1a28:A (LEU687) to (LYS769) HORMONE-BOUND HUMAN PROGESTERONE RECEPTOR LIGAND-BINDING DOMAIN | PROGESTERONE RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION
3e7c:A (VAL533) to (GLN615) GLUCOCORTICOID RECEPTOR LBD BOUND TO GSK866 | GR, GLUCOCORTICOID RECEPTOR, NUCLEAR RECEPTOR, ALTERNATIVE INITIATION, CHROMATIN REGULATOR, DISEASE MUTATION, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, PSEUDOHERMAPHRODITISM, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER, ACTIVATOR
3e7c:B (THR531) to (GLN615) GLUCOCORTICOID RECEPTOR LBD BOUND TO GSK866 | GR, GLUCOCORTICOID RECEPTOR, NUCLEAR RECEPTOR, ALTERNATIVE INITIATION, CHROMATIN REGULATOR, DISEASE MUTATION, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, PSEUDOHERMAPHRODITISM, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER, ACTIVATOR
1a4f:A (PRO37) to (ARG92) BAR-HEADED GOOSE HEMOGLOBIN (OXY FORM) | OXYGEN TRANSPORT, HEME, RESPIRATORY PROTEIN, ERYTHROCYTE
3roc:A (ASN269) to (ALA309) CRYSTAL STRUCTURE OF HUMAN P38 ALPHA COMPLEXED WITH A PYRIMIDINONE COMPOUND | TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gxe:A (ILE52) to (ALA113) T. VULCANUS PHYCOCYANIN CRYSTALLIZED IN 4M UREA | PHOTOSYNTHESIS, LIGHT HARVESTING, UREA DENATURATION, GLOBIN-TYPE, PHOTOSYNTHETIC ANTENNA, N-METHYL ASPARAGINE, PHYCOCYANOBLILIN, THYLAKOID MEMBRANE ATTACHED
3rqe:C (GLY57) to (ARG124) CEREBRAL CAVERNOUS MALFORMATION 3 (CCM3) IN COMPLEX WITH PAXILLIN LD1 | PROTEIN-PEPTIDE COMPLEX, PROTEIN BINDING, FAT DOMAIN, DIMERIZATION, CEREBRAL CAVERNOUS MALFORMATION
3rrw:B (LEU73) to (ASN148) CRYSTAL STRUCTURE OF THE TL29 PROTEIN FROM ARABIDOPSIS THALIANA | CHLOROPLAST THYLAKOID LUMEN, PLANT PROTEIN
2ax6:A (PRO671) to (ASN758) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN T877A MUTANT IN COMPLEX WITH HYDROXYFLUTAMIDE | TRANSCRIPTION
2ax8:A (ILE672) to (ASN758) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN W741L MUTANT IN COMPLEX WITH S-1 | TRANSCRIPTION
2ay1:A (HIS301) to (HIS356) AROMATIC AMINO ACID AMINOTRANSFERASE WITH 4-AMINOHYDROCINNAMIC ACID | AMINOTRANSFERASE
2ay2:A (HIS301) to (HIS356) AROMATIC AMINO ACID AMINOTRANSFERASE WITH CYCLOHEXANE PROPIONIC ACID | AMINOTRANSFERASE
2ay4:A (HIS301) to (HIS356) AROMATIC AMINO ACID AMINOTRANSFERASE WITH 3-(P-TOLYL)PROPIONIC ACID | AMINOTRANSFERASE
1nl3:A (ALA616) to (ILE757) CRYSTAL STRUCTURE OF THE SECA PROTEIN TRANSLOCATION ATPASE FROM MYCOBACTERIUM TUBERCULOSIS IN APO FORM | PREPROTEIN TRANSLOCATION, ATPASE, TRANSMEMBRANE TRANSPORT, HELICASE-LIKE MOTOR DOMAIN, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PROTEIN TRANSPORT
1nl3:B (MET618) to (ALA758) CRYSTAL STRUCTURE OF THE SECA PROTEIN TRANSLOCATION ATPASE FROM MYCOBACTERIUM TUBERCULOSIS IN APO FORM | PREPROTEIN TRANSLOCATION, ATPASE, TRANSMEMBRANE TRANSPORT, HELICASE-LIKE MOTOR DOMAIN, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PROTEIN TRANSPORT
2ay9:A (HIS301) to (HIS356) AROMATIC AMINO ACID AMINOTRANSFERASE WITH 5-PHENYLVALERIC ACID | AMINOTRANSFERASE
2azk:A (LEU220) to (LEU273) CRYSTAL STRUCTURE FOR THE MUTANT W136E OF SULFOLOBUS SOLFATARICUS HEXAPRENYL PYROPHOSPHATE SYNTHASE | HEXPPS, TRANS-PRENYLTRANSFERASE, ISOPRENYL PYROPHOSPHATE SYNTHASE
2b23:B (THR311) to (SER395) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN AND A GLUCOCORTICOID RECEPTOR-INTERACTING PROTEIN 1 NR BOX II PEPTIDE | ESTROGEN RECEPTOR, LBD, GRIP PEPTIDE, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
1noo:A (LEU127) to (THR185) CYTOCHROME P450-CAM COMPLEXED WITH 5-EXO-HYDROXYCAMPHOR | MONOOXYGENASE, OXIDOREDUCTASE (OXYGENASE)
1nvb:B (ASP176) to (ARG222) CRYSTAL STRUCTURE OF 3-DEHYDROQUINATE SYNTHASE (DHQS) IN COMPLEX WITH ZN2+ AND CARBAPHOSPHONATE | SHIKIMATE PATHWAY, AROMATIC AMINO ACID BIOSYNTHESIS, DHQS, CLOSED FORM, FORM C, DOMAIN MOVEMENT, CYCLASE, LYASE
1nvd:A (ASP176) to (ARG223) CRYSTAL STRUCTURE OF 3-DEHYDROQUINATE SYNTHASE (DHQS) IN COMPLEX WITH ZN2+ AND CARBAPHOSPHONATE | SHIKIMATE PATHWAY, AROMATIC AMINO ACID BIOSYNTHESIS, DHQS, OPEN FORM, FORM B, DOMAIN MOVEMENT, CYCLASE, LYASE
1nvd:B (ASP176) to (ARG222) CRYSTAL STRUCTURE OF 3-DEHYDROQUINATE SYNTHASE (DHQS) IN COMPLEX WITH ZN2+ AND CARBAPHOSPHONATE | SHIKIMATE PATHWAY, AROMATIC AMINO ACID BIOSYNTHESIS, DHQS, OPEN FORM, FORM B, DOMAIN MOVEMENT, CYCLASE, LYASE
1ay5:A (HIS301) to (HIS356) AROMATIC AMINO ACID AMINOTRANSFERASE COMPLEX WITH MALEATE | TRANSFERASE, AMINOTRANSFERASE
1ay8:A (HIS301) to (HIS356) AROMATIC AMINO ACID AMINOTRANSFERASE COMPLEX WITH 3-PHENYLPROPIONATE | TRANSFERASE, AMINOTRANSFERASE
3eqx:A (THR27) to (LEU113) CRYSTAL STRUCTURE OF A FIC FAMILY PROTEIN (SO_4266) FROM SHEWANELLA ONEIDENSIS AT 1.6 A RESOLUTION | FIC FAMILY PROTEIN, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, DNA BINDING PROTEIN
3eqx:B (LEU28) to (LEU113) CRYSTAL STRUCTURE OF A FIC FAMILY PROTEIN (SO_4266) FROM SHEWANELLA ONEIDENSIS AT 1.6 A RESOLUTION | FIC FAMILY PROTEIN, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, DNA BINDING PROTEIN
4hgv:A (GLY93) to (MSE146) CRYSTAL STRUCTURE OF A FUMARATE HYDRATASE | NYSGRC, PSI-BIOLOGY, STRUCTURAL GENOMICS, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, SMALL MOLECULE METABOLISM, ENERGY, LYASE
4hi0:A (ALA160) to (GLU224) CRYSTAL STRUCTURE OF HELICOBACTER PYLORI UREASE ACCESSORY PROTEIN UREF/H/G COMPLEX | METALLOCHAPERONE, METAL BINDING PROTEIN, UREASE, CYTOSOL
4hi0:C (ALA160) to (GLU224) CRYSTAL STRUCTURE OF HELICOBACTER PYLORI UREASE ACCESSORY PROTEIN UREF/H/G COMPLEX | METALLOCHAPERONE, METAL BINDING PROTEIN, UREASE, CYTOSOL
1beq:A (TYR16) to (ALA83) INTERACTION BETWEEN PROXIMAL AND DISTALS REGIONS OF CYTOCHROME C PEROXIDASE | PEROXIDASE, OXIDOREDUCTASE
3eyb:B (VAL269) to (ILE347) STRUCTURAL AND FUNCTIONAL INSIGHTS INTO THE LIGAND BINDING DOMAIN OF A NON-DUPLICATED RXR FROM THE INVERTEBRATE CHORDATE AMPHIOXUS | AMPHIOXUS, RETINOID X RECEPTOR, NUCLEAR RECEPTOR, LIGAND BINDING, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER, STRUCTURAL GENOMICS, STRUCTURAL PROTEOMICS IN EUROPE, SPINE
4hjz:A (ASN113) to (ASP170) 1.9 A CRYSTAL STRUCTURE OF E. COLI MLTE-E64Q WITH BOUND CHITOPENTAOSE | GOOSE TYPE LYSOZYME-LIKE STRUCTURE, LYTIC TRANSGLYCOSYLASE, LYASE
4x2c:B (ASN3) to (SER78) CLOSTRIDIUM DIFFICILE FIC PROTEIN_0569 MUTANT S31A, E35A | FIC PROTEIN, A-HELICAL, SE/AA MUTANT, STRUCTURAL PROTEIN
4x2s:A (VAL209) to (VAL274) CRYSTAL STRUCTURE OF 276S/M395R-GLTPH IN INWARD-FACING CONFORMATION | AMINO ACID SECONDARY TRANSPORTERS, SODIUM COUPLED ASPARTATE TRANSPORTER
4x2s:B (TYR204) to (VAL274) CRYSTAL STRUCTURE OF 276S/M395R-GLTPH IN INWARD-FACING CONFORMATION | AMINO ACID SECONDARY TRANSPORTERS, SODIUM COUPLED ASPARTATE TRANSPORTER
4x2s:C (TYR204) to (VAL274) CRYSTAL STRUCTURE OF 276S/M395R-GLTPH IN INWARD-FACING CONFORMATION | AMINO ACID SECONDARY TRANSPORTERS, SODIUM COUPLED ASPARTATE TRANSPORTER
3f0t:B (PRO209) to (ALA294) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH N-METHYL-DHBT | TRANSFERASE, THYMIDINE KINASE, DNA-SYNTHESIS, PET TRACER, ATP- BINDING, DNA SYNTHESIS, EARLY PROTEIN, NUCLEOTIDE-BINDING
4x3n:C (ALA28) to (LYS80) CRYSTAL STRUCTURE OF 34 KDA F-ACTIN BUNDLING PROTEIN FROM DICTYOSTELIUM DISCOIDEUM | ACTIN, CYTOSKELETON, BUNDLING, PROTEIN BINDING
1o9x:A (GLY399) to (THR467) HUMAN SERUM ALBUMIN COMPLEXED WITH TETRADECANOIC ACID (MYRISTIC ACID) AND HEMIN | PLASMA PROTEIN, LIPID-BINDING, FATTY ACID TRANSPORT, HEME- BINDING
2bxi:A (GLY399) to (THR467) HUMAN SERUM ALBUMIN COMPLEXED WITH MYRISTATE AND AZAPROPAZONE | TRANSPORT PROTEIN, ALBUMIN, CARRIER PROTEIN, LIPID-BINDING, METAL-BINDING, DRUG-BINDING, AZAPROPAZONE, MYRISTATE
2bxl:A (GLU400) to (THR467) HUMAN SERUM ALBUMIN COMPLEXED WITH MYRISTATE AND 3,5- DIIODOSALICYLIC ACID | TRANSPORT PROTEIN, ALBUMIN, CARRIER PROTEIN, LIPID-BINDING, METAL-BINDING, DRUG-BINDING, 3, 5-DIIODOSALICYLIC ACID, MYRISTATE
2bxm:A (GLY399) to (THR467) HUMAN SERUM ALBUMIN COMPLEXED WITH MYRISTATE AND INDOMETHACIN | TRANSPORT PROTEIN, ALBUMIN, CARRIER PROTEIN, LIPID-BINDING, METAL-BINDING, DRUG-BINDING, MYRISTATE, INDOMETHACIN
2bxo:A (GLY399) to (THR467) HUMAN SERUM ALBUMIN COMPLEXED WITH MYRISTATE AND OXYPHENBUTAZONE | TRANSPORT PROTEIN, ALBUMIN, CARRIER PROTEIN, LIPID-BINDING, METAL-BINDING, DRUG-BINDING, MYRISTATE, OXYPHENBUTAZONE
2bxp:A (GLU400) to (THR467) HUMAN SERUM ALBUMIN COMPLEXED WITH MYRISTATE AND PHENYLBUTAZONE | ALBUMIN, CARRIER PROTEIN, LIPID-BINDING, PHENYLBUTAZONE, METAL- BINDING, DRUG-BINDING, MYRISTATE, TRANSPORT PROTEIN
2bxq:A (GLU400) to (THR467) HUMAN SERUM ALBUMIN COMPLEXED WITH MYRISTATE, PHENYLBUTAZONE AND INDOMETHACIN | TRANSPORT PROTEIN, ALBUMIN, CARRIER PROTEIN, LIPID-BINDING, METAL-BINDING, DRUG- BINDING, MYRISTATE, PHENYLBUTAZONE, INDOMETHACIN
1ogk:A (SER235) to (ALA277) THE CRYSTAL STRUCTURE OF TRYPANOSOMA CRUZI DUTPASE IN COMPLEX WITH DUDP | DIMER, HYDROLASE
3sf5:A (ALA160) to (LEU225) CRYSTAL STRUCTURE OF HELICOBACTER PYLORI UREASE ACCESSORY PROTEIN UREF/H COMPLEX | UREASE ACCESSORY PROTEIN, UREF, UREH, CHAPERONE
3sf5:C (ALA160) to (GLU224) CRYSTAL STRUCTURE OF HELICOBACTER PYLORI UREASE ACCESSORY PROTEIN UREF/H COMPLEX | UREASE ACCESSORY PROTEIN, UREF, UREH, CHAPERONE
4i5l:B (ASP142) to (GLY187) STRUCTURAL MECHANISM OF TRIMERIC PP2A HOLOENZYME INVOLVING PR70: INSIGHT FOR CDC6 DEPHOSPHORYLATION | EF HAND, PHOSPHATASE, CDC6 (SUBSTRATE), HYDROLASE-TOXIN COMPLEX
4i5l:E (ASN140) to (GLY187) STRUCTURAL MECHANISM OF TRIMERIC PP2A HOLOENZYME INVOLVING PR70: INSIGHT FOR CDC6 DEPHOSPHORYLATION | EF HAND, PHOSPHATASE, CDC6 (SUBSTRATE), HYDROLASE-TOXIN COMPLEX
4i5n:E (VAL141) to (GLY187) STRUCTURAL MECHANISM OF TRIMERIC PP2A HOLOENZYME INVOLVING PR70: INSIGHT FOR CDC6 DEPHOSPHORYLATION | EF HAND, PHOSPHATASE, CDC6 (SUBSTRATE), TRANSFERASE-TOXIN COMPLEX, HYDROLASE-TOXIN COMPLEX
2c4c:B (GLY405) to (TYR483) CRYSTAL STRUCTURE OF THE NADPH-TREATED MONOOXYGENASE DOMAIN OF MICAL | CYTOSKELETON, FAD, FLAVOPROTEIN, LIM DOMAIN, METAL-BINDING, SIGNALING PROTEIN, TRANSPORT
4i6z:A (ASP110) to (GLY197) CRYSTAL STRUCTURE OF THE TRANSCRIPTIONAL REGULATOR TM1030 WITH 24BP DNA OLIGONUCLEOTIDE | STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, PFAM TETR_N, HELIX-TURN-HELIX, TRANSCRIPTIONAL REGULATOR, DNA BINDING, TRANSCRIPTION REGULATOR-DNA COMPLEX
4i6z:B (ASP110) to (GLY197) CRYSTAL STRUCTURE OF THE TRANSCRIPTIONAL REGULATOR TM1030 WITH 24BP DNA OLIGONUCLEOTIDE | STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, PFAM TETR_N, HELIX-TURN-HELIX, TRANSCRIPTIONAL REGULATOR, DNA BINDING, TRANSCRIPTION REGULATOR-DNA COMPLEX
3ftu:A (PRO400) to (LEU448) LEUKOTRIENE A4 HYDROLASE IN COMPLEX WITH DIHYDRORESVERATROL | LEUKOTRIENE A4 HYDROLASE, LTA4H, FRAGMENT CRYSTALLOGRAPHY, FRAGMENTS OF LIFE, FOL, RESVERATROL, ALTERNATIVE SPLICING, CYTOPLASM, HYDROLASE, LEUKOTRIENE BIOSYNTHESIS, METAL- BINDING, METALLOPROTEASE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, PROTEASE, ZINC
3sqg:A (LEU297) to (GLY373) CRYSTAL STRUCTURE OF A METHYL-COENZYME M REDUCTASE PURIFIED FROM BLACK SEA MATS | ANAEROBIC METHANE OXIDATION, TRANSFERASE
3sqg:B (VAL192) to (GLY255) CRYSTAL STRUCTURE OF A METHYL-COENZYME M REDUCTASE PURIFIED FROM BLACK SEA MATS | ANAEROBIC METHANE OXIDATION, TRANSFERASE
3sqg:E (VAL192) to (GLY255) CRYSTAL STRUCTURE OF A METHYL-COENZYME M REDUCTASE PURIFIED FROM BLACK SEA MATS | ANAEROBIC METHANE OXIDATION, TRANSFERASE
3sqg:G (LEU297) to (GLY373) CRYSTAL STRUCTURE OF A METHYL-COENZYME M REDUCTASE PURIFIED FROM BLACK SEA MATS | ANAEROBIC METHANE OXIDATION, TRANSFERASE
3ftz:A (GLY399) to (LEU448) LEUKOTRIENE A4 HYDROLASE IN COMPLEX WITH FRAGMENT 2-(PYRIDIN-3- YLMETHOXY)ANILINE | LEUKOTRIENE A4 HYDROLASE, LTA4H, FRAGMENT CRYSTALLOGRAPHY, FRAGMENTS OF LIFE, FOL, HYDROLASE-HYDROLASE INHIBITOR COMPLEX, LEUKOTRIENE BIOSYNTHESIS, METAL-BINDING, METALLOPROTEASE, MULTIFUNCTIONAL ENZYME, PROTEASE
3fu6:A (GLY399) to (LEU448) LEUKOTRIENE A4 HYDROLASE IN COMPLEX WITH FRAGMENT (4- THIOPHEN-2-YLPHENYL)METHANAMINE | LEUKOTRIENE A4 HYDROLASE, LTA4H, FRAGMENT CRYSTALLOGRAPHY, FRAGMENTS OF LIFE, FOL, ALTERNATIVE SPLICING, CYTOPLASM, HYDROLASE, LEUKOTRIENE BIOSYNTHESIS, METAL-BINDING, METALLOPROTEASE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, PROTEASE, ZINC
3fuf:A (PRO400) to (LEU448) LEUKOTRIENE A4 HYDROLASE IN COMPLEX WITH FRAGMENT 5- FLUOROINDOLE AND BESTATIN | LEUKOTRIENE A4 HYDROLASE, LTA4H, FRAGMENT CRYSTALLOGRAPHY, FRAGMENTS OF LIFE, FOL, ALTERNATIVE SPLICING, CYTOPLASM, HYDROLASE, LEUKOTRIENE BIOSYNTHESIS, METAL-BINDING, METALLOPROTEASE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, PROTEASE, ZINC
3fuj:A (PRO400) to (LEU448) LEUKOTRIENE A4 HYDROLASE IN COMPLEX WITH 5-[2-(1H-PYRROL-1- YL)ETHOXY]-1H-INDOLE | LEUKOTRIENE A4 HYDROLASE, LTA4H, FRAGMENT CRYSTALLOGRAPHY, FRAGMENTS OF LIFE, FOL, ALTERNATIVE SPLICING, CYTOPLASM, HYDROLASE, LEUKOTRIENE BIOSYNTHESIS, METAL-BINDING, METALLOPROTEASE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, PROTEASE, ZINC
3g0w:A (ILE672) to (THR755) CRYSTAL STRUCTURE OF THE RAT ANDROGEN RECEPTOR LIGAND BINDING DOMAIN COMPLEX WITH AN N-ARYL-OXAZOLIDIN 2-IMINE INHIBITOR | ANDROGEN RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, LIGAND-BINDING DOMAIN, DISEASE MUTATION, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, UBL CONJUGATION, ZINC, ZINC-FINGER, HORMONE/GROWTH FACTOR COMPLEX
3g1q:A (THR135) to (LEU208) CRYSTAL STRUCTURE OF STEROL 14-ALPHA DEMETHYLASE (CYP51) FROM TRYPANOSOMA BRUCEI IN LIGAND FREE STATE | STEROL 14-ALPHA DEMETHYLASE, CYP51, CYTOCHROME P450, HEME, OXIDOREDUCTASE, MONOOXYGENASE, MEMBRANE PROTEIN, STEROL BIOSYNTHESIS
3g1q:C (PHE142) to (SER206) CRYSTAL STRUCTURE OF STEROL 14-ALPHA DEMETHYLASE (CYP51) FROM TRYPANOSOMA BRUCEI IN LIGAND FREE STATE | STEROL 14-ALPHA DEMETHYLASE, CYP51, CYTOCHROME P450, HEME, OXIDOREDUCTASE, MONOOXYGENASE, MEMBRANE PROTEIN, STEROL BIOSYNTHESIS
2qd9:A (ASN269) to (ALA309) P38 ALPHA MAP KINASE INHIBITOR BASED ON HETEROBICYCLIC SCAFFOLDS | SERINE/THREONINE-PROTEIN KINASE, KINASE, TRANSFERASE, P38 MAP KINASE
1p93:A (THR531) to (ARG614) CRYSTAL STRUCTURE OF THE AGONIST FORM OF GLUCOCORTICOID RECEPTOR | PROTIEN-LIGAND COMPLEX, ANTI PARALLEL ALPHA HELIX SANDWICH, HORMONE RECEPTOR
1p93:B (THR531) to (ARG614) CRYSTAL STRUCTURE OF THE AGONIST FORM OF GLUCOCORTICOID RECEPTOR | PROTIEN-LIGAND COMPLEX, ANTI PARALLEL ALPHA HELIX SANDWICH, HORMONE RECEPTOR
1p93:D (THR531) to (ARG614) CRYSTAL STRUCTURE OF THE AGONIST FORM OF GLUCOCORTICOID RECEPTOR | PROTIEN-LIGAND COMPLEX, ANTI PARALLEL ALPHA HELIX SANDWICH, HORMONE RECEPTOR
4il3:B (GLN120) to (ASN222) CRYSTAL STRUCTURE OF S. MIKATAE STE24P | MEMBRANE PROTEIN, ALPHA HELICAL, CAAX PROTEASE, A-FACTOR, STRUCTURAL GENOMICS, MPSBC, PSI-BIOLOGY, MEMBRANE PROTEIN STRUCTURAL BIOLOGY CONSORTIUM, HYDROLASE
1phf:A (LEU127) to (THR185) CRYSTAL STRUCTURES OF METYRAPONE-AND PHENYLIMIDAZOLE- INHIBITED COMPLEXES OF CYTOCHROME P450-CAM | OXIDOREDUCTASE(OXYGENASE)
2qmq:A (GLY177) to (ALA224) CRYSTAL STRUCTURE OF A N-MYC DOWNSTREAM REGULATED 2 PROTEIN (NDRG2, SYLD, NDR2, AI182517, AU040374) FROM MUS MUSCULUS AT 1.70 A RESOLUTION | ALPHA/BETA-HYDROLASES FOLD, NDR FAMILY, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, NEUROGENESIS, PHOSPHORYLATION, REGULATORY PROTEIN, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, SIGNALING PROTEIN
4iui:B (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DYNAMIC WAY DERIVATIVE, 4A | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, NUCLEUS, TRANSCRIPTION
3t5n:A (PRO180) to (PRO227) 1.8A CRYSTAL STRUCTURE OF LASSA VIRUS NUCLEOPROTEIN IN COMPLEX WITH SSRNA | SSRNA, SINGLE STRANDED RNA, VIRAL PROTEIN-RNA COMPLEX
4ivp:B (GLU210) to (ALA294) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH IN51/20 | DNA SYNTHESIS, PET IMAGING TRACER, ATP BINDING, NUCLEOTIDE BINDING, TRANSFERASE
4ivq:A (PRO209) to (ALA294) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH IN43/5 | DNA SYNTHESIS, PET IMAGING TRACER, ATP BINDING, NUCLEOTIDE BINDING, TRANSFERASE
4ivr:A (PRO209) to (SER263) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH IN52/10 | DNA SYNTHESIS, PET IMAGING TRACER, ATP BINDING, NUCLEOTIDE BINDING, TRANSFERASE
4ivr:B (GLU210) to (LEU262) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH IN52/10 | DNA SYNTHESIS, PET IMAGING TRACER, ATP BINDING, NUCLEOTIDE BINDING, TRANSFERASE
4iwc:A (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A DYNAMIC THIOPHENE-DERIVATIVE | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, TRANSCRIPTION
2qti:A (SER8) to (LEU73) CRYSTAL STRUCTURE OF THE UPF0352 PROTEIN SO_2176 FROM SHEWANELLA ONEIDENSIS. NESG TARGET SOR77. | Y2176_SHEON, UPF0352, SO_2176, PF07208, NESG, SOR77, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, UNKNOWN FUNCTION
2cyd:C (MET1) to (LEU80) CRYSTAL STRUCTURE OF LITHIUM BOUND ROTOR RING OF THE V-ATPASE FROM ENTEROCOCCUS HIRAE | NTPK, V-ATPASE, NA(+)-ATPASE, LITHIUM, PROTEOLIPID, ENTEROCOCCUS, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, HYDROLASE
2cyd:F (MET1) to (LEU80) CRYSTAL STRUCTURE OF LITHIUM BOUND ROTOR RING OF THE V-ATPASE FROM ENTEROCOCCUS HIRAE | NTPK, V-ATPASE, NA(+)-ATPASE, LITHIUM, PROTEOLIPID, ENTEROCOCCUS, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, HYDROLASE
2quy:A (ALA214) to (ASN260) TRUNCATED MUTANT ASN175ALA OF PENICILLIN V ACYLASE FROM BACILLUS SPHAERICUS | PENICILLIN, AUTOPROTEOLYSIS, NTN, OXY-ANION HOLE, ANTIBIOTIC RESISTANCE, HYDROLASE, ZYMOGEN
2quy:B (ALA214) to (ASN260) TRUNCATED MUTANT ASN175ALA OF PENICILLIN V ACYLASE FROM BACILLUS SPHAERICUS | PENICILLIN, AUTOPROTEOLYSIS, NTN, OXY-ANION HOLE, ANTIBIOTIC RESISTANCE, HYDROLASE, ZYMOGEN
2quy:C (ALA214) to (ASN260) TRUNCATED MUTANT ASN175ALA OF PENICILLIN V ACYLASE FROM BACILLUS SPHAERICUS | PENICILLIN, AUTOPROTEOLYSIS, NTN, OXY-ANION HOLE, ANTIBIOTIC RESISTANCE, HYDROLASE, ZYMOGEN
2quy:D (ALA214) to (ASN260) TRUNCATED MUTANT ASN175ALA OF PENICILLIN V ACYLASE FROM BACILLUS SPHAERICUS | PENICILLIN, AUTOPROTEOLYSIS, NTN, OXY-ANION HOLE, ANTIBIOTIC RESISTANCE, HYDROLASE, ZYMOGEN
2quy:F (ALA214) to (ASN260) TRUNCATED MUTANT ASN175ALA OF PENICILLIN V ACYLASE FROM BACILLUS SPHAERICUS | PENICILLIN, AUTOPROTEOLYSIS, NTN, OXY-ANION HOLE, ANTIBIOTIC RESISTANCE, HYDROLASE, ZYMOGEN
2quy:G (ALA214) to (ASN260) TRUNCATED MUTANT ASN175ALA OF PENICILLIN V ACYLASE FROM BACILLUS SPHAERICUS | PENICILLIN, AUTOPROTEOLYSIS, NTN, OXY-ANION HOLE, ANTIBIOTIC RESISTANCE, HYDROLASE, ZYMOGEN
2quy:H (ALA214) to (ASN260) TRUNCATED MUTANT ASN175ALA OF PENICILLIN V ACYLASE FROM BACILLUS SPHAERICUS | PENICILLIN, AUTOPROTEOLYSIS, NTN, OXY-ANION HOLE, ANTIBIOTIC RESISTANCE, HYDROLASE, ZYMOGEN
2qvw:A (SER698) to (GLN749) STRUCTURE OF GIARDIA DICER REFINED AGAINST TWINNED DATA | DICER, RNAI,PSEUDO-MEROHEDRAL TWIN, HYDROLASE
2qvw:B (SER698) to (GLN749) STRUCTURE OF GIARDIA DICER REFINED AGAINST TWINNED DATA | DICER, RNAI,PSEUDO-MEROHEDRAL TWIN, HYDROLASE
2qvw:D (SER698) to (GLN749) STRUCTURE OF GIARDIA DICER REFINED AGAINST TWINNED DATA | DICER, RNAI,PSEUDO-MEROHEDRAL TWIN, HYDROLASE
1e2h:B (ASP211) to (LEU262) THE NUCLEOSIDE BINDING SITE OF HERPES SIMPLEX TYPE 1 THYMIDINE KINASE ANALYZED BY X-RAY CRYSTALLOGRAPHY | TRANSFERASE, ADENINE ANALOG, ENZYME-PRODRUG GENE THERAPY, NUCLEOSIDE- BINDING, THYMIDINE KINASE, X-RAY CRYSTALLOGRAPHY
1e2i:B (PRO209) to (LEU262) THE NUCLEOSIDE BINDING SITE OF HERPES SIMPLEX TYPE 1 THYMIDINE KINASE ANALYZED BY X-RAY CRYSTALLOGRAPHY | TRANSFERASE, ADENINE ANALOG, ENZYME-PRODRUG GENE THERAPY, NUCLEOSIDE- BINDING, THYMIDINE KINASE, X-RAY CRYSTALLOGRAPHY
1e2j:B (PRO209) to (ALA294) THE NUCLEOSIDE BINDING SITE OF HERPES SIMPLEX TYPE 1 THYMIDINE KINASE ANALYZED BY X-RAY CRYSTALLOGRAPHY | TRANSFERASE, ADENINE ANALOG, ENZYME-PRODRUG GENE THERAPY, NUCLEOSIDE- BINDING, THYMIDINE KINASE, X-RAY CRYSTALLOGRAPHY
1e2k:B (ASP211) to (ALA294) KINETICS AND CRYSTAL STRUCTURE OF THE WILD-TYPE AND THE ENGINEERED Y101F MUTANT OF HERPES SIMPLEX VIRUS TYPE 1 THYMIDINE KINASE INTERACTING WITH (NORTH)-METHANOCARBA-THYMIDINE | TRANSFERASE, THYMIDINE KINASE, ANTIVIRAL DRUG, ENZYME-PRODRUG GENE THERAPY, X-RAY STRUCTURE, SUGAR RING PUCKER
1e2n:B (PRO209) to (LEU262) HPT + HMTT | TRANSFERASE, NULL
1e3k:A (PRO686) to (LYS769) HUMAN PROGESTERON RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH THE LIGAND METRIBOLONE (R1881) | HUMAN PROGESTERONE RECEPTOR, LIGAND BINDING DOMAIN
2d96:A (GLY13) to (THR53) SOLUTION STRUCTURE OF THE DEATH DOMAIN OF NUCLEAR FACTOR NF- KAPPA-B P100 | SIX HELIX BUNDLE, PROCESSING, PROTEASOME, SIGNAL TRANSDUCTION, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, TRANSCRIPTION
2db4:I (MET1) to (LEU61) CRYSTAL STRUCTURE OF ROTOR RING WITH DCCD OF THE V- ATPASE FROM ENTEROCOCCUS HIRAE | NTPK, V-ATPASE, NA(+)-ATPASE, DCCD, PROTEOLIPID, ENTEROCOCCUS HIRAE, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, HYDROLASE
2dbt:A (THR238) to (GLY285) CRYSTAL STRUCTURE OF CHITINASE C FROM STREPTOMYCES GRISEUS HUT6037 | FAMILY 19 CHITINASE, HYDROLASE
2r40:A (ILE210) to (LEU302) CRYSTAL STRUCTURE OF 20E BOUND ECR/USP | NUCLEAR RECEPTOR LIGAND-BINDING DOMAIN, ANTI-PARALLEL ALPHA-HELICAL SANDWICH, ECDYSONE RECEPTOR, ECR, GENE REGULATION
1e6v:A (PRO285) to (TYR361) METHYL-COENZYME M REDUCTASE FROM METHANOPYRUS KANDLERI | BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE, NI ENZYME
1e6v:D (PRO285) to (TYR361) METHYL-COENZYME M REDUCTASE FROM METHANOPYRUS KANDLERI | BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE, NI ENZYME
4j5w:C (VAL232) to (SER317) CRYSTAL STRUCTURE OF THE APO-PXR/RXRALPHA LBD HETEROTETRAMER COMPLEX | PREGNANE X RECEPTOR, RETINOID X RECEPTOR ALPHA, LIGAND BINDING DOMAIN, NUCLEAR RECEPTOR, ALPHA HELICAL SANDWICH, UNIQUE INTERMOLECULAR BETA-SHEET DIMERIZATION, XENOBIOTIC SENSING, UPREGULATION OF DRUG METABOLISM ENZYMES, RETINOIC ACID-BINDING PROTEIN
2r70:A (GLY420) to (VAL465) CRYSTAL STRUCTURE OF INFECTIOUS BURSAL DISEASE VIRUS VP1 POLYMERASE, COCRYSTALLIZED WITH AN OLIGOPEPTIDE MIMICKING THE VP3 C-TERMINUS. | IBDV, INFECTIOUS BURSAL DISEASE VIRUS, BIRNAVIRUS, POLYMERASE, VP1, VP3, ACTIVATION, TRANSFERASE
4ja4:A (TYR125) to (THR219) INWARD OPEN CONFORMATION OF THE XYLOSE TRANSPORTER XYLE FROM E. COLI | MFS GENERAL SUBSTRATE TRANSPORTER, XYLOSE TRANSPORTER, TRANSPORT PROTEIN
4ja4:B (TYR125) to (THR219) INWARD OPEN CONFORMATION OF THE XYLOSE TRANSPORTER XYLE FROM E. COLI | MFS GENERAL SUBSTRATE TRANSPORTER, XYLOSE TRANSPORTER, TRANSPORT PROTEIN
3tik:A (PHE142) to (LEU208) STEROL 14-ALPHA DEMETHYLASE (CYP51) FROM TRYPANOSOMA BRUCEI IN COMPLEX WITH THE TIPIFARNIB DERIVATIVE 6-((4-CHLOROPHENYL)(METHOXY)(1-METHYL- 1H-IMIDAZOL-5-YL)METHYL)-4-(2,6-DIFLUOROPHENYL)-1-METHYLQUINOLIN- 2(1H)-ONE | STEROL 14-ALPHA DEMETHYLASE, CYP51, HEME, MONOOXYGENASE, STEROL BIOSYNTHESIS, CYTOCHROME P450 FOLD, OXIDOREDUCTASE, CYTOCHROME P450 REDUCTASE, ENDOPLASMIC RETICULUM MEMBRANE
4jbv:A (ASP324) to (ASP415) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1268 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jbx:B (PRO209) to (LEU262) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH SK-78 | DNA SYNTHESIS, PET IMAGING TRACER, ATP BINDING, NUCLEOTIDE BINDING, TRANSFERASE
4jby:B (PRO209) to (LEU262) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH F-SK78 | DNA SYNTHESIS, PET IMAGING TRACER, ATP BINDING, NUCLEOTIDE BINDING, TRANSFERASE
2dqb:B (HIS310) to (GLY350) CRYSTAL STRUCTURE OF DNTP TRIPHOSPHOHYDROLASE FROM THERMUS THERMOPHILUS HB8, WHICH IS HOMOLOGOUS TO DGTP TRIPHOSPHOHYDROLASE | DNTPASE, DNTP, TRIPHOSPHOHYDROLASE, SINGLE-STRANDED DNA, DNA, DGTPASE, HD SUPERFAMILY, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, HYDROLASE, DNA BINDING PROTEIN
3gw9:A (PHE142) to (LEU208) CRYSTAL STRUCTURE OF STEROL 14-ALPHA DEMETHYLASE (CYP51) FROM TRYPANOSOMA BRUCEI BOUND TO AN INHIBITOR N-(1-(2,4- DICHLOROPHENYL)-2-(1H-IMIDAZOL-1-YL)ETHYL)-4-(5-PHENYL-1,3, 4-OXAZIAZOL-2-YL)BENZAMIDE | STEROL 14ALPHA-DEMETHYLASE, CYP51, CYTOCHROME P450, HEME, OXIDOREDUCTASE, MONOOXYGENASE, STEROL BIOSYNTHESIS, LIPIDS, ENDOPLASMIC RETICULUM, IRON, HEME-THIOLATE PROTEIN
3gw9:B (PHE139) to (LEU208) CRYSTAL STRUCTURE OF STEROL 14-ALPHA DEMETHYLASE (CYP51) FROM TRYPANOSOMA BRUCEI BOUND TO AN INHIBITOR N-(1-(2,4- DICHLOROPHENYL)-2-(1H-IMIDAZOL-1-YL)ETHYL)-4-(5-PHENYL-1,3, 4-OXAZIAZOL-2-YL)BENZAMIDE | STEROL 14ALPHA-DEMETHYLASE, CYP51, CYTOCHROME P450, HEME, OXIDOREDUCTASE, MONOOXYGENASE, STEROL BIOSYNTHESIS, LIPIDS, ENDOPLASMIC RETICULUM, IRON, HEME-THIOLATE PROTEIN
2drd:B (VAL904) to (SER992) CRYSTAL STRUCTURE OF A MULTIDRUG TRANSPORTER REVEAL A FUNCTIONALLY ROTATING MECHANISM | MEMBRANE TRANSPORTER, MEMBRANE PROTEIN, MULTIDRUG EFFLUX, DRUG RESISTANCE, TRANSPORTER, EXPORTER, ANTIPORTER
3h0d:A (GLU78) to (TYR129) CRYSTAL STRUCTURE OF CTSR IN COMPLEX WITH A 26BP DNA DUPLEX | PROTEIN DNA COMPLEX, WINGED HTH DOMAIN, 4-HELIX BUNDLE, DNA TANDEM REPEAT, TRANSCRIPTION/DNA COMPLEX
3h0d:B (SER77) to (TYR129) CRYSTAL STRUCTURE OF CTSR IN COMPLEX WITH A 26BP DNA DUPLEX | PROTEIN DNA COMPLEX, WINGED HTH DOMAIN, 4-HELIX BUNDLE, DNA TANDEM REPEAT, TRANSCRIPTION/DNA COMPLEX
1qhi:B (GLU210) to (LEU262) HERPES SIMPLEX VIRUS TYPE-I THYMIDINE KINASE COMPLEXED WITH A NOVEL NON-SUBSTRATE INHIBITOR, 9-(4-HYDROXYBUTYL)-N2- PHENYLGUANINE | TRANSFERASE, TRANSFERASE (PHOSPHOTRANSFERASE) THYMIDINE, TRANSFERASE (PHOSPHOTRANSFERASE) THYMIDINE KINASE; VIRIDAE; DS-DNA ENVELOPED VIRUSES; HERPESVIRIDAE; ALPHAHERPESVIRINAE NOVEL INHIBITOR
3tx7:B (GLU315) to (VAL396) CRYSTAL STRUCTURE OF LRH-1/BETA-CATENIN COMPLEX | LRH-1, BETA-CATENIN, ARMADILLO REPEAT, NUCLEAR RECEPTOR LIGAND BINDING DOMAIN, PROTEIN BINDING
4jr7:A (PRO318) to (ALA364) CRYSTAL STRUCTURE OF SCCK2 ALPHA IN COMPLEX WITH GMPPNP | PROTEIN KINASE, PROTEIN PHOSPHORYLATION, TRANSFERASE
4yi9:A (LEU102) to (GLY160) CRYSTAL STRUCTURE OF NON-MYRISTOYLATED E153A RECOVERIN AT 1.35 A RESOLUTION WITH A SODIUM ION BOUND TO EF-HAND 2 AND CALCIUM ION BOUND TO EF-HAND 3 | CALCIUM BINDING PROTEIN, EF HAND, NCS FAMILY
1qvr:B (THR522) to (LYS558) CRYSTAL STRUCTURE ANALYSIS OF CLPB | COILED COIL, AAA ATPASE, CHAPERONE
3hd6:A (PRO148) to (SER237) CRYSTAL STRUCTURE OF THE HUMAN RHESUS GLYCOPROTEIN RHCG | AMMONIA, CHANNEL, RHESUS, GLYCOPROTEIN, TRANSPORTER, MEMBRANE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, CENTER FOR STRUCTURES OF MEMBRANE PROTEINS, CSMP, AMMONIA TRANSPORT, CELL MEMBRANE, TRANSMEMBRANE, TRANSPORT, MEMBRANE PROTEIN, TRANSPORT PROTEIN
1fc3:A (LYS141) to (TYR197) THE CRYSTAL STRUCTURE OF TRANS-ACTIVATION DOMAIN OF THE SPORULATION RESPONSE REGULATOR, SPO0A | RESPONSE REGULATOR, SIGNALING PROTEIN
1fc3:B (LYS141) to (TYR197) THE CRYSTAL STRUCTURE OF TRANS-ACTIVATION DOMAIN OF THE SPORULATION RESPONSE REGULATOR, SPO0A | RESPONSE REGULATOR, SIGNALING PROTEIN
1fc3:C (LYS141) to (TYR197) THE CRYSTAL STRUCTURE OF TRANS-ACTIVATION DOMAIN OF THE SPORULATION RESPONSE REGULATOR, SPO0A | RESPONSE REGULATOR, SIGNALING PROTEIN
2uza:A (ASP545) to (LYS594) CRYSTAL STRUCTURE OF THE FREE RADICAL INTERMEDIATE OF PYRUVATE:FERREDOXIN OXIDOREDUCTASE FROM DESULFOVIBRIO AFRICANUS | TPP-DEPENDENT ENZYME, PYRUVATE CATABOLISM, OXIDOREDUCTASE, ELECTRON TRANSPORT
4yru:D (ASP44) to (LEU110) CRYSTAL STRUCTURE OF C-TERMINALLY TRUNCATED NEURONAL CALCIUM SENSOR (NCS-1) FROM RATTUS NORVEGICUS | EF-HAND, CALCIUM SENSOR, C-TERMINAL TRUNCATION, SIGNALING PROTEIN
4yrw:A (GLY915) to (GLU990) RAT XANTHINE OXIDOREDUCTASE, C-TERMINAL DELETION PROTEIN VARIANT | XANTHINE OXIDOREDUCTASE, XANTHINE OXIDASE, XANTHINE DEHYDROGENASE, D/O CONVERSION, OXIDOREDUCTASE
4ys0:A (HIS616) to (GLY743) CONFORMATIONAL CHANGES OF THE CLAMP OF THE PROTEIN TRANSLOCATION ATPASE SECA FROM THERMOTOGA MARITIMA | PROTEIN TRANSLOCATION, SECA, ATPASE, PROTEIN TRANSPORT
2ewp:B (ILE237) to (SER317) CRYSTAL STRUCTURE OF ESTROGEN RELATED RECEPTOR-3 (ERR-GAMMA) LIGAND BINDING DOMAIND WITH TAMOXIFEN ANALOG GSK5182 | TAMOXIFEN, ERR, ESTROGEN RELATED RECEPTOR, ORPHAN RECEPTOR, TRANSCRIPTION
4yty:A (GLY916) to (GLU990) STRUCTURE OF RAT XANTHINE OXIDOREDUCTASE, C535A/C992R/C1324S, NADH BOUND FORM | XANTHINE OXIDOREDUCTASE, XANTHINE OXIDASE, XANTHINE DEHYDROGENASE, D/O CONVERSION, OXIDOREDUCTASE
1rec:A (LEU102) to (GLY160) THREE-DIMENSIONAL STRUCTURE OF RECOVERIN, A CALCIUM SENSOR IN VISION | CALCIUM-BINDING PROTEIN
1req:A (GLY242) to (LEU284) METHYLMALONYL-COA MUTASE | ISOMERASE, MUTASE, INTRAMOLECULAR TRANSFERASE
4ytz:B (MET920) to (GLU990) RAT XANTHINE OXIDOREDUCTASE, C-TERMINAL DELETION PROTEIN VARIANT, CRYSTAL GROWN WITHOUT DITHIOTHREITOL | XANTHINE OXIDOREDUCTASE, XANTHINE OXIDASE, XANTHINE DEHYDROGENASE, D/O CONVERSION, OXIDOREDUCTASE
4k8v:A (SER420) to (LEU507) STRUCTURE OF CYCLIC GMP-AMP SYNTHASE (CGAS) | NUCLEOTIDYLTRANSFERASE, DNA, TRANSFERASE
3una:A (GLY915) to (GLU990) CRYSTAL STRUCTURE OF BOVINE MILK XANTHINE DEHYDROGENASE WITH NAD BOUND | XANTHINE DEHYDROGENASE, OXIDOREDUCTASE
1g3i:B (GLU82) to (GLY252) CRYSTAL STRUCTURE OF THE HSLUV PROTEASE-CHAPERONE COMPLEX | CHAPERONE/HYDROLASE
1g4b:E (GLU82) to (GLU228) CRYSTAL STRUCTURES OF THE HSLVU PEPTIDASE-ATPASE COMPLEX REVEAL AN ATP-DEPENDENT PROTEOLYSIS MECHANISM | HSLVU, PEPTIDASE-ATPASE COMPLEX, CHAPERONE/HYDROLASE COMPLEX
1g4b:K (GLU82) to (GLU228) CRYSTAL STRUCTURES OF THE HSLVU PEPTIDASE-ATPASE COMPLEX REVEAL AN ATP-DEPENDENT PROTEOLYSIS MECHANISM | HSLVU, PEPTIDASE-ATPASE COMPLEX, CHAPERONE/HYDROLASE COMPLEX
2ffl:B (SER698) to (VAL750) CRYSTAL STRUCTURE OF DICER FROM GIARDIA INTESTINALIS | RNA INTERFERENCE; RNAI; PAZ DOMAIN, TRANSLATION, HYDROLASE, TRANSLATION,HYDROLASE
2ffl:C (SER698) to (VAL750) CRYSTAL STRUCTURE OF DICER FROM GIARDIA INTESTINALIS | RNA INTERFERENCE; RNAI; PAZ DOMAIN, TRANSLATION, HYDROLASE, TRANSLATION,HYDROLASE
2ffl:D (SER698) to (VAL750) CRYSTAL STRUCTURE OF DICER FROM GIARDIA INTESTINALIS | RNA INTERFERENCE; RNAI; PAZ DOMAIN, TRANSLATION, HYDROLASE, TRANSLATION,HYDROLASE
3upz:A (LEU323) to (ASP415) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH BUMPLESS BKI ANALOG UW1243 | SERINE/THREONINE PROTEIN KINASE, CALCIUM-BINDING, ATP-BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4z49:B (SER2340) to (LEU2390) HOMO SAPIENS FATTY ACID SYNTHETASE, THIOESTERASE DOMAIN AT 1.7 ANGSTROMS RESOLUTION | FATTY ACID SYNTHETASE, THIOESTERASE, FAS-TE, HYDROLASE
4kit:B (GLU983) to (LYS1025) CRYSTAL STRUCTURE OF HUMAN BRR2 IN COMPLEX WITH THE PRP8 JAB1/MPN DOMAIN | RECA DOMAIN, WINGED HELIX DOMAIN, SEC63 UNIT, JAB1/MPN DOMAIN, PRE- MRNA SPLICING, ATP BINDING, RNA BINDING, UBIQUITIN BINDING, RNA BINDING PROTEIN
4kit:B (ASN1814) to (ASN1857) CRYSTAL STRUCTURE OF HUMAN BRR2 IN COMPLEX WITH THE PRP8 JAB1/MPN DOMAIN | RECA DOMAIN, WINGED HELIX DOMAIN, SEC63 UNIT, JAB1/MPN DOMAIN, PRE- MRNA SPLICING, ATP BINDING, RNA BINDING, UBIQUITIN BINDING, RNA BINDING PROTEIN
4kjt:B (GLY1) to (MET49) STRUCTURE OF THE L100F MUTANT OF DEHALOPEROXIDASE-HEMOGLOBIN A FROM AMPHITRITE ORNATA WITH OXYGEN | GLOBIN, OXYGEN STORAGE, PEROXIDASE, OXIDOREDUCTASE
3uuc:B (THR311) to (SER395) CRYSTAL STRUCTURE OF HERA-LBD (WT) IN COMPLEX WITH BISPHENOL-C | LIGAND-BINDING DOMAIN OF NUCLEAR HORMONE RECEPTOR, HORMONE RECEPTOR
3uy4:A (SER184) to (LYS234) CRYSTAL STRUCTURE OF PANTOATE--BETA-ALANINE LIGASE FROM CAMPYLOBACTER JEJUNI COMPLEXED WITH AMP AND VITAMIN B5 | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA-BETA-ALPHA STRUCTURE, CYTOSOL, LIGASE
4kmv:B (GLY1) to (MET49) STRUCTURE OF THE L100F MUTANT OF DEHALOPEROXIDASE-HEMOGLOBIN A FROM AMPHITRITE ORNATA WITH 2,4,6-TRICHLOROPHENOL | GLOBIN, OXYGEN STORAGE, PEROXIDASE, OXIDOREDUCTASE, OXIDOREDUCTASE- OXIDOREDUCTASE INHIBITOR COMPLEX
2fsl:X (ASN269) to (ALA309) MITOGEN ACTIVATED PROTEIN KINASE P38ALPHA (D176A+F327S) ACTIVATING MUTANT FORM-A | MITOGEN ACTIVATED PROTEIN KINASE, P38, ACTIVE MUTANTS, LIPIDS, MAP KINASE INSERTION, AUTOPHOSPHORYLATION, TRANSFERASE
1s9p:D (LYS236) to (SER317) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAIN OF THE ESTROGEN-RELATED RECEPTOR GAMMA IN COMPLEX WITH DIETHYLSTILBESTROL | LIGAND-BINDING DOMAIN, ANTAGONIST COMPLEX, TRANSCRIPTION
3hwk:B (GLN308) to (ARG357) CRYSTAL STRUCTURE OF METHYLCITRATE SYNTHASE FROM MYCOBACTERIUM TUBERCULOSIS | NIAID, SSGCID, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, TUBERCLUOSIS, UW, SBRI, DECODE, ACYLTRANSFERASE, TRANSFERASE
3hwk:E (GLN308) to (ARG357) CRYSTAL STRUCTURE OF METHYLCITRATE SYNTHASE FROM MYCOBACTERIUM TUBERCULOSIS | NIAID, SSGCID, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, TUBERCLUOSIS, UW, SBRI, DECODE, ACYLTRANSFERASE, TRANSFERASE
2fup:A (ALA81) to (ARG130) CRYSTAL STRUCTURE OF A PUTATIVE FLAGELLA SYNTHESIS PROTEIN FLGN (PA3352) FROM PSEUDOMONAS AERUGINOSA AT 1.48 A RESOLUTION | STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, BIOSYNTHETIC PROTEIN
3i1i:B (PRO182) to (GLU270) X-RAY CRYSTAL STRUCTURE OF HOMOSERINE O-ACETYLTRANSFERASE FROM BACILLUS ANTHRACIS | STRUCTURAL GENOMICS, IDP01610, HOMOSERINE, O-ACETYLTRANSFERASE, BACILLUS ANTHRACIS, TRANSFERASE, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID
3v9r:B (SER3) to (MSE80) CRYSTAL STRUCTURE OF SACCHAROMYCES CEREVISIAE MHF COMPLEX | MHF1, MHF2, HISTONE FOLD, FANCONI ANEMIA, DNA REPAIR, DNA BINDING PROTEIN
1sr7:B (PRO686) to (LYS769) PROGESTERONE RECEPTOR HORMONE BINDING DOMAIN WITH BOUND MOMETASONE FUROATE | PROGESTERONE RECEPTOR, MOMETASONE, PROGESTERONE, NUCLEAR RECEPTOR, HORMONE RECEPTOR, TRANSCRIPTION
1sra:A (TYR207) to (ASP257) STRUCTURE OF A NOVEL EXTRACELLULAR CA2+-BINDING MODULE IN BM-40(SLASH)SPARC(SLASH)OSTEONECTIN | EXTRACELLULAR MATRIX PROTEIN, CALCIUM-BINDING PROTEIN
1gws:A (GLY443) to (HIS509) HEXADECAHEME HIGH MOLECULAR WEIGHT CYTOCHROME HMC FROM DESULFOVIBRIO VULGARIS HILDENBOROUGH | ELECTRON TRANSPORT, MULTIHEME CYTOCHROME, SULFATE REDUCING BACTERIA, PERIPLASMIC, HEME
1svl:A (ASN332) to (ASN415) CO-CRYSTAL STRUCTURE OF SV40 LARGE T ANTIGEN HELICASE DOMAIN AND ADP | AAA+ FOLD, VIRAL PROTEIN
4l0f:A (LEU119) to (ALA179) STRUCTURE OF P450SKY (CYP163B3), A CYTOCHROME P450 FROM SKYLLAMYCIN BIOSYNTHESIS (OPEN ACTIVE SITE) | CYTOCHROME P450, SKYLLAMYCIN BIOSYNTHESIS, BETA-AMINOACYL CARRIER PROTEIN OXIDASE, SKYLLAMYCIN NONRIBOSOMAL PEPTIDE SYNTHETASE, OXIDOREDUCTASE
3vh5:D (ARG9) to (PHE79) CRYSTAL STRUCTURE OF THE CHICKEN CENP-T HISTONE FOLD/CENP-W/CENP- S/CENP-X HETEROTETRAMERIC COMPLEX, CRYSTAL FORM I | HISTONE FOLD, CHROMOSOME SEGREGATION, DNA BINDING, NUCLEUS, DNA BINDING PROTEIN
1h29:B (GLY474) to (HIS540) SULFATE RESPIRATION IN DESULFOVIBRIO VULGARIS HILDENBOROUGH: STRUCTURE OF THE 16-HEME CYTOCHROME C HMCA AT 2.5 A RESOLUTION AND A VIEW OF ITS ROLE IN TRANSMEMBRANE ELECTRON TRANSFER | ELECTRON TRANSPORT, HIGH MOLECULAR MASS CYTOCHROME, SULFATE RESPIRATION, HYDROGEN CYCLE, TRANSMEMBRANE REDOX COMPLEX, ENERGY CONSERVATION, PROTON GRADIENT, TETRA-HEME, C3-LIKE DOMAIN
1h29:D (GLY474) to (HIS540) SULFATE RESPIRATION IN DESULFOVIBRIO VULGARIS HILDENBOROUGH: STRUCTURE OF THE 16-HEME CYTOCHROME C HMCA AT 2.5 A RESOLUTION AND A VIEW OF ITS ROLE IN TRANSMEMBRANE ELECTRON TRANSFER | ELECTRON TRANSPORT, HIGH MOLECULAR MASS CYTOCHROME, SULFATE RESPIRATION, HYDROGEN CYCLE, TRANSMEMBRANE REDOX COMPLEX, ENERGY CONSERVATION, PROTON GRADIENT, TETRA-HEME, C3-LIKE DOMAIN
2gl8:C (VAL14) to (VAL99) HUMAN RETINOIC ACID RECEPTOR RXR-GAMMA LIGAND-BINDING DOMAIN | NUCLEAR RECEPTOR, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
1t3q:A (LEU95) to (ASN140) CRYSTAL STRUCTURE OF QUINOLINE 2-OXIDOREDUCTASE FROM PSEUDOMONAS PUTIDA 86 | QOR, MOLYBDENUM, MCD, OXIDOREDUCTASE
1t3q:D (ASN93) to (ASN140) CRYSTAL STRUCTURE OF QUINOLINE 2-OXIDOREDUCTASE FROM PSEUDOMONAS PUTIDA 86 | QOR, MOLYBDENUM, MCD, OXIDOREDUCTASE
4l49:A (LEU127) to (PRO187) STRUCTURE OF L358A MUTANT OF P450CAM BOUND TO CAMPHOR | MONO-OXYGENASE, CYTOCHROME P450, OXIDOREDUCTASE
1t6j:A (ALA648) to (LEU715) CRYSTAL STRUCTURE OF PHENYLALANINE AMMONIA LYASE FROM RHODOSPORIDIUM TORULOIDES | TRIPLE HELIX COILED COIL; MIO; CINNAMATE, LYASE
2gpv:A (ASN235) to (LEU318) ESTROGEN RELATED RECEPTOR-GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH 4-HYDROXY-TAMOXIFEN AND A SMRT PEPTIDE | ESTROGEN RELATED RECEPTOR, ERR, ERRG, ESRRG, NUCLEAR RECEPTOR, STEROID RECEPTOR, SMRT, TAMOXIFEN, TRANSCRIPTION
3ih2:A (LEU121) to (MSE198) TM1030 CRYSTALLIZED AT 323K | TM1030, TRANSCRIPTIONAL REGULATOR, TEMPERATURE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, DNA-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSCRIPTION REGULATOR
3ih3:A (LEU121) to (MSE198) TM1030 CRYSTALLIZED AT 310K | TRANSCRIPTIONAL REGULATOR, TM1030, TEMPERATURE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, DNA-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSCRIPTION REGULATOR
3ih4:A (LEU121) to (MSE198) TM1030 CRYSTALLIZED AT 277K | TRANSCRIPTIONAL REGULATOR, TM1030, TEMPERATURE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, DNA-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSCRIPTION REGULATOR
4l8u:A (GLU400) to (PRO468) X-RAY STUDY OF HUMAN SERUM ALBUMIN COMPLEXED WITH 9 AMINO CAMPTOTHECIN | PLASMA PROTEIN, ONCOLOGY DRUGS, PROTEIN DRUG COMPLEX, TRANSPORT PROTEIN
1ha2:A (GLY399) to (THR467) HUMAN SERUM ALBUMIN COMPLEXED WITH MYRISTIC ACID AND THE S- (-) ENANTIOMER OF WARFARIN | TRANSPORT PROTEIN, SERUM PROTEIN, DRUG BINDING, ANTI-COAGULANT
1h9z:A (GLY399) to (THR467) HUMAN SERUM ALBUMIN COMPLEXED WITH MYRISTIC ACID AND THE R-(+) ENANTIOMER OF WARFARIN | TRANSPORT PROTEIN, SERUM PROTEIN, DRUG BINDING, ANTI-COAGULANT
1hbn:A (PRO282) to (TYR358) METHYL-COENZYME M REDUCTASE | METHANOGENESIS, BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE
1hbn:D (PRO282) to (TYR358) METHYL-COENZYME M REDUCTASE | METHANOGENESIS, BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE
1hbo:A (PRO282) to (TYR358) METHYL-COENZYME M REDUCTASE MCR-RED1-SILENT | METHANOGENESIS, BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE
1hbo:D (PHE283) to (TYR358) METHYL-COENZYME M REDUCTASE MCR-RED1-SILENT | METHANOGENESIS, BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE
1hbu:A (PRO282) to (TYR358) METHYL-COENZYME M REDUCTASE IN THE MCR-RED1-SILENT STATE IN COMPLEX WITH COENZYME M | METHANOGENESIS, BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE
1hbu:D (PRO282) to (TYR358) METHYL-COENZYME M REDUCTASE IN THE MCR-RED1-SILENT STATE IN COMPLEX WITH COENZYME M | METHANOGENESIS, BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE
4zti:A (GLY291) to (PRO314) EBOLA VIRUS NUCLEOPROTEIN BOUND TO VP35 CHAPERONING PEPTIDE P212121 | NUCLEOPROTEIN, CHAPERONE, RNA-BINDNG, VIRAL PROTEIN
1tfb:A (LYS226) to (GLY279) NMR STUDIES OF HUMAN GENERAL TRANSCRIPTION FACTOR TFIIB: DYNAMICS AND INTERACTION WITH VP16 ACTIVATION DOMAIN, 20 STRUCTURES | TRANSCRIPTION FACTOR, HUMAN GENERAL TRANSCRIPTION FACTOR TFIIB, C-TERMINAL CORE DOMAIN, CYCLIN BOX FOLD
2h1l:A (ASN332) to (VAL413) THE STRUCTURE OF THE ONCOPROTEIN SV40 LARGE T ANTIGEN AND P53 TUMOR SUPPRESSOR COMPLEX | P53 LOOP-3 CONFORMATION CHANGE, VIRAL PROTEIN
2h1l:F (ASN332) to (ASN415) THE STRUCTURE OF THE ONCOPROTEIN SV40 LARGE T ANTIGEN AND P53 TUMOR SUPPRESSOR COMPLEX | P53 LOOP-3 CONFORMATION CHANGE, VIRAL PROTEIN
2h1l:H (ASN332) to (VAL413) THE STRUCTURE OF THE ONCOPROTEIN SV40 LARGE T ANTIGEN AND P53 TUMOR SUPPRESSOR COMPLEX | P53 LOOP-3 CONFORMATION CHANGE, VIRAL PROTEIN
2h1l:J (GLN333) to (ASN415) THE STRUCTURE OF THE ONCOPROTEIN SV40 LARGE T ANTIGEN AND P53 TUMOR SUPPRESSOR COMPLEX | P53 LOOP-3 CONFORMATION CHANGE, VIRAL PROTEIN
4lil:A (PHE223) to (SER262) CRYSTAL STRUCTURE OF THE CATALYTIC SUBUNIT OF HUMAN PRIMASE BOUND TO UTP AND MN | PRIM FOLD, TRANSFERASE
1hk4:A (GLY399) to (THR467) HUMAN SERUM ALBUMIN COMPLEXED WITH THYROXINE (3,3',5,5'-TETRAIODO-L-THYRONINE) AND MYRISTIC ACID (TETRADECANOIC ACID) | PLASMA PROTEIN, HORMONE-BINDING, LIPID-BINDING, THYROXINE, FAMILIAL DYSALBUMINEMIC HYPERTHYROXINEMIA
3vkh:A (ASP4300) to (ASN4370) X-RAY STRUCTURE OF A FUNCTIONAL FULL-LENGTH DYNEIN MOTOR DOMAIN | AAA+ PROTEIN, MOLECULAR MOTOR, MICROTUBLES, MOTOR PROTEIN
3vkh:B (GLU3985) to (GLY4049) X-RAY STRUCTURE OF A FUNCTIONAL FULL-LENGTH DYNEIN MOTOR DOMAIN | AAA+ PROTEIN, MOLECULAR MOTOR, MICROTUBLES, MOTOR PROTEIN
3vlm:B (ASP443) to (GLU500) CRYSTAL STRUCTURE ANALYSIS OF THE MET244ALA VARIANT OF KATG FROM HALOARCULA MARISMORTUI | CATALASE-PEROXIDASE, OXIDOREDUCTASE
2hfp:A (ILE267) to (MET334) CRYSTAL STRUCTURE OF PPAR GAMMA WITH N-SULFONYL-2-INDOLE CARBOXAMIDE LIGANDS | PPAR PPARGAMMA LBD, TRANSCRIPTION
3ixp:A (ILE210) to (LEU302) CRYSTAL STRUCTURE OF THE ECDYSONE RECEPTOR BOUND TO BYI08346 | ANTI-PARALLEL ALPHA-HELICES, TRANSCRIPTION, TRANSCRIPTION REGULATION
1tt5:C (VAL315) to (ASN386) STRUCTURE OF APPBP1-UBA3-UBC12N26: A UNIQUE E1-E2 INTERACTION REQUIRED FOR OPTIMAL CONJUGATION OF THE UBIQUITIN-LIKE PROTEIN NEDD8 | CELL CYCLE, LIGASE
5a0g:B (SER163) to (LEU243) N-TERMINAL THIOESTER DOMAIN OF SURFACE PROTEIN FROM CLOSTRIDIUM PERFRINGENS | CELL ADHESION, SURFACE-ASSOCIATED PROTEIN, GRAM-POSITIVE, ADHESIN, INTERNAL THIOESTER, THIOESTER DOMAIN
1ht2:F (GLU82) to (VAL234) NUCLEOTIDE-DEPENDENT CONFORMATIONAL CHANGES IN A PROTEASE-ASSOCIATED ATPASE HSLU | HSLVU, PEPTIDASE-ATPASE COMPLEX, CHAPERONE
5a0y:A (PRO282) to (GLY359) METHYL-COENZYME M REDUCTASE FROM METHANOTHERMOBACTER MARBURGENSIS AT 1.1 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, CATALYSIS, COENZYMES, DISULFIDES, HYDROGEN, HYDROGEN BONDING, LIGANDS, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, MODELS, MOLECULAR, NICKEL, OXIDATION-REDUCTION, OXIDOREDUCTASES, PHOSPHOTHREONINE, PROTEIN CONFORMATION, PROTEIN FOLDING, PROTEIN STRUCTURE,
5a0y:D (PRO282) to (GLY359) METHYL-COENZYME M REDUCTASE FROM METHANOTHERMOBACTER MARBURGENSIS AT 1.1 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, CATALYSIS, COENZYMES, DISULFIDES, HYDROGEN, HYDROGEN BONDING, LIGANDS, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, MODELS, MOLECULAR, NICKEL, OXIDATION-REDUCTION, OXIDOREDUCTASES, PHOSPHOTHREONINE, PROTEIN CONFORMATION, PROTEIN FOLDING, PROTEIN STRUCTURE,
2wio:A (PRO108) to (ASP176) STRUCTURE OF THE HISTIDINE TAGGED, OPEN CYTOCHROME P450 ERYK FROM S. ERYTHRAEA | SUBSTRATE SPECIFICITY, ANTIBIOTIC BIOSYNTHESIS, METAL-BINDING, OXIDOREDUCTASE, CYTOCHROME P450, IRON, HEME, ERYTHROMICYN, MONOOXYGENASE
3vuq:B (PRO118) to (GLY184) CRYSTAL STRUCTURE OF TTHA0167, A TRANSCRIPTIONAL REGULATOR, TETR/ACRR FAMILY FROM THERMUS THERMOPHILUS HB8 | HELIX-TURN-HELIX, TRANSCRIPTIONAL REGULATOR, DNA BINDING, TRANSCRIPTION REGULATOR
1u75:A (ARG31) to (ALA83) ELECTRON TRANSFER COMPLEX BETWEEN HORSE HEART CYTOCHROME C AND ZINC- PORPHYRIN SUBSTITUTED CYTOCHROME C PEROXIDASE | PROTEIN-PROTEIN COMPLEX, HEME, OXIDOREDUCTASE
2wss:N (GLY392) to (ALA474) THE STRUCTURE OF THE MEMBRANE EXTRINSIC REGION OF BOVINE ATP SYNTHASE | HYDROGEN ION TRANSPORT, ATP SYNTHESIS, PHOSPHOPROTEIN, UBL CONJUGATION, TRANSIT PEPTIDE, NUCLEOTIDE-BINDING, ACETYLATION, ATP-BINDING, ION TRANSPORT, MITOCHONDRION, PYRROLIDONE CARBOXYLIC ACID, HYDROLASE, TRANSPORT
3w4t:A (SER235) to (PHE349) CRYSTAL STRUCTURE OF MATE P26A MUTANT | MATE, MULTIDRUG TRANSPORTER, TRANSPORT PROTEIN
5a8k:A (PRO282) to (TYR358) METHYL-COENZYME M REDUCTASE FROM METHANOTHERMOBACTER WOLFEII AT 1.4 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, CATALYSIS, COENZYMES, DISULFIDES, HYDROGEN, HYDROGEN BONDING, LIGANDS, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, MODELS, MOLECULAR, NICKEL, OXIDATION-REDUCTION, OXIDOREDUCTASES, PHOSPHOTHREONINE, PROTEIN CONFORMATION, PROTEIN FOLDING, PROTEIN STRUCTURE,
5a8k:D (PRO282) to (TYR358) METHYL-COENZYME M REDUCTASE FROM METHANOTHERMOBACTER WOLFEII AT 1.4 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, CATALYSIS, COENZYMES, DISULFIDES, HYDROGEN, HYDROGEN BONDING, LIGANDS, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, MODELS, MOLECULAR, NICKEL, OXIDATION-REDUCTION, OXIDOREDUCTASES, PHOSPHOTHREONINE, PROTEIN CONFORMATION, PROTEIN FOLDING, PROTEIN STRUCTURE,
5a8w:A (ALA286) to (PHE361) METHYL-COENZYME M REDUCTASE II FROM METHANOTHERMOBACTER WOLFEII AT 1.8 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, COENZYMES, DISULFIDES, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, NICKEL, OXIDATION-REDUCTION, PHOSPHOTHREONINE,
5a8w:D (ALA286) to (PHE361) METHYL-COENZYME M REDUCTASE II FROM METHANOTHERMOBACTER WOLFEII AT 1.8 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, COENZYMES, DISULFIDES, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, NICKEL, OXIDATION-REDUCTION, PHOSPHOTHREONINE,
5a8w:G (ALA286) to (PHE361) METHYL-COENZYME M REDUCTASE II FROM METHANOTHERMOBACTER WOLFEII AT 1.8 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, COENZYMES, DISULFIDES, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, NICKEL, OXIDATION-REDUCTION, PHOSPHOTHREONINE,
5a8w:J (ALA286) to (PHE361) METHYL-COENZYME M REDUCTASE II FROM METHANOTHERMOBACTER WOLFEII AT 1.8 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, COENZYMES, DISULFIDES, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, NICKEL, OXIDATION-REDUCTION, PHOSPHOTHREONINE,
4m58:A (LEU106) to (GLU215) CRYSTAL STRUCTURE OF AN TRANSITION METAL TRANSPORTER | MEMBRANE PROTEIN, TRANSPORTER, NICKEL
4m5b:A (LEU106) to (HIS212) CRYSTAL STRUCTURE OF AN TRUNCATED TRANSITION METAL TRANSPORTER | MEMBRANE PROTEIN, TRANSPORTER, NICKEL
4m5c:A (LEU106) to (HIS212) CRYSTAL STRUCTURE OF AN TRUNCATED TRANSITION METAL TRANSPORTER | MEMBRANE PROTEIN, TRANSPORTER, COBALT
1up6:A (ASP352) to (ASN408) STRUCTURE OF THE 6-PHOSPHO-BETA GLUCOSIDASE FROM THERMOTOGA MARITIMA AT 2.55 ANGSTROM RESOLUTION IN THE TETRAGONAL FORM WITH MANGANESE, NAD+ AND GLUCOSE-6-PHOSPHATE | HYDROLASE, 6-PHOSPHO-BETA-GLUCOSIDASE, FAMILY4 HYDROLASE, NAD DEPENDENT
1up6:B (ASP352) to (ASN408) STRUCTURE OF THE 6-PHOSPHO-BETA GLUCOSIDASE FROM THERMOTOGA MARITIMA AT 2.55 ANGSTROM RESOLUTION IN THE TETRAGONAL FORM WITH MANGANESE, NAD+ AND GLUCOSE-6-PHOSPHATE | HYDROLASE, 6-PHOSPHO-BETA-GLUCOSIDASE, FAMILY4 HYDROLASE, NAD DEPENDENT
2id6:A (LEU121) to (MSE198) CRYSTAL STRUCTURE OF TRANSCRIPTIONAL REGULATOR (TM1030) AT 1.75A RESOLUTION | TRANSCRIPTIONAL REGULATOR; TETR FAMILY
3wbn:A (SER235) to (PHE349) CRYSTAL STRUCTURE OF MATE IN COMPLEX WITH MAL6 | MATE, MULTIDRUG TRANSPORTER, TRANSPORT PROTEIN-INHIBITOR COMPLEX
4md8:E (ARG280) to (TYR325) CRYSTAL STRUCTURE OF FULL-LENGTH SYMMETRIC CK2 HOLOENZYME WITH MUTATED ALPHA SUBUNIT (F121E) | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
4md8:F (ARG280) to (TYR325) CRYSTAL STRUCTURE OF FULL-LENGTH SYMMETRIC CK2 HOLOENZYME WITH MUTATED ALPHA SUBUNIT (F121E) | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
4md8:G (ARG280) to (TYR325) CRYSTAL STRUCTURE OF FULL-LENGTH SYMMETRIC CK2 HOLOENZYME WITH MUTATED ALPHA SUBUNIT (F121E) | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
2iwh:B (ASP336) to (THR391) STRUCTURE OF YEAST ELONGATION FACTOR 3 IN COMPLEX WITH ADPNP | PROTEIN BIOSYNTHESIS, TRANSLATION, PHOSPHORYLATION, ELONGATION FACTOR, NUCLEOTIDE-BINDING, RNA-BINDING, ACETYLATION, ATP-BINDING, RRNA-BINDING
1jfz:D (LYS618) to (GLU688) CRYSTAL STRUCTURE OF MN(II)-COMPLEX OF RNASE III ENDONUCLEASE DOMAIN FROM AQUIFEX AEOLICUS AT 2.10 ANGSTROM RESOLUTION | RIBONUCLEASE, RNASE III, DOUBLE-STRANDED RNA, RNA INTERFERENCE, ENDONUCLEASE DOMAIN, ENDONUCLEOLYTIC CLEAVAGE, HYDROLASE
5aqd:K (ASN47) to (ALA111) CRYSTAL STRUCTURE OF PHORMIDIUM PHYCOERYTHRIN AT PH 8.5 | PHOTOSYNTHESIS, PHYCOBILISOME PROTEIN, PHYCOERYTHRIN ALPHA CHAIN, PHYCOERYTHRIN BETA CHAIN, PEB CHROMOPHORE, PROTEIN-CHROMOPHORE LINKAGE
4ms3:B (THR334) to (THR406) CRYSTAL STRUCTURE OF THE EXTRACELLULAR DOMAIN OF HUMAN GABA(B) RECEPTOR BOUND TO THE ENDOGENOUS AGONIST GABA | HETERODIMERIC PROTEIN COMPLEX, VENUS FLYTRAP MODULE, NEUROTRANSMITTER RECEPTOR, SIGNALING PROTEIN-AGONIST COMPLEX
4ms4:B (THR334) to (THR406) CRYSTAL STRUCTURE OF THE EXTRACELLULAR DOMAIN OF HUMAN GABA(B) RECEPTOR BOUND TO THE AGONIST BACLOFEN | HETERODIMERIC PROTEIN COMPLEX, VENUS FLYTRAP MODULE, NEUROTRANSMITTER RECEPTOR, SIGNALING PROTEIN-AGONIST COMPLEX
1vtk:A (PRO209) to (ALA294) THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH ADP AND DEOXYTHYMIDINE-MONOPHOSPHATE | KEY ENZYME IN THYMIDINE SALVAGE PATHWAY, ADDITIONAL THYMIDYLATE KINASE ACTIVITY, TARGET FOR ANTI-HERPES VIRAL DRUGS, TRANSFERASE
2xmr:B (TRP164) to (ALA210) CRYSTAL STRUCTURE OF HUMAN NDRG2 PROTEIN PROVIDES INSIGHT INTO ITS ROLE AS A TUMOR SUPPRESSOR | SIGNALING PROTEIN, NDRG FAMILY
3wz4:D (ASP75) to (LYS132) STRUCTURE OF THE PERIPLASMIC DOMAIN OF DOTI (CRYSTAL FORM I) | TYPE IVB SECRETION, UNKNOWN FUNCTION
5b02:C (LEU200) to (LEU254) STRUCTURE OF THE PRENYLTRANSFERASE MOEN5 WITH A FUSION PROTEIN TAG OF SSO7D | PRENYLTRANSFERASE, ALPHA-HELICAL FOLD, DNA-BINDING, TRANSFERASE, DNA BINDING PROTEIN
5b0i:C (LEU200) to (LEU254) STRUCTURE OF MOEN5-SSO7D FUSION PROTEIN IN COMPLEX WITH BETA-OCTYL GLUCOSIDE | PRENYLTRANSFERASE, ALPHA-HELICAL FOLD, FUSION TAG, LIGAND COMPLEX, TRANSFERASE, DNA BINDING PROTEIN
4n1y:C (THR249) to (ILE333) CRYSTAL STRUCTURE OF THE PACIFIC OYSTER ESTROGEN RECEPTOR LIGAND BINDING DOMAIN | ESTROGEN, NUCLEAR HORMONE RECEPTOR, ENDOCRINE SIGNALING, TRANSCRIPTION
4n1y:D (THR249) to (ILE333) CRYSTAL STRUCTURE OF THE PACIFIC OYSTER ESTROGEN RECEPTOR LIGAND BINDING DOMAIN | ESTROGEN, NUCLEAR HORMONE RECEPTOR, ENDOCRINE SIGNALING, TRANSCRIPTION
1w27:A (SER559) to (GLY644) PHENYLALANINE AMMONIA-LYASE (PAL) FROM PETROSELINUM CRISPUM | LYASE, PHENYLPROPANOID METABOLISM, MIO
1w27:B (SER559) to (GLY644) PHENYLALANINE AMMONIA-LYASE (PAL) FROM PETROSELINUM CRISPUM | LYASE, PHENYLPROPANOID METABOLISM, MIO
3zcn:B (LEU28) to (LEU113) FIC PROTEIN FROM SHEWANELLA ONEIDENSIS IN COMPLEX WITH ATP | TRANSFERASE, AMPYLATION, ADENYLYLATION
2xsb:A (GLU258) to (THR338) OGOGA PUGNAC COMPLEX | O-GLCNACYLATION, O-GLCNACASE, GLYCOSYL HYDROLASE, HYDROLASE
4n5g:B (VAL232) to (ILE318) CRYSTAL STRUCTURE OF RXRA LBD COMPLEXED WITH A SYNTHETIC MODULATOR K8012 | RETINOID X RECEPTOR-ALPHA NUCLEAR RECEPTOR, NUCLEUS, SIGNALING PROTEIN
4n5g:C (VAL232) to (SER317) CRYSTAL STRUCTURE OF RXRA LBD COMPLEXED WITH A SYNTHETIC MODULATOR K8012 | RETINOID X RECEPTOR-ALPHA NUCLEAR RECEPTOR, NUCLEUS, SIGNALING PROTEIN
3zec:A (LEU28) to (LEU113) FIC PROTEIN FROM SHEWANELLA ONEIDENSIS (E73G MUTANT) IN COMPLEX WITH AMPPNP | AMPYLATION, ADENYLYLATION, TRANSFERASE
3zec:B (THR27) to (LEU113) FIC PROTEIN FROM SHEWANELLA ONEIDENSIS (E73G MUTANT) IN COMPLEX WITH AMPPNP | AMPYLATION, ADENYLYLATION, TRANSFERASE
2xvw:A (GLY399) to (THR467) HUMAN SERUM ALBUMIN COMPLEXED WITH DANSYL-L-ARGININE AND MYRISTIC ACID | TRANSPORT PROTEIN
5bs7:D (LYS31) to (GLN93) STRUCTURE OF HISTONE H3/H4 IN COMPLEX WITH SPT2 | CHAPERONE, TRANSCRIPTION, TRANSCRIPTION REGULATOR
4ne6:B (LYS12) to (PHE81) HUMAN MHF1-MHF2 COMPLEX | HISTONE FOLD, DNA REPAIR, GENOME MAINTENANCE, FANCONI ANEMIA, FANCM, NUCLEUS, DNA BINDING PROTEIN
4ne6:D (LYS12) to (PHE81) HUMAN MHF1-MHF2 COMPLEX | HISTONE FOLD, DNA REPAIR, GENOME MAINTENANCE, FANCONI ANEMIA, FANCM, NUCLEUS, DNA BINDING PROTEIN
1k7l:E (ALA256) to (MET325) THE 2.5 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE HUMAN PPARALPHA LIGAND BINDING DOMAIN BOUND WITH GW409544 AND A CO-ACTIVATOR PEPTIDE. | THE 2.5 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF THE HUMAN PPARALPHA LIGAND BINDING DOMAIN BOUND WITH GW409544 AND A COACTIVATOR PEPTIDE, TRANSCRIPTION
2jq4:A (MET1) to (SER65) COMPLETE RESONANCE ASSIGNMENTS AND SOLUTION STRUCTURE CALCULATION OF ATC2521 (NESG ID: ATT6) FROM AGROBACTERIUM TUMEFACIENS | AGROBACTERIUM TUMEFACIENS, ATC2521, UNKNOWN FUNCTION, ATC, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, NESG
1wgz:B (VAL417) to (GLY475) CRYSTAL STRUCTURE OF CARBOXYPEPTIDASE 1 FROM THERMUS THERMOPHILUS | NEUROLYSIN-LIKE CARBOXYPEPTIDASE, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, STRUCTURAL GENOMICS, HYDROLASE
4nh1:A (ARG280) to (TYR325) CRYSTAL STRUCTURE OF A HETEROTETRAMERIC CK2 HOLOENZYME COMPLEX CARRYING THE ANDANTE-MUTATION IN CK2BETA AND CONSISTENT WITH PROPOSED MODELS OF AUTOINHIBITION AND TRANS-AUTOPHOSPHORYLATION | EUKARYOTIC PROTEIN KINASE FOLD, PHOSPHOTRANSFERASE (KINASE), PHOSPHORYLATION, TRANSFERASE
4nh1:B (ARG280) to (TYR325) CRYSTAL STRUCTURE OF A HETEROTETRAMERIC CK2 HOLOENZYME COMPLEX CARRYING THE ANDANTE-MUTATION IN CK2BETA AND CONSISTENT WITH PROPOSED MODELS OF AUTOINHIBITION AND TRANS-AUTOPHOSPHORYLATION | EUKARYOTIC PROTEIN KINASE FOLD, PHOSPHOTRANSFERASE (KINASE), PHOSPHORYLATION, TRANSFERASE
1wmg:F (LEU860) to (ALA897) CRYSTAL STRUCTURE OF THE UNC5H2 DEATH DOMAIN | SIX HELIX BUNDLE, DEATH DOMAIN, APOPTOSIS, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
2ki5:B (ASP211) to (LEU262) HERPES SIMPLEX TYPE-1 THYMIDINE KINASE IN COMPLEX WITH THE DRUG ACICLOVIR AT 1.9A RESOLUTION | TRANSFERASE (PHOSPHOTRANSFERASE) THYMID, TRANSFERASE (PHOSPHOTRANSFERASE) THYMIDINE KINASE; VIRIDAE; DS-DNA ENVELOPED VIRUSES; HERPESVIRIDAE; ALPHAHERPESVIRINAE ANTIVIRAL DRUG (ACICLOVIR)
2km6:A (SER5) to (ALA51) NMR STRUCTURE OF THE NLRP7 PYRIN DOMAIN | NLRP7, PYRIN DOMAIN, INNATE IMMUNE SYSTEM, NALP, ATP-BINDING, DISEASE MUTATION, LEUCINE-RICH REPEAT, NUCLEOTIDE-BINDING, IMMUNE SYSTEM, SIGNALING PROTEIN, PROTEIN BINDING
5c0t:B (VAL25) to (ALA60) CRYSTAL STRUCTURE OF THE MERCURY-BOUND FORM OF MERB MUTANT D99S | BACTERIAL PROTEINS, CYSTEINE, ESCHERICHIA COLI, LYASES, MERCURY, MUTATION, LYASE, METAL BINDING PROTEIN
2kzt:A (LEU226) to (SER305) STRUCTURE OF THE TANDEM MA-3 REGION OF PDCD4 | PDCD4, MA-3, EIF4A, HEAT, APOPTOSIS
1ki2:A (GLU210) to (ALA294) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE I COMPLEXED WITH GANCICLOVIR | PHOSPHOTRANSFERASE, THYMIDINE KINASE, VIRIDAE, DS-DNA ENVELOPED VIRUSES, HERPESVIRIDAE, ALPHAHERPESVIRINAE, ANTIVIRAL DRUG, GANCICLOVIR
1ki2:B (GLU210) to (LEU262) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE I COMPLEXED WITH GANCICLOVIR | PHOSPHOTRANSFERASE, THYMIDINE KINASE, VIRIDAE, DS-DNA ENVELOPED VIRUSES, HERPESVIRIDAE, ALPHAHERPESVIRINAE, ANTIVIRAL DRUG, GANCICLOVIR
1ki3:B (PRO209) to (LEU262) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE I COMPLEXED WITH PENCICLOVIR | PHOSPHOTRANSFERASE, THYMIDINE KINASE, VIRIDAE, DS-DNA ENVELOPED VIRUSES, HERPESVIRIDAE, ALPHAHERPESVIRINAE, ANTIVIRAL DRUG PENCICLOVIR
1ki6:B (GLU210) to (LEU262) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE I COMPLEXED WITH A 5-IODOURACIL ANHYDROHEXITOL NUCLEOSIDE | PHOSPHOTRANSFERASE, THYMIDINE KINASE, VIRIDAE, DS-DNA ENVELOPED VIRUSES, HERPESVIRIDAE, ALPHAHERPESVIRINAE, SUBSTRATE ANALOG, 5-IODOURACIL ANHYDROHEXITOL NUCLEOSIDE
1ki7:B (GLU210) to (LEU262) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE I COMPLEXED WITH 5-IODODEOXYURIDINE | PHOSPHOTRANSFERASE, THYMIDINE KINASE, VIRIDAE, DS-DNA ENVELOPED VIRUSES, HERPESVIRIDAE, ALPHAHERPESVIRINAE, SUBSTRATE ANALOG, 5-IODODEOXYURIDINE
3zr7:A (PRO686) to (LYS769) STRUCTURAL BASIS FOR AGONISM AND ANTAGONISM FOR A SET OF CHEMICALLY RELATED PROGESTERONE RECEPTOR MODULATORS | RECEPTOR, AGONIST, ANTAGONIST
3zr7:B (PRO686) to (LYS769) STRUCTURAL BASIS FOR AGONISM AND ANTAGONISM FOR A SET OF CHEMICALLY RELATED PROGESTERONE RECEPTOR MODULATORS | RECEPTOR, AGONIST, ANTAGONIST
3zra:A (PRO686) to (LYS769) STRUCTURAL BASIS FOR AGONISM AND ANTAGONISM FOR A SET OF CHEMICALLY RELATED PROGESTERONE RECEPTOR MODULATORS | HORMONE RECEPTOR
3zra:B (PRO686) to (LYS769) STRUCTURAL BASIS FOR AGONISM AND ANTAGONISM FOR A SET OF CHEMICALLY RELATED PROGESTERONE RECEPTOR MODULATORS | HORMONE RECEPTOR
3zry:A (ALA414) to (GLU487) ROTOR ARCHITECTURE IN THE F(1)-C(10)-RING COMPLEX OF THE YEAST F-ATP SYNTHASE | HYDROLASE, ATP-BINDING, F(1)-F(O)ATP SYNTHASE, MITOCHONDRIA, MOLECULAR MOTOR, CENTRAL STALK, MEMBRANE PROTEIN, C-RING
5c3j:C (PHE100) to (THR183) CRYSTAL STRUCTURE OF MITOCHONDRIAL RHODOQUINOL-FUMARATE REDUCTASE FROM ASCARIS SUUM WITH UBIQUINONE-1 | RHODOQUINOL-FUMARATE REDUCTASE, COMPLEX II, OXIDOREDUCTASE- OXIDOREDUCTASE INHIBITOR COMPLEX
3zsn:A (ALA104) to (LEU169) STRUCTURE OF THE MIXED-FUNCTION P450 MYCG F286A MUTANT IN COMPLEX WITH MYCINAMICIN IV | OXIDOREDUCTASE, MYCINAMICIN BIOSYNTHESIS
1kv1:A (ASN269) to (ALA309) P38 MAP KINASE IN COMPLEX WITH INHIBITOR 1 | PROTEIN-INHIBITOR COMPLEX, TRANSFERASE
2np3:A (LEU153) to (VAL208) CRYSTAL STRUCTURE OF TETR-FAMILY REGULATOR (SCO0857) FROM STREPTOMYCES COELICOLOR A3. | TETR, TRANSCRIPTIONAL REGULATOR, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSCRIPTION
2np3:B (ARG142) to (ASP210) CRYSTAL STRUCTURE OF TETR-FAMILY REGULATOR (SCO0857) FROM STREPTOMYCES COELICOLOR A3. | TETR, TRANSCRIPTIONAL REGULATOR, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSCRIPTION
1xf6:C (ALA48) to (LEU110) HIGH RESOLUTION CRYSTAL STRUCTURE OF PHYCOERYTHRIN 545 FROM THE MARINE CRYPTOPHYTE RHODOMONAS CS24 | PHYCOERYTHRIN, LIGHT-HARVESTING PROTEIN, CRYPTOPHYTE, PHOTOSYNTHESIS
2yja:B (THR311) to (SER395) STAPLED PEPTIDES BINDING TO ESTROGEN RECEPTOR ALPHA. | HORMONE RECEPTOR-PEPTIDE COMPLEX
2nr7:A (ASN120) to (LEU192) STRUCTURAL GENOMICS, THE CRYSTAL STRUCTURE OF PUTATIVE SECRETION ACTIVATOR PROTEIN FROM PORPHYROMONAS GINGIVALIS W83 | APCC85792, SECRETION ACTIVATOR, PORPHYROMONAS GINGIVALIS W83, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MCSG, MIDWEST CENTER FOR STRUCTURAL GENOMICS, UNKNOWN FUNCTION
2nun:A (SER268) to (LEU316) THE STRUCTURE OF THE TYPE III EFFECTOR AVRB COMPLEXED WITH ADP | TYPE III EFFECTOR, AVRB, NUCLOTIDE, POCKET, ADP, TOXIN/PROTEIN BINDING COMPLEX
3jv2:B (SER571) to (PHE703) CRYSTAL STRUCTURE OF B. SUBTILIS SECA WITH BOUND PEPTIDE | PROTEIN TRANSLOCATION, ATPASE, CONFORMATIONAL CHANGE, PEPTIDE BINDING, ATP-BINDING, CELL MEMBRANE, CYTOPLASM, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PROTEIN TRANSPORT, TRANSLOCATION, TRANSPORT, ZINC
4oar:A (GLN838) to (LEU921) PROGESTERONE RECEPTOR WITH BOUND ULIPRISTAL ACETATE AND A PEPTIDE FROM THE CO-REPRESSOR SMRT | PROGESTERONE RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, WOMEN HEALTH, CONTRACEPTION, TRANSCRIPTION- PEPTIDE COMPLEX
2yvx:A (TRP352) to (GLU448) CRYSTAL STRUCTURE OF MAGNESIUM TRANSPORTER MGTE | MEMBRANE PROTEIN, TRANSPORT PROTEIN
2yvx:B (TRP352) to (GLU448) CRYSTAL STRUCTURE OF MAGNESIUM TRANSPORTER MGTE | MEMBRANE PROTEIN, TRANSPORT PROTEIN
2yvx:C (TRP352) to (GLU448) CRYSTAL STRUCTURE OF MAGNESIUM TRANSPORTER MGTE | MEMBRANE PROTEIN, TRANSPORT PROTEIN
2yvx:D (TRP352) to (GLU448) CRYSTAL STRUCTURE OF MAGNESIUM TRANSPORTER MGTE | MEMBRANE PROTEIN, TRANSPORT PROTEIN
5cig:C (ARG31) to (ALA83) COMPLEX OF YEAST CYTOCHROME C PEROXIDASE (W191G) WITH ISO-1 CYTOCHROME C | ELECTRON TRANSFER, HEME PROTEINS, ELECTRON HOPPING, MULTI-STEP TUNNELING, PHOTOCHEMISTRY, ELECTRON TRANSPORT-OXIDOREDUCTASE COMPLEX, ELECTRON TRANSPORT-OXIDOREDUCTASE
2nxx:A (LEU183) to (SER263) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE T.CASTANEUM (COLEOPTERA) HETERODIMER ECRUSP BOUND TO PONASTERONE A | HORMONE RECEPTOR, APO AND HOLO LIGAND BINDING POCKET, HORMONE/GROWTH FACTOR COMPLEX
2nxx:B (LEU183) to (SER263) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE T.CASTANEUM (COLEOPTERA) HETERODIMER ECRUSP BOUND TO PONASTERONE A | HORMONE RECEPTOR, APO AND HOLO LIGAND BINDING POCKET, HORMONE/GROWTH FACTOR COMPLEX
2nxx:C (LEU183) to (SER263) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE T.CASTANEUM (COLEOPTERA) HETERODIMER ECRUSP BOUND TO PONASTERONE A | HORMONE RECEPTOR, APO AND HOLO LIGAND BINDING POCKET, HORMONE/GROWTH FACTOR COMPLEX
2nxx:D (LEU183) to (SER263) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE T.CASTANEUM (COLEOPTERA) HETERODIMER ECRUSP BOUND TO PONASTERONE A | HORMONE RECEPTOR, APO AND HOLO LIGAND BINDING POCKET, HORMONE/GROWTH FACTOR COMPLEX
3k22:B (VAL533) to (GLN615) GLUCOCORTICOID RECEPTOR WITH BOUND ALANINAMIDE 10 WITH TIF2 PEPTIDE | GLUCOCORTICOID RECEPTOR, STEROID HORMONE RECEPTOR, NUCLEAR RECEPTOR, GR, GLUCOCORTICOIDS, ALPHA HELICAL SANDWICH, META-CHANNEL, ALTERNATIVE INITIATION, CHROMATIN REGULATOR, DISEASE MUTATION, DNA- BINDING, ISOPEPTIDE BOND, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, PSEUDOHERMAPHRODITISM, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3k23:A (LEU532) to (SER617) GLUCOCORTICOID RECEPTOR WITH BOUND D-PROLINAMIDE 11 | GLUCOCORTICOID RECEPTOR, STEROID HORMONE RECEPTOR, NUCLEAR RECEPTOR, GR, GLUCOCORTICOIDS, ALPHA HELICAL SANDWICH, META-CHANNEL, ALTERNATIVE INITIATION, CHROMATIN REGULATOR, DISEASE MUTATION, DNA- BINDING, METAL-BINDING, NUCLEUS, PSEUDOHERMAPHRODITISM, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC- FINGER, ACTIVATOR
3k23:C (LEU532) to (GLN615) GLUCOCORTICOID RECEPTOR WITH BOUND D-PROLINAMIDE 11 | GLUCOCORTICOID RECEPTOR, STEROID HORMONE RECEPTOR, NUCLEAR RECEPTOR, GR, GLUCOCORTICOIDS, ALPHA HELICAL SANDWICH, META-CHANNEL, ALTERNATIVE INITIATION, CHROMATIN REGULATOR, DISEASE MUTATION, DNA- BINDING, METAL-BINDING, NUCLEUS, PSEUDOHERMAPHRODITISM, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC- FINGER, ACTIVATOR
2z71:A (ALA214) to (ASN260) STRUCTURE OF TRUNCATED MUTANT CYS1GLY OF PENICILLIN V ACYLASE FROM BACILLUS SPHAERICUS CO-CRYSTALLIZED WITH PENICILLIN V | ZYMOGEN, HYDROLASE, PRECURSOR, PENICILLIN, AUTOPROTEOLYSIS, ANTIBIOTIC RESISTANCE, CATALYSIS, PENICILLIN V ACYLASE
4a4z:A (LEU1112) to (GLN1193) CRYSTAL STRUCTURE OF THE S. CEREVISIAE DEXH HELICASE SKI2 BOUND TO AMPPNP | HYDROLASE, ATPASE, MRNA DEGRADATION, EXOSOME
5cqg:B (LEU27) to (THR79) STRUCTURE OF TRIBOLIUM TELOMERASE IN COMPLEX WITH THE HIGHLY SPECIFIC INHIBITOR BIBR1532 | TELOMERASE REVERSE TRANSCRIPTASE FOLD TERT BIBR15312, TELOMERASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5cs6:A (ARG280) to (VAL328) CRYSTAL STRUCTURE OF CK2ALPHA WITH COMPOUND 3 BOUND | TRANSFERASE, CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION
4ona:A (ASP324) to (VAL414) CALCIUM-DEPENDENT PROTEIN KINASE 1 FROM TOXOPLASMA GONDII (TGCDPK1) IN COMPLEX WITH INHIBITOR UW1517 | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE, CALCIUM-BINDING, ATP- BINDING, BUMPED KINASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ct0:A (ARG280) to (VAL328) CRYSTAL STRUCTURE OF CK2ALPHA WITH 3-(3-CHLORO-4-(PHENYL)BENZYLAMINO) PROPAN-1-OL BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
5cvf:A (ARG280) to (VAL328) CRYSTAL STRUCTURE OF CK2ALPHA WITH COMPOUND 5 BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
5cvh:A (ARG280) to (VAL328) CRYSTAL STRUCTURE OF CK2ALPHA | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
5cvh:B (ARG280) to (VAL327) CRYSTAL STRUCTURE OF CK2ALPHA | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
2zk4:B (GLN271) to (MET334) HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA LIGAND BINDING DOMAIN COMPLEXED WITH 15-OXO- EICOSATETRAENOIC ACID | ANTI PARALLEL HELIX SANDWICH, ACTIVATOR, ALTERNATIVE SPLICING, DIABETES MELLITUS, DISEASE MUTATION, DNA-BINDING, METAL-BINDING, NUCLEUS, OBESITY, PHOSPHOPROTEIN, POLYMORPHISM, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
5cvv:A (ASP45) to (SER91) CONIFERYL ALCOHOL BOUND MONOLIGNOL 4-O-METHYLTRANSFERASE 9 | MONOLIGNOL-4-O METHYLTRANSFERASE, LIGNIN, CONIFERYL ALCOHOL, S- ADENOSYLMETHIONINE, TRANSFERASE
4opx:A (ARG78) to (GLY290) STRUCTURE OF HUMAN PARP-1 BOUND TO A DNA DOUBLE STRAND BREAK IN COMPLEX WITH (2R)-5-FLUORO-2-METHYL-2,3-DIHYDRO-1-BENZOFURAN-7- CARBOXAMIDE | ZINC FINGER, DNA BINDING, PARP, POLYMERASE, DNA REPAIR, POLY(ADP- RIBOSYL)ATION, TRANSFERASE-DNA-TRANSFERASE INHIBITOR COMPLEX
4opx:D (ARG78) to (GLY290) STRUCTURE OF HUMAN PARP-1 BOUND TO A DNA DOUBLE STRAND BREAK IN COMPLEX WITH (2R)-5-FLUORO-2-METHYL-2,3-DIHYDRO-1-BENZOFURAN-7- CARBOXAMIDE | ZINC FINGER, DNA BINDING, PARP, POLYMERASE, DNA REPAIR, POLY(ADP- RIBOSYL)ATION, TRANSFERASE-DNA-TRANSFERASE INHIBITOR COMPLEX
4oqb:A (ARG78) to (GLY290) STRUCTURE OF HUMAN PARP-1 BOUND TO A DNA DOUBLE STRAND BREAK IN COMPLEX WITH (2Z)-2-{4-[2-(MORPHOLIN-4-YL)ETHOXY]BENZYLIDENE}-3-OXO- 2,3-DIHYDRO-1-BENZOFURAN-7-CARBOXAMIDE | ZINC FINGER, DNA BINDING, PARP, POLYMERASE, DNA REPAIR, POLY(ADP- RIBOSYL)ATION, TRANSFERASE-DNA-TRANSFERASE INHIBITOR COMPLEX
4oqb:D (ARG78) to (GLY290) STRUCTURE OF HUMAN PARP-1 BOUND TO A DNA DOUBLE STRAND BREAK IN COMPLEX WITH (2Z)-2-{4-[2-(MORPHOLIN-4-YL)ETHOXY]BENZYLIDENE}-3-OXO- 2,3-DIHYDRO-1-BENZOFURAN-7-CARBOXAMIDE | ZINC FINGER, DNA BINDING, PARP, POLYMERASE, DNA REPAIR, POLY(ADP- RIBOSYL)ATION, TRANSFERASE-DNA-TRANSFERASE INHIBITOR COMPLEX
4oql:B (GLU210) to (LEU262) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH DF-EDU | DNA SYNTHESIS, THYMIDINE KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, TRANSFERASE, 5-ETHYNYLURIDINE NUCLEOSIDE DERIVATIVE
4oqm:B (PRO209) to (LEU262) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH F-ARA-EDU | DNA SYNTHESIS, THYMIDINE KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, TRANSFERASE, 5-ETHYNYLURIDINE NUCLEOSIDE DERIVATIVE
4oqx:B (PRO209) to (LEU262) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH ME-ARA-EDU | DNA SYNTHESIS, THYMIDINE KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, TRANSFERASE, 5-ETHYNYLURIDINE NUCLEOSIDE DERIVATIVE
3khk:A (ASN10) to (ASN100) CRYSTAL STRUCTURE OF TYPE-I RESTRICTION-MODIFICATION SYSTEM METHYLATION SUBUNIT (MM_0429) FROM METHANOSARCHINA MAZEI. | STRUCTURAL GENOMICS, TYPE I RESTRICTION-MODIFICATION SYSTEM METHYLATION SUBUNIT., PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
3khk:B (PHE8) to (ASN100) CRYSTAL STRUCTURE OF TYPE-I RESTRICTION-MODIFICATION SYSTEM METHYLATION SUBUNIT (MM_0429) FROM METHANOSARCHINA MAZEI. | STRUCTURAL GENOMICS, TYPE I RESTRICTION-MODIFICATION SYSTEM METHYLATION SUBUNIT., PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC
4oye:A (ILE341) to (GLU416) CRYSTAL STRUCTURE OF GLTPH R397A IN APO | TRANSPORTER, ALPHA-HELIX, MEMBRANE PROTEIN
4oye:B (ILE341) to (GLU416) CRYSTAL STRUCTURE OF GLTPH R397A IN APO | TRANSPORTER, ALPHA-HELIX, MEMBRANE PROTEIN
4oye:C (ILE341) to (GLU416) CRYSTAL STRUCTURE OF GLTPH R397A IN APO | TRANSPORTER, ALPHA-HELIX, MEMBRANE PROTEIN
4oye:D (ILE341) to (GLU416) CRYSTAL STRUCTURE OF GLTPH R397A IN APO | TRANSPORTER, ALPHA-HELIX, MEMBRANE PROTEIN
4oye:E (ILE341) to (GLU416) CRYSTAL STRUCTURE OF GLTPH R397A IN APO | TRANSPORTER, ALPHA-HELIX, MEMBRANE PROTEIN
4oye:F (ILE341) to (GLU416) CRYSTAL STRUCTURE OF GLTPH R397A IN APO | TRANSPORTER, ALPHA-HELIX, MEMBRANE PROTEIN
4oye:G (ILE341) to (GLU416) CRYSTAL STRUCTURE OF GLTPH R397A IN APO | TRANSPORTER, ALPHA-HELIX, MEMBRANE PROTEIN
4oye:H (ILE341) to (GLU416) CRYSTAL STRUCTURE OF GLTPH R397A IN APO | TRANSPORTER, ALPHA-HELIX, MEMBRANE PROTEIN
4oye:I (ILE341) to (GLU416) CRYSTAL STRUCTURE OF GLTPH R397A IN APO | TRANSPORTER, ALPHA-HELIX, MEMBRANE PROTEIN
4oye:J (ILE341) to (GLU416) CRYSTAL STRUCTURE OF GLTPH R397A IN APO | TRANSPORTER, ALPHA-HELIX, MEMBRANE PROTEIN
4oye:K (ILE341) to (GLU416) CRYSTAL STRUCTURE OF GLTPH R397A IN APO | TRANSPORTER, ALPHA-HELIX, MEMBRANE PROTEIN
4oye:L (ILE341) to (GLU416) CRYSTAL STRUCTURE OF GLTPH R397A IN APO | TRANSPORTER, ALPHA-HELIX, MEMBRANE PROTEIN
4oys:A (PRO511) to (ASN584) CRYSTAL STRUCTURE OF VPS34 IN COMPLEX WITH SAR405. | LIPID KINASE
1y2m:A (ALA648) to (LEU715) CRYSTAL STRUCTURE OF PHENYLALANINE AMMONIA-LYASE FROM YEAST RHODODPORIDIUM TORULOIDES | ALPHA HELICES, LYASE
1y2m:B (ALA648) to (ALA716) CRYSTAL STRUCTURE OF PHENYLALANINE AMMONIA-LYASE FROM YEAST RHODODPORIDIUM TORULOIDES | ALPHA HELICES, LYASE
5d1w:C (SER138) to (HIS205) CRYSTAL STRUCTURE OF MYCOBACTERIUM TUBERCULOSIS RV3249C TRANSCRIPTIONAL REGULATOR. | MYCOBACTERIUM TUBERCULOSIS, TRANSCRIPTIONAL REGULATOR, TRANSCRIPTION
4p19:C (VAL335) to (GLU416) CLOSED, APO INWARD-FACING STATE OF THE GLUTAMATE TRANSPORTER HOMOLOGUE GLTPH | MEMBRANE PROTEIN, SODIUM-COUPLED ASPARTATE TRANSPORTER, INWARD-FACING STATE, APO FORM, TRANSPORT PROTEIN
5d3u:A (THR107) to (SER177) CRYSTAL STRUCTURE OF THE 5-SELECTIVE H176F MUTANT OF CYTOCHROME TXTE | CYTOCHROME, P450, HEME, REGIOSELECTIVITY, F/G LOOP, OXIDOREDUCTASE
5d3u:B (THR107) to (SER177) CRYSTAL STRUCTURE OF THE 5-SELECTIVE H176F MUTANT OF CYTOCHROME TXTE | CYTOCHROME, P450, HEME, REGIOSELECTIVITY, F/G LOOP, OXIDOREDUCTASE
5d40:B (THR107) to (SER177) CRYSTAL STRUCTURE OF THE 5-SELECTIVE H176Y MUTANT OF CYTOCHROME TXTE | CYTOCHROME, P450, HEME, REGIOSELECTIVITY, F/G LOOP, OXIDOREDUCTASE
2zy9:A (TRP352) to (ALA449) IMPROVED CRYSTAL STRUCTURE OF MAGNESIUM TRANSPORTER MGTE | MEMBRANE PROTIEN, METAL TRANSPORT
2zy9:B (GLY361) to (GLU448) IMPROVED CRYSTAL STRUCTURE OF MAGNESIUM TRANSPORTER MGTE | MEMBRANE PROTIEN, METAL TRANSPORT
4p6v:E (ASN119) to (VAL196) CRYSTAL STRUCTURE OF THE NA+-TRANSLOCATING NADH: UBIQUINONE OXIDOREDUCTASE FROM VIBRIO CHOLERAE | RESPIRATORY COMPLEX, NADH:UBIQUINONE OXIDOREDUCTASE, SODIUM TRANSLOCATION, FAD, COVALENT FMN, RIBOFLAVIN, OXIDOREDUCTASE
1ya3:A (PRO738) to (LYS820) CRYSTAL STRUCTURE OF THE HUMAN MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN BOUND TO PROGESTERONE AND HARBORING THE S810L MUTATION RESPONSIBLE FOR A SEVERE FORM OF HYPERTENSION | MINERALOCORTICOID RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR TRANSCRIPTION REGULATION, ACTIVATING MUTATION, HYPERTENSION
1mro:A (PRO282) to (TYR358) METHYL-COENZYME M REDUCTASE | BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE, METHANOGENESIS
1mro:D (PRO282) to (TYR358) METHYL-COENZYME M REDUCTASE | BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE, METHANOGENESIS
4aiu:A (LYS381) to (GLU456) A COMPLEX STRUCTURE OF BTGH84 | HYDROLASE, GLYCOSIDE HYDROLASE, INHIBITOR COMPLEX
1mzn:A (VAL232) to (LYS321) CRYSTAL STRUCTURE AT 1.9 ANGSTROEMS RESOLUTION OF THE HOMODIMER OF HUMAN RXR ALPHA LIGAND BINDING DOMAIN BOUND TO THE SYNTHETIC AGONIST COMPOUND BMS 649 AND A COACTIVATOR PEPTIDE | TRANSCRIPTION, NUCLEAR RECEPTOR, RETINOIC ACID RECEPTORS, AGONIST
5dca:A (SER1848) to (VAL1892) CRYSTAL STRUCTURE OF YEAST FULL LENGTH BRR2 IN COMPLEX WITH PRP8 JAB1 DOMAIN | PROTEIN COMPLEX, HELICASE, RNP REMODELING, SPLICEOSOME ACTIVATION, HYDROLASE
5dlb:A (PRO169) to (PHE207) CRYSTAL STRUCTURE OF CHAPERONE ESPG3 OF ESX-3 TYPE VII SECRETION SYSTEM FROM MYCOBACTERIUM MARINUM M | CHAPERONE, VIRULENCE, ESX, SECRETION, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC
5dlq:B (SER737) to (ASN788) CRYSTAL STRUCTURE OF RANGTP-EXPORTIN 4-EIF5A COMPLEX | ACTIVE TRANSPORT, NUCLEAR TRANSPORT, NUCLEAR EXPORT IMPORTIN-BETA FAMILY, EXPORTIN, HEAT REPEAT, GTPASE, NUCLEOTIDE BINDING, EIF5A, TRANSLATION FACTOR, HYPUSINE, UNUSUAL AMINO ACID, PROTEIN TRANSPORT
3lb1:B (GLY1) to (MET49) TWO-SITE COMPETITIVE INHIBITION IN DEHALOPEROXIDASE-HEMOGLOBIN | PEROXIDASE, GLOBIN, OXIDOREDUCTASE, HEME, OXYGEN TRANSPORT, TRANSPORT
3ajb:A (SER86) to (VAL190) CRYSTAL STRUCTURE OF HUMAN PEX3P IN COMPLEX WITH N-TERMINAL PEX19P PEPTIDE | ALL ALPHA, PROTEIN-PROTEIN COMPLEX, PROTEIN TRANSPORT
1z77:A (LEU121) to (MSE198) CRYSTAL STRUCTURE OF TRANSCRIPTIONAL REGULATOR PROTEIN FROM THERMOTOGA MARITIMA. | TRANSCRIPTIONAL REGULATOR, TETR FAMILY, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG
3aka:A (ARG27) to (ARG101) STRUCTURAL BASIS FOR PROKARYOTIC CALCIUM-MEDIATED REGULATION BY A STREPTOMYCES COELICOLOR CALCIUM-BINDING PROTEIN | CALCIUM-BINDING PROTEIN, EF-HAND, METAL BINDING PROTEIN
4apu:A (PRO686) to (ARG766) PR X-RAY STRUCTURES IN AGONIST CONFORMATIONS REVEAL TWO DIFFERENT MECHANISMS FOR PARTIAL AGONISM IN 11BETA-SUBSTITUTED STEROID | TRANSCRIPTION, ASOPRISNIL, PARTIAL AGONIST
5dv5:A (TYR153) to (SER221) THE FATTY ACID-RESPONSIVE FADR REPRESSOR OF VIBRIO ALGINOLYTICUS COMPLEX WITH PALMITOYL-COA | FATTY ACID-RESPONSIVE FADR REPRESSOR, PALMITOYL1-COA ESTER BINDING, DNA BINDING, TRANSCRIPTION
5dwe:B (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 2-CHLORO-SUBSTITUTED TRIARYL-IMINE ANALOG 4,4'-[(2- CHLOROPHENYL)CARBONIMIDOYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
1zkg:B (ARG126) to (GLY197) CRYSTAL STRUCTURE OF TRANSCRIPTIONAL REGULATOR, TETR FAMILY (TM1030) FROM THERMOTOGA MARITIMA AT 2.30 A RESOLUTION | TM1030, TRANSCRIPTIONAL REGULATOR, TETR FAMILY, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI, TRANSCRIPTION REGULATOR
5dxg:A (THR311) to (SER395) ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN Y537S MUTANT IN COMPLEX WITH STAPLED PEPTIDE SRC2-P5 | ESTROGEN RECEPTOR, HORMONE, STAPLED PEPTIDE, PEPTIDE MIMETIC, BREAST CANCER, HORMONE RECEPTOR-PEPTIDE COMPLEX
5dxe:A (THR311) to (SER395) ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN Y537S MUTANT IN COMPLEX WITH STAPLED PEPTIDE SRC2-P4 AND ESTRADIOL | ESTROGEN RECEPTOR ALPHA, STAPLED PEPTIDE, PEPTIDE MIMETIC, BREAST CANCER, HORMONE, SOMATIC MUTATION, HORMONE RECEPTOR-PEPTIDE COMPLEX
4q2e:A (ILE29) to (TYR88) CRYSTAL STRUCTURE OF AN INTRAMEMBRANE CDP-DAG SYNTHETASE CENTRAL FOR PHOSPHOLIPID BIOSYNTHESIS (S200C/S258C, ACTIVE MUTANT) | INTRAMEMBRANE ENZYME, CDSA FOLD, PHOSPHOLIPID BIOSYNTHESIS LIPID METABOLISM, CTP AND PHOSPHATIDIC ACID BINDING, NUCLEOTIDYLTRANSFERASE, MEMBRANE, TRANSFERASE
4q2e:B (ARG27) to (TYR88) CRYSTAL STRUCTURE OF AN INTRAMEMBRANE CDP-DAG SYNTHETASE CENTRAL FOR PHOSPHOLIPID BIOSYNTHESIS (S200C/S258C, ACTIVE MUTANT) | INTRAMEMBRANE ENZYME, CDSA FOLD, PHOSPHOLIPID BIOSYNTHESIS LIPID METABOLISM, CTP AND PHOSPHATIDIC ACID BINDING, NUCLEOTIDYLTRANSFERASE, MEMBRANE, TRANSFERASE
5e15:A (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH THE CYCLOFENIL DERIVATIVE 4,4'-{[4-(2-HYDROXYETHYL) CYCLOHEXYLIDENE]METHANEDIYL}DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
3aou:A (MET1) to (LEU61) STRUCTURE OF THE NA+ UNBOUND ROTOR RING MODIFIED WITH N,N F- DICYCLOHEXYLCARBODIIMIDE OF THE NA+-TRANSPORTING V-ATPASE | SODIUM ION TRANSPORT, V-ATPASE, DCCD, MEMBRANE ROTOR RING, HYDROLASE
3aou:C (MET1) to (LEU61) STRUCTURE OF THE NA+ UNBOUND ROTOR RING MODIFIED WITH N,N F- DICYCLOHEXYLCARBODIIMIDE OF THE NA+-TRANSPORTING V-ATPASE | SODIUM ION TRANSPORT, V-ATPASE, DCCD, MEMBRANE ROTOR RING, HYDROLASE
4aw3:A (ALA104) to (LEU169) STRUCTURE OF THE MIXED-FUNCTION P450 MYCG F286V MUTANT IN COMPLEX WITH MYCINAMICIN V IN P1 SPACE GROUP | OXIDOREDUCTASE, MYCINAMICIN BIOSYNTHESIS
4aw3:B (ALA104) to (LEU169) STRUCTURE OF THE MIXED-FUNCTION P450 MYCG F286V MUTANT IN COMPLEX WITH MYCINAMICIN V IN P1 SPACE GROUP | OXIDOREDUCTASE, MYCINAMICIN BIOSYNTHESIS
4aw6:D (ILE98) to (GLY192) CRYSTAL STRUCTURE OF THE HUMAN NUCLEAR MEMBRANE ZINC METALLOPROTEASE ZMPSTE24 (FACE1) | HYDROLASE, M48 PEPTIDASE, INTEGRAL MEMBRANE PROTEIN, PRELAMIN A PROCESSING, AGEING, PROGERIA
4q71:A (GLY57) to (LEU99) CRYSTAL STRUCTURE OF BRADYRHIZOBIUM JAPONICUM PROLINE UTILIZATION A (PUTA) MUTANT D779W | PROLINE UTILIZATION A, PUTA, BETA-ALPHA BARREL, ROSSMANN FOLD, PROLINE DEHYDROGENASE, 1-PYRROLINE-5-CARBOXYLATE DEHYDROGENASE, FAD BINDING, OXIDOREDUCTASE
3m2r:A (PRO282) to (TYR358) STRUCTURAL INSIGHT INTO METHYL-COENZYME M REDUCTASE CHEMISTRY USING COENZYME B ANALOGUES | METHYL-COENZYME M REDUCTASE, NICKEL, METAL-BINDING, METHANOGENESIS, METHYLATION, TRANSFERASE
3m2r:D (PHE283) to (ASP356) STRUCTURAL INSIGHT INTO METHYL-COENZYME M REDUCTASE CHEMISTRY USING COENZYME B ANALOGUES | METHYL-COENZYME M REDUCTASE, NICKEL, METAL-BINDING, METHANOGENESIS, METHYLATION, TRANSFERASE
3m2v:A (PHE283) to (TYR358) STRUCTURAL INSIGHT INTO METHYL-COENZYME M REDUCTASE CHEMISTRY USING COENZYME B ANALOGUES | METHYL-COENZYME M REDUCTASE, NICKEL, METAL-BINDING, METHANOGENESIS, METHYLATION, TRANSFERASE
3m2v:D (PHE283) to (TYR358) STRUCTURAL INSIGHT INTO METHYL-COENZYME M REDUCTASE CHEMISTRY USING COENZYME B ANALOGUES | METHYL-COENZYME M REDUCTASE, NICKEL, METAL-BINDING, METHANOGENESIS, METHYLATION, TRANSFERASE
3m30:A (PRO282) to (TYR358) STRUCTURAL INSIGHT INTO METHYL-COENZYME M REDUCTASE CHEMISTRY USING COENZYME B ANALOGUES | METHYL-COENZYME M REDUCTASE, NICKEL, METAL-BINDING, METHANOGENESIS, METHYLATION, TRANSFERASE
3m30:D (PRO282) to (LYS357) STRUCTURAL INSIGHT INTO METHYL-COENZYME M REDUCTASE CHEMISTRY USING COENZYME B ANALOGUES | METHYL-COENZYME M REDUCTASE, NICKEL, METAL-BINDING, METHANOGENESIS, METHYLATION, TRANSFERASE
3b0b:C (LYS10) to (PHE79) CRYSTAL STRUCTURE OF THE CHICKEN CENP-S/CENP-X COMPLEX | HISTONE FOLD, DNA BINDING, DNA, NUCLEUS, DNA BINDING PROTEIN
3b0b:D (ARG9) to (PHE79) CRYSTAL STRUCTURE OF THE CHICKEN CENP-S/CENP-X COMPLEX | HISTONE FOLD, DNA BINDING, DNA, NUCLEUS, DNA BINDING PROTEIN
3b7r:L (PRO400) to (LEU448) LEUKOTRIENE A4 HYDROLASE COMPLEXED WITH INHIBITOR RB3040 | TRANSITION STATE, ANALOGUE PEPTIDE, HYDROLYSIS, ALTERNATIVE SPLICING, CYTOPLASM, HYDROLASE, LEUKOTRIENE BIOSYNTHESIS, METAL-BINDING, METALLOPROTEASE, MULTIFUNCTIONAL ENZYME, PROTEASE, ZINC
3b7t:A (PRO400) to (LEU448) [E296Q]LTA4H IN COMPLEX WITH ARG-ALA-ARG SUBSTRATE | TRANSITION STATE, ANALOGUE PEPTIDE, HYDROLYSIS, ALTERNATIVE SPLICING, CYTOPLASM, HYDROLASE, LEUKOTRIENE BIOSYNTHESIS, METAL-BINDING, METALLOPROTEASE, MULTIFUNCTIONAL ENZYME, PROTEASE, ZINC, TRIPEPTIDE SUBSTRATE
4bcr:A (GLY262) to (MET320) STRUCTURE OF PPARALPHA IN COMPLEX WITH WY14643 | TRANSCRIPTION, NUCLEAR RECEPTOR, PPAR, FIBRATE
3bcg:A (MET123) to (CYS205) CONFORMATIONAL CHANGES OF THE ACRR REGULATOR REVEAL A MECHANISM OF INDUCTION | ACRB REGULATOR, DNA-BINDING, REPRESSOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, DNA BINDING PROTEIN, TRANSCRIPTION REGULATOR
3bcg:B (MET123) to (CYS205) CONFORMATIONAL CHANGES OF THE ACRR REGULATOR REVEAL A MECHANISM OF INDUCTION | ACRB REGULATOR, DNA-BINDING, REPRESSOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, DNA BINDING PROTEIN, TRANSCRIPTION REGULATOR
3mji:D (ALA217) to (ASN263) ACTIVATION OF CATALYTIC CYSTEINE WITHOUT A BASE IN A MUTANT PENICILLIN ACYLASE PRECURSOR | ZYMOGEN, HYDROLASE, PENICILLIN, AUTOPROTEOLYSIS, ANTIBIOTIC RESISTANCE, CATALYSIS, PENICILLIN V ACYLASE, AMIDASE
3mk4:A (SER86) to (GLY192) X-RAY STRUCTURE OF HUMAN PEX3 IN COMPLEX WITH A PEX19 DERIVED PEPTIDE | MEMBRANE, PEROXISOME, PROTEIN TRANSPORT
4bem:J (ASN6) to (LEU93) CRYSTAL STRUCTURE OF THE F-TYPE ATP SYNTHASE C-RING FROM ACETOBACTERIUM WOODII. | HYDROLASE
5epg:A (LYS474) to (ASP538) HUMAN ALDEHYDE OXIDASE SNP S1271L | OXIDOREDUCTASE, DRUG METABOLISM, SNP
4qr8:A (TYR270) to (PRO334) CRYSTAL STRUCTURE OF E COLI PEPQ | PEPQ, PROTEASE, HYDROLASE
4qr8:B (ASP269) to (PRO334) CRYSTAL STRUCTURE OF E COLI PEPQ | PEPQ, PROTEASE, HYDROLASE
3bg5:B (HIS333) to (ASN361) CRYSTAL STRUCTURE OF STAPHYLOCOCCUS AUREUS PYRUVATE CARBOXYLASE | TIM BARREL, ATP-BINDING, LIGASE, NUCLEOTIDE-BINDING, PYRUVATE
3mno:A (LEU538) to (ALA622) CRYSTAL STRUCTURE OF THE AGONIST FORM OF MOUSE GLUCOCORTICOID RECEPTOR STABILIZED BY (A611V, F608S) MUTATIONS AT 1.55A | PROTEIN-LIGAND COMPLEX, STEROID NUCLEAR RECEPTOR, MOUSE GR, AGONIST, CO-ACTIVATOR, HORMONE RECEPTOR
3mnp:A (LEU538) to (SER623) CRYSTAL STRUCTURE OF THE AGONIST FORM OF MOUSE GLUCOCORTICOID RECEPTOR STABILIZED BY (A611V, V708A, E711G) MUTATIONS AT 1.50A | PROTEIN-LIGAND COMPLEX, STEROID NUCLEAR RECEPTOR, MOUSE GR, AGONIST, CO-ACTIVATOR, HORMONE RECEPTOR
4bjk:C (THR135) to (SER206) CYP51 OF TRYPANOSOMA BRUCEI BOUND TO (S)-N-(3-(1H-INDOL-3- YL)-1-OXO-1-(PYRIDIN-4-YLAMINO)PROPAN-2-YL)-3,3'-DIFLUORO-( 1,1'-BIPHENYL)-4-CARBOXAMIDE | OXIDOREDUCTASE, ERGOSTEROL BIOSYNTHESIS
4quw:A (ALA185) to (VAL231) CRYSTAL STRUCTURE OF THE APO FORM OF CYANOBACTERIAL ALDEHYDE- DEFORMYLATING OXYGENASE | OXYGENASE, LYASE
4qvg:A (PRO80) to (PRO141) CRYSTAL STRUCTURE OF S-ADENOSYLMETHIONINE-DEPENDENT METHYLTRANSFERASE SIBL IN ITS APO FORM | METHYLTRANSFERASE, TRANSFERASE
5f15:A (PRO87) to (PHE154) CRYSTAL STRUCTURE OF ARNT FROM CUPRIAVIDUS METALLIDURANS BOUND TO UNDECAPRENYL PHOSPHATE | MEMBRANE PROTEIN, LIPID GLYCOSYLTRANSFERASE, GT-C FOLD, UNDECAPRENYL PHOSPHATE, STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK CONSORTIUM ON MEMBRANE PROTEIN STRUCTURE, NYCOMPS, TRANSFERASE
3brj:A (SER8) to (LEU67) CRYSTAL STRUCTURE OF MANNITOL OPERON REPRESSOR (MTLR) FROM VIBRIO PARAHAEMOLYTICUS RIMD 2210633 | APC85967.1, MANNITOL OPERON REPRESSOR, MTLR, VIBRIO PARAHAEMOLYTICUS RIMD 2210633, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSCRIPTION
3brj:B (ILE5) to (LEU67) CRYSTAL STRUCTURE OF MANNITOL OPERON REPRESSOR (MTLR) FROM VIBRIO PARAHAEMOLYTICUS RIMD 2210633 | APC85967.1, MANNITOL OPERON REPRESSOR, MTLR, VIBRIO PARAHAEMOLYTICUS RIMD 2210633, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSCRIPTION
3brj:C (ASN6) to (LEU67) CRYSTAL STRUCTURE OF MANNITOL OPERON REPRESSOR (MTLR) FROM VIBRIO PARAHAEMOLYTICUS RIMD 2210633 | APC85967.1, MANNITOL OPERON REPRESSOR, MTLR, VIBRIO PARAHAEMOLYTICUS RIMD 2210633, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSCRIPTION
3brj:D (ILE5) to (LEU67) CRYSTAL STRUCTURE OF MANNITOL OPERON REPRESSOR (MTLR) FROM VIBRIO PARAHAEMOLYTICUS RIMD 2210633 | APC85967.1, MANNITOL OPERON REPRESSOR, MTLR, VIBRIO PARAHAEMOLYTICUS RIMD 2210633, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSCRIPTION
3mwt:C (PRO180) to (PRO227) CRYSTAL STRUCTURE OF LASSA FEVER VIRUS NUCLEOPROTEIN IN COMPLEX WITH MN2+ | NUCLEOPROTEIN, LASSA FEVER VIRUS, STRUCTURAL GENOMICS, SCOTTISH STRUCTURAL PROTEOMICS FACILITY, SSPF, NUCLEAR PROTEIN
3mx2:A (PRO180) to (PRO227) LASSA FEVER VIRUS NUCLEOPROTEIN COMPLEXED WITH DTTP | NUCLEOPROTEIN, LASSA FEVER VIRUS, STRUCTURAL GENOMICS, SCOTTISH STRUCTURAL PROTEOMICS FACILITY, SSPF, NUCLEAR PROTEIN
3mx5:B (PRO180) to (PRO227) LASSA FEVER VIRUS NUCLEOPROTEIN COMPLEXED WITH UTP | NUCLEOPROTEIN, LASSA FEVER VIRUS, STRUCTURAL GENOMICS, SCOTTISH STRUCTURAL PROTEOMICS FACILITY, SSPF, NUCLEAR PROTEIN
4buj:A (LEU1112) to (GLN1193) CRYSTAL STRUCTURE OF THE S. CEREVISIAE SKI2-3-8 COMPLEX | HYDROLASE, DEXH BOX HELICASE, RNA DEGRADATION, TPR, PROTEIN COMPLEX
4buj:E (LEU1112) to (GLN1193) CRYSTAL STRUCTURE OF THE S. CEREVISIAE SKI2-3-8 COMPLEX | HYDROLASE, DEXH BOX HELICASE, RNA DEGRADATION, TPR, PROTEIN COMPLEX
4r3u:B (GLY243) to (LEU285) CRYSTAL STRUCTURE OF 2-HYDROXYISOBUTYRYL-COA MUTASE | TIM ROSSMANN FOLD, MUTASE, COA, ISOMERASE
4c0c:A (PHE142) to (LEU208) CRYSTAL STRUCTURE OF TRYPANOSOMA CRUZI CYP51 BOUND TO THE INHIBITOR (R)-N-(3-(1H-INDOL-3-YL)-1-OXO-1-(PYRIDIN-4- YLAMINO)PROPAN-2-YL)-4-(4-(2,4-DIFLUOROPHENYL)PIPERAZIN-1- YL)-2-FLUOROBENZAMIDE. | OXIDOREDUCTASE, STEROL BIOSYNTHESIS, CHAGAS DISEASE
4c27:A (PHE142) to (SER207) CRYSTAL STRUCTURE OF TRYPANOSOMA CRUZI CYP51 BOUND TO THE INHIBITOR (R)-N-(3-(1H-INDOL-3-YL)-1-OXO-1-(PYRIDIN-4- 4-YLAMINO)PROPAN-2-YL)-2-FLUORO-4-(4-(4-(TRIFLUOROMETHYL) PHENYL)PIPERAZIN-1-YL)BENZAMIDE | OXIDOREDUCTASE, STEROL BIOSYNTHESIS, CHAGAS DISEASE
4c27:B (PHE142) to (SER207) CRYSTAL STRUCTURE OF TRYPANOSOMA CRUZI CYP51 BOUND TO THE INHIBITOR (R)-N-(3-(1H-INDOL-3-YL)-1-OXO-1-(PYRIDIN-4- 4-YLAMINO)PROPAN-2-YL)-2-FLUORO-4-(4-(4-(TRIFLUOROMETHYL) PHENYL)PIPERAZIN-1-YL)BENZAMIDE | OXIDOREDUCTASE, STEROL BIOSYNTHESIS, CHAGAS DISEASE
4req:A (GLY242) to (LEU284) METHYLMALONYL-COA MUTASE SUBSTRATE COMPLEX | ISOMERASE, MUTASE, INTRAMOLECULAR TRANSFERASE
4req:C (GLY242) to (LEU284) METHYLMALONYL-COA MUTASE SUBSTRATE COMPLEX | ISOMERASE, MUTASE, INTRAMOLECULAR TRANSFERASE
3cjw:A (SER174) to (SER261) CRYSTAL STRUCTURE OF THE HUMAN COUP-TFII LIGAND BINDING DOMAIN | COUP-TFII, NUCLEAR RECEPTOR, LIGAND BINDING DOMAIN, ORPHAN RECEPTOR, THREE-LAYERED HELICAL SANDWICH, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER
5fru:A (THR44) to (GLY106) CRYSTAL STRUCTURE OF THE PHENOL-RESPONSIVE SENSORY DOMAIN OF THE TRANSCRIPTION ACTIVATOR POXR | TRANSCRIPTION, PHENOL, POXR, DMPR, ENHANCER-BINDING PROTEIN, ACTIVATOR, ATPASE FAMILY
5frv:A (THR44) to (GLY106) CRYSTAL STRUCTURE OF THE PHENOL-RESPONSIVE SENSORY DOMAIN OF THE TRANSCRIPTION ACTIVATOR POXR IN COMPLEX WITH 4-METHYLPHENOL (CRESOL) | TRANSCRIPTION, PHENOL, POXR, DMPR, ENHANCER-BINDING PROTEIN, ACTIVATOR, ATPASE FAMILY
5frv:B (HIS43) to (GLY106) CRYSTAL STRUCTURE OF THE PHENOL-RESPONSIVE SENSORY DOMAIN OF THE TRANSCRIPTION ACTIVATOR POXR IN COMPLEX WITH 4-METHYLPHENOL (CRESOL) | TRANSCRIPTION, PHENOL, POXR, DMPR, ENHANCER-BINDING PROTEIN, ACTIVATOR, ATPASE FAMILY
5frw:B (THR44) to (GLU105) CRYSTAL STRUCTURE OF THE PHENOL-RESPONSIVE SENSORY DOMAIN OF THE TRANSCRIPTION ACTIVATOR POXR WITH PHENOL | TRANSCRIPTION, PHENOL, DMPR, ENHANCER-BINDING PROTEIN, ACTIVATOR, ATPASE FAMILY
5frx:A (THR44) to (GLU105) CRYSTAL STRUCTURE OF THE PHENOL-RESPONSIVE SENSORY DOMAIN OF THE TRANSCRIPTION ACTIVATOR POXR IN COMPLEX WITH 4-NITROPHENOL | TRANSCRIPTION, PHENOL, DMPR, ENHANCER-BINDING PROTEIN, ACTIVATOR, ATPASE FAMILY
5frx:B (THR44) to (GLY106) CRYSTAL STRUCTURE OF THE PHENOL-RESPONSIVE SENSORY DOMAIN OF THE TRANSCRIPTION ACTIVATOR POXR IN COMPLEX WITH 4-NITROPHENOL | TRANSCRIPTION, PHENOL, DMPR, ENHANCER-BINDING PROTEIN, ACTIVATOR, ATPASE FAMILY
5fry:B (THR44) to (GLY106) CRYSTAL STRUCTURE OF THE PHENOL-RESPONSIVE SENSORY DOMAIN OF THE TRANSCRIPTION ACTIVATOR POXR WITH 3,5-DIMETHYLPHENOL | TRANSCRIPTION, PHENOL, DMPR, ENHANCER-BINDING PROTEIN, ACTIVATOR, ATPASE FAMILY
5frz:A (THR44) to (GLY106) CRYSTAL STRUCTURE OF THE PHENOL-RESPONSIVE SENSORY DOMAIN OF THE TRANSCRIPTION ACTIVATOR POXR WITH 3,4-DIMETHYLPHENOL | TRANSCRIPTION, PHENOL, DMPR, ENHANCER-BINDING PROTEIN, ACTIVATOR, ATPASE FAMILY
5frz:B (HIS43) to (GLU105) CRYSTAL STRUCTURE OF THE PHENOL-RESPONSIVE SENSORY DOMAIN OF THE TRANSCRIPTION ACTIVATOR POXR WITH 3,4-DIMETHYLPHENOL | TRANSCRIPTION, PHENOL, DMPR, ENHANCER-BINDING PROTEIN, ACTIVATOR, ATPASE FAMILY
3nv5:A (GLU129) to (MET185) CRYSTAL STRUCTURE OF CYTOCHROME P450 CYP101D2 | CYTOCHROME P450 FOLD, OXIDIZING CAMPHOR, OXIDOREDUCTASE
3nv6:A (GLU129) to (MET185) CRYSTAL STRUCTURE OF CAMPHOR-BOUND CYP101D2 | CYTOCHROME P450 FOLD, OXIDIZING CAMPHOR, OXIDOREDUCTASE
4rsy:A (GLY399) to (LEU448) CRYSTAL STRUCTURES OF THE HUMAN LEUKOTRIENE A4 HYDROLASE COMPLEX WITH A POTENTIAL INHIBITOR H7 | HUMAN LEUKOTRIENE A4 HYDROLASE, LTA4H', HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5fwq:A (GLY399) to (LEU448) APO STRUCTURE OF HUMAN LEUKOTRIENE A4 HYDROLASE | HYDROLASE, LEUKOTRIENE (LT) A4 HYDROLASE/AMINOPEPTIDASE, LTA4H
3o1e:A (TYR179) to (ARG302) STRUCTURE-FUNCTION OF GEMINI DERIVATIVES WITH TWO DIFFERENT SIDE CHAINS AT C-20, GEMINI-0072 AND GEMINI-0097. | TRANSCRIPTION FACTOR, VITAMIN D, NUCLEUS, TRANSCRIPTION-TRANSCRIPTION ACTIVATOR COMPLEX
3o7n:B (GLY1) to (MET49) THE V59W MUTATION BLOCKS THE DISTAL POCKET OF THE HEMOGLOBIN - DEHALOPEROXIDASE FROM AMPHITRITE ORNATA | PEROXIDASE, GLOBIN, OXYGEN TRANSPORT
5g04:I (THR238) to (THR326) STRUCTURE OF THE HUMAN APC-CDC20-HSL1 COMPLEX | CELL CYCLE, PHOSPHORYLATION, MITOSIS, UBIQUITINATION
3o8u:A (ASN269) to (ALA309) CONFORMATIONAL PLASTICITY OF P38 MAP KINASE DFG MOTIF MUTANTS IN RESPONSE TO INHIBITOR BINDING | TRANSFERASE
5g0r:A (PRO282) to (TYR358) METHYL-COENZYME M REDUCTASE I FROM METHANOTHERMOBACTER MARBURGENSIS EXPOSED TO 3-NITROOXYPROPANOL | TRANSFERASE, METHYL-COENZYMEM, METHYL-COENZYMEM REDUCTASE EXPOSED TO 3-NITROOXYPROPANOL, POSTTRANSLATIONAL MODIFICATION, BINDING SITES, CATALYSIS, COENZYMES, DISULFIDES, HYDROGEN, LIGANDS, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, NICKEL, OXIDATION-REDUCTION, OXDOREDUCTASES, PHOSPHOTHREONINE, THIOGLYCINE, 3- NITROOXYPROPANOL, INHIBITOR, GREENHOUSE GAS
5g0r:D (PRO282) to (TYR358) METHYL-COENZYME M REDUCTASE I FROM METHANOTHERMOBACTER MARBURGENSIS EXPOSED TO 3-NITROOXYPROPANOL | TRANSFERASE, METHYL-COENZYMEM, METHYL-COENZYMEM REDUCTASE EXPOSED TO 3-NITROOXYPROPANOL, POSTTRANSLATIONAL MODIFICATION, BINDING SITES, CATALYSIS, COENZYMES, DISULFIDES, HYDROGEN, LIGANDS, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, NICKEL, OXIDATION-REDUCTION, OXDOREDUCTASES, PHOSPHOTHREONINE, THIOGLYCINE, 3- NITROOXYPROPANOL, INHIBITOR, GREENHOUSE GAS
3oaa:E (GLY378) to (LEU459) STRUCTURE OF THE E.COLI F1-ATP SYNTHASE INHIBITED BY SUBUNIT EPSILON | ROSSMANN FOLD, HYDROLASE, SYNTHASE, HYDROLASE-TRANSPORT PROTEIN COMPLEX
3oaa:M (GLY378) to (LEU459) STRUCTURE OF THE E.COLI F1-ATP SYNTHASE INHIBITED BY SUBUNIT EPSILON | ROSSMANN FOLD, HYDROLASE, SYNTHASE, HYDROLASE-TRANSPORT PROTEIN COMPLEX
3oaa:U (GLY378) to (LEU459) STRUCTURE OF THE E.COLI F1-ATP SYNTHASE INHIBITED BY SUBUNIT EPSILON | ROSSMANN FOLD, HYDROLASE, SYNTHASE, HYDROLASE-TRANSPORT PROTEIN COMPLEX
4csj:A (VAL533) to (GLN615) THE DISCOVERY OF POTENT SELECTIVE GLUCOCORTICOID RECEPTOR MODULATORS, SUITABLE FOR INHALATION | SIGNALING PROTEIN, NUCLEAR HORMONE RECEPTOR, LIGAND COMPLEX, PEPTIDE COMPLEX
3ofm:A (ARG281) to (TYR326) STRUCTURE OF A HUMAN CK2ALPHA PRIME, THE PARALOG ISOFORM OF THE CATALYTIC SUBUNIT OF PROTEIN KINASE CK2 FROM HOMO SAPIENS | EUKARYPTIC PROTEIN KINASE FOLD, PHOSPHO TRANSFERASE, ATP BINDING, PHOSPHORYLATION, CYTOPLASM AND NUCLEUS, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3ofs:C (PHE59) to (LEU112) DYNAMIC CONFORMATIONS OF THE CD38-MEDIATED NAD CYCLIZATION CAPTURED USING MULTI-COPY CRYSTALLOGRAPHY | CD38, CYCLIZATION, HYDROLYSIS, CADPR, ADPR, ARA-2'F-NAD, ARA-2'F- ADPR, HYDROLASE
3ofs:D (PHE59) to (LEU112) DYNAMIC CONFORMATIONS OF THE CD38-MEDIATED NAD CYCLIZATION CAPTURED USING MULTI-COPY CRYSTALLOGRAPHY | CD38, CYCLIZATION, HYDROLYSIS, CADPR, ADPR, ARA-2'F-NAD, ARA-2'F- ADPR, HYDROLASE
3ofs:F (ARG58) to (LEU112) DYNAMIC CONFORMATIONS OF THE CD38-MEDIATED NAD CYCLIZATION CAPTURED USING MULTI-COPY CRYSTALLOGRAPHY | CD38, CYCLIZATION, HYDROLYSIS, CADPR, ADPR, ARA-2'F-NAD, ARA-2'F- ADPR, HYDROLASE
4tvq:A (LEU58) to (ARG124) CCM3 IN COMPLEX WITH CCM2 LD-LIKE MOTIF | FAT-HOMOLOGY DOMAIN, PROTEIN BINDING
4d9i:A (SER315) to (ALA364) CRYSTAL STRUCTURE OF HOLO DIAMINOPROPIONATE AMMONIA LYASE FROM ESCHERICHIA COLI | FOLD TYPE II PLP-DEPENDENT ENZYME, TRYPTOPHAN SYNTHASE BETA SUBUNIT- LIKE PLP-DEPENDENT ENZYMES SUPERFAMILY, LYASE
3ord:B (GLY1) to (MET49) STRUCTURAL EVIDENCE FOR STABILIZATION OF INHIBITOR BINDING BY A PROTEIN CAVITY IN THE DEHALOPEROXIDASE-HEMOGLOBIN FROM AMPHITRITE ORNATA | GLOBIN, PEROXIDASE, OXIDOREDUCTASE
5hi9:A (LEU498) to (ASN650) STRUCTURE OF THE FULL-LENGTH TRPV2 CHANNEL BY CRYO-ELECTRON MICROSCOPY | TRPV2 ION CHANNEL, TRANSPORT PROTEIN
5hi9:B (LEU498) to (ASN650) STRUCTURE OF THE FULL-LENGTH TRPV2 CHANNEL BY CRYO-ELECTRON MICROSCOPY | TRPV2 ION CHANNEL, TRANSPORT PROTEIN
5hi9:C (LEU498) to (ASN650) STRUCTURE OF THE FULL-LENGTH TRPV2 CHANNEL BY CRYO-ELECTRON MICROSCOPY | TRPV2 ION CHANNEL, TRANSPORT PROTEIN
5hi9:D (LEU498) to (ASN650) STRUCTURE OF THE FULL-LENGTH TRPV2 CHANNEL BY CRYO-ELECTRON MICROSCOPY | TRPV2 ION CHANNEL, TRANSPORT PROTEIN
4u67:G (GLU117) to (ARG147) CRYSTAL STRUCTURE OF THE LARGE RIBOSOMAL SUBUNIT (50S) OF DEINOCOCCUS RADIODURANS CONTAINING A THREE RESIDUE INSERTION IN L22 | RIBOSOME, ANTIBIOTICS, RESISTANCE, ERYTHROMYCIN
3p5k:A (ASN269) to (ALA309) P38 INHIBITOR-BOUND | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4u8v:A (ASN361) to (PHE459) COUPLING OF REMOTE ALTERNATING-ACCESS TRANSPORT MECHANISMS FOR PROTONS AND SUBSTRATES IN THE MULTIDRUG EFFLUX PUMP ACRB | MEMBRANE PROTEIN, TRANSPORT PROTEIN, DARPIN, MULTIDRUG EFFLUX PROTEIN
3p99:B (PHE139) to (SER206) STEROL 14ALPHA-DEMETHYLASE (CYP51) FROM TRYPANOSOMA BRUCEI IN COMPLEX WITH DELTA7-14ALPHA-METHYLENE-CYCLOPROPYL-DIHYDROLANOSTEROL | CYTOCHROME P450 FOLD/STEROL 14-ALPHA DEMETHYLASE, CYP51, OXIDOREDUCTASE, MONOOXYGENASE, HEMOPROTEIN, STEROL BIOSYNTHESIS, CYTOCHROME P450 REDUCTASE (CPR), ENDOPLASMIC RETICULUM, MEMBRANE
4u9l:B (ARG353) to (LEU446) STRUCTURE OF A MEMBRANE PROTEIN | CHANNEL, MAGNESIUM, METAL TRANSPORT
4u9n:A (GLU307) to (GLY382) STRUCTURE OF A MEMBRANE PROTEIN | CHANNEL, MAGNESIUM, METAL TRANSPORT
4drb:J (ARG11) to (PHE81) THE CRYSTAL STRUCTURE OF FANCM BOUND MHF COMPLEX | DNA REPAIR, DNA BINDING COMPLEX, HISTONE FOLD, DNA DAMAGE REPAIR, DNA BINDING, DNA BINDING-PROTEIN BINDING COMPLEX, DNA BINDING PROTEIN- PROTEIN BINDING COMPLEX
4drb:K (ARG11) to (PHE81) THE CRYSTAL STRUCTURE OF FANCM BOUND MHF COMPLEX | DNA REPAIR, DNA BINDING COMPLEX, HISTONE FOLD, DNA DAMAGE REPAIR, DNA BINDING, DNA BINDING-PROTEIN BINDING COMPLEX, DNA BINDING PROTEIN- PROTEIN BINDING COMPLEX
4drb:L (ARG11) to (PHE81) THE CRYSTAL STRUCTURE OF FANCM BOUND MHF COMPLEX | DNA REPAIR, DNA BINDING COMPLEX, HISTONE FOLD, DNA DAMAGE REPAIR, DNA BINDING, DNA BINDING-PROTEIN BINDING COMPLEX, DNA BINDING PROTEIN- PROTEIN BINDING COMPLEX
4drb:M (ARG11) to (PHE81) THE CRYSTAL STRUCTURE OF FANCM BOUND MHF COMPLEX | DNA REPAIR, DNA BINDING COMPLEX, HISTONE FOLD, DNA DAMAGE REPAIR, DNA BINDING, DNA BINDING-PROTEIN BINDING COMPLEX, DNA BINDING PROTEIN- PROTEIN BINDING COMPLEX
4drb:N (LYS12) to (PHE81) THE CRYSTAL STRUCTURE OF FANCM BOUND MHF COMPLEX | DNA REPAIR, DNA BINDING COMPLEX, HISTONE FOLD, DNA DAMAGE REPAIR, DNA BINDING, DNA BINDING-PROTEIN BINDING COMPLEX, DNA BINDING PROTEIN- PROTEIN BINDING COMPLEX
4drb:O (LYS12) to (PHE81) THE CRYSTAL STRUCTURE OF FANCM BOUND MHF COMPLEX | DNA REPAIR, DNA BINDING COMPLEX, HISTONE FOLD, DNA DAMAGE REPAIR, DNA BINDING, DNA BINDING-PROTEIN BINDING COMPLEX, DNA BINDING PROTEIN- PROTEIN BINDING COMPLEX
5hw2:B (PRO55) to (PHE88) CRYSTAL STRUCTURE OF ADENYLOSUCCINATE LYASE FROM FRANCISELLA TULARENSIS COMPLEXED WITH FUMARIC ACID | STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, LYASE
4udd:A (THR531) to (SER617) GR IN COMPLEX WITH DESISOBUTYRYLCICLESONIDE | SIGNALING PROTEIN, NUCLEAR HORMONE RECEPTOR, LIGAND COMPLEX, PEPTIDE COMPLEX
5hyn:C (TRP591) to (GLY644) STRUCTURE OF HUMAN POLYCOMB REPRESSIVE COMPLEX 2 (PRC2) WITH ONCOGENIC HISTONE H3K27M PEPTIDE | CHROMATIN MODIFICATION COMPLEX, TRANSFERASE
5i20:C (SER25) to (LEU88) CRYSTAL STRUCTURE OF PROTEIN | ALPHA HELICAL, MEMBRANE PROTEIN
5i20:E (SER2) to (LEU88) CRYSTAL STRUCTURE OF PROTEIN | ALPHA HELICAL, MEMBRANE PROTEIN
4uhw:A (LYS474) to (ASP538) HUMAN ALDEHYDE OXIDASE | OXIDOREDUCTASE, DRUG METABOLISM, MOLYBDENUM ENZYMES, XANTHINE OXIDASE ENZYMES,
4uhx:A (ASN475) to (MET537) HUMAN ALDEHYDE OXIDASE IN COMPLEX WITH PHTHALAZINE AND THIORIDAZINE | OXIDOREDUCTASE, ALDEHYDE OXIDASE, DRUG METABOLISM, MOLYBDENUM ENZYMES, XANTHINE OXIDASE, PHTHALAZINE, THIORIDAZINE
3pm0:A (ARG161) to (VAL235) STRUCTURAL CHARACTERIZATION OF THE COMPLEX BETWEEN ALPHA- NAPHTHOFLAVONE AND HUMAN CYTOCHROME P450 1B1 (CYP1B1) | CYP1B1, P450 1B1, P450, MONOOXYGENASE, ALPHA-NAPHTHOFLAVONE, HEME, 17BETA-ESTRADIOL, OXIDOREDUCTASE
3pot:A (PRO282) to (TYR358) STRUCTURAL ANALYSIS OF A NI(III)-METHYL SPECIES IN METHYL-COENZYME M REDUCTASE FROM METHANOTHERMOBACTER MARBURGENSIS | METAL-BINDING, NICKEL, METHYL-COENZYME M REDUCTASE, METHANOGENESIS, METHYLATION, TRANSFERASE
3pot:D (PRO282) to (ASP356) STRUCTURAL ANALYSIS OF A NI(III)-METHYL SPECIES IN METHYL-COENZYME M REDUCTASE FROM METHANOTHERMOBACTER MARBURGENSIS | METAL-BINDING, NICKEL, METHYL-COENZYME M REDUCTASE, METHANOGENESIS, METHYLATION, TRANSFERASE
4e45:B (LYS12) to (PHE81) CRYSTAL STRUCTURE OF THE HMHF1/HMHF2 HISTONE-FOLD TETRAMER IN COMPLEX WITH FANCONI ANEMIA ASSOCIATED HELICASE HFANCM | HISTONE-FOLD, PENTAMER, FANCONI ANEMIA, HELICASE, FANCM, MHF, DNA BINDING PROTEIN-HYDROLASE COMPLEX
4e45:D (LYS12) to (PHE81) CRYSTAL STRUCTURE OF THE HMHF1/HMHF2 HISTONE-FOLD TETRAMER IN COMPLEX WITH FANCONI ANEMIA ASSOCIATED HELICASE HFANCM | HISTONE-FOLD, PENTAMER, FANCONI ANEMIA, HELICASE, FANCM, MHF, DNA BINDING PROTEIN-HYDROLASE COMPLEX
4e45:G (LYS12) to (PHE81) CRYSTAL STRUCTURE OF THE HMHF1/HMHF2 HISTONE-FOLD TETRAMER IN COMPLEX WITH FANCONI ANEMIA ASSOCIATED HELICASE HFANCM | HISTONE-FOLD, PENTAMER, FANCONI ANEMIA, HELICASE, FANCM, MHF, DNA BINDING PROTEIN-HYDROLASE COMPLEX
4e45:I (LYS12) to (PHE81) CRYSTAL STRUCTURE OF THE HMHF1/HMHF2 HISTONE-FOLD TETRAMER IN COMPLEX WITH FANCONI ANEMIA ASSOCIATED HELICASE HFANCM | HISTONE-FOLD, PENTAMER, FANCONI ANEMIA, HELICASE, FANCM, MHF, DNA BINDING PROTEIN-HYDROLASE COMPLEX
4e45:L (ARG11) to (PHE81) CRYSTAL STRUCTURE OF THE HMHF1/HMHF2 HISTONE-FOLD TETRAMER IN COMPLEX WITH FANCONI ANEMIA ASSOCIATED HELICASE HFANCM | HISTONE-FOLD, PENTAMER, FANCONI ANEMIA, HELICASE, FANCM, MHF, DNA BINDING PROTEIN-HYDROLASE COMPLEX
4e45:N (LYS12) to (PHE81) CRYSTAL STRUCTURE OF THE HMHF1/HMHF2 HISTONE-FOLD TETRAMER IN COMPLEX WITH FANCONI ANEMIA ASSOCIATED HELICASE HFANCM | HISTONE-FOLD, PENTAMER, FANCONI ANEMIA, HELICASE, FANCM, MHF, DNA BINDING PROTEIN-HYDROLASE COMPLEX
4us3:A (ASP76) to (GLY167) CRYSTAL STRUCTURE OF THE BACTERIAL NSS MEMBER MHST IN AN OCCLUDED INWARD-FACING STATE | TRANSPORT PROTEIN, NEUROTRANSMITTER, NEUROTRANSMITTER SODIUM SYMPORTER FAMILY, LEUT FOLD, AMINO ACID TRANSPORTER, SECONDARY TRANSPORTER, MEMBRANE PROTEIN
3psf:A (SER340) to (SER400) CRYSTAL STRUCTURE OF THE SPT6 CORE DOMAIN FROM SACCHAROMYCES CEREVISIAE, FORM SPT6(236-1259) | TRANSCRIPTION ELONGATION, NUCLEUS, TRANSCRIPTION
3psi:A (SER340) to (SER400) CRYSTAL STRUCTURE OF THE SPT6 CORE DOMAIN FROM SACCHAROMYCES CEREVISIAE, FORM SPT6(239-1451) | TRANSCRIPTION ELONGATION, NUCLEUS, TRANSCRIPTION
4eei:A (PRO55) to (PHE88) CRYSTAL STRUCTURE OF ADENYLOSUCCINATE LYASE FROM FRANCISELLA TULARENSIS COMPLEXED WITH AMP AND SUCCINATE | STRUCTURAL GENOMICS, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, ALPHA STRUCTURE, LYASE, AMP BINDING, BETA- ELIMINATION, CYTOSOLE
3pva:A (ALA214) to (ASN260) PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE, HYDROLASE
3pva:B (ALA214) to (ASN260) PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE, HYDROLASE
3pva:C (ALA214) to (ASN260) PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE, HYDROLASE
3pva:D (ALA214) to (ASN260) PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE, HYDROLASE
3pva:F (ALA214) to (ASN260) PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE, HYDROLASE
3pva:H (ALA214) to (ASN260) PENICILLIN V ACYLASE FROM B. SPHAERICUS | AMIDOHYDROLASE, NTN HYDROLASE, PENICILLIN V ACYLASE, HYDROLASE
4eh5:A (ASN269) to (ALA309) HUMAN P38 MAP KINASE IN COMPLEX WITH NP-F4 AND RL87 | MAP KINASE INSERT, KINASE-LIGAND COMPLEX, NP-FRAGMENT, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3pxp:A (MSE125) to (ARG152) CRYSTAL STRUCTURE OF A PAS AND DNA BINDING DOMAIN CONTAINING PROTEIN (CAUR_2278) FROM CHLOROFLEXUS AURANTIACUS J-10-FL AT 2.30 A RESOLUTION | DNA-BINDING, BASIC HELIX-LOOP-HELIX MOTIF, BHLH MOTIF, LAMBDA REPRESSOR-LIKE DNA-BINDING FOLD, PER ARNT SIM DOMAIN, PAS DOMAIN, PROFILIN-LIKE FOLD, TRANSCRIPTION, TRANSCRIPTION REGULATION, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, TRANSCRIPTION REGULATOR
3pyb:C (SER560) to (SER663) CRYSTAL STRUCTURE OF ENT-COPALYL DIPHOSPHATE SYNTHASE FROM ARABIDOPSIS THALIANA IN COMPLEX WITH 13-AZA-13,14-DIHYDROCOPALYL DIPHOSPHATE | CLASS I AND II TERPENE CYCLASE FOLD, CLASS II DITERPENE CYCLASE, DXXDD MOTIF, GIBBERELLIN BIOSYNTHESIS, BIOSYNTHESIS OF ENT-COPALYL DIPHOSPHATE, ISOMERASE
3q95:B (THR311) to (SER395) CRYSTAL STRUCTURE OF HUMAN ESTROGEN RECEPTOR ALPHA LBD IN COMPLEX WITH GRIP PEPTIDE AND ESTRIOL | TRANSCRIPTIONAL REGULATOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATOR
4ezd:A (ASN69) to (SER132) CRYSTAL STRUCTURE OF THE UT-B UREA TRANSPORTER FROM BOS TAURUS BOUND TO SELENOUREA | MEMBRANE PROTEIN, CHANNEL, UREA TRANSPORT, SLC14, STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK CONSORTIUM ON MEMBRANE PROTEIN STRUCTURE, NYCOMPS, TRANSPORT PROTEIN
3qea:Z (GLU212) to (LYS262) CRYSTAL STRUCTURE OF HUMAN EXONUCLEASE 1 EXO1 (WT) IN COMPLEX WITH DNA (COMPLEX II) | EXONUCLEASE, HYDROLASE-DNA COMPLEX
4f5s:A (PRO516) to (ALA583) CRYSTAL STRUCTURE OF BOVINE SERUM ALBUMIN | BOVINE SERUM ALBUMIN, TRANSPORT PROTEIN
4f91:B (LEU1813) to (ILE1858) BRR2 HELICASE REGION | RNP REMODELING, PRE-MRNA SPLICING, SPLICEOSOME CATALYTIC ACTIVATION, DEXD/H-BOX RNA HELICASE, RNA AND ATP BINDING, NUCLEUS, HYDROLASE
4f92:B (LEU1813) to (ILE1858) BRR2 HELICASE REGION S1087L | RNP REMODELING, PRE-MRNA SPLICING, SPLICEOSOME CATALYTIC ACTIVATION, DEXD/H-BOX RNA HELICASE, RNA AND ATP BINDING, NUCLEUS, HYDROLASE
4uwh:A (PRO511) to (ASN584) DISCOVERY OF (2S)-8-((3R)-3-METHYLMORPHOLIN-4-YL)-1-(3- METHYL-2-OXO-BUTYL)-2-(TRIFLUOROMETHYL)-3,4-DIHYDRO-2H- PYRIMIDO(1,2-A)PYRIMIDIN-6-ONE: A NOVEL POTENT AND SELECTIVE INHIBITOR OF VPS34 FOR THE TREATMENT OF SOLID TUMORS | TRANSFERASE, LIPID KINASE, AUTOPHAGY INHIBITOR
4f93:B (GLU983) to (THR1028) BRR2 HELICASE REGION S1087L, MG-ATP | RNP REMODELING, PRE-MRNA SPLICING, SPLICEOSOME CATALYTIC ACTIVATION, DEXD/H-BOX RNA HELICASE, RNA AND ATP BINDING, NUCLEUS, HYDROLASE
4f93:B (ASN1814) to (ILE1858) BRR2 HELICASE REGION S1087L, MG-ATP | RNP REMODELING, PRE-MRNA SPLICING, SPLICEOSOME CATALYTIC ACTIVATION, DEXD/H-BOX RNA HELICASE, RNA AND ATP BINDING, NUCLEUS, HYDROLASE
4fc4:E (THR3) to (THR64) FNT FAMILY ION CHANNEL | ALPHA-HELICAL INNER MEMBRANE PROTEIN, ION CHANNEL, CYTOPLASMIC MEMBRANE, TRANSPORT PROTEIN
4fc4:G (ASP4) to (THR64) FNT FAMILY ION CHANNEL | ALPHA-HELICAL INNER MEMBRANE PROTEIN, ION CHANNEL, CYTOPLASMIC MEMBRANE, TRANSPORT PROTEIN
4fc4:H (PHE2) to (ILE73) FNT FAMILY ION CHANNEL | ALPHA-HELICAL INNER MEMBRANE PROTEIN, ION CHANNEL, CYTOPLASMIC MEMBRANE, TRANSPORT PROTEIN
4fcy:A (SER126) to (VAL165) CRYSTAL STRUCTURE OF THE BACTERIOPHAGE MU TRANSPOSOSOME | RNASEH, DDE TRANSPOSASE, DNA BINDING PROTEIN-DNA COMPLEX
4fcy:B (SER126) to (VAL165) CRYSTAL STRUCTURE OF THE BACTERIOPHAGE MU TRANSPOSOSOME | RNASEH, DDE TRANSPOSASE, DNA BINDING PROTEIN-DNA COMPLEX
4fhh:A (TYR179) to (ARG302) DEVELOPMENT OF SYNTHETICALLY ACCESSIBLE NON-SECOSTEROIDAL HYBRID MOLECULES COMBINING VITAMIN D RECEPTOR AGONISM AND HISTONE DEACETYLASE INHIBITION | LIGAND BINDING DOMAIN, APHA HELICAL SANDWICH, ALPHA HELICAL SANDWICH, TRANSCRIPTION FACTOR, ADN COREGULATORS, PHOSPHORYLATION AND HDAC INHIBITOR, NUCLEUS, TRANSCRIPTION-PROTEIN BINDING-INHIBITOR COMPLEX
3qxi:C (PRO185) to (LYS252) CRYSTAL STRUCTURE OF ENOYL-COA HYDRATASE ECHA1 FROM MYCOBACTERIUM MARINUM | STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, SSGCID, MYCOBACTERIUM, TUBERCULOSIS, MARINUM, WATER-BORNE PATHOGEN, FATTY ACID SYNTHESIS, ENOYL-COA, COENZYME A, HYDRATASE, LYASE
3r3l:A (PRO180) to (PRO227) STRUCTURE OF NP PROTEIN FROM LASSA AV STRAIN | NUCLEAR PROTEIN, REPLICATION, VIRAL PROTEIN, STRUCTURAL PROTEIN
3rdp:B (GLU210) to (ALA294) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH N-METHYL-FHBT | TRANSFERASE, THYMIDINE KINASE, DNA-SYNTHESIS, PET TRACER, ATP- BINDING, DNA SYNTHESIS, EARLY PROTEIN, NUCLEOTIDE-BINDING
5jj7:A (THR225) to (SER320) FIC-1 (AA134 - 508 E274G) FROM C. ELEGANS | AMPYLASE, HYPE, FIDO DOMAIN, TRANSFERASE
5jxm:A (GLU112) to (PRO155) CRYSTAL STRUCTURE OF PRENYLTRANSFERASE PRIB APO FORM | PRENYLTRANSFERASE, INDOLE-PT, ABBA FAMILY, PT FOLD, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, ENZYME DISCOVERY FOR NATURAL PRODUCT BIOSYNTHESIS, NATPRO, TRANSFERASE
4g7g:B (LYS138) to (LEU208) STEROL 14-ALPHA DEMETHYLASE (CYP51) FROM TRYPANOSOMA BRUCEI IN COMPLEX WITH THE VNI DERIVATIVE (R)-N-(1-(3,4'-DIFLUOROBIPHENYL-4-YL)-2-(1H- IMIDAZOL-1-YL)ETHYL)-4-(5-PHENYL-1,3,4-OXADIAZOL-2-YL)BENZAMIDE [VNI/VNF (VFV)] | CYTOCHROME P450 FOLD, HEME, MONOOXYGENASE, STEROL BIOSYNTHESIS, EUKARYOTIC MEMBRANE BIOGENESIS, CYTOCHROME P450 REDUCTASE, ENDOPLASMIC RETICULUM MEMBRANE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
5kcf:B (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-ETHYL, 4-METHOXYBENZYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4gfk:B (GLU117) to (ILE195) STRUCTURES OF NO FACTORS | NO, SLMA, DNA BINDING PROTEIN, NUCLEOID OCCLUSION, FTSZ, TETR FAMILY
5req:C (TYR243) to (LEU284) METHYLMALONYL-COA MUTASE, Y89F MUTANT, SUBSTRATE COMPLEX | ISOMERASE, MUTASE, INTRAMOLECULAR TRANSFERASE
5sv1:C (VAL12) to (PHE78) STRUCTURE OF THE EXBB/EXBD COMPLEX FROM E. COLI AT PH 4.5 | EXBB, MEMBRANE PROTEINS, PORE, CHANNEL, TRANSPORT PROTEIN
5syt:A (GLY97) to (LYS190) CRYSTAL STRUCTURE OF ZMPSTE24 | HYDROLASE, MEMBRANE PROTEIN, CAAX PROTEASE, ZINC METALLOPROTEASE, STE24, ISOPRENYLATION, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MEMBRANE PROTEIN STRUCTURAL BIOLOGY CONSORTIUM, MPSBC
5tcm:A (HIS24) to (CYS45) FIRST BROMODOMAIN FROM LEISHMANIA DONOVANI LDBPK.091320 COMPLEXED WITH BI-2536 | BROMODOMAIN, INHIBITOR, STRUCTURAL GENOMICS CONSORTIUM (SGC), UNKNOWN FUNCTION
5tcm:B (HIS24) to (CYS45) FIRST BROMODOMAIN FROM LEISHMANIA DONOVANI LDBPK.091320 COMPLEXED WITH BI-2536 | BROMODOMAIN, INHIBITOR, STRUCTURAL GENOMICS CONSORTIUM (SGC), UNKNOWN FUNCTION
5tcm:C (HIS24) to (CYS45) FIRST BROMODOMAIN FROM LEISHMANIA DONOVANI LDBPK.091320 COMPLEXED WITH BI-2536 | BROMODOMAIN, INHIBITOR, STRUCTURAL GENOMICS CONSORTIUM (SGC), UNKNOWN FUNCTION
6cpp:A (LEU127) to (THR185) CRYSTAL STRUCTURES OF CYTOCHROME P450-CAM COMPLEXED WITH CAMPHANE, THIOCAMPHOR, AND ADAMANTANE: FACTORS CONTROLLING P450 SUBSTRATE HYDROXYLATION | OXIDOREDUCTASE(OXYGENASE)
6req:A (GLY242) to (LEU284) METHYLMALONYL-COA MUTASE, 3-CARBOXYPROPYL-COA INHIBITOR COMPLEX | ISOMERASE, MUTASE, INTRAMOLECULAR TRANSFERASE
6req:C (GLY242) to (LEU284) METHYLMALONYL-COA MUTASE, 3-CARBOXYPROPYL-COA INHIBITOR COMPLEX | ISOMERASE, MUTASE, INTRAMOLECULAR TRANSFERASE
4gt9:A (SER102) to (LEU150) T. MARITIMA FDTS WITH FAD, DUMP AND FOLATE. | FLAVIN-DEPENDENT THYMIDYLATE SYNTHASE, TM0449, FAD, DUMP, 5,10- METHYLENETETRAHYDROFOLATE, TRANSFERASE
2ocf:A (THR311) to (SER395) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH ESTRADIOL AND THE E2#23 FN3 MONOBODY | ESTROGEN RECEPTOR, LBD, MONOBODY, ESTRADIOL, HORMONE-GROWTH FACTOR COMPLEX
1nkt:A (LYS617) to (GLY759) CRYSTAL STRUCTURE OF THE SECA PROTEIN TRANSLOCATION ATPASE FROM MYCOBACTERIUM TUBERCULOSIS COMPLEX WITH ADPBS | PREPROTEIN TRANSLOCATION, ATPASE, TRANSMEMBRANE TRANSPORT, HELICASE-LIKE MOTOR DOMAIN, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PROTEIN TRANSPORT
1nkt:B (ALA616) to (ILE757) CRYSTAL STRUCTURE OF THE SECA PROTEIN TRANSLOCATION ATPASE FROM MYCOBACTERIUM TUBERCULOSIS COMPLEX WITH ADPBS | PREPROTEIN TRANSLOCATION, ATPASE, TRANSMEMBRANE TRANSPORT, HELICASE-LIKE MOTOR DOMAIN, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, TB STRUCTURAL GENOMICS CONSORTIUM, TBSGC, PROTEIN TRANSPORT
2ay6:B (HIS301) to (HIS356) AROMATIC AMINO ACID AMINOTRANSFERASE WITH 3-INDOLEBUTYRIC ACID | AMINOTRANSFERASE
2ay7:A (HIS301) to (HIS356) AROMATIC AMINO ACID AMINOTRANSFERASE WITH 4-PHENYLBUTYRIC ACID | AMINOTRANSFERASE, AROMATIC AMINO ACID BIOSYNTHESIS
2oxx:A (PRO280) to (GLN325) PROTEIN KINASE CK2 IN COMPLEX WITH TETRABROMOBENZOIMIDAZOLE DERIVATIVES K17, K22 AND K32 | PROTEIN KINASE CK2, INHIBITORS, TETRABROMOBENZOIMIDAZOLE DERIVATIVES, TRANSFERASE
1b33:H (ARG46) to (GLY119) STRUCTURE OF LIGHT HARVESTING COMPLEX OF ALLOPHYCOCYANIN ALPHA AND BETA CHAINS/CORE-LINKER COMPLEX AP*LC7.8 | LIGHT-HARVESTING PROTEIN, CYANOBACTERIA, ALLOPHYCOCYANIN, LINKER POLYPEPTIDES, COMPLEX STRUCTURE, PHOTOSYNTHESIS
2bl2:I (MET1) to (LEU80) THE MEMBRANE ROTOR OF THE V-TYPE ATPASE FROM ENTEROCOCCUS HIRAE | V-TYPE ATPASE, K-RING, MEMBRANE ROTOR, SODIUM TRANSPORTER, HYDROGEN ION TRANSPORT, HYDROLASE, TRANSMEMBRANE
3f2b:A (THR1391) to (LEU1435) DNA POLYMERASE POLC FROM GEOBACILLUS KAUSTOPHILUS COMPLEX WITH DNA, DGTP, MG AND ZN | DNA POLYMERASE C, DNA POLYMERASE III, TERNARY COMPLEX, PROTEIN-DNA COMPLEX, REPLICATIVE DNA POLYMERASE, DNA REPLICATION, DNA-DIRECTED DNA POLYMERASE, EXONUCLEASE, HYDROLASE, NUCLEASE, NUCLEOTIDYLTRANSFERASE, TRANSFERASE, TRANSFERASE-DNA COMPLEX
1of1:B (GLU210) to (ALA294) KINETICS AND CRYSTAL STRUCTURE OF THE HERPES SIMPLEX VIRUS TYPE 1 THYMIDINE KINASE INTERACTING WITH (SOUTH)-METHANOCARBA-THYMIDINE | TRANSFERASE, THYMIDINE KINASE, ANTIVIRAL DRUG, ENZYME- PRODRUG GENE, KINASE, DNA SYNTHESIS, ATP-BINDING
2pru:A (SER1) to (GLU67) NMR STRUCTURE OF HUMAN APOS100B AT 10C | S100, CALCIUM BINDING PROTEIN, EF-HAND, ALL ALPHA HELICAL PROTEIN, METAL BINDING PROTEIN
2pru:B (SER1) to (GLU67) NMR STRUCTURE OF HUMAN APOS100B AT 10C | S100, CALCIUM BINDING PROTEIN, EF-HAND, ALL ALPHA HELICAL PROTEIN, METAL BINDING PROTEIN
1cqw:A (ASP167) to (LEU205) NAI COCRYSTALLISED WITH HALOALKANE DEHALOGENASE FROM A RHODOCOCCUS SPECIES | A/B HYDROLASE FOLD, DEHALOGENASE I-S BOND
3fud:A (PRO400) to (LEU448) LEUKOTRIENE A4 HYDROLASE IN COMPLEX WITH N-METHYL-1-(2- THIOPHEN-2-YLPHENYL)METHANAMINE | LEUKOTRIENE A4 HYDROLASE, LTA4H, FRAGMENT CRYSTALLOGRAPHY, FRAGMENTS OF LIFE, FOL, ALTERNATIVE SPLICING, CYTOPLASM, HYDROLASE, LEUKOTRIENE BIOSYNTHESIS, METAL-BINDING, METALLOPROTEASE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, PROTEASE, ZINC
3fuk:A (GLY399) to (LEU448) LEUKOTRIENE A4 HYDROLASE IN COMPLEX WITH 1-[2-(1H-INDOL-5- YLOXY)ETHYL]PIPERIDINE-4-CARBOXYLIC ACID | LEUKOTRIENE A4 HYDROLASE, LTA4H, FRAGMENT CRYSTALLOGRAPHY, FRAGMENTS OF LIFE, FOL, ALTERNATIVE SPLICING, CYTOPLASM, HYDROLASE, LEUKOTRIENE BIOSYNTHESIS, METAL-BINDING, METALLOPROTEASE, MULTIFUNCTIONAL ENZYME, POLYMORPHISM, PROTEASE, ZINC
1phd:A (LEU127) to (THR185) CRYSTAL STRUCTURES OF METYRAPONE-AND PHENYLIMIDAZOLE-INHIBITED COMPLEXES OF CYTOCHROME P450-CAM | OXIDOREDUCTASE(OXYGENASE)
1e1c:C (GLY242) to (LEU284) METHYLMALONYL-COA MUTASE H244A MUTANT | ISOMERASE, MUTASE, INTRAMOLECULAR TRANSFERASE
1e2l:B (ASP211) to (LEU262) KINETICS AND CRYSTAL STRUCTURE OF THE WILD-TYPE AND THE ENGINEERED Y101F MUTANT OF HERPES SIMPLEX VIRUS TYPE 1 THYMIDINE KINASE INTERACTING WITH (NORTH)-METHANOCARBA-THYMIDINE | THYMIDINE KINASE, ANTIVIRAL DRUG, ENZYME-PRODRUG GENE THERAPY, X-RAY STRUCTURE, SUGAR RING PUCKER
1e6y:A (SER1296) to (ASN1372) METHYL-COENZYME M REDUCTASE FROM METHANOSARCINA BARKERI | BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE, NI ENZYME
1e6y:B (ASN2195) to (GLY2260) METHYL-COENZYME M REDUCTASE FROM METHANOSARCINA BARKERI | BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE, NI ENZYME
1e6y:D (SER4296) to (ASN4372) METHYL-COENZYME M REDUCTASE FROM METHANOSARCINA BARKERI | BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE, NI ENZYME
1e6y:E (ASN5195) to (GLY5260) METHYL-COENZYME M REDUCTASE FROM METHANOSARCINA BARKERI | BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE, NI ENZYME
3hbl:C (HIS333) to (ASN361) CRYSTAL STRUCTURE OF S. AUREUS PYRUVATE CARBOXYLASE T908A MUTANT | TIM BARREL, PYRUVATE, LIGASE
4ysw:A (GLY915) to (GLU990) STRUCTURE OF RAT XANTHINE OXIDOREDUCTASE, C-TERMINAL DELETION PROTEIN VARIANT, NADH BOUND FORM | XANTHINE OXIDASE, XANTHINE, DEHYDROGENASE, OXIDOREDUCTASE, D/O CONVERSION
1rc5:D (SER619) to (GLU688) CRYSTAL STRUCTURE OF MG(II)-COMPLEX OF RNASE III ENDONUCLEASE DOMAIN FROM AQUIFEX AEOLICUS AT 2.30 ANGSTROM RESOLUTION | RIBONUCLEASE, RNASE III, DOUBLE-STRANDED RNA, RNA INTERFERENCE, ENDONUCLEASE DOMAIN, ENDONUCLEOLYTIC CLEAVAGE, HYDROLASE
2vdb:A (GLY399) to (PRO468) STRUCTURE OF HUMAN SERUM ALBUMIN WITH S-NAPROXEN AND THE GA MODULE | LIPID-BINDING, METAL-BINDING, PROTEIN BINDING, PEPTIDOGLYCAN-ANCHOR, BACTERIAL ALBUMIN-BINDING, DISEASE MUTATION, THREE-HELIX BUNDLE, GA MODULE, DRUG BINDING, GLYCOPROTEIN, CLEAVAGE ON PAIR OF BASIC RESIDUES, HUMAN SERUM ALBUMIN, SECRETED, NAPROXEN, CELL WALL, GLYCATION
3v48:A (ASN118) to (HIS171) CRYSTAL STRUCTURE OF THE PUTATIVE ALPHA/BETA HYDROLASE RUTD FROM E.COLI | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, HYDROLASE
3v48:B (ASN118) to (HIS171) CRYSTAL STRUCTURE OF THE PUTATIVE ALPHA/BETA HYDROLASE RUTD FROM E.COLI | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, HYDROLASE
4kvi:D (SER55) to (ASP133) CRYSTAL STRUCTURE OF ASPERGILLUS TERREUS ARISTOLOCHENE SYNTHASE COMPLEXED WITH (4AS,7S)-4A-METHYL-7-(PROP-1-EN-2-YL)-2,3,4,4A,5,6,7, 8-OCTAHYDROQUINOLIN-1-IUM | CLASS I TERPENE CYCLASE, ALPHA-HELICAL FOLD, FARNESYL DIPHOSPHATE, METAL-BINDING, MAGNESIUM, LYASE-LYASE INHIBITOR COMPLEX
2vtk:A (PRO209) to (ALA294) THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH ADP AND DEOXYTHYMIDINE | KEY ENZYME IN THYMIDINE SALVAGE PATHWAY, ADDITIONAL THYMIDYLATE KINASE ACTIVITY, TARGET FOR ANTI-HERPES VIRAL DRUGS, TRANSFERASE
1sqm:A (PRO400) to (LEU448) STRUCTURE OF [R563A] LEUKOTRIENE A4 HYDROLASE | EPOXIDE HYDROLASE; ALPHA-BETA PROTEIN; LEUKOTRIENE BIOSYNTHESIS; METALLOPROTEASE
1svm:A (ASN332) to (VAL413) CO-CRYSTAL STRUCTURE OF SV40 LARGE T ANTIGEN HELICASE DOMAIN AND ATP | AAA+ FOLD, VIRAL PROTEIN
1svm:E (ASN332) to (VAL413) CO-CRYSTAL STRUCTURE OF SV40 LARGE T ANTIGEN HELICASE DOMAIN AND ATP | AAA+ FOLD, VIRAL PROTEIN
2ghm:A (ASN269) to (ALA309) MUTATED MAP KINASE P38 (MUS MUSCULUS) IN COMPLEX WITH INHBITOR PG-895449 | MAP KINASE P38, TRANSFERASE
3vh6:D (ARG9) to (PHE79) CRYSTAL STRUCTURE OF THE CHICKEN CENP-T HISTONE FOLD/CENP-W/CENP- S/CENP-X HETEROTETRAMERIC COMPLEX, CRYSTAL FORM II | HISTONE FOLD, CHROMOSOME SEGREGATION, DNA BINDING, NUCLEUS, DNA BINDING PROTEIN
3ihy:A (PRO511) to (ASN584) HUMAN PIK3C3 CRYSTAL STRUCTURE | ALPHA/BETA PROTEIN, STRUCTURAL GENOMICS, SGC STOCKHOLM, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, MANGANESE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, TRANSFERASE
3ihy:E (PRO511) to (ASN584) HUMAN PIK3C3 CRYSTAL STRUCTURE | ALPHA/BETA PROTEIN, STRUCTURAL GENOMICS, SGC STOCKHOLM, STRUCTURAL GENOMICS CONSORTIUM, SGC, ATP-BINDING, KINASE, MANGANESE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, TRANSFERASE
1hbm:A (PHE283) to (TYR358) METHYL-COENZYME M REDUCTASE ENZYME PRODUCT COMPLEX | METHANOGENESIS, BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE
1hbm:D (PHE283) to (TYR358) METHYL-COENZYME M REDUCTASE ENZYME PRODUCT COMPLEX | METHANOGENESIS, BIOLOGICAL METHANOGENESIS, NI-ENZYME, OXIDOREDUCTASE
2wgl:C (ALA160) to (LEU225) CRYSTAL STRUCTURE OF HELICOBACTOR PYLORI UREF | CYTOPLASM, VIRULENCE, CHAPERONE, NICKEL INSERTION, METAL BINDING PROTEIN
3vtk:A (PRO209) to (ALA294) THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH ADP AND 5-IODO-DEOXYURIDINE-MONOPHOSPHATE | KEY ENZYME IN THYMIDINE SALVAGE PATHWAY, ADDITIONAL THYMIDYLATE KINASE ACTIVITY, TARGET FOR ANTI-HERPES VIRAL DRUGS, TRANSFERASE
2i2z:A (GLY399) to (THR467) HUMAN SERUM ALBUMIN COMPLEXED WITH MYRISTATE AND ASPIRIN | PLASMA PROTEIN, METAL-BINDING, LIPID-BINDING, LIPID BINDING PROTEIN
4m2s:A (VAL732) to (GLY826) CORRECTED STRUCTURE OF MOUSE P-GLYCOPROTEIN BOUND TO QZ59-RRR | ATP-BINDING CASSETTE TRANSPORTER, MULTIDRUG EFFLUX, ADENOSINE TRIPHOSPHATE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5a8r:A (ALA285) to (TYR360) METHYL-COENZYME M REDUCTASE II FROM METHANOTHERMOBACTER MARBURGENSIS AT 2.15 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, CATALYSIS, COENZYMES, DISULFIDES, HYDROGEN, HYDROGEN BONDING, LIGANDS, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, MODELS, MOLECULAR, NICKEL, OXIDATION-REDUCTION, OXIDOREDUCTASES, PHOSPHOTHREONINE, PROTEIN CONFORMATION, PROTEIN FOLDING, PROTEIN STRUCTURE
5a8r:B (ALA197) to (ASN259) METHYL-COENZYME M REDUCTASE II FROM METHANOTHERMOBACTER MARBURGENSIS AT 2.15 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, CATALYSIS, COENZYMES, DISULFIDES, HYDROGEN, HYDROGEN BONDING, LIGANDS, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, MODELS, MOLECULAR, NICKEL, OXIDATION-REDUCTION, OXIDOREDUCTASES, PHOSPHOTHREONINE, PROTEIN CONFORMATION, PROTEIN FOLDING, PROTEIN STRUCTURE
5a8r:D (ALA285) to (TYR360) METHYL-COENZYME M REDUCTASE II FROM METHANOTHERMOBACTER MARBURGENSIS AT 2.15 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, CATALYSIS, COENZYMES, DISULFIDES, HYDROGEN, HYDROGEN BONDING, LIGANDS, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, MODELS, MOLECULAR, NICKEL, OXIDATION-REDUCTION, OXIDOREDUCTASES, PHOSPHOTHREONINE, PROTEIN CONFORMATION, PROTEIN FOLDING, PROTEIN STRUCTURE
5a8r:E (ALA197) to (GLY260) METHYL-COENZYME M REDUCTASE II FROM METHANOTHERMOBACTER MARBURGENSIS AT 2.15 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, CATALYSIS, COENZYMES, DISULFIDES, HYDROGEN, HYDROGEN BONDING, LIGANDS, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, MODELS, MOLECULAR, NICKEL, OXIDATION-REDUCTION, OXIDOREDUCTASES, PHOSPHOTHREONINE, PROTEIN CONFORMATION, PROTEIN FOLDING, PROTEIN STRUCTURE
5a8r:G (ALA285) to (TYR360) METHYL-COENZYME M REDUCTASE II FROM METHANOTHERMOBACTER MARBURGENSIS AT 2.15 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, CATALYSIS, COENZYMES, DISULFIDES, HYDROGEN, HYDROGEN BONDING, LIGANDS, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, MODELS, MOLECULAR, NICKEL, OXIDATION-REDUCTION, OXIDOREDUCTASES, PHOSPHOTHREONINE, PROTEIN CONFORMATION, PROTEIN FOLDING, PROTEIN STRUCTURE
5a8r:H (ALA197) to (ASN247) METHYL-COENZYME M REDUCTASE II FROM METHANOTHERMOBACTER MARBURGENSIS AT 2.15 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, CATALYSIS, COENZYMES, DISULFIDES, HYDROGEN, HYDROGEN BONDING, LIGANDS, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, MODELS, MOLECULAR, NICKEL, OXIDATION-REDUCTION, OXIDOREDUCTASES, PHOSPHOTHREONINE, PROTEIN CONFORMATION, PROTEIN FOLDING, PROTEIN STRUCTURE
5a8r:J (ALA285) to (TYR360) METHYL-COENZYME M REDUCTASE II FROM METHANOTHERMOBACTER MARBURGENSIS AT 2.15 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, CATALYSIS, COENZYMES, DISULFIDES, HYDROGEN, HYDROGEN BONDING, LIGANDS, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, MODELS, MOLECULAR, NICKEL, OXIDATION-REDUCTION, OXIDOREDUCTASES, PHOSPHOTHREONINE, PROTEIN CONFORMATION, PROTEIN FOLDING, PROTEIN STRUCTURE
5a8r:K (ALA197) to (ASN247) METHYL-COENZYME M REDUCTASE II FROM METHANOTHERMOBACTER MARBURGENSIS AT 2.15 A RESOLUTION | TRANSFERASE, POST-TRANSLATIONAL MODIFICATION, BINDING SITES, CATALYSIS, COENZYMES, DISULFIDES, HYDROGEN, HYDROGEN BONDING, LIGANDS, MESNA, METALLOPORPHYRINS, METHANE, METHANOBACTERIUM, MODELS, MOLECULAR, NICKEL, OXIDATION-REDUCTION, OXIDOREDUCTASES, PHOSPHOTHREONINE, PROTEIN CONFORMATION, PROTEIN FOLDING, PROTEIN STRUCTURE
4mck:A (ASP129) to (ARG189) CRYSTAL STRUCTURE OF FAMILY GH19, CLASS IV CHITINASE FROM ZEA MAYS | HYDROLASE
4md7:E (ARG280) to (TYR325) CRYSTAL STRUCTURE OF FULL-LENGTH SYMMETRIC CK2 HOLOENZYME | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
4md7:G (ARG280) to (TYR325) CRYSTAL STRUCTURE OF FULL-LENGTH SYMMETRIC CK2 HOLOENZYME | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
4md7:H (ARG280) to (TYR325) CRYSTAL STRUCTURE OF FULL-LENGTH SYMMETRIC CK2 HOLOENZYME | PROTEIN SERINE/THREONINE KINASE, TRANSFERASE
1iw8:D (THR58) to (ILE103) CRYSTAL STRUCTURE OF A MUTANT OF ACID PHOSPHATASE FROM ESCHERICHIA BLATTAE (G74D/I153T) | ALL ALPHA, HYDROLASE
3wil:A (ARG280) to (VAL328) CRYSTAL STRUCTURE OF THE CK2ALPHA/COMPOUND3 COMPLEX | KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4mlb:B (SER235) to (PHE349) REVERSE POLARITY OF BINDING POCKET SUGGESTS DIFFERENT FUNCTION OF A MOP SUPERFAMILY TRANSPORTER FROM PYROCOCCUS FURIOSUS VC1 (DSM3638) | LIPID TRANSLOCASE, FLIPPASE, MEMBRANE PROTEIN, TRANSPORT PROTEIN
1jkm:B (ASP241) to (TRP285) BREFELDIN A ESTERASE, A BACTERIAL HOMOLOGUE OF HUMAN HORMONE SENSITIVE LIPASE | SERINE HYDROLASE, DEGRADATION OF BREFELDIN A, ALPHA/BETA HYDROLASE FAMILY
3wz5:C (ASP75) to (ALA131) STRUCTURE OF THE PERIPLASMIC DOMAIN OF DOTI (CRYSTAL FORM II) | TYPE IVB SECRETION, UNKNOWN FUNCTION
2le9:B (THR7) to (VAL65) RAGEC2-S100A13 TETRAMERIC COMPLEX | RECEPTOR FOR ADVANCED GLYCATION END PRODUCTS, S100A13, TETRAMERIC COMPLEX, MEMBRANE PROTEIN-METAL BINDING PROTEIN COMPLEX
3zrb:A (PRO686) to (LYS769) STRUCTURAL BASIS FOR AGONISM AND ANTAGONISM FOR A SET OF CHEMICALLY RELATED PROGESTERONE RECEPTOR MODULATORS | RECEPTOR, AGONIST, ANTAGONIST
2m49:B (SER1) to (GLY64) STRUCTURAL INSIGHTS INTO HUMAN S100B AND BASIC FIBROBLAST GROWTH FACTOR (FGF2) INTERACTION | S100B, FGF2, CYTOKINE-METAL BINDING PROTEIN COMPLEX
4nsl:B (GLU76) to (PHE119) X-RAY CRYSTAL STRUCTURE OF ADENYLOSUCCINATE LYASE FROM SALMONELLA TYPHIMURIUM | PURINE BIOSYNTHESIS, HOMOTETRAMER, ASPARTASE/FUMARASE SUPERFAMILY, LYASE, INTERFACE BINDING SITE
2mph:A (THR11) to (THR53) SOLUTION STRUCTURE OF HUMAN FK506 BINDING PROTEIN 25 | HFKBP25, ISOMERASE
2ypt:D (ILE98) to (GLY192) CRYSTAL STRUCTURE OF THE HUMAN NUCLEAR MEMBRANE ZINC METALLOPROTEASE ZMPSTE24 MUTANT (E336A) IN COMPLEX WITH A SYNTHETIC CSIM TETRAPEPTIDE FROM THE C-TERMINUS OF PRELAMIN A | HYDROLASE-PEPTIDE COMPLEX, M48 PEPTIDASE, INTEGRAL MEMBRANE PROTEIN, PRELAMIN A PROCESSING, AGEING, PROGERIA
1m2z:A (THR531) to (ARG614) CRYSTAL STRUCTURE OF A DIMER COMPLEX OF THE HUMAN GLUCOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN BOUND TO DEXAMETHASONE AND A TIF2 COACTIVATOR MOTIF | GLUCOCORTICOID RECEPTOR, DEXAMETHASONE, TIF2, DIMER INTERFACE, HORMONE BINDING POCKET, CHARGE CLAMP, COACTIVATOR, HORMONE/HORMONE ACTIVATOR COMPLEX
1m2z:D (THR531) to (ARG614) CRYSTAL STRUCTURE OF A DIMER COMPLEX OF THE HUMAN GLUCOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN BOUND TO DEXAMETHASONE AND A TIF2 COACTIVATOR MOTIF | GLUCOCORTICOID RECEPTOR, DEXAMETHASONE, TIF2, DIMER INTERFACE, HORMONE BINDING POCKET, CHARGE CLAMP, COACTIVATOR, HORMONE/HORMONE ACTIVATOR COMPLEX
5cu0:A (ARG280) to (VAL328) CRYSTAL STRUCTURE OF CK2ALPHA WITH 2-HYDROXY-5-METHYLBENZOIC ACID AND N-(3-(3-CHLORO-4-(PHENYL)BENZYLAMINO)PROPYL)ACETAMIDE BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
5cu0:B (ARG280) to (VAL328) CRYSTAL STRUCTURE OF CK2ALPHA WITH 2-HYDROXY-5-METHYLBENZOIC ACID AND N-(3-(3-CHLORO-4-(PHENYL)BENZYLAMINO)PROPYL)ACETAMIDE BOUND | CK2ALPHA, CK2A, FRAGMENT BASED DRUG DISCOVERY, HIGH CONCENTRATION SCREENING, SELECTIVE ATP COMPETITIVE INHIBITORS, SURFACE ENTROPHY REDUCTION, TRANSFERASE
1ypt:A (SER422) to (GLY462) CRYSTAL STRUCTURE OF YERSINIA PROTEIN TYROSINE PHOSPHATASE AT 2.5 ANGSTROMS AND THE COMPLEX WITH TUNGSTATE | HYDROLASE, PROTEIN TYROSINE PHOSPHATASE
1ypt:B (SER422) to (GLY462) CRYSTAL STRUCTURE OF YERSINIA PROTEIN TYROSINE PHOSPHATASE AT 2.5 ANGSTROMS AND THE COMPLEX WITH TUNGSTATE | HYDROLASE, PROTEIN TYROSINE PHOSPHATASE
1z1n:X (LEU460) to (HIS525) CRYSTAL STRUCTURE OF THE SIXTEEN HEME CYTOCHROME FROM DESULFOVIBRIO GIGAS | ELECTRON TRANSPORT
5dqt:J (ASP169) to (THR227) CRYSTAL STRUCTURE OF CAS-DNA-22 COMPLEX | PROTEIN-DNA COMPLEX, HYDROLASE-DNA COMPLEX
1zac:A (SER15) to (GLY69) N-DOMAIN OF TROPONIN C FROM CHICKEN SKELETAL MUSCLE, NMR, MINIMIZED AVERAGE STRUCTURE | CALCIUM-BINDING, EF-HAND, MUSCLE PROTEIN, LOW-TEMPERATURE
3an1:A (GLY915) to (GLU990) CRYSTAL STRUCTURE OF RAT D428A MUTANT, URATE BOUND FORM | PRODUCT BOUND FORM, OXIDOREDUCTASE, URATE BINDING
3an1:B (GLY915) to (GLU990) CRYSTAL STRUCTURE OF RAT D428A MUTANT, URATE BOUND FORM | PRODUCT BOUND FORM, OXIDOREDUCTASE, URATE BINDING
5dvs:A (THR311) to (MET396) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A 2-METHYL-SUBSTITUTED TRIARYL-IMINE 4,4'-[(2-METHYLPHENYL) CARBONIMIDOYL]DIPHENOL | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
3m1v:A (PRO282) to (TYR358) STRUCTURAL INSIGHT INTO METHYL-COENZYME M REDUCTASE CHEMISTRY USING COENZYME B ANALOGUES | METHYL-COENZYME M REDUCTASE, METAL-BINDING, METHANOGENESIS, METHYLATION, NICKEL, TRANSFERASE
3m1v:D (PRO282) to (TYR358) STRUCTURAL INSIGHT INTO METHYL-COENZYME M REDUCTASE CHEMISTRY USING COENZYME B ANALOGUES | METHYL-COENZYME M REDUCTASE, METAL-BINDING, METHANOGENESIS, METHYLATION, NICKEL, TRANSFERASE
3m2u:A (PRO282) to (TYR358) STRUCTURAL INSIGHT INTO METHYL-COENZYME M REDUCTASE CHEMISTRY USING COENZYME B ANALOGUES | METHYL-COENZYME M REDUCTASE, NICKEL, METAL-BINDING, METHANOGENESIS, METHYLATION, TRANSFERASE
3m2u:D (PRO282) to (TYR358) STRUCTURAL INSIGHT INTO METHYL-COENZYME M REDUCTASE CHEMISTRY USING COENZYME B ANALOGUES | METHYL-COENZYME M REDUCTASE, NICKEL, METAL-BINDING, METHANOGENESIS, METHYLATION, TRANSFERASE
3m32:A (PRO282) to (TYR358) STRUCTURAL INSIGHT INTO METHYL-COENZYME M REDUCTASE CHEMISTRY USING COENZYME B ANALOGUES | METHYL-COENZYME M REDUCTASE, NICKEL, METAL-BINDING, METHANOGENESIS, METHYLATION, TRANSFERASE
3m32:D (PRO282) to (TYR358) STRUCTURAL INSIGHT INTO METHYL-COENZYME M REDUCTASE CHEMISTRY USING COENZYME B ANALOGUES | METHYL-COENZYME M REDUCTASE, NICKEL, METAL-BINDING, METHANOGENESIS, METHYLATION, TRANSFERASE
5efy:D (TRP127) to (SER193) APO-FORM OF SCO3201 | TETR-REGULATOR, APO-FORM, HTH-MOTIF, BACTERIAL TRANSCRIPTION REGULATOR, TRANSCRIPTION
4ql8:A (PRO671) to (THR755) CRYSTAL STRUCTURE OF ANDROGEN RECEPTOR IN COMPLEX WITH THE LIGAND | TRANSCRIPTION REGULATION, RECEPTOR, TRANSCRIPTION
3mne:A (LEU538) to (GLN621) CRYSTAL STRUCTURE OF THE AGONIST FORM OF MOUSE GLUCOCORTICOID RECEPTOR STABILIZED BY F608S MUTATION AT 1.96A | PROTEIN-LIGAND COMPLEX, STEROID NUCLEAR RECEPTOR, MOUSE, AGONIST, CO- ACTIVATOR, HORMONE RECEPTOR
3mxt:A (SER184) to (LYS234) CRYSTAL STRUCTURE OF PANTOATE-BETA-ALANINE LIGASE FROM CAMPYLOBACTER JEJUNI | ALPHA-BETA-ALPHA, STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID, LIGASE
4c28:B (PHE142) to (SER207) CRYSTAL STRUCTURE OF TRYPANOSOMA CRUZI CYP51 BOUND TO THE INHIBITOR (R)-N-(3-(1H-INDOL-3-YL)-1-OXO-1-(PYRIDIN-4- YLAMINO)PROPAN-2-YL)-4-(4-(4-CHLOROPHENYL)PIPERAZIN-1-YL)- 2-FLUOROBENZAMIDE. | OXIDOREDUCTASE, STEROL BIOSYNTHESIS, CHAGAS DISEASE
5fs0:B (ALA45) to (GLU105) CRYSTAL STRUCTURE OF THE PHENOL-RESPONSIVE SENSORY DOMAIN OF THE TRANSCRIPTION ACTIVATOR POXR WITH 2,4-DICHLOROPHENOL | TRANSCRIPTION, PHENOL, DMPR, ENHANCER-BINDING PROTEIN, ACTIVATOR, ATPASE FAMILY
4ck8:B (PHE142) to (GLU205) STEROL 14-ALPHA DEMETHYLASE (CYP51)FROM TRYPANOSOMA CRUZI IN COMPLEX WITH (R)-1-(2,4-DICHLOROPHENYL)-2-(1H-IMIDAZOL-1-YL)ETHYL 4-(4-(3,4-DICHLOROPHENYL)PIPERAZIN-1-YL)PHENYLCARBAMATE (LFD) | CYTOCHROME P450, OXIDOREDUCTASE, MONOOXYGENASE, STEROL BIOSYNTHESIS, EUKARYOTIC MEMBRANES, CYTOCHROME P450 FOLD, ENDOPLASMIC RETICULUM MEMBRANE
3o1q:A (ALA160) to (LEU225) NATIVE CRYSTAL STRUCTURE OF HELICOBACTER PYLORI UREASE ACCESSORY PROTEIN UREF | UREASE MATURATION, METAL BINDING PROTEIN
3dbl:G (VAL315) to (ASN386) STRUCTURAL DISSECTION OF A GATING MECHANISM PREVENTING MISACTIVATION OF UBIQUITIN BY NEDD8'S E1 (APPBP1- UBA3ARG190WT-NEDD8ALA72GLN) | CELL CYCLE, ACTIVATING ENZYME, APOPTOSIS, MEMBRANE, UBL CONJUGATION PATHWAY, ATP-BINDING, LIGASE, NUCLEOTIDE- BINDING, POLYMORPHISM, NUCLEUS
3oj1:A (GLY1) to (MET49) STRUCTURE OF THE H55D MUTANT OF DEHALOPEROXIDASE-HEMOGLOBIN A FROM AMPHITRITE ORNATA | GLOBIN, PEOXIDASE, DEHALOPEOXIDASE, OXIDOREDUCTASE
3dxl:A (VAL208) to (LYS257) CRYSTAL STRUCTURE OF AED7 FROM AEDES AEGYPTI | ODORANT-BINDING PROTEIN, ALL-HELICAL, ALLERGEN, SECRETED
4e44:D (LYS12) to (PHE81) CRYSTAL STRUCTURE OF THE HMHF1/HMHF2 HISTONE-FOLD TETRAMER | HISTONE-FOLD, TETRAMER, FANCONI ANEMIA, FANCM, MHF, DNA BINDING PROTEIN
5ij7:S (LEU592) to (GLY644) STRUCTURE OF HS/ACPRC2 IN COMPLEX WITH A PYRIDONE INHIBITOR | LYSINE METHYLTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ij7:T (GLU590) to (GLY644) STRUCTURE OF HS/ACPRC2 IN COMPLEX WITH A PYRIDONE INHIBITOR | LYSINE METHYLTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ij8:S (PRO589) to (GLY644) STRUCTURE OF THE PRIMARY ONCOGENIC MUTANT Y641N HS/ACPRC2 IN COMPLEX WITH A PYRIDONE INHIBITOR | LYSINE METHYLTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5ij8:T (TRP591) to (GLY644) STRUCTURE OF THE PRIMARY ONCOGENIC MUTANT Y641N HS/ACPRC2 IN COMPLEX WITH A PYRIDONE INHIBITOR | LYSINE METHYLTRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5imn:D (GLY53) to (HIS132) CRYSTAL STRUCTURE OF N299A/S303A ASPERGILLUS TERREUS ARISTOLOCHENE SYNTHASE COMPLEXED WITH (1S,8S,9AR)-1,9A-DIMETHYL-8-(PROP-1-EN-2-YL) DECAHYDROQUINOLIZIN-5-IUM | LYASE, TERPENE CYCLASES, LYASE-LYASE INHIBITOR COMPLEX
3qeb:Z (GLU212) to (LEU261) CRYSTAL STRUCTURE OF HUMAN EXONUCLEASE 1 EXO1 (WT) IN COMPLEX WITH DNA AND MN2+ (COMPLEX III) | EXONUCLEASE, HYDROLASE-DNA COMPLEX
4uwk:A (PRO511) to (ASN584) DISCOVERY OF (2S)-8-((3R)-3-METHYLMORPHOLIN-4-YL)-1-(3- METHYL-2-OXO-BUTYL)-2-(TRIFLUOROMETHYL)-3,4-DIHYDRO-2H- PYRIMIDO(1,2-A)PYRIMIDIN-6-ONE: A NOVEL POTENT AND SELECTIVE INHIBITOR OF VPS34 FOR THE TREATMENT OF SOLID TUMORS | TRANSFERASE, LIPID KINASE, AUTOPHAGY INHIBITOR
4geh:A (LEU58) to (ARG124) CRYSTAL STRUCTURE OF MST4 DIMERIZATION DOMAIN COMPLEX WITH PDCD10 | ALPHA HELIX-RICH PROTEIN, SERINE/THREONINE-PROTEIN KINASE, PROTEIN BINDING, CELL PROLIFERATION, CELL GROWTH, PROTEIN BINDING- TRANSFERASE COMPLEX
5l08:A (PRO31) to (ASN70) CRYO-EM STRUCTURE OF CASP-8 TDED FILAMENT | CASP-8, FILAMENT, DED, DEATH DOMAIN, APOPTOSIS
5liv:A (VAL155) to (VAL213) CRYSTAL STRUCTURE OF MYXOBACTERIAL CYP260A1 | 1-ALPHA-HYDROXYLASE, STEROID, SORANGIUM CELLULOSUM, REDOX POOL, OXIDOREDUCTASE