4gs8:B (PRO856) to (LEU931) STRUCTURE ANALYSIS OF CYSTEINE FREE INSULIN DEGRADING ENZYME (IDE) WITH COMPOUND BDM43079 [{[(S)-2-(1H-IMIDAZOL-4-YL)-1-METHYLCARBAMOYL- ETHYLCARBAMOYL]-METHYL}-(3-PHENYL-PROPYL)-AMINO]-ACETIC ACID | INSULIN DEGRADING ENZYME, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3e6i:A (ASP264) to (PRO365) HUMAN CYTOCHROME P450 2E1 IN COMPLEX WITH THE INHIBITOR INDAZOLE | CYP2E1, P450 2E1, MONOOXYGENASE, ACETAMINOPHEN, OXIDOREDUCTASE, HEME, ENDOPLASMIC RETICULUM, IRON, MEMBRANE, METAL-BINDING, MICROSOME
2of7:A (MSE145) to (GLU202) STRUCTURAL GENOMICS, THE CRYSTAL STRUCTURE OF A TETR-FAMILY TRANSCRIPTIONAL REGULATOR FROM STREPTOMYCES COELICOLOR A3 | APC7240, TETR-FAMILY TRANSCRIPTIONAL REGULATOR, STREPTOMYCES COELICOLOR A3, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSCRIPTION
2ama:A (SER696) to (SER740) CRYSTAL STRUCTURE OF HUMAN ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH DIHYDROTESTOSTERONE | NUCLEAR RECEPTOR, ANDROGEN RECEPTOR, LIGAND BINDING DOMAIN, DHT, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
1a8i:A (VAL715) to (MET766) SPIROHYDANTOIN INHIBITOR OF GLYCOGEN PHOSPHORYLASE | GLYCOGEN PHOSPHORYLASE, GLUCOPYRANOSE SPIROHYDANTOIN, WATER STRUCTURE, INHIBITOR BINDING, ANTI-HYPERGLYCEMIC AGENT
2au3:A (SER76) to (ASP142) CRYSTAL STRUCTURE OF THE AQUIFEX AEOLICUS PRIMASE (ZINC BINDING AND RNA POLYMERASE DOMAINS) | ZINC RIBBON, TOPRIM, RNA POLYMERASE, DNA REPLICATION, TRANSFERASE
2ax9:A (ILE672) to (TRP741) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH R-3 | TRANSCRIPTION
1nok:A (ARG714) to (MET766) COMPLEX OF GLYCOGEN PHOSPHORYLASE WITH A TRANSITION STATE ANALOGUE NOJIRIMYCIN TETRAZOLE AND PHOSPHATE IN THE T STATE | GLYCOGEN PHOSPHORYLASE, TRANSFERASE, GLYCOSYLTRANSFERASE
2oun:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 IN COMPLEX WITH AMP | PDE, PRODUCT BINDING, HYDROLASE
2our:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 MUTANT D674A IN COMPLEX WITH CAMP | PDE10, CAMP, SUBSTRATE SPECIFICITY, HYDROLASE
2ous:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 MUTANT D674A | PDE, HYDROLASE
2ous:B (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 MUTANT D674A | PDE, HYDROLASE
2ouu:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 MUTANT D674A IN COMPLEX WITH CGMP | PDE, CGMP, SUBSTRATE SPECIFICITY, HYDROLASE
2ouv:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 MUTANT OF D564N | PDE, HYDROLASE
2ouz:A (THR311) to (ALA382) CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR ALPHA-LASOFOXIFENE COMPLEX | NUCLEAR RECEPTOR, SERM, ESTROGEN, HORMONE-GROWTH FACTOR COMPLEX
3ek1:G (VAL48) to (VAL127) CRYSTAL STRUCTURE OF ALDEHYDE DEHYDROGENASE FROM BRUCELLA MELITENSIS BIOVAR ABORTUS 2308 | SSGCID, ALDEHYDE DEHYDROGENASE,, OXIDOREDUCTASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE
3ek1:H (SER47) to (VAL127) CRYSTAL STRUCTURE OF ALDEHYDE DEHYDROGENASE FROM BRUCELLA MELITENSIS BIOVAR ABORTUS 2308 | SSGCID, ALDEHYDE DEHYDROGENASE,, OXIDOREDUCTASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE
2ovv:A (ASN562) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF RAT PHOSPHODIESTERASE 10A | PHOSPHODIESTERASE 10A; ZN-BINDING SITE, HYDROLASE
2ovy:A (ASN562) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF RAT PHOSPHODIESTERASE 10A | PHOSPHODIESTERASE 10A; ZN-BINDING SITE, HYDROLASE
1nux:A (THR1012) to (SER1088) FRUCTOSE-1,6-BISPHOSPHATASE COMPLEX WITH MAGNESIUM, FRUCTOSE-6- PHOSPHATE, PHOSPHATE AND INHIBITORY CONCENTRATIONS OF POTASSIUM (200MM) | BISPHOSPHATASE, ALLOSTERIC ENZYMES, GLUCONEOGENESIS, HYDROLASE
1nv2:A (THR1012) to (SER1088) FRUCTOSE-1,6-BISPHOSPHATASE COMPLEX WITH MAGNESIUM, FRUCTOSE-6- PHOSPHATE, PHOSPHATE AND THALLIUM (20 MM) | BISPHOSPHATASE, ALLOSTERIC ENZYMES, GLUCONEOGENESIS, HYDROLASE
1nv3:A (THR1012) to (SER1088) FRUCTOSE-1,6-BISPHOSPHATASE COMPLEX WITH MAGNESIUM, FRUCTOSE-6- PHOSPHATE, PHOSPHATE AND THALLIUM (100 MM) | BISPHOSPHATASE, ALLOSTERIC ENZYMES, GLUCONEOGENESIS, HYDROLASE
1nv6:A (THR1012) to (SER1088) FRUCTOSE-1,6-BISPHOSPHATASE COMPLEX WITH MAGNESIUM, FRUCTOSE-6- PHOSPHATE, PHOSPHATE, EDTA AND THALLIUM (20 MM) | BISPHOSPHATASE, ALLOSTERIC ENZYMES, GLUCONEOGENESIS, HYDROLASE
2p15:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF THE ER ALPHA LIGAND BINDING DOMAIN WITH THE AGONIST ORTHO-TRIFLUOROMETHYLPHENYLVINYL ESTRADIOL | NULEAR RECEPTOR, LIGAND BINDING DOMAIN, HELIX 12, HORMONE RECEPTOR
4he0:A (THR12) to (SER88) CRYSTAL STRUCTURE OF HUMAN MUSCLE FRUCTOSE-1,6-BISPHOSPHATASE | ALLOSTERIC ENZYME, HYDROLASE
1b4d:A (ARG714) to (MET766) AMIDOCARBAMATE INHIBITOR OF GLYCOGEN PHOSPHORYLASE | GLYCOGEN PHOSPHORYLASE, INHIBITOR BINDING, AMIDOCARBAMATE, TRANSFERASE
4heu:A (SER561) to (THR623) CRYSTAL STRUCTURE OF PDE10A WITH A BIARYL ETHER INHIBITOR ((1-(3-(4- ((1H-BENZO[D]IMIDAZOL-2-YL)AMINO)PHENOXY)PYRIDIN-2-YL)PIPERIDIN-4- YL)METHANOL) | PDE10A, INHIBITORS, PHOSPHODIESTERASE 10A, BIARYL ETHERS, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4heu:B (SER561) to (THR623) CRYSTAL STRUCTURE OF PDE10A WITH A BIARYL ETHER INHIBITOR ((1-(3-(4- ((1H-BENZO[D]IMIDAZOL-2-YL)AMINO)PHENOXY)PYRIDIN-2-YL)PIPERIDIN-4- YL)METHANOL) | PDE10A, INHIBITORS, PHOSPHODIESTERASE 10A, BIARYL ETHERS, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1o2d:A (LEU254) to (GLY312) CRYSTAL STRUCTURE OF ALCOHOL DEHYDROGENASE, IRON-CONTAINING (TM0920) FROM THERMOTOGA MARITIMA AT 1.30 A RESOLUTION | TM0920, ALCOHOL DEHYDROGENASE, IRON-CONTAINING, STRUCTURAL GENOMICS, JCSG, PSI, PROTEIN STRUCTURE INITIATIVE, JOINT CENTER FOR STRUCTURAL GENOMICS, OXIDOREDUCTASE
1o2d:B (LEU254) to (GLY312) CRYSTAL STRUCTURE OF ALCOHOL DEHYDROGENASE, IRON-CONTAINING (TM0920) FROM THERMOTOGA MARITIMA AT 1.30 A RESOLUTION | TM0920, ALCOHOL DEHYDROGENASE, IRON-CONTAINING, STRUCTURAL GENOMICS, JCSG, PSI, PROTEIN STRUCTURE INITIATIVE, JOINT CENTER FOR STRUCTURAL GENOMICS, OXIDOREDUCTASE
3s5r:A (ILE129) to (GLY200) CRYSTAL STRUCTURE OF A PUTATIVE TRANSCRIPTIONAL REGULATOR OF THE TETR FAMILY (SYN_02108) FROM SYNTROPHUS ACIDITROPHICUS AT 2.60 A RESOLUTION | DNA/RNA-BINDING 3-HELICAL BUNDLE, TETRACYCLIN REPRESSOR-LIKE, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, DNA BINDING PROTEIN
4xai:B (MET338) to (GLN1246) CRYSTAL STRUCTURE OF RED FLOUR BEETLE NR2E1/TLX | HELICAL SANDWICH, TRANSPORT PROTEIN-TRANSCRIPTION COMPLEX
2pfm:A (GLN378) to (LEU430) CRYSTAL STRUCTURE OF ADENYLOSUCCINATE LYASE (PURB) FROM BACILLUS ANTHRACIS | ADENYLOSUCCINATE LYASE, PURB, PURINE BIOSYNTHESIS, BA0290, BACILLUS ANTHRACIS, LYASE
4htz:D (ASN704) to (THR768) CRYSTAL STRUCTURE OF PDE2 CATALYTIC DOMAIN IN SPACE GROUP P1 | HYDROLASE
4hxd:D (CYS40) to (LYS95) DIVERSITY OF UBIQUITIN AND ISG15 SPECIFICITY AMONGST NAIROVIRUSES VIRAL OVARIAN TUMOR DOMAIN PROTEASES | OTU-LIKE CYSTEINE PROTEASE, DUGBE VIRUS, DEUBIQUITINASE, 3- AMINOPROPANE, UBIQUITIN HYDROLASE, VIRAL PROTEIN, HYDROLASE, UBIQUITIN., HYDROLASE-VIRAL PROTEIN COMPLEX
2ptm:A (GLU516) to (LEU561) STRUCTURE AND REARRANGEMENTS IN THE CARBOXY-TERMINAL REGION OF SPIH CHANNELS | ION CHANNEL, CYCLIC NUCLEOTIDE BINDING DOMAIN, C-LINKER, CAMP, CGMP, SPHCN1, HCN, TRANSPORT PROTEIN
4xk4:A (LEU134) to (ILE209) E. COLI TRANSCRIPTIONAL REGULATOR RUTR WITH DIHYDROURACIL | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, HELIX-TURN-HELIX, TRANSCRIPTIONAL REGULATOR, TRANSCRIPTION REGULATOR
4xk4:B (LEU134) to (ILE209) E. COLI TRANSCRIPTIONAL REGULATOR RUTR WITH DIHYDROURACIL | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, HELIX-TURN-HELIX, TRANSCRIPTIONAL REGULATOR, TRANSCRIPTION REGULATOR
4xk4:C (LEU134) to (ILE209) E. COLI TRANSCRIPTIONAL REGULATOR RUTR WITH DIHYDROURACIL | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, HELIX-TURN-HELIX, TRANSCRIPTIONAL REGULATOR, TRANSCRIPTION REGULATOR
4xk4:D (LEU134) to (ILE209) E. COLI TRANSCRIPTIONAL REGULATOR RUTR WITH DIHYDROURACIL | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, HELIX-TURN-HELIX, TRANSCRIPTIONAL REGULATOR, TRANSCRIPTION REGULATOR
3sl3:B (HIS105) to (TYR153) CRYSTAL STRUCTURE OF THE APO FORM OF THE CATALYTIC DOMAIN OF PDE4D2 | CATALYTIC MECHANISM, CAMP HYDROLYSIS, HYDROLASE
3sn7:A (ASN562) to (THR623) HIGHLY POTENT, SELECTIVE, AND ORALLY ACTIVE PHOSPHODIESTARASE 10A INHIBITORS | HYDROLASE, HYDROLASE INHIBITOR, ZN BINDING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2pyi:A (ARG714) to (MET766) CRYSTAL STRUCTURE OF GLYCOGEN PHOSPHORYLASE IN COMPLEX WITH GLUCOSYL TRIAZOLEACETAMIDE | GLYCOGENOLYSIS, INHIBITION, TYPE 2 DIABETES, TRANSFERASE
3sni:A (SER561) to (THR623) HIGHLY POTENT, SELECTIVE, AND ORALLY ACTIVE PHOSPHODIESTARASE 10A INHIBITORS | HYDROLASE, HYDROLASE INHIBITOR, ZN BINDING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3snl:A (SER561) to (THR623) HIGHLY POTENT, SELECTIVE, AND ORALLY ACTIVE PHOSPHODIESTARASE 10A INHIBITORS | HYDROLASE, HYDROLASE INHIBITOR, ZN BINDING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1ord:A (THR548) to (ASN588) CRYSTALLOGRAPHIC STRUCTURE OF A PLP-DEPENDENT ORNITHINE DECARBOXYLASE FROM LACTOBACILLUS 30A TO 3.1 ANGSTROMS RESOLUTION | CARBOXY-LYASE
1ord:B (THR548) to (ASN588) CRYSTALLOGRAPHIC STRUCTURE OF A PLP-DEPENDENT ORNITHINE DECARBOXYLASE FROM LACTOBACILLUS 30A TO 3.1 ANGSTROMS RESOLUTION | CARBOXY-LYASE
1cls:B (THR4) to (ASN57) CROSS-LINKED HUMAN HEMOGLOBIN DEOXY | OXYGEN TRANSPORT, HEMOGLOBIN, HUMAN, DEOXY, CROSS-LINKED
1cnq:A (THR12) to (SER88) FRUCTOSE-1,6-BISPHOSPHATASE COMPLEXED WITH FRUCTOSE-6-PHOSPHATE AND ZINC IONS | BISPHOSPHATASE, HYDROLASE
1coh:B (THR4) to (ASN57) STRUCTURE OF HAEMOGLOBIN IN THE DEOXY QUATERNARY STATE WITH LIGAND BOUND AT THE ALPHA HAEMS | OXYGEN TRANSPORT
3fs3:A (THR36) to (VAL126) CRYSTAL STRUCTURE OF MALARIA PARASITE NUCLEOSOME ASSEMBLY PROTEIN (NAP) | PLASMODIUM FALCIPARUM, NUCLEOSOME ASSEMBLY PROTEIN, PROTEIN LOCALIZATION, HISTONE RECOGNITION, STRUCTURAL ANALYSIS, CHAPERONE
4ia7:A (TYR179) to (ALA295) DIASTEREOTOPIC AND DEUTERIUM EFFECTS IN GEMINI | VDR-AGONIST COMPLEX, ALPHA HELICAL SANDWICH, TRANSCRIPTION REGULATION, DNA, RXR, PHOSPHORYLATION, NUCLEUS, TRANSCRIPTION- TRANSCRIPTION ACTIVATOR COMPLEX
1out:A (ALA21) to (SER82) TROUT HEMOGLOBIN I | HEME, OXYGEN TRANSPORT, RESPIRATORY PROTEIN, ERYTHROCYTE
1ouu:A (ALA21) to (MET81) CARBONMONOXY TROUT HEMOGLOBIN I | HEME, OXYGEN TRANSPORT, RESPIRATORY PROTEIN, ERYTHROCYTE
1ouu:C (ALA21) to (MET81) CARBONMONOXY TROUT HEMOGLOBIN I | HEME, OXYGEN TRANSPORT, RESPIRATORY PROTEIN, ERYTHROCYTE
2qe0:B (THR39) to (MET118) THIOACYLENZYME INTERMEDIATE OF GAPN FROM S. MUTANS, NEW DATA INTEGRATION AND REFINEMENT. | ALDH, GAPN, TERNARY COMPLEX, OXIDOREDUCTASE
2qe0:C (THR39) to (MET118) THIOACYLENZYME INTERMEDIATE OF GAPN FROM S. MUTANS, NEW DATA INTEGRATION AND REFINEMENT. | ALDH, GAPN, TERNARY COMPLEX, OXIDOREDUCTASE
2qe0:D (THR39) to (MET118) THIOACYLENZYME INTERMEDIATE OF GAPN FROM S. MUTANS, NEW DATA INTEGRATION AND REFINEMENT. | ALDH, GAPN, TERNARY COMPLEX, OXIDOREDUCTASE
3g3n:A (GLN261) to (ASP322) PDE7A CATALYTIC DOMAIN IN COMPLEX WITH 3-(2,6- DIFLUOROPHENYL)-2-(METHYLTHIO)QUINAZOLIN-4(3H)-ONE | PDE7, CRYSTAL, INHIBITOR COMPLEX, ALTERNATIVE SPLICING, CAMP, HYDROLASE, PHOSPHOPROTEIN
1d9q:C (THR20) to (LEU93) OXIDIZED PEA FRUCTOSE-1,6-BISPHOSPHATASE FORM 1 | CHLOROPLAST, PHOTOSYNTHESIS, REDOX REGULATION, THIOREDOXIN, ALLOSTERY, DISULFIDE BRIDGE, CALVIN CYCLE, HYDROLASE
1d9q:D (LEU21) to (LEU93) OXIDIZED PEA FRUCTOSE-1,6-BISPHOSPHATASE FORM 1 | CHLOROPLAST, PHOTOSYNTHESIS, REDOX REGULATION, THIOREDOXIN, ALLOSTERY, DISULFIDE BRIDGE, CALVIN CYCLE, HYDROLASE
3g58:C (ASN375) to (ASP438) CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 4D WITH D155988/PMNPQ | PHOSPHODIESTERASE, PDE4D, ALTERNATIVE SPLICING, CAMP, CYTOPLASM, CYTOSKELETON, HYDROLASE, MEMBRANE, METAL- BINDING, PHOSPHOPROTEIN
1dbz:D (LEU21) to (LEU93) C153S MUTANT OF PEA FRUCTOSE-1,6-BISPHOSPHATASE | CHLOROPLAST, PHOTOSYNTHESIS, REDOX REGULATION, THIOREDOXIN, ALLOSTERY, DISULFIDE BRIDGE, CALVIN CYCLE, HYDROLASE
2qfz:B (LEU432) to (ASN483) CRYSTAL STRUCTURE OF HUMAN TBC1 DOMAIN FAMILY MEMBER 22A | RAB-GAP, GTPASE ACTIVATOR, TBC1, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, HYDROLASE ACTIVATOR
1dcu:A (THR20) to (CYS92) REDOX SIGNALING IN THE CHLOROPLAST: STRUCTURE OF OXIDIZED PEA FRUCTOSE-1,6-BISPHOSPHATE PHOSPHATASE | CHLOROPLAST, PHOTOSYNTHESIS, REDOX REGULATION, THIOREDOXIN, ALLOSTERY, HYDROLASE
1dcu:D (THR20) to (CYS92) REDOX SIGNALING IN THE CHLOROPLAST: STRUCTURE OF OXIDIZED PEA FRUCTOSE-1,6-BISPHOSPHATE PHOSPHATASE | CHLOROPLAST, PHOTOSYNTHESIS, REDOX REGULATION, THIOREDOXIN, ALLOSTERY, HYDROLASE
2qg7:A (ASN215) to (ASN287) PLASMODIUM VIVAX ETHANOLAMINE KINASE PV091845 | MALARIA, ETHANOLAMINE KINASE, PV091845, SGC, STRUCTURAL GENOMICS CONSORTIUM, TRANSFERASE
4iod:B (SER90) to (VAL154) PRELIMINARY STRUCTURAL INVESTIGATIONS OF A MALARIAL PROTEIN SECRETION SYSTEM. | MALARIA, AAA+ ATPASE CLPB CHAPERONE, N-TERMINAL CARGO-BINDING DOMAIN, PROTEIN TRANSLOCATION AND UNFOLDING, PARASITOPHOROUS VACUOLE, CHAPERONE
4is8:A (GLU315) to (CYS381) DIVERGENT SEQUENCE TUNES LIGAND SENSITIVITY IN PHOSPHOLIPID-REGULATED HORMONE RECEPTORS | LIGAND BINDING DOMAIN, TRANSCRIPTION
3t3z:A (ASP264) to (PRO365) HUMAN CYTOCHROME P450 2E1 IN COMPLEX WITH PILOCARPINE | CYP2E1, CYTOCHROME P450 2E1, P450 2E1, HEME PROTEIN, MONOOXYGENASE, DRUG METABOLISM, XENOBIOTIC METABOLISM, ENDOPLASMIC RETICULUM, MEMBRANE, OXIDOREDUCTASE
3t3z:B (LEU265) to (PRO365) HUMAN CYTOCHROME P450 2E1 IN COMPLEX WITH PILOCARPINE | CYP2E1, CYTOCHROME P450 2E1, P450 2E1, HEME PROTEIN, MONOOXYGENASE, DRUG METABOLISM, XENOBIOTIC METABOLISM, ENDOPLASMIC RETICULUM, MEMBRANE, OXIDOREDUCTASE
3t3z:D (ASP267) to (PRO365) HUMAN CYTOCHROME P450 2E1 IN COMPLEX WITH PILOCARPINE | CYP2E1, CYTOCHROME P450 2E1, P450 2E1, HEME PROTEIN, MONOOXYGENASE, DRUG METABOLISM, XENOBIOTIC METABOLISM, ENDOPLASMIC RETICULUM, MEMBRANE, OXIDOREDUCTASE
4itb:A (PRO22) to (HIS97) STRUCTURE OF BACTERIAL ENZYME IN COMPLEX WITH COFACTOR AND SUBSTRATE | ROSSMANN FOLD, OXIDOREDUCTASE, OXIDOREDUCTASE-SUBSTRATE COMPLEX
4xy2:B (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A IN COMPLEX WITH ASP9436 | PHOSPHODIESTERASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2qrp:A (VAL715) to (MET766) GLYCOGEN PHOSPHORYLASE B IN COMPLEX WITH (1R)-3'-(2- NAPHTHYL)-SPIRO[1,5-ANHYDRO-D-GLUCITOL-1,5'-ISOXAZOLINE] | GLYCOGENOLYSIS, TYPE 2 DIABETES, ACETYLATION, ALLOSTERIC ENZYME, CARBOHYDRATE METABOLISM, GLYCOGEN METABOLISM, GLYCOSYLTRANSFERASE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, PYRIDOXAL PHOSPHATE, TRANSFERASE
2qrq:A (VAL715) to (MET766) GLYCOGEN PHOSPHORYLASE B IN COMPLEX WITH (1R)-3'-(4- METHYLPHENYL)-SPIRO[1,5-ANHYDRO-D-GLUCITOL-1,5'- ISOXAZOLINE] | GLYCOGENOLYSIS, TYPE 2 DIABETES, ACETYLATION, ALLOSTERIC ENZYME, CARBOHYDRATE METABOLISM, GLYCOGEN METABOLISM, GLYCOSYLTRANSFERASE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, PYRIDOXAL PHOSPHATE, TRANSFERASE
1pqk:A (SER38) to (MET106) REPACKING OF THE CORE OF T4 LYSOZYME BY AUTOMATED DESIGN | HYDROLASE (O-GLYCOSYL), T4 LYSOZYME, DESIGNED CORE MUTANT, AUTOMATED PROTEIN DESIGN, PROTEIN ENGINEERING, PROTEIN FOLDING, PROTEIN STABILITY, CORE REPACKING, BACK REVERTANT, DEAD-END ELIMINATION THEOREM, SIDE-CHAIN PACKING, OPTIMIZED ROTAMER COMBINATIONS, ORBIT
1dxt:B (THR5) to (ASN58) HIGH-RESOLUTION X-RAY STUDY OF DEOXY RECOMBINANT HUMAN HEMOGLOBINS SYNTHESIZED FROM BETA-GLOBINS HAVING MUTATED AMINO TERMINI | OXYGEN TRANSPORT
4y06:A (GLN430) to (ALA496) CRYSTAL STRUCTURE OF THE DAP BII (G675R) DIPEPTIDE COMPLEX | HYDROLASE
4y06:B (GLN430) to (ALA496) CRYSTAL STRUCTURE OF THE DAP BII (G675R) DIPEPTIDE COMPLEX | HYDROLASE
4y0b:A (THR164) to (MSE225) THE STRUCTURE OF ARABIDOPSIS CLPT1 | CASEINOLYTIC PROTEASE, N-DOMAIN, ALPHA HELICAL BUNDLE, PLASTID
4y0b:B (THR164) to (ASN226) THE STRUCTURE OF ARABIDOPSIS CLPT1 | CASEINOLYTIC PROTEASE, N-DOMAIN, ALPHA HELICAL BUNDLE, PLASTID
1ps1:A (TYR50) to (GLY107) PENTALENENE SYNTHASE | ANTIBIOTIC BIOSYNTHESIS, SESQUITERPENE CYCLASE, LYASE
3gph:A (LEU265) to (PRO365) HUMAN CYTOCHROME P450 2E1 IN COMPLEX WITH OMEGA-IMIDAZOLYL-DECANOIC ACID | CYP2E1, P450 2E1, MONOOXYGENASE, ACETAMINOPHEN, OXIDOREDUCTASE, HEME, FATTY ACID HYDROXYLASE, METAL-BINDING
3gqr:D (THR4) to (ASN57) CRYSTAL STRUCTURE DETERMINATION OF CAT (FELIS SILVESTRIS CATUS) HEMOGLOBIN AT 2.4 ANGSTROM RESOLUTION | LOW OXYGEN AFFINITY, METHEMOGLOBIN, ORTHORHOMBIC, HEME, IRON, OXYGEN TRANSPORT, TRANSPORT, POLYMORPHISM, OXYGEN STORAGE
1pyg:B (ARG714) to (MET766) STRUCTURAL BASIS FOR THE ACTIVATION OF GLYCOGEN PHOSPHORYLASE B BY ADENOSINE MONOPHOSPHATE | GLYCOGEN PHOSPHORYLASE
4j72:A (GLY264) to (MET355) CRYSTAL STRUCTURE OF POLYPRENYL-PHOSPHATE N-ACETYL HEXOSAMINE 1- PHOSPHATE TRANSFERASE | ALPHA-HELICAL MEMBRANE PROTEIN, MEMBRANE ENZYME, MAGNESIUM BINDING, UNDECAPRENYL PHOSPHATE BINDING, UDP-MURNAC-PENTAPEPTIDE BINDING, MEMBRANE, TRANSFERASE
4j72:B (GLY264) to (MET355) CRYSTAL STRUCTURE OF POLYPRENYL-PHOSPHATE N-ACETYL HEXOSAMINE 1- PHOSPHATE TRANSFERASE | ALPHA-HELICAL MEMBRANE PROTEIN, MEMBRANE ENZYME, MAGNESIUM BINDING, UNDECAPRENYL PHOSPHATE BINDING, UDP-MURNAC-PENTAPEPTIDE BINDING, MEMBRANE, TRANSFERASE
4jag:B (ILE1117) to (SER1166) STRUCTURAL DETERMINATION OF THE A50T:S279G:S280K:V281K:K282E:H283N VARIANT OF CITRATE SYNTHASE FROM E. COLI COMPLEXED WITH OXALOACETATE | CITRATE SYNTHASE, GRAM-NEGATIVE BACTERIA, ALLOSTERY, OXALOACETATE, ACETYL-COA, NADH, PROTEIN FOLDING, S-CARBOXYMETHYL-COA, ALLOSTERIC ENZYME, TRANSFERASE, TRICARBOXYLIC ACID CYCLE
1q5n:A (ARG382) to (LYS427) CRYSTAL STRUCTURE OF BETA-CARBOXY-CIS,CIS-MUCONATE CYCLOISOMERASE (CMLE) FROM ACINETOBACTER CALCOACETICUS SP. ADP1 | CMLE, CYCLOISOMERASE, AROMATIC DEGRADATION, ISOMERASE
3tor:A (ALA97) to (HIS144) CRYSTAL STRUCTURE OF ESCHERICHIA COLI NRFA WITH EUROPIUM BOUND | MULTIHAEM CYTOCHROME, DECAHEME, REDUCTASE, ELECTRON TRANSPORT, IRON, METAL-BINDING, OXIDOREDUCTASE, NITRITE, CALCIUM BINDING
3tor:B (ALA97) to (HIS144) CRYSTAL STRUCTURE OF ESCHERICHIA COLI NRFA WITH EUROPIUM BOUND | MULTIHAEM CYTOCHROME, DECAHEME, REDUCTASE, ELECTRON TRANSPORT, IRON, METAL-BINDING, OXIDOREDUCTASE, NITRITE, CALCIUM BINDING
3tor:C (ALA97) to (HIS144) CRYSTAL STRUCTURE OF ESCHERICHIA COLI NRFA WITH EUROPIUM BOUND | MULTIHAEM CYTOCHROME, DECAHEME, REDUCTASE, ELECTRON TRANSPORT, IRON, METAL-BINDING, OXIDOREDUCTASE, NITRITE, CALCIUM BINDING
3tor:D (ALA97) to (HIS144) CRYSTAL STRUCTURE OF ESCHERICHIA COLI NRFA WITH EUROPIUM BOUND | MULTIHAEM CYTOCHROME, DECAHEME, REDUCTASE, ELECTRON TRANSPORT, IRON, METAL-BINDING, OXIDOREDUCTASE, NITRITE, CALCIUM BINDING
3gyv:A (PRO77) to (VAL126) CRYSTAL STRUCTURE OF NUCLEOSOME ASSEMBLY PROTEIN FROM PLASMODIUM FALCIPARUM | IODIDE-SAD, NUCLEOSOME ASSEMBLY PROTEIN, HISTONE RECOGNITION, CHAPERONE
3gyw:A (PRO77) to (VAL126) CRYSTAL STRUCTURE OF NUCLEOSOME ASSEMBLY PROTEIN FROM PLASMODIUM FALCIPARUM AT 2.4 A RESOLUTION | SIR, SIRAS, NUCLEOSOME ASSEMBLY PROTEIN, HISTONE RECOGNITION, CHAPERONE
2rdz:A (ALA97) to (HIS144) HIGH RESOLUTION CRYSTAL STRUCTURE OF THE ESCHERICHIA COLI CYTOCHROME C NITRITE REDUCTASE. | DECAHEME, REDUCTASE, ELECTRON TRANSPORT, IRON, METAL-BINDING, OXIDOREDUCTASE, TRANSPORT
2rdz:B (ALA97) to (HIS144) HIGH RESOLUTION CRYSTAL STRUCTURE OF THE ESCHERICHIA COLI CYTOCHROME C NITRITE REDUCTASE. | DECAHEME, REDUCTASE, ELECTRON TRANSPORT, IRON, METAL-BINDING, OXIDOREDUCTASE, TRANSPORT
2rdz:C (ALA97) to (HIS144) HIGH RESOLUTION CRYSTAL STRUCTURE OF THE ESCHERICHIA COLI CYTOCHROME C NITRITE REDUCTASE. | DECAHEME, REDUCTASE, ELECTRON TRANSPORT, IRON, METAL-BINDING, OXIDOREDUCTASE, TRANSPORT
2rdz:D (ALA97) to (HIS144) HIGH RESOLUTION CRYSTAL STRUCTURE OF THE ESCHERICHIA COLI CYTOCHROME C NITRITE REDUCTASE. | DECAHEME, REDUCTASE, ELECTRON TRANSPORT, IRON, METAL-BINDING, OXIDOREDUCTASE, TRANSPORT
2rf7:A (ALA97) to (HIS144) CRYSTAL STRUCTURE OF THE ESCHERICHIA COLI NRFA MUTANT Q263E | OXIDOREDUCTASE, CALCIUM LIGAND, ELECTRON TRANSPORT, HEME, IRON, METAL-BINDING, PERIPLASM, TRANSPORT
2rf7:B (ALA97) to (HIS144) CRYSTAL STRUCTURE OF THE ESCHERICHIA COLI NRFA MUTANT Q263E | OXIDOREDUCTASE, CALCIUM LIGAND, ELECTRON TRANSPORT, HEME, IRON, METAL-BINDING, PERIPLASM, TRANSPORT
2rf7:C (ALA97) to (HIS144) CRYSTAL STRUCTURE OF THE ESCHERICHIA COLI NRFA MUTANT Q263E | OXIDOREDUCTASE, CALCIUM LIGAND, ELECTRON TRANSPORT, HEME, IRON, METAL-BINDING, PERIPLASM, TRANSPORT
2rf7:D (ALA97) to (HIS144) CRYSTAL STRUCTURE OF THE ESCHERICHIA COLI NRFA MUTANT Q263E | OXIDOREDUCTASE, CALCIUM LIGAND, ELECTRON TRANSPORT, HEME, IRON, METAL-BINDING, PERIPLASM, TRANSPORT
2dxm:B (THR4) to (ASN57) NEUTRON STRUCTURE ANALYSIS OF DEOXY HUMAN HEMOGLOBIN | ALPHA2-BETA2, OXYGEN STORAGE-TRANSPORT COMPLEX
1qi6:A (THR39) to (ARG117) SECOND APO FORM OF AN NADP DEPENDENT ALDEHYDE DEHYDROGENASE WITH GLU250 SITUATED 3.7 A FROM CYS284 | OXIDOREDUCTASE
1qi6:B (THR39) to (ARG117) SECOND APO FORM OF AN NADP DEPENDENT ALDEHYDE DEHYDROGENASE WITH GLU250 SITUATED 3.7 A FROM CYS284 | OXIDOREDUCTASE
1qi6:C (THR39) to (ARG117) SECOND APO FORM OF AN NADP DEPENDENT ALDEHYDE DEHYDROGENASE WITH GLU250 SITUATED 3.7 A FROM CYS284 | OXIDOREDUCTASE
1qi6:D (THR39) to (ARG117) SECOND APO FORM OF AN NADP DEPENDENT ALDEHYDE DEHYDROGENASE WITH GLU250 SITUATED 3.7 A FROM CYS284 | OXIDOREDUCTASE
1qi1:C (THR39) to (MET118) TERNARY COMPLEX OF AN NADP DEPENDENT ALDEHYDE DEHYDROGENASE | OXIDOREDUCTASE
1qi1:D (THR39) to (MET118) TERNARY COMPLEX OF AN NADP DEPENDENT ALDEHYDE DEHYDROGENASE | OXIDOREDUCTASE
1euh:A (THR39) to (MET118) APO FORM OF A NADP DEPENDENT ALDEHYDE DEHYDROGENASE FROM STREPTOCOCCUS MUTANS | DEHYDROGENASE, OXIDOREDUCTASE
1euh:D (THR39) to (MET118) APO FORM OF A NADP DEPENDENT ALDEHYDE DEHYDROGENASE FROM STREPTOCOCCUS MUTANS | DEHYDROGENASE, OXIDOREDUCTASE
1ewa:A (GLY1) to (MET49) DEHALOPEROXIDASE AND 4-IODOPHENOL | PEROXIDASE, GLOBIN, OXIDOREDUCTASE
1ewa:B (GLY1) to (MET49) DEHALOPEROXIDASE AND 4-IODOPHENOL | PEROXIDASE, GLOBIN, OXIDOREDUCTASE
1f0l:A (HIS223) to (VAL288) 1.55 ANGSTROM CRYSTAL STRUCTURE OF WILD TYPE DIPHTHERIA TOXIN | BACTERIAL TOXIN, ADP-RIBOSYLATION, TRANSMEMBRANE
2e50:A (GLN65) to (MET104) CRYSTAL STRUCTURE OF SET/TAF-1BETA/INHAT | HISTONE CHAPERONE, INHAT, SET, PP2AI, PROTEIN BINDING
2e50:B (LYS26) to (MET104) CRYSTAL STRUCTURE OF SET/TAF-1BETA/INHAT | HISTONE CHAPERONE, INHAT, SET, PP2AI, PROTEIN BINDING
2e50:Q (GLN65) to (HIS105) CRYSTAL STRUCTURE OF SET/TAF-1BETA/INHAT | HISTONE CHAPERONE, INHAT, SET, PP2AI, PROTEIN BINDING
2uum:E (THR3) to (ILE100) CRYSTAL STRUCTURE OF C-PHYCOCYANIN FROM PHORMIDIUM, LYNGBYA SPP. (MARINE) AND SPIRULINA SP. (FRESH WATER) SHOWS TWO DIFFERENT WAYS OF ENERGY TRANSFER BETWEEN TWO HEXAMERS. | PHOTOSYNTHESIS, ELECTRON TRANSPORT, SPIRULINA SP, C-PHYCOCYANIN, PHYCOBILISOME, MARINE, TRANSPORT, LYNGBYA SP, PHORMIDIUM, CHROMOPHORE, FRESH WATER, METHYLATION, BILE PIGMENT
3u11:B (ASP565) to (LEU611) TETRAMERIZATION DYNAMICS OF THE C-TERMINUS UNDERLIES ISOFORM-SPECIFIC CAMP-GATING IN HCN CHANNELS | TRANSPORT PROTEIN
3u1n:A (PHE165) to (ASN248) STRUCTURE OF THE CATALYTIC CORE OF HUMAN SAMHD1 | HD-DOMAIN, DEOXYNUCLEOTIDE TRIPHOSPHOHYDROLASE, HYDROLASE
3u1n:B (PHE213) to (GLY274) STRUCTURE OF THE CATALYTIC CORE OF HUMAN SAMHD1 | HD-DOMAIN, DEOXYNUCLEOTIDE TRIPHOSPHOHYDROLASE, HYDROLASE
3u1n:C (PHE165) to (ASN248) STRUCTURE OF THE CATALYTIC CORE OF HUMAN SAMHD1 | HD-DOMAIN, DEOXYNUCLEOTIDE TRIPHOSPHOHYDROLASE, HYDROLASE
3u1n:D (PHE165) to (ASN248) STRUCTURE OF THE CATALYTIC CORE OF HUMAN SAMHD1 | HD-DOMAIN, DEOXYNUCLEOTIDE TRIPHOSPHOHYDROLASE, HYDROLASE
1qvr:A (THR7) to (LEU71) CRYSTAL STRUCTURE ANALYSIS OF CLPB | COILED COIL, AAA ATPASE, CHAPERONE
1qvr:B (THR7) to (LEU71) CRYSTAL STRUCTURE ANALYSIS OF CLPB | COILED COIL, AAA ATPASE, CHAPERONE
1qvr:C (THR7) to (LEU71) CRYSTAL STRUCTURE ANALYSIS OF CLPB | COILED COIL, AAA ATPASE, CHAPERONE
1qvt:A (THR109) to (SER187) CRYSTAL STRUCTURE OF THE MULTIDRUG BINDING TRANSCRIPTIONAL REPRESSOR QACR BOUND TO THE DRUG PROFLAVINE | MULTIDRUG BINDING PROTEIN, REPRESSOR, TRANSCRIPTION, QACR
3hc8:A (ASN662) to (THR723) INVESTIGATION OF AMINOPYRIDIOPYRAZINONES AS PDE5 INHIBITORS: EVALUATION OF MODIFICATIONS TO THE CENTRAL RING SYSTEM. | PDE5, PDE-5,INHIBITION, ALTERNATIVE SPLICING, CAMP, HYDROLASE, PHOSPHOPROTEIN, POLYMORPHISM ALLOSTERIC ENZYME, CGMP, CGMP-BINDING, MAGNESIUM, METAL-BINDING, NUCLEOTIDE- BINDING, ZINC
1r1y:B (THR4) to (ASN57) CRYSTAL STRUCTURE OF DEOXY-HUMAN HEMOGLOBIN BASSETT AT 1.8 ANGSTROM | DEOXYHEMOGLOBIN, MUTANT, ROCHESTER, OXYGEN AFFINITY, CRYSTAL STRUCTURE, OXYGEN TRANSPORT
1r20:D (THR291) to (ALA374) CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAINS OF THE HETERODIMER ECR/USP BOUND TO THE SYNTHETIC AGONIST BYI06830 | NUCLEAR RECEPTOR, HETERODIMER, ALPHA-HELICAL SANDWICH, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, STRUCTURAL GENOMICS, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
4jyk:A (LEU134) to (ILE209) STRUCTURE OF E. COLI TRANSCRIPTIONAL REGULATOR RUTR WITH BOUND URACIL | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, HELIX-TURN-HELIX, TRANSCRIPTIONAL REGULATOR, TRANSCRIPTION REGULATOR
4jyk:B (LEU134) to (ILE209) STRUCTURE OF E. COLI TRANSCRIPTIONAL REGULATOR RUTR WITH BOUND URACIL | STRUCTURAL GENOMICS, PSI-BIOLOGY, NEW YORK STRUCTURAL GENOMICS RESEARCH CONSORTIUM, NYSGRC, HELIX-TURN-HELIX, TRANSCRIPTIONAL REGULATOR, TRANSCRIPTION REGULATOR
4jyq:A (GLY1) to (MET49) DHP-CO CRYSTAL STRUCTURE | GLOBIN, PEROXIDASE, OXIDOREDUCTASE
3hfd:A (THR36) to (VAL126) NUCLEOSOME ASSEMBLY PROTEIN 1 FROM PLASMODIUM KNOWLESI | HISTONE BINDING, STRUCTURAL GENOMICS, MEDICAL STRUCTURAL GENOMICS OF PATHOGENIC PROTOZOA, MSGPP, CHAPERONE, PROTEIN TRANSPORT
4ynk:A (LEU220) to (ALA263) CRYSTAL STRUCTURE OF VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH A 19-NORVITAMIN D COMPOUND | TRANSCRIPTION, HORMONE RECEPTOR
3hhc:B (ASP48) to (CYS103) INTERFERON-LAMBDA IS FUNCTIONALLY AN INTERFERON BUT STRUCTURALLY RELATED TO THE IL-10 FAMILY | INTERFERON, IL-22, ANTIVIRAL, ANTIVIRAL DEFENSE, CYTOKINE, SECRETED
4k1p:H (SER243) to (VAL357) STRUCTURE OF THE NHEA COMPONENT OF THE NHE TOXIN FROM BACILLUS CEREUS | HELICAL BUNDLE, BETA TONGUE, CLYA-LIKE FOLD, PORE-FORMING TOXIN COMPONENT, TOXIN
1r6o:B (THR81) to (SER139) ATP-DEPENDENT CLP PROTEASE ATP-BINDING SUBUNIT CLPA/ATP-DEPENDENT CLP PROTEASE ADAPTOR PROTEIN CLPS | CLPA, AAA+, N-TERMINAL DOMAIN, CLPS, CRYSTAL, BINDING MECHANISM, HYDROLASE
1r6q:B (THR81) to (SER139) CLPNS WITH FRAGMENTS | CLPA, AAA+, N-TERMINAL DOMAIN, CLPS, CRYSTAL, BINDING MECHANISM, CHAPERONE-PROTEIN BINDING COMPLEX
4yqh:A (SER571) to (THR633) 2-[2-(4-PHENYL-1H-IMIDAZOL-2-YL)ETHYL]QUINOXALINE (SUNOVION COMPOUND 14) CO-CRYSTALLIZED WITH PDE10A | INHIBITOR, PDE10A, CO-CRYSTAL
4yqh:B (SER571) to (THR633) 2-[2-(4-PHENYL-1H-IMIDAZOL-2-YL)ETHYL]QUINOXALINE (SUNOVION COMPOUND 14) CO-CRYSTALLIZED WITH PDE10A | INHIBITOR, PDE10A, CO-CRYSTAL
1fj6:A (THR12) to (SER88) FRUCTOSE-1,6-BISPHOSPHATASE (MUTANT Y57W) PRODUCT/ZN COMPLEX (R-STATE) | BISPHOSPHATASE, ALLOSTERIC ENZYMES, GLUCONEOGENESIS, HYDROLASE
2euh:A (THR39) to (ARG117) HOLO FORM OF A NADP DEPENDENT ALDEHYDE DEHYDROGENASE COMPLEX WITH NADP+ | OXIDOREDUCTASE, DEHYDROGENASE
2euh:B (THR39) to (ARG117) HOLO FORM OF A NADP DEPENDENT ALDEHYDE DEHYDROGENASE COMPLEX WITH NADP+ | OXIDOREDUCTASE, DEHYDROGENASE
2euh:C (THR39) to (ARG117) HOLO FORM OF A NADP DEPENDENT ALDEHYDE DEHYDROGENASE COMPLEX WITH NADP+ | OXIDOREDUCTASE, DEHYDROGENASE
2euh:D (THR39) to (ARG117) HOLO FORM OF A NADP DEPENDENT ALDEHYDE DEHYDROGENASE COMPLEX WITH NADP+ | OXIDOREDUCTASE, DEHYDROGENASE
4ys7:A (SER571) to (THR633) CO-CRYSTAL STRUCTURE OF 2-[2-(5,8-DIMETHYL[1,2,4]TRIAZOLO[1,5- A]PYRAZIN-2-YL)ETHYL]-3-METHYL-3H-IMIDAZO[4,5-F]QUINOLINE (COMPOUND 39) WITH PDE10A | PDE10A, INHIBITOR, CO-CRYSTAL, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4ys7:B (ASN572) to (THR633) CO-CRYSTAL STRUCTURE OF 2-[2-(5,8-DIMETHYL[1,2,4]TRIAZOLO[1,5- A]PYRAZIN-2-YL)ETHYL]-3-METHYL-3H-IMIDAZO[4,5-F]QUINOLINE (COMPOUND 39) WITH PDE10A | PDE10A, INHIBITOR, CO-CRYSTAL, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1rdf:B (THR41) to (ILE97) G50P MUTANT OF PHOSPHONOACETALDEHYDE HYDROLASE IN COMPLEX WITH SUBSTRATE ANALOGUE VINYL SULFONATE | HALOACID DEHALOGENASE, SPECIFICITY LOOP, PHOSPHONATASE, SCHIFF-BASE, HYDROLASE
2va8:B (ASN501) to (ASP586) DNA REPAIR HELICASE HEL308 | HEL308, SSO2462, HELICASE, HYDROLASE, DNA REPAIR, ATP-BINDING, NUCLEOTIDE-BINDING
1rjk:A (TYR147) to (SER262) CRYSTAL STRUCTURE OF THE RAT VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH 2MD AND A SYNTHETIC PEPTIDE CONTAINING THE NR2 BOX OF DRIP 205 | NUCLEAR RECEPTOR-SUPERAGONIST COMPLEX, NUCLEAR RECEPTOR- COACTIVATOR INTERACTIONS,, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
2f3b:A (THR12) to (SER88) MECHANISM OF DISPLACEMENT OF A CATALYTICALLY ESSENTIAL LOOP FROM THE ACTIVE SITE OF FRUCTOSE-1,6-BISPHOSPHATASE | ALLOSTERY, ALLOSTERIC REGULATION, LOOP DIENGAGEMENT, ENZYME CATALYSIS, FBPASE, FRUCTOSE-1,6-BISPHOSPHATASE, HYDROLASE
1rk3:A (TYR147) to (SER262) CRYSTAL STRUCTURE OF THE RAT VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH 1,25-DIHYDROXYVITAMIN D3 AND A SYNTHETIC PEPTIDE CONTAINING THE NR2 BOX OF DRIP 205 | NUCLEAR RECEPTOR-LIGAND COMPLEX, NUCLEAR RECEPTOR- COACTIVATOR INTERACTIONS, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
1rkg:A (TYR147) to (SER262) CRYSTAL STRUCTURE OF THE RAT VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH 2MBISP AND A SYNTHETIC PEPTIDE CONTAINING THE NR2 BOX OF DRIP 205 | NUCLEAR RECEPTOR-LIGAND COMPLEX, NUCLEAR RECEPTOR- COACTIVATOR INTERACTIONS, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
4yxd:C (PHE70) to (MET143) CRYSTAL STRUCTURE OF PORCINE HEART MITOCHONDRIAL COMPLEX II BOUND WITH FLUTOLANIL | OXIDOREDUCTASE, SUCCINATE DEHYDROGENASE, COMPLEX II, INHIBITOR, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
3umc:A (ARG16) to (GLY80) CRYSTAL STRUCTURE OF THE L-2-HALOACID DEHALOGENASE PA0810 | HALOACID DEHALOGENASE-LIKE HYDROLASE PROTEIN SUPERFAMILY, HYDROLASE
3umg:F (GLN62) to (LEU115) CRYSTAL STRUCTURE OF THE DEFLUORINATING L-2-HALOACID DEHALOGENASE RHA0230 | HALOACID DEHALOGENASE-LIKE HYDROLASE PROTEIN SUPERFAMILY, DEFLUORINASE, HYDROLASE
1fz3:B (ASP365) to (ASN412) METHANE MONOOXYGENASE HYDROXYLASE, FORM III SOAK AT PH 6.2 (0.1 M PIPES) | DINUCLEAR IRON CENTER, MONOOXYGENASE, OXIDOREDUCTASE
1fzh:B (ASP365) to (ASN412) METHANE MONOOXYGENASE HYDROXYLASE, FORM II PRESSURIZED WITH XENON GAS | DINUCLEAR IRON CENTER, MONOOXYGENASE, OXIDOREDUCTASE
2fbq:A (TYR134) to (ALA209) THE CRYSTAL STRUCTURE OF TRANSCRIPTIONAL REGULATOR PA3006 | PA3006, APC5893, TRANSCRIPTIONAL REGULATOR, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, TRANSCRIPTION
4kfe:B (THR117) to (LYS150) CRYSTAL STRUCTURE OF HANSENULA POLYMORPHA COPPER AMINE OXIDASE-1 REDUCED BY METHYLAMINE AT PH 7.0 | AMINE OXIDASE, OXIDOREDUCTASE, PEROXISOME
3utf:A (ASN109) to (PHE158) CRYSTAL STRUCTURE OF ASPERGILLUS FUMIGATUS UDP GALACTOPYRANOSE MUTASE IN REDUCED STATE | NUCLEOTIDE BINDING, MUTASE, FLAVIN ADENINE DINUCLEOTIDE BINDING, ISOMERASE
4z6y:B (PRO216) to (ASN265) STRUCTURE OF THE TBC1D7-TSC1 COMPLEX | COILED COIL, HETEROTETRAMER, HYDROLASE INHIBITOR-PROTEIN BINDING COMPLEX
4z6y:G (PRO216) to (ASN265) STRUCTURE OF THE TBC1D7-TSC1 COMPLEX | COILED COIL, HETEROTETRAMER, HYDROLASE INHIBITOR-PROTEIN BINDING COMPLEX
4z6y:E (PRO216) to (ASN265) STRUCTURE OF THE TBC1D7-TSC1 COMPLEX | COILED COIL, HETEROTETRAMER, HYDROLASE INHIBITOR-PROTEIN BINDING COMPLEX
4z6y:A (PRO216) to (ASN265) STRUCTURE OF THE TBC1D7-TSC1 COMPLEX | COILED COIL, HETEROTETRAMER, HYDROLASE INHIBITOR-PROTEIN BINDING COMPLEX
4kl1:B (GLU566) to (LEU611) HCN4 CNBD IN COMPLEX WITH CGMP | CNBD, CAMP, CGMP, C-DI-GMP, C-DI-AMP, ION CHANNEL, HCN, POTASSIUM/SODIUM HYPERPOLARIZATION-ACTIVATED CYCLIC NUCLEOTIDE-GATED CHANNEL, CAMP BINDING, CGMP BINDING, PROTEIN TRANSPORT
3uuo:A (ASN572) to (THR633) THE DISCOVERY OF POTENT, SELECTIVITY, AND ORALLY BIOAVAILABLE PYROZOLOQUINOLINES AS PDE10 INHIBITORS FOR THE TREATMENT OF SCHIZOPHRENIA | INHIBITOR COMPLEX, HYDROLASE, ZN BINDING, MG BINDING, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3uuo:B (SER571) to (THR633) THE DISCOVERY OF POTENT, SELECTIVITY, AND ORALLY BIOAVAILABLE PYROZOLOQUINOLINES AS PDE10 INHIBITORS FOR THE TREATMENT OF SCHIZOPHRENIA | INHIBITOR COMPLEX, HYDROLASE, ZN BINDING, MG BINDING, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1s0z:A (LEU224) to (SER266) CRYSTAL STRUCTURE OF THE VDR LBD COMPLEXED TO SEOCALCITOL. | NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, ALPHA-HELICAL SANDWICH, GENE REGULATION
3hqw:A (ASN562) to (THR623) DISCOVERY OF NOVEL INHIBITORS OF PDE10A | PHOSPHODIESTERASE 10A PDE10A PDE INHIBITORS, ALLOSTERIC ENZYME, ALTERNATIVE SPLICING, CAMP, CAMP-BINDING, CGMP, CGMP-BINDING, CYTOPLASM, HYDROLASE, MAGNESIUM, METAL- BINDING, NUCLEOTIDE-BINDING, ZINC, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
3hqy:A (ASN562) to (THR623) DISCOVERY OF NOVEL INHIBITORS OF PDE10A | PHOSPHODIESTERASE 10A PDE 10A PDE10 INHIBITORS, ALLOSTERIC ENZYME, ALTERNATIVE SPLICING, CAMP, CAMP-BINDING, CGMP, CGMP-BINDING, CYTOPLASM, HYDROLASE, MAGNESIUM, METAL- BINDING, NUCLEOTIDE-BINDING, ZINC, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
3hr1:A (ASN562) to (THR623) DISCOVERY OF NOVEL INHIBITORS OF PDE10A | PHOSPHODIESTERASE 10A, PDE 10A, PDE10 INHIBITORS, ALLOSTERIC ENZYME, ALTERNATIVE SPLICING, CAMP, CAMP-BINDING, CGMP, CGMP-BINDING, CYTOPLASM, HYDROLASE, MAGNESIUM, METAL- BINDING, NUCLEOTIDE-BINDING, ZINC, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
4kmw:A (GLY1) to (MET49) STRUCTURE OF THE Y34N MUTANT OF DEHALOPEROXIDASE-HEMOGLOBIN A FROM AMPHITRITE ORNATA WITH 2,4,6-TRICHLOROPHENOL | GLOBIN, OXYGEN STORAGE, PEROXIDASE, OXIDOREDUCTASE, OXIDOREDUCTASE- OXIDOREDUCTASE INHIBITOR COMPLEX
4kmw:B (GLY1) to (MET49) STRUCTURE OF THE Y34N MUTANT OF DEHALOPEROXIDASE-HEMOGLOBIN A FROM AMPHITRITE ORNATA WITH 2,4,6-TRICHLOROPHENOL | GLOBIN, OXYGEN STORAGE, PEROXIDASE, OXIDOREDUCTASE, OXIDOREDUCTASE- OXIDOREDUCTASE INHIBITOR COMPLEX
4kn3:A (GLY1) to (MET49) STRUCTURE OF THE Y34NS91G DOUBLE MUTANT OF DEHALOPEROXIDASE FROM AMPHITRITE ORNATA WITH 2,4,6-TRICHLOROPHENOL | GLOBIN, OXYGEN STORAGE, PEROXIDASE, OXIDOREDUCTASE, OXIDOREDUCTASE- OXIDOREDUCTASE INHIBITOR COMPLEX
4kn3:B (GLY1) to (MET49) STRUCTURE OF THE Y34NS91G DOUBLE MUTANT OF DEHALOPEROXIDASE FROM AMPHITRITE ORNATA WITH 2,4,6-TRICHLOROPHENOL | GLOBIN, OXYGEN STORAGE, PEROXIDASE, OXIDOREDUCTASE, OXIDOREDUCTASE- OXIDOREDUCTASE INHIBITOR COMPLEX
1gh0:Q (PRO4) to (ILE100) CRYSTAL STRUCTURE OF C-PHYCOCYANIN FROM SPIRULINA PLATENSIS | C-PHYCOCYANIN FROM SPIRULINA PLATENSIS, PHOTOSYNTHESIS
4kna:B (SER36) to (LYS105) CRYSTAL STRUCTURE OF AN N-SUCCINYLGLUTAMATE 5-SEMIALDEHYDE DEHYDROGENASE FROM BURKHOLDERIA THAILANDENSIS | NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, SSGCID, STRUCTURAL GENOMICS, NAD-DEPENDENT, N-SUCCINYL-L-GLUTAMATE, AMIDO ACID DEGRADATION, AST PATHWAY, ALDEHYDE DEHYDROGENASE, OXIDOREDUCTASE
3v49:A (PRO671) to (SER740) STRUCTURE OF AR LBD WITH ACTIVATOR PEPTIDE AND SARM INHIBITOR 1 | DIARYLHYDANTOIN, SYNTHESIS, SARM, ANTIANDROGEN, LIGAND BINDING DOMAIN, TESTOSTERONE, DIHYDROTESTOSTERONE, TRANSCRIPTION, SARM (SELECTIVE ANDROGEN RECEPTOR MODULATOR)
3v4a:A (PRO671) to (TRP741) STRUCTURE OF AR LBD WITH ACTIVATOR PEPTIDE AND SARM INHIBITOR 2 | DIARYLHYDANTOIN, SYNTHESIS, ANTIANDROGEN, ANDROGEN RECEPTOR, TESTOSTERONE, SELECTIVE ANDROGEN RECEPTOR MODULATOR, DIHYDROTESTOSTERONE, TRANSCRIPTION
3hzj:A (LEU710) to (ARG756) CRYSTAL STRUCTURE OF THE RABGAP DOMAIN OF THE RABGAP1L PROTEIN | STRUCTURAL GENOMICS CONSORTIUM, GTPASE ACTIVATING PROTEIN, SGC, ALTERNATIVE SPLICING, GTPASE ACTIVATION, PHOSPHOPROTEIN, POLYMORPHISM, HYDROLASE ACTIVATOR
3hzj:B (LEU710) to (ARG756) CRYSTAL STRUCTURE OF THE RABGAP DOMAIN OF THE RABGAP1L PROTEIN | STRUCTURAL GENOMICS CONSORTIUM, GTPASE ACTIVATING PROTEIN, SGC, ALTERNATIVE SPLICING, GTPASE ACTIVATION, PHOSPHOPROTEIN, POLYMORPHISM, HYDROLASE ACTIVATOR
3i2g:A (ASP198) to (PRO229) COCAINE ESTERASE WITH MUTATION G173Q, BOUND TO DTT ADDUCT | ALPHA/BETA HYDROLASE, HYDROLASE
3i2h:A (ASP198) to (PRO229) COCAINE ESTERASE WITH MUTATION L169K, BOUND TO DTT ADDUCT | ALPHA/BETA HYDROLASE, HYDROLASE
3i2k:A (ASP198) to (PRO229) COCAINE ESTERASE, WILD TYPE, BOUND TO A DTT ADDUCT | ALPHA/BETA HYDROLASE, HYDROLASE
3v94:A (THR417) to (THR480) TCRPDEC1 CATALYTIC DOMAIN IN COMPLEX WITH INHIBITOR WYQ16 | TRYPANOSOMA PDE PARASITE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3v94:B (THR417) to (THR480) TCRPDEC1 CATALYTIC DOMAIN IN COMPLEX WITH INHIBITOR WYQ16 | TRYPANOSOMA PDE PARASITE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3v94:C (THR417) to (THR480) TCRPDEC1 CATALYTIC DOMAIN IN COMPLEX WITH INHIBITOR WYQ16 | TRYPANOSOMA PDE PARASITE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3v94:D (THR417) to (THR480) TCRPDEC1 CATALYTIC DOMAIN IN COMPLEX WITH INHIBITOR WYQ16 | TRYPANOSOMA PDE PARASITE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3v94:E (THR417) to (THR480) TCRPDEC1 CATALYTIC DOMAIN IN COMPLEX WITH INHIBITOR WYQ16 | TRYPANOSOMA PDE PARASITE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3v94:F (THR417) to (ASP481) TCRPDEC1 CATALYTIC DOMAIN IN COMPLEX WITH INHIBITOR WYQ16 | TRYPANOSOMA PDE PARASITE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3v94:G (THR417) to (THR480) TCRPDEC1 CATALYTIC DOMAIN IN COMPLEX WITH INHIBITOR WYQ16 | TRYPANOSOMA PDE PARASITE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3v94:H (THR417) to (THR480) TCRPDEC1 CATALYTIC DOMAIN IN COMPLEX WITH INHIBITOR WYQ16 | TRYPANOSOMA PDE PARASITE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3v93:A (THR417) to (THR480) UNLIGANDED STRUCTURE OF TCRPDEC1 CATALYTIC DOMAIN | PARASITE, PHOSPHODIESTERASES,, HYDROLASE
3v93:B (THR417) to (THR480) UNLIGANDED STRUCTURE OF TCRPDEC1 CATALYTIC DOMAIN | PARASITE, PHOSPHODIESTERASES,, HYDROLASE
3v93:C (THR417) to (THR480) UNLIGANDED STRUCTURE OF TCRPDEC1 CATALYTIC DOMAIN | PARASITE, PHOSPHODIESTERASES,, HYDROLASE
3v93:D (THR417) to (THR480) UNLIGANDED STRUCTURE OF TCRPDEC1 CATALYTIC DOMAIN | PARASITE, PHOSPHODIESTERASES,, HYDROLASE
3v93:E (THR417) to (THR480) UNLIGANDED STRUCTURE OF TCRPDEC1 CATALYTIC DOMAIN | PARASITE, PHOSPHODIESTERASES,, HYDROLASE
3v93:G (THR417) to (THR480) UNLIGANDED STRUCTURE OF TCRPDEC1 CATALYTIC DOMAIN | PARASITE, PHOSPHODIESTERASES,, HYDROLASE
3v93:H (THR417) to (THR480) UNLIGANDED STRUCTURE OF TCRPDEC1 CATALYTIC DOMAIN | PARASITE, PHOSPHODIESTERASES,, HYDROLASE
4ksl:B (THR207) to (HIS276) GUMBY/FAM105B IN COMPLEX WITH LINEAR DI-UBIQUITIN | OTU DOMAIN, DEUBIQUITINASE, LINEAR DIUBIQUITIN, HYDROLASE
4ksl:E (ALA208) to (ARG274) GUMBY/FAM105B IN COMPLEX WITH LINEAR DI-UBIQUITIN | OTU DOMAIN, DEUBIQUITINASE, LINEAR DIUBIQUITIN, HYDROLASE
4ksl:I (ALA208) to (HIS276) GUMBY/FAM105B IN COMPLEX WITH LINEAR DI-UBIQUITIN | OTU DOMAIN, DEUBIQUITINASE, LINEAR DIUBIQUITIN, HYDROLASE
1gs4:A (PRO671) to (TYR739) STRUCTURAL BASIS FOR THE GLUCOCORTICOID RESPONSE IN A MUTANT HUMAN ANDROGEN RECEPTOR (ARCCR) DERIVED FROM AN ANDROGEN-INDEPENDENT PROSTATE CANCER | ANDROGEN RECEPTOR, HUMAN ANDROGEN RECEPTOR, LIGAND-BINDING DOMAIN, CORTISOL/ CORTISONE RESPONSE, PROSTATE CANCER
1so2:C (THR829) to (THR893) CATALYTIC DOMAIN OF HUMAN PHOSPHODIESTERASE 3B IN COMPLEX WITH A DIHYDROPYRIDAZINE INHIBITOR | PDE3B PHOSPHODIESTERASE, HYDROLASE
1sww:B (ARG46) to (ILE97) CRYSTAL STRUCTURE OF THE PHOSPHONOACETALDEHYDE HYDROLASE D12A MUTANT COMPLEXED WITH MAGNESIUM AND SUBSTRATE PHOSPHONOACETALDEHYDE | PHOPSHONOACETALDEHYDE HYDROLASE, PHOSPHONATASE, HAD ENZYM SUPERFAMILY, METAL BINDING
4kyn:A (ARG74) to (GLN147) CRYSTAL STRUCTURE OF ODORANT BINDING PROTEIN 48 FROM ANOPHELES GAMBIAE AT 3.3 ANGSTROM RESOLUTION | INSECT ODORANT BINDING PROTEIN, OBP48, OLFACTION, ANOPHELES GAMBIAE, TRANSPORT PROTEIN
4kyn:C (ARG74) to (ALA146) CRYSTAL STRUCTURE OF ODORANT BINDING PROTEIN 48 FROM ANOPHELES GAMBIAE AT 3.3 ANGSTROM RESOLUTION | INSECT ODORANT BINDING PROTEIN, OBP48, OLFACTION, ANOPHELES GAMBIAE, TRANSPORT PROTEIN
4kyn:D (ARG74) to (ALA146) CRYSTAL STRUCTURE OF ODORANT BINDING PROTEIN 48 FROM ANOPHELES GAMBIAE AT 3.3 ANGSTROM RESOLUTION | INSECT ODORANT BINDING PROTEIN, OBP48, OLFACTION, ANOPHELES GAMBIAE, TRANSPORT PROTEIN
1t1f:A (LEU81) to (ILE119) CRYSTAL STRUCTURE OF NATIVE ANTITHROMBIN IN ITS MONOMERIC FORM | SERINE-CYSTEINE PROTEINASE INHIBITOR; THROMBIN; HUMAN; X-RAY CRYSTALLOGRAPHY, BLOOD CLOTTING
1t1f:B (LEU81) to (ILE119) CRYSTAL STRUCTURE OF NATIVE ANTITHROMBIN IN ITS MONOMERIC FORM | SERINE-CYSTEINE PROTEINASE INHIBITOR; THROMBIN; HUMAN; X-RAY CRYSTALLOGRAPHY, BLOOD CLOTTING
1t1f:C (LEU81) to (ILE119) CRYSTAL STRUCTURE OF NATIVE ANTITHROMBIN IN ITS MONOMERIC FORM | SERINE-CYSTEINE PROTEINASE INHIBITOR; THROMBIN; HUMAN; X-RAY CRYSTALLOGRAPHY, BLOOD CLOTTING
3vjs:A (TYR147) to (SER262) VITAMIN D RECEPTOR COMPLEX WITH A CARBORANE COMPOUND | NUCLEAR RECEPTOR, SYNTHETIC AGONIST, CARBORANE, TRANSCRIPTION
1t6h:A (THR115) to (THR152) CRYSTAL STRUCTURE T4 LYSOZYME INCORPORATING AN UNNATURAL AMINO ACID P-IODO-L-PHENYLALANINE AT POSITION 153 | IODOPHE, SAD PHASING, UNNATURAL AMINO ACID, HYDROLASE
4zo5:A (SER561) to (THR623) PDE10 COMPLEXED WITH 4-ISOPROPOXY-2-(2-(3-(4-METHOXYPHENYL)-4-OXO-3,4- DIHYDROQUINAZOLIN-2-YL)ETHYL)ISOINDOLINE-1,3-DIONE | PHOSPHODIESTERASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4zo5:B (SER561) to (THR623) PDE10 COMPLEXED WITH 4-ISOPROPOXY-2-(2-(3-(4-METHOXYPHENYL)-4-OXO-3,4- DIHYDROQUINAZOLIN-2-YL)ETHYL)ISOINDOLINE-1,3-DIONE | PHOSPHODIESTERASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1t73:A (SER696) to (TYR739) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH A FXXFF MOTIF | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING DOMAIN, AF-2, ANDROGEN, TESTOSTERONE, DHT, ALPHA-HELICAL SANDWICH, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
1t74:A (SER696) to (TYR739) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH A WXXLF MOTIF | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING DOMAIN, AF-2, ANDROGEN, TESTOSTERONE, DHT, ALPHA-HELICAL SANDWICH, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
1t79:A (SER696) to (TYR739) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH A FXXLW MOTIF | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING DOMAIN, AF-2, ANDROGEN, TESTOSTERONE, DHT, ALPHA-HELICAL SANDWICH, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
2gr9:C (ARG199) to (GLU275) CRYSTAL STRUCTURE OF P5CR COMPLEXED WITH NADH | CRYSTAL STRUCUTRE, HUMAN PYRROLINE-5-CARBOXYLATE REDUCTASE, NADH, OXIDOREDUCTASE
2w3r:B (PHE344) to (ASN441) CRYSTAL STRUCTURE OF XANTHINE DEHYDROGENASE (DESULFO FORM) FROM RHODOBACTER CAPSULATUS IN COMPLEX WITH HYPOXANTHINE | XDH, GOUT, IRON, XANTHINE, IRON-SULFUR, MOLYBDENUM COFACTOR, HYPOXANTHINE, METAL-BINDING, OXIDOREDUCTASE
2w3r:D (PHE344) to (ASN441) CRYSTAL STRUCTURE OF XANTHINE DEHYDROGENASE (DESULFO FORM) FROM RHODOBACTER CAPSULATUS IN COMPLEX WITH HYPOXANTHINE | XDH, GOUT, IRON, XANTHINE, IRON-SULFUR, MOLYBDENUM COFACTOR, HYPOXANTHINE, METAL-BINDING, OXIDOREDUCTASE
2w3r:H (GLY345) to (ASN441) CRYSTAL STRUCTURE OF XANTHINE DEHYDROGENASE (DESULFO FORM) FROM RHODOBACTER CAPSULATUS IN COMPLEX WITH HYPOXANTHINE | XDH, GOUT, IRON, XANTHINE, IRON-SULFUR, MOLYBDENUM COFACTOR, HYPOXANTHINE, METAL-BINDING, OXIDOREDUCTASE
1t90:D (LYS43) to (ALA116) CRYSTAL STRUCTURE OF METHYLMALONATE SEMIALDEHYDE DEHYDROGENASE FROM BACILLUS SUBTILIS | OXIDOREDUCTASE, NAD
3vkg:B (LEU3913) to (LYS3977) X-RAY STRUCTURE OF AN MTBD TRUNCATION MUTANT OF DYNEIN MOTOR DOMAIN | AAA+ PROTEIN, MOLECULAR MOTOR, MICROTUBLES, MOTOR PROTEIN
2w55:D (GLY345) to (ASN441) CRYSTAL STRUCTURE OF XANTHINE DEHYDROGENASE (E232Q VARIANT) FROM RHODOBACTER CAPSULATUS IN COMPLEX WITH HYPOXANTHINE | XDH, GOUT, IRON, XANTHINE, IRON-SULFUR, MOLYBDENUM COFACTOR, HYPOXANTHINE, METAL-BINDING, OXIDOREDUCTASE
2w55:F (GLY346) to (ASN441) CRYSTAL STRUCTURE OF XANTHINE DEHYDROGENASE (E232Q VARIANT) FROM RHODOBACTER CAPSULATUS IN COMPLEX WITH HYPOXANTHINE | XDH, GOUT, IRON, XANTHINE, IRON-SULFUR, MOLYBDENUM COFACTOR, HYPOXANTHINE, METAL-BINDING, OXIDOREDUCTASE
2w55:H (GLY345) to (ASN441) CRYSTAL STRUCTURE OF XANTHINE DEHYDROGENASE (E232Q VARIANT) FROM RHODOBACTER CAPSULATUS IN COMPLEX WITH HYPOXANTHINE | XDH, GOUT, IRON, XANTHINE, IRON-SULFUR, MOLYBDENUM COFACTOR, HYPOXANTHINE, METAL-BINDING, OXIDOREDUCTASE
2h12:B (HIS122) to (ALA174) STRUCTURE OF ACETOBACTER ACETI CITRATE SYNTHASE COMPLEXED WITH OXALOACETATE AND CARBOXYMETHYLDETHIA COENZYME A (CMX) | ACIDOPHILE, CITRATE SYNTHASE, ACETIC ACID RESISTANCE, ALLOSTERY, TRANSFERASE
4zul:B (SER56) to (SER133) STRUCTURE ALDH7A1 COMPLEXED WITH ALPHA-AMINOADIPATE | ALDEHYDE DEHYDROGENASE, NAD, OXIDOREDUCTASE, LYSINE CATABOLISM
4zul:C (SER56) to (SER133) STRUCTURE ALDH7A1 COMPLEXED WITH ALPHA-AMINOADIPATE | ALDEHYDE DEHYDROGENASE, NAD, OXIDOREDUCTASE, LYSINE CATABOLISM
4zul:G (SER56) to (SER133) STRUCTURE ALDH7A1 COMPLEXED WITH ALPHA-AMINOADIPATE | ALDEHYDE DEHYDROGENASE, NAD, OXIDOREDUCTASE, LYSINE CATABOLISM
2h1j:A (GLU357) to (ASN437) 3.1 A X-RAY STRUCTURE OF PUTATIVE OLIGOENDOPEPTIDASE F: CRYSTALS GROWN BY MICROFLUIDIC SEEDING | STRUCTURAL GENOMICS, MICROFLUIDIC SEEDING, PSI-2, PROTEIN STRUCTURE INITIATIVE, ACCELERATED TECHNOLOGIES CENTER FOR GENE TO 3D STRUCTURE, ATCG3D, HYDROLASE
2h1j:B (GLU357) to (ASN437) 3.1 A X-RAY STRUCTURE OF PUTATIVE OLIGOENDOPEPTIDASE F: CRYSTALS GROWN BY MICROFLUIDIC SEEDING | STRUCTURAL GENOMICS, MICROFLUIDIC SEEDING, PSI-2, PROTEIN STRUCTURE INITIATIVE, ACCELERATED TECHNOLOGIES CENTER FOR GENE TO 3D STRUCTURE, ATCG3D, HYDROLASE
4zv5:A (GLY8) to (PRO77) CRYSTAL STRUCTURE OF N-MYRISTOYLATED MOUSE MAMMARY TUMOR VIRUS MATRIX PROTEIN | RETROVIRAL MATRIX PROTEIN, N-MYRISTOYLATION, VIRAL PROTEIN
2w8n:A (VAL95) to (VAL174) THE CRYSTAL STRUCTURE OF THE OXIDIZED FORM OF HUMAN SSADH | MITOCHONDRION, OXIDOREDUCTASE, TRANSIT PEPTIDE, DISEASE MUTATION, SSA, NAD, POLYMORPHISM, MITOCHONDRIA
4zvw:B (SER56) to (MET135) STRUCTURE OF APO HUMAN ALDH7A1 IN SPACE GROUP C2 | ALDEHYDE DEHYDROGENASE, NAD, OXIDOREDUCTASE, LYSINE CATABOLISM
3irh:A (TYR117) to (LYS165) STRUCTURE OF AN ENTEROCOCCUS FAECALIS HD-DOMAIN PROTEIN COMPLEXED WITH DGTP AND DATP | HD DOMAIN, PHOSPHOHYDROLASE, DNTPASE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, UNKNOWN FUNCTION, HYDROLASE
4zw9:A (LEU355) to (GLY428) CRYSTAL STRUCTURE OF HUMAN GLUT3 BOUND TO D-GLUCOSE IN THE OUTWARD- OCCLUDED CONFORMATION AT 1.5 ANGSTROM | TRANSPORTER, TRANSPORT PROTEIN
4zwe:C (MET216) to (ILE272) CRYSTAL STRUCTURE OF THE DGTP-BOUND CATALYTIC CORE OF SAMHD1 T592V MUTANT | PHOSPHORYLATION, TETRAMER STABILITY, DNTPASE, HIV-1 RESTRICTION, HYDROLASE
4zwe:D (MET216) to (ILE272) CRYSTAL STRUCTURE OF THE DGTP-BOUND CATALYTIC CORE OF SAMHD1 T592V MUTANT | PHOSPHORYLATION, TETRAMER STABILITY, DNTPASE, HIV-1 RESTRICTION, HYDROLASE
4zwg:C (PHE213) to (ILE272) CRYSTAL STRUCTURE OF THE GTP-DATP-BOUND CATALYTIC CORE OF SAMHD1 PHOSPHOMIMETIC T592E MUTANT | PHOSPHORYLATION, TETRAMER STABILITY, DNTPASE, HIV-1 RESTRICTION, HYDROLASE
1tox:A (GLY224) to (VAL288) DIPHTHERIA TOXIN DIMER COMPLEXED WITH NAD | TOXIN, ADP-RIBOSYLATION, GLUCOSYLTRANSFERASE, TRANSFERASE, NAD
3vm9:A (SER3) to (SER58) DIMERIC HORSE MYOGLOBIN | MYOGLOBIN, OXYGEN STORAGE, OXYGEN BINDING, OXYGEN TRANSPORT
2hek:A (THR94) to (GLY140) CRYSTAL STRUCTURE OF O67745, A HYPOTHETICAL PROTEIN FROM AQUIFEX AEOLICUS AT 2.0 A RESOLUTION. | PREDOMINANTLY ALPHA HELICAL PROTEIN WITH GDP BINDING SITE AND ACTIVE SITE BEING FAR FROM EACH OTHER, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, BERKELEY STRUCTURAL GENOMICS CENTER, BSGC, UNKNOWN FUNCTION
4lkq:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT017 | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2wey:A (SER571) to (THR633) HUMAN PDE-PAPAVERINE COMPLEX OBTAINED BY LIGAND SOAKING OF CROSS-LINKED PROTEIN CRYSTALS | METAL-BINDING, CROSS-LINKING, PHOSPHOPROTEIN, PHOSPHODIESTERASE, ALLOSTERIC ENZYME, CGMP, CAMP, ZINC, HYDROLASE, CYTOPLASM, MAGNESIUM, PAPAVERINE, POLYMORPHISM, CGMP-BINDING, CAMP-BINDING, NUCLEOTIDE-BINDING, ALTERNATIVE SPLICING
2wey:B (SER571) to (THR633) HUMAN PDE-PAPAVERINE COMPLEX OBTAINED BY LIGAND SOAKING OF CROSS-LINKED PROTEIN CRYSTALS | METAL-BINDING, CROSS-LINKING, PHOSPHOPROTEIN, PHOSPHODIESTERASE, ALLOSTERIC ENZYME, CGMP, CAMP, ZINC, HYDROLASE, CYTOPLASM, MAGNESIUM, PAPAVERINE, POLYMORPHISM, CGMP-BINDING, CAMP-BINDING, NUCLEOTIDE-BINDING, ALTERNATIVE SPLICING
3ixp:D (THR291) to (ALA374) CRYSTAL STRUCTURE OF THE ECDYSONE RECEPTOR BOUND TO BYI08346 | ANTI-PARALLEL ALPHA-HELICES, TRANSCRIPTION, TRANSCRIPTION REGULATION
2hhb:B (THR4) to (ASN57) THE CRYSTAL STRUCTURE OF HUMAN DEOXYHAEMOGLOBIN AT 1.74 ANGSTROMS RESOLUTION | OXYGEN TRANSPORT
4llp:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT401 | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4lm1:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT450 | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4lm1:B (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT450 | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4lm4:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT902 | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3vru:A (TYR147) to (ALA263) VDR LIGAND BINDING DOMAIN IN COMPLEX WITH 2-METHYLIDENE-19,24-DINOR- 1ALPHA,25-DIHYDROXY VITAMIND3 | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION, VITAMIN D3, VDRE, RXR, CO- FACTORS, NUCLEAR
3vrv:A (TYR147) to (ALA263) VDR LIGAND BINDING DOMAIN IN COMPLEX WITH 2-METHYLIDENE-26,27- DIMETHYL-19,24-DINOR-1ALPHA,25-DIHYDROXYVITAMIN D3 | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION, VITAMIN D3, VDRE, RXR, CO- FACTORS, NUCLEAR
3vrw:A (TYR147) to (ALA263) VDR LIGAND BINDING DOMAIN IN COMPLEX WITH 22S-BUTYL-2-METHYLIDENE-26, 27-DIMETHYL-19,24-DINOR-1ALPHA,25-DIHYDROXYVITAMIN D3 | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION, VITAMIN D3, VDRE, RXR, CO- FACTORS, NUCLEAR
3vt3:A (TYR147) to (ALA263) CRYSTAL STRUCTURES OF RAT VDR-LBD WITH R270L MUTATION | TRANSCRIPTION, HORMONE RECEPTOR
3vt4:A (TYR147) to (ALA263) CRYSTAL STRUCTURES OF RAT VDR-LBD WITH R270L MUTATION | TRANSCRIPTION, HORMONE RECEPTOR
3vt7:A (TYR147) to (ALA263) CRYSTAL STRUCTURES OF RAT VDR-LBD WITH W282R MUTATION | TRANSCRIPTION, HORMONE RECEPTOR
3vvl:B (PRO180) to (PHE272) CRYSTAL STRUCTURE OF L-SERINE-O-ACETYLTRANSFERASE FOUND IN D- CYCLOSERINE BIOSYNTHETIC PATHWAY | D-CYCLOSERINE, ALPHA/BETA HYDROLASE DOMAIN, L-SERINE-O- ACETYLTRANSFERASE, TRANSFERASE
3vvm:B (PRO180) to (PHE272) CRYSTAL STRUCTURE OF G52A-P55G MUTANT OF L-SERINE-O-ACETYLTRANSFERASE FOUND IN D-CYCLOSERINE BIOSYNTHETIC PATHWAY | D-CYCLOSERINE, ALPHA/BETA HYDROLASE DOMAIN, L-SERINE-O- ACETYLTRANSFERASE, TRANSFERASE
1i38:A (ILE672) to (TYR739) CRYSTAL STRUCTURE OF THE RAT ANDROGEN RECEPTOR LIGAND BINDING DOMAIN T877A MUTANT COMPLEX WITH DIHYDROTESTOSTERONE | ANDROGEN RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, LIGAND-BINDING DOMAIN, HORMONE/GROWTH FACTOR COMPLEX
3w0j:A (TYR147) to (ALA263) CRYSTAL STRUCTURE OF RAT VDR LIGAND BINDING DOMAIN IN COMPLEX WITH NOVEL NONSECOSTEROIDAL LIGANDS | GENE REGULATION, TRANSCRIPTION
4lxl:A (PRO213) to (LYS242) CRYSTAL STRUCTURE OF JMJD2B COMPLEXED WITH PYRIDINE-2,4-DICARBOXYLIC ACID AND H3K9ME3 | JMJC DOMAIN, DEMETHYLATION, HISTONE, METHYLATION, NUCLEUS, OXIDOREDUCTASE-PEPTIDE COMPLEX
2i15:A (GLN50) to (GLY124) CRYSTAL STRUCTURE OF MPN423 FROM MYCOPLASMA PNEUMONIAE | STRUCTURAL GENOMICS, MPN423, HYPOTHETICAL PROTIEN, CRYSTAL STRUCTURE, ALL ALPHA STRUCTURE, PSI, PROTEIN STRUCTURE INITIATIVE, BERKELEY STRUCTURAL GENOMICS CENTER, BSGC, UNKNOWN FUNCTION
3izx:A (PRO84) to (GLY158) 3.1 ANGSTROM CRYOEM STRUCTURE OF CYTOPLASMIC POLYHEDROSIS VIRUS | CYTOPLASMIC POLYHEDROSIS VIRUS, 3D RECONSTRUCTION, CRYOEM, FULL ATOM MODEL, VIRUS
3w5q:A (TYR147) to (ALA263) CRYSTAL STRUCTURE OF COMPLEXES OF VITAMIN D RECEPTOR LIGAND BINDING DOMAIN WITH LITHOCHOLIC ACID DERIVATIVES | ZINC-FINGER, NUCLEAR RECEPTOR-AGONIST COMPLEX, TRANSCRIPTION, RECEPTOR, TRANSCRIPTION REGULATION, ACTIVATOR, DNA-BINDING, METAL- BINDING, PHOSPHOPROTEIN, NUCLEUS
3w5t:A (TYR147) to (ALA263) CRYSTAL STRUCTURE OF COMPLEXES OF VITAMIN D RECEPTOR LIGAND BINDING DOMAIN WITH LITHOCHOLIC ACID DERIVATIVES | ZINC-FINGER, NUCLEAR RECEPTOR-AGONIST COMPLEX, TRANSCRIPTION, RECEPTOR, TRANSCRIPTION REGULATION, ACTIVATOR, DNA-BINDING, METAL- BINDING, PHOSPHOPROTEIN, NUCLEUS
2ibp:B (PRO95) to (ALA156) CRYSTAL STRUCTURE OF CITRATE SYNTHASE FROM PYROBACULUM AEROPHILUM | DISULFIDE BOND, HOMODIMER, CITRATE SYNTHASE, THERMOPHILIC, CATENANE, TRANSFERASE
2id2:A (THR39) to (MET118) GAPN T244S MUTANT X-RAY STRUCTURE AT 2.5 A | ALDH, T244, ACYLATION STEP, HYDRIDE TRANSFER, CONFORMATION OF NICOTINAMIDE, OXIDOREDUCTASE
2id2:B (THR39) to (MET118) GAPN T244S MUTANT X-RAY STRUCTURE AT 2.5 A | ALDH, T244, ACYLATION STEP, HYDRIDE TRANSFER, CONFORMATION OF NICOTINAMIDE, OXIDOREDUCTASE
2id2:D (THR39) to (MET118) GAPN T244S MUTANT X-RAY STRUCTURE AT 2.5 A | ALDH, T244, ACYLATION STEP, HYDRIDE TRANSFER, CONFORMATION OF NICOTINAMIDE, OXIDOREDUCTASE
3wdc:A (THR81) to (GLU147) N-TERMINAL DOMAIN OF MYCOBACTERIUM TUBERCULOSIS CLPC1 BOUND TO CYCLOMARIN A | CHAPERONE, CHAPERONE-ANTIMICROBIAL PROTEIN COMPLEX
3wde:A (THR81) to (GLU147) MUTANT N-TERMINAL DOMAIN OF MYCOBACTERIUM TUBERCULOSIS CLPC1, F80Y, BOUND TO CYCLOMARIN A | CHAPERONE, CHAPERONE-ANTIMICROBIAL PROTEIN COMPLEX
2ihq:A (PRO671) to (TRP741) CRYSTAL STRUCTURE OF THE RAT ANDROGEN RECEPTOR LIGAND BINDING DOMIAN COMPLEX WITH AN N-ARYL- HYDROXYBICYCLOHYDANTOIN | ANDROGEN RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, LIGAND-BINDING DOMAIN, HORMONE/GROWTH FACTOR COMPLEX
5agc:A (HIS11) to (ILE83) CRYSTALLOGRAPHIC FORMS OF THE VPS75 TETRAMER | TRANSPORT PROTEIN, VPS75, VACUOLAR PROTEIN SORTING 75, HISTONE CHAPERONE, NAP1, CHROMATIN
5agc:B (GLU6) to (ILE83) CRYSTALLOGRAPHIC FORMS OF THE VPS75 TETRAMER | TRANSPORT PROTEIN, VPS75, VACUOLAR PROTEIN SORTING 75, HISTONE CHAPERONE, NAP1, CHROMATIN
5agc:C (GLU10) to (ILE83) CRYSTALLOGRAPHIC FORMS OF THE VPS75 TETRAMER | TRANSPORT PROTEIN, VPS75, VACUOLAR PROTEIN SORTING 75, HISTONE CHAPERONE, NAP1, CHROMATIN
5agc:D (GLU10) to (ILE83) CRYSTALLOGRAPHIC FORMS OF THE VPS75 TETRAMER | TRANSPORT PROTEIN, VPS75, VACUOLAR PROTEIN SORTING 75, HISTONE CHAPERONE, NAP1, CHROMATIN
1uzf:A (ASN374) to (GLY474) COMPLEX OF THE ANTI-HYPERTENSIVE DRUG CAPTOPRIL AN THE HUMAN TESTICULAR ANGIOTENSIN I-CONVERTING ENZYME | METALLOPROTEASE, HYDROLASE, INHIBITOR, CAPTOPRIL, ZINC DEPENDANT PEPTIDASE, ANTI-HYPERTENSIVE DRUG
2iul:A (ASN374) to (GLY474) HUMAN TACE G13 MUTANT | HYDROLASE, PHOSPHORYLATION, CARBOXYPEPTIDASE, METAL-BINDING, TRANSMEMBRANE, METALLOPROTEASE, PEPTIDYL DIPEPTIDASE, ALTERNATIVE SPLICING, TYPE-I MEMBRANE-ANCHORED PROTEIN, GLYCOSIDASE, POLYMORPHISM, GLYCOPROTEIN, AC, ZINC, MUTANT, MEMBRANE, CHLORIDE, PROTEASE
2x8z:A (THR358) to (LEU436) CRYSTAL STRUCTURE OF ANCE-CAPTOPRIL COMPLEX | HYDROLASE, ACE INHIBITOR, ZINC METALLOPEPTIDASE
2x8y:A (THR358) to (LEU436) CRYSTAL STRUCTURE OF ANCE | HYDROLASE, ACE INHIBITOR, ZINC METALLOPEPTIDASE
2iux:A (ASN374) to (GLY474) HUMAN TACE MUTANT G1234 | GLYCOSIDASE, POLYMORPHISM, GLYCOPROTEIN, METAL-BINDING, ALTERNATIVE SPLICING, METALLOPROTEASE, PHOSPHORYLATION, AC, ZINC, MEMBRANE, CHLORIDE, PROTEASE, HYDROLASE, TYPE-I MEMBRANE-ANCHORED PROTEIN, CARBOXYPEPTIDASE, PEPTIDYL DIPEPTIDASE, TRANSMEMBRANE
3woj:A (GLN430) to (ALA496) CRYSTAL STRUCTURE OF THE DAP BII | CHYMOTRYPSIN FOLD, S46 PEPTIDASE, HYDROLASE
3wok:A (GLN430) to (ALA496) CRYSTAL STRUCTURE OF THE DAP BII (SPACE) | CHYMOTRYPSIN FOLD, S46 PEPTIDASE, HYDROLASE
3wok:B (GLN430) to (ALA496) CRYSTAL STRUCTURE OF THE DAP BII (SPACE) | CHYMOTRYPSIN FOLD, S46 PEPTIDASE, HYDROLASE
3wom:A (GLN430) to (ALA496) CRYSTAL STRUCTURE OF THE DAP BII DIPEPTIDE COMPLEX II | CHYMOTRYPSIN FOLD, HYDROLASE
3wom:B (GLN430) to (ALA496) CRYSTAL STRUCTURE OF THE DAP BII DIPEPTIDE COMPLEX II | CHYMOTRYPSIN FOLD, HYDROLASE
3woo:B (GLN430) to (ALA496) CRYSTAL STRUCTURE OF THE DAP BII HEXAPEPTIDE COMPLEX I | CHYMOTRYPSIN FOLD, S46 PEPTIDASE, HYDROLASE-HORMONE COMPLEX
3wop:B (GLN430) to (ALA496) CRYSTAL STRUCTURE OF THE DAP BII HEXAPEPTIDE COMPLEX II | CHYMOTRYPSIN FOLD, S46 PEPTIDASE, HYDROLASE-HORMONE COMPLEX
3woq:B (GLN430) to (ALA496) CRYSTAL STRUCTURE OF THE DAP BII HEXAPEPTIDE COMPLEX III | CHYMOTRYPSIN FOLD, S46 PEPTIDASE, HYDROLASE-HORMONE COMPLEX
3wor:A (GLN430) to (ALA496) CRYSTAL STRUCTURE OF THE DAP BII OCTAPEPTIDE COMPLEX | CHYMOTRYPSIN FOLD, S46 PEPTIDASE, HYDROLASE-HORMONE COMPLEX
5ao0:B (MET216) to (GLY274) CRYSTAL STRUCTURE OF HUMAN SAMHD1 (AMINO ACID RESIDUES 41-583) BOUND TO DDGTP | HYDROLASE, DEOXYNUCLEOSIDE, DEOXYNUCLEOSIDE TRIPHOSPHATE TRIPHOSPHOHYDROLASE, HIV RESTRICTION FACTOR
2xdr:C (SER42) to (LEU119) CRYSTALLOGRAPHIC STRUCTURE OF BETAINE ALDEHYDE DEHYDROGENASE MUTANT E252A FROM PSEUDOMONAS AERUGINOSA | ALDEHYDE OXIDATION, NADPH COMPLEX, OXIDOREDUCTASE
1vhd:A (LEU254) to (GLY312) CRYSTAL STRUCTURE OF AN IRON CONTAINING ALCOHOL DEHYDROGENASE | STRUCTURAL GENOMICS, OXIDOREDUCTASE
1vhd:B (LEU254) to (GLY312) CRYSTAL STRUCTURE OF AN IRON CONTAINING ALCOHOL DEHYDROGENASE | STRUCTURAL GENOMICS, OXIDOREDUCTASE
3ws9:B (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A IN COMPLEX WITH A BENZIMDAZOLE INHIBITOR | PHOSPHODIESTERASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3ws9:B (GLN659) to (VAL722) CRYSTAL STRUCTURE OF PDE10A IN COMPLEX WITH A BENZIMDAZOLE INHIBITOR | PHOSPHODIESTERASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4mrw:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT0120 (7-CHLOROQUINOLIN-4- OL) | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4mrw:B (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT0120 (7-CHLOROQUINOLIN-4- OL) | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3ws8:B (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A IN COMPLEX WITH A BENZIMIDAZOLE INHIBITOR | PHOSPHODIESTERASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4mrz:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT0429 (4-METHYL-3- NITROPYRIDIN-2-AMINE) | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4ms0:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT0443 (6-CHLOROPYRIMIDINE- 2,4-DIAMINE) | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4ms0:B (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT0443 (6-CHLOROPYRIMIDINE- 2,4-DIAMINE) | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4msa:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT0449 (5-NITRO-1H- BENZIMIDAZOLE) | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4mse:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT1597 (2-({[(2S)-2-METHYL- 2,3-DIHYDRO-1,3-BENZOTHIAZOL-5-YL]OXY}METHYL)QUINOLINE) | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4msh:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT0143 ((2S)-4-CHLORO-2,3- DIHYDRO-1,3-BENZOTHIAZOL-2-AMINE) | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4msh:B (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT0143 ((2S)-4-CHLORO-2,3- DIHYDRO-1,3-BENZOTHIAZOL-2-AMINE) | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1vlj:A (TRP265) to (GLY338) CRYSTAL STRUCTURE OF NADH-DEPENDENT BUTANOL DEHYDROGENASE A (TM0820) FROM THERMOTOGA MARITIMA AT 1.78 A RESOLUTION | TM0820, NADH-DEPENDENT BUTANOL DEHYDROGENASE A, STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI, JOINT CENTER FOR STRUCTURAL GENOMICS, OXIDOREDUCTASE
1vlj:B (TRP265) to (GLY338) CRYSTAL STRUCTURE OF NADH-DEPENDENT BUTANOL DEHYDROGENASE A (TM0820) FROM THERMOTOGA MARITIMA AT 1.78 A RESOLUTION | TM0820, NADH-DEPENDENT BUTANOL DEHYDROGENASE A, STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI, JOINT CENTER FOR STRUCTURAL GENOMICS, OXIDOREDUCTASE
4muw:A (ASN562) to (THR623) CRYSTAL STRUCTURE OF PDE10A WITH NOVEL KETO-BENZIMIDAZOLE INHIBITOR | PDE10A, PHOSPHODIESTERASE 10A, INHIBITORS, KETO-BENZIMIDAZOLES, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4muw:B (ASN562) to (THR623) CRYSTAL STRUCTURE OF PDE10A WITH NOVEL KETO-BENZIMIDAZOLE INHIBITOR | PDE10A, PHOSPHODIESTERASE 10A, INHIBITORS, KETO-BENZIMIDAZOLES, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4mvh:A (ASN562) to (THR623) CRYSTAL STRUCTURE OF PDE10A WITH NOVEL KETO-BENZIMIDAZOLE INHIBITOR | PDE10A, PHOSPHODIESTERASE 10A, INHIBITORS, KETO-BENZIMIDAZOLES, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4mvh:B (SER561) to (THR623) CRYSTAL STRUCTURE OF PDE10A WITH NOVEL KETO-BENZIMIDAZOLE INHIBITOR | PDE10A, PHOSPHODIESTERASE 10A, INHIBITORS, KETO-BENZIMIDAZOLES, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1vqq:A (LYS28) to (LEU73) STRUCTURE OF PENICILLIN BINDING PROTEIN 2A FROM METHICILLIN RESISTANT STAPHYLOCOCCUS AUREUS STRAIN 27R AT 1.80 A RESOLUTION. | PENICILLIN BINDING PROTEIN, BETA-LACTAM, D, D- TRANSPEPTIDASE, D-CARBOXYPEPTIDASE, BIOSYNTHETIC PROTEIN
1vqq:B (LYS28) to (LEU73) STRUCTURE OF PENICILLIN BINDING PROTEIN 2A FROM METHICILLIN RESISTANT STAPHYLOCOCCUS AUREUS STRAIN 27R AT 1.80 A RESOLUTION. | PENICILLIN BINDING PROTEIN, BETA-LACTAM, D, D- TRANSPEPTIDASE, D-CARBOXYPEPTIDASE, BIOSYNTHETIC PROTEIN
5awf:A (GLY441) to (HIS492) CRYSTAL STRUCTURE OF SUFB-SUFC-SUFD COMPLEX FROM ESCHERICHIA COLI | IRON-SULFUR CLUSTERS, IRON-SULFUR PROTEINS, ABC PROTEINS, ABC ATPASE, TRANSPORT PROTEIN-PROTEIN BINDING COMPLEX
5awf:E (GLY441) to (GLY495) CRYSTAL STRUCTURE OF SUFB-SUFC-SUFD COMPLEX FROM ESCHERICHIA COLI | IRON-SULFUR CLUSTERS, IRON-SULFUR PROTEINS, ABC PROTEINS, ABC ATPASE, TRANSPORT PROTEIN-PROTEIN BINDING COMPLEX
1vr0:A (THR176) to (LYS219) CRYSTAL STRUCTURE OF PUTATIVE 2-PHOSPHOSULFOLACTATE PHOSPHATASE (15026306) FROM CLOSTRIDIUM ACETOBUTYLICUM AT 2.6 A RESOLUTION | 15026306, PUTATIVE 2-PHOSPHOSULFOLACTATE PHOSPHATASE, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI, HYDROLASE
1vr0:B (THR176) to (LYS219) CRYSTAL STRUCTURE OF PUTATIVE 2-PHOSPHOSULFOLACTATE PHOSPHATASE (15026306) FROM CLOSTRIDIUM ACETOBUTYLICUM AT 2.6 A RESOLUTION | 15026306, PUTATIVE 2-PHOSPHOSULFOLACTATE PHOSPHATASE, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI, HYDROLASE
1vr0:C (THR176) to (LYS219) CRYSTAL STRUCTURE OF PUTATIVE 2-PHOSPHOSULFOLACTATE PHOSPHATASE (15026306) FROM CLOSTRIDIUM ACETOBUTYLICUM AT 2.6 A RESOLUTION | 15026306, PUTATIVE 2-PHOSPHOSULFOLACTATE PHOSPHATASE, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI, HYDROLASE
5awg:A (GLY441) to (HIS492) CRYSTAL STRUCTURE OF HG-BOUND SUFB-SUFC-SUFD COMPLEX FROM ESCHERICHIA COLI | IRON-SULFUR CLUSTERS, IRON-SULFUR PROTEINS, ABC PROTEINS, ABC ATPASE, TRANSPORT PROTEIN-PROTEIN BINDING COMPLEX
5awg:E (GLY441) to (GLU491) CRYSTAL STRUCTURE OF HG-BOUND SUFB-SUFC-SUFD COMPLEX FROM ESCHERICHIA COLI | IRON-SULFUR CLUSTERS, IRON-SULFUR PROTEINS, ABC PROTEINS, ABC ATPASE, TRANSPORT PROTEIN-PROTEIN BINDING COMPLEX
5awg:F (ASP368) to (LEU418) CRYSTAL STRUCTURE OF HG-BOUND SUFB-SUFC-SUFD COMPLEX FROM ESCHERICHIA COLI | IRON-SULFUR CLUSTERS, IRON-SULFUR PROTEINS, ABC PROTEINS, ABC ATPASE, TRANSPORT PROTEIN-PROTEIN BINDING COMPLEX
5awk:A (LEU220) to (ALA263) CRYSTAL STRUCTURE OF VDR-LBD/PARTIAL AGONIST COMPLEX: 22S-ETHYL ANALOGUE | TRANDCRIPTION, VITAMIN D, VDRE, RXR, CO-FACTORS, HORMONE, TRANSCRIPTION
4mxm:B (SER122) to (MSE193) CRYSTAL STRUCTURE OF SUPERANTIGEN PFIT | SUPERANTIGEN, DNA BINDING PROTEIN
5axp:A (ASN562) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF PDE10A COMPLEXED WITH 1- (2-FLUORO-4-(2-OXO-1,3-OXAZOLIDIN-3-YL)PHENYL)-5-METHOXY-3-(1-PHENYL- 1H-PYRAZOL-5-YL)PYRIDAZIN-4(1H)-ONE | HYDROLASE/HYDROLASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5axp:B (SER561) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF PDE10A COMPLEXED WITH 1- (2-FLUORO-4-(2-OXO-1,3-OXAZOLIDIN-3-YL)PHENYL)-5-METHOXY-3-(1-PHENYL- 1H-PYRAZOL-5-YL)PYRIDAZIN-4(1H)-ONE | HYDROLASE/HYDROLASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5axq:B (SER561) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF PDE10A COMPLEXED WITH HIGHLY POTENT AND BRAIN-PENETRANT PDE10A INHIBITOR WITH 2-OXINDOLE SCAFFOLD | HYDROLASE/HYDROLASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4myh:A (PRO129) to (MET232) STRUCTURE OF THE GLUTATHIONE BOUND MITOCHONDRIAL ABC TRANSPORTER, ATM1 | ABC TRANSPORTER, MEMBRANE TRANSPORT, MITOCHONDRIAL INNER MEMBRANE, GLUTATHIONE, TRANSPORT PROTEIN
2xmo:B (ASP345) to (GLY402) THE CRYSTAL STRUCTURE OF LMO2642 | PHOSPHODIESTERASE, HYDROLASE
2xmz:A (GLU121) to (SER176) STRUCTURE OF MENH FROM S. AUREUS | MENAQUINONE BIOSYNTHESIS, LYASE
4mz7:A (ARG164) to (GLY258) STRUCTURAL INSIGHT INTO DGTP-DEPENDENT ACTIVATION OF TETRAMERIC SAMHD1 DEOXYNUCLEOSIDE TRIPHOSPHATE TRIPHOSPHOHYDROLASE | HD-DOMAIN, HYDROLASE, DNTP BINDING, PHOSPHORYLATION
3wyk:A (ASN562) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF PDE10A COMPLEXED WITH 3- (1-PHENYL-1H-PYRAZOL-5-YL)-1-(3-(TRIFLUOROMETHYL)PHENYL)PYRIDAZIN- 4(1H)-ONE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3wyk:B (SER561) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF PDE10A COMPLEXED WITH 3- (1-PHENYL-1H-PYRAZOL-5-YL)-1-(3-(TRIFLUOROMETHYL)PHENYL)PYRIDAZIN- 4(1H)-ONE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3wyl:A (SER561) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF PDE10A COMPLEXED WITH 5- METHOXY-3-(1-PHENYL-1H-PYRAZOL-5-YL)-1-(3-(TRIFLUOROMETHYL)PHENYL) PYRIDAZIN-4(1H)-ONE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3wyl:B (ASN562) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF PDE10A COMPLEXED WITH 5- METHOXY-3-(1-PHENYL-1H-PYRAZOL-5-YL)-1-(3-(TRIFLUOROMETHYL)PHENYL) PYRIDAZIN-4(1H)-ONE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3wym:A (SER561) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF PDE10A COMPLEXED WITH 1- (2-FLUORO-4-(1H-PYRAZOL-1-YL)PHENYL)-5-METHOXY-3-(1-PHENYL-1H- PYRAZOL-5-YL)PYRIDAZIN-4(1H)-ONE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3wym:B (SER561) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF PDE10A COMPLEXED WITH 1- (2-FLUORO-4-(1H-PYRAZOL-1-YL)PHENYL)-5-METHOXY-3-(1-PHENYL-1H- PYRAZOL-5-YL)PYRIDAZIN-4(1H)-ONE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5azb:A (TRP25) to (PHE93) CRYSTAL STRUCTURE OF ESCHERICHIA COLI LGT IN COMPLEX WITH PHOSPHATIDYLGLYCEROL AND THE INHIBITOR PALMITIC ACID | INHIBITOR, COMPLEX, TRANSFERASE
5azc:A (TRP25) to (PHE93) CRYSTAL STRUCTURE OF ESCHERICHIA COLI LGT IN COMPLEX WITH PHOSPHATIDYLGLYCEROL | INHIBITOR, COMPLEX, TRANSFERASE
2xo3:A (LEU66) to (LYS101) HUMAN ANNEXIN V WITH INCORPORATED METHIONINE ANALOGUE HOMOPROPARGYLGLYCINE | MEMBRANE BINDING PROTEIN, APOPTOSIS, ION CHANNEL
4n1k:A (LEU15) to (ALA53) CRYSTAL STRUCTURES OF NLRP14 PYRIN DOMAIN REVEAL A CONFORMATIONAL SWITCH MECHANISM, REGULATING ITS MOLECULAR INTERACTIONS | DEATH DOMAIN FOLD, PYRIN DOMAIN, NOD-LIKE RECEPTOR, SIGNALING PROTEIN, PROTEIN BINDING, SPERMATOGENESIS, INNATE IMMUNITY
1w36:B (ASP634) to (LEU701) RECBCD:DNA COMPLEX | RECOMBINATION, HELICASE, NUCLEASE, HYDROLASE, DNA REPAIR
1w36:E (TRP638) to (LEU701) RECBCD:DNA COMPLEX | RECOMBINATION, HELICASE, NUCLEASE, HYDROLASE, DNA REPAIR
4n4n:C (THR333) to (GLY425) NITROSOMONAS EUROPEA HAO | C-TYPE CYTOCHROME, OXIDOREDUCTASE
4n4o:A (THR333) to (GLY425) NITROSOMONAS EUROPEA HAO SOAKED IN NH2OH | C-TYPE CYTOCHROME, OXIDOREDUCTASE
4n4o:E (THR333) to (GLY425) NITROSOMONAS EUROPEA HAO SOAKED IN NH2OH | C-TYPE CYTOCHROME, OXIDOREDUCTASE
5b4k:A (SER561) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN PDE10A COMPLEXED WITH N-(4-((5-METHYL-5H-PYRROLO[3,2-D]PYRIMIDIN-4-YL)OXY)PHENYL)-1H- BENZIMIDAZOL-2-AMINE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5b4k:B (SER561) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN PDE10A COMPLEXED WITH N-(4-((5-METHYL-5H-PYRROLO[3,2-D]PYRIMIDIN-4-YL)OXY)PHENYL)-1H- BENZIMIDAZOL-2-AMINE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5b4l:A (SER561) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN PDE10A COMPLEXED WITH 1-(CYCLOPROPYLMETHYL)-5-(2-(2,3-DIHYDRO-1H-IMIDAZO[1,2- A]BENZIMIDAZOL-1-YL)ETHOXY)-3-(1-PHENYL-1H-PYRAZOL-5-YL)PYRIDAZIN- 4(1H)-ONE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5b4l:B (SER561) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN PDE10A COMPLEXED WITH 1-(CYCLOPROPYLMETHYL)-5-(2-(2,3-DIHYDRO-1H-IMIDAZO[1,2- A]BENZIMIDAZOL-1-YL)ETHOXY)-3-(1-PHENYL-1H-PYRAZOL-5-YL)PYRIDAZIN- 4(1H)-ONE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3jab:C (ASN661) to (THR723) DOMAIN ORGANIZATION AND CONFORMATIONAL PLASTICITY OF THE G PROTEIN EFFECTOR, PDE6 | PHOSPHODIESTERASE, PHOTORECEPTOR, HYDROLASE-IMMUNE SYSTEM COMPLEX
3jab:O (ASN661) to (THR723) DOMAIN ORGANIZATION AND CONFORMATIONAL PLASTICITY OF THE G PROTEIN EFFECTOR, PDE6 | PHOSPHODIESTERASE, PHOTORECEPTOR, HYDROLASE-IMMUNE SYSTEM COMPLEX
3zfz:A (LYS28) to (LEU73) CRYSTAL STRUCTURE OF CEFTAROLINE ACYL-PBP2A FROM MRSA WITH NON-COVALENTLY BOUND CEFTAROLINE AND MURAMIC ACID AT ALLOSTERIC SITE OBTAINED BY SOAKING | HYDROLASE, PENICILLIN BINDING PROTEINS, MRSA, ALLOSTERIC SITE, B- LACTAM ANTIBIOTICS
3zg5:A (ASP27) to (GLY74) CRYSTAL STRUCTURE OF PBP2A FROM MRSA IN COMPLEX WITH PEPTIDOGLYCAN ANALOGUE AT ALLOSTERIC | HYDROLASE, PENICILLIN BINDING PROTEINS, ALLOSTERIC SITE, B- LACTAM ANTIBIOTICS
4nc6:A (LEU738) to (ARG784) TBC DOMAIN OF HUMAN RAB GTPASE-ACTIVATING PROTEIN 1 | TBC DOMAIN, GTPASE ACTIVATION, HYDROLASE ACTIVATOR
1k6k:A (THR81) to (GLY141) CRYSTAL STRUCTURE OF CLPA, AN AAA+ CHAPERONE-LIKE REGULATOR OF CLPAP PROTEASE IMPLICATION TO THE FUNCTIONAL DIFFERENCE OF TWO ATPASE DOMAINS | CLPA, CHAPERONE, ATPASE, ADAPTOR BINDING, X-RAY, STRUCTURE, N-DOMAIN, HYDROLASE
1wer:A (LYS815) to (LEU904) RAS-GTPASE-ACTIVATING DOMAIN OF HUMAN P120GAP | GTPASE ACTIVATION, RAS, GAP, SIGNAL TRANSDUCTION, GROWTH REGULATION, CANCER
3zjg:A (MET105) to (SER176) A20 OTU DOMAIN WITH IRREVERSIBLY OXIDISED CYS103 FROM 60 MIN H2O2 SOAK. | HYDROLASE, UBIQUITIN, DEUBIQUITINATING ENZYME, REVERSIBLE OXIDATION, SULPHENIC ACID, SULPHINIC ACID, SULPHONIC ACID, CYS PROTEASE
2k2f:A (GLU3) to (ASP50) SOLUTION STRUCTURE OF CA2+-S100A1-RYRP12 | S100, EF HAND, RYANODINE RECEPTOR, CALCIUM BINDING, ALTERNATIVE SPLICING, CALCIUM CHANNEL, CALCIUM TRANSPORT, GLYCOPROTEIN, ION TRANSPORT, IONIC CHANNEL, MEMBRANE, POLYMORPHISM, TRANSMEMBRANE, TRANSPORT, CYTOPLASM, METAL- BINDING, ZINC, METAL BINDING PROTEIN
2k2f:B (SER2) to (ASP50) SOLUTION STRUCTURE OF CA2+-S100A1-RYRP12 | S100, EF HAND, RYANODINE RECEPTOR, CALCIUM BINDING, ALTERNATIVE SPLICING, CALCIUM CHANNEL, CALCIUM TRANSPORT, GLYCOPROTEIN, ION TRANSPORT, IONIC CHANNEL, MEMBRANE, POLYMORPHISM, TRANSMEMBRANE, TRANSPORT, CYTOPLASM, METAL- BINDING, ZINC, METAL BINDING PROTEIN
3jb2:A (ALA85) to (LEU157) ATOMIC MODEL OF CYTOPLASMIC POLYHEDROSIS VIRUS WITH SAM AND GTP | VIRAL ATPASE, HISTIDINE-MEDIATED GUANYLYL TRANSFER, CONFORMATIONAL CHANGES, REGULATION OF TRANSCRIPTION, VIRUS
2kil:A (LEU47) to (GLY97) NMR STRUCTURE OF THE H103G MUTANT SO2144 H-NOX DOMAIN FROM SHEWANELLA ONEIDENSIS IN THE FE(II)CO LIGATION STATE | H-NOX, UNKNOWN FUNCTION
3jb3:A (PRO84) to (LEU157) ATOMIC MODEL OF CYTOPLASMIC POLYHEDROSIS VIRUS WITH SAM, GTP AND ATP | VIRAL ATPASE, HISTIDINE-MEDIATED GUANYLYL TRANSFER, CONFORMATIONAL CHANGES, REGULATION OF TRANSCRIPTION, VIRUS
4nm2:A (PRO108) to (LYS148) STRUCTURE OF HUMAN DNA POLYMERASE BETA COMPLEXED WITH A NICKED DNA CONTAINING A 8BRG-G AT N-1 POSITION AND G-C AT N POSITION | DNA BINDING, HELIX-TURN-HELIX MOTIF, POLYMERASE FOLD, NUCLEOTIDYL TRANSFERASE, NUCLEUS, TRANSFERASE, LYASE-DNA COMPLEX
2y5d:B (ASP41) to (GLY120) CRYSTAL STRUCTURE OF C296A MUTANT OF THE BOX PATHWAY ENCODED ALDH FROM BURKHOLDERIA XENOVORANS LB400 | OXIDOREDUCTASE
3znv:A (ALA208) to (HIS276) CRYSTAL STRUCTURE OF THE OTU DOMAIN OF OTULIN AT 1.3 ANGSTROMS. | HYDROLASE
3znz:A (ALA208) to (HIS276) CRYSTAL STRUCTURE OF OTULIN OTU DOMAIN (C129A) IN COMPLEX WITH MET1-DI UBIQUITIN | HYDROLASE
5c1w:A (SER561) to (THR623) PDE10 COMPLEXED WITH 4,6-DICHLORO-2-CYCLOPROPYL-5-METHYL-PYRIMIDINE | PHOSPHODIESTERASE, INHIBITOR, COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5c28:A (SER561) to (THR623) PDE10 COMPLEXED WITH 6-CHLORO-2-CYCLOPROPYL-5-METHYL-PYRIMIDIN-4-AMINE | PHOSPHODIESTERASE, INHIBITOR, COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5c29:A (SER561) to (THR623) PDE10 COMPLEXED WITH 6-CHLORO-2-CYCLOPROPYL-5-METHYL-N-PROPYL- PYRIMIDIN-4-AMINE | PHOSPHODIESTERASE, INHIBITOR, COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5c2a:A (SER561) to (THR623) PDE10 COMPLEXED WITH 6-CHLORO-2-CYCLOPROPYL-N-[(2,4-DIMETHYLTHIAZOL-5- YL)METHYL]-5-METHYL-PYRIMIDIN-4-AMINE | PHOSPHODIESTERASE, INHIBITOR, COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5c2a:B (SER561) to (THR623) PDE10 COMPLEXED WITH 6-CHLORO-2-CYCLOPROPYL-N-[(2,4-DIMETHYLTHIAZOL-5- YL)METHYL]-5-METHYL-PYRIMIDIN-4-AMINE | PHOSPHODIESTERASE, INHIBITOR, COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3zqa:B (SER42) to (LEU119) CRYSTALLOGRAPHIC STRUCTURE OF BETAINE ALDEHYDE DEHYDROGENASE MUTANT C286A FROM PSEUDOMONAS AERUGINOSA IN COMPLEX WITH NADPH | ALDEHYDE OXIDATION, NADPH COMPLEX, OXIDOREDUCTASE
3zqa:D (SER42) to (LEU119) CRYSTALLOGRAPHIC STRUCTURE OF BETAINE ALDEHYDE DEHYDROGENASE MUTANT C286A FROM PSEUDOMONAS AERUGINOSA IN COMPLEX WITH NADPH | ALDEHYDE OXIDATION, NADPH COMPLEX, OXIDOREDUCTASE
5c2h:A (SER561) to (THR623) PDE10 COMPLEXED WITH 6-CHLORO-N-[(2,4-DIMETHYLTHIAZOL-5-YL)METHYL]-5- METHYL-2-[3-(2-QUINOLYL)PROPOXY]PYRIMIDIN-4-AMINE | PHOSPHODIESTERASE, INHIBITOR, COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5c2h:B (SER561) to (THR623) PDE10 COMPLEXED WITH 6-CHLORO-N-[(2,4-DIMETHYLTHIAZOL-5-YL)METHYL]-5- METHYL-2-[3-(2-QUINOLYL)PROPOXY]PYRIMIDIN-4-AMINE | PHOSPHODIESTERASE, INHIBITOR, COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2li6:A (GLU14) to (LEU80) 1H, 13C, AND 15N CHEMICAL SHIFT ASSIGNMENTS FOR YEAST PROTEIN | LIGAND BINDING, DNA BINDING PROTEIN
3jbq:B (ASN662) to (THR723) DOMAIN ORGANIZATION AND CONFORMATIONAL PLASTICITY OF THE G PROTEIN EFFECTOR, PDE6 | PHOSPHODIESTERASE, PHOTORECEPTOR, PDE6, HYDROLASE-IMMUNE SYSTEM COMPLEX
3jbq:F (ASN662) to (THR723) DOMAIN ORGANIZATION AND CONFORMATIONAL PLASTICITY OF THE G PROTEIN EFFECTOR, PDE6 | PHOSPHODIESTERASE, PHOTORECEPTOR, PDE6, HYDROLASE-IMMUNE SYSTEM COMPLEX
3zrj:A (ASN14) to (THR74) COMPLEX OF CLPV N-DOMAIN WITH VIPB PEPTIDE | CHAPERONE-PEPTIDE COMPLEX, HSP100 PROTEINS, AAA+ PROTEINS, T6SS, SECRETION, VIRULENCE
3zrj:B (ASN14) to (SER73) COMPLEX OF CLPV N-DOMAIN WITH VIPB PEPTIDE | CHAPERONE-PEPTIDE COMPLEX, HSP100 PROTEINS, AAA+ PROTEINS, T6SS, SECRETION, VIRULENCE
2lwd:A (GLU135) to (ARG179) SOLUTION STRUCTURE OF SECOND CARD OF HUMAN RIG-I | RIG-I, CARD, SENSOR, VIRAL RNA, HELICASE, SIGNALING PROTEIN
1x7r:A (THR311) to (TRP383) CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR ALPHA COMPLEXED WITH GENISTEIN | ESTROGEN RECEPTOR, ESTROGEN RECEPTOR BETA, ER-BETA, ER, ESTROGEN RECEPTOR ALPHA, ER-ALPHA, ESTROGEN, NUCLEAR RECEPT TRANSCRIPTION FACTOR, AGONIST
5c78:A (TYR56) to (ILE136) ATP-DRIVEN LIPID-LINKED OLIGOSACCHARIDE FLIPPASE PGLK IN APO-INWARD STATE (1) | ABC TRANSPORTER FLIPPASE, HYDROLASE
5c78:B (TYR56) to (ILE136) ATP-DRIVEN LIPID-LINKED OLIGOSACCHARIDE FLIPPASE PGLK IN APO-INWARD STATE (1) | ABC TRANSPORTER FLIPPASE, HYDROLASE
1xdt:T (HIS223) to (GLN287) COMPLEX OF DIPHTHERIA TOXIN AND HEPARIN-BINDING EPIDERMAL GROWTH FACTOR | COMPLEX (TOXIN-GROWTH FACTOR), DIPHTHERIA TOXIN, RECEPTOR, HEPARIN- BINDING EPIDERMAL GROWTH FACTOR, EPIDERMAL GROWTH FACTOR, COMPLEX (TOXIN-GROWTH FACTOR) COMPLEX
2yk0:A (CYS608) to (LYS672) STRUCTURE OF THE N-TERMINAL NTS-DBL1-ALPHA AND CIDR-GAMMA DOUBLE DOMAIN OF THE PFEMP1 PROTEIN FROM PLASMODIUM FALCIPARUM VARO STRAIN. | ADHESIN, MEMBRANE PROTEIN, PFEMP1
2ylp:A (ILE672) to (TYR739) TARGETING THE BINDING FUNCTION 3 SITE OF THE ANDROGEN RECEPTOR THROUGH IN SILICO MOLECULAR MODELING | HORMONE RECEPTOR, BINDING FUNCTION 3
2ylq:A (PRO671) to (TYR739) TARGETING THE BINDING FUNCTION 3 SITE OF THE ANDROGEN RECEPTOR THROUGH IN SILICO MOLECULAR MODELING | HORMONE RECEPTOR, BINDING FUNCTION 3
3jwr:A (ASN661) to (THR723) CRYSTAL STRUCTURE OF CHIMERIC PDE5/PDE6 CATALYTIC DOMAIN COMPLEXED WITH 3-ISOBUTYL-1-METHYLXANTHINE (IBMX) AND PDE6 GAMMA-SUBUNIT INHIBITORY PEPTIDE 70-87. | MOSTLY ALPHA, CGMP, HYDROLASE, POLYMORPHISM, SENSORY TRANSDUCTION, VISION
3jwr:B (ASN661) to (THR723) CRYSTAL STRUCTURE OF CHIMERIC PDE5/PDE6 CATALYTIC DOMAIN COMPLEXED WITH 3-ISOBUTYL-1-METHYLXANTHINE (IBMX) AND PDE6 GAMMA-SUBUNIT INHIBITORY PEPTIDE 70-87. | MOSTLY ALPHA, CGMP, HYDROLASE, POLYMORPHISM, SENSORY TRANSDUCTION, VISION
4a2j:B (GLN838) to (GLY923) PR X-RAY STRUCTURES IN AGONIST CONFORMATIONS REVEAL TWO DIFFERENT MECHANISMS FOR PARTIAL AGONISM IN 11BETA- SUBSTITUTED STEROIDS | TRANSCRIPTION, PARTIAL AGONIST
2yyv:A (GLY162) to (THR206) CRYSTAL STRUCTURE OF UNCHARACTERIZED CONSERVED PROTEIN FROM THERMOTOGA MARITIMA | UNCHARACTERIZED CONSERVED PROTEIN, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, HYDROLASE
2yyv:B (GLY162) to (THR206) CRYSTAL STRUCTURE OF UNCHARACTERIZED CONSERVED PROTEIN FROM THERMOTOGA MARITIMA | UNCHARACTERIZED CONSERVED PROTEIN, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, HYDROLASE
2z0j:B (ASP172) to (GLN214) CRYSTAL STRUCTURE OF UNCHARACTERIZED CONSERVED PROTEIN FROM THERMUS THERMOPHILUS HB8 | UNCHARACTERIZED CONSERVED PROTEIN, STRUCTURAL GENOMICS, UNKNOWN FUNCTION, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
2z0j:E (ASP172) to (GLN214) CRYSTAL STRUCTURE OF UNCHARACTERIZED CONSERVED PROTEIN FROM THERMUS THERMOPHILUS HB8 | UNCHARACTERIZED CONSERVED PROTEIN, STRUCTURAL GENOMICS, UNKNOWN FUNCTION, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
2z0j:F (ASP172) to (GLN214) CRYSTAL STRUCTURE OF UNCHARACTERIZED CONSERVED PROTEIN FROM THERMUS THERMOPHILUS HB8 | UNCHARACTERIZED CONSERVED PROTEIN, STRUCTURAL GENOMICS, UNKNOWN FUNCTION, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
2z0j:G (ASP172) to (GLN214) CRYSTAL STRUCTURE OF UNCHARACTERIZED CONSERVED PROTEIN FROM THERMUS THERMOPHILUS HB8 | UNCHARACTERIZED CONSERVED PROTEIN, STRUCTURAL GENOMICS, UNKNOWN FUNCTION, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
3k2w:G (LYS47) to (ASP121) CRYSTAL STRUCTURE OF BETAINE-ALDEHYDE DEHYDROGENASE FROM PSEUDOALTEROMONAS ATLANTICA T6C | STRUCTURAL GENOMICS, PSI-2, ALDEHYDE DEHYDROGENASE, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, OXIDOREDUCTASE
4ogb:B (HIS105) to (HIS152) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF PDE4D2 WITH COMPOUND 2 | CATALYTIC MECHANISM, CAMP HYDROLYSIS, HYDROLASE-INHIBITOR COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2o4j:A (TYR147) to (SER262) CRYSTAL STRUCTURE OF RAT VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH VITIII 17-20Z AND THE NR2 BOX OF DRIP 205 | NUCLEAR RECEPTOR-LIGAND COMPLEX, HORMONE/GROWTH FACTOR RECEPTOR COMPLEX
3k70:B (GLU635) to (LEU701) CRYSTAL STRUCTURE OF THE COMPLETE INITIATION COMPLEX OF RECBCD | RECOMBINATION, HELICASE, NUCLEASE, HYDROLASE, DNA REPAIR, ATP-BINDING, DNA DAMAGE, ENDONUCLEASE, EXONUCLEASE, NUCLEOTIDE-BINDING, HYDROLASE/DNA COMPLEX
3k70:E (GLU635) to (LEU701) CRYSTAL STRUCTURE OF THE COMPLETE INITIATION COMPLEX OF RECBCD | RECOMBINATION, HELICASE, NUCLEASE, HYDROLASE, DNA REPAIR, ATP-BINDING, DNA DAMAGE, ENDONUCLEASE, EXONUCLEASE, NUCLEOTIDE-BINDING, HYDROLASE/DNA COMPLEX
1lzw:B (THR172) to (SER230) STRUCTURAL BASIS OF CLPS-MEDIATED SWITCH IN CLPA SUBSTRATE RECOGNITION | ALPHA-BETA-PROTEIN (CLPS), ALPHA-PROTEIN (CLPA-ND), CHAPERONE
2zd7:A (MET40) to (ILE83) THE STRUCTURE OF VPS75 (VACUOLAR PROTEIN SORTING-ASSOCIATED PROTEIN 75) | HISTONE CHAPERONE, VPS75, NAP1, NUCLEUS, PHOSPHOPROTEIN, PROTEIN TRANSPORT, TRANSPORT
2zd7:B (ALA12) to (ILE83) THE STRUCTURE OF VPS75 (VACUOLAR PROTEIN SORTING-ASSOCIATED PROTEIN 75) | HISTONE CHAPERONE, VPS75, NAP1, NUCLEUS, PHOSPHOPROTEIN, PROTEIN TRANSPORT, TRANSPORT
1xos:A (SER282) to (THR345) CATALYTIC DOMAIN OF HUMAN PHOSPHODIESTERASE 4B IN COMPLEX WITH SILDENAFIL | PHOSPHODIESTERASE, PDE, PDE4B, SILDENAFIL, VIAGRA, HYDROLASE
1xow:A (ILE672) to (SER740) CRYSTAL STRUCTURE OF THE HUMAN ANDROGEN RECEPTOR LIGAND BINDING DOMAIN BOUND WITH AN ANDROGEN RECEPTOR NH2- TERMINAL PEPTIDE, AR20-30, AND R1881 | CRYSTAL STRUCTURE; HUMAN ANDROGEN RECEPTOR LIGAND BINDING DOMAIN; ANDROGEN RECEPTOR NH2-TERMINAL PEPTIDE AR20-30; R1881, TRANSCRIPTION
1xp1:A (THR311) to (ALA382) HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH COMPOUND 15 | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, ER-ALPHA, ANTAGONIST, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
3k9d:B (ASP7) to (SER78) CRYSTAL STRUCTURE OF PROBABLE ALDEHYDE DEHYDROGENASE FROM LISTERIA MONOCYTOGENES EGD-E | STRUCTURAL GENOMICS, PSI-2, ALDEHYDE DEHYDROGENASE, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, OXIDOREDUCTASE
3kby:A (HIS0) to (LEU58) CRYSTAL STRUCTURE OF HYPOTHETICAL PROTEIN FROM STAPHYLOCOCCUS AUREUS | PUTATIVE UNCHARACTERIZED PROTEIN, ALL HELICAL, UNKNOWN FUNCTION
4aa2:A (THR358) to (LEU436) CRYSTAL STRUCTURE OF ANCE IN COMPLEX WITH BRADYKININ POTENTIATING PEPTIDE B | HYDROLASE-PEPTIDE COMPLEX, HYDROLASE, SUBSTRATE BINDING, INHIBITOR
2zla:A (TYR147) to (ALA263) 2-SUBSTITUTED-16-ENE-22-THIA-1ALPHA,25-DIHYDROXY-26,27- DIMETHYL-19-NORVITAMIN D3 ANALOGS: SYNTHESIS, BIOLOGICAL EVALUATION AND CRYSTAL STRUCTURE | PROTEIN-LIGAND COMPLEX, DNA-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, HORMONE
2zlc:A (TYR147) to (ALA263) 2-SUBSTITUTED-16-ENE-22-THIA-1ALPHA,25-DIHYDROXY-26,27- DIMETHYL-19-NORVITAMIN D3 ANALOGS: SYNTHESIS, BIOLOGICAL EVALUATION AND CRYSTAL STRUCTURE | PROTEIN-LIGAND COMPLEX, DNA-BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, HORMONE
1xu3:B (ASP365) to (ASN412) SOLUBLE METHANE MONOOXYGENASE HYDROXYLASE-SOAKED WITH BROMOPHENOL | METHANE, SUBSTRATE BINDING, DIIRON, FOUR-HELIX BUNDLE, CAVITIES, OXIDOREDUCTASE
3kfc:B (THR221) to (SER307) COMPLEX STRUCTURE OF LXR WITH AN AGONIST | NUCLEAR RECEPTOR, LXR, LIVER X RECEPTOR, LXR AGONIST, LXR LIGAND, DNA-BINDING, METAL-BINDING, NUCLEUS, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
2zmi:A (TYR147) to (ALA263) CRYSTAL STRUCTURE OF RAT VITAMIN D RECEPTOR BOUND TO ADAMANTYL VITAMIN D ANALOGS: STRUCTURAL BASIS FOR VITAMIN D RECEPTOR ANTAGONISM AND/OR PARTIAL AGONISM | NUCLEAR RECEPTOR-ANTAGONIST COMPLEX, DNA-BINDING, METAL- BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACTIVATOR
1mbu:B (THR81) to (SER139) CRYSTAL STRUCTURE ANALYSIS OF CLPSN HETERODIMER | PROTEIN BINDING
2zu0:A (ASP369) to (LEU418) CRYSTAL STRUCTURE OF SUFC-SUFD COMPLEX INVOLVED IN THE IRON- SULFUR CLUSTER BIOSYNTHESIS | IRON-SULFUR CLUSTER, ABC-ATPASE, ATP-BINDING, CYTOPLASM, NUCLEOTIDE-BINDING, TRANSPORT, BIOSYNTHETIC PROTEIN/PROTEIN BINDING COMPLEX
2zu6:E (LEU226) to (GLY272) CRYSTAL STRUCTURE OF THE EIF4A-PDCD4 COMPLEX | PROTEIN-PROTEIN COMPLEX, ATP-BINDING, HELICASE, HYDROLASE, INITIATION FACTOR, NUCLEOTIDE-BINDING, PROTEIN BIOSYNTHESIS, RNA-BINDING, ANTI-ONCOGENE, APOPTOSIS, CELL CYCLE, CYTOPLASM, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM
1mdt:B (HIS223) to (VAL288) THE REFINED STRUCTURE OF MONOMERIC DIPHTHERIA TOXIN AT 2.3 ANGSTROMS RESOLUTION | TOXIN
1mg9:B (THR81) to (ILE138) THE STRUCTURAL BASIS OF CLPS-MEDIATED SWITCH IN CLPA SUBSTRATE RECOGNITION | AAA+ATPASE, SUBSTRATE SENSOR, CHAPERONE
4ae0:A (HIS223) to (VAL288) CRYSTAL STRUCTURE OF DIPHTHERIA TOXIN MUTANT CRM197 | TOXIN
4p0n:A (SER561) to (THR623) CRYSTAL STRUCTURE OF PDE10A WITH A NOVEL IMIDAZO[4,5-B]PYRIDINE INHIBITOR | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4p0n:B (SER561) to (THR623) CRYSTAL STRUCTURE OF PDE10A WITH A NOVEL IMIDAZO[4,5-B]PYRIDINE INHIBITOR | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4ael:A (SER571) to (THR633) PDE10A IN COMPLEX WITH THE INHIBITOR AZ5 | HYDROLASE, HIT-TO-LEAD, ENZYME INHIBITOR, NAPHTYRIDINE
4ael:B (SER571) to (THR633) PDE10A IN COMPLEX WITH THE INHIBITOR AZ5 | HYDROLASE, HIT-TO-LEAD, ENZYME INHIBITOR, NAPHTYRIDINE
4p1r:A (SER561) to (THR623) CRYSTAL STRUCTURE OF PDE10A WITH IMIDAZO[4,5-B]PYRIDINES AS POTENT AND SELECTIVE INHIBITORS | HYDROLASE-HYDROLASE INHIBITOR COMPLEX, HYDROLASE-HYDROLASE INBHITOR COMPLEX
4p1r:B (SER561) to (THR623) CRYSTAL STRUCTURE OF PDE10A WITH IMIDAZO[4,5-B]PYRIDINES AS POTENT AND SELECTIVE INHIBITORS | HYDROLASE-HYDROLASE INHIBITOR COMPLEX, HYDROLASE-HYDROLASE INBHITOR COMPLEX
2zxm:A (TYR147) to (SER262) A NEW CLASS OF VITAMIN D RECEPTOR LIGANDS THAT INDUCE STRUCTURAL REARRANGEMENT OF THE LIGAND-BINDING POCKET | NUCLEAR RECEPTOR-ANTAGONIST COMPLEX, TRANSCRIPTION, DNA- BINDING, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, RECEPTOR, TRANSCRIPTION REGULATION, ZINC, ZINC-FINGER, ACTIVATOR
4p3z:A (GLY158) to (THR211) CHLAMYDIA PNEUMONIAE COPN (D29 CONSTRUCT) | SECRETION REGULATION, T3SS, VIRULENCE, TRANSPORT, TUBULIN, TRANSPORT PROTEIN
4p4s:A (GLN283) to (LYS337) GMPPCP-BOUND STALKLESS-MXA | GTPASE, DYNAMIN-RELATED PROTEIN, ANTIVIRAL, SIGNALING PROTEIN, ANTIVIRAL PROTEIN-HYDROLASE COMPLEX
4p4t:A (GLY282) to (LEU342) GDP-BOUND STALKLESS-MXA | GTPASE, DYNAMIN-RELATED PROTEIN, ANTIVIRAL, MECHANO-ENZYME, HYDROLASE, GTP-BINDING PROTEIN, ANTIVIRAL PROTEIN-HYDROLASE COMPLEX
4p4u:A (GLY282) to (GLY361) NUCLEOTIDE-FREE STALKLESS-MXA | GTPASE, DYNAMIN-RELATED PROTEIN, ANTIVIRAL, MECHANO-ENZYME, HYDROLASE, GTP-BINDING PROTEIN, ANTIVIRAL PROTEIN-HYDROLASE COMPLEX
4ajd:A (SER571) to (THR633) IDENTIFICATION AND STRUCTURAL CHARACTERIZATION OF PDE10 FRAGMENT INHIBITORS | HYDROLASE
4ajd:D (SER571) to (THR633) IDENTIFICATION AND STRUCTURAL CHARACTERIZATION OF PDE10 FRAGMENT INHIBITORS | HYDROLASE
4ajg:A (SER571) to (THR633) IDENTIFICATION AND STRUCTURAL CHARACTERIZATION OF PDE10 FRAGMENT INHIBITORS | HYDROLASE
4ajg:D (SER571) to (THR633) IDENTIFICATION AND STRUCTURAL CHARACTERIZATION OF PDE10 FRAGMENT INHIBITORS | HYDROLASE
4ajm:A (SER571) to (THR633) DEVELOPMENT OF A PLATE-BASED OPTICAL BIOSENSOR METHODOLOGY TO IDENTIFY PDE10 FRAGMENT INHIBITORS | HYDROLASE
4ajm:D (SER571) to (THR633) DEVELOPMENT OF A PLATE-BASED OPTICAL BIOSENSOR METHODOLOGY TO IDENTIFY PDE10 FRAGMENT INHIBITORS | HYDROLASE
1mws:A (LYS28) to (LEU73) STRUCTURE OF NITROCEFIN ACYL-PENICILLIN BINDING PROTEIN 2A FROM METHICILLIN RESISTANT STAPHYLOCOCCUS AUREUS STRAIN 27R AT 2.00 A RESOLUTION. | PENICILLIN BINDING PROTEIN, BETA-LACTAM, D, D- TRANSPEPTIDASE, D-CARBOXYPEPTIDASE, NITROCEFIN, BIOSYNTHETIC PROTEIN
1mws:B (LYS28) to (GLY74) STRUCTURE OF NITROCEFIN ACYL-PENICILLIN BINDING PROTEIN 2A FROM METHICILLIN RESISTANT STAPHYLOCOCCUS AUREUS STRAIN 27R AT 2.00 A RESOLUTION. | PENICILLIN BINDING PROTEIN, BETA-LACTAM, D, D- TRANSPEPTIDASE, D-CARBOXYPEPTIDASE, NITROCEFIN, BIOSYNTHETIC PROTEIN
1yhu:A (ALA5) to (SER58) CRYSTAL STRUCTURE OF RIFTIA PACHYPTILA C1 HEMOGLOBIN REVEALS NOVEL ASSEMBLY OF 24 SUBUNITS. | HEMOGLOBIN, GLOBIN FOLD, OXYGEN STORAGE-TRANSPORT COMPLEX
1mwu:A (GLU29) to (LEU73) STRUCTURE OF METHICILLIN ACYL-PENICILLIN BINDING PROTEIN 2A FROM METHICILLIN RESISTANT STAPHYLOCOCCUS AUREUS STRAIN 27R AT 2.60 A RESOLUTION. | PENICILLIN BINDING PROTEIN, BETA-LACTAM, D,D-TRANSPEPTIDASE, D,D- CARBOXYPEPTIDASE, METHICILLIN, BIOSYNTHETIC PROTEIN
3kur:H (THR546) to (ASP589) CRYSTAL STRUCTURE OF THE MLLE DOMAIN OF POLY(A)-BINDING PROTEIN | ALL-HELICAL DOMAIN, METHYLATION, MRNA PROCESSING, MRNA SPLICING, NUCLEUS, PHOSPHOPROTEIN, RNA-BINDING, SPLICEOSOME, RNA BINDING PROTEIN
5dbv:A (MET35) to (THR102) STRUCTURE OF A C269A MUTANT OF PROPIONALDEHYDE DEHYDROGENASE FROM THE CLOSTRIDIUM PHYTOFERMENTANS FUCOSE UTILISATION BACTERIAL MICROCOMPARTMENT | ACYLATING ALDEHYDE DEHYDROGENASE, COA, PROPIONALDEHYDE, BMC, OXIDOREDUCTASE
1yow:A (ASP236) to (CYS301) HUMAN STEROIDOGENIC FACTOR 1 LBD WITH BOUND CO-FACTOR PEPTIDE | STEROIDOGENIC FACTOR 1, SF1, PHOSPHOLIPID, PHOSPHATIDYL ETHANOLAMINE, PHOSPHATIDYL GLYCEROL, TRANSCRIPTION
4phw:A (SER561) to (THR623) CRYSTAL STRUCTURE OF PDE10A WITH 1H-BENZIMIDAZOL-2-YL(4-((3- (TETRAHYDRO-2H-PYRAN-4-YL)-2-PYRIDINYL)OXY)PHENYL)METHANONE | INHIBITOR, PHOSPHODIESTERASE, KETO-BENZIMIDAZOLE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4phw:B (SER561) to (ALA622) CRYSTAL STRUCTURE OF PDE10A WITH 1H-BENZIMIDAZOL-2-YL(4-((3- (TETRAHYDRO-2H-PYRAN-4-YL)-2-PYRIDINYL)OXY)PHENYL)METHANONE | INHIBITOR, PHOSPHODIESTERASE, KETO-BENZIMIDAZOLE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5dh4:A (SER561) to (THR623) PDE10 COMPLEXED WITH 5-CHLORO-N-[(2,4-DIMETHYLTHIAZOL-5-YL) METHYL]PYRAZOLO[1,5-A]PYRIMIDIN-7-AMINE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5dh4:B (SER561) to (THR623) PDE10 COMPLEXED WITH 5-CHLORO-N-[(2,4-DIMETHYLTHIAZOL-5-YL) METHYL]PYRAZOLO[1,5-A]PYRIMIDIN-7-AMINE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5dh5:A (SER561) to (THR623) PDE10 COMPLEXED WITH N-[(1-METHYLPYRAZOL-4-YL)METHYL]-5-[[(1S,2S)-2- (2-PYRIDYL)CYCLOPROPYL]METHOXY]PYRAZOLO[1,5-A]PYRIMIDIN-7-AMINE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5dh5:B (SER561) to (THR623) PDE10 COMPLEXED WITH N-[(1-METHYLPYRAZOL-4-YL)METHYL]-5-[[(1S,2S)-2- (2-PYRIDYL)CYCLOPROPYL]METHOXY]PYRAZOLO[1,5-A]PYRIMIDIN-7-AMINE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1yuu:A (LEU9) to (LEU56) SOLUTION STRUCTURE OF CALCIUM-S100A13 | S100A13, EF HAND CALCIUM-BINDING PROTEINS, COPPER(II), NMR STRUCTURE, STRUCTURAL GENOMICS, STRUCTURAL PROTEOMICS IN EUROPE, SPINE, METAL BINDING PROTEIN
1yxi:A (THR12) to (SER88) R-STATE AMP COMPLEX REVEALS INITIAL STEPS OF THE QUATERNARY TRANSITION OF FRUCTOSE-1,6-BISPHOSPHATASE | GLYCOLYSIS; GLUCONEOGENESIS; ALLOSTERIC ENZYMES; FRUCTOSE-1,6- BISPHOSPHATASE; INTERMEDIATE STATES, HYDROLASE
3ahd:A (PRO95) to (PHE133) PHOSPHOKETOLASE FROM BIFIDOBACTERIUM BREVE COMPLEXED WITH 2-ACETYL- THIAMINE DIPHOSPHATE | THIAMINE DIPHOSPHATE-DEPENDENT ENZYME, ALPHA-BETA FOLD, HOMODIMER, ACETYL THIAMINE DIPHOSPHATE, LYASE
3ahe:A (PRO95) to (GLN132) PHOSPHOKETOLASE FROM BIFIDOBACTERIUM BREVE COMPLEXED WITH DIHYDROXYETHYL THIAMINE DIPHOSPHATE | THIAMINE DIPHOSPHATE-DEPENDENT ENZYME, ALPHA-BETA FOLD, HOMODIMER, DIHYDROXYETHYL THIAMINE DIPHOSPHATE, LYASE
3ahh:A (PRO95) to (PHE133) H142A MUTANT OF PHOSPHOKETOLASE FROM BIFIDOBACTERIUM BREVE COMPLEXED WITH ACETYL THIAMINE DIPHOSPHATE | THIAMINE DIPHOSPHATE-DEPENDENT ENZYME, ALPHA-BETA FOLD, HOMODIMER, ACETYL THIAMINE DIPHOSPHATE, LYASE
3ahi:A (PRO95) to (PHE133) H320A MUTANT OF PHOSPHOKETOLASE FROM BIFIDOBACTERIUM BREVE COMPLEXED WITH ACETYL THIAMINE DIPHOSPHATE | THIAMINE DIPHOSPHATE-DEPENDENT ENZYME, ALPHA-BETA FOLD, HOMODIMER, ACETYL THIAMINE DIPHOSPHATE, LYASE
3ahj:A (PRO95) to (PHE133) H553A MUTANT OF PHOSPHOKETOLASE FROM BIFIDOBACTERIUM BREVE | THIAMINE DIPHOSPHATE-DEPENDENT ENZYME, ALPHA-BETA FOLD, HOMODIMER, LYASE
1yz0:A (LEU13) to (SER88) R-STATE AMP COMPLEX REVEALS INITIAL STEPS OF THE QUATERNARY TRANSITION OF FRUCTOSE-1,6-BISPHOSPHATASE | ALLOSTERIC ENZYMES; INTERMEDIATE STATES; GLYCOLYSIS; GLUCONEOGENESIS, HYDROLASE
3ai7:H (PRO95) to (PHE133) CRYSTAL STRUCTURE OF BIFIDOBACTERIUM LONGUM PHOSPHOKETOLASE | THIAMINE-DIPHOSPHATE PROTEIN, LYASE
4pov:A (VAL87) to (LYS172) THIT WITH LMG135 BOUND | S-COMPONENT, THIAMINE-BINDING PROTEIN, ECF MODULE, MEMBRANE, PROTEIN BINDING
3lb1:A (GLY1) to (MET49) TWO-SITE COMPETITIVE INHIBITION IN DEHALOPEROXIDASE-HEMOGLOBIN | PEROXIDASE, GLOBIN, OXIDOREDUCTASE, HEME, OXYGEN TRANSPORT, TRANSPORT
3lb2:A (GLY1) to (MET49) TWO-SITE COMPETITIVE INHIBITION IN DEHALOPEROXIDASE-HEMOGLOBIN | PEROXIDASE, GLOBIN, OXIDOREDUCTASE
3lb3:A (GLY1) to (MET49) TWO-SITE COMPETITIVE INHIBITION IN DEHALOPEROXIDASE-HEMOGLOBIN | PEROXIDASE, GLOBIN, OXIDOREDUCTASE, HEME, OXYGEN TRANSPORT, TRANSPORT
3lb3:B (GLY1) to (MET49) TWO-SITE COMPETITIVE INHIBITION IN DEHALOPEROXIDASE-HEMOGLOBIN | PEROXIDASE, GLOBIN, OXIDOREDUCTASE, HEME, OXYGEN TRANSPORT, TRANSPORT
1z6q:A (VAL715) to (MET766) GLYCOGEN PHOSPHORYLASE WITH INHIBITOR IN THE AMP SITE | GLYCOGEN METABOLISM; GLYCOGEN PHOSPHORYLASE B; INHIBITION; ALLOSTERIC, TRANSFERASE
3akb:A (ARG27) to (ARG101) STRUCTURAL BASIS FOR PROKARYOTIC CALCIUM-MEDIATED REGULATION BY A STREPTOMYCES COELICOLOR CALCIUM-BINDING PROTEIN | CALCIUM-BINDING PROTEIN, EF-HAND, METAL BINDING PROTEIN
1z8d:A (ARG714) to (MET766) CRYSTAL STRUCTURE OF HUMAN MUSCLE GLYCOGEN PHOSPHORYLASE A WITH AMP AND GLUCOSE | TRANSFERASE
5dq6:A (ASP100) to (MET174) MUS MUSCULUS A20 OTU DOMAIN | A20 OTU, HYDROLASE
1z95:A (SER696) to (SER740) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND-BINDING DOMAIN W741L MUTANT COMPLEX WITH R-BICALUTAMIDE | STEROID HORMONES; RECEPTORS; CELLULAR PROLIFERATION; CELLULAR DIFFERENTIATION, TRANSCRIPTION REGULATION, RECEPTOR
3lj1:A (MET1034) to (PHE1088) IRE1 COMPLEXED WITH CDK1/2 INHIBITOR III | KINASE, KINASE INHIBITOR, NUCLEASE ACTIVATOR, ATP-BINDING, ENDOPLASMIC RETICULUM, GLYCOPROTEIN, HYDROLASE, MAGNESIUM, MEMBRANE, METAL-BINDING, MULTIFUNCTIONAL ENZYME, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, TRANSMEMBRANE, UNFOLDED PROTEIN RESPONSE
3lj1:B (MET1034) to (PHE1088) IRE1 COMPLEXED WITH CDK1/2 INHIBITOR III | KINASE, KINASE INHIBITOR, NUCLEASE ACTIVATOR, ATP-BINDING, ENDOPLASMIC RETICULUM, GLYCOPROTEIN, HYDROLASE, MAGNESIUM, MEMBRANE, METAL-BINDING, MULTIFUNCTIONAL ENZYME, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, TRANSMEMBRANE, UNFOLDED PROTEIN RESPONSE
3ang:B (ASP115) to (GLY192) CRYSTAL STRUCTURE OF THERMUS THERMOPHILUS FADR IN COMPLEX WITH E. COLI-DERIVED DODECYL-COA | ALL ALPHA PROTEIN, TETRACYCLIN REPRESSOR-LIKE, C-TERMINAL DOMAIN, TRANSCRIPTIONAL REPRESSOR, DNA BINDING, ACYL-COA, TRANSCRIPTION
5duh:B (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH A SULFOXIDE-BRIDGED OXABICYCLIC HEPTENE SULFONATE (SOBHS)-3 ANALOG PHENYL (1S,2S,4S,7S)-5,6-BIS(4-HYDROXY-3-METHYLPHENYL)-7- THIABICYCLO[2.2.1]HEPT-5-ENE-2-SULFONATE 7-OXIDE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
1zkn:B (ASN209) to (ASP272) STRUCTURE OF PDE4D2-IBMX | PROTEIN-INHIBITOR COMPLEX, INHIBITOR SELECTIVITY, HYDROLASE
3loc:A (LEU133) to (ARG209) CRYSTAL STRUCTURE OF PUTATIVE TRANSCRIPTIONAL REGULATOR YCDC | HELIX-TURN-HELIX, PUTATIVE TRANSCRIPTIONAL REGULATOR, DIMER, URACIL, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, DNA-BINDING, REPRESSOR, TRANSCRIPTION, TRANSCRIPTION REGULATION
3loc:B (LEU133) to (ARG209) CRYSTAL STRUCTURE OF PUTATIVE TRANSCRIPTIONAL REGULATOR YCDC | HELIX-TURN-HELIX, PUTATIVE TRANSCRIPTIONAL REGULATOR, DIMER, URACIL, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, DNA-BINDING, REPRESSOR, TRANSCRIPTION, TRANSCRIPTION REGULATION
3loc:C (MSE126) to (ARG209) CRYSTAL STRUCTURE OF PUTATIVE TRANSCRIPTIONAL REGULATOR YCDC | HELIX-TURN-HELIX, PUTATIVE TRANSCRIPTIONAL REGULATOR, DIMER, URACIL, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, DNA-BINDING, REPRESSOR, TRANSCRIPTION, TRANSCRIPTION REGULATION
3loc:D (MSE126) to (ARG209) CRYSTAL STRUCTURE OF PUTATIVE TRANSCRIPTIONAL REGULATOR YCDC | HELIX-TURN-HELIX, PUTATIVE TRANSCRIPTIONAL REGULATOR, DIMER, URACIL, STRUCTURAL GENOMICS, PSI, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, DNA-BINDING, REPRESSOR, TRANSCRIPTION, TRANSCRIPTION REGULATION
3lrb:B (GLY71) to (GLY143) STRUCTURE OF E. COLI ADIC | TRANSPORTER, ANTIPORTER, ADIC, AMINO-ACID TRANSPORT, ANTIPORT, CELL INNER MEMBRANE, CELL MEMBRANE, MEMBRANE, TRANSMEMBRANE, TRANSPORT, TRANSPORT PROTEIN
3lrc:A (GLY71) to (GLY143) STRUCTURE OF E. COLI ADIC (P1) | ADIC, TRANSPORTER, ANTIPORTER, AMINO-ACID TRANSPORT, ANTIPORT, CELL INNER MEMBRANE, CELL MEMBRANE, MEMBRANE, TRANSMEMBRANE, TRANSPORT, TRANSPORT PROTEIN
3lrc:B (GLY71) to (GLY143) STRUCTURE OF E. COLI ADIC (P1) | ADIC, TRANSPORTER, ANTIPORTER, AMINO-ACID TRANSPORT, ANTIPORT, CELL INNER MEMBRANE, CELL MEMBRANE, MEMBRANE, TRANSMEMBRANE, TRANSPORT, TRANSPORT PROTEIN
3lrc:C (GLY71) to (GLY143) STRUCTURE OF E. COLI ADIC (P1) | ADIC, TRANSPORTER, ANTIPORTER, AMINO-ACID TRANSPORT, ANTIPORT, CELL INNER MEMBRANE, CELL MEMBRANE, MEMBRANE, TRANSMEMBRANE, TRANSPORT, TRANSPORT PROTEIN
3lrc:D (GLY71) to (GLY143) STRUCTURE OF E. COLI ADIC (P1) | ADIC, TRANSPORTER, ANTIPORTER, AMINO-ACID TRANSPORT, ANTIPORT, CELL INNER MEMBRANE, CELL MEMBRANE, MEMBRANE, TRANSMEMBRANE, TRANSPORT, TRANSPORT PROTEIN
4aw6:A (LYS46) to (GLY154) CRYSTAL STRUCTURE OF THE HUMAN NUCLEAR MEMBRANE ZINC METALLOPROTEASE ZMPSTE24 (FACE1) | HYDROLASE, M48 PEPTIDASE, INTEGRAL MEMBRANE PROTEIN, PRELAMIN A PROCESSING, AGEING, PROGERIA
4aw6:B (LYS46) to (GLY154) CRYSTAL STRUCTURE OF THE HUMAN NUCLEAR MEMBRANE ZINC METALLOPROTEASE ZMPSTE24 (FACE1) | HYDROLASE, M48 PEPTIDASE, INTEGRAL MEMBRANE PROTEIN, PRELAMIN A PROCESSING, AGEING, PROGERIA
3lxg:A (ASN562) to (THR623) CRYSTAL STRUCTURE OF RAT PHOSPHODIESTERASE 10A IN COMPLEX WITH LIGAND WEB-3 | PHOSPHODIESTERASE 10A; CATALYTIC DOMAIN, ALLOSTERIC ENZYME, CAMP, CAMP-BINDING, CGMP, CGMP-BINDING, HYDROLASE, METAL-BINDING, NUCLEOTIDE-BINDING
5edg:A (SER571) to (THR633) HUMAN PDE10A IN COMPLEX WITH 3-(2-CHLORO-5-PHENYL-3H-IMIDAZOL-4-YL)-1- (3-TRIFLUOROMETHOXY-PHENYL)-1H-PYRIDAZIN-4-ONE AT 2.30A | PHOSPHODIESTERASE, PDE10, HYDROLASE
5edg:B (SER571) to (THR633) HUMAN PDE10A IN COMPLEX WITH 3-(2-CHLORO-5-PHENYL-3H-IMIDAZOL-4-YL)-1- (3-TRIFLUOROMETHOXY-PHENYL)-1H-PYRIDAZIN-4-ONE AT 2.30A | PHOSPHODIESTERASE, PDE10, HYDROLASE
5edg:C (ASN572) to (THR633) HUMAN PDE10A IN COMPLEX WITH 3-(2-CHLORO-5-PHENYL-3H-IMIDAZOL-4-YL)-1- (3-TRIFLUOROMETHOXY-PHENYL)-1H-PYRIDAZIN-4-ONE AT 2.30A | PHOSPHODIESTERASE, PDE10, HYDROLASE
5edg:D (ASN572) to (THR633) HUMAN PDE10A IN COMPLEX WITH 3-(2-CHLORO-5-PHENYL-3H-IMIDAZOL-4-YL)-1- (3-TRIFLUOROMETHOXY-PHENYL)-1H-PYRIDAZIN-4-ONE AT 2.30A | PHOSPHODIESTERASE, PDE10, HYDROLASE
5ede:A (SER571) to (THR633) HUMAN PDE10A IN COMPLEX WITH 1-(4-CHLORO-PHENYL)-3-METHYL-1H-THIENO[2, 3-C]PYRAZOLE-5-CARBOXYLIC ACID (TETRAHYDRO-FURAN-2-YLMETHYL)-AMIDE AT 2.2A | PHOSPHODIESTERASE, PDE10, HYDROLASE
5ede:B (SER571) to (THR633) HUMAN PDE10A IN COMPLEX WITH 1-(4-CHLORO-PHENYL)-3-METHYL-1H-THIENO[2, 3-C]PYRAZOLE-5-CARBOXYLIC ACID (TETRAHYDRO-FURAN-2-YLMETHYL)-AMIDE AT 2.2A | PHOSPHODIESTERASE, PDE10, HYDROLASE
5ede:C (SER571) to (THR633) HUMAN PDE10A IN COMPLEX WITH 1-(4-CHLORO-PHENYL)-3-METHYL-1H-THIENO[2, 3-C]PYRAZOLE-5-CARBOXYLIC ACID (TETRAHYDRO-FURAN-2-YLMETHYL)-AMIDE AT 2.2A | PHOSPHODIESTERASE, PDE10, HYDROLASE
5ede:D (SER571) to (THR633) HUMAN PDE10A IN COMPLEX WITH 1-(4-CHLORO-PHENYL)-3-METHYL-1H-THIENO[2, 3-C]PYRAZOLE-5-CARBOXYLIC ACID (TETRAHYDRO-FURAN-2-YLMETHYL)-AMIDE AT 2.2A | PHOSPHODIESTERASE, PDE10, HYDROLASE
5edh:A (SER571) to (THR633) HUMAN PDE10A, 8-ETHYL-5-METHYL-2-[2-(2-METHYL-5-PYRROLIDIN-1-YL-1,2,4- TRIAZOL-3-YL)ETHYL]-[1,2,4]TRIAZOLO[1,5-C]PYRIMIDINE, 2.03A, H3, RFREE=22.7% | PHOSPHODIESTERASE, PDE10, HYDROLASE
5edh:B (SER571) to (THR633) HUMAN PDE10A, 8-ETHYL-5-METHYL-2-[2-(2-METHYL-5-PYRROLIDIN-1-YL-1,2,4- TRIAZOL-3-YL)ETHYL]-[1,2,4]TRIAZOLO[1,5-C]PYRIMIDINE, 2.03A, H3, RFREE=22.7% | PHOSPHODIESTERASE, PDE10, HYDROLASE
5edh:C (SER571) to (THR633) HUMAN PDE10A, 8-ETHYL-5-METHYL-2-[2-(2-METHYL-5-PYRROLIDIN-1-YL-1,2,4- TRIAZOL-3-YL)ETHYL]-[1,2,4]TRIAZOLO[1,5-C]PYRIMIDINE, 2.03A, H3, RFREE=22.7% | PHOSPHODIESTERASE, PDE10, HYDROLASE
5edh:D (SER571) to (THR633) HUMAN PDE10A, 8-ETHYL-5-METHYL-2-[2-(2-METHYL-5-PYRROLIDIN-1-YL-1,2,4- TRIAZOL-3-YL)ETHYL]-[1,2,4]TRIAZOLO[1,5-C]PYRIMIDINE, 2.03A, H3, RFREE=22.7% | PHOSPHODIESTERASE, PDE10, HYDROLASE
5edi:A (SER571) to (ALA632) HUMAN PDE10A, 6-CHLORO-5,8-DIMETHYL-2-[2-(2-METHYL-5-PYRROLIDIN-1-YL- 2H-[1,2,4]TRIAZOL-3-YL)-ETHYL]-[1,2,4]TRIAZOLO[1,5-A]PYRIDINE, 2.20A, H3, RFREE=23.5% | PHOSPHODIESTERASE, PDE10, HYDROLASE
5edi:B (SER571) to (THR633) HUMAN PDE10A, 6-CHLORO-5,8-DIMETHYL-2-[2-(2-METHYL-5-PYRROLIDIN-1-YL- 2H-[1,2,4]TRIAZOL-3-YL)-ETHYL]-[1,2,4]TRIAZOLO[1,5-A]PYRIDINE, 2.20A, H3, RFREE=23.5% | PHOSPHODIESTERASE, PDE10, HYDROLASE
5edi:C (SER571) to (THR633) HUMAN PDE10A, 6-CHLORO-5,8-DIMETHYL-2-[2-(2-METHYL-5-PYRROLIDIN-1-YL- 2H-[1,2,4]TRIAZOL-3-YL)-ETHYL]-[1,2,4]TRIAZOLO[1,5-A]PYRIDINE, 2.20A, H3, RFREE=23.5% | PHOSPHODIESTERASE, PDE10, HYDROLASE
5edi:D (ASN572) to (THR633) HUMAN PDE10A, 6-CHLORO-5,8-DIMETHYL-2-[2-(2-METHYL-5-PYRROLIDIN-1-YL- 2H-[1,2,4]TRIAZOL-3-YL)-ETHYL]-[1,2,4]TRIAZOLO[1,5-A]PYRIDINE, 2.20A, H3, RFREE=23.5% | PHOSPHODIESTERASE, PDE10, HYDROLASE
5edl:A (GLU100) to (LEU162) CRYSTAL STRUCTURE OF AN S-COMPONENT OF ECF TRANSPORTER | MEMBRANE TRANSPORT PROTEIN, TRANSPORT PROTEIN
4qg2:B (PHE213) to (GLN271) CRYSTAL STRUCTURE OF THE TETRAMERIC GTP/DATP/ATP-BOUND SAMHD1 (RN206) MUTANT CATALYTIC CORE | DEOXYNUCLEOSIDE TRIPHOSPHATE TRIPHOSPHOHYDROLASE, 2'-DEOXYADENOSINE- 5'-TRIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, HIV RESTRICTION FACTOR, DNTPASE, HYDROLASE
4qg0:C (PHE213) to (VAL273) CRYSTAL STRUCTURE OF THE TETRAMERIC DGTP/DUTP-BOUND SAMHD1 (RN206) MUTANT CATALYTIC CORE | DEOXYNUCLEOSIDE TRIPHOSPHATE TRIPHOSPHOHYDROLASE, 2'-DEOXYNUCLEOTIDE- 5'-TRIPHOSPHATE, HIV RESTRICTION FACTOR, DNTPASE, HYDROLASE
4qg4:D (PHE165) to (GLY258) CRYSTAL STRUCTURE OF THE TETRAMERIC GTP/DATP/ATP-BOUND SAMHD1 (H210A) MUTANT CATALYTIC CORE | DEOXYNUCLEOSIDE TRIPHOSPHATE TRIPHOSPHOHYDROLASE, 2'-DEOXYADENOSINE- 5'-TRIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, HIV RESTRICTION FACTOR, DNTPASE, HYDROLASE
2aa1:B (ASP5) to (ASN57) CRYSTAL STRUCTURE OF THE CATHODIC HEMOGLOBIN ISOLATED FROM THE ANTARCTIC FISH TREMATOMUS NEWNESI | HEMOGLOBIN, ROOT EFFECT, COOPERATIVITY, ANTARCTIC FISH, OXYGEN STORAGE/TRANSPORT COMPLEX
3b66:A (PRO671) to (TRP741) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH SARM S-21 | ANDROGEN RECEPTOR, SARM, DISEASE MUTATION, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRIPLET REPEAT EXPANSION, UBL CONJUGATION, ZINC, ZINC-FINGER
3b67:A (PRO671) to (TRP741) CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH SARM C-23 | ANDROGEN RECEPTOR, SARM, DISEASE MUTATION, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, POLYMORPHISM, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRIPLET REPEAT EXPANSION, UBL CONJUGATION, ZINC, ZINC-FINGER
4bbx:A (SER561) to (THR623) DISCOVERY OF A POTENT, SELECTIVE AND ORALLY ACTIVE PDE10A INHIBITOR FOR THE TREATMENT OF SCHIZOPHRENIA | PHOSPHODIESTERASE INHIBITOR, INHIBITOR COMPLEX, HYDROLASE, ZINC BINDING, MAGNESIUM BINDING
4bbx:B (ASN562) to (THR623) DISCOVERY OF A POTENT, SELECTIVE AND ORALLY ACTIVE PDE10A INHIBITOR FOR THE TREATMENT OF SCHIZOPHRENIA | PHOSPHODIESTERASE INHIBITOR, INHIBITOR COMPLEX, HYDROLASE, ZINC BINDING, MAGNESIUM BINDING
3b9z:A (ASP162) to (HIS254) CRYSTAL STRUCTURE OF THE NITROSOMONAS EUROPAEA RH PROTEIN COMPLEXED WITH CARBON DIOXIDE | CARBON DIOXIDE, CHANNEL, RH PROTEIN, CO2, TRANSPORT PROTEIN
3mqt:U (LYS67) to (LEU117) CRYSTAL STRUCTURE OF A MANDELATE RACEMASE/MUCONATE LACTONIZING ENZYME FROM SHEWANELLA PEALEANA | PSI-II, NYSGXRC, MANDELATE RACEMASE, MUCONATE LACTONIZING ENZYME, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, ISOMERASE
4bl3:A (LYS28) to (GLY74) CRYSTAL STRUCTURE OF PBP2A CLINICAL MUTANT N146K FROM MRSA | HYDROLASE, MRSA, ALLOSTERIC SITE, B-LACTAM ANTIBIOTICS
4bl3:B (LYS28) to (GLY74) CRYSTAL STRUCTURE OF PBP2A CLINICAL MUTANT N146K FROM MRSA | HYDROLASE, MRSA, ALLOSTERIC SITE, B-LACTAM ANTIBIOTICS
4qvg:D (TYR111) to (SER158) CRYSTAL STRUCTURE OF S-ADENOSYLMETHIONINE-DEPENDENT METHYLTRANSFERASE SIBL IN ITS APO FORM | METHYLTRANSFERASE, TRANSFERASE
5f0a:A (ARG260) to (THR303) CRYSTAL STRUCTURE OF PVX_084705 WITH BOUND 1-TERT-BUTYL-3-(3- CHLOROPHENOXY)-1H-PYRAZOLO[3,4-D]PYRIMIDIN-4-AMINE INHIBITOR | STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4boz:A (ALA160) to (ARG215) STRUCTURE OF OTUD2 OTU DOMAIN IN COMPLEX WITH K11-LINKED DI UBIQUITIN | HYDROLASE
4bzb:A (CYS205) to (ILE272) CRYSTAL STRUCTURE OF THE TETRAMERIC DGTP-BOUND SAMHD1 MUTANT CATALYTIC CORE | HYDROLASE, HIV RESTRICTION FACTOR, DNTPASE
4bzb:C (CYS205) to (ILE272) CRYSTAL STRUCTURE OF THE TETRAMERIC DGTP-BOUND SAMHD1 MUTANT CATALYTIC CORE | HYDROLASE, HIV RESTRICTION FACTOR, DNTPASE
4bzb:D (CYS205) to (ILE272) CRYSTAL STRUCTURE OF THE TETRAMERIC DGTP-BOUND SAMHD1 MUTANT CATALYTIC CORE | HYDROLASE, HIV RESTRICTION FACTOR, DNTPASE
4bzc:A (PHE165) to (GLY258) CRYSTAL STRUCTURE OF THE TETRAMERIC DGTP-BOUND WILD TYPE SAMHD1 CATALYTIC CORE | HYDROLASE, HIV RESTRICTION FACTOR, DNTPASE
3c9b:B (LEU18) to (ILE83) CRYSTAL STRUCTURE OF SEMET VPS75 | CHROMATIN, HAT, HISTONE CHAPERONE, NUCLEUS, PHOSPHOPROTEIN, PROTEIN TRANSPORT, TRANSPORT, CHAPERONE
3cem:A (ARG714) to (PHE766) HUMAN GLYCOGEN PHOSPHORYLASE (TENSE STATE) IN COMPLEX WITH THE ALLOSTERIC INHIBITOR AVE9423 | PROTEIN LIGAND COMPLEX, TENSE STATE, ALLOSTERIC INHIBITOR, ALLOSTERIC ENZYME, CARBOHYDRATE METABOLISM, DISEASE MUTATION, GLYCOGEN METABOLISM, GLYCOGEN STORAGE DISEASE, GLYCOSYLTRANSFERASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PYRIDOXAL PHOSPHATE, TRANSFERASE
4rdq:A (ASP104) to (GLY161) CALCIUM-ACTIVATED CHLORIDE CHANNEL BESTROPHIN-1, FROM CHICKEN, IN COMPLEX WITH FAB ANTIBODY FRAGMENTS, CHLORIDE AND CALCIUM | TRANSMEMBRANE PROTEIN, MEMBRANE PROTEIN, ION CHANNEL, CALCIUM- ACTIVATED CHLORIDE CHANNEL, CACC, ANION CHANNEL, MEMBRANE, TRANSPORT PROTEIN
4rdq:B (ASP104) to (GLY161) CALCIUM-ACTIVATED CHLORIDE CHANNEL BESTROPHIN-1, FROM CHICKEN, IN COMPLEX WITH FAB ANTIBODY FRAGMENTS, CHLORIDE AND CALCIUM | TRANSMEMBRANE PROTEIN, MEMBRANE PROTEIN, ION CHANNEL, CALCIUM- ACTIVATED CHLORIDE CHANNEL, CACC, ANION CHANNEL, MEMBRANE, TRANSPORT PROTEIN
4rdq:C (ASP104) to (GLY161) CALCIUM-ACTIVATED CHLORIDE CHANNEL BESTROPHIN-1, FROM CHICKEN, IN COMPLEX WITH FAB ANTIBODY FRAGMENTS, CHLORIDE AND CALCIUM | TRANSMEMBRANE PROTEIN, MEMBRANE PROTEIN, ION CHANNEL, CALCIUM- ACTIVATED CHLORIDE CHANNEL, CACC, ANION CHANNEL, MEMBRANE, TRANSPORT PROTEIN
4rdq:D (ASP104) to (GLY161) CALCIUM-ACTIVATED CHLORIDE CHANNEL BESTROPHIN-1, FROM CHICKEN, IN COMPLEX WITH FAB ANTIBODY FRAGMENTS, CHLORIDE AND CALCIUM | TRANSMEMBRANE PROTEIN, MEMBRANE PROTEIN, ION CHANNEL, CALCIUM- ACTIVATED CHLORIDE CHANNEL, CACC, ANION CHANNEL, MEMBRANE, TRANSPORT PROTEIN
4rdq:E (ASP104) to (GLY161) CALCIUM-ACTIVATED CHLORIDE CHANNEL BESTROPHIN-1, FROM CHICKEN, IN COMPLEX WITH FAB ANTIBODY FRAGMENTS, CHLORIDE AND CALCIUM | TRANSMEMBRANE PROTEIN, MEMBRANE PROTEIN, ION CHANNEL, CALCIUM- ACTIVATED CHLORIDE CHANNEL, CACC, ANION CHANNEL, MEMBRANE, TRANSPORT PROTEIN
4c2p:A (LEU375) to (GLY474) CRYSTAL STRUCTURE OF HUMAN TESTIS ANGIOTENSIN-I CONVERTING ENZYME MUTANT R522K IN COMPLEX WITH CAPTOPRIL | HYDROLASE, CHLORIDE ACTIVATION, HYPERTENSION
3ng6:B (ASP5) to (ASN57) THE CRYSTAL STRUCTURE OF HEMOGLOBIN I FROM TREMATOMUS NEWNESI IN DEOXYGENATED STATE OBTAINED THROUGH AN OXIDATION/REDUCTION CYCLE IN WHICH POTASSIUM HEXACYANOFERRATE AND SODIUM DITHIONITE WERE ALTERNATIVELY ADDED | ROOT EFFECT, FISH HEMOGLOBIN, ANTARCTIC FISH, OXYGEN TRANSPORT
4ca7:A (THR358) to (LEU436) DROSOPHILA ANGIOTENSIN CONVERTING ENZYME (ANCE) IN COMPLEX WITH A PHOSPHINIC TRIPEPTIDE FI | HYDROLASE, ZINC METALLOPEPTIDASE, INHIBITOR BINDING
4ca8:A (THR358) to (LEU436) DROSOPHILA ANGIOTENSIN CONVERTING ENZYME (ANCE) IN COMPLEX WITH A PHOSPHINIC TRIPEPTIDE FII | HYDROLASE, ZINC METALLOPEPTIDASE, INHIBITOR BINDING
4cbb:A (SER42) to (LEU119) APO FORM OF BETAINE ALDEHYDE DEHYDROGENASE FROM PSEUDOMONAS AERUGINOSA | OXIDOREDUCTASE, ALDEHYDE OXIDATION
4cbb:B (SER42) to (LEU119) APO FORM OF BETAINE ALDEHYDE DEHYDROGENASE FROM PSEUDOMONAS AERUGINOSA | OXIDOREDUCTASE, ALDEHYDE OXIDATION
4cjn:A (LYS28) to (LEU73) CRYSTAL STRUCTURE OF PBP2A FROM MRSA IN COMPLEX WITH QUINAZOLINONE LIGAND | HYDROLASE, IMMUNE SYSTEM, ALLOSTERIC SITE
4rxr:A (ARG164) to (GLY258) THE STRUCTURE OF GTP-DCTP-BOUND SAMHD1 | HD-DOMAIN, HYDROLASE, DNTP AND GTP BINDING, PHOSPHORYLATION
4rxr:B (ARG164) to (GLY258) THE STRUCTURE OF GTP-DCTP-BOUND SAMHD1 | HD-DOMAIN, HYDROLASE, DNTP AND GTP BINDING, PHOSPHORYLATION
3o65:C (CYS15) to (GLN65) CRYSTAL STRUCTURE OF A JOSEPHIN-UBIQUITIN COMPLEX: EVOLUTIONARY RESTRAINTS ON ATAXIN-3 DEUBIQUITINATING ACTIVITY | PAPAIN-LIKE FOLD, UBIQUITIN THIOLESTERASE, HYDROLASE-PROTEIN BINDING COMPLEX
4s1b:A (ALA522) to (HIS592) CRYSTAL STRUCTURE OF L. MONOCYTOGENES PHOSPHODIESTERASE PGPH HD DOMAIN IN COMPLEX WITH CYCLIC-DI-AMP | C-DI-AMP, LISTERIA MONOCYTOGENES, PHOSPHODIESTERASE, HD DOMAIN, HYDROLASE
3ob4:A (GLU1086) to (ASN1132) MBP-FUSION PROTEIN OF THE MAJOR PEANUT ALLERGEN ARA H 2 | ALPHA-AMYLASE INHIBITORS (AAI), LIPID TRANSFER (LT) AND SEED STORAGE (SS) PROTEIN FAMILY, SEED STORAGE PROTEIN, ALLERGEN, FUSION PROTEIN, CHIMERA PROTEIN
3d9v:B (SER6) to (LEU69) CRYSTAL STRUCTURE OF ROCK I BOUND TO H-1152P A DI- METHYLATED VARIANT OF FASUDIL | DIMER, DIMERIZATION, KINASE, PHOSPHORYLATION, FASUDIL, APOPTOSIS, ATP-BINDING, COILED COIL, CYTOPLASM, GOLGI APPARATUS, MEMBRANE, METAL-BINDING, NUCLEOTIDE-BINDING, PHORBOL-ESTER BINDING, PHOSPHOPROTEIN, POLYMORPHISM, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ZINC, ZINC- FINGER
4tnr:C (ARG164) to (GLY258) STRUCTURE BASIS OF CELLULAR DNTP REGULATION, SAMHD1-GTP-DATP-DATP COMPLEX | SAMHD1, HIV, RESTRICTION FACTOR, DNTPASE, DNTP REGULATION, HOST PATHOGEN INTERACTION
4tnr:B (ARG164) to (GLY258) STRUCTURE BASIS OF CELLULAR DNTP REGULATION, SAMHD1-GTP-DATP-DATP COMPLEX | SAMHD1, HIV, RESTRICTION FACTOR, DNTPASE, DNTP REGULATION, HOST PATHOGEN INTERACTION
4tnr:A (ARG164) to (GLY258) STRUCTURE BASIS OF CELLULAR DNTP REGULATION, SAMHD1-GTP-DATP-DATP COMPLEX | SAMHD1, HIV, RESTRICTION FACTOR, DNTPASE, DNTP REGULATION, HOST PATHOGEN INTERACTION
4tnx:A (ARG164) to (GLY258) STRUCTURE BASIS OF CELLULAR DNTP REGULATION, SAMHD1-GTP-DGTP COMPLEX | SAMHD1, HIV, RESTRICTION FACTOR, DNTPASE, DNTP REGULATION, HOST PATHOGEN INTERACTION
4tny:A (ARG164) to (GLY258) STRUCTURAL BASIS OF CELLULAR DNTP REGULATION, SAMHD1-DGTP-DATP-DGTP COMPLEX | SAMHD1, HIV, RESTRICTION FACTOR, DNTPASE, DNTP REGULATION, HOST PATHOGEN INTERACTION
4tny:B (ARG164) to (GLY258) STRUCTURAL BASIS OF CELLULAR DNTP REGULATION, SAMHD1-DGTP-DATP-DGTP COMPLEX | SAMHD1, HIV, RESTRICTION FACTOR, DNTPASE, DNTP REGULATION, HOST PATHOGEN INTERACTION
4tnz:C (ARG164) to (GLY258) STRUCTURE BASIS OF CELLULAR DNTP REGULATION, SAMHD1-GTP-DATP-DTTP COMPLEX | SAMHD1, HIV, RESTRICTION FACTOR, DNTPASE, DNTP REGULATION, HOST PATHOGEN INTERACTION
4to1:D (PHE213) to (GLN271) STRUCTURE BASIS OF CELLULAR DNTP REGULATION, SAMHD1-GTP-DATP/DCTP-DCTP COMPLEX | SAMHD1, HIV, RESTRICTION FACTOR, DNTPASE, DNTP REGULATION, HOST PATHOGEN INTERACTION
3dd1:B (ARG714) to (PHE766) CRYSTAL STRUCTURE OF GLYCOGEN PHOPHORYLASE COMPLEXED WITH AN ANTHRANILIMIDE BASED INHIBITOR GSK254 | GLYCOGEN PHOSPHORYLASE HLGP, DIABETES, ALLOSTERIC ENZYME, CARBOHYDRATE METABOLISM, DISEASE MUTATION, GLYCOGEN METABOLISM, GLYCOGEN STORAGE DISEASE, GLYCOSYLTRANSFERASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PYRIDOXAL PHOSPHATE, TRANSFERASE
4tpm:A (ASN562) to (THR623) CRYSTAL STRUCTURE OF 2-(3-ALKOXY-1-AZETIDINYL) QUINOLINES AS PDE10A INHIBITORS | PDE10A, QUINOLINES, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4tpm:B (ASN562) to (THR623) CRYSTAL STRUCTURE OF 2-(3-ALKOXY-1-AZETIDINYL) QUINOLINES AS PDE10A INHIBITORS | PDE10A, QUINOLINES, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4tpp:B (ASN562) to (THR623) 2-(3-ALKOXY-1-AZETIDINYL) QUINOLINES AS NOVEL PDE10A INHIBITORS | PHOSPHODIESTERASE 10A, QUINOLINES, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4d08:B (ASN705) to (ALA767) PDE2A CATALYTIC DOMAIN IN COMPLEX WITH A BRAIN PENETRANT INHIBITOR | HYDROLASE, BINDING SITES, CATALYTIC DOMAIN, CYCLIC NUCLEOTIDE PHOSPHODIESTERASES, TYPE 2, TYPE 4, DISEASE MODELS, ANIMAL, DRUG EVALUATION, PRECLINICAL, PHOSPHODIESTERASE 2 INHIBITORS, PHOSPHODIESTERASE INHIBITORS, PROTEIN BINDING, STRUCTURE-ACTIVITY RELATIONSHIP
4trq:E (GLN293) to (LYS337) CRYSTAL STRUCTURE OF SAC3/THP1/SEM1 | PCI DOMAIN, TREX-2, GENE EXPRESSION, GENE REGULATION
4d09:C (ASN705) to (THR768) PDE2A CATALYTIC DOMAIN IN COMPLEX WITH A BRAIN PENETRANT INHIBITOR | HYDROLASE, CYCLIC NUCLEOTIDE PHOSPHODIESTERASES, TYPE 2, TYPE 4, DISEASE MODELS, ANIMAL, DRUG EVALUATION, PRECLINICAL, PHOSPHODIESTERASE 2 INHIBITORS, PHOSPHODIESTERASE INHIBITORS, PROTEIN BINDING, STRUCTURE-ACTIVITY RELATIONSHIP
3ok5:A (GLY1) to (MET49) STRUCTURE OF THE H55D MUTANT OF DEHALOPEROXIDASE-HEMOGLOBIN A FROM AMPHITRITI ORNATA WITH 4-BROMOPHENOL INHIBITOR | GLOBIN, PEROXIDASE, DEHALOPEROXIDASE, OXIDOREDUCTASE
5gpb:A (VAL715) to (MET766) COMPARISON OF THE BINDING OF GLUCOSE AND GLUCOSE-1-PHOSPHATE DERIVATIVES TO T-STATE GLYCOGEN PHOSPHORYLASE B | GLYCOGEN PHOSPHORYLASE
5gpk:A (GLN33) to (GLU74) CRYSTAL STRUCTURE OF CCP1 MUTANT | CCP1 DIMER, NUCLEOSOME ASSEMBLY PROTEIN, CHAPERONE
5gpl:A (GLN33) to (GLU74) CRYSTAL STRUCTURE OF CCP1 | CCP1 DIMER, NUCLEOSOME ASSEMBLY PROTEIN, CHAPERONE
5gpl:B (PHE32) to (LEU73) CRYSTAL STRUCTURE OF CCP1 | CCP1 DIMER, NUCLEOSOME ASSEMBLY PROTEIN, CHAPERONE
4d5c:A (PHE110) to (LEU203) TETRACYCLINE REPRESSOR CLASS J, APO FORM | TRANSCRIPTION, INDUCTION, ALLOSTERY
4tyw:A (GLU509) to (SER557) DEAD-BOX HELICASE MSS116 BOUND TO SSRNA AND ADP-BEF | DEAD-BOX, RNA HELICASE, HYDROLASE, RNA BINDING PROTEIN-RNA COMPLEX
3dr9:A (GLY1) to (MET49) INCREASED DISTAL HISTIDINE CONFORMATIONAL FLEXIBILITY IN THE DEOXY FORM OF DEHALOPEROXIDASE FROM AMPHITRITE ORNATA | DEOXY FORM OF DEHALOPEROXIDASE, DHP, HEME PEROXIDASE, GLOBIN-LIKE, GLOBIN, HEME PROTEIN, HEME, OXYGEN TRANSPORT, PEROXIDASE, TRANSPORT, OXIDOREDUCTASE
3os8:A (THR311) to (SER395) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
3os8:B (THR311) to (SER395) ESTROGEN RECEPTOR | ESTROGEN RECEPTOR COMPLEX, SIGNALING PROTEIN
4ddl:A (ASN562) to (THR623) PDE10A CRYSTAL STRUCTURE COMPLEXED WITH NOVEL INHIBITOR | PHOSPHODIESTERASE 10A, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4ddl:B (ASN562) to (THR623) PDE10A CRYSTAL STRUCTURE COMPLEXED WITH NOVEL INHIBITOR | PHOSPHODIESTERASE 10A, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4dff:A (SER571) to (THR633) THE SAR DEVELOPMENT OF DIHYDROIMIDAZOISOQUINOLINE DERIVATIVES AS PHOSPHODIESTERASE 10A INHIBITORS FOR THE TREATMENT OF SCHIZOPHRENIA | ZN BINDING, MG BINDING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4dhj:L (THR152) to (ILE206) THE STRUCTURE OF A CEOTUB1 UBIQUITIN ALDEHYDE UBC13~UB COMPLEX | UBIQUITINATION, HYDROLASE-SIGNALING PROTEIN-LIGASE COMPLEX
4dji:B (GLY270) to (THR359) STRUCTURE OF GLUTAMATE-GABA ANTIPORTER GADC | LEUT FOLD, GLUTAMATE-GABA ANTIPORTER, TRANSPORT PROTEIN
4djk:A (GLY270) to (THR359) STRUCTURE OF GLUTAMATE-GABA ANTIPORTER GADC | LEUT, GLUTAMATE-GABA ANTIPORTER, TRANSPORT PROTEIN
3dzx:A (LEU420) to (ASN471) CRYSTAL STRUCTURE OF THE RABGAP DOMAIN OF HUMAN TBC1D22B | RAB-GAP, GTPASE ACTIVATOR, TBC1, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, GTPASE ACTIVATION, SIGNALING PROTEIN, HYDROLASE ACTIVATOR
3e3l:B (ARG714) to (MET766) THE R-STATE GLYCOGEN PHOSPHORYLASE | GLYCOGENOLYSIS, INHIBITION, TYPE 2 DIABETES, ALLOSTERIC ENZYME, CARBOHYDRATE METABOLISM, GLYCOGEN METABOLISM, GLYCOSYLTRANSFERASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PYRIDOXAL PHOSPHATE, TRANSFERASE
3e3n:H (ARG714) to (MET766) THE GLYCOGEN PHOSPHORYLASE B R STATE- AMP COMPLEX | GLYCOGENOLYSIS, INHIBITION, TYPE 2 DIABETES, ALLOSTERIC ENZYME, CARBOHYDRATE METABOLISM, GLYCOGEN METABOLISM, GLYCOSYLTRANSFERASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PYRIDOXAL PHOSPHATE, TRANSFERASE
4dsh:B (ASN105) to (PHE152) CRYSTAL STRUCTURE OF REDUCED UDP-GALACTOPYRANOSE MUTASE | ROSSMANN FOLD, FLAVIN ADENINE DINUCLEOTIDE, ISOMERASE
5i1u:A (ILE50) to (GLY107) CRYSTAL STRUCTURE OF GERMACRADIEN-4-OL SYNTHASE FROM STREPTOMYCES CITRICOLOR | LYASE, SESQUITERPENE CYCLASE
5i2r:A (ASN572) to (THR633) HUMAN PDE10A IN COMPLEX WITH 3-(2-PHENYLPYRAZOL-3-YL)-1-[3- (TRIFLUOROMETHOXY)PHENYL]PYRIDAZIN-4-ONE | PHOSPHODIESTERASE, PDE10, HYDROLASE
5i2r:B (ASN572) to (THR633) HUMAN PDE10A IN COMPLEX WITH 3-(2-PHENYLPYRAZOL-3-YL)-1-[3- (TRIFLUOROMETHOXY)PHENYL]PYRIDAZIN-4-ONE | PHOSPHODIESTERASE, PDE10, HYDROLASE
5i2r:C (ASN572) to (THR633) HUMAN PDE10A IN COMPLEX WITH 3-(2-PHENYLPYRAZOL-3-YL)-1-[3- (TRIFLUOROMETHOXY)PHENYL]PYRIDAZIN-4-ONE | PHOSPHODIESTERASE, PDE10, HYDROLASE
5i2r:D (SER571) to (ALA632) HUMAN PDE10A IN COMPLEX WITH 3-(2-PHENYLPYRAZOL-3-YL)-1-[3- (TRIFLUOROMETHOXY)PHENYL]PYRIDAZIN-4-ONE | PHOSPHODIESTERASE, PDE10, HYDROLASE
3pjw:A (ASP276) to (THR315) STRUCTURE OF PSEUDOMONAS FLUORESCENCE LAPD GGDEF-EAL DUAL DOMAIN, I23 | GGDEF-EAL TANDEM DOMAIN, C-DI-GMP RECEPTOR, LYASE
5i6c:A (SER450) to (MET542) THE STRUCTURE OF THE EUKARYOTIC PURINE/H+ SYMPORTER, UAPA, IN COMPLEX WITH XANTHINE | MEMBRANE PROTEIN EUKARYOTIC URIC ACID/XANTHINE H+ SYMPORTER, TRANSPORT PROTEIN
5i6c:B (PRO448) to (ILE541) THE STRUCTURE OF THE EUKARYOTIC PURINE/H+ SYMPORTER, UAPA, IN COMPLEX WITH XANTHINE | MEMBRANE PROTEIN EUKARYOTIC URIC ACID/XANTHINE H+ SYMPORTER, TRANSPORT PROTEIN
5i6x:A (SER404) to (THR482) X-RAY STRUCTURE OF THE TS3 HUMAN SEROTONIN TRANSPORTER COMPLEXED WITH PAROXETINE AT THE CENTRAL SITE | MEMBRANE PROTEIN
5i73:A (SER404) to (THR482) X-RAY STRUCTURE OF THE TS3 HUMAN SEROTONIN TRANSPORTER COMPLEXED WITH S-CITALOPRAM AT THE CENTRAL AND ALLOSTERIC SITES | MEMBRANE PROTEIN
5i82:A (PRO225) to (VAL288) FIRST CRYSTAL STRUCTURE OF E.COLI BASED RECOMBINANT DIPHTHERIA TOXIN MUTANT CRM197 | DIPHTHERIA TOXIN, CRM197, CSGID, RECOMBINANT, STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, TRANSFERASE
5i82:B (GLY224) to (VAL288) FIRST CRYSTAL STRUCTURE OF E.COLI BASED RECOMBINANT DIPHTHERIA TOXIN MUTANT CRM197 | DIPHTHERIA TOXIN, CRM197, CSGID, RECOMBINANT, STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, TRANSFERASE
5i82:D (PRO225) to (VAL288) FIRST CRYSTAL STRUCTURE OF E.COLI BASED RECOMBINANT DIPHTHERIA TOXIN MUTANT CRM197 | DIPHTHERIA TOXIN, CRM197, CSGID, RECOMBINANT, STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, TRANSFERASE
4us4:A (ALA77) to (ASN145) CRYSTAL STRUCTURE OF THE BACTERIAL NSS MEMBER MHST IN AN OCCLUDED INWARD-FACING STATE (LIPIDIC CUBIC PHASE FORM) | TRANSPORT PROTEIN, NEUROTRANSMITTER, NEUROTRANSMITTER SODIUM SYMPORTER FAMILY, LEUT FOLD, AMINO ACID TRANSPORTER, SECONDARY TRANSPORTER, MEMBRANE PROTEIN
5ik2:E (SER348) to (SER386) CALDALAKLIBACILLUS THERMARUM F1-ATPASE (EPSILON MUTANT) | HYDROLASE, F1-ATPASE, COMPLEX
5ik2:M (SER348) to (SER386) CALDALAKLIBACILLUS THERMARUM F1-ATPASE (EPSILON MUTANT) | HYDROLASE, F1-ATPASE, COMPLEX
3q33:B (VAL25) to (ILE83) STRUCTURE OF THE RTT109-ACCOA/VPS75 COMPLEX AND IMPLICATIONS FOR CHAPERONE-MEDIATED HISTONE ACETYLATION | RTT109:VPS75=2:2 STOICHIOMETRY COMPLEX, HISTONE ACETYLTRANSFERASE, WITH ACETYL COENZYME A (ACOA) BOUND, AUTOACETYLATION ON RTT109 LYS290, NUCLEAR, TRANSFERASE-CHAPERONE-TRANSCRIPTION REGULATOR COMPLEX, TRANSFERASE-CHAPERONE COMPLEX, TRANSFERASE,CHAPERONE-GENE REGULATION COMPLEX, TRANSFERASE, CHAPERONE-GENE REGULATION COMPLEX
3q35:B (GLU10) to (ILE83) STRUCTURE OF THE RTT109-ACCOA/VPS75 COMPLEX AND IMPLICATIONS FOR CHAPERONE-MEDIATED HISTONE ACETYLATION | RTT109:VPS75=2:2 STOICHIOMETRY COMPLEX, ACETYL COENZYME A (ACOA) BOUND, AUTOACETYLATION AT RTT109 LYS290, NUCLEAR, TRANSFERASE- CHAPERONE COMPLEX
3q66:B (ASN9) to (ILE83) STRUCTURE OF THE VPS75-RTT109 HISTONE CHAPERONE-LYSINE ACETYLTRANSFERASE COMPLEX (FULL-LENGTH PROTEINS IN SPACE GROUP P6122) | HISTONE CHAPERONE, LYSINE ACETYLTRANSFERASE, CHAPERONE-TRANSFERASE COMPLEX
4fcb:A (SER561) to (THR623) POTENT AND SELECTIVE PHOSPHODIESTERASE 10A INHIBITORS | BINDING SITES, CYCLIC AMP, CYCLIC GMP,LIGANDS, PHOSPHODIESTERASE INHIBITORS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4fcd:A (SER561) to (THR623) POTENT AND SELECTIVE PHOSPHODIESTERASE 10A INHIBITORS | BINDING SITES, CYCLIC AMP, CYCLIC GMP, HUMANS, HYDROLYSIS, LIGANDS, PHOSPHODIESTERASE INHIBITORS, PHOSPHORIC DIESTER HYDROLASES, RECOMBINANT PROTEINS, STRUCTURE-ACTIVITY RELATIONSHIP, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3qpn:A (SER561) to (THR623) STRUCTURE OF PDE10-INHIBITOR COMPLEX | PHOSPHODIESTERASE INHIBITORS, STRUCTURE-BASED DRUG DESIGN, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3qpo:A (ASN562) to (THR623) STRUCTURE OF PDE10-INHIBITOR COMPLEX | PHOSPHODIESTERASE INHIBITORS, STRUCTURE-BASED DRUG DESIGN, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3qwl:A (PRO216) to (ASN265) CRYSTAL STRUCTURE OF HUMAN TBC1 DOMAIN FAMILY MEMBER 7 | RAB GTPASE ACTIVATION, STRUCTURAL GENOMICS CONSORTIUM, TBC DOMAIN, SGC, HYDROLASE ACTIVATOR
4fp9:B (GLU252) to (SER327) HUMAN MTERF4-NSUN4 PROTEIN COMPLEX | MODIFICATION ENZYME, TRANSFERASE
4fp9:E (GLU252) to (SER327) HUMAN MTERF4-NSUN4 PROTEIN COMPLEX | MODIFICATION ENZYME, TRANSFERASE
4fp9:G (GLU252) to (SER327) HUMAN MTERF4-NSUN4 PROTEIN COMPLEX | MODIFICATION ENZYME, TRANSFERASE
4fp9:H (GLU252) to (SER327) HUMAN MTERF4-NSUN4 PROTEIN COMPLEX | MODIFICATION ENZYME, TRANSFERASE
5jj6:B (ILE328) to (HIS404) FIC-1 (AA134 - 508) FROM C. ELEGANS | AMPYLASE, TRANSFERASE
4fzv:B (GLU252) to (GLU328) CRYSTAL STRUCTURE OF THE HUMAN MTERF4:NSUN4:SAM TERNARY COMPLEX | MTERF FOLD, METHYLTRANSFERASE FOLD, RRNA METHYLTRANSFERASE, MITOCHONDRIA, TRANSFERASE
4g21:A (TYR179) to (ALA295) STRUCTURAL BASIS FOR THE ACCOMMODATION OF BIS- AND TRIS-AROMATIC DERIVATIVES IN VITAMIN D NUCLEAR RECEPTOR | VDR, TRANSCRIPTION REGULATION, NUCLEAR RECEPTOR, ALPHA HELICAL SANDWICH, LIGAND, DNA, PHOSPHORYLATION, NUCLEUS, TRANSCRIPTION- TRANSCRIPTION INHIBITOR COMPLEX
4g51:D (ASP5) to (ASN57) CRYSTALLOGRAPHIC ANALYSIS OF THE INTERACTION OF NITRIC OXIDE WITH HEMOGLOBIN FROM TREMATOMUS BERNACCHII IN THE T QUATERNARY STRUCTURE (FULLY LIGATED STATE). | ALL ALPHA PROTEINS, OXYGEN TRANSPORTER, N-TERMINAL ACETYLATED SERINE, OXYGEN TRANSPORT
5k3i:A (PRO62) to (GLU104) CRYSTAL STRUCTURE OF ACYL-COA OXIDASE-1 IN CAENORHABDITIS ELEGANS COMPLEXED WITH FAD AND ATP | DAUER PHEROMONE, ASCAROSIDES, B-OXIDATION, ATP, OXIDOREDUCTASE
5k3i:B (PRO62) to (LEU106) CRYSTAL STRUCTURE OF ACYL-COA OXIDASE-1 IN CAENORHABDITIS ELEGANS COMPLEXED WITH FAD AND ATP | DAUER PHEROMONE, ASCAROSIDES, B-OXIDATION, ATP, OXIDOREDUCTASE
5k3i:H (PRO62) to (GLY107) CRYSTAL STRUCTURE OF ACYL-COA OXIDASE-1 IN CAENORHABDITIS ELEGANS COMPLEXED WITH FAD AND ATP | DAUER PHEROMONE, ASCAROSIDES, B-OXIDATION, ATP, OXIDOREDUCTASE
5k9r:A (SER561) to (THR623) PDE10A WITH IMIDAZOPYRAZINE INHIBITOR | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5k9r:B (SER561) to (THR623) PDE10A WITH IMIDAZOPYRAZINE INHIBITOR | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4gbv:A (THR12) to (SER88) CRYSTAL STRUCTURE OF AMP COMPLEXES OF PORCINE LIVER FRUCTOSE-1,6- BISPHOSPHATASE MUTANT A54L WITH 1,2-ETHANEDIOL AS CRYO-PROTECTANT | ALLOSTERIC ENZYMES, FBPASE, AMP, 1,2-ETHANEDIOL, HYDROLASE
5kcu:B (THR311) to (SER395) CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH AN N-ETHYL, ALPHA-NAPHTHYL OBHS-N DERIVATIVE | NUCLEAR RECEPTOR, TRANSCRIPTION FACTOR, LIGAND BINDING, PROTEIN- LIGAND COMPLEX, TRANSCRIPTION
4gfj:A (ARG351) to (GLU393) CRYSTAL STRUCTURE OF TOPO-78, AN N-TERMINAL 78KDA FRAGMENT OF TOPOISOMERASE V | HELIX-HAIRPIN-HELIX, DNA REPAIR ENZYME, TOPOISOMERASE, DNA BINDING, ISOMERASE
4ghk:D (ILE3) to (LEU91) X-RAY CRYSTAL STRUCTURE OF GAMMA-GLUTAMYL PHOSPHATE REDUCTASE FROM BURKHOLDERIA THAILANDENSIS | STRUCTURAL GENOMICS, NIAID, NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, SSGCID, GAMMA-GLUTAMYL PHOSPHATE REDUCTASE, OXIDOREDUCTASE
5l11:A (ASP314) to (CYS381) HUMAN LIVER RECEPTOR HOMOLOGUE-1 (LRH-1) BOUND TO RJW100 AND A FRAGMENT OF TIF-2 | NUCLEAR RECEPTOR, AGONIST, TRANSCRIPTION-INHIBITOR COMPLEX
5syz:A (ASP314) to (CYS381) HUMAN LIVER RECEPTOR HOMOLOGUE-1 (LRH-1) BOUND TO A RJW100 STEREOISOMER AND A FRAGMENT OF TIF-2 | NUCLEAR RECEPTOR, AGONIST, COACTIVATOR, NUCLEAR PROTEIN
5t5n:A (ASP104) to (GLY161) CALCIUM-ACTIVATED CHLORIDE CHANNEL BESTROPHIN-1 (BEST1), TRIPLE MUTANT: I76A, F80A, F84A; IN COMPLEX WITH AN FAB ANTIBODY FRAGMENT, CHLORIDE, AND CALCIUM | ION CHANNEL, ANION, CHLORIDE, CALCIUM-ACTIVATED, EUKARYOTIC MEMBRANE PROTEIN, CACC, MEMBRANE PROTEIN
5t5n:B (ASP104) to (GLY161) CALCIUM-ACTIVATED CHLORIDE CHANNEL BESTROPHIN-1 (BEST1), TRIPLE MUTANT: I76A, F80A, F84A; IN COMPLEX WITH AN FAB ANTIBODY FRAGMENT, CHLORIDE, AND CALCIUM | ION CHANNEL, ANION, CHLORIDE, CALCIUM-ACTIVATED, EUKARYOTIC MEMBRANE PROTEIN, CACC, MEMBRANE PROTEIN
5t5n:C (ASP104) to (GLY161) CALCIUM-ACTIVATED CHLORIDE CHANNEL BESTROPHIN-1 (BEST1), TRIPLE MUTANT: I76A, F80A, F84A; IN COMPLEX WITH AN FAB ANTIBODY FRAGMENT, CHLORIDE, AND CALCIUM | ION CHANNEL, ANION, CHLORIDE, CALCIUM-ACTIVATED, EUKARYOTIC MEMBRANE PROTEIN, CACC, MEMBRANE PROTEIN
5t5n:D (ASP104) to (GLY161) CALCIUM-ACTIVATED CHLORIDE CHANNEL BESTROPHIN-1 (BEST1), TRIPLE MUTANT: I76A, F80A, F84A; IN COMPLEX WITH AN FAB ANTIBODY FRAGMENT, CHLORIDE, AND CALCIUM | ION CHANNEL, ANION, CHLORIDE, CALCIUM-ACTIVATED, EUKARYOTIC MEMBRANE PROTEIN, CACC, MEMBRANE PROTEIN
5t5n:E (ASP104) to (GLY161) CALCIUM-ACTIVATED CHLORIDE CHANNEL BESTROPHIN-1 (BEST1), TRIPLE MUTANT: I76A, F80A, F84A; IN COMPLEX WITH AN FAB ANTIBODY FRAGMENT, CHLORIDE, AND CALCIUM | ION CHANNEL, ANION, CHLORIDE, CALCIUM-ACTIVATED, EUKARYOTIC MEMBRANE PROTEIN, CACC, MEMBRANE PROTEIN
9gpb:B (GLU716) to (HIS768) THE ALLOSTERIC TRANSITION OF GLYCOGEN PHOSPHORYLASE | GLYCOGEN PHOSPHORYLASE
2amb:A (PRO671) to (TRP741) CRYSTAL STRUCTURE OF HUMAN ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH TETRAHYDROGESTRINONE | NUCLEAR RECEPTOR, ANDROGEN RECEPTOR, LIGAND BINDING DOMAIN, THG, AGONIST, DESIGNER ANDROGEN, HORMONE-GROWTH FACTOR RECEPTOR COMPLEX
3ecn:A (ILE502) to (TYR549) CRYSTAL STRUCTURE OF PDE8A CATALYTIC DOMAIN IN COMPLEX WITH IBMX | IBMX, PDE8A CATALYTIC DOMAIN, REFOLDING, ALTERNATIVE SPLICING, CAMP, HYDROLASE, MAGNESIUM, MANGANESE, METAL- BINDING
2oup:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A | PDE10, HYDROLASE
2ouy:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 MUTANT D564A IN COMPLEX WITH CAMP. | PDE, SUBSTRATE SPECIFICITY, CAMP, HYDROLASE
4wx7:A (ASN144) to (THR196) CRYSTAL STRUCTURE OF ADENOVIRUS 8 PROTEASE WITH A NITRILE INHIBITOR | CYSTEINE PROTEASE, INHIBITOR, COVALENT, HYDROLASE
4wx7:C (ASN144) to (THR196) CRYSTAL STRUCTURE OF ADENOVIRUS 8 PROTEASE WITH A NITRILE INHIBITOR | CYSTEINE PROTEASE, INHIBITOR, COVALENT, HYDROLASE
4hf4:A (SER561) to (THR623) CRYSTAL STRUCTURE OF PDE10A WITH A BIARYL ETHER INHIBITOR (1-(1-(3-(4- (BENZO[D]THIAZOL-2-YLAMINO)PHENOXY)PYRAZIN-2-YL)PIPERIDIN-4-YL) ETHANOL) | PDE10A, PHOSPHODIESTERASE 10A, BIARYL ETHERS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4hf4:B (SER561) to (THR623) CRYSTAL STRUCTURE OF PDE10A WITH A BIARYL ETHER INHIBITOR (1-(1-(3-(4- (BENZO[D]THIAZOL-2-YLAMINO)PHENOXY)PYRAZIN-2-YL)PIPERIDIN-4-YL) ETHANOL) | PDE10A, PHOSPHODIESTERASE 10A, BIARYL ETHERS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4x3q:B (TYR111) to (SER158) CRYSTAL STRUCTURE OF S-ADENOSYLMETHIONINE-DEPENDENT METHYLTRANSFERASE SIBL IN COMPLEX WITH SAH | SIBIROMYCIN BIOSYNTHESIS, SAM-DEPENDENT METHYLTRANSFERASE, C- METHYLATION., LIGASE
4x3q:D (TYR111) to (SER158) CRYSTAL STRUCTURE OF S-ADENOSYLMETHIONINE-DEPENDENT METHYLTRANSFERASE SIBL IN COMPLEX WITH SAH | SIBIROMYCIN BIOSYNTHESIS, SAM-DEPENDENT METHYLTRANSFERASE, C- METHYLATION., LIGASE
1bp3:A (ASN63) to (GLU129) THE XRAY STRUCTURE OF A GROWTH HORMONE-PROLACTIN RECEPTOR COMPLEX | HORMONE, RECEPTOR, HORMONE/GROWTH FACTOR
3ffq:B (ASP487) to (LEU533) HCN2I 443-640 APO-STATE | ION TRANSPORT, ION CHANNEL, MEMBRANE, NUCLEOTIDE-BINDING, POTASSIUM, POTASSIUM CHANNEL, SODIUM CHANNEL, TRANSMEMBRANE, VOLTAGE-GATED CHANNEL, CAMP, CAMP-BINDING, GLYCOPROTEIN, IONIC CHANNEL, PHOSPHOPROTEIN, POTASSIUM TRANSPORT, SODIUM TRANSPORT, TRANSPORT, METAL TRANSPORT
3sl8:A (SER208) to (ASP272) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF PDE4D2 WITH COMPOUND 10O | CATALYTIC MECHANISM, CAMP HYDROLYSIS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2qxs:A (THR311) to (ALA382) CRYSTAL STRUCTURE OF ANTAGONIZING MUTANT 536S OF THE ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN COMPLEXED TO RALOXIFENE | PROTEIN-LIGAND COMPLEX, DNA-BINDING, LIPID-BINDING, METAL-BINDING, NUCLEUS, PHOSPHORYLATION, RECEPTOR, STEROID-BINDING, TRANSCRIPTION, TRANSCRIPTION REGULATION, ZINC-FINGER
3gqp:B (THR4) to (ASN57) CRYSTAL STRUCTURE DETERMINATION OF CAT (FELIS SILVESTRIS CATUS) HEMOGLOBIN AT 2.0 ANGSTROM RESOLUTION | LOW OXYGEN AFFINITY, METHEMOGLOBIN, CHROMATOGRAPHY, MONOCLINIC, HEME, IRON, OXYGEN TRANSPORT, TRANSPORT, POLYMORPHISM, OXYGEN STORAGE
2r9g:C (ASP257) to (LEU308) CRYSTAL STRUCTURE OF THE C-TERMINAL FRAGMENT OF AAA ATPASE FROM ENTEROCOCCUS FAECIUM | STRUCTURAL GENOMICS, ATPASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, HYDROLASE
2r9g:D (ASP257) to (LEU308) CRYSTAL STRUCTURE OF THE C-TERMINAL FRAGMENT OF AAA ATPASE FROM ENTEROCOCCUS FAECIUM | STRUCTURAL GENOMICS, ATPASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, HYDROLASE
2r9g:E (VAL256) to (LEU308) CRYSTAL STRUCTURE OF THE C-TERMINAL FRAGMENT OF AAA ATPASE FROM ENTEROCOCCUS FAECIUM | STRUCTURAL GENOMICS, ATPASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, HYDROLASE
2r9g:F (VAL256) to (LEU308) CRYSTAL STRUCTURE OF THE C-TERMINAL FRAGMENT OF AAA ATPASE FROM ENTEROCOCCUS FAECIUM | STRUCTURAL GENOMICS, ATPASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, HYDROLASE
2r9g:G (VAL256) to (LEU308) CRYSTAL STRUCTURE OF THE C-TERMINAL FRAGMENT OF AAA ATPASE FROM ENTEROCOCCUS FAECIUM | STRUCTURAL GENOMICS, ATPASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, HYDROLASE
2r9g:H (ASP257) to (LEU308) CRYSTAL STRUCTURE OF THE C-TERMINAL FRAGMENT OF AAA ATPASE FROM ENTEROCOCCUS FAECIUM | STRUCTURAL GENOMICS, ATPASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, HYDROLASE
2r9g:I (VAL256) to (LEU308) CRYSTAL STRUCTURE OF THE C-TERMINAL FRAGMENT OF AAA ATPASE FROM ENTEROCOCCUS FAECIUM | STRUCTURAL GENOMICS, ATPASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, HYDROLASE
2r9g:J (VAL256) to (LEU308) CRYSTAL STRUCTURE OF THE C-TERMINAL FRAGMENT OF AAA ATPASE FROM ENTEROCOCCUS FAECIUM | STRUCTURAL GENOMICS, ATPASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, HYDROLASE
2r9g:K (VAL256) to (LEU308) CRYSTAL STRUCTURE OF THE C-TERMINAL FRAGMENT OF AAA ATPASE FROM ENTEROCOCCUS FAECIUM | STRUCTURAL GENOMICS, ATPASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, HYDROLASE
2r9g:L (VAL256) to (LEU308) CRYSTAL STRUCTURE OF THE C-TERMINAL FRAGMENT OF AAA ATPASE FROM ENTEROCOCCUS FAECIUM | STRUCTURAL GENOMICS, ATPASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, HYDROLASE
2r9g:N (ASP257) to (LEU308) CRYSTAL STRUCTURE OF THE C-TERMINAL FRAGMENT OF AAA ATPASE FROM ENTEROCOCCUS FAECIUM | STRUCTURAL GENOMICS, ATPASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, HYDROLASE
2r9g:O (ASP257) to (LEU308) CRYSTAL STRUCTURE OF THE C-TERMINAL FRAGMENT OF AAA ATPASE FROM ENTEROCOCCUS FAECIUM | STRUCTURAL GENOMICS, ATPASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, HYDROLASE
2r9g:P (ASP257) to (LEU308) CRYSTAL STRUCTURE OF THE C-TERMINAL FRAGMENT OF AAA ATPASE FROM ENTEROCOCCUS FAECIUM | STRUCTURAL GENOMICS, ATPASE, PSI-2, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, NYSGXRC, ATP- BINDING, NUCLEOTIDE-BINDING, HYDROLASE
4jib:B (ASN704) to (THR768) CRYSTAL STRUCTURE OF OF PDE2-INHIBITOR COMPLEX | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4jib:C (ASN705) to (THR768) CRYSTAL STRUCTURE OF OF PDE2-INHIBITOR COMPLEX | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4jib:D (ASN704) to (THR768) CRYSTAL STRUCTURE OF OF PDE2-INHIBITOR COMPLEX | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1f99:M (THR3) to (VAL100) CRYSTAL STRUCTURE OF R-PHYCOCYANIN FROM POLYSIPHONIA AT 2.4 A RESOLUTION | LIGHT HARVESTING PROTEIN, R-PHYCOCYANIN, PHOTOSYNTHESIS, ELECTRON TRASNPORT
3ubr:A (ALA94) to (LYS141) LAUE STRUCTURE OF SHEWANELLA ONEIDENSIS CYTOCHROME-C NITRITE REDUCTASE | DECA-HEME, ELECTRON TRANSFER, REDOX, CYMA, OXIDOREDUCTASE
3ubr:B (ALA94) to (LYS141) LAUE STRUCTURE OF SHEWANELLA ONEIDENSIS CYTOCHROME-C NITRITE REDUCTASE | DECA-HEME, ELECTRON TRANSFER, REDOX, CYMA, OXIDOREDUCTASE
2esd:B (THR39) to (MET118) CRYSTAL STRUCTURE OF THIOACYLENZYME INTERMEDIATE OF AN NADP DEPENDENT ALDEHYDE DEHYDROGENASE | ALDH, GAPN, TERNARY COMPLEX, OXIDOREDUCTASE
2esd:C (THR39) to (MET118) CRYSTAL STRUCTURE OF THIOACYLENZYME INTERMEDIATE OF AN NADP DEPENDENT ALDEHYDE DEHYDROGENASE | ALDH, GAPN, TERNARY COMPLEX, OXIDOREDUCTASE
2esd:D (SER38) to (MET118) CRYSTAL STRUCTURE OF THIOACYLENZYME INTERMEDIATE OF AN NADP DEPENDENT ALDEHYDE DEHYDROGENASE | ALDH, GAPN, TERNARY COMPLEX, OXIDOREDUCTASE
3ui7:A (ASN572) to (THR633) DISCOVERY OF ORALLY ACTIVE PYRAZOLOQUINOLINE AS A POTENT PDE10 INHIBITOR FOR THE MANAGEMENT OF SCHIZOPHRENIA | INHIBITOR COMPLEX, HYDROLASE, ZN BINDING, MG BINDING, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3ui7:B (SER571) to (THR633) DISCOVERY OF ORALLY ACTIVE PYRAZOLOQUINOLINE AS A POTENT PDE10 INHIBITOR FOR THE MANAGEMENT OF SCHIZOPHRENIA | INHIBITOR COMPLEX, HYDROLASE, ZN BINDING, MG BINDING, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3hqz:A (ASN562) to (THR623) DISCOVERY OF NOVEL INHIBITORS OF PDE10A | PHOSPHODIESTERASE 10A PDE 10A PDE10 INHIBITORS, ALLOSTERIC ENZYME, ALTERNATIVE SPLICING, CAMP, CAMP-BINDING, CGMP, CGMP-BINDING, CYTOPLASM, HYDROLASE, MAGNESIUM, METAL- BINDING, NUCLEOTIDE-BINDING, ZINC, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1sgk:A (HIS223) to (VAL288) NUCLEOTIDE-FREE DIPHTHERIA TOXIN | TOXIN, ADP-RIBOSYLATION, TRANSFERASE, GLYCOSYLTRANSFERASE, NAD, ADP- RIBOSYL TRANSFERASE
3vjt:A (TYR147) to (SER262) VITAMIN D RECEPTOR COMPLEX WITH A CARBORANE COMPOUND | NUCLEAR RECEPTOR, SYNTHETIC AGONIST, CARBORANE, TRANSCRIPTION
2hb7:A (LEU224) to (SER266) CRYSTAL STRUCTURE OF VDR LBD IN COMPLEX WITH 2ALPHA(3- HYDROXY-1-PROPYL) CALCITRIOL | ALPHA HELICAL SANDWICH, GENE REGULATION
3ixf:A (GLY1) to (MET49) CRYSTAL STRUCTURE OF DEHALOPEROXIDASE B AT 1.58 AND STRUCTURAL CHARACTERIZATION OF THE AB DIMER FROM AMPHITRITE ORNATA | PEROXIDASE, GLOBIN, HEME, OXYGEN TRANSPORT, TRANSPORT, OXIDOREDUCTASE
4llj:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT214 | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4llj:B (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT214 | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4llk:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT217 | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4llx:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT434 | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4lm0:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT448 | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4lm2:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT462 | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4lm3:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT464 | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5a1s:B (PRO27) to (GLY97) CRYSTAL STRUCTURE OF THE SODIUM-DEPENDENT CITRATE SYMPORTER SECITS FORM SALMONELLA ENTERICA. | TRANSPORT PROTEIN, MEMBRANE PROTEIN, SYMPORTER, TRANSPORTER, DI-CARBOXYLATE TRANSPORTER
4lrl:C (SER118) to (LYS165) STRUCTURE OF AN ENTEROCOCCUS FAECALIS HD-DOMAIN PROTEIN COMPLEXED WITH DGTP AND DTTP | STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, HD DOMAIN, PHOSPHOHYDROLASE, DNTPASE, ALLOSTERIC REGULATION, METAL BINDING PROTEIN, HYDROLASE
1i37:A (SER696) to (GLN738) CRYSTAL STRUCTURE OF THE RAT ANDROGEN RECEPTOR LIGAND BINDING DOMAIN COMPLEX WITH DIHYDROTESTOSTERONE | ANDROGEN RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, LIGAND-BINDING DOMAIN, HORMONE/GROWTH FACTOR COMPLEX
2hyd:A (PHE27) to (ASN141) MULTIDRUG ABC TRANSPORTER SAV1866 | TRANSPORT PROTEIN
2hyd:B (PHE27) to (ASN141) MULTIDRUG ABC TRANSPORTER SAV1866 | TRANSPORT PROTEIN
3w5c:A (TRP832) to (TYR949) CRYSTAL STRUCTURE OF THE CALCIUM PUMP IN THE E2 STATE FREE FROM EXOGENOUS INHIBITORS | P-TYPE ATPASE, HYDROLASE, CALCIUM TRANSPORT, CALCIUM BINDING, ATP BINDING, ENDOPLASMIC RETICULUM, SARCOPLASMIC RETICULUM, METAL TRANSPORT
5aav:A (THR311) to (ALA382) OPTIMIZATION OF A NOVEL BINDING MOTIF TO TO (E)-3-(3,5- DIFLUORO-4-((1R,3R)-2-(2-FLUORO-2-METHYLPROPYL)-3-METHYL-2, 3,4,9-TETRAHYDRO-1H-PYRIDO(3,4-B)INDOL-1-YL)PHENYL)ACRYLIC ACID (AZD9496), A POTENT AND ORALLY BIOAVAILABLE SELECTIVE ESTROGEN RECEPTOR DOWNREGULATOR AND ANTAGONIST | SIGNALING PROTEIN, BREAST CANCER, ESTROGEN RECEPTOR DOWNREGULATOR, FULVESTRANT, AZD9496, NUCLEAR HORMONE RECEPTOR
2x90:A (THR358) to (LEU436) CRYSTAL STRUCTURE OF ANCE-ENALAPRILAT COMPLEX | HYDROLASE, ACE INHIBITOR, ZINC METALLOPEPTIDASE
2x93:A (THR358) to (LEU436) CRYSTAL STRUCTURE OF ANCE-TRANDOLAPRILAT COMPLEX | METALLOPROTEASE, CARBOXYPEPTIDASE, ACE INHIBITOR, HYDROLASE, GLYCOPROTEIN
2x96:A (THR358) to (LEU436) CRYSTAL STRUCTURE OF ANCE-RXPA380 COMPLEX | HYDROLASE, ACE INHIBITOR, ZINC METALLOPEPTIDASE
3won:B (GLN430) to (ALA496) CRYSTAL STRUCTURE OF THE DAP BII DIPEPTIDE COMPLEX III | CHYMOTRYPSIN FOLD, S46 PEPTIDASE, HYDROLASE
5ao3:B (PHE213) to (GLY274) CRYSTAL STRUCTURE OF HUMAN SAMHD1 (AMINO ACID RESIDUES 115-626) BOUND TO GTP | HYDROLASE, DEOXYNUCLEOSIDE TRIPHOSPHATE TRIPHOSPHOHYDROLASE, HIV RESTRICTION FACTOR
1vh4:A (ASP369) to (LEU418) CRYSTAL STRUCTURE OF A STABILIZER OF IRON TRANSPORTER | STRUCTURAL GENOMICS, PROTEIN BINDING PROTEIN
4msc:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT1595 (2-[(QUINOLIN-7- YLOXY)METHYL]QUINOLINE) | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4msc:B (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT1595 (2-[(QUINOLIN-7- YLOXY)METHYL]QUINOLINE) | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4msn:A (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT0451 (8-NITROQUINOLINE) | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4msn:B (SER571) to (THR633) CRYSTAL STRUCTURE OF PDE10A2 WITH FRAGMENT ZT0451 (8-NITROQUINOLINE) | FRAGMENT SCREENING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5bml:A (SER6) to (LEU69) ROCK 1 BOUND TO A PYRIDINE THIAZOLE INHIBITOR | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5bml:B (SER6) to (LEU69) ROCK 1 BOUND TO A PYRIDINE THIAZOLE INHIBITOR | KINASE, DIMER, DIMERIZATION, MYOSIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2y0j:A (SER561) to (THR623) TRIAZOLOQUINAZOLINES AS A NOVEL CLASS OF PHOSPHODIESTERASE 10A (PDE10A) INHIBITORS, PART 2, LEAD-OPTIMISATION. | HYDROLASE
5c2e:A (SER561) to (THR623) PDE10 COMPLEXED WITH6-CHLORO-N-[(2,4-DIMETHYLTHIAZOL-5-YL)METHYL]-5- METHYL-2-[2-(2-PYRIDYL)ETHOXY]PYRIMIDIN-4-AMINE | PHOSPHODIESTERASE, INHIBITOR, COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5c2e:B (SER561) to (THR623) PDE10 COMPLEXED WITH6-CHLORO-N-[(2,4-DIMETHYLTHIAZOL-5-YL)METHYL]-5- METHYL-2-[2-(2-PYRIDYL)ETHOXY]PYRIMIDIN-4-AMINE | PHOSPHODIESTERASE, INHIBITOR, COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1khy:C (THR7) to (LEU71) THE CRYSTAL STRUCTURE OF CLPB N TERMINAL DOMAIN, IMPLICATION TO THE PEPTIDE BINDING FUNCTION OF CLPB | ALPHA HELIX, CHAPERONE
1khy:C (SER84) to (MSE143) THE CRYSTAL STRUCTURE OF CLPB N TERMINAL DOMAIN, IMPLICATION TO THE PEPTIDE BINDING FUNCTION OF CLPB | ALPHA HELIX, CHAPERONE
1khy:D (THR7) to (LEU71) THE CRYSTAL STRUCTURE OF CLPB N TERMINAL DOMAIN, IMPLICATION TO THE PEPTIDE BINDING FUNCTION OF CLPB | ALPHA HELIX, CHAPERONE
1khy:D (SER84) to (MSE143) THE CRYSTAL STRUCTURE OF CLPB N TERMINAL DOMAIN, IMPLICATION TO THE PEPTIDE BINDING FUNCTION OF CLPB | ALPHA HELIX, CHAPERONE
3zrb:A (GLN838) to (GLY923) STRUCTURAL BASIS FOR AGONISM AND ANTAGONISM FOR A SET OF CHEMICALLY RELATED PROGESTERONE RECEPTOR MODULATORS | RECEPTOR, AGONIST, ANTAGONIST
2yhd:A (ILE672) to (TYR739) HUMAN ANDROGEN RECEPTOR IN COMPLEX WITH AF2 SMALL MOLECULE INHIBITOR | TRANSCRIPTION, ACTIVATION FUNCTION 2 SITE (AF2), SMALL MOLECULE INHIBITOR
3jwq:B (ASN661) to (THR723) CRYSTAL STRUCTURE OF CHIMERIC PDE5/PDE6 CATALYTIC DOMAIN COMPLEXED WITH SILDENAFIL | MOSTLY ALPHA, ALLOSTERIC ENZYME, CGMP, CGMP-BINDING, HYDROLASE, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, CELL MEMBRANE, LIPOPROTEIN, MEMBRANE, METHYLATION, PRENYLATION, SENSORY TRANSDUCTION, VISION
2yzo:A (GLY162) to (THR206) CRYSTAL STRUCTURE OF UNCHARACTERIZED CONSERVED PROTEIN FROM THERMOTOGA MARITIMA | UNCHARACTERIZED CONSERVED PROTEIN, HYDROLASE, MAGNESIUM, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
2yzo:B (GLY162) to (THR206) CRYSTAL STRUCTURE OF UNCHARACTERIZED CONSERVED PROTEIN FROM THERMOTOGA MARITIMA | UNCHARACTERIZED CONSERVED PROTEIN, HYDROLASE, MAGNESIUM, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
4oh6:A (PRO671) to (TYR739) CRYSTAL STRUCTURE OF T877A-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE | ALPHA-HELIX, HORMONE/GROWTH FACTOR RECEPTOR, PHOSPHORYLATION, HORMONE RECEPTOR-PEPTIDE COMPLEX
4ok1:A (ILE672) to (LEU741) CRYSTAL STRUCTURE OF W741L-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE | ALPHA-HELIX, HORMONE/GROWTH FACTOR RECEPTOR, PHOSPHORYLATION, HORMONE RECEPTOR-PEPTIDE COMPLEX, SIGNAL TRANSDUCTION
1xmy:B (SER282) to (THR345) CATALYTIC DOMAIN OF HUMAN PHOSPHODIESTERASE 4B IN COMPLEX WITH (R)- ROLIPRAM | PHOSPHODIESTERASE, PDE, PDE4B, ROLIPRAM, (R)-ROLIPRAM, HYDROLASE
2o8h:A (SER561) to (THR623) CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF RAT PHOSPHODIESTERASE 10A | PHOSPHODIESTERASE 10A; ZN-BINDING SITE, HYDROLASE
4ae1:B (HIS223) to (VAL288) CRYSTAL STRUCTURE OF DIPHTHERIA TOXIN MUTANT CRM197 IN COMPLEX WITH NICOTINAMIDE | TOXIN
5day:B (PRO65) to (LYS104) THE STRUCTURE OF NAP1-RELATED PROTEIN(NRP1) IN ARABIDOPSIS | HISTONE CHAPERONE, NAP1-RELATED PROTEIN, TRANSCRIPTIONAL ACTIVATION, CHAPERONE
3l1t:A (ALA97) to (HIS144) E. COLI NRFA SULFITE OCMPLEX | MULTIHEME, SULFITE, NITRITE REDUCTASE, C-TYPE CYTOCHROME, ELECTRON TRANSPORT, HEME, IRON, METAL-BINDING, OXIDOREDUCTASE, TRANSPORT
3l1t:C (ALA97) to (HIS144) E. COLI NRFA SULFITE OCMPLEX | MULTIHEME, SULFITE, NITRITE REDUCTASE, C-TYPE CYTOCHROME, ELECTRON TRANSPORT, HEME, IRON, METAL-BINDING, OXIDOREDUCTASE, TRANSPORT
3ahc:A (PRO95) to (PHE133) RESTING FORM OF PHOSPHOKETOLASE FROM BIFIDOBACTERIUM BREVE | THIAMINE DIPHOSPHATE-DEPENDENT ENZYME, ALPHA-BETA FOLD, HOMODIMER, LIGAND-FREE STRUCTURE, LYASE
4ppp:A (THR311) to (ALA382) CRYSTAL STRUCTURE OF THE ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH FLUORO-RESVERATROL | NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, LIGAND-BINDING, NUCLEUS, PROTEIN BINDING
5dru:A (MET35) to (ALA99) STRUCTURE OF HIS387ALA MUTANT OF THE PROPIONALDEHYDE DEHYDROGENASE FROM THE CLOSTRIDIUM PHYTOFERMENTANS FUCOSE UTILISATION BACTERIAL MICROCOMPARTMENT | ACYLATING ALDEHYDE DEHYDROGENASE, BACTERIAL MICROCOMPARTMENT, OXIDOREDUCTASE
3lj2:A (ASP1030) to (PHE1088) IRE1 COMPLEXED WITH JAK INHIBITOR I | KINASE, KINASE INHIBITOR, NUCLEASE ACTIVATOR, ATP-BINDING, ENDOPLASMIC RETICULUM, GLYCOPROTEIN, HYDROLASE, MAGNESIUM, MEMBRANE, METAL-BINDING, MULTIFUNCTIONAL ENZYME, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, TRANSMEMBRANE, UNFOLDED PROTEIN RESPONSE
3lj2:B (ASP1030) to (PHE1088) IRE1 COMPLEXED WITH JAK INHIBITOR I | KINASE, KINASE INHIBITOR, NUCLEASE ACTIVATOR, ATP-BINDING, ENDOPLASMIC RETICULUM, GLYCOPROTEIN, HYDROLASE, MAGNESIUM, MEMBRANE, METAL-BINDING, MULTIFUNCTIONAL ENZYME, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE, TRANSMEMBRANE, UNFOLDED PROTEIN RESPONSE
3c9d:A (GLU8) to (ILE83) CRYSTAL STRUCTURE OF VPS75 | CHROMATIN, HISTONE CHAPERONE, NUCLEUS, PHOSPHOPROTEIN, PROTEIN TRANSPORT, TRANSPORT, CHAPERONE
3nnr:A (ASP108) to (THR191) CRYSTAL STRUCTURE OF A TETR-FAMILY TRANSCRIPTIONAL REGULATOR (MAQU_3571) FROM MARINOBACTER AQUAEOLEI VT8 AT 2.49 A RESOLUTION | TETR-FAMILY TRANSCRIPTIONAL REGULATOR, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-2, TRANSCRIPTION
4rxp:A (ARG164) to (GLY258) THE STRUCTURE OF GTP-DATP-BOUND SAMHD1 | HD-DOMAIN, HYDROLASE, DNTP AND GTP BINDING, PHOSPHORYLATION
4rxp:B (ARG164) to (GLY258) THE STRUCTURE OF GTP-DATP-BOUND SAMHD1 | HD-DOMAIN, HYDROLASE, DNTP AND GTP BINDING, PHOSPHORYLATION
4rxq:A (ARG164) to (GLY258) THE STRUCTURE OF GTP-DUTP-BOUND SAMHD1 | HD-DOMAIN, HYDROLASE, DNTP AND GTP BINDING, PHOSPHORYLATION
4rxs:A (ARG164) to (GLY258) THE STRUCTURE OF GTP-DTTP-BOUND SAMHD1 | HD-DOMAIN, HYDROLASE, DNTP AND GTP BINDING, PHOSPHORYLATION
4rxs:B (ARG164) to (GLY258) THE STRUCTURE OF GTP-DTTP-BOUND SAMHD1 | HD-DOMAIN, HYDROLASE, DNTP AND GTP BINDING, PHOSPHORYLATION
4tnq:A (ARG164) to (GLY258) STRUCTURAL BASIS OF CELLULAR DNTP REGULATION, SAMHD1-GTP-DTTP-DTTP COMPLEX | SAMHD1, HIV, RESTRICTION FACTOR, DNTPASE, DNTP REGULATION, HOST PATHOGEN INTERACTION
4to2:A (PHE213) to (VAL273) STRUCTURE BASIS OF CELLULAR DNTP REGULATION, SAMHD1-DGTP-DGTP- DGTP/DTTP COMPLEX | SAMHD1, HIV, RESTRICTION FACTOR, DNTPASE, DNTP REGULATION, HOST PATHOGEN INTERACTION, HYDROLASE
4to2:B (PHE213) to (VAL273) STRUCTURE BASIS OF CELLULAR DNTP REGULATION, SAMHD1-DGTP-DGTP- DGTP/DTTP COMPLEX | SAMHD1, HIV, RESTRICTION FACTOR, DNTPASE, DNTP REGULATION, HOST PATHOGEN INTERACTION, HYDROLASE
4to2:C (PHE213) to (GLN271) STRUCTURE BASIS OF CELLULAR DNTP REGULATION, SAMHD1-DGTP-DGTP- DGTP/DTTP COMPLEX | SAMHD1, HIV, RESTRICTION FACTOR, DNTPASE, DNTP REGULATION, HOST PATHOGEN INTERACTION, HYDROLASE
4to6:A (ARG164) to (GLY258) STRUCTURE BASIS OF CELLULAR DNTP REGULATION, SAMHD1-DGTP-DATP- DTTP/DGTP COMPLEX | SAMHD1, HIV, RESTRICTION FACTOR, DNTPASE, DNTP REGULATION, HOST PATHOGEN INTERACTION, HYDROLASE
4to6:B (ARG164) to (GLY258) STRUCTURE BASIS OF CELLULAR DNTP REGULATION, SAMHD1-DGTP-DATP- DTTP/DGTP COMPLEX | SAMHD1, HIV, RESTRICTION FACTOR, DNTPASE, DNTP REGULATION, HOST PATHOGEN INTERACTION, HYDROLASE
4dwt:A (GLY1) to (MET49) CARBONMONOXY DEHALOPEROXIDASE-HEMOGLOBIN A STRUCTURE AT 2.05 ANGSTROM RESOLUTION | PEROXIDASE, GLOBIN, HYDROGEN PEROXIDE, 2,4,6-TRIHALOPHENOL, OXIDOREDUCTASE
3ppb:A (PHE130) to (MSE191) CRYSTAL STRUCTURE OF A PUTATIVE TETR FAMILY TRANSCRIPTION REGULATOR (SHEW_3104) FROM SHEWANELLA SP. PV-4 AT 2.10 A RESOLUTION | DNA-BINDING, HELIX-TURN-HELIX MOTIF, HTH MOTIF, DNA/RNA-BINDING 3- HELICAL BUNDLE FOLD, TETRACYCLIN REPRESSOR-LIKE FOLD, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSCRIPTION REGULATOR, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI
3ppb:B (PHE130) to (MSE191) CRYSTAL STRUCTURE OF A PUTATIVE TETR FAMILY TRANSCRIPTION REGULATOR (SHEW_3104) FROM SHEWANELLA SP. PV-4 AT 2.10 A RESOLUTION | DNA-BINDING, HELIX-TURN-HELIX MOTIF, HTH MOTIF, DNA/RNA-BINDING 3- HELICAL BUNDLE FOLD, TETRACYCLIN REPRESSOR-LIKE FOLD, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSCRIPTION REGULATOR, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI
3qpp:A (ASN562) to (THR623) STRUCTURE OF PDE10-INHIBITOR COMPLEX | PHOSPHODIESTERASE INHIBITORS, STRUCTURE-BASED DRUG DESIGN, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
5l08:C (ASP2) to (GLU36) CRYO-EM STRUCTURE OF CASP-8 TDED FILAMENT | CASP-8, FILAMENT, DED, DEATH DOMAIN, APOPTOSIS
5ld2:C (PRO449) to (GLU499) CRYO-EM STRUCTURE OF RECBCD+DNA COMPLEX REVEALING ACTIVATED NUCLEASE DOMAIN | HELICASE, NUCLEASE, SH3, HOMOLOGOUS RECOMBINATION, HYDROLASE