRADING ENZYME, UBIQUITIN, EXOSITE
3ogu:A (THR121) to (LYS148) DNA POLYMERASE BETA MUTANT 5P20 COMPLEXED WITH 6BP OF DNA | DNA POLYMERASE, DNA REPAIR, TRANSFERASE-DNA COMPLEX
5gm2:A (SER229) to (LYS276) CRYSTAL STRUCTURE OF METHYLTRANSFERASE TLED COMPLEXED WITH SAH AND TELEOCIDIN A1 | TLED, TELEOCIDIN, METHYLTRANSFERASES, TERPENE CYCLIZATION, TRANSFERASE
5gm2:D (SER229) to (LYS276) CRYSTAL STRUCTURE OF METHYLTRANSFERASE TLED COMPLEXED WITH SAH AND TELEOCIDIN A1 | TLED, TELEOCIDIN, METHYLTRANSFERASES, TERPENE CYCLIZATION, TRANSFERASE
5gm2:H (SER229) to (LYS276) CRYSTAL STRUCTURE OF METHYLTRANSFERASE TLED COMPLEXED WITH SAH AND TELEOCIDIN A1 | TLED, TELEOCIDIN, METHYLTRANSFERASES, TERPENE CYCLIZATION, TRANSFERASE
5gm2:M (SER229) to (ILE274) CRYSTAL STRUCTURE OF METHYLTRANSFERASE TLED COMPLEXED WITH SAH AND TELEOCIDIN A1 | TLED, TELEOCIDIN, METHYLTRANSFERASES, TERPENE CYCLIZATION, TRANSFERASE
4tuu:A (THR974) to (ASP1045) ISOLATED P110A SUBUNIT OF PI3KA PROVIDES A PLATFORM FOR STRUCTURE- BASED DRUG DESIGN | LIPID KINASE ACTIVITY, ATPASE ACTIVITY, SURFACE PLASMON RESONANCE (SPR), ISOTHERMAL TITRATION CALORIMETRY (ITC)., TRANSFERASE
3dpd:A (SER1003) to (GLY1079) ACHIEVING MULTI-ISOFORM PI3K INHIBITION IN A SERIES OF SUBSTITUTED 3,4-DIHYDRO-2H-BENZO[1,4]OXAZINES | PHOSPHOINOSITIDE 3-KINASE GAMMA, SECONDARY MESSENGER GENERATION, PI3K, PI 3K, KINASE, TRANSFERASE
4u16:A (ILE64) to (ASN131) M3-MT4L RECEPTOR BOUND TO NMS | GPCR CRYSTALLOGRAPHY T4 LYSOZYME, MEMBRANE PROTEIN-INHIBITOR COMPLEX
4ddj:A (SER1) to (ASN77) CRYSTAL STRUCTURE OF SAPOSIN A IN COMPLEX WITH LAURYLDIMETHYLAMINE-N- OXIDE (LDAO) | SAPOSIN FOLD, SPHINGOLIPID ACTIVATOR PROTEIN, GALACTOSYLCERAMIDE, LAURYLDIMETHYLAMINE-N-OXIDE, LIPID, DETERGENT, LYSOSOME, LIPID BINDING PROTEIN
3dy8:A (PHE254) to (LEU294) HUMAN PHOSPHODIESTERASE 9 IN COMPLEX WITH PRODUCT 5'-GMP (E+P COMPLEX) | PHOSPHODIESTRASE, ENZYME MECHANISM, CGMP, HYDROLASE, MANGANESE, METAL-BINDING, PHOSPHOPROTEIN
3dy8:B (PHE254) to (LEU294) HUMAN PHOSPHODIESTERASE 9 IN COMPLEX WITH PRODUCT 5'-GMP (E+P COMPLEX) | PHOSPHODIESTRASE, ENZYME MECHANISM, CGMP, HYDROLASE, MANGANESE, METAL-BINDING, PHOSPHOPROTEIN
3dyn:A (PHE254) to (LEU294) HUMAN PHOSPHODIESTRASE 9 IN COMPLEX WITH CGMP (ZN INHIBITED) | PHOPHODIESTRASE, ENZYME MECHANISM, CGMP, HYDROLASE, MANGANESE, METAL- BINDING, PHOSPHOPROTEIN
3dyn:B (PHE254) to (LEU294) HUMAN PHOSPHODIESTRASE 9 IN COMPLEX WITH CGMP (ZN INHIBITED) | PHOPHODIESTRASE, ENZYME MECHANISM, CGMP, HYDROLASE, MANGANESE, METAL- BINDING, PHOSPHOPROTEIN
4dk5:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF HUMAN PI3K-GAMMA IN COMPLEX WITH A PYRIDYL- TRIAZINE INHIBITOR | PHOSPHOTRANSFERASE, CANCER, P85-ALPHA, P85-BETA, RAS, TRANSFERASE- INHIBITOR COMPLEX
3dys:A (PHE254) to (LEU294) HUMAN PHOSPHODIESTRASE-5'GMP COMPLEX (EP), PRODUCED BY SOAKING WITH 20MM CGMP+20 MM MNCL2+20 MM MGCL2 FOR 2 HOURS, AND FLASH-COOLED TO LIQUID NITROGEN TEMPERATURE WHEN SUBSTRATE WAS STILL ABUDANT. | PHOSPHODIESTRASE, ENZYME MECHANISM, CGMP, HYDROLASE, MANGANESE, METAL-BINDING, PHOSPHOPROTEIN
3dys:B (PHE254) to (LEU294) HUMAN PHOSPHODIESTRASE-5'GMP COMPLEX (EP), PRODUCED BY SOAKING WITH 20MM CGMP+20 MM MNCL2+20 MM MGCL2 FOR 2 HOURS, AND FLASH-COOLED TO LIQUID NITROGEN TEMPERATURE WHEN SUBSTRATE WAS STILL ABUDANT. | PHOSPHODIESTRASE, ENZYME MECHANISM, CGMP, HYDROLASE, MANGANESE, METAL-BINDING, PHOSPHOPROTEIN
3p7l:A (LYS656) to (LEU720) RAT INSULIN DEGRADING ENZYME (INSULYSIN) | PEPTIDASE, HYDROLASE
3p7o:A (ASP655) to (SER721) RAT INSULIN DEGRADING ENZYME (INSULYSIN) E111F MUTANT WITH TWO BOUND PEPTIDES | METALLOPEPTIDASE, HYDROLASE
4doc:A (THR121) to (LYS148) TERNARY COMPLEX OF DNA POLYMERASE BETA WITH A DIDEOXY TERMINATED PRIMER AND 2'-DEOXYGUANOSINE 5'-BETA, GAMMA-MONOCHLOROROMETHYLENE TRIPHOSPHATE:BINDING OF S-ISOMER | STEREOSELECTIVITY, POLYMERASE, DNA POLYMERASE, TRANSFERASE-DNA COMPLEX
4ucd:B (ASN37) to (GLY87) N-TERMINAL GLOBULAR DOMAIN OF THE RSV NUCLEOPROTEIN IN COMPLEX WITH THE NUCLEOPROTEIN PHOSPHOPROTEIN INTERACTION INHIBITOR M81 | VIRAL PROTEIN, RESPIRATORY SYNCYTIAL VIRUS, RIBONUCLEOPROTEIN, NUCLEOCAPSID, PHOSPHOPROTEIN, ANTIVIRAL COMPOUNDS, HALOGEN BOND
3e4a:A (ASP655) to (SER721) HUMAN IDE-INHIBITOR COMPLEX AT 2.6 ANGSTROM RESOLUTION | INSULIN, HYDROXAMATE, INSULIN DEGRADING ENZYME, HYDROLASE, METAL- BINDING, METALLOPROTEASE, PROTEASE
3e4z:B (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN DEGRADING ENZYME IN COMPLEX WITH INSULIN-LIKE GROWTH FACTOR II | IDE, IGF-II, DEGRADING, COMPLEX, ALTERNATIVE SPLICING, GLYCOPROTEIN, GROWTH FACTOR, MITOGEN, POLYMORPHISM, SECRETED, HYDROLASE/HORMONE COMPLEX
4uf5:B (PHE49) to (ASP113) CRYSTAL STRUCTURE OF UCH-L5 IN COMPLEX WITH INHIBITORY FRAGMENT OF INO80G | HYDROLASE, DEUBIQUITINATING ENZYME
4dwk:A (GLU656) to (SER721) STRUCTURE OF CYSTEIN FREE INSULIN DEGRADING ENZYME WITH COMPOUND BDM41671 ((S)-2-{2-[CARBOXYMETHYL-(3-PHENYL-PROPYL)-AMINO]- ACETYLAMINO}-3-(1H-IMIDAZOL-4-YL)-PROPIONIC ACID METHYL ESTER) | METALLOENDOPEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4dwk:B (GLU656) to (SER721) STRUCTURE OF CYSTEIN FREE INSULIN DEGRADING ENZYME WITH COMPOUND BDM41671 ((S)-2-{2-[CARBOXYMETHYL-(3-PHENYL-PROPYL)-AMINO]- ACETYLAMINO}-3-(1H-IMIDAZOL-4-YL)-PROPIONIC ACID METHYL ESTER) | METALLOENDOPEPTIDASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5i85:A (TRP84) to (GLY162) ASMASE WITH ZINC AND PHOSPHOCHOLINE | ACID SPHINGOMYELINASE, PHOSPHOCHOLINE, HYDROLASE
3pre:A (SER1003) to (GLY1079) QUINAZOLINES WITH INTRA-MOLECULAR HYDROGEN BONDING SCAFFOLD (IMHBS) AS PI3K/MTOR DUAL INHIBITORS. | PHOSPHOINOSITIDE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3prz:A (PRO1004) to (GLY1079) QUINAZOLINES WITH INTRA-MOLECULAR HYDROGEN BONDING SCAFFOLD (IMHBS) AS PI3K/MTOR DUAL INHIBITORS. | PHOSPHOINOSITIDE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5is5:A (ASN949) to (SER1026) DISCOVERY AND PHARMACOLOGICAL CHARACTERIZATION OF NOVEL QUINAZOLINE- BASED PI3K DELTA-SELECTIVE INHIBITORS | PHOSPHOINOSITIDE 3-KINASE, ISOFORM-SEPCIFIC INHIBITORS, TRANSFERASE
5itd:A (THR974) to (HIS1048) CRYSTAL STRUCTURE OF PI3K ALPHA WITH PI3K DELTA INHIBITOR | INHIBITOR, LIPID KINASE, PI3K, ALPHA, DELTA, TRANSFERASE-PROTEIN TRANSPORT-INHIBITOR COMPLEX
5iwa:B (PHE105) to (LYS156) CRYSTAL STRUCTURE OF THE 30S RIBOSOMAL SUBUNIT FROM THERMUS THERMOPHILUS IN COMPLEX WITH THE GE81112 PEPTIDE ANTIBIOTIC | PROTEIN SYNTHESIS, TRANSLATION INITIATION, RIBOSOME, ANTIBIOTIC, TRANSCRIPTION
3qaq:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF PI3K-GAMMA IN COMPLEX WITH TRIAZINE-BENZIMIDAZOLE 1 | INHIBITOR, P110, KINASE, TRANSFERASE, ATP BINDING, P84, P101, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4ezj:A (SER1003) to (GLY1079) POTENT AND SELECTIVE INHIBITORS OF PI3K-DELTA: OBTAINING ISOFORM SELECTIVITY FROM THE AFFINITY POCKET AND TRYPTOPHAN SHELF | KINASE P110, P110-GAMMA, LIPID KINASE, CYTOPLASMIC, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4ezk:A (SER1003) to (GLY1079) POTENT AND SELECTIVE INHIBITORS OF PI3K-DELTA: OBTAINING ISOFORM SELECTIVITY FROM THE AFFINITY POCKET AND TRYPTOPHAN SHELF | KINASE P110, P110-GAMMA, LIPID KINASE, CYTOPLASMIC, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4f1s:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF HUMAN PI3K-GAMMA IN COMPLEX WITH A PYRIDYL- TRIAZINE-SULFONAMIDE INHIBITOR | PHOSPHOTRANSFERASE, LIPID KINASE, P85, TRANSFERASE-INHIBITOR COMPLEX
5j0p:A (LEU122) to (LYS148) BINARY COMPLEX CRYSTAL STRUCTURE OF DNA POLYMERASE BETA WITH A:C MISMATCH AT THE PRIMER TERMINUS | DNA POLYMERASE BETA, MISMATCH EXTENSION, BINARY COMPLEX, TRANSFERASE- DNA COMPLEX
5j0q:A (THR121) to (LYS148) BINARY COMPLEX CRYSTAL STRUCTURE OF DNA POLYMERASE BETA WITH A:G MISMATCH AT THE PRIMER TERMINUS | DNA POLYMERASE BETA, MISMATCH EXTENSION, BINARY COMPLEX, TRANSFERASE- DNA COMPLEX
5j0t:A (LEU122) to (LYS148) BINARY COMPLEX CRYSTAL STRUCTURE OF DNA POLYMERASE BETA WITH G:A MISMATCH AT THE PRIMER TERMINUS | DNA POLYMERASE BETA, MISMATCH EXTENSION, BINARY COMPLEX, TRANSFERASE- DNA COMPLEX
5j0w:A (THR121) to (LYS148) BINARY COMPLEX CRYSTAL STRUCTURE OF DNA POLYMERASE BETA WITH T:C MISMATCH AT THE PRIMER TERMINUS | DNA POLYMERASE BETA, MISMATCH EXTENSION, BINARY COMPLEX, TRANSFERASE- DNA COMPLEX
5j0y:A (THR121) to (LYS148) BINARY COMPLEX CRYSTAL STRUCTURE OF DNA POLYMERASE BETA WITH T:T MISMATCH AT THE PRIMER TERMINUS | DNA POLYMERASE BETA, MISMATCH EXTENSION, BINARY COMPLEX, TRANSFERASE- DNA COMPLEX
4f5q:A (THR121) to (LYS148) CLOSED TERNARY COMPLEX OF R283K DNA POLYMERASE BETA | TRANSFERASE, LYASE/DNA, LYASE-DNA COMPLEX
3qi4:B (PHE254) to (LEU294) CRYSTAL STRUCTURE OF PDE9A(Q453E) IN COMPLEX WITH IBMX | PDE, HYDROLASE
3qjz:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF PI3K-GAMMA IN COMPLEX WITH BENZOTHIAZOLE 1 | P110, TRANSFERASE, KINASE, INHIBITOR, ATP-BINDING, P84, P101, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qk0:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF PI3K-GAMMA IN COMPLEX WITH BENZOTHIAZOLE 82 | P110, TRANSFERASE, KINASE, INHIBITOR, ATP-BINDING, P84, P101, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4uwg:A (GLU793) to (ALA869) DISCOVERY OF (2S)-8-((3R)-3-METHYLMORPHOLIN-4-YL)-1-(3- METHYL-2-OXO-BUTYL)-2-(TRIFLUOROMETHYL)-3,4-DIHYDRO-2H- PYRIMIDO(1,2-A)PYRIMIDIN-6-ONE: A NOVEL POTENT AND SELECTIVE INHIBITOR OF VPS34 FOR THE TREATMENT OF SOLID TUMORS | TRANSFERASE
4uwh:A (GLN794) to (ALA873) DISCOVERY OF (2S)-8-((3R)-3-METHYLMORPHOLIN-4-YL)-1-(3- METHYL-2-OXO-BUTYL)-2-(TRIFLUOROMETHYL)-3,4-DIHYDRO-2H- PYRIMIDO(1,2-A)PYRIMIDIN-6-ONE: A NOVEL POTENT AND SELECTIVE INHIBITOR OF VPS34 FOR THE TREATMENT OF SOLID TUMORS | TRANSFERASE, LIPID KINASE, AUTOPHAGY INHIBITOR
4uwl:A (GLU793) to (VAL867) DISCOVERY OF (2S)-8-((3R)-3-METHYLMORPHOLIN-4-YL)-1-(3- METHYL-2-OXO-BUTYL)-2-(TRIFLUOROMETHYL)-3,4-DIHYDRO-2H- PYRIMIDO(1,2-A)PYRIMIDIN-6-ONE: A NOVEL POTENT AND SELECTIVE INHIBITOR OF VPS34 FOR THE TREATMENT OF SOLID TUMORS | TRANSFERASE, LIPID KINASE, AUTOPHAGY INHIBITOR
4fa6:A (SER1003) to (GLY1079) DESIGN AND SYNTHESIS OF A NOVEL PYRROLIDINYL PYRIDO PYRIMIDINONE DERIVATIVE AS A POTENT INHIBITOR OF PI3KA AND MTOR | PHOSPHOINOSITIDE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qqs:A (ASP293) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS172) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
3qqs:B (ASP293) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS172) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
3qqs:C (ASP293) to (ARG365) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS172) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
3qqs:D (ALA294) to (GLN369) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS172) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
3qr9:A (ALA294) to (GLN369) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (APO STRUCTURE) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
3qsa:A (ASP293) to (ARG368) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR TAMU-A7) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
3qsa:B (ALA294) to (GLN369) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR TAMU-A7) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
4fhk:A (SER1003) to (LYS1078) CRYSTAL STRUCTURE OF PI3K-GAMMA IN COMPLEX WITH IMIDAZOPYRIDAZINE 19E | P110, KINASE, ATP-BINDING, P84, P101, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3qz2:B (ASP655) to (SER721) THE STRUCTURE OF CYSTEINE-FREE HUMAN INSULIN DEGRADING ENZYME | INSULIN DEGRADING ENZYME, HYDROLASE
4fjy:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF PI3K-GAMMA IN COMPLEX WITH QUINOLINE-INDOLINE INHIBITOR 24F | INFLAMMATION, CANCER, P110, C2 DOMAIN, LEUKOCYTES, KINASE, P85, PHOSPHOTRANSFERASE, TRANSFERASE-INHIBITOR COMPLEX
4fjz:A (SER1003) to (LYS1078) CRYSTAL STRUCTURE OF PI3K-GAMMA IN COMPLEX WITH PYRROLO-PYRIDINE INHIBITOR 63 | INFLAMMATION, CANCER, P110, C2 DOMAIN, LEUKOCYTES, KINASE, P85, PHOSPHOTRANSFERASE, TRANSFERASE-INHIBITOR COMPLEX
4flh:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF HUMAN PI3K-GAMMA IN COMPLEX WITH AMG511 | P110, PHOSPHOTRANSFERASE, CANCER, P85, PHOSPHORYLATION, TRANSFERASE- INHIBITOR COMPLEX
3r6c:A (ASP293) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS179) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r6c:B (ASP293) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS179) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r7q:A (PRO1004) to (GLY1079) STRUCTURE-BASED DESIGN OF THIENOBENZOXEPIN INHIBITORS OF PI3- KINASE | KINASE P110, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r7r:A (SER1003) to (GLY1079) STRUCTURE-BASED DESIGN OF THIENOBENZOXEPIN INHIBITORS OF PI3-KINASE | KINASE P110, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r88:A (ALA294) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS145) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3r88:B (ASP293) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS145) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5jhx:A (GLY158) to (GLY210) CRYSTAL STRUCTURE OF FUNGAL MAGKATG2 AT PH 3.0 | OXIDOREDUCTASE
5jhx:B (GLY158) to (GLY210) CRYSTAL STRUCTURE OF FUNGAL MAGKATG2 AT PH 3.0 | OXIDOREDUCTASE
5jhz:A (GLY158) to (GLY210) CRYSTAL STRUCTURE OF FUNGAL MAGKATG2 AT PH 7.0 | OXIDOREDUCTASE
3rey:A (VAL8) to (GLY69) THERMOSTABILISED ADENOSINE A2A RECEPTOR IN COMPLEX WITH XAC | 7TM, GPCR, SIGNALING PROTEIN, G-PROTEIN, MEMBRANE PROTEIN
4ful:A (SER1003) to (GLY1079) PI3 KINASE GAMMA BOUND TO A PYRMIDINE INHIBITOR | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fy0:A (LYS398) to (GLU478) CRYSTAL STRUCTURE OF LEUT-F253A BOUND TO L-SELENOMETHIONINE FROM LIPID BICELLES | AMINO ACID TRANSPORTER, TRANSPORT PROTEIN
5k3g:A (ILE557) to (SER617) CRYSTALS STRUCTURE OF ACYL-COA OXIDASE-1 IN CAENORHABDITIS ELEGANS, APO FORM-I | DAUER PHEROMONE, ASCAROSIDES, B-OXIDATION, ATP, OXIDOREDUCTASE
5k3g:C (ILE557) to (SER617) CRYSTALS STRUCTURE OF ACYL-COA OXIDASE-1 IN CAENORHABDITIS ELEGANS, APO FORM-I | DAUER PHEROMONE, ASCAROSIDES, B-OXIDATION, ATP, OXIDOREDUCTASE
5k3g:D (ILE557) to (SER617) CRYSTALS STRUCTURE OF ACYL-COA OXIDASE-1 IN CAENORHABDITIS ELEGANS, APO FORM-I | DAUER PHEROMONE, ASCAROSIDES, B-OXIDATION, ATP, OXIDOREDUCTASE
4gb9:A (SER1003) to (LYS1078) POTENT AND HIGHLY SELECTIVE BENZIMIDAZOLE INHIBITORS OF PI3K-DELTA | KINASE P110 GAMMA-ISOFORM, KINASE, LIPID KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4giu:A (ASP293) to (GLN369) BIANTHRANILATE-LIKE ANALOGUE BOUND IN INNER SITE OF ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD). | MAGNESIUM BINDING, PHOPHORIBOSYLPYROPHOSPHATE, PRPP, INHIBITOR COMPLEX, BI-ANTHRANILATE-LIKE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4giu:B (ASP293) to (GLN369) BIANTHRANILATE-LIKE ANALOGUE BOUND IN INNER SITE OF ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD). | MAGNESIUM BINDING, PHOPHORIBOSYLPYROPHOSPHATE, PRPP, INHIBITOR COMPLEX, BI-ANTHRANILATE-LIKE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4gkm:A (ASP293) to (ILE370) BIANTHRANILATE-LIKE ANALOGUE BOUND IN THE OUTER SITE OF ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | MAGNESIUM BINDING, PHOSPHORIBOSYLPYROPHOSPHATE, PRPP, INHIBITOR COMPLEX, BI-ANTHRANILATE-LIKE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4gkm:B (ASP293) to (ILE370) BIANTHRANILATE-LIKE ANALOGUE BOUND IN THE OUTER SITE OF ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) | MAGNESIUM BINDING, PHOSPHORIBOSYLPYROPHOSPHATE, PRPP, INHIBITOR COMPLEX, BI-ANTHRANILATE-LIKE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5ko2:A (MET107) to (GLU180) MOUSE PGP 34 LINKER DELETED MUTANT HG DERIVATIVE | MOUSE PGP, MULTIDRUG RESISTANCE, DRUG TRANSPORT, MERCURY DERIVATIVE, HYDROLASE
5kpd:A (GLU93) to (ILE182) MOUSE PGP 34 LINKER DELETED DOUBLE EQ MUTANT | MULTIDRUG RESISTANCE, ABC TRANSPORTER, MEMBRANE PROTEIN, DRUG EFFLUX, HYDROLASE
5kpd:B (GLU93) to (ILE182) MOUSE PGP 34 LINKER DELETED DOUBLE EQ MUTANT | MULTIDRUG RESISTANCE, ABC TRANSPORTER, MEMBRANE PROTEIN, DRUG EFFLUX, HYDROLASE
5kpi:B (GLU93) to (ILE182) MOUSE NATIVE PGP | MOUSE PGP, MULTIDRUG RESISTANCE, DRUG TRANSPORT, NATIVE, HYDROLASE
5l02:A (ALA503) to (ASN565) S324T VARIANT OF B. PSEUDOMALLEI KATG | CATALASE, PEROXIDASE, KATG, S324T VARIANT, OXIDOREDUCTASE
5l05:A (GLY129) to (GLY181) CRYSTAL STRUCTURE OF CATALASE-PEROXIDASE KATG OF BURKHOLDERIA PSEUDOMALLEI TREATED WITH INH | CATALASE, PEROXIDASE, KATG, OXIDOREDUCTASE
5l05:B (ALA503) to (GLY567) CRYSTAL STRUCTURE OF CATALASE-PEROXIDASE KATG OF BURKHOLDERIA PSEUDOMALLEI TREATED WITH INH | CATALASE, PEROXIDASE, KATG, OXIDOREDUCTASE
5sw4:A (GLY129) to (GLY181) CRYSTAL STRUCTURE OF NATIVE CATALASE-PEROXIDASE KATG AT PH8.0 | CATALASE, PEROXIDASE, PH CHANGE, MOLECULAR SWITCH, OXIDOREDUCTASE
5sw4:A (ALA503) to (GLY567) CRYSTAL STRUCTURE OF NATIVE CATALASE-PEROXIDASE KATG AT PH8.0 | CATALASE, PEROXIDASE, PH CHANGE, MOLECULAR SWITCH, OXIDOREDUCTASE
5sw4:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF NATIVE CATALASE-PEROXIDASE KATG AT PH8.0 | CATALASE, PEROXIDASE, PH CHANGE, MOLECULAR SWITCH, OXIDOREDUCTASE
5sw5:A (ALA503) to (ASN565) CRYSTAL STRUCTURE OF NATIVE CATALASE-PEROXIDASE KATG AT PH7.5 | CATALASE, PEROXIDASE, PH CHANGE, MOLECULAR SWITCH, OXIDOREDUCTASE
5sw5:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF NATIVE CATALASE-PEROXIDASE KATG AT PH7.5 | CATALASE, PEROXIDASE, PH CHANGE, MOLECULAR SWITCH, OXIDOREDUCTASE
5sx0:A (GLY129) to (GLY181) CRYSTAL STRUCTURE OF AN OXOFERRYL SPECIES OF CATALASE-PEROXIDASE KATG AT PH7.5 | CATALASE-PEROXIDASE, KATG, COMPOUND I, OXOFERRYL SPECIES, OXIDOREDUCTASE
5sx0:A (ALA503) to (GLY567) CRYSTAL STRUCTURE OF AN OXOFERRYL SPECIES OF CATALASE-PEROXIDASE KATG AT PH7.5 | CATALASE-PEROXIDASE, KATG, COMPOUND I, OXOFERRYL SPECIES, OXIDOREDUCTASE
5sx0:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF AN OXOFERRYL SPECIES OF CATALASE-PEROXIDASE KATG AT PH7.5 | CATALASE-PEROXIDASE, KATG, COMPOUND I, OXOFERRYL SPECIES, OXIDOREDUCTASE
5sx1:A (ALA503) to (GLY567) CRYSTAL STRUCTURE OF D141E VARIANT OF B. PSEUDOMALLEI KATG | KATG, CATALASE-PEROXIDASE, OXIDOREDUCTASE
5sx1:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF D141E VARIANT OF B. PSEUDOMALLEI KATG | KATG, CATALASE-PEROXIDASE, OXIDOREDUCTASE
5sx2:A (GLY129) to (GLY181) CRYSTAL STRUCTURE OF THE D141E MUTANT OF B. PSEUDOMALLEI KATG AT PH 8.0. | CATALASE-PEROXIDASE, KATG, OXIDOREDUCTASE
5sx2:A (ALA503) to (ASN565) CRYSTAL STRUCTURE OF THE D141E MUTANT OF B. PSEUDOMALLEI KATG AT PH 8.0. | CATALASE-PEROXIDASE, KATG, OXIDOREDUCTASE
5sx2:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF THE D141E MUTANT OF B. PSEUDOMALLEI KATG AT PH 8.0. | CATALASE-PEROXIDASE, KATG, OXIDOREDUCTASE
5sx6:A (ALA503) to (ASN565) CRYSTAL STRUCTURE OF THE CATALASE-PEROXIDASE KATG OF B. PSEUDOMALLEI AT PH 6.5 | CATALASE-PEROXIDASE, PH CHANGES, OXIDOREDUCTASE, KATG
5sx6:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF THE CATALASE-PEROXIDASE KATG OF B. PSEUDOMALLEI AT PH 6.5 | CATALASE-PEROXIDASE, PH CHANGES, OXIDOREDUCTASE, KATG
5sxq:A (ALA503) to (ASN565) CRYSTAL STRUCTURE OF B. PSEUDOMALLEI KATG WITH ISONICOTINIC ACID HYDRAZIDE BOUND | CATALASE-PEROXIDASE, TUBERCULOSIS, ISONIAZID-COMPLEX, OXIDOREDUCTASE, KATG
5sxq:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF B. PSEUDOMALLEI KATG WITH ISONICOTINIC ACID HYDRAZIDE BOUND | CATALASE-PEROXIDASE, TUBERCULOSIS, ISONIAZID-COMPLEX, OXIDOREDUCTASE, KATG
5sxs:A (ALA503) to (ASN565) CRYSTAL STRUCTURE OF CATALASE-PEROXIDASE KATG WITH ISONICOTINIC ACID HYDRAZIDE AND AMP BOUND | CATALASE-PEROXIDASE, TUBERCULOSIS, ISONIAZID, PRO-DRUG ACTIVATION, OXIDOREDUCTASE
5sxs:B (ALA503) to (GLY567) CRYSTAL STRUCTURE OF CATALASE-PEROXIDASE KATG WITH ISONICOTINIC ACID HYDRAZIDE AND AMP BOUND | CATALASE-PEROXIDASE, TUBERCULOSIS, ISONIAZID, PRO-DRUG ACTIVATION, OXIDOREDUCTASE
5sxt:A (ALA503) to (ASN565) CRYSTAL STRUCTURE OF THE S324T VARIANT OF BURKHOLDERIA PSEUDOMALLEI KATG WITH ISONICOTINIC ACID HYDRAZIDE BOUND | CATALASE-PEROXIDASE, S324T VARIANT, ISONIAZID, PRO-DRUG ACTIVATION, TUBERCULOSIS, OXIDOREDUCTASE, KATG
5sxw:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF THE E198A VARIANT OF CATALASE-PEROXIDASE KATG OF BURKHOLDERIA PSEUDOMALLEI | CATALASE-PEROXIDASE, E198A VARIANT, TUBERCULOSIS ISONICOTINIC ACID HYDRAZIDE, OXIDOREDUCTASE, KATG
5sxx:A (ALA503) to (GLY567) CRYSTAL STRUCTURE OF THE E198A VARIANT OF BURKHOLDERIA PSEUDOMALLEI CATALASE-PEROXIDASE KATG WITH INH | CATALASE-PEROXIDASE, ISONIAZID, PRO-DRUG ACTIVATION, TUBERCULOSIS, OXIDOREDUCTASE, KATG
5sxx:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF THE E198A VARIANT OF BURKHOLDERIA PSEUDOMALLEI CATALASE-PEROXIDASE KATG WITH INH | CATALASE-PEROXIDASE, ISONIAZID, PRO-DRUG ACTIVATION, TUBERCULOSIS, OXIDOREDUCTASE, KATG
5syh:A (GLY129) to (GLY181) STRUCTURE OF D141A VARIANT OF B. PSEUDOMALLEI KATG | CATALASE-PEROXIDASE, KATG, D141A VARIANT, OXIDOREDUCTASE
5syh:B (ALA503) to (ASN565) STRUCTURE OF D141A VARIANT OF B. PSEUDOMALLEI KATG | CATALASE-PEROXIDASE, KATG, D141A VARIANT, OXIDOREDUCTASE
5syi:A (ALA503) to (ASN565) STRUCTURE OF D141A VARIANT OF B. PSEUDOMALLEI KATG COMPLEXED WITH INH | CATALASE-PEROXIDASE, KATG, ISONIAZID, D141A VARIANT, OXIDOREDUCTASE
5syi:B (ALA503) to (ASN565) STRUCTURE OF D141A VARIANT OF B. PSEUDOMALLEI KATG COMPLEXED WITH INH | CATALASE-PEROXIDASE, KATG, ISONIAZID, D141A VARIANT, OXIDOREDUCTASE
5syj:A (ALA503) to (GLY567) CRYSTAL STRUCTURE OF THE D141A VARIANT OF B. PSEUDOMALLEI KATGIN COMPLEX WITH ISONIAZID | KATG, CATALASE-PEROXIDASE, OXIDOREDUCTASE, ISONIAZID
5syj:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF THE D141A VARIANT OF B. PSEUDOMALLEI KATGIN COMPLEX WITH ISONIAZID | KATG, CATALASE-PEROXIDASE, OXIDOREDUCTASE, ISONIAZID
5syk:A (ALA503) to (ASN565) CRYSTAL STRUCTURE OF B. PSEUDOMALLEI KATG TREATED WITH HYDROGEN PEROXIDE | CATALASE-PEROXIDASE, KATG, HYDROGEN PEROXIDE, OXIDREDUCTASE, INH, OXIDOREDUCTASE
5syk:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF B. PSEUDOMALLEI KATG TREATED WITH HYDROGEN PEROXIDE | CATALASE-PEROXIDASE, KATG, HYDROGEN PEROXIDE, OXIDREDUCTASE, INH, OXIDOREDUCTASE
5syu:A (ALA503) to (ASN565) CRYSTAL STRUCTURE OF BURKHOLDERIA PSEUDOMALLEI KATG E242Q VARIANT | CATALASE-PEROXIDASE, KATG, E242Q VARIANT, OXIDOREDUCTASE
5syu:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF BURKHOLDERIA PSEUDOMALLEI KATG E242Q VARIANT | CATALASE-PEROXIDASE, KATG, E242Q VARIANT, OXIDOREDUCTASE
5syv:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF BURKHOLDERIA PSEUDOMALLEI KATG N240D VARIANT | CATALASE-PEROXIDASE, KATG, N240D VARIANT, OXIDOREDUCTASE
5syw:A (ALA503) to (ASN565) CRYSTAL STRUCTURE OF BURKHODERIA PSEUDOMALLEI KATG VARIANT Q233E | CATALASE-PEROXIDASE, KATG, Q233E VARIANT, OXIDOREDUCTASE
5syx:A (ALA503) to (GLY567) CRYSTAL STRUCTURE OF BURKHOLDERIA PSEUDOMALLEI KATG VARIANT W139F | CATALASE-PEROXIDASE, KATG W139F VARIANT, OXIDOREDUCTASE
5syx:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF BURKHOLDERIA PSEUDOMALLEI KATG VARIANT W139F | CATALASE-PEROXIDASE, KATG W139F VARIANT, OXIDOREDUCTASE
5syy:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF THE S324G VARIANT OF CATALASE-PEROXIDASE FROM B. PSEUDOMALLEI | CATALASE-PEROXIDASE, KATG, S324G, OXIDOREDUCTASE
2aw6:A (ILE4) to (GLY66) STRUCTURE OF A BACTERIAL PEPTIDE PHEROMONE/RECEPTOR COMPLEX AND ITS MECHANISM OF GENE REGULATION | REPRESSOR, PHEROMONE, DNA BINDING, REGULATORY, TRANSCRIPTION
2aw6:B (ILE4) to (ALA65) STRUCTURE OF A BACTERIAL PEPTIDE PHEROMONE/RECEPTOR COMPLEX AND ITS MECHANISM OF GENE REGULATION | REPRESSOR, PHEROMONE, DNA BINDING, REGULATORY, TRANSCRIPTION
2b2k:B (LEU144) to (THR179) STRUCTURE OF Y104F IDI-1 MUTANT IN COMPLEX WITH EIPP | COMPLEX, ISOMERASE
4x5d:A (GLN295) to (ARG368) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE VARIANT R193A FROM MYCOBACTERIUM TUBERCULOSIS WITH ANTHRANILATE BOUND | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MYCOBACTERIUM TUBERCULOSIS, MAGNESIUM, TRYPTOPHAN, MUTATION, TRANSFERASE, MAGNESIUM BINDING, PHOSPHORIBOSYL PYROPHOSPHATE
3s5i:A (ASN499) to (LYS559) CRYSTAL STRUCTURES OF FALCILYSIN, A M16 METALLOPROTEASE FROM THE MALARIA PARASITE PLASMODIUM FALCIPARUM | M16 METALLOPROTEASE, PEPTIDASE, HYDROLASE
4ij1:A (ALA294) to (ILE370) BIANTHRANILATE-LIKE ANALOGUE BOUND TO ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) IN ABSENCE OF SUBSTRATES. | INHIBITOR COMPLEX, BI-ANTHRANILATE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4ij1:B (ALA294) to (ILE370) BIANTHRANILATE-LIKE ANALOGUE BOUND TO ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (ANPRT; TRPD) IN ABSENCE OF SUBSTRATES. | INHIBITOR COMPLEX, BI-ANTHRANILATE ANALOGUE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PHOSPHORIBOSYLTRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
2ddh:A (LYS549) to (ALA609) CRYSTAL STRUCTURE OF ACYL-COA OXIDASE COMPLEXED WITH 3-OH-DODECANOATE | BETA BARREL, ALPHA UP-DOWN BUNDLE, OXIDOREDUCTASE
1e8z:A (SER1003) to (GLY1079) STRUCTURE DETERMINANTS OF PHOSPHOINOSITIDE 3-KINASE INHIBITION BY WORTMANNIN, LY294002, QUERCETIN, MYRICETIN AND STAUROSPORINE | TRANSFERASE, PHOSPHOINOSITIDE 3-KINASE GAMMA, SECONDARY MESSENGER GENERATION, PI3K, PI 3K, STAUROSPORINE
1e90:A (LEU1004) to (LYS1078) STRUCTURE DETERMINANTS OF PHOSPHOINOSITIDE 3-KINASE INHIBITION BY WORTMANNIN, LY294002, QUERCETIN, MYRICETIN AND STAUROSPORINE | PHOSPHOINOSITIDE 3-KINASE GAMMA, SECONDARY MESSENGER GENERATION, PI3K, PI 3K, MYRICETIN
3tl5:A (SER1003) to (GLY1079) DISCOVERY OF GDC-0980: A POTENT, SELECTIVE, AND ORALLY AVAILABLE CLASS I PHOSPHATIDYLINOSITOL 3-KINASE (PI3K)/MAMMALIAN TARGET OF RAPAMYCIN (MTOR) KINASE INHIBITOR FOR THE TREATMENT OF CANCER | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4yek:A (ASN252) to (LYS321) X-RAY STRUCTURE OF THE THYMIDINE PHOSPHORYLASE FROM SALMONELLA TYPHIMURIUM IN COMPLEX WITH THYMIDINE | THYMIDINE PHOSPHORYLASE, NUCLEOSIDE, METABOLISM, TRANSFERASE
1euz:C (PRO339) to (GLY415) GLUTAMATE DEHYDROGENASE FROM THERMOCOCCUS PROFUNDUS IN THE UNLIGATED STATE | GLUTAMATE, HYPERTHERMOSTABILITY, DOMAIN CLOSURE MOVEMENT, OXIDOREDUCTASE
2tmg:A (ASP337) to (ARG411) THERMOTOGA MARITIMA GLUTAMATE DEHYDROGENASE MUTANT S128R, T158E, N117R, S160E | METABOLIC ROLE, GLUTAMATE, DEHYDROGENASE, MUTANT, OXIDOREDUCTASE
2tmg:B (ASP337) to (ARG411) THERMOTOGA MARITIMA GLUTAMATE DEHYDROGENASE MUTANT S128R, T158E, N117R, S160E | METABOLIC ROLE, GLUTAMATE, DEHYDROGENASE, MUTANT, OXIDOREDUCTASE
2tmg:C (ASP337) to (ARG411) THERMOTOGA MARITIMA GLUTAMATE DEHYDROGENASE MUTANT S128R, T158E, N117R, S160E | METABOLIC ROLE, GLUTAMATE, DEHYDROGENASE, MUTANT, OXIDOREDUCTASE
2tmg:D (ASP337) to (ARG411) THERMOTOGA MARITIMA GLUTAMATE DEHYDROGENASE MUTANT S128R, T158E, N117R, S160E | METABOLIC ROLE, GLUTAMATE, DEHYDROGENASE, MUTANT, OXIDOREDUCTASE
2tmg:E (ASP337) to (ARG411) THERMOTOGA MARITIMA GLUTAMATE DEHYDROGENASE MUTANT S128R, T158E, N117R, S160E | METABOLIC ROLE, GLUTAMATE, DEHYDROGENASE, MUTANT, OXIDOREDUCTASE
2tmg:F (ASP337) to (ARG411) THERMOTOGA MARITIMA GLUTAMATE DEHYDROGENASE MUTANT S128R, T158E, N117R, S160E | METABOLIC ROLE, GLUTAMATE, DEHYDROGENASE, MUTANT, OXIDOREDUCTASE
1f07:C (LYS2221) to (VAL2265) STRUCTURE OF COENZYME F420 DEPENDENT TETRAHYDROMETHANOPTERIN REDUCTASE FROM METHANOBACTERIUM THERMOAUTOTROPHICUM | (BETA, ALPHA)8 BARREL, TIM BARREL, OXIDOREDUCTASE
4yi7:A (SER270) to (GLU345) ANTHRANILATE BOUND AT ACTIVE SITE OF ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE FROM ACINETOBACTER (ANPRT; TRPD) | TRANSFERASE, PHOSPHORIBOSYL BINDING, ANTHRANILATE BOUND
1r0d:B (LEU779) to (ASN865) HIP1R THATCH DOMAIN CORE | ENDOCYTOSIS, ACTIN-BINDING, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, STRUCTURAL PROTEIN
4ywu:B (LEU45) to (MET104) STRUCTURAL INSIGHT INTO THE SUBSTRATE INHIBITION MECHANISM OF NADP+- DEPENDENT SUCCINIC SEMIALDEHYDE DEHYDROGENASE FROM STREPTOCOCCUS PYOGENES | SUCCINIC SEMIALDEHYDE DEHYDROGENASE, STREPTOCOCCUS PYOGENES, SUBSTRATE INHIBITION, ES-COMPLEX STRUCTURE, OXIDOREDUCTASE
1sj2:B (GLY495) to (GLY560) CRYSTAL STRUCTURE OF MYCOBACTERIUM TUBERCULOSIS CATALASE-PEROXIDASE | HOMODIMER, OXIDOREDUCTASE
2g3v:C (ASP35) to (PHE110) CRYSTAL STRUCTURE OF CAGS (HP0534, CAG13) FROM HELICOBACTER PYLORI | HELICOBACTER PYLORI, PATHOGENICITY ISLAND, TYPE IV SECRETION SYSTEM, UNKNOWN FUNCTION
2g47:A (GLU656) to (SER721) CRYSTAL STRUCTURE OF HUMAN INSULIN-DEGRADING ENZYME IN COMPLEX WITH AMYLOID-BETA (1-40) | PROTEIN-PEPTIDE COMPLEX, HYDROLASE
1gxb:A (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE IN COMPLEX WITH PYROPHOSPHATE AND MAGNESIUM | TRANSFERASE, TRYPTOPHANE BIOSYNTHESIS, ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE, PRPP, MG2+, PYROPHOSPHATE
1gxb:B (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE IN COMPLEX WITH PYROPHOSPHATE AND MAGNESIUM | TRANSFERASE, TRYPTOPHANE BIOSYNTHESIS, ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE, PRPP, MG2+, PYROPHOSPHATE
1gxb:C (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE IN COMPLEX WITH PYROPHOSPHATE AND MAGNESIUM | TRANSFERASE, TRYPTOPHANE BIOSYNTHESIS, ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE, PRPP, MG2+, PYROPHOSPHATE
1gxb:D (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE IN COMPLEX WITH PYROPHOSPHATE AND MAGNESIUM | TRANSFERASE, TRYPTOPHANE BIOSYNTHESIS, ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE, PRPP, MG2+, PYROPHOSPHATE
2grl:A (ILE4) to (ALA65) CRYSTAL STRUCTURE OF DCT/ICF10 COMPLEX | RECEPTOR, INHIBITOR, TRANSCRIPTION
2grl:B (ILE4) to (GLY66) CRYSTAL STRUCTURE OF DCT/ICF10 COMPLEX | RECEPTOR, INHIBITOR, TRANSCRIPTION
2grl:C (ILE4) to (GLY66) CRYSTAL STRUCTURE OF DCT/ICF10 COMPLEX | RECEPTOR, INHIBITOR, TRANSCRIPTION
2grl:D (ILE4) to (GLY66) CRYSTAL STRUCTURE OF DCT/ICF10 COMPLEX | RECEPTOR, INHIBITOR, TRANSCRIPTION
3ihy:B (GLN794) to (PHE871) HUMAN PIK3C3 CRYSTAL STRUCTURE | ALPHA/BETA PROTEIN, STRUCTURAL GENOMICS, SGC STOCKHOLM, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, MANGANESE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, TRANSFERASE
2gvq:A (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYL-TRANSFERASE (TRPD) FROM S. SOLFATARICUS IN COMPLEX WITH ANTHRANILATE | PROTEIN-LIGAND COMPLEX, TRANSFERASE
2gvq:B (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYL-TRANSFERASE (TRPD) FROM S. SOLFATARICUS IN COMPLEX WITH ANTHRANILATE | PROTEIN-LIGAND COMPLEX, TRANSFERASE
2gvq:C (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYL-TRANSFERASE (TRPD) FROM S. SOLFATARICUS IN COMPLEX WITH ANTHRANILATE | PROTEIN-LIGAND COMPLEX, TRANSFERASE
2gvq:D (SER265) to (ASN330) ANTHRANILATE PHOSPHORIBOSYL-TRANSFERASE (TRPD) FROM S. SOLFATARICUS IN COMPLEX WITH ANTHRANILATE | PROTEIN-LIGAND COMPLEX, TRANSFERASE
3iyl:B (ASP505) to (LEU584) ATOMIC CRYOEM STRUCTURE OF A NONENVELOPED VIRUS SUGGESTS HOW MEMBRANE PENETRATION PROTEIN IS PRIMED FOR CELL ENTRY | NON-ENVELOPED VIRUS, MEMBRANE PENETRATION PROTEIN, AUTOCLEAVAGE, MYRISTOL GROUP, ICOSAHEDRAL VIRUS, VIRUS
3iyl:D (ASP505) to (LEU584) ATOMIC CRYOEM STRUCTURE OF A NONENVELOPED VIRUS SUGGESTS HOW MEMBRANE PENETRATION PROTEIN IS PRIMED FOR CELL ENTRY | NON-ENVELOPED VIRUS, MEMBRANE PENETRATION PROTEIN, AUTOCLEAVAGE, MYRISTOL GROUP, ICOSAHEDRAL VIRUS, VIRUS
3iyl:F (ASP505) to (LEU584) ATOMIC CRYOEM STRUCTURE OF A NONENVELOPED VIRUS SUGGESTS HOW MEMBRANE PENETRATION PROTEIN IS PRIMED FOR CELL ENTRY | NON-ENVELOPED VIRUS, MEMBRANE PENETRATION PROTEIN, AUTOCLEAVAGE, MYRISTOL GROUP, ICOSAHEDRAL VIRUS, VIRUS
3iyl:H (ASP505) to (LEU584) ATOMIC CRYOEM STRUCTURE OF A NONENVELOPED VIRUS SUGGESTS HOW MEMBRANE PENETRATION PROTEIN IS PRIMED FOR CELL ENTRY | NON-ENVELOPED VIRUS, MEMBRANE PENETRATION PROTEIN, AUTOCLEAVAGE, MYRISTOL GROUP, ICOSAHEDRAL VIRUS, VIRUS
3iyl:J (ASP505) to (LEU584) ATOMIC CRYOEM STRUCTURE OF A NONENVELOPED VIRUS SUGGESTS HOW MEMBRANE PENETRATION PROTEIN IS PRIMED FOR CELL ENTRY | NON-ENVELOPED VIRUS, MEMBRANE PENETRATION PROTEIN, AUTOCLEAVAGE, MYRISTOL GROUP, ICOSAHEDRAL VIRUS, VIRUS
3iyl:L (ASP505) to (LEU584) ATOMIC CRYOEM STRUCTURE OF A NONENVELOPED VIRUS SUGGESTS HOW MEMBRANE PENETRATION PROTEIN IS PRIMED FOR CELL ENTRY | NON-ENVELOPED VIRUS, MEMBRANE PENETRATION PROTEIN, AUTOCLEAVAGE, MYRISTOL GROUP, ICOSAHEDRAL VIRUS, VIRUS
3iyl:P (ASP505) to (LEU584) ATOMIC CRYOEM STRUCTURE OF A NONENVELOPED VIRUS SUGGESTS HOW MEMBRANE PENETRATION PROTEIN IS PRIMED FOR CELL ENTRY | NON-ENVELOPED VIRUS, MEMBRANE PENETRATION PROTEIN, AUTOCLEAVAGE, MYRISTOL GROUP, ICOSAHEDRAL VIRUS, VIRUS
3iyl:R (ASP505) to (LEU584) ATOMIC CRYOEM STRUCTURE OF A NONENVELOPED VIRUS SUGGESTS HOW MEMBRANE PENETRATION PROTEIN IS PRIMED FOR CELL ENTRY | NON-ENVELOPED VIRUS, MEMBRANE PENETRATION PROTEIN, AUTOCLEAVAGE, MYRISTOL GROUP, ICOSAHEDRAL VIRUS, VIRUS
1u2j:A (ALA490) to (GLY545) CRYSTAL STRUCTURE OF THE C-TERMINAL DOMAIN FROM THE CATALASE-PEROXIDASE KATG OF ESCHERICHIA COLI (P21 21 21) | KATG, CATALASE-PEROXIDASE, C-TERMINAL DOMAIN, OXIDOREDUCTASE
1u2j:B (ALA490) to (GLY545) CRYSTAL STRUCTURE OF THE C-TERMINAL DOMAIN FROM THE CATALASE-PEROXIDASE KATG OF ESCHERICHIA COLI (P21 21 21) | KATG, CATALASE-PEROXIDASE, C-TERMINAL DOMAIN, OXIDOREDUCTASE
4lz6:A (ARG89) to (GLU163) STRUCTURE OF MATE MULTIDRUG TRANSPORTER DINF-BH | MULTIDRUG TRANSPORTER, TRANSPORT PROTEIN
4m1c:A (GLU656) to (SER721) CRYSTAL STRUCTURE ANALYSIS OF FAB-BOUND HUMAN INSULIN DEGRADING ENZYME (IDE) IN COMPLEX WITH AMYLOID-BETA (1-40) | HYDROLASE, ZINC METALLOPROTEASE
4m1c:B (GLU656) to (SER721) CRYSTAL STRUCTURE ANALYSIS OF FAB-BOUND HUMAN INSULIN DEGRADING ENZYME (IDE) IN COMPLEX WITH AMYLOID-BETA (1-40) | HYDROLASE, ZINC METALLOPROTEASE
2i2z:A (SER65) to (LYS106) HUMAN SERUM ALBUMIN COMPLEXED WITH MYRISTATE AND ASPIRIN | PLASMA PROTEIN, METAL-BINDING, LIPID-BINDING, LIPID BINDING PROTEIN
4m2s:A (SER92) to (GLU180) CORRECTED STRUCTURE OF MOUSE P-GLYCOPROTEIN BOUND TO QZ59-RRR | ATP-BINDING CASSETTE TRANSPORTER, MULTIDRUG EFFLUX, ADENOSINE TRIPHOSPHATE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4m2s:B (MET91) to (ASP184) CORRECTED STRUCTURE OF MOUSE P-GLYCOPROTEIN BOUND TO QZ59-RRR | ATP-BINDING CASSETTE TRANSPORTER, MULTIDRUG EFFLUX, ADENOSINE TRIPHOSPHATE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4mcw:A (MET322) to (ARG360) METALLO-ENZYME FROM P. MARINA | STRUCTURAL GENOMICS, OXFORD PROTEIN PRODUCTION FACILITY, OPPF, HYDROLASE
4mcw:B (MET322) to (ARG360) METALLO-ENZYME FROM P. MARINA | STRUCTURAL GENOMICS, OXFORD PROTEIN PRODUCTION FACILITY, OPPF, HYDROLASE
1uxq:A (GLY76) to (LYS132) STRUCTURAL BASIS FOR ALLOSTERIC REGULATION AND SUBSTRATE SPECIFICITY OF THE NON-PHOSPHORYLATING GLYCERALDEHYDE-3-PHOSPHATE DEHYDROGENASE (GAPN) FROM THERMOPROTEUS TENAX | GAPN, ALDH, GLUCOSE 1-PHOSPHATE, GLYCOLYSIS, REGULATION, CATALYSIS, OXIDOREDUCTASE
1uxt:A (GLY76) to (LYS132) STRUCTURAL BASIS FOR ALLOSTERIC REGULATION AND SUBSTRATE SPECIFICITY OF THE NON-PHOSPHORYLATING GLYCERALDEHYDE-3-PHOSPHATE DEHYDROGENASE (GAPN) FROM THERMOPROTEUS TENAX | GAPN, ALDH, GLUCOSE 1-PHOSPHATE, NAD, GLYCOLYSIS, REGULATION, CATATYSIS, OXIDOREDUCTASE
2x38:A (ASN949) to (SER1026) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH IC87114. | PHOSPHOINOSITIDE 3-KINASE, ISOFORM-SPECIFIC INHIBITORS, CANCER, TRANSFERASE
2x3w:C (GLU18) to (GLN140) STRUCTURE OF MOUSE SYNDAPIN I (CRYSTAL FORM 2) | ENDOCYTOSIS, N-WASP, DYNAMIN, PACSIN I, TRANSFERASE
2x6i:A (SER854) to (MET933) THE CRYSTAL STRUCTURE OF THE DROSOPHILA CLASS III PI3-KINASE VPS34 IN COMPLEX WITH PIK-90 | TRANSFERASE
4mlb:A (LYS90) to (GLY164) REVERSE POLARITY OF BINDING POCKET SUGGESTS DIFFERENT FUNCTION OF A MOP SUPERFAMILY TRANSPORTER FROM PYROCOCCUS FURIOSUS VC1 (DSM3638) | LIPID TRANSLOCASE, FLIPPASE, MEMBRANE PROTEIN, TRANSPORT PROTEIN
4mlb:C (LEU105) to (GLY164) REVERSE POLARITY OF BINDING POCKET SUGGESTS DIFFERENT FUNCTION OF A MOP SUPERFAMILY TRANSPORTER FROM PYROCOCCUS FURIOSUS VC1 (DSM3638) | LIPID TRANSLOCASE, FLIPPASE, MEMBRANE PROTEIN, TRANSPORT PROTEIN
5anl:A (SER792) to (ALA869) CRYSTAL STRUCTURE OF VPS34 IN COMPLEX WITH (2S)-8-((3R)-3- METHYLMORPHOLIN-4-YL)-1-(3-METHYL-2-OXO- BUTYL)-2-( TRIFLUOROMETHYL)-3,4-DIHYDRO-2H-PYRIMIDO(1,2-A)PYRIMIDIN-6- ONE, PROCESSED WITH THE CRYSTALDIRECT AUTOMATED MOUNTING AND CRYO-COOLING TECHNOLOGY | TRANSFERASE, LIPID KINASE, AUTOMATED CRYSTAL HARVESTING, AUTOMATED CRYO- COOLING, CRYSTALDIRECT
1jn3:A (THR121) to (LYS148) FIDELITY PROPERTIES AND STRUCTURE OF M282L MUTATOR MUTANT OF DNA POLYMERASE: SUBTLE STRUCTURAL CHANGES INFLUENCE THE MECHANISM OF NUCLEOTIDE DISCRIMINATION | DNA POLYMERASE BETA (FRAGMENT), MUTANT, NUCLEOTIDE DISCRIMINATION, TRANSFERASE
5c1r:A (ASP293) to (GLN369) STEREOISOMER OF PRPP BOUND IN THE ACTIVE SITE OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYL (ANPRT; TRPD) | STEREOISOMER OF PRPP, PHOSPHORIBOYSL PYROPHOSPHATE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, MAGNESIUM BINDING, TRANSFERASE, PSI-2, PROTEIN STRUCTURE INITIATIVE
5c1r:B (ASP293) to (ILE370) STEREOISOMER OF PRPP BOUND IN THE ACTIVE SITE OF MYCOBACTERIUM TUBERCULOSIS ANTHRANILATE PHOSPHORIBOSYL (ANPRT; TRPD) | STEREOISOMER OF PRPP, PHOSPHORIBOYSL PYROPHOSPHATE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, MAGNESIUM BINDING, TRANSFERASE, PSI-2, PROTEIN STRUCTURE INITIATIVE
3zw3:A (SER1003) to (GLY1079) FRAGMENT BASED DISCOVERY OF A NOVEL AND SELECTIVE PI3 KINASE INHIBITOR | TRANSFERASE
4ovv:A (ARG975) to (HIS1047) CRYSTAL STRUCTURE OF PI3KALPHA IN COMPLEX WITH DIC4-PIP2 | P110, P85, PI3KCA, PI3K, PIK3R1, PHOSPHATIDILYNOSITOL 3, 4, 5 TRIPHOSPHATE, PIP2, PHOSPHATIDYLINOSITOL 4, 5 BISPHOSPHATE, LIPID KINASE, PHOSPHOINOSITIDE, 3-KINASE, SIGNALING, PHOSPHATIDYLINOSITOL 3-KINASE, TRANSFERASE-TRANSFERASE REGULATOR COMPLEX
4ows:B (ASP293) to (GLN369) ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH 4-METHYLANTHRANILATE, PRPP AND MAGNESIUM | ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE
4owv:A (ASP293) to (GLN369) ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH ANTHRANILATE | ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE
4owv:B (GLN295) to (ILE370) ANTHRANILATE PHOSPHORIBOSYL TRANSFERASE FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH ANTHRANILATE | ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, INHIBITOR, TRANSFERASE
4pae:A (GLY112) to (GLY164) CRYSTAL STRUCTURE OF CATALASE-PEROXIDASE (KATG) W78F MUTANT FROM SYNECHOCOCCUS ELONGATUS PCC7942 | OXIDOREDUCTASE
4pae:A (ALA485) to (GLY541) CRYSTAL STRUCTURE OF CATALASE-PEROXIDASE (KATG) W78F MUTANT FROM SYNECHOCOCCUS ELONGATUS PCC7942 | OXIDOREDUCTASE
5db6:A (THR121) to (LYS148) STRUCTURE OF HUMAN DNA POLYMERASE BETA HOST-GUEST COMPLEX WITH THE N7MG BASE PAIRED WITH A DC | HUMAN DNA POLYMERASE, TRANSFERASE-DNA COMPLEX
5dbb:A (THR121) to (LYS148) STRUCTURE OF HUMAN DNA POLYMERASE BETA HOST-GUEST COMPLEX WITH THE DG BASE PAIRED WITH A DA | HUMAN DNA POLYMERASE, TRANSFERASE-DNA COMPLEX
3l16:A (SER1003) to (LYS1078) DISCOVERY OF (THIENOPYRIMIDIN-2-YL)AMINOPYRIMIDINES AS POTENT, SELECTIVE, AND ORALLY AVAILABLE PAN-PI3-KINASE AND DUAL PAN-PI3- KINASE/MTOR INHIBITORS FOR THE TREATMENT OF CANCER | KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, TRANSFERASE, PI3K-GAMMA P110 GAMMA
4anu:A (SER1003) to (GLY1079) COMPLEXES OF PI3KGAMMA WITH ISOFORM SELECTIVE INHIBITORS. | TRANSFERASE
5ds4:D (LEU213) to (LEU272) CRYSTAL STRUCTURE THE ESCHERICHIA COLI CAS1-CAS2 COMPLEX BOUND TO PROTOSPACER DNA | CRISPR-CAS SYSTEMS, CLUSTERED REGULARLY INTERSPACED SHORT PALINDROMIC REPEATS, INTEGRASES, ENDODEOXYRIBONUCLEASES, ENDONUCLEASES, DNA BINDING PROTEIN, HYDROLASE-DNA COMPLEX
4q4a:A (PHE49) to (ASN152) IMPROVED MODEL OF AMP-PNP BOUND TM287/288 | ABC EXPORTER, MULTIDRUG TRANSPORT, ABC TRANSPORTER, MEMBRANE TRANSPORTER, HYDROLASE-TRANSPORT PROTEIN COMPLEX
5eds:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF HUMAN PI3K-GAMMA IN COMPLEX WITH BENZIMIDAZOLE INHIBITOR 5 | INHIBITOR, PHOSPHOTRANSFERASE, P110, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ejs:A (ASP2166) to (GLN2221) STRUCTURE OF DICTYOSTELIUM DISCOIDEUM MYOSIN VII MYTH4-FERM MF2 DOMAIN, MUTANT 1 | MYOSIN, MOTOR MYOSIN, MYOSIN TAIL, MYTH4-FERM, MOTOR PROTEIN
5ejs:B (ASP2166) to (GLN2221) STRUCTURE OF DICTYOSTELIUM DISCOIDEUM MYOSIN VII MYTH4-FERM MF2 DOMAIN, MUTANT 1 | MYOSIN, MOTOR MYOSIN, MYOSIN TAIL, MYTH4-FERM, MOTOR PROTEIN
4qp7:A (ALA195) to (LEU267) CRYSTAL STRUCTURE OF ERK2 IN COMPLEX WITH 2-(1H-PYRAZOL-4-YL)-5H- PYRROLO[2,3-B]PYRAZINE | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4rid:A (PRO373) to (ARG424) HUMAN FAN1 NUCLEASE | NUCLEASE, HYDROLASE
4rid:B (PRO373) to (ARG424) HUMAN FAN1 NUCLEASE | NUCLEASE, HYDROLASE
4rpx:A (THR121) to (LYS148) PRECATALYTIC TERNARY COMPLEX OF HUMAN DNA POLYMERASE BETA WITH GAPPED DNA CONTAINING AN 8-OXO-7,8-DIHYDRO-GUANINE (8-OXOG) AND DCTP IN THE PRESENCE OF CACL2 | X-FAMILY, POL BETA, TRANSFERASE-DNA COMPLEX
4rq0:A (THR121) to (LYS148) HUMAN DNA POLYMERASE BETA WITH GAPPED DNA CONTAINING AN 8-OXO-7,8- DIHYDRO-GUANINE (8-OXOG)AND DCTP SOAKED WITH MGCL2 FOR 80 S | X-FAMILY, POL BETA, TRANSFERASE-DNA COMPLEX
5gm1:F (SER229) to (LYS276) CRYSTAL STRUCTURE OF METHYLTRANSFERASE TLED COMPLEXED WITH SAH | TLED, TELEOCIDIN, METHYLTRANSFERASES, TERPENE CYCLIZATION, TRANSFERASE
5gm1:L (SER229) to (LYS276) CRYSTAL STRUCTURE OF METHYLTRANSFERASE TLED COMPLEXED WITH SAH | TLED, TELEOCIDIN, METHYLTRANSFERASES, TERPENE CYCLIZATION, TRANSFERASE
4tv3:A (GLU976) to (ASP1045) ISOLATED P110A SUBUNIT OF PI3KA PROVIDES A PLATFORM FOR STRUCTURE- BASED DRUG DESIGN | LIPID KINASE ACTIVITY, ATPASE ACTIVITY, SURFACE PLASMON RESONANCE (SPR), ISOTHERMAL TITRATION CALORIMETRY (ITC)., TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3p2b:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF PI3K GAMMA WITH 3-(2-MORPHOLINO-6-(PYRIDIN-3- YLAMINO)PYRIMIDIN-4-YL)PHENOL | PI3-KINASE P110 SUBUNIT GAMMA, TRANSFERASE, LIPID KINASE, ATP BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5i8r:B (TRP84) to (GLY162) ASMASE WITH ZINC | ACID SPHINGOMYELINASE, OLIPUDASE ALFA, ZINC, HYDROLASE
5i8r:C (TRP84) to (GLY162) ASMASE WITH ZINC | ACID SPHINGOMYELINASE, OLIPUDASE ALFA, ZINC, HYDROLASE
4ezl:A (PRO1004) to (GLY1079) POTENT AND SELECTIVE INHIBITORS OF PI3K-DELTA: OBTAINING ISOFORM SELECTIVITY FROM THE AFFINITY POCKET AND TRYPTOPHAN SHELF | KINASE P110, P110-GAMMA, LIPID KINASE, CYTOPLASMIC, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5j0o:A (THR121) to (LYS148) BINARY COMPLEX CRYSTAL STRUCTURE OF DNA POLYMERASE BETA WITH A:A MISMATCH AT THE PRIMER TERMINUS | DNA POLYMERASE BETA, MISMATCH EXTENSION, BINARY COMPLEX, TRANSFERASE- DNA COMPLEX
4f5o:A (THR121) to (LYS148) OPEN TERNARY COMPLEX OF R283K DNA POLYMERASE BETA WITH A ONE METAL BOUND DCTP ANALOG | TRANSFERASE, LYASE/DNA, LYASE-DNA COMPLEX
4uwk:A (GLU793) to (ALA869) DISCOVERY OF (2S)-8-((3R)-3-METHYLMORPHOLIN-4-YL)-1-(3- METHYL-2-OXO-BUTYL)-2-(TRIFLUOROMETHYL)-3,4-DIHYDRO-2H- PYRIMIDO(1,2-A)PYRIMIDIN-6-ONE: A NOVEL POTENT AND SELECTIVE INHIBITOR OF VPS34 FOR THE TREATMENT OF SOLID TUMORS | TRANSFERASE, LIPID KINASE, AUTOPHAGY INHIBITOR
3qs8:A (GLN295) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS174) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
3qs8:B (ALA294) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS174) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
3qs8:C (GLN295) to (ILE370) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS174) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
3qs8:D (ASP293) to (GLN369) ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE (TRPD) FROM MYCOBACTERIUM TUBERCULOSIS (COMPLEX WITH INHIBITOR ACS174) | ANTHRANILATE PHOSPHORIBOSYLTRANSFERASE, ANTHRANILIC ACIDS, MAGNESIUM, TRYPTOPHAN, MAGNESIUM BINDING PHOSPHORIBOSYL PYROPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, STRUCTURAL GENOMICS, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
4fhj:A (SER1003) to (GLY1079) CRYSTAL STRUCTURE OF PI3K-GAMMA IN COMPLEX WITH IMIDAZOPYRIDINE 2 | INHIBITOR, P110, KINASE, TRANSFERASE, ATP-BINDING, P84, P101, TRANSFERASE-INHIBITOR COMPLEX
5jhy:A (GLY158) to (GLY210) CRYSTAL STRUCTURE OF FUNGAL MAGKATG2 AT PH 5.5 | OXIDOREDUCTASE
5jhy:B (GLY158) to (GLY210) CRYSTAL STRUCTURE OF FUNGAL MAGKATG2 AT PH 5.5 | OXIDOREDUCTASE
5sx3:A (ALA503) to (GLY567) CRYSTAL STRUCTURE OF THE CATALASE-PEROXIDASE KATG OF B. PSEUDOMAALLEI AT PH 4.5 | CATALASE-PEROXIDASE, KATG, PH CHANGES, OXIDOREDUCTASE
5sx3:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF THE CATALASE-PEROXIDASE KATG OF B. PSEUDOMAALLEI AT PH 4.5 | CATALASE-PEROXIDASE, KATG, PH CHANGES, OXIDOREDUCTASE
5sx7:A (ALA503) to (GLY567) CRYSTAL STRUCTURE OF CATALASE-PEROXIDASE KATG OF B. PSEUDOMALLEI AT PH 8.5 | CATALASE-PEROXIDASE, PH CHANGES, KATG OXIDOREDUCTASE, OXIDOREDUCTASE
5sx7:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF CATALASE-PEROXIDASE KATG OF B. PSEUDOMALLEI AT PH 8.5 | CATALASE-PEROXIDASE, PH CHANGES, KATG OXIDOREDUCTASE, OXIDOREDUCTASE
5sxr:B (ALA503) to (ASN565) CRYSTAL STRUCTURE OF B. PSEUDOMALLEI KATG WITH NAD BOUND | CATALASE-PEROXIDASE, TUBERCULOSIS, ISONIAZID NAD, OXIDOREDUCTASE, PRO-DRUG ACTIVATION